gene_claim_name	gene_concept_id	gene_name	interaction_source_db_name	interaction_source_db_version	interaction_type	interaction_score	drug_claim_name	drug_concept_id	drug_name	approved	immunotherapy	anti_neoplastic
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	RACLOPRIDE	ncit:C152139	RACLOPRIDE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	KALOPANAX-SAPONIN F	chembl:CHEMBL1833984	CHEMBL:CHEMBL1833984	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	RO-5-3335	chembl:CHEMBL91609	CHEMBL:CHEMBL91609	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.034318739	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.6674703970639131	ANGIOTENSIN II	rxcui:1999003	ANGIOTENSIN II	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.026412309	HKI-272	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	2.100306849	CEP-9722	drugbank:DB14882	CEP-9722	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1625	ncit:C80578	ETORPHINE	FALSE	FALSE	FALSE
NCBIGENE:1838	hgnc:3058	DTNB	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8137	iuphar.ligand:8137	COMPOUND 8E [PMID: 24432909]	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:12708	iuphar.ligand:12708	GDC-0339	FALSE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:4303	iuphar.ligand:4303	RYANODINE	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DoCM	10-Apr-24	NULL	1.029066006546944	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CCL4	hgnc:10630	CCL4	NCI	14-Sep-17	NULL	3.182283105193606	CLODRONATE	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.070010228	PLATINUM	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00767656	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.5707355569097228	BENZENETHIOL	chembl:CHEMBL119405	BENZENETHIOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SJ000114961	chembl:CHEMBL590168	CHEMBL:CHEMBL590168	FALSE	FALSE	FALSE
CSNK2A3	hgnc:2458	CSNK2A3	PharmGKB	4/5/24	NULL	0.7242437411819931	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	1.790034246671403	ARBUTAMINE	rxcui:61609	ARBUTAMINE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.2302968036653267	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.8899605294185507	YM-358	chembl:CHEMBL347610	CHEMBL:CHEMBL347610	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2060	iuphar.ligand:2060	[125I]TYR11-SRIF-14	FALSE	FALSE	FALSE
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	0.1547594520630995	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.1666910197958555	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	1.250182648468916	LANOTEPLASE	ncit:C96707	LANOTEPLASE	FALSE	FALSE	FALSE
KCND3	hgnc:6239	KCND3	ChEMBL	33	blocker	1.093909817410302	VERNAKALANT HYDROCHLORIDE	ncit:C152865	VERNAKALANT HYDROCHLORIDE	FALSE	FALSE	FALSE
RPL28	hgnc:10330	RPL28	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.056622219	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.201178817	MAREIN	chembl:CHEMBL490510	MAREIN	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.546954909	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.017709164	Tetrabenazine	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
UNIPROT:Q16665	hgnc:4910	HIF1A	TdgClinicalTrial	Jan-14	NULL	0.090530468	NOSCAPINE	rxcui:7533	NOSCAPINE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1037701012563132	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:1502	iuphar.ligand:1502	NEUROPEPTIDE B-29	FALSE	FALSE	FALSE
NCBIGENE:1252	hgnc:5187	PRMT1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7029	iuphar.ligand:7029	RM65	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1090501998664475	RO5126766	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.2692701089009974	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.011452055	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	7.501095891	Amsilarotene	ncit:C38684	AMSILAROTENE	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.2143170254518143	IUPHAR.LIGAND:8784	iuphar.ligand:8784	SGI-1776	FALSE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:6981	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	THEONELLASTEROL E	chembl:CHEMBL1782601	THEONELLASTEROL E	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	GNF-PF-5052	chembl:CHEMBL601367	CHEMBL:CHEMBL601367	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.00809055	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.043756393	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
IL6R	hgnc:6019	IL6R	DTC	9/2/20	NULL	1.615620653405984	BAZEDOXIFENE	rxcui:1441386	BAZEDOXIFENE	TRUE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.019440086	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.036087747	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.2524407270946851	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	S-NITROSOGLUTATHIONE	drugbank:DB17877	S-NITROSOGLUTATHIONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.1640864726115453	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:3850	iuphar.ligand:3850	[SAR9,MET(O2)11]SP	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	agonist	0.760980743	VASOPRESSIN TANNATE	chembl:CHEMBL1201528	VASOPRESSIN TANNATE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	2.917092846427472	PITAVASTATIN MAGNESIUM	rxcui:2001252	PITAVASTATIN MAGNESIUM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	CARBETAPENTANE CITRATE	rxcui:283547	CARBETAPENTANE CITRATE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	MyCancerGenome	20-Jun-17	immunotherapy	0.6177373086552294	MDX-1105	ncit:C78852	ANTI-PD-L1 MONOCLONAL ANTIBODY MDX-1105	FALSE	TRUE	TRUE
CD274	hgnc:17635	CD274	MyCancerGenome	20-Jun-17	antibody	0.6177373086552294	MDX-1105	ncit:C78852	ANTI-PD-L1 MONOCLONAL ANTIBODY MDX-1105	FALSE	TRUE	TRUE
NCBIGENE:2651	hgnc:4204	GCNT2	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:7014	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
PAK-4 PROTEIN KINASE	hgnc:16059	PAK4	TTD	2020.06.01	NULL	2.187819634820604	KPT-9274	ncit:C126646	PADNARSERTIB	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.040814358	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	blocker	0.2282942227638891	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	blocker	0.5556367326528517	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	2.917092846427472	THIOURACIL	ncit:C29856	THIOURACIL	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.5834185692854944	BACILLUS CALMETTE-GUERIN	hemonc:59	BCG VACCINE	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.182318303	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	AM-404	iuphar.ligand:12556	AM404	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	ARACHIDONOYL GABA	iuphar.ligand:5494	N-ARACHIDONYL-&GAMMA;-AMINOBUTYRIC ACID	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	DNDI1417006	chembl:CHEMBL1415258	CHEMBL:CHEMBL1415258	FALSE	FALSE	FALSE
UNIPROT:Q03181	hgnc:9235	PPARD	TdgClinicalTrial	Jan-14	NULL	1.579178082276526	CER-002	chembl:CHEMBL3544958	CER-002	FALSE	FALSE	FALSE
UNIPROT:Q13324	hgnc:2358	CRHR2	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	CORTICOTROPIN-RELEASING FACTOR	iuphar.ligand:913	CORTICOTROPIN-RELEASING FACTOR	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.09969811	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.083478015	IUPHAR.LIGAND:7135	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.1808115400678185	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.089501712	MESALAZINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
N-FORMYL PEPTIDE RECEPTOR	hgnc:3826	FPR1	TTD	2020.06.01	NULL	1.166837138570988	Rebamipide	ncit:C29852	REBAMIPIDE	FALSE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	1.193356164447602	ABBV-3067	chembl:CHEMBL4802150	NAVOCAFTOR	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.060077427	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
C10ORF67	hgnc:28716	C10orf67	PharmGKB	4/5/24	NULL	1.193356164447602	mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.1736364789540161	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.035358701	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2917092846427472	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
RARG	hgnc:9866	RARG	NCI	14-Sep-17	NULL	0.2989051493493045	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.4055851016423223	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.4953553890159858	BMS-695735	chembl:CHEMBL459729	CHEMBL:CHEMBL459729	FALSE	FALSE	FALSE
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	1.312691780892362	DS-3032	ncit:C141432	MILADEMETAN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.020029629	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
TERT	hgnc:11730	TERT	CGI	2/1/22	NULL	0.4800701370120639	Eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.007123548	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	CGI	2/1/22	NULL	2.080014029626545	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.1244257612220248	SRT-1720	drugbank:DB17057	SRT-1720	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	4-BENZYLOXYANILINE	chembl:CHEMBL1351571	4-BENZYLOXYANILINE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	MyCancerGenome	20-Jun-17	inhibitor	1.826353782111112	X-396	drugbank:DB13104	X-396	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	umifenovir	ncit:C152799	UMIFENOVIR	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:5290	iuphar.ligand:5290	Y27632	FALSE	FALSE	FALSE
NCBIGENE:1232	hgnc:1604	CCR3	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:11776	iuphar.ligand:11776	DALUTRAFUSP ALFA	FALSE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	ChEMBL	33	inhibitor	4.039051633514961	ELOBIXIBAT	ncit:C171820	ELOBIXIBAT	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.1547594520630995	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.3454452054979901	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.108040476	ARRY-614	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	METHYLPREDNISOLONE SODIUM SUCCINATE	rxcui:203189	METHYLPREDNISOLONE SODIUM SUCCINATE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	0.9723642821424906	FLUVASTATIN SODIUM	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	modulator	0.046965717	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	1.779921058837101	TASOSARTAN	ncit:C152517	TASOSARTAN	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	0.8751278539282416	FARICIMAB	rxcui:2591519	FARICIMAB	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.059219178	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.6168664383892681	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.009662803	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.002270406	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.1154014752432845	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.7955707762984013	Nepafenac	rxcui:298665	NEPAFENAC	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.2044691247495891	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.054695491	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	DTC	9/2/20	NULL	8.353493151133215	LUMACAFTOR	rxcui:1655922	LUMACAFTOR	TRUE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	negative modulator	3.281729452230906	PRILIXIMAB	ncit:C188634	PRILIXIMAB	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	SOFALCONE	ncit:C81118	SOFALCONE	FALSE	FALSE	FALSE
CHKA	hgnc:1937	CHKA	NCI	14-Sep-17	NULL	0.6105543166941221	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	agonist	0.035430277	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.5357925636295356	IUPHAR.LIGAND:6440	iuphar.ligand:6440	AZD6538	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:9442	iuphar.ligand:9442	LV-2172	FALSE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	ChEMBL	33	modulator	0.3977853881492006	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.040437175	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.055740628	DP001	iuphar.ligand:2776	2MD	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE	chembl:CHEMBL1371413	2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE	FALSE	FALSE	FALSE
PLCG2	hgnc:9066	PLCG2	CGI	2/1/22	NULL	4.773424657790409	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
UNIPROT:P18084	hgnc:6160	ITGB5	TdgClinicalTrial	Jan-14	NULL	7.876150685354174	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:499	iuphar.ligand:499	WB 4101	FALSE	FALSE	FALSE
NCBIGENE:390	hgnc:671	RND3	GuideToPharmacology	2024.1	activator	0.3804903712731485	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
CXCL12	hgnc:10672	CXCL12	PharmGKB	4/5/24	NULL	1.312691780892362	chlorambucil	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.06823609	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.035430277	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.5147810905460245	Antibiotics	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	Vilanterol	rxcui:1424884	VILANTEROL	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE	chembl:CHEMBL1371413	2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.015036561	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.085378327	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.2154897588332195	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1117184494376478	PROPANTHELINE BROMIDE	rxcui:8762	PROPANTHELINE BROMIDE	TRUE	FALSE	FALSE
YWHAE	hgnc:12851	YWHAE	NCI	14-Sep-17	NULL	1.981421556063943	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:2595	iuphar.ligand:2595	R-L3	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	CIViC	10-Apr-24	NULL	0.014484875	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P41595	hgnc:5294	HTR2B	TEND	1-Aug-11	NULL	0.4375639269641209	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:8520	iuphar.ligand:8520	COMPOUND 58 [PMID: 25037917]	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.030688294	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:287	iuphar.ligand:287	(-)-YM796	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:10003	iuphar.ligand:10003	GNE-131	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:2226	rxcui:358257	TOLVAPTAN	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1905904582057876	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.007737647	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.7095631248066824	BEFIRADOL	ncit:C81392	BEFIRADOL	FALSE	FALSE	FALSE
RPL35	hgnc:10344	RPL35	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	LOBELINE HYDROCHLORIDE	chembl:CHEMBL1257005	LOBELINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.061412481	NONIVAMIDE	rxcui:31945	NONIVAMIDE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.029766254	IUPHAR.LIGAND:7247	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
CDK20	hgnc:21420	CDK20	ChEMBL	33	inhibitor	0.6250913242344582	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.2019525816757481	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.03394161	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.091796628	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
NCBIGENE:2650	hgnc:4203	GCNT1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:7019	ncit:C103179	PINOMETOSTAT	FALSE	FALSE	TRUE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5749	rxcui:1665496	ROLAPITANT	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.009433646	IUPHAR.LIGAND:5659	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2332563532602643	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	5-(2-PHENYLETHYL)ISATIN	chembl:CHEMBL1642672	CHEMBL:CHEMBL1642672	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.4930297768609811	NALTREXONE HYDROCHLORIDE	rxcui:105069	NALTREXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.036847489	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2035181055647073	OT-730	drugbank:DB16112	OT-730	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.078545507	TAE226	iuphar.ligand:9382	NVP-TAE 226	FALSE	FALSE	FALSE
LPAR1	hgnc:3166	LPAR1	ChEMBL	33	inhibitor	26.25383561784724	BMS-986020	drugbank:DB14948	BMS-986020	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000093004	chembl:CHEMBL590914	CHEMBL:CHEMBL590914	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.096264064	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
GUCA2A	hgnc:4682	GUCA2A	NCI	14-Sep-17	NULL	8.751278539282415	LACTOSE	rxcui:6211	LACTOSE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	0.3671865121377238	ERGOTAMINE	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1229687850953032	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.050246575	IUPHAR.LIGAND:150	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
UNIPROT:P51787	hgnc:6294	KCNQ1	TdgClinicalTrial	Jan-14	NULL	1.432027397337122	INDAPAMIDE	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1787	hgnc:2977	TRDMT1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8144	iuphar.ligand:8144	COMPOUND 13R [PMID: 23639540]	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	0.5498185469706229	RO-5212054	chembl:CHEMBL3545080	RG-7256	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.092933931	IUPHAR.LIGAND:1642	iuphar.ligand:1642	NOR-BINALTORPHIMINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.9546849315580818	LIRAGLUTIDE	rxcui:475968	LIRAGLUTIDE	TRUE	FALSE	FALSE
RPS10	hgnc:10383	RPS10	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	0.6731752722524935	GSK525762	ncit:C101538	MOLIBRESIB	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:441	iuphar.ligand:441	AS95	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.095468493	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
HEAT SHOCK PROTEIN	hgnc:12099	HSP90B2P	TTD	2020.06.01	NULL	52.50767123569449	Arimoclomol	ncit:C79744	ARIMOCLOMOL	FALSE	FALSE	FALSE
NCBIGENE:415	hgnc:719	ARSL	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.1268301237577161	TERAZOSIN HYDROCHLORIDE	rxcui:235224	TERAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.172722603	Conatumumab	ncit:C71015	CONATUMUMAB	FALSE	TRUE	TRUE
NCBIGENE:1993	hgnc:3313	ELAVL2	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:8161	iuphar.ligand:8161	COMPOUND 17 [PMID: 23642479]	FALSE	FALSE	FALSE
NCBIGENE:664	hgnc:1084	BNIP3	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:9675	drugbank:DB05767	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:2626	iuphar.ligand:2626	VERATRIDINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ALLISAN	chembl:CHEMBL504381	ALLISAN	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.1842374429322613	XL880	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.039960176	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.7955707762984013	N-(3-OXODODECANOYL)HOMOSERINELACTONE	chembl:CHEMBL8483	CHEMBL:CHEMBL8483	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.018570352	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.4487835148349957	RAMIPRIL	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.032572997	Ergotidine	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:3218	iuphar.ligand:3218	(R)-UH 301	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:12758	iuphar.ligand:12758	GLOFITAMAB	FALSE	FALSE	FALSE
NCBIGENE:697	ncbigene:697	BTNL1	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
DELTA-LIKE PROTEIN 4	hgnc:2910	DLL4	TTD	2020.06.01	NULL	31.50460274141669	OMP-21M18	ncit:C80041	DEMCIZUMAB	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.003384317	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TNIK	hgnc:30765	TNIK	PharmGKB	4/5/24	NULL	0.3918482928036902	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
PSMA2	hgnc:9531	PSMA2	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	agonist	1.381780822	FLUDROCORTISONE ACETATE	rxcui:165516	FLUDROCORTISONE ACETATE	TRUE	FALSE	FALSE
ITGA2B	hgnc:6138	ITGA2B	ChEMBL	33	inhibitor	3.500511415712967	EPTIFIBATIDE	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.090530468	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(+)-VENTILOQUINONE	chembl:CHEMBL594257	CHEMBL:CHEMBL594257	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.6105543166941221	PEITC	ncit:C2233	PHENETHYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1325951293830669	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 23 MEMBER 1	hgnc:10974	SLC23A1	TTD	2020.06.01	NULL	2.019525816757481	Vitamin C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M4	hgnc:1953	CHRM4	TTD	2020.06.01	NULL	0.3241214273808302	Methacholine Chloride	rxcui:40165	METHACHOLINE CHLORIDE	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1013661606866689	E6201	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	chembl:CHEMBL1449651	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	FALSE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TEND	1-Aug-11	NULL	0.08914715	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
IMPDH2	hgnc:6053	IMPDH2	ChEMBL	33	inhibitor	2.625383561784724	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	AM-404	iuphar.ligand:12556	AM404	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:11491	iuphar.ligand:11491	CPN-219	FALSE	FALSE	FALSE
HCN4	hgnc:16882	HCN4	ChEMBL	33	blocker	17.50255707856483	IVABRADINE HYDROCHLORIDE	rxcui:1649479	IVABRADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.116943588	METHANDROSTENOLONE	rxcui:6818	METHANDROSTENOLONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	5-(4-PHENYLBUTOXY)PSORALEN	iuphar.ligand:9583	PSORA-4	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	CGS-15943	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	1.129197231	OZORALIZUMAB	ncit:C175183	OZORALIZUMAB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00903591	quinine	rxcui:9071	QUININE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2209	iuphar.ligand:2209	[PHAA1,D-TYR(ET)2,VAL4,LYS6,TYR-NH28,DES-GLY9]AVP	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.015466177	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	potentiator	0.6963882126749933	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1000146118775133	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	modulator	1.458546423213736	ABT-560	drugbank:DB06093	ABT-560	FALSE	FALSE	FALSE
DHCR24	hgnc:2859	DHCR24	ChEMBL	33	inhibitor	3.281729452230906	TRIPARANOL	ncit:C152752	TRIPARANOL	TRUE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.053145416	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.039214094	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	TCMDC-123516	chembl:CHEMBL547304	CHEMBL:CHEMBL547304	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.023482858	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	THYMOL IODIDE	rxcui:89717	THYMOL IODIDE	TRUE	FALSE	FALSE
OSM	hgnc:8506	OSM	NCI	14-Sep-17	NULL	2.187819634820604	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.1842374429322613	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:64	iuphar.ligand:64	(-)-TERTATOLOL	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.069089041	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.004589831	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.4565884455277783	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	SJ000111093	chembl:CHEMBL585045	CHEMBL:CHEMBL585045	FALSE	FALSE	FALSE
UNIPROT:P14060	hgnc:5217	HSD3B1	TEND	1-Aug-11	NULL	8.751278539282415	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00675253	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
NCBIGENE:2353	hgnc:3796	FOS	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:6478	iuphar.ligand:6478	ODANACATIB	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:12065	iuphar.ligand:12065	BI-167107	FALSE	FALSE	FALSE
NCBIGENE:2603	hgnc:2861	DHFR	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:7613	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.095468493	Sapanisertib	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	6.300920548	Ledipasvir	rxcui:1591922	LEDIPASVIR	TRUE	FALSE	FALSE
GPC3	hgnc:4451	GPC3	ChEMBL	33	inhibitor	10.50153424713889	CODRITUZUMAB	ncit:C80043	CODRITUZUMAB	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.1178623372293928	PAMIDRONATE	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	GNF-PF-3792	chembl:CHEMBL582983	CHEMBL:CHEMBL582983	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1363835616511545	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:443	iuphar.ligand:443	BW-A1433	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.2051080907644316	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	1.712206670729168	Conivaptan	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	1.779921058837101	Tasosartan	ncit:C152517	TASOSARTAN	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.2333674277141977	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	DNDI1417461	chembl:CHEMBL1520282	CHEMBL:CHEMBL1520282	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	modulator	0.210030685	ARHALOFENATE	ncit:C83536	ARHALOFENATE	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.1875273972703375	GW405833	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.010213911	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CAV1	hgnc:1527	CAV1	NCI	14-Sep-17	NULL	0.3323270331373069	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
ADM	hgnc:259	ADM	PharmGKB	4/5/24	NULL	0.525076712	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	LY-255283	chembl:CHEMBL15766	LY-255283	FALSE	FALSE	FALSE
SIRT3	hgnc:14931	SIRT3	TALC	12-May-16	inhibitor	0.3977853881492008	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.065675636	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	0.6731752722524936	Ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	8.751278539282417	TZP-101	ncit:C102755	ULIMORELIN HYDROCHLORIDE	FALSE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	4.375639269641208	SAR-566658	chembl:CHEMBL2109635	SAR-566658	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	NSC-636948	chembl:CHEMBL1998001	CHEMBL:CHEMBL1998001	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	2.019525817	NSC-640583	chembl:CHEMBL1287895	CHEMBL:CHEMBL1287895	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	1.093909817410302	2X-121	drugbank:DB16063	2X-121	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	TRICLOSAN	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-574	chembl:CHEMBL582737	CHEMBL:CHEMBL582737	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	ChEMBL	33	inhibitor	0.1904575128526865	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-2374	chembl:CHEMBL600298	CHEMBL:CHEMBL600298	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	NCI	14-Sep-17	NULL	0.015655239	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NCBIGENE:3015	hgnc:4741	H2AZ1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10048	iuphar.ligand:10048	ERW1041E	FALSE	FALSE	FALSE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	8.751278539282415	LEBRIKIZUMAB	ncit:C87767	LEBRIKIZUMAB	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	PharmGKB	4/5/24	NULL	0.072775705	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1875273972703375	Trimethoprim	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	blocker	0.2243917574174979	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
UNIPROT:P35346	hgnc:11334	SSTR5	TdgClinicalTrial	Jan-14	NULL	0.729273212	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.03124062	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CTSC	hgnc:2528	CTSC	NCI	14-Sep-17	NULL	3.000438356	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.5834185692854944	vardenafil	rxcui:306674	VARDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9386	iuphar.ligand:9386	BMS-536924	FALSE	FALSE	TRUE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.2853677784548614	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.7440358272264402	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.1056492378987816	VISTUSERTIB	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	GITOXIN	chembl:CHEMBL109317	GITOXIN	FALSE	FALSE	FALSE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	3.500511415712966	itopride	ncit:C65991	ITOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:473	iuphar.ligand:473	MRS1505	FALSE	FALSE	FALSE
NCBIGENE:688	hgnc:6349	KLF5	GuideToPharmacology	2024.1	blocker	6.563458904461812	IUPHAR.LIGAND:10939	iuphar.ligand:10939	5-HYDROXYMETHYL-2-FURFURAL	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.008475815	IUPHAR.LIGAND:4920	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NCBIGENE:2397	hgnc:3908	FRA5D	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8559	iuphar.ligand:8559	COMPOUND 9 [PMID: 3514912]	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:4573	iuphar.ligand:4573	THREO-3-METHYLGLUTAMATE	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.1286952726365061	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
ADCYAP1	hgnc:241	ADCYAP1	NCI	14-Sep-17	NULL	1.093909817410302	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.010586224	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	WAY-629	chembl:CHEMBL258465	CHEMBL:CHEMBL258465	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	OncoKB	23-Jul-20	NULL	0.060772768	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	ERGOCRISTINE	chembl:CHEMBL446315	ERGOCRISTINE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:9286	iuphar.ligand:9286	PZM21	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.055563673	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.036038209	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:12084	iuphar.ligand:12084	PIFUSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.007596596	IUPHAR.LIGAND:9381	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
RRM1	hgnc:10451	RRM1	CIViC	10-Apr-24	NULL	0.028598949	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:4239	iuphar.ligand:4239	L689560	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.055681518	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.059330702	IUPHAR.LIGAND:8014	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	6-O-BENZYLGUANINE	drugbank:DB11919	6-O-BENZYLGUANINE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.4150804050252529	QUINAGOLIDE	rxcui:76887	QUINAGOLIDE	FALSE	FALSE	FALSE
NCBIGENE:2149	hgnc:3537	F2R	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:6062	drugbank:DB06836	N-(5-{4-CHLORO-3-[(2-HYDROXYETHYL)SULFAMOYL]PHENYL}-4-METHYL-1,3-THIAZOL-2-YL)ACETAMIDE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	PALMITOYL-DL-CARNITINE CHLORIDE	chembl:CHEMBL1256761	CHEMBL:CHEMBL1256761	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	THYMOL IODIDE	rxcui:89717	THYMOL IODIDE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.064505739	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	negative modulator	0.1530835896084387	ESKETAMINE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.2586584789935689	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.6731752722524935	NSC-119911	chembl:CHEMBL502775	CHEMBL:CHEMBL502775	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1875273972703375	TCMDC-124522	chembl:CHEMBL526776	CHEMBL:CHEMBL526776	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,7-BIS[3-(ETHYLAMINO)PROPIONAMIDO]ANTHRAQUINONE	chembl:CHEMBL481161	CHEMBL:CHEMBL481161	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	CIViC	10-Apr-24	NULL	0.1121958787087489	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	CIViC	10-Apr-24	NULL	0.1935766681500258	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	8-{[(4-BROMOPHENYL)METHYL]SULFANYL}CAFFEINE	chembl:CHEMBL1927670	CHEMBL:CHEMBL1927670	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:5691	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	4.375639269641208	BRIAKINUMAB	ncit:C95321	BRIAKINUMAB	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.08780547	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIA	chembl:CHEMBL1094691	AESCULIOSIDE IIA	FALSE	FALSE	FALSE
NCBIGENE:724	hgnc:1327	C4BPAP2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.2573905452730122	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
ITGA2B	hgnc:6138	ITGA2B	ChEMBL	33	inhibitor	2.187819634820604	ZALUNFIBAN	ncit:C180665	ZALUNFIBAN	FALSE	FALSE	FALSE
NCBIGENE:2371	hgnc:3879	FRA1L	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8596	iuphar.ligand:8596	NTE-1	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.7440358272264402	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	SB-242084	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
FANCC	hgnc:3584	FANCC	CIViC	10-Apr-24	NULL	0.5000730593875666	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	N-ETHYLMALEIMIDE	drugbank:DB02967	N-ETHYLMALEIMIDE	FALSE	FALSE	FALSE
EYA4	hgnc:3522	EYA4	PharmGKB	4/5/24	NULL	0.6731752722524936	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	0.9053046764774912	GSK2245840	iuphar.ligand:9515	SRT2104	FALSE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA2.2	hgnc:6291	KCNN2	TTD	2020.06.01	NULL	3.281729452230906	dequalinium	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00410569	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR DELTA	hgnc:4084	GABRD	TTD	2020.06.01	NULL	0.075768645	Ganaxolone	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	SILVER SULFADIAZINE	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.054355767	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	DNDI1416988	chembl:CHEMBL1389794	CHEMBL:CHEMBL1389794	FALSE	FALSE	FALSE
EFR3A	hgnc:28970	EFR3A	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
WBP2NL	hgnc:28389	WBP2NL	PharmGKB	4/5/24	NULL	1.093909817410302	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1100789753368857	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.030868707	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	blocker	0.1442518440541058	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.003811809	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:9342	iuphar.ligand:9342	ALARELIN	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.546954909	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.1620607136904151	E-GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	inhibitor	1.640864726115453	TICLOPIDINE HYDROCHLORIDE	rxcui:97	TICLOPIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.637458239	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
NCBIGENE:585	hgnc:969	BBS4	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:10119	iuphar.ligand:10119	AM-6120	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ORBIFLOXACIN	rxcui:995897	ORBIFLOXACIN	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.5834185692854944	TCMDC-124416	chembl:CHEMBL530664	CHEMBL:CHEMBL530664	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:5192	iuphar.ligand:5192	G&OUML; 6983	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.036770078	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
UNIPROT:P42263	hgnc:4573	GRIA3	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	BGG-492	chembl:CHEMBL3545042	SELURAMPANEL	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.1600843635234588	IUPHAR.LIGAND:1936	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	E-4031	iuphar.ligand:2605	E4031	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	GNF-PF-107	chembl:CHEMBL578675	CHEMBL:CHEMBL578675	FALSE	FALSE	FALSE
UNIPROT:Q70Z44	hgnc:24004	HTR3D	TdgClinicalTrial	Jan-14	NULL	1.500219178	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.088866948	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.2631963470460877	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	4.565884455277782	MLN1202	ncit:C88308	PLOZALIZUMAB	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	CGI	2/1/22	NULL	0.3302369260106572	Tegafur	rxcui:10995	URACIL	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.037666909	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.063034419	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.3281729452230906	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.072424374	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P16444	hgnc:3002	DPEP1	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	CILASTATIN	rxcui:2540	CILASTATIN	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.037398626	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.297915865	amlodipine	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	NSC-693571	chembl:CHEMBL1287983	CHEMBL:CHEMBL1287983	FALSE	FALSE	FALSE
RXRG	hgnc:10479	RXRG	ChEMBL	33	modulator	0.7955707762984013	MOFAROTENE	ncit:C63667	MOFAROTENE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	2-(2'-METHOXYPHENYL)-1H-INDOLE	chembl:CHEMBL1449007	2-(2'-METHOXYPHENYL)-1H-INDOLE	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:10224	iuphar.ligand:10224	CASOXIN C	FALSE	FALSE	FALSE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.081597003	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.4953553890159858	N-(BENZYLCARBAMOTHIOYL)BENZAMIDE	chembl:CHEMBL1478462	CHEMBL:CHEMBL1478462	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	NSC-724440	chembl:CHEMBL515617	CHEMBL:CHEMBL515617	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.098328972	IUPHAR.LIGAND:8915	iuphar.ligand:8915	AZD8835	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1071585127259071	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	2.187819634820604	Ivosidenib	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.014977128	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.08334551	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.025827679	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.01689436	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1651184630053286	VORICONAZOLE	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.035617739	sertindole	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	1.093909817410302	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.071439008	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.596678082	ROFLUMILAST	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
NCBIGENE:1836	hgnc:10994	SLC26A2	GuideToPharmacology	2024.1	NULL	3.750547945	IUPHAR.LIGAND:5050	iuphar.ligand:5050	PROTEIN S	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.3182283105193605	PEXIDARTINIB HYDROCHLORIDE	rxcui:2183103	PEXIDARTINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.192335792	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	S-49076	drugbank:DB16821	S-49076	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	0.06714536	Masitinib	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.005235062	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
AURORA KINASE C	hgnc:11391	AURKC	TTD	2020.06.01	NULL	1.312691780892362	PHA-739358	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.8899605294185507	IUPHAR.LIGAND:3217	iuphar.ligand:3217	E6801	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	5,7-DICHLOROKYNURENIC ACID	drugbank:DB01931	5,7-DICHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MESTANOLONE	ncit:C83939	MESTANOLONE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.033148782	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.05814803	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.9634435089118256	ALPHA-ENDORPHIN	chembl:CHEMBL255300	CHEMBL:CHEMBL255300	FALSE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	3.621218705909965	Chi Lob 7/4	ncit:C101366	ANTI-CD40 MONOCLONAL ANTIBODY CHI LOB 7/4	FALSE	FALSE	FALSE
TFAP2A	hgnc:11742	TFAP2A	NCI	14-Sep-17	NULL	2.917092846427472	NELFINAVIR	rxcui:134527	NELFINAVIR	TRUE	FALSE	TRUE
FAM178B	hgnc:28036	FAM178B	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
UNIPROT:P31785	hgnc:6010	IL2RG	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	INTERLEUKIN-2	ncit:C587	RECOMBINANT INTERLEUKIN-2	FALSE	FALSE	FALSE
FSHR	hgnc:3969	FSHR	PharmGKB	4/5/24	NULL	18.37768493249307	follitropin beta	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	SUFENTANIL	rxcui:56795	SUFENTANIL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	Protokylol Hydrochloride	ncit:C66496	PROTOKYLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.729273212	DECAMETHONIUM	ncit:C77363	DECAMETHONIUM	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:392	iuphar.ligand:392	MRS1041	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.054243462	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:523	ncit:C75049	XYLAZINE	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:916	iuphar.ligand:916	[125I]SAUVAGINE (FROG)	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.065634589	mepivacaine	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:277	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.100976291	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.011419676	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	E-GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
CYP27A1	hgnc:2605	CYP27A1	NCI	14-Sep-17	NULL	0.4234489615781814	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.1553481397505754	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.032252869	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.1193356164447602	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.088945801	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1017590527823536	SULOCHRIN	chembl:CHEMBL61133	SULOCHRIN	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.276356164	PARTHENOLIDE	rxcui:32941	PARTHENOLIDE	FALSE	FALSE	FALSE
ADCYAP1R1	hgnc:242	ADCYAP1R1	NCI	14-Sep-17	NULL	0.6250913242344582	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	4.145342465975881	CHLORMEZANONE	rxcui:2373	CHLORMEZANONE	TRUE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.1154014752432846	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:423	iuphar.ligand:423	N(6)-CYCLOHEXYLADENOSINE	FALSE	FALSE	FALSE
CA9	hgnc:1383	CA9	PharmGKB	4/5/24	NULL	0.1119566550867686	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.057574201	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	ALTANSERIN	ncit:C77258	ALTANSERIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.3977853881492006	OX-914	chembl:CHEMBL4297287	HT-0712	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:5191	iuphar.ligand:5191	FR122047	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	CGI	2/1/22	NULL	0.4735540335109532	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.027476542	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
ZNF816	hgnc:26995	ZNF816	PharmGKB	4/5/24	NULL	0.8468979231563629	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
TBXAS1	hgnc:11609	TBXAS1	PharmGKB	4/5/24	NULL	0.093098708	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.3231241306811969	PROPERICIAZINE	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	OncoKB	23-Jul-20	NULL	2.212697851403848	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.1346350544504987	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2327	hgnc:3770	FMO2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8559	iuphar.ligand:8559	COMPOUND 9 [PMID: 3514912]	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.019695301	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5754	iuphar.ligand:5754	R116031	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.085332077	TSU-68	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.052948912	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2386712328895204	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.030368809	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.7001022831425933	DIMETHYLFORMAMIDE	chembl:CHEMBL268291	DIMETHYLFORMAMIDE	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	3.182283105193606	TRIAZENE COMPOUNDS	ncit:C902	TRIAZENE COMPOUND	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	AMBUNOL	chembl:CHEMBL454893	AMBUNOL	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.088248187	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.029918901	ANTICONVULSANTS	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
STRBP	hgnc:16462	STRBP	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.2051080907644316	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.4070362111294147	Inavolisib	ncit:C132166	INAVOLISIB	FALSE	FALSE	TRUE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1349	iuphar.ligand:1349	GR 196429	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.3571950424196904	DIHYDROSPHINGOSINE	iuphar.ligand:2453	DIHYDROSPHINGOSINE	FALSE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 3	hgnc:11332	SSTR3	TTD	2020.06.01	NULL	1.458546423213736	Pasireotide	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	CLOFAZIMINE	rxcui:2592	CLOFAZIMINE	TRUE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.049723174	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1198	iuphar.ligand:1198	UR-PG131A	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:4460	ncit:C169980	FILOREXANT	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.016764901	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.030386384	Navitoclax	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.006077277	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	SKF-10047	chembl:CHEMBL101510	CHEMBL:CHEMBL101510	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10424	iuphar.ligand:10424	HSD1590	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.096264064	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABL	hgnc:76	ABL1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.637458239	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1400204566285186	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014993624	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004207345	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.063110182	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.048483538	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.007119684	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	0.084146909	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.018874073	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
ALCAM	hgnc:400	ALCAM	CIViC	10-Apr-24	NULL	0.01131387	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	0.4327555321623173	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:846	iuphar.ligand:846	CXCL12-(1-17)	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.5609793935437446	TARIQUIDAR	ncit:C2246	TARIQUIDAR	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.048663273	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.026519026	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
NCBIGENE:735	hgnc:1358	C9	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.031254566	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	CID 5310655	chembl:CHEMBL408563	CHEMBL:CHEMBL408563	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.061628722	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:446	iuphar.ligand:446	I-ABOPX	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.3571950424196904	LEVOFLOXACIN	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1377	iuphar.ligand:1377	DCG-IV	FALSE	FALSE	FALSE
NCBIGENE:1630	hgnc:2701	DCC	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	SJ000147784	chembl:CHEMBL590186	CHEMBL:CHEMBL590186	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.041344623	INDOCYANINE GREEN	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
UNIPROT:Q14568	hgnc:5256	HSP90AA2P	TdgClinicalTrial	Jan-14	NULL	7.001022831425932	RETASPIMYCIN	ncit:C80378	RETASPIMYCIN	FALSE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.8468979231563628	Vapitadine	ncit:C96721	VAPITADINE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	Metipranolol	rxcui:10824	METIPRANOLOL	TRUE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	6.563458904461812	PRX-08066	drugbank:DB05607	PRX-08066	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	ChEMBL	33	inhibitor	0.1342907192728759	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1185944014357865	DOMPERIDONE	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TdgClinicalTrial	Jan-14	NULL	3.750547945	DINOPROST TROMETHAMINE	rxcui:23321	DINOPROST TROMETHAMINE	TRUE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:12057	iuphar.ligand:12057	TP0556351	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:2613	iuphar.ligand:2613	AFT-II	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:5610	iuphar.ligand:5610	MSX-2	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:2924	iuphar.ligand:2924	FINGOLIMOD-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.2206204673768676	IUPHAR.LIGAND:10947	iuphar.ligand:10947	NIK INHIBITOR 12F	FALSE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	0.175610941	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-123808	chembl:CHEMBL546493	CHEMBL:CHEMBL546493	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	ADEFOVIR DIPIVOXIL	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.5357925636295356	IUPHAR.LIGAND:1426	iuphar.ligand:1426	MPEP	FALSE	FALSE	FALSE
NCBIGENE:2379	hgnc:3891	FRA2G	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8493	iuphar.ligand:8493	COMPOUND 11 [PMID: 16413183]	FALSE	FALSE	FALSE
ARAF	hgnc:646	ARAF	CIViC	10-Apr-24	NULL	0.019093699	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.050805681	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
ABCG1	hgnc:73	ABCG1	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.041639708	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.006525935	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	0.1689436011444482	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.1535312024435511	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.5303805175322677	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1017590527823536	ZK-93423	drugbank:DB17063	ZK-93423	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.071004288	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.060772768	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
NCBIGENE:3248	hgnc:5154	HPGD	GuideToPharmacology	2024.1	inhibitor	0.070574827	IUPHAR.LIGAND:12972	ncit:C81529	DALCETRAPIB	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
RECEPTOR-INTERACTING PROTEIN 1	hgnc:10019	RIPK1	TTD	2020.06.01	NULL	26.25383561784724	GSK2982772	iuphar.ligand:9554	GSK2982772	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	inhibitor	0.030246354	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
UNIPROT:P00492	hgnc:5157	HPRT1	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.04344264	NVP-BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	GNF-PF-1295	chembl:CHEMBL579837	CHEMBL:CHEMBL579837	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	ONC1-13B	ncit:C148485	ANDROGEN RECEPTOR ANTAGONIST ONC1-0013B	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002358411	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.1100789753368857	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.033295923	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P02745	hgnc:1241	C1QA	TEND	1-Aug-11	NULL	52.50767123569449	IMMUNE GLOBULIN	ncit:C2701	THERAPEUTIC IMMUNE GLOBULIN	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:482	iuphar.ligand:482	HEAT (BE2254)	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1226814748497534	PHENDIMETRAZINE TARTRATE	rxcui:33272	PHENDIMETRAZINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	HYDROCORTISONE SODIUM PHOSPHATE	rxcui:235482	HYDROCORTISONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.061055432	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1204304386139782	CODEINE POLISTIREX	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.051027863	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.039097298	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	1.175544878411071	PF-03814735	drugbank:DB13059	PF-03814735	FALSE	FALSE	TRUE
PTK2	hgnc:9611	PTK2	TALC	12-May-16	inhibitor	0.09003373	PF-00562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.089298761	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:10452	iuphar.ligand:10452	NMRA-140	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.1312691780892362	IUPHAR.LIGAND:2020	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:1508	iuphar.ligand:1508	NPY-(2-36) (PIG)	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	N-PHENETHYL-NICOTINAMIDE	chembl:CHEMBL309848	CHEMBL:CHEMBL309848	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.020117882	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	MONOCILLIN I	chembl:CHEMBL215853	MONOCILLIN I	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	SJ000119988	chembl:CHEMBL589694	CHEMBL:CHEMBL589694	FALSE	FALSE	FALSE
NR1D1	hgnc:7962	NR1D1	DTC	9/2/20	NULL	17.50255707856483	GSK-4112	iuphar.ligand:2903	GSK4112	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.064033745	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
SCGB1A1	hgnc:12523	SCGB1A1	NCI	14-Sep-17	NULL	26.25383561784724	RHIGF-1	rxcui:274403	MECASERMIN	TRUE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:12320	iuphar.ligand:12320	SLC-391	FALSE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.2991890098899972	GDC-0032	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	0.106290832	IUPHAR.LIGAND:2448	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SKF-83565 HYDROBROMIDE	chembl:CHEMBL541585	CHEMBL:CHEMBL541585	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:2221	iuphar.ligand:2221	D(CH2)5[TYR(ME)2,THR4,TYR-NH29]OVT	FALSE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.6886251965336985	Norgestimate	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.065145994	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	0.3777530304726222	BAFETINIB	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	0.1458546423213736	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.002852903	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.072165573	Exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.00961679	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.023759127	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
PALB2	hgnc:26144	PALB2	CIViC	10-Apr-24	NULL	0.5966780822238011	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.2019525816757481	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DL2	hgnc:6330	KIR2DL2	TTD	2020.06.01	NULL	7.876150685354174	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.1204304386139782	MARAVIROC	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	GNF-PF-1134	chembl:CHEMBL600694	CHEMBL:CHEMBL600694	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.024932417	AZD1305	chembl:CHEMBL3545169	AZD1305	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.3977853881492007	MURAGLITAZAR	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.7395446652914718	ALACIZUMAB PEGOL	ncit:C61438	ALACIZUMAB PEGOL	FALSE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	1.875273972703375	RISANKIZUMAB	rxcui:2166040	RISANKIZUMAB	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:11510	iuphar.ligand:11510	M4205	FALSE	FALSE	FALSE
RPE65	hgnc:10294	RPE65	ChEMBL	33	inhibitor	7.501095891	EMIXUSTAT HYDROCHLORIDE	ncit:C171670	EMIXUSTAT HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1758	hgnc:2932	DMP1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:5051	ncit:C63958	RESIQUIMOD	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.100589408	AMPICILLIN TRIHYDRATE	rxcui:203115	AMPICILLIN TRIHYDRATE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	DTC	9/2/20	NULL	0.031254566	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002610374	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P05771	hgnc:9395	PRKCB	TdgClinicalTrial	Jan-14	NULL	0.2051080907644316	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
CYCSP5	hgnc:24416	CYCSP5	PharmGKB	4/5/24	NULL	2.917092846427472	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	ESTROGEN	chembl:CHEMBL592868	ESTROGEN	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.3889457128569962	MEPAZINE ACETATE	chembl:CHEMBL1712842	MEPAZINE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.063262255	IUPHAR.LIGAND:121	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.042276708	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
UNIPROT:P11473	hgnc:12679	VDR	TEND	1-Aug-11	NULL	0.1486416737033106	PARICALCITOL	rxcui:73710	PARICALCITOL	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.026385764	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.2917092846427472	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.006705961	VERAPAMIL HYDROCHLORIDE	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.008804103	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	POTASSIUM DICHROMATE	rxcui:8595	POTASSIUM DICHROMATE	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1591141552596802	DOLUTEGRAVIR SODIUM	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.016236138	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.0191914	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
KCNH3	hgnc:6252	KCNH3	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.1744440904840348	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	2.917092846427472	MACIMORELIN ACETATE	rxcui:1999419	MACIMORELIN ACETATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.021335909	doxycycline	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
AREG	hgnc:651	AREG	CIViC	10-Apr-24	NULL	0.5250767123569451	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	6-HYDROXYFLAVONE	chembl:CHEMBL138649	6-HYDROXYFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:227	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:1059	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1221108633388244	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:1389	iuphar.ligand:1389	YM298198	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1500219178162699	succimer	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	IPI-504	ncit:C48401	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	TRUE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.1773907812016706	IUPHAR.LIGAND:198	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	1,3-DIBENZYLTHIOUREA	chembl:CHEMBL1388908	CHEMBL:CHEMBL1388908	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.3125456621172291	benztropine	rxcui:1424	BENZTROPINE	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:1720	iuphar.ligand:1720	MRS2179	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.693795846312725	MEQUITAZINE	rxcui:29528	MEQUITAZINE	TRUE	FALSE	FALSE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.3750547945406749	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.9010915075351876	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3771	iuphar.ligand:3771	[125I]BH-NMB (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.052824619	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.7721716358190367	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1465330360065893	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	NCG-C00093990-01	chembl:CHEMBL1255966	CHEMBL:CHEMBL1255966	FALSE	FALSE	FALSE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.7160136986685613	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.078136416	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.029465584	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.4039051633514962	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:12515	iuphar.ligand:12515	DF3016A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	MECHLORETHAMINE HYDROCHLORIDE	rxcui:155036	MECHLORETHAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.1041818873724097	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.003944979	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	2.917092846427472	VS-6063	ncit:C79809	DEFACTINIB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1852122442176172	NERATINIB MALEATE	rxcui:1940642	NERATINIB MALEATE	TRUE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1875273972703375	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
THYROTROPIN-RELEASING HORMONE RECEPTOR	hgnc:12299	TRHR	TTD	2020.06.01	NULL	17.50255707856483	Protirelin	rxcui:10580	THYROTROPIN-RELEASING HORMONE	TRUE	FALSE	FALSE
NCBIGENE:2348	hgnc:3791	FOLR1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:6542	iuphar.ligand:6542	COMPOUND 1 [PMID: 11425539]	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.039688338	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.067403943	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:6557	iuphar.ligand:6557	RS-25344	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.108374966	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	INTERFERON ALPHA	chembl:CHEMBL2108506	INTERFERON ALFA	TRUE	FALSE	FALSE
UNIPROT:P40261	hgnc:7861	NNMT	TdgClinicalTrial	Jan-14	NULL	3.750547945406749	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Zalifrelimab	ncit:C126113	ZALIFRELIMAB	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	WAY-629	chembl:CHEMBL258465	CHEMBL:CHEMBL258465	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.009529523	FLUFENAMIC ACID	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.023060023	IUPHAR.LIGAND:6058	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
CXCR1	hgnc:6026	CXCR1	ChEMBL	33	inhibitor	3.750547945	NAVARIXIN	ncit:C156730	NAVARIXIN	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.2083637747448194	AZD1305	chembl:CHEMBL3545169	AZD1305	FALSE	FALSE	FALSE
TGFB2	hgnc:11768	TGFB2	ChEMBL	33	inhibitor	2.500365296937833	FRESOLIMUMAB	ncit:C63546	FRESOLIMUMAB	FALSE	FALSE	FALSE
NCBIGENE:2394	hgnc:3906	FRA5B	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:6498	iuphar.ligand:6498	WX-UK1	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:9569	iuphar.ligand:9569	ASP4058	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	6-METHYLFLAVONE	iuphar.ligand:12466	6-METHYLFLAVONE	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.033232703	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:P79483	hgnc:4951	HLA-DRB3	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	1D09C3	drugbank:DB05121	1D09C3	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.030281241	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8970	iuphar.ligand:8970	HUMAN GIP(3-42)NH2	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:3204	hgnc:5108	HOXA7	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:12138	iuphar.ligand:12138	MS8815	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.031032903	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	BRL-52537	chembl:CHEMBL1256835	CHEMBL:CHEMBL1256835	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.1286952726365061	Eltoprazine	ncit:C73286	ELTOPRAZINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	METHYLPARABEN	rxcui:29903	METHYLPARABEN	TRUE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	DTC	9/2/20	NULL	1.640864726115453	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	NSC-102045	chembl:CHEMBL483633	CHEMBL:CHEMBL483633	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TCMDC-123904	chembl:CHEMBL586061	CHEMBL:CHEMBL586061	FALSE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.051127236	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
POLE2	hgnc:9178	POLE2	ChEMBL	33	inhibitor	0.108040476	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.019896806	ALL-TRANS RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.031479419	IUPHAR.LIGAND:12575	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:11223	iuphar.ligand:11223	ISAM-140	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.082559232	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	0.8751278539282416	IUPHAR.LIGAND:2316	iuphar.ligand:2316	LEIUROTOXIN I	FALSE	FALSE	FALSE
NCBIGENE:2890	hgnc:4571	GRIA1	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:9137	iuphar.ligand:9137	NEOCEPTIN-3	FALSE	FALSE	FALSE
NCBIGENE:981	hgnc:23089	SLC13A5	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12851	iuphar.ligand:12851	ETG-5773	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC KAINATE 1	hgnc:4579	GRIK1	TTD	2020.06.01	NULL	1.432027397337122	Topiramate	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.029416062	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.2592971419046642	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.1088116604009326	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SMAD4	hgnc:6770	SMAD4	CIViC	10-Apr-24	NULL	0.2917092846427472	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.6482428547616604	CIDOFOVIR	rxcui:1546007	CIDOFOVIR ANHYDROUS	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006265458	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	E-GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	CIViC	10-Apr-24	NULL	0.1307787577476824	REPOTRECTINIB	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.078682824	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6074	iuphar.ligand:6074	M1160	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.210030685	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1341	iuphar.ligand:1341	PG-901	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:9585	iuphar.ligand:9585	AZ8838	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.027781837	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.2500365296937833	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	8.353493151133215	Lumacaftor	rxcui:1655922	LUMACAFTOR	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.015153729	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	4.039051633514961	Oxypurinol	ncit:C87294	OXYPURINOL	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	7.501095891	Peretinoin	ncit:C87202	PERETINOIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	BROMPERIDOL	rxcui:19777	BROMPERIDOL	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.3006164383722967	FLUOROMETHOLONE	rxcui:4491	FLUOROMETHOLONE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.023737645	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.032134438	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:6155	iuphar.ligand:6155	CP-195543	FALSE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:5530	iuphar.ligand:5530	COMPOUND 2 [PMID: 19230660]	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:6155	iuphar.ligand:6155	CP-195543	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:10110	iuphar.ligand:10110	PGN-9856	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:7839	iuphar.ligand:7839	ILGINATINIB	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	agonist	0.087952548	IUPHAR.LIGAND:1763	iuphar.ligand:1710	2MESADP	FALSE	FALSE	FALSE
NCBIGENE:1307	hgnc:2193	COL16A1	GuideToPharmacology	2024.1	inhibitor	0.1861974157294131	IUPHAR.LIGAND:4807	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:2442	hgnc:3840	FRA11E	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:8849	iuphar.ligand:8849	PEPTIDE LIGAND 2 [PMID: 19055415]	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:2778	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
CIC	hgnc:14214	CIC	CIViC	10-Apr-24	NULL	0.4861821410712454	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
NR1H3	hgnc:7966	NR1H3	ChEMBL	33	agonist	1.250182648468916	ROVAZOLAC	ncit:C152263	ROVAZOLAC	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.2419708351875322	NEZULCITINIB	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	TCMDC-125298	chembl:CHEMBL581152	CHEMBL:CHEMBL581152	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.00962384	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	1.193356164447602	cotinine	ncit:C70941	COTININE	FALSE	FALSE	FALSE
DELTA-LIKE PROTEIN 4	hgnc:2910	DLL4	TTD	2020.06.01	NULL	5.250767123569449	ABT-165	ncit:C116750	DILPACIMAB	FALSE	FALSE	FALSE
NME2	hgnc:7850	NME2	PharmGKB	4/5/24	NULL	0.4375639269641208	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	2.838252499226729	MK-869	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	1.029562181092048	TCMDC-125764	chembl:CHEMBL586670	CHEMBL:CHEMBL586670	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.045579576	CGP41251	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.2408608772279564	METHYLNALTREXONE BROMIDE	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.2453629496995069	MK-6913	chembl:CHEMBL3545274	MK-6913	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	0.8255923150266431	AMG 479	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
SRMS	hgnc:11298	SRMS	ChEMBL	33	inhibitor	0.4102161815288632	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	potentiator	0.4526523382387456	NAMINIDIL	ncit:C77076	NAMINIDIL	FALSE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TEND	1-Aug-11	NULL	1.666910197958555	AMINOCAPROIC ACID	rxcui:99	6-AMINOCAPROIC ACID	TRUE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:1096	iuphar.ligand:1096	[125I][TYR4]GHRELIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	blocker	0.2243917574174978	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.305277158	TCMDC-124530	chembl:CHEMBL582593	CHEMBL:CHEMBL582593	FALSE	FALSE	FALSE
NCBIGENE:2084	hgnc:6861	MAP3K9	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9355	iuphar.ligand:9355	GNE-3511	FALSE	FALSE	FALSE
NCBIGENE:3240	hgnc:5141	HP	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12814	iuphar.ligand:12814	GNE-7883	FALSE	FALSE	FALSE
MPST	hgnc:7223	MPST	NCI	14-Sep-17	NULL	8.751278539282415	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.039068208	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
CSNK1G3	hgnc:2456	CSNK1G3	DTC	9/2/20	NULL	0.1591141552596803	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1840222122746302	DESVENLAFAXINE SUCCINATE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.047518255	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1583941817064691	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:9099	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.1103102336884338	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1715936968486748	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.150021918	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.1458546423213736	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.5556367326528519	RO5083945	chembl:CHEMBL2109389	IMGATUZUMAB	FALSE	TRUE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	NECA	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.2243917574174978	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.088996053	TREQUINSIN HYDROCHLORIDE	chembl:CHEMBL1256910	TREQUINSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.081533651	IUPHAR.LIGAND:958	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.069454592	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O60840	hgnc:1393	CACNA1F	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	MK-6913	chembl:CHEMBL3545274	MK-6913	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.03729238	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1048	iuphar.ligand:1048	WKYMVM	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3197	iuphar.ligand:3197	COMPOUND 47 [PMID: 18800762]	FALSE	FALSE	FALSE
UNIPROT:Q9NSA0	hgnc:18120	SLC22A11	TEND	1-Aug-11	NULL	4.773424657790409	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.03319069	econazole	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	NCI	14-Sep-17	NULL	0.1202465753489187	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
SPSB2	hgnc:29522	SPSB2	PharmGKB	4/5/24	NULL	1.141471113819445	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.2734774543525755	PHENDIMETRAZINE	rxcui:33272	PHENDIMETRAZINE	TRUE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	blocker	0.2243917574174979	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12710	iuphar.ligand:12710	DOSIMERTINIB	FALSE	FALSE	FALSE
CUL4A	hgnc:2554	CUL4A	ChEMBL	33	inhibitor	0.3547815624033412	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
NCBIGENE:234	hgnc:4044	FZD6	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:10327	iuphar.ligand:10327	SAG1.3	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	agonist	0.087952548	IUPHAR.LIGAND:1710	iuphar.ligand:1710	2MESADP	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	0.4234489615781814	IUPHAR.LIGAND:1755	iuphar.ligand:1755	ADP&BETA;S	FALSE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.3977853881492006	HALOBETASOL PROPIONATE	rxcui:41208	HALOBETASOL	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.2263261691193728	GANCOTAMAB	ncit:C170020	GANCOTAMAB	FALSE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TdgClinicalTrial	Jan-14	NULL	0.4412409347537352	MECLOFENAMIC ACID	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
STAT1	hgnc:11362	STAT1	DTC	9/2/20	NULL	0.9723642821424908	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
NCBIGENE:2472	hgnc:3882	FRA20B	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:6646	rxcui:72937	TOLCAPONE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TOLUIC ACID	chembl:CHEMBL114957	TOLUIC ACID	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.039598545	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NSC-83217	chembl:CHEMBL120806	CHEMBL:CHEMBL120806	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	1.750255707856483	SULFONES	ncit:C849	SULFONE ANTI-INFECTIVE AGENT	FALSE	FALSE	FALSE
UNIPROT:P41594	hgnc:4597	GRM5	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	ADX10059	drugbank:DB05070	ADX10059	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.019929531	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	ESCULETIN	iuphar.ligand:5180	ESCULETIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003981473	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	3.500511415712966	ombitasvir / paritaprevir / ritonavir	wikidata:Q19858657	OMBITASVIR/PARITAPREVIR/RITONAVIR	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	NILVADIPINE	rxcui:53692	NILVADIPINE	FALSE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	0.2406768735020374	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	DTC	9/2/20	NULL	0.5834185692854945	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
NCBIGENE:3082	hgnc:4893	HGF	GuideToPharmacology	2024.1	NULL	1.944728564284981	IUPHAR.LIGAND:10363	iuphar.ligand:10363	BT-11	FALSE	FALSE	FALSE
NCBIGENE:2985	hgnc:3621	FCGRT	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:9959	iuphar.ligand:9959	DX-2507	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:1378	iuphar.ligand:1378	LY341495	FALSE	FALSE	FALSE
NCBIGENE:1014	hgnc:1755	CDH16	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8890	iuphar.ligand:8890	COMPOUND 9 [PMID: 15615544]	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.012878997	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
NCBIGENE:347	hgnc:612	APOD	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:9255	iuphar.ligand:9255	F16357	FALSE	FALSE	FALSE
RBX1	hgnc:9928	RBX1	PharmGKB	4/5/24	NULL	0.1260688385010672	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	2.100306849	9Z-RETINOIC ACID	chembl:CHEMBL451158	CHEMBL:CHEMBL451158	FALSE	FALSE	FALSE
HIST4H4	hgnc:20510	H4C16	NCI	14-Sep-17	NULL	2.625383561784725	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	0.03409589	Ebselen	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.049256727	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007866318	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
TNIK	hgnc:30765	TNIK	DTC	9/2/20	NULL	2.917092846427472	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	1.381780822	NITD609	ncit:C169853	CIPARGAMIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	4-HYDROXYFLAVONOL	chembl:CHEMBL272682	CHEMBL:CHEMBL272682	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	GRINIMIBINE	chembl:CHEMBL1477760	GRINIMIBINE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.014354202	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002542744	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
EYA1	hgnc:3519	EYA1	PharmGKB	4/5/24	NULL	0.1489579325835304	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1750255707856483	HARMAN	chembl:CHEMBL12014	HARMAN	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.036237178	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	0.5556367326528519	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	modulator	0.4884434533552977	SUVECALTAMIDE	ncit:C174710	SUVECALTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	NULL	0.42006137	IUPHAR.LIGAND:4505	iuphar.ligand:4505	[3H]BSP	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006182465	fluticasone propionate	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.067317527	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
CDKN1B	hgnc:1785	CDKN1B	CIViC	10-Apr-24	NULL	0.094099769	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.019461702	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
CDC25C	hgnc:1727	CDC25C	NCI	14-Sep-17	NULL	0.2206204673768676	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.2169738480813822	propafenone	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.201178817	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	CIViC	10-Apr-24	NULL	0.3906820776465364	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	inhibitor	0.046549354	IUPHAR.LIGAND:4807	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.09869863	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.018359326	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	ZOLANTIDINE	chembl:CHEMBL419296	ZOLANTIDINE	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.01741548	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:11274	iuphar.ligand:11274	GSK'547	FALSE	FALSE	FALSE
MTRR	hgnc:7473	MTRR	NCI	14-Sep-17	NULL	3.000438356325399	VITAMIN B12	rxcui:11248	VITAMIN B12	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SJ000113107	chembl:CHEMBL589245	CHEMBL:CHEMBL589245	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.364636606	LAROTRECTINIB SULFATE	rxcui:2104548	LAROTRECTINIB SULFATE	TRUE	FALSE	FALSE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	blocker	0.2243917574174979	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.080781033	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2269	iuphar.ligand:2269	BAY 55-9837	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7810	iuphar.ligand:7810	COMPOUND 2 [PMID: 25408830]	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010629083	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.008585296	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	ChEMBL	33	inhibitor	0.9376369863516875	AVAGACESTAT	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.1691976516724849	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	agonist	0.1286952726365061	FENFLURAMINE HYDROCHLORIDE	rxcui:82018	FENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BACE1	hgnc:933	BACE1	ChEMBL	33	inhibitor	1.346350544504987	VERUBECESTAT	ncit:C152868	VERUBECESTAT	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.038104261	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.1097339001790898	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	MyCancerGenome	20-Jun-17	antibody	5.834185692854944	IBRITUMOMAB TIUXETAN	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.064824285	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
IL4	hgnc:6014	IL4	PharmGKB	4/5/24	NULL	0.1489579325835304	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.054695491	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
UNIPROT:P27361	hgnc:6877	MAPK3	TdgClinicalTrial	Jan-14	NULL	0.1415301111474245	RDEA119	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.2706580991530644	IUPHAR.LIGAND:5598	iuphar.ligand:5598	CP608,039	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:8191	iuphar.ligand:8191	COMPOUND 18 [PMID: 20873740]	FALSE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3964	iuphar.ligand:3964	&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:7114	rxcui:236612	ANAGRELIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.050597611	Brexpiprazole	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:342	iuphar.ligand:342	BRUCINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	MK-571	iuphar.ligand:10346	MK-571	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.3977853881492006	DENBUFYLLINE	ncit:C76316	DENBUFYLLINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.019889269	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
RXFP2	hgnc:17318	RXFP2	DTC	9/2/20	NULL	1.093909817410302	N6-CYCLOPENTYLADENOSINE	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.1108075556053025	GLEEVEC	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3194	iuphar.ligand:3194	COMPOUND 14 [PMID: 18800762]	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	TRYPAN BLUE	rxcui:10878	TRYPAN BLUE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	TCMDC-123480	chembl:CHEMBL588683	CHEMBL:CHEMBL588683	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005905046	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.040682597	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	1.009762908	REMTOLUMAB	ncit:C152189	REMTOLUMAB	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.030959712	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:755	iuphar.ligand:755	CCL23	FALSE	FALSE	FALSE
NCBIGENE:2499	hgnc:3991	FTH1P4	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:2844	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10218	iuphar.ligand:10218	COMPOUND 27D [PMID: 28231433]	FALSE	FALSE	FALSE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	0.364636606	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.008394512	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	METHOXYVONE	chembl:CHEMBL1591080	METHOXYVONE	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:2787	iuphar.ligand:2787	LG190178	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.6775183385250904	STEEL FACTOR	ncit:C1410	RECOMBINANT HUMAN STEM CELL FACTOR	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.027840759	NDGA	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.001351375	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	1.050153425	cannabinoids	chembl:CHEMBL3833333	NABIXIMOLS	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.1773907812016706	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004919212	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	DTC	9/2/20	NULL	0.4861821410712453	ALENDRONIC ACID	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9315	iuphar.ligand:9315	B-TPMF	FALSE	FALSE	FALSE
NCBIGENE:545	hgnc:882	ATR	GuideToPharmacology	2024.1	blocker	0.038894571	IUPHAR.LIGAND:2406	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:8839	iuphar.ligand:8839	TORIN 2	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	Ganitumab	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.3431873936973496	AG-024322	ncit:C52182	CDK1/2/4 INHIBITOR AG-024322	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.03409589	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.5147810905460245	DOCOSAPENTAENOIC ACID	chembl:CHEMBL496634	DOCOSAPENTAENOIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003100908	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
AIFM1	hgnc:8768	AIFM1	NCI	14-Sep-17	NULL	5.250767124	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
MARCKSL1	hgnc:7142	MARCKSL1	NCI	14-Sep-17	NULL	0.921187215	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.252440727	ASENAPINE MALEATE	rxcui:860647	ASENAPINE MALEATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.133607306	HALCINONIDE	rxcui:5084	HALCINONIDE	TRUE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	5.250767123569449	CVX-060	chembl:CHEMBL4594470	CVX-060	FALSE	FALSE	TRUE
CHAT	hgnc:1912	CHAT	NCI	14-Sep-17	NULL	0.4167275494896388	SODIUM CHLORIDE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	0.084146909	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:12143	iuphar.ligand:12143	WNY0824	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:8245	iuphar.ligand:8245	ZM-306416	FALSE	FALSE	FALSE
PROTEIN KINASE C ALPHA	hgnc:9393	PRKCA	TTD	2020.06.01	NULL	0.1215455352678113	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:10082	ncit:C171711	FIRUGLIPEL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.002904025	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
LGALS8	hgnc:6569	LGALS8	DTC	9/2/20	NULL	35.00511415712966	LACTOSE, ANHYDROUS	chembl:CHEMBL417016	LACTOSE, ANHYDROUS	FALSE	FALSE	FALSE
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	0.3125456621172291	Urokinase	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.04636439	ZINC CHLORIDE	rxcui:39937	ZINC CHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.4605936073306534	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	BUSPIRONE HYDROCHLORIDE	rxcui:203116	BUSPIRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2778183663264259	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
FK506-BINDING PROTEIN 1A	hgnc:3711	FKBP1A	TTD	2020.06.01	NULL	8.751278539282415	GPI-1485	drugbank:DB05814	GPI-1485	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.027010119	zafirlukast	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	0.4735540335109532	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.006375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CancerCommons	25-Jul-13	inhibitor	3.500511415712966	ARQ 197	ncit:C62437	TIVANTINIB	FALSE	FALSE	TRUE
HSPB1	hgnc:5246	HSPB1	CancerCommons	25-Jul-13	inhibitor	4.375639269641208	OGX-427	ncit:C71740	APATORSEN	FALSE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CGI	2/1/22	NULL	NULL	Platinum Agent	NULL	NULL	NULL	NULL	NULL
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1041818873724097	AZD-8186	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	CGI	2/1/22	NULL	NULL	Platinum Agent	NULL	NULL	NULL	NULL	NULL
BRCA2	hgnc:1101	BRCA2	CGI	2/1/22	NULL	0.3860858179095183	Veliparib	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.4487835148349957	CLEBOPRIDE	rxcui:21224	CLEBOPRIDE	TRUE	FALSE	FALSE
CBL	hgnc:1541	CBL	CGI	2/1/22	NULL	0.1022876712383659	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.9010915075351876	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	NULL	LHRH analogues or antagonist	NULL	NULL	NULL	NULL	NULL
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	NULL	LHRH analogues or antagonist	NULL	NULL	NULL	NULL	NULL
MKNK1	hgnc:7110	MKNK1	ChEMBL	33	inhibitor	26.25383561784724	TOMIVOSERTIB	ncit:C125062	TOMIVOSERTIB	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	CGI	2/1/22	NULL	0.2944355396394084	Lucitanib	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
GNAQ	hgnc:4390	GNAQ	CGI	2/1/22	NULL	4.773424657790409	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
GNA11	hgnc:4379	GNA11	CGI	2/1/22	NULL	1.750255707856483	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	CGI	2/1/22	NULL	0.007390242	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	CGI	2/1/22	NULL	1.494525746746522	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	R1295	drugbank:DB05122	R1295	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.013179636	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
MLL	hgnc:7132	KMT2A	CGI	2/1/22	NULL	1.640864726115453	EPZ-5676	ncit:C103179	PINOMETOSTAT	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.091159151	MEK inhibitor	ncit:C69145	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	FALSE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.0296486	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
LRP1B	hgnc:6693	LRP1B	CGI	2/1/22	NULL	4.375639269641208	Liposomal Doxorubicin	wikidata:Q29004943	CAELYX	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	CGI	2/1/22	NULL	0.043629141	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005899738	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	0.760980743	ET-1	iuphar.ligand:989	ENDOTHELIN-1	FALSE	FALSE	FALSE
TSC1	hgnc:12362	TSC1	CGI	2/1/22	NULL	2.625383561784725	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
TRHR	hgnc:12299	TRHR	ChEMBL	33	agonist	17.50255707856483	PROTIRELIN	rxcui:10580	THYROTROPIN-RELEASING HORMONE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	DESLORATADINE	rxcui:275635	DESLORATADINE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.4565884455277783	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	2.917092846427472	CHLOROTHIAZIDE SODIUM	rxcui:91217	CHLOROTHIAZIDE SODIUM	TRUE	FALSE	FALSE
SLC12A1	hgnc:10910	SLC12A1	ChEMBL	33	inhibitor	7.501095891	ETHACRYNATE SODIUM	rxcui:4108	ETHACRYNATE SODIUM	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.596678082	LEVOBETAXOLOL HYDROCHLORIDE	rxcui:261718	LEVOBETAXOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.6945459158160648	NIMOTUZUMAB	ncit:C2733	NIMOTUZUMAB	FALSE	TRUE	TRUE
EMBA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ETHAMBUTOL HYDROCHLORIDE	rxcui:142435	ETHAMBUTOL HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	0.3241214273808303	CHLORTHALIDONE	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.038187397	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003405608	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.043629141	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	VENLAFAXINE HYDROCHLORIDE	rxcui:235988	VENLAFAXINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.640864726115453	CANAGLIFLOZIN	rxcui:1373458	CANAGLIFLOZIN	TRUE	FALSE	FALSE
CA4	hgnc:1375	CA4	ChEMBL	33	inhibitor	0.6250913242344582	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
GLP2R	hgnc:4325	GLP2R	ChEMBL	33	agonist	13.12691780892362	TEDUGLUTIDE	rxcui:1364468	TEDUGLUTIDE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	agonist	0.038159645	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.8607814956671229	DESOGESTREL	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.034727296	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:3285	iuphar.ligand:3285	PSB36	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.024354207	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.033295923	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:997	iuphar.ligand:997	BQ123	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.031631127	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.042863405	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.1944728564284981	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.1346350544504987	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.03043923	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.1682938180631233	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.1056492378987816	TETRAHYDROZOLINE HYDROCHLORIDE	rxcui:57983	TETRAHYDROZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.1056492378987816	NAPHAZOLINE HYDROCHLORIDE	rxcui:82054	NAPHAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.078136416	NAPHAZOLINE HYDROCHLORIDE	rxcui:82054	NAPHAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.046965717	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.070129236	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.052142673	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.09745299	NANDROLONE PHENPROPIONATE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	modulator	0.1256164383629055	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2907401508067248	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMPIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.760980743	Gandotinib	ncit:C116857	GANDOTINIB	FALSE	FALSE	TRUE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMPIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMPIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMPIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFABUTIN	rxcui:55672	RIFABUTIN	TRUE	FALSE	FALSE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFABUTIN	rxcui:55672	RIFABUTIN	TRUE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFABUTIN	rxcui:55672	RIFABUTIN	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	0.096264064	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFABUTIN	rxcui:55672	RIFABUTIN	TRUE	FALSE	FALSE
COL6A3	hgnc:2213	COL6A3	ChEMBL	33	cleavage	0.3454452054979901	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
COL4A4	hgnc:2206	COL4A4	ChEMBL	33	cleavage	0.4605936073306535	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
MARK4	hgnc:13538	MARK4	DTC	9/2/20	NULL	0.1591141552596803	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
COL5A3	hgnc:14864	COL5A3	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
PBP1A	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN	rxcui:26797	HETACILLIN	TRUE	FALSE	FALSE
PBP1B	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN	rxcui:26797	HETACILLIN	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.013159817	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
PBP2A	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN	rxcui:26797	HETACILLIN	TRUE	FALSE	FALSE
PBP2B	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN	rxcui:26797	HETACILLIN	TRUE	FALSE	FALSE
PBP2X	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN	rxcui:26797	HETACILLIN	TRUE	FALSE	FALSE
PBP3	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN	rxcui:26797	HETACILLIN	TRUE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 2	hgnc:6871	MAPK1	TTD	2020.06.01	NULL	0.016669102	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.2302968036653267	TOLTERODINE TARTRATE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.096167896	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.089298761	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.047886613	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.048083948	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	BUSPIRONE HYDROCHLORIDE	rxcui:203116	BUSPIRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.030527716	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.038608582	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.093763699	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.083257407	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.01924768	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	OncoKB	23-Jul-20	NULL	0.3314878234576672	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXALACTAM DISODIUM	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXALACTAM DISODIUM	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXALACTAM DISODIUM	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXALACTAM DISODIUM	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXALACTAM DISODIUM	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXALACTAM DISODIUM	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXALACTAM DISODIUM	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIZOXIME SODIUM	rxcui:82126	CEFTIZOXIME SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIZOXIME SODIUM	rxcui:82126	CEFTIZOXIME SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIZOXIME SODIUM	rxcui:82126	CEFTIZOXIME SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIZOXIME SODIUM	rxcui:82126	CEFTIZOXIME SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIZOXIME SODIUM	rxcui:82126	CEFTIZOXIME SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIZOXIME SODIUM	rxcui:82126	CEFTIZOXIME SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIZOXIME SODIUM	rxcui:82126	CEFTIZOXIME SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.09699693	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERTAPENEM SODIUM	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERTAPENEM SODIUM	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERTAPENEM SODIUM	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.051511777	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CGI	2/1/22	NULL	0.088866948	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	ChEMBL	33	inhibitor	0.1250182648468916	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	modulator	0.036692992	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	modulator	0.1944728564284981	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	modulator	0.1296485709523321	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	modulator	0.1944728564284981	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	modulator	0.045226246	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.062139256	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.045898314	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.065145994	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.159436249	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.068458502	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.069454592	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.068369364	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.050488145	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.055155117	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.044763573	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.027635616	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR1	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR2	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB1	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB2	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG1	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG2	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMB1	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMB2	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMG1	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMG2	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.4070362111294147	METHSUXIMIDE	rxcui:47858	METHSUXIMIDE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.1465330360065893	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
MME	hgnc:7154	MME	ChEMBL	33	inhibitor	4.773424657790408	SACUBITRIL	rxcui:1656328	SACUBITRIL	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.2734774543525755	PARITAPREVIR	rxcui:1597373	PARITAPREVIR	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.1166837138570989	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.2917092846427472	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
PSMA6	hgnc:9535	PSMA6	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMA5	hgnc:9534	PSMA5	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.046965717	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.02804897	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.051782713	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.032055965	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.049256727	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.049302978	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
PRKACG	hgnc:9382	PRKACG	ChEMBL	33	inhibitor	3.088686543276147	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.096521454	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
PRKCH	hgnc:9403	PRKCH	ChEMBL	33	inhibitor	0.280789686	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
PRKCB	hgnc:9395	PRKCB	ChEMBL	33	inhibitor	0.1930429089547592	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.097962073	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.2430910705356226	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1223955040459079	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	ChEMBL	33	inhibitor	1.250182648468916	BRICICLIB	ncit:C141431	BRICICLIB	FALSE	FALSE	FALSE
FZD2	hgnc:4040	FZD2	ChEMBL	33	inhibitor	3.750547945406749	VANTICTUMAB	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
MLNR	hgnc:4495	MLNR	ChEMBL	33	agonist	10.50153424713889	ATILMOTIN	ncit:C77604	ATILMOTIN	FALSE	FALSE	FALSE
FZD1	hgnc:4038	FZD1	ChEMBL	33	inhibitor	1.875273972703374	VANTICTUMAB	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	ChEMBL	33	inhibitor	0.039899446	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1875273972703375	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1041818873724097	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1764963739014941	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.075732218	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PRKCG	hgnc:9402	PRKCG	ChEMBL	33	inhibitor	0.1141471113819445	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	ChEMBL	33	inhibitor	0.2187819634820604	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.1630673019742065	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	ChEMBL	33	inhibitor	0.065634589	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	inhibitor	0.3889457128569962	ODELEPRAN	chembl:CHEMBL2103878	ODELEPRAN	FALSE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	1.193356164447602	LEMBOREXANT	rxcui:2272403	LEMBOREXANT	TRUE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	negative modulator	2.917092846427472	AZD2516	chembl:CHEMBL3545346	AZD2516	FALSE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	ChEMBL	33	inhibitor	0.9376369863516875	PRATOSARTAN	ncit:C72935	PRATOSARTAN	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	inhibitor	1.750255707856483	SURINABANT	ncit:C87598	SURINABANT	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	1.419126249613364	VOFOPITANT	ncit:C72949	VOFOPITANT	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	inhibitor	0.2536602475154323	RELCOVAPTAN	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	FRAKEFAMIDE	ncit:C77290	FRAKEFAMIDE	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.1209854175937661	GW468816	chembl:CHEMBL1207366	GW468816	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.1861974157294131	AZD1305	chembl:CHEMBL3545169	AZD1305	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	3.281729452230906	CNV2197944	chembl:CHEMBL3545172	CNV2197944	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	3.424413341458336	SSR180711	chembl:CHEMBL559478	SSR180711	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.5357925636295356	TRAXOPRODIL	ncit:C87769	TRAXOPRODIL	FALSE	FALSE	FALSE
KCNA4	hgnc:6222	KCNA4	ChEMBL	33	blocker	0.150021918	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.017799211	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.016408647	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNC4	hgnc:6236	KCNC4	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.033875917	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.016669102	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1481697953740938	OSIMERTINIB	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.2520944435184235	PACRITINIB	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1458546423213736	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	3.000438356	FOSTAMATINIB	rxcui:2044896	FOSTAMATINIB	TRUE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.1250182648468916	SARIZOTAN HYDROCHLORIDE	ncit:C76654	SARIZOTAN HYDROCHLORIDE	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.084146909	ESMIRTAZAPINE MALEATE	ncit:C76940	ESMIRTAZAPINE MALEATE	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	inverse agonist	2.333674277141977	TARANABANT	ncit:C81420	TARANABANT	FALSE	FALSE	FALSE
PTGIR	hgnc:9602	PTGIR	ChEMBL	33	agonist	3.750547945	ESUBERAPROST	ncit:C166506	ESUBERAPROST	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.1204304386139782	NALDEMEDINE	rxcui:1876597	NALDEMEDINE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.064347636	ESMIRTAZAPINE MALEATE	ncit:C76940	ESMIRTAZAPINE MALEATE	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.070956312	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	1.009762908	IFERANSERIN	ncit:C90945	IFERANSERIN	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	modulator	0.6226206075378794	PRIDOPIDINE	ncit:C170349	PRIDOPIDINE	FALSE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	activator	0.729273212	FLINDOKALNER	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.064505739	DICYCLOMINE HYDROCHLORIDE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	activator	0.6563458904461812	FLINDOKALNER	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
MMP12	hgnc:7158	MMP12	ChEMBL	33	inhibitor	0.3889457128569963	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	inhibitor	0.5585922471882393	DEXMECAMYLAMINE	ncit:C166871	DEXMECAMYLAMINE	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.042344896	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.042344896	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.044498026	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.041672755	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
NGF	hgnc:7808	NGF	ChEMBL	33	inhibitor	3.750547945	FULRANUMAB	ncit:C84838	FULRANUMAB	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	1.372749574789398	PATRITUMAB	ncit:C78853	PATRITUMAB	FALSE	TRUE	TRUE
CD33	hgnc:1659	CD33	ChEMBL	33	other/unknown	8.078103267029922	LINTUZUMAB	ncit:C1716	LINTUZUMAB	FALSE	FALSE	FALSE
TGFB2	hgnc:11768	TGFB2	ChEMBL	33	inhibitor	15.00219178	LERDELIMUMAB	ncit:C170107	LERDELIMUMAB	FALSE	FALSE	FALSE
HTR6	hgnc:5301	HTR6	ChEMBL	33	inhibitor	8.751278539282417	INTEPIRDINE	ncit:C166572	INTEPIRDINE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.041672755	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.042174836	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	negative modulator	0.042174836	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	negative modulator	0.038894571	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.03151721	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	0.760980743	TROPIFEXOR	ncit:C152764	TROPIFEXOR	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.037213091	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	negative modulator	0.041672755	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.036770078	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	ChEMBL	33	inhibitor	6.563458904461812	LITRONESIB	ncit:C88328	LITRONESIB	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	modulator	0.2302968036653267	ERTUMAXOMAB	ncit:C2658	ERTUMAXOMAB	FALSE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	AD-159	chembl:CHEMBL2109444	AD-159	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFADIMETHOXINE	rxcui:10172	SULFADIMETHOXINE	TRUE	FALSE	FALSE
CPT1B	hgnc:2329	CPT1B	ChEMBL	33	inhibitor	0.1403948428761885	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	blocker	0.2019525816757481	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	blocker	0.096167896	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	blocker	0.1553481397505754	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	inhibitor	0.079197091	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	blocker	0.2243917574174979	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	blocker	0.2243917574174979	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	ChEMBL	33	inhibitor	0.1029562181092049	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.02271093	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	inhibitor	14.58546423213736	EPRATUZUMAB	ncit:C1887	EPRATUZUMAB	FALSE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	ChEMBL	33	agonist	11.66837138570988	APOMAB	ncit:C71693	APOMAB	FALSE	TRUE	TRUE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	binder	1.944728564284981	J591 177LU	chembl:CHEMBL2109559	J591 177LU	FALSE	FALSE	FALSE
G	NULL	NULL	ChEMBL	33	inhibitor	NULL	CL-184	chembl:CHEMBL2109564	CL-184	FALSE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	0.084146909	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	IDRAPARINUX	drugbank:DB06406	IDRAPARINUX	FALSE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.1442518440541058	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	0.2430910705356227	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.042898424	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEDI-564	chembl:CHEMBL2109567	MEDI-564	FALSE	FALSE	FALSE
CD44	hgnc:1681	CD44	ChEMBL	33	binder	2.763561643983921	BIVATUZUMAB	ncit:C175749	BIVATUZUMAB	FALSE	FALSE	FALSE
PCRV	NULL	NULL	ChEMBL	33	inhibitor	NULL	KB-001	chembl:CHEMBL2109536	KB-001	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:171	iuphar.ligand:171	ORG-37684	FALSE	FALSE	FALSE
GB	NULL	NULL	ChEMBL	33	inhibitor	NULL	REGAVIRUMAB	ncit:C188625	REGAVIRUMAB	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	FELVIZUMAB	ncit:C188649	FELVIZUMAB	FALSE	FALSE	FALSE
BLAT-3	NULL	NULL	ChEMBL	33	inhibitor	NULL	RELEBACTAM	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
BLAT-4	NULL	NULL	ChEMBL	33	inhibitor	NULL	RELEBACTAM	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:191	iuphar.ligand:191	SB 221284	FALSE	FALSE	FALSE
BLAT-5	NULL	NULL	ChEMBL	33	inhibitor	NULL	RELEBACTAM	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
BLAT-6	NULL	NULL	ChEMBL	33	inhibitor	NULL	RELEBACTAM	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.092443083	AVIPTADIL	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.100976291	AVIPTADIL	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	SOVAPREVIR	ncit:C152411	SOVAPREVIR	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.095122593	AVIPTADIL	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
SLAMF7	hgnc:21394	SLAMF7	ChEMBL	33	binder	2.187819634820604	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1981421556063943	NILVADIPINE	rxcui:53692	NILVADIPINE	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.2500365296937833	NILVADIPINE	rxcui:53692	NILVADIPINE	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADALBUVIR	ncit:C152141	RADALBUVIR	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	ChEMBL	33	inhibitor	2.386712328895204	ZIMLOVISERTIB	ncit:C185226	ZIMLOVISERTIB	FALSE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	positive modulator	1.009762908	OLINCIGUAT	ncit:C153148	OLINCIGUAT	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2917092846427472	TETOMILAST	ncit:C90922	TETOMILAST	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
GRM3	hgnc:4595	GRM3	PharmGKB	4/5/24	NULL	0.2351089756822141	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PHENETHICILLIN	rxcui:33277	PHENETHICILLIN	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PHENETHICILLIN	rxcui:33277	PHENETHICILLIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PHENETHICILLIN	rxcui:33277	PHENETHICILLIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PHENETHICILLIN	rxcui:33277	PHENETHICILLIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PHENETHICILLIN	rxcui:33277	PHENETHICILLIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PHENETHICILLIN	rxcui:33277	PHENETHICILLIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PHENETHICILLIN	rxcui:33277	PHENETHICILLIN	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMOCILLIN	rxcui:37775	TEMOCILLIN	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMOCILLIN	rxcui:37775	TEMOCILLIN	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMOCILLIN	rxcui:37775	TEMOCILLIN	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMOCILLIN	rxcui:37775	TEMOCILLIN	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMOCILLIN	rxcui:37775	TEMOCILLIN	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMOCILLIN	rxcui:37775	TEMOCILLIN	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMOCILLIN	rxcui:37775	TEMOCILLIN	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOXACILLIN	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAVIDASVIR	ncit:C152158	RAVIDASVIR	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	MERICITABINE	ncit:C98959	MERICITABINE	FALSE	FALSE	FALSE
TTR	hgnc:12405	TTR	ChEMBL	33	modulator	4.375639269641208	ACORAMIDIS	ncit:C170791	ACORAMIDIS	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEMONOXACIN	ncit:C174838	NEMONOXACIN	FALSE	FALSE	FALSE
PA	hgnc:8549	BLOC1S6	ChEMBL	33	inhibitor	17.50255707856483	BALOXAVIR	rxcui:2197842	BALOXAVIR	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	TESOFENSINE	ncit:C66589	TESOFENSINE	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	TESOFENSINE	ncit:C66589	TESOFENSINE	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	ALX-0171	chembl:CHEMBL4297692	ALX-0171	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.1221108633388244	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
ASGR1	hgnc:742	ASGR1	ChEMBL	33	binder	3.750547945	VUPANORSEN SODIUM	ncit:C174943	VUPANORSEN SODIUM	FALSE	FALSE	FALSE
TCDA	NULL	NULL	ChEMBL	33	binder	NULL	TOLEVAMER SODIUM	chembl:CHEMBL2108872	TOLEVAMER SODIUM	FALSE	FALSE	FALSE
TCDB	NULL	NULL	ChEMBL	33	binder	NULL	TOLEVAMER SODIUM	chembl:CHEMBL2108872	TOLEVAMER SODIUM	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	BALAPIRAVIR	ncit:C87439	BALAPIRAVIR	FALSE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.8078103267029924	ATACIGUAT	ncit:C79587	ATACIGUAT	FALSE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.6177373086552295	ATACIGUAT	ncit:C79587	ATACIGUAT	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.036770078	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.03151721	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
GLP2R	hgnc:4325	GLP2R	ChEMBL	33	agonist	13.12691780892362	FE 203799	chembl:CHEMBL4563522	FE 203799	FALSE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	ChEMBL	33	inhibitor	5.834185692854944	ACEBILUSTAT	ncit:C169757	ACEBILUSTAT	FALSE	FALSE	FALSE
ICOS	hgnc:5351	ICOS	ChEMBL	33	agonist	35.00511415712966	VOPRATELIMAB	ncit:C129876	VOPRATELIMAB	FALSE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	agonist	2.187819634820604	CDX-1140	chembl:CHEMBL4297721	CDX-1140	FALSE	FALSE	FALSE
NPR2	hgnc:7944	NPR2	ChEMBL	33	agonist	2.917092846427472	CARPERITIDE	ncit:C169829	CARPERITIDE	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ZOLIFLODACIN	ncit:C152962	ZOLIFLODACIN	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ZOLIFLODACIN	ncit:C152962	ZOLIFLODACIN	FALSE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	ALBACONAZOLE	ncit:C72952	ALBACONAZOLE	FALSE	FALSE	FALSE
TGFA	hgnc:11765	TGFA	ChEMBL	33	inhibitor	6.563458904461812	FEPIXNEBART	ncit:C188574	FEPIXNEBART	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	ChEMBL	33	inhibitor	0.3977853881492007	PRI-724	drugbank:DB15034	PRI-724	FALSE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	ChEMBL	33	inhibitor	0.5357925636295356	CTS-1027	drugbank:DB08490	CTS-1027	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	EDRALBRUTINIB	ncit:C175775	EDRALBRUTINIB	FALSE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	2.019525817	VUNAKIZUMAB	ncit:C152923	VUNAKIZUMAB	FALSE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	agonist	1.500219178	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	1.853211925965688	SOCAZOLIMAB	ncit:C162504	SOCAZOLIMAB	FALSE	FALSE	FALSE
IL18R1	hgnc:5988	IL18R1	ChEMBL	33	agonist	17.50255707856483	IBOCTADEKIN	ncit:C1680	IBOCTADEKIN	FALSE	FALSE	FALSE
EEF2	hgnc:3214	EEF2	ChEMBL	33	inhibitor	1.458546423213736	RESIMMUNE	chembl:CHEMBL4297555	RESIMMUNE	FALSE	FALSE	FALSE
IMPDH2	hgnc:6053	IMPDH2	ChEMBL	33	inhibitor	2.625383561784724	MYCOPHENOLATE SODIUM	rxcui:408142	MYCOPHENOLATE SODIUM	TRUE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	0.7001022831425933	E-7016	chembl:CHEMBL3527000	E-7016	FALSE	FALSE	FALSE
IL10RB	hgnc:5965	IL10RB	ChEMBL	33	agonist	8.751278539282415	EFLEPEDOCOKIN ALFA	ncit:C141419	EFLEPEDOCOKIN ALFA	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.068637479	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.037213091	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	vaccine	NULL	ABDAVOMERAN	ncit:C173052	ABDAVOMERAN	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	REGDANVIMAB	ncit:C177084	REGDANVIMAB	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	CASIRIVIMAB	rxcui:2465242	CASIRIVIMAB	TRUE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	vaccine	NULL	CX-024414	chembl:CHEMBL4650491	CX-024414	FALSE	FALSE	FALSE
S1PR2	hgnc:3169	S1PR2	ChEMBL	33	binder	1.500219178	FINGOLIMOD LAURYL SULFATE	rxcui:2610292	FINGOLIMOD LAURYL SULFATE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.081533651	NEZULCITINIB	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	NULL	RAFAMETINIB	NULL	NULL	NULL	NULL	NULL
CCND2	hgnc:1583	CCND2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.5527123287967842	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3070624048871023	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
CCND3	hgnc:1585	CCND3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.5527123287967842	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.087952548	ROBINETIN	chembl:CHEMBL170405	ROBINETIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2917092846427472	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	NULL	RAFAMETINIB	NULL	NULL	NULL	NULL	NULL
NF1	hgnc:7765	NF1	ClearityFoundationBiomarkers	26-Jul-13	NULL	NULL	RAFAMETINIB	NULL	NULL	NULL	NULL	NULL
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1324279224103266	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1154014752432846	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.066213961	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.364636606	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.088695391	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
NCBIGENE:1994	hgnc:3312	ELAVL1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8074	iuphar.ligand:8074	NG-25	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1374032518317239	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
IL-12A	hgnc:5969	IL12A	ClearityFoundationClinicalTrial	15-Jun-13	other/unknown	2.625383561784724	CID 446414	drugbank:DB05953	EGEN-001	FALSE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2853677784548614	LY2228820	ncit:C105853	RALIMETINIB MESYLATE	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	COSMIC	4-Sep-20	NULL	NULL	Tyrosine kinase inhibitor - NS	NULL	NULL	NULL	NULL	NULL
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3983	iuphar.ligand:3983	&ALPHA;-CONOTOXIN GI	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	COSMIC	4-Sep-20	NULL	NULL	Tyrosine kinase inhibitor - NS	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	COSMIC	4-Sep-20	NULL	0.179119736	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	COSMIC	4-Sep-20	NULL	1.184383561707394	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.007292732	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.092606122	IUPHAR.LIGAND:3482	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1640864726115453	TRYPAN BLUE	rxcui:10878	TRYPAN BLUE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	XANTHONE	chembl:CHEMBL186784	XANTHONE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.4412409347537352	STILONIUM IODIDE	ncit:C73168	STILONIUM IODIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	(R,S)-IFENPRODIL	chembl:CHEMBL49623	(R,S)-IFENPRODIL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	TCMDC-125319	chembl:CHEMBL527586	CHEMBL:CHEMBL527586	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	3-(DIMETHYLAMINO)PHENOL	chembl:CHEMBL225257	CHEMBL:CHEMBL225257	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	ISOBOLDINE	chembl:CHEMBL462880	ISOBOLDINE	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.017679351	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	1.400204566285186	ISOSILYBIN B	chembl:CHEMBL3542340	ISOSILYBIN B	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	2-AMINOBIPHENYL	chembl:CHEMBL296021	CHEMBL:CHEMBL296021	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIIF	chembl:CHEMBL1095026	AESCULIOSIDE IIIF	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.077217164	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
OPRL1	hgnc:8155	OPRL1	DTC	9/2/20	NULL	4.375639269641208	JTC-801	iuphar.ligand:1692	JTC-801	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.210030685	PHENAMIPHOS	chembl:CHEMBL1313005	PHENAMIPHOS	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	AMBUNOL	chembl:CHEMBL454893	AMBUNOL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.007416338	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	LEUCINE	rxcui:6308	LEUCINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005860885	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.007548544	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DNDI1417599	chembl:CHEMBL2094833	CHEMBL:CHEMBL2094833	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.03729238	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	DTC	9/2/20	NULL	4.039051633514961	GSK9772	iuphar.ligand:8693	GSK9772	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	MEFLOQUINE HYDROCHLORIDE	rxcui:82130	MEFLOQUINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.3621218705909965	HALICLONADIAMINE	chembl:CHEMBL2177349	HALICLONADIAMINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	1.193356164447602	TCMDC-125319	chembl:CHEMBL527586	CHEMBL:CHEMBL527586	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.00962384	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.024767769	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	LIMONIN	chembl:CHEMBL517449	LIMONIN	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	INDOLE-3-BUTYRIC ACID	chembl:CHEMBL582878	INDOLE-3-BUTYRIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	ANGUIDIN	chembl:CHEMBL433680	ANGUIDIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.069824031	GW405833	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.008799677	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.016352436	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.029783137	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00239313	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	ChEMBL	33	agonist	0.8751278539282418	SOMATOSTATIN	rxcui:9939	SOMATOSTATIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.060008767	TCMDC-123781	chembl:CHEMBL581194	CHEMBL:CHEMBL581194	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	DAIDZIN	drugbank:DB02115	DAIDZIN	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1848861663228679	PIRENOXINE	rxcui:228080	PIRENOXINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.01609924	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.015853765	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	METHOXYVONE	chembl:CHEMBL1591080	METHOXYVONE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.182318303	CAFFEIC ACID	rxcui:1311397	CAFFEIC ACID	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.017092341	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.07458476	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	NIFUROXAZIDE	rxcui:31782	NIFUROXAZIDE	FALSE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	DTC	9/2/20	NULL	5.250767123569449	BELACTOSIN A	chembl:CHEMBL491636	BELACTOSIN A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	GNF-PF-1184	chembl:CHEMBL600347	CHEMBL:CHEMBL600347	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	NORTRIPTYLINE HYDROCHLORIDE	rxcui:203130	NORTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002097622	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.021240967	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.02832129	PIRARUBICIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.006982403	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006570029	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	DEHYDROVARIABILIN	chembl:CHEMBL1520512	DEHYDROVARIABILIN	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1591141552596803	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002936671	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.546954909	CEFUROXIME	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
UNIPROT:P26358	hgnc:2976	DNMT1	TdgClinicalTrial	Jan-14	NULL	0.1909369863116163	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	2.625383561784724	DNDI1417478	chembl:CHEMBL1972216	CHEMBL:CHEMBL1972216	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	SCOULERINE	chembl:CHEMBL1235966	SCOULERINE	FALSE	FALSE	FALSE
BCL2L1	hgnc:992	BCL2L1	DTC	9/2/20	NULL	7.501095891	APOGOSSYPOL	chembl:CHEMBL551288	APOGOSSYPOL	FALSE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	DTC	9/2/20	NULL	0.1750255707856483	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	5.250767123569449	ETILEFRINE	rxcui:4169	ETILEFRINE	FALSE	FALSE	FALSE
GUANYLATE CYCLASE	hgnc:4187	GC	TTD	2020.06.01	NULL	4.375639269641208	Pirsidomine	ncit:C166919	PIRSIDOMINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	COLCHICEINE	rxcui:2174385	COLCHICEINE	TRUE	FALSE	FALSE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	0.364636606	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
RXFP2	hgnc:17318	RXFP2	DTC	9/2/20	NULL	0.9723642821424908	NECA	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.067059606	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	CID 1540545	chembl:CHEMBL259784	CHEMBL:CHEMBL259784	FALSE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	DTC	9/2/20	NULL	0.1403948428761885	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.018874073	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ACIVICIN	ncit:C986	ACIVICIN	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1810609352954983	BENZOQUINONE	iuphar.ligand:6307	BENZOQUINONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.010685322	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1640864726115453	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	ZERANOL	rxcui:1368476	ZERANOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.014405397	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	DTC	9/2/20	NULL	0.3500511415712967	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	TRYPAN BLUE	rxcui:10878	TRYPAN BLUE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.4449802647092754	T-1032	chembl:CHEMBL77971	CHEMBL:CHEMBL77971	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE	chembl:CHEMBL1569494	CHEMBL:CHEMBL1569494	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	DTC	9/2/20	NULL	4.375639269641208	VOACANGINE	chembl:CHEMBL182120	VOACANGINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	GNF-PF-4068	chembl:CHEMBL584668	CHEMBL:CHEMBL584668	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.050246575	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.1166837138570989	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
KLRD1	hgnc:6378	KLRD1	PharmGKB	4/5/24	NULL	0.8078103267029924	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.076541795	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.01609924	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.020836377	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.035083077	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.3947945205691315	STILONIUM IODIDE	ncit:C73168	STILONIUM IODIDE	FALSE	FALSE	FALSE
MIXED LINEAGE KINASE 1	hgnc:6861	MAP3K9	TTD	2020.06.01	NULL	2.625383561784725	CEP1347	iuphar.ligand:8173	CEP-1347	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.029465584	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.019233579	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.031822831	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.041672755	NSC-7387	chembl:CHEMBL119878	CHEMBL:CHEMBL119878	FALSE	FALSE	FALSE
DUSP3	hgnc:3069	DUSP3	DTC	9/2/20	NULL	0.5000730593875666	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009009552	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.49187514	LEVONORGESTREL	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.046965717	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	TENONITROZOLE	rxcui:236186	TENONITROZOLE	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.1187956362798518	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.2019525816757481	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	RILMENIDINE HEMIFUMARATE	chembl:CHEMBL1256674	RILMENIDINE HEMIFUMARATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	PHENYLGLYOXAL	chembl:CHEMBL233632	PHENYLGLYOXAL	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	BITHIONOLOXIDE	ncit:C78040	BITHIONOLOXIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	(R)-ALPHA-METHYLHISTAMINE	iuphar.ligand:1236	(R)-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.3201687270469177	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1693795846312726	BENZOQUINONE	iuphar.ligand:6307	BENZOQUINONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	(R)-PINOCEMBRIN	chembl:CHEMBL399249	(R)-PINOCEMBRIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002016269	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	DNDI1417319	chembl:CHEMBL1392244	CHEMBL:CHEMBL1392244	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ERAP1	hgnc:18173	ERAP1	DTC	9/2/20	NULL	1.250182648468916	ESCULETIN	iuphar.ligand:5180	ESCULETIN	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.018131102	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.043611023	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.081365193	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	1.479089330582943	6,6'-DISELANEDIYLBIS(N-PHENYLHEXANAMIDE)	chembl:CHEMBL1086397	CHEMBL:CHEMBL1086397	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.072324616	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CAMKK2	hgnc:1470	CAMKK2	DTC	9/2/20	NULL	0.2561349816375341	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	15.00219178	hygromycin b	rxcui:1426887	HYGROMYCIN B	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.028184472	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	PRALIDOXIME IODIDE	rxcui:55052	PRALIDOXIME IODIDE	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.028850369	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.4375639269641209	MK-571	iuphar.ligand:10346	MK-571	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	SJ000114741	chembl:CHEMBL591370	CHEMBL:CHEMBL591370	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.005469549	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	NSC-102045	chembl:CHEMBL483633	CHEMBL:CHEMBL483633	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	QUERCITRIN	chembl:CHEMBL82242	QUERCITRIN	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.039778539	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	N-PHENYLMALEIMIDE	chembl:CHEMBL76012	CHEMBL:CHEMBL76012	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001750547	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	NSC-37031	chembl:CHEMBL222993	CHEMBL:CHEMBL222993	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002622106	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	ZALCITABINE	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.043466615	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.2465148884304905	IRSOGLADINE MALEATE	chembl:CHEMBL1712923	IRSOGLADINE MALEATE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	ROSE BENGAL	rxcui:9471	ROSE BENGAL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.3947945205691315	BITHIONOLOXIDE	ncit:C78040	BITHIONOLOXIDE	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	DTC	9/2/20	NULL	0.6141248097742047	NECA	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.1094923635591405	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	4-NONYLPHENOL	rxcui:1788868	4-NONYLPHENOL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.09055649	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.090922374	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.022730594	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:254	hgnc:6585	LHCGR	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:3793	iuphar.ligand:3793	[125I]LH	FALSE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	DTC	9/2/20	NULL	7.001022831425932	RIBOPRINE	rxcui:1376156	RIBOPRINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	IMIDAZOLE-4-ACETIC ACID HCL	chembl:CHEMBL1256325	CHEMBL:CHEMBL1256325	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.019483366	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	OXATOMIDE	rxcui:54236	OXATOMIDE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW290597X	chembl:CHEMBL272026	GW290597X	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.048618214	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PITAVASTATIN CALCIUM	rxcui:861640	PITAVASTATIN CALCIUM	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-2547	chembl:CHEMBL601994	CHEMBL:CHEMBL601994	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	PLICAMYCIN	rxcui:6995	PLICAMYCIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	GAMOLENIC ACID	rxcui:25605	GAMMA-LINOLENIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	CIS-RESVERATROL	chembl:CHEMBL87333	CIS-RESVERATROL	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	2.333674277141977	AW-01208	chembl:CHEMBL560532	CHEMBL:CHEMBL560532	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1363835616511545	FUROXAN	chembl:CHEMBL336467	FUROXAN	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.068637479	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FENARIMOL	chembl:CHEMBL28971	FENARIMOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	NSC-747261	chembl:CHEMBL593366	CHEMBL:CHEMBL593366	FALSE	FALSE	FALSE
LMNA	hgnc:6636	LMNA	DTC	9/2/20	NULL	1.591141552596803	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	5.527123287967842	PRT2527	ncit:C185868	CDK9 INHIBITOR PRT2527	FALSE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	2.386712328895204	DNDI1417461	chembl:CHEMBL1520282	CHEMBL:CHEMBL1520282	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	EQUILIN	ncit:C29020	EQUILIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	MESO-HEXESTROL	drugbank:DB07931	HEXESTROL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	3-(DIMETHYLAMINO)PHENOL	chembl:CHEMBL225257	CHEMBL:CHEMBL225257	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.016116535	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.080781033	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
DHRS9	hgnc:16888	DHRS9	DTC	9/2/20	NULL	15.00219178	(+/-)-HYATELLAQUINONE	chembl:CHEMBL456414	CHEMBL:CHEMBL456414	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.010084054	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	N-(4-HYDROXYPHENYL)RHODANINE	chembl:CHEMBL462430	CHEMBL:CHEMBL462430	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	2.282942227638891	CYCLOPROPARADICICOL	chembl:CHEMBL468439	CYCLOPROPARADICICOL	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.064111931	rocuronium	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.033658764	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	SJ000114741	chembl:CHEMBL591370	CHEMBL:CHEMBL591370	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.016352436	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.028413242	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	0.4150804050252529	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014160645	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.2885036881082115	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.030832455	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.006007743	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.042863405	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.6141248097742046	4',6,7-TRIHYDROXYISOFLAVAN	chembl:CHEMBL8328	CHEMBL:CHEMBL8328	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.2059124362184098	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.002413591	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.00453826	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	DIHYDROERGOTAMINE	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	DTC	9/2/20	NULL	0.032362201	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.033148782	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.023420014	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	GNF-PF-3725	chembl:CHEMBL598695	CHEMBL:CHEMBL598695	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	OXYBENZONE	rxcui:32673	OXYBENZONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003279475	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	THIOLACTOMYCIN	drugbank:DB04302	4-HYDROXY-3,5-DIMETHYL-5-(2-METHYL-BUTA-1,3-DIENYL)-5H-THIOPHEN-2-ONE	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	agonist	0.2885036881082115	RAPASTINEL	ncit:C152156	RAPASTINEL	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	DTC	9/2/20	NULL	1.591141552596803	SODIUM 2-PHENOXYBENZOATE	chembl:CHEMBL2172378	CHEMBL:CHEMBL2172378	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.018560506	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-123748	chembl:CHEMBL530609	CHEMBL:CHEMBL530609	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GITOXIGENIN	chembl:CHEMBL464658	GITOXIGENIN	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	DTC	9/2/20	NULL	4.773424657790409	O6-[3-(AMINOMETHYL)BENZYL]GUANINE	chembl:CHEMBL485756	CHEMBL:CHEMBL485756	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	2-(2-HYDROXYBENZYL)PHENOL	chembl:CHEMBL148831	CHEMBL:CHEMBL148831	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.038467158	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.002318219	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.016764901	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.008773212	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.5527123287967841	IUPHAR.LIGAND:350	iuphar.ligand:350	SCH 57790	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.033985548	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.03505185	ZERANOL	rxcui:1368476	ZERANOL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	GAMOLENIC ACID	rxcui:25605	GAMMA-LINOLENIC ACID	FALSE	FALSE	FALSE
RXFP2	hgnc:17318	RXFP2	DTC	9/2/20	NULL	0.7955707762984016	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	METHAPHIT	chembl:CHEMBL41541	METHAPHIT	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1396480617970598	TCMDC-123480	chembl:CHEMBL588683	CHEMBL:CHEMBL588683	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	FPL-64176	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2035181055647073	PROCATEROL HYDROCHLORIDE	rxcui:58918	PROCATEROL HYDROCHLORIDE	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.031784305	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.039361073	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004579424	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	EDARAVONE	rxcui:1921877	EDARAVONE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	HEMICHOLINIUM-3	iuphar.ligand:4494	HEMICHOLINIUM-3	FALSE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.7292732116068681	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	BMS-182874	chembl:CHEMBL267458	BMS-182874	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005117707	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.058083707	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-2059	chembl:CHEMBL601968	CHEMBL:CHEMBL601968	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.2273059360852575	BITHIONOLOXIDE	ncit:C78040	BITHIONOLOXIDE	FALSE	FALSE	FALSE
SMAD2	hgnc:6768	SMAD2	DTC	9/2/20	NULL	2.187819634820604	DEMETHOXYCURCUMIN	chembl:CHEMBL179512	DEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	ALX-5407	iuphar.ligand:4618	(R)-NFPS	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-4864	chembl:CHEMBL583558	CHEMBL:CHEMBL583558	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	ITRAZOLE	chembl:CHEMBL64391	ITRACONAZOLE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.032412143	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.012794267	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.028459442	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.022164488	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.038894571	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.002731502	ESTRADIOL ACETATE	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.4375639269641208	8-FLUOROTRYPTANTHRIN	chembl:CHEMBL1098875	CHEMBL:CHEMBL1098875	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	6.563458904461812	RICININE	chembl:CHEMBL1329957	RICININE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	5-FLUOROINDOLE-2-CARBOXYLIC ACID	chembl:CHEMBL23507	5-FLUOROINDOLE-2-CARBOXYLIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	DEQUALINIUM CHLORIDE	rxcui:3120	DEQUALINIUM CHLORIDE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	BORIC ACID	rxcui:1700	BORIC ACID	TRUE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	1.944728564284981	CHLORPYRAMIN HYDROCHLORIDE	chembl:CHEMBL550011	CHLORPYRAMIN HYDROCHLORIDE	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	1.166837138570988	HELIPARVIFOLINE	chembl:CHEMBL455007	HELIPARVIFOLINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.028598949	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	GNF-PF-1233	chembl:CHEMBL585788	CHEMBL:CHEMBL585788	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.097870776	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CARBENOXOLONE DISODIUM	chembl:CHEMBL1697717	CARBENOXOLONE SODIUM	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	GNF-PF-2359	chembl:CHEMBL610622	CHEMBL:CHEMBL610622	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	DNDI1417484	chembl:CHEMBL1308677	CHEMBL:CHEMBL1308677	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	2.561349816375341	FERRUGINENE B	chembl:CHEMBL1775032	FERRUGINENE B	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.6250913242344582	METHYLERGONOVINE MALEATE	rxcui:84158	METHYLERGONOVINE MALEATE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-2941	chembl:CHEMBL602413	CHEMBL:CHEMBL602413	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.026227608	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.021129848	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004339477	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.052090944	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.013957382	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.027276712	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
ADCY2	hgnc:233	ADCY2	DTC	9/2/20	NULL	6.563458904461812	NSC-270718	chembl:CHEMBL401844	CHEMBL:CHEMBL401844	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.026227608	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	SARAFLOXACIN HYDROCHLORIDE	ncit:C72844	SARAFLOXACIN HYDROCHLORIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	DOCUSATE	rxcui:82003	DOCUSATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MITOBRONITOL	rxcui:6996	MITOBRONITOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	FLUAZINAM	chembl:CHEMBL1878267	FLUAZINAM	FALSE	FALSE	FALSE
RPS6KA1	hgnc:10430	RPS6KA1	DTC	9/2/20	NULL	1.944728564284981	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.4167275494896389	NECA	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.2282942227638891	DIHYDROTANSHINONE I	chembl:CHEMBL227075	DIHYDROTANSHINONE I	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.070197421	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.7778914257139926	DIHYDROTANSHINONE I	chembl:CHEMBL227075	DIHYDROTANSHINONE I	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.00937637	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	ETIDRONIC ACID	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.039778539	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IV-23D1	chembl:CHEMBL1094675	CHEMBL:CHEMBL1094675	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.088996053	THIOLACTOMYCIN	drugbank:DB04302	4-HYDROXY-3,5-DIMETHYL-5-(2-METHYL-BUTA-1,3-DIENYL)-5H-THIOPHEN-2-ONE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.044498026	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.034544521	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	DTC	9/2/20	NULL	7.876150685354174	MK-0893	drugbank:DB12044	MK-0893	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009320613	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.020834311	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
UQCR10	hgnc:30863	UQCR10	DTC	9/2/20	NULL	105.0153424713889	FAMOXADONE	chembl:CHEMBL10118	FAMOXADONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	AMINACRINE HYDROCHLORIDE	rxcui:81949	AMINACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.9376369863516875	DIPHYLLIN	chembl:CHEMBL221190	DIPHYLLIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	STILONIUM IODIDE	ncit:C73168	STILONIUM IODIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002169738	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	GNF-PF-1872	chembl:CHEMBL600103	CHEMBL:CHEMBL600103	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.008217163	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.078722146	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	AMCINAFIDE	ncit:C80807	AMCINAFIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	METHOXYVERAPAMIL HYDROCHLORIDE	chembl:CHEMBL1256940	METHOXYVERAPAMIL HYDROCHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.3125456621172291	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01823183	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	DNDI1417599	chembl:CHEMBL2094833	CHEMBL:CHEMBL2094833	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006434764	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-699479	chembl:CHEMBL1701915	CHEMBL:CHEMBL1701915	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2075402025126264	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2273059360852575	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003099626	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.017945205	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	BMS-182874	chembl:CHEMBL267458	BMS-182874	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2430910705356226	GNF-PF-4864	chembl:CHEMBL583558	CHEMBL:CHEMBL583558	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.2476776945079929	GNF-PF-2260	chembl:CHEMBL601351	CHEMBL:CHEMBL601351	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-4786	chembl:CHEMBL602363	CHEMBL:CHEMBL602363	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.007737647	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	PD-0118057	iuphar.ligand:7676	PD-118057	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.012738397	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-4665	chembl:CHEMBL601744	CHEMBL:CHEMBL601744	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.008047153	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NSC-123526	chembl:CHEMBL271165	CHEMBL:CHEMBL271165	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	SALICYLURIC ACID	chembl:CHEMBL586	SALICYLURIC ACID	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.082300425	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.018786287	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	DTC	9/2/20	NULL	3.500511415712966	CYPATE	chembl:CHEMBL2071606	CYPATE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	TRICLOSAN	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	BIX-01294	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
UNIPROT:P54710	hgnc:4026	FXYD2	TEND	1-Aug-11	NULL	0.9723642821424908	CYCLOTHIAZIDE	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.2083637747448194	CHLORMADINONE ACETATE	rxcui:2369	CHLORMADINONE ACETATE	TRUE	FALSE	FALSE
DDAH1	hgnc:2715	DDAH1	DTC	9/2/20	NULL	105.0153424713889	2-ETHYL-BENZIMIDAZOLE	chembl:CHEMBL351569	CHEMBL:CHEMBL351569	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	TDR78109	chembl:CHEMBL1304363	CHEMBL:CHEMBL1304363	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	1.141471113819445	CUCURBITACIN D	chembl:CHEMBL493646	CUCURBITACIN D	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	NSC-133896	chembl:CHEMBL512908	CHEMBL:CHEMBL512908	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007831122	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.013360731	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
GCK	hgnc:4195	GCK	DTC	9/2/20	NULL	7.001022831425932	PIRAGLIATIN	ncit:C77587	PIRAGLIATIN	FALSE	FALSE	FALSE
CDC42	hgnc:1736	CDC42	DTC	9/2/20	NULL	17.50255707856483	SECRAMINE A	chembl:CHEMBL1222038	SECRAMINE A	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009875432	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1041818873724097	NSC-638080	chembl:CHEMBL136344	CHEMBL:CHEMBL136344	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.033487035	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.008143249	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	E232	chembl:CHEMBL1903906	E232	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	ANTHRALIN	rxcui:873	ANTHRALIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	METCONAZOLE	chembl:CHEMBL1883512	METCONAZOLE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.210030685	DNDI1383301	chembl:CHEMBL1509103	CHEMBL:CHEMBL1509103	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	SJ000193360	chembl:CHEMBL607253	CHEMBL:CHEMBL607253	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	DTC	9/2/20	NULL	0.1842374429322614	PIPERTRAMINE AMIDE	chembl:CHEMBL130835	PIPERTRAMINE AMIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.035670972	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	BRONOPOL	rxcui:1114345	BRONOPOL	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.021590325	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.1555782851427985	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.1715936968486748	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	OXAPIUM IODIDE	ncit:C90697	OXAPIUM IODIDE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	CID 1225609	chembl:CHEMBL444376	CHEMBL:CHEMBL444376	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	NSC-83217	chembl:CHEMBL120806	CHEMBL:CHEMBL120806	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005563432	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NSC-117079	chembl:CHEMBL471225	CHEMBL:CHEMBL471225	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001259177	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	GNF-PF-4997	chembl:CHEMBL306147	CHEMBL:CHEMBL306147	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	IODOCARB	chembl:CHEMBL1893913	IODOCARB	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	GNF-PF-4542	chembl:CHEMBL585999	CHEMBL:CHEMBL585999	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	NSC-102045	chembl:CHEMBL483633	CHEMBL:CHEMBL483633	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	3,3',4,4',5,5'-HEXAMETHOXYCHALCONE	chembl:CHEMBL17442	CHEMBL:CHEMBL17442	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.012913839	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.021074723	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.084146909	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	AMINACRINE HYDROCHLORIDE	rxcui:81949	AMINACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	2'-METHOXYFORMONETIN	chembl:CHEMBL1087126	2'-METHOXYFORMONETIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	SIMETRIDE	ncit:C72129	SIMETRIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CGS-12066A MALEATE	chembl:CHEMBL1256689	CHEMBL:CHEMBL1256689	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.100589408	MRS-1220	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.081533651	ZERANOL	rxcui:1368476	ZERANOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.004542186	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-2121	chembl:CHEMBL577365	CHEMBL:CHEMBL577365	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ALLETHRIN	rxcui:513	ALLETHRIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	MALINAMIDE	chembl:CHEMBL64379	MALINAMIDE	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.4375639269641208	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.040452751	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	GNF-PF-3191	chembl:CHEMBL581865	CHEMBL:CHEMBL581865	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	HELIOMYCIN	ncit:C75147	HELIOMYCIN	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.047647615	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.3302369260106572	TUBASTATIN A	iuphar.ligand:9702	TUBASTATIN A	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.006077277	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
PDK1	hgnc:8809	PDK1	DTC	9/2/20	NULL	5.000730593875666	DICHLOROACETIC ACID	rxcui:155021	DICHLOROACETIC ACID	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	NSC-7387	chembl:CHEMBL119878	CHEMBL:CHEMBL119878	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.1396480617970598	FIDUXOSIN	ncit:C65682	FIDUXOSIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.022439176	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.026227608	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.03223307	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.088935758	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	MOFEGILINE	ncit:C83968	MOFEGILINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006987979	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	DTC	9/2/20	NULL	0.1458546423213736	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	VALRUBICIN	rxcui:31435	VALRUBICIN	TRUE	FALSE	TRUE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.8204323630577265	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	2.333674277141977	RIMEGEPANT	rxcui:2282307	RIMEGEPANT	TRUE	FALSE	FALSE
ADM	hgnc:259	ADM	DTC	9/2/20	NULL	4.375639269641208	NSC-87877	chembl:CHEMBL472004	CHEMBL:CHEMBL472004	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.02832129	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	TENOXICAM	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
FPR1	hgnc:3826	FPR1	DTC	9/2/20	NULL	0.2500365296937833	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	1.640864726115453	MI-503	iuphar.ligand:9526	MI-503	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	SYM004	ncit:C91381	FUTUXIMAB/MODOTUXIMAB MIXTURE	FALSE	TRUE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	1-NAPHTHYLISOTHIOCYANATE	chembl:CHEMBL1381098	1-NAPHTHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004579424	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.3017682254924971	Ipatasertib	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.1816874437221263	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.025814981	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.009734459	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.037693949	FLUORESCEIN	rxcui:25138	FLUORESCEIN	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.021878196	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1666910197958555	BITHIONOLOXIDE	ncit:C78040	BITHIONOLOXIDE	FALSE	FALSE	FALSE
FGB	hgnc:3662	FGB	DTC	9/2/20	NULL	0.1346350544504987	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	TCMDC-123808	chembl:CHEMBL546493	CHEMBL:CHEMBL546493	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	QUIFENADINE	ncit:C81147	QUIFENADINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW779439X	chembl:CHEMBL468963	GW779439X	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.078958904	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.005834186	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NUCLEOBINDIN-1	hgnc:8043	NUCB1	TTD	2020.06.01	NULL	52.50767123569449	GS-5734	rxcui:2284718	REMDESIVIR	TRUE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.6482428547616604	DIPHENYLUREA	chembl:CHEMBL354676	DIPHENYLUREA	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.3040984820600068	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	TDR78109	chembl:CHEMBL1304363	CHEMBL:CHEMBL1304363	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2885036881082115	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GERONTOXANTHONE I	chembl:CHEMBL478791	GERONTOXANTHONE I	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.3125456621172292	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	SB-242084	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	GNF-PF-2755	chembl:CHEMBL600738	CHEMBL:CHEMBL600738	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.027121731	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	GNF-PF-1872	chembl:CHEMBL600103	CHEMBL:CHEMBL600103	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	PROPYLPARABEN	rxcui:34706	PROPYLPARABEN	TRUE	FALSE	FALSE
PTBP1	hgnc:9583	PTBP1	DTC	9/2/20	NULL	0.4861821410712454	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.041672755	2,6-DIMETHOXYQUINONE	chembl:CHEMBL448515	2,6-DIMETHOXYQUINONE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.015193192	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00402481	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.023759127	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.02321294	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.729273212	CEFMETAZOLE	rxcui:2182	CEFMETAZOLE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	ALLOXAN	rxcui:2466730	ALLOXAN	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	1.250182648468916	CEFMETAZOLE	rxcui:2182	CEFMETAZOLE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1041818873724097	ACRIDIN-1-YLAMINE	chembl:CHEMBL146525	CHEMBL:CHEMBL146525	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	SYROSINGOPINE	ncit:C152485	SYROSINGOPINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	TCMDC-124063	chembl:CHEMBL534535	CHEMBL:CHEMBL534535	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	MyCancerGenome	20-Jun-17	inhibitor	0.2853677784548614	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.043629141	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	MyCancerGenome	20-Jun-17	inhibitor	0.03337352	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.8751278539282416	EMD1214063	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.272767123	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	1.458546423213736	Ibutamoren	rxcui:1805438	IBUTAMOREN	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.7160136986685613	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.06697407	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547592	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547592	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	GNF-PF-5052	chembl:CHEMBL601367	CHEMBL:CHEMBL601367	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.2500365296937833	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.063331621	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4735540335109532	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.736088849	GUANADREL SULFATE	rxcui:91239	GUANADREL SULFATE	TRUE	FALSE	FALSE
AKT2	hgnc:392	AKT2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2430910705356226	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSP90AB2	NULL	NULL	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	NULL	RETASPIMYCIN HYDROCHLORIDE	ncit:C48401	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3409589041278863	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
CDK1	hgnc:1722	CDK1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3431873936973496	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
MIR21	hgnc:31586	MIR21	CIViC	10-Apr-24	NULL	0.3621218705909965	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1944728564284981	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.053798843	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1944728564284981	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
WNT7A	hgnc:12786	WNT7A	NCI	14-Sep-17	NULL	3.182283105193606	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
VEGFC	hgnc:12682	VEGFC	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.051177067	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.008013991	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.2243917574174978	EPIPODOPHYLLOTOXINS	ncit:C1331	EPIPODOPHYLLOTOXIN COMPOUND	FALSE	FALSE	FALSE
AKR1B1	hgnc:381	AKR1B1	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.009304921	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
AGTR2	hgnc:338	AGTR2	NCI	14-Sep-17	NULL	1.193356164447602	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	NCI	14-Sep-17	NULL	0.092118721	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
NCBIGENE:3237	hgnc:5134	HOXD11	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12791	iuphar.ligand:12791	CW85319	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.1286952726365061	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	NCI	14-Sep-17	NULL	0.1826353782111113	IL-10	iuphar.ligand:4975	IL-10	FALSE	FALSE	FALSE
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	0.280789686	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
NCBIGENE:2084	hgnc:6861	MAP3K9	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:8173	iuphar.ligand:8173	CEP-1347	FALSE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.085239726	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	NCI	14-Sep-17	NULL	0.052771529	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.034819411	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.06466462	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.084254928	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
BCL6	hgnc:1001	BCL6	NCI	14-Sep-17	NULL	1.346350544504987	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.3750547945406749	IUPHAR.LIGAND:9130	iuphar.ligand:9130	ZM336372	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.044935962	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.035574303	ICI 182780	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.056918885	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.076709527	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	PharmGKB	4/5/24	NULL	0.065226921	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.066297565	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.1193356164447602	IL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.2983390411119005	RAS INHIBITOR	ncit:C1902	RAS INHIBITOR	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.046549354	MITOMYCIN C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	NCI	14-Sep-17	NULL	0.050978322	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
CAMK2B	hgnc:1461	CAMK2B	NCI	14-Sep-17	NULL	0.09969811	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	NCI	14-Sep-17	NULL	0.7778914257139926	ACTIVIN	ncit:C2689	IH636 GRAPE SEED PROANTHOCYANIDIN EXTRACT	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	FAS-LIGAND	ncit:C1538	RECOMBINANT FAS LIGAND	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.729273212	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.1576806944014849	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.052090944	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CHST11	hgnc:17422	CHST11	NCI	14-Sep-17	NULL	NULL	CHONDROITIN	NULL	NULL	NULL	NULL	NULL
CISH	hgnc:1984	CISH	NCI	14-Sep-17	NULL	3.088686543276147	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.006811217	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.048017989	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	1.29648571	TETRANDRINE	ncit:C28952	TETRANDRINE	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.2187819634820604	TOLMETIN SODIUM	rxcui:42935	TOLMETIN SODIUM	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.1470803115845784	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.08854582	O6-BENZYLGUANINE	ncit:C1306	O6-BENZYLGUANINE	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.187193124	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.09969811	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.1640864726115453	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.026259671	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.027781837	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.002553627	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.005339401	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.068637479	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	NCI	14-Sep-17	NULL	1.250182648468916	CHLORZOXAZONE	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
DBP	hgnc:2697	DBP	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	FDA	10-Apr-24	NULL	0.042793538	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.064268875	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.4070362111294147	MANNITOL	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.05309168	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
DEFB4	hgnc:2767	DEFB4A	NCI	14-Sep-17	NULL	1.166837138570989	IMMUNOSUPPRESSIVE AGENTS	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1831662950082366	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	(+)-THALIPORPHINE	chembl:CHEMBL1397308	CHEMBL:CHEMBL1397308	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	TIRATRICOL	rxcui:13982	TIRATRICOL	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	1.640864726115453	ZD1694	ncit:C1804	RALTITREXED	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.1904575128526865	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	1.193356164447602	FTI	ncit:C2020	FARNESYL TRANSFERASE INHIBITOR	FALSE	FALSE	FALSE
DTYMK	hgnc:3061	DTYMK	NCI	14-Sep-17	NULL	0.1661635165686534	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	0.062065805	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	NCI	14-Sep-17	NULL	0.014977128	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.1782942996118658	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.3947945205691315	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
EMP1	hgnc:3333	EMP1	NCI	14-Sep-17	NULL	0.3088686543276147	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.035560536	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.018672714	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
ERCC1	hgnc:3433	ERCC1	NCI	14-Sep-17	NULL	0.073540156	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.1810609352954983	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:295	iuphar.ligand:295	ARECAIDINE PROPARGYL ESTER	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.6604738520213144	IL-18	iuphar.ligand:4983	IL-18	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.3977853881492007	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1973972602845657	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	0.1329308132549227	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.037398626	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.6863747873946994	ROFECOXIB	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	agonist	0.032899543	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.561579372	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
GNMT	hgnc:4415	GNMT	NCI	14-Sep-17	NULL	5.000730593875666	VITAMIN B12	rxcui:11248	VITAMIN B12	TRUE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.038608582	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
GLS	hgnc:4331	GLS	NCI	14-Sep-17	NULL	0.013206155	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
GLS	hgnc:4331	GLS	NCI	14-Sep-17	NULL	0.1232574442152452	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.106290832	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.3977853881492006	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	1.570742301922485	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	NULL	XANTHOPHYLLS	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.4375639269641208	ADM	ncit:C186783	ACELLULAR DERMAL MATRIX	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.4375639269641208	BPDE	ncit:C196	BENZO(A)PYRENE-7,8-DIOL 9,10-EPOXIDE	FALSE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	0.2375912725597036	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.4102161815288632	CYCLOOXYGENASE INHIBITOR	ncit:C1323	CYCLOOXYGENASE INHIBITOR	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.2059124362184098	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	NULL	TOTAL PARENTERAL NUTRITION	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.6863747873946993	DINITROCHLOROBENZENE	ncit:C439	DINITROCHLOROBENZENE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.2287915957982331	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1470803115845784	DIDEOXYINOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.1440539677248134	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.2592971419046642	RECOMBINANT HUMAN IL-4	rxcui:1426682	BINETRAKIN	FALSE	FALSE	FALSE
IRS1	hgnc:6125	IRS1	NCI	14-Sep-17	NULL	0.7292732116068681	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.030430409	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1293292394967844	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.3241214273808302	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.013876234	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
JUNB	hgnc:6205	JUNB	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
UBE2I	hgnc:12485	UBE2I	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.729273212	PROTEOLYTIC ENZYMES	ncit:C38728	PANCREATIC PROTEOLYTIC ENZYMES	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.08334551	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.2083637747448194	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	NCI	14-Sep-17	NULL	0.2130128650535274	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
KRT19	hgnc:6436	KRT19	NCI	14-Sep-17	NULL	1.419126249613364	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.4375639269641208	PANTOPRAZOLE SODIUM	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	1.750255707856483	RHENIUM-186 HYDROXYETHYLIDENE DIPHOSPHONATE	ncit:C1562	RHENIUM RE 186 ETIDRONATE	FALSE	FALSE	FALSE
LCAT	hgnc:6522	LCAT	NCI	14-Sep-17	NULL	0.5385402178019948	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.09963505	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
LIPC	hgnc:6619	LIPC	NCI	14-Sep-17	NULL	0.2215513554248712	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.019177382	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.1500219178162699	PI3-KINASE INHIBITORS	ncit:C2152	PHOSPHATIDYLINOSITIDE 3-KINASE INHIBITOR	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.016669102	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.1091635576625665	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
MDH2	hgnc:6971	MDH2	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
MDM2	hgnc:6973	MDM2	NCI	14-Sep-17	NULL	0.2187819634820604	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.4375639269641208	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	0.8078103267029924	ISOSORBIDE-5-MONONITRATE	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	1.458546423213736	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.086861325	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	0.045051627	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:5263	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	NULL	CHONDROITIN	NULL	NULL	NULL	NULL	NULL
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1071585127259071	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
MYB	hgnc:7545	MYB	NCI	14-Sep-17	NULL	0.5645986154375753	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	0.1141471113819445	RETASPIMYCIN HYDROCHLORIDE	ncit:C48401	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.013990853	SELECTIVE ESTROGEN RECEPTOR MODULATORS	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.001937195	TAM	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1479089330582944	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	NULL	PHOSPHOROTHIOATE OLIGONUCLEOTIDE	NULL	NULL	NULL	NULL	NULL
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	3.182283105193605	ENDOTHELIN RECEPTOR ANTAGONIST	ncit:C28313	ENDOTHELIN RECEPTOR ANTAGONIST	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	GNF-PF-372	chembl:CHEMBL580155	CHEMBL:CHEMBL580155	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.027010119	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	NCI	14-Sep-17	NULL	0.056459862	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.3125456621172291	HEREGULIN	ncit:C1426	RECOMBINANT HEREGULIN	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	NCI	14-Sep-17	NULL	0.158394182	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	NCI	14-Sep-17	NULL	0.066213961	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.026519026	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	NULL	PHOSPHOROTHIOATE OLIGONUCLEOTIDE	NULL	NULL	NULL	NULL	NULL
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	0.4039051633514962	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	0.252440727	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	ARACHIDONOYL GABA	iuphar.ligand:5494	N-ARACHIDONYL-&GAMMA;-AMINOBUTYRIC ACID	FALSE	FALSE	FALSE
POU5F1	hgnc:9221	POU5F1	NCI	14-Sep-17	NULL	0.3323270331373069	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	NCI	14-Sep-17	NULL	0.041540879	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.049026771	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ADH1C	hgnc:251	ADH1C	PharmGKB	4/5/24	NULL	0.016094305	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
RBP3	hgnc:9921	RBP3	NCI	14-Sep-17	NULL	1.693795846312725	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	NCI	14-Sep-17	NULL	0.099587807	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
CSNK2A1	hgnc:2457	CSNK2A1	NCI	14-Sep-17	NULL	0.1640864726115453	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
SI	hgnc:10856	SI	NCI	14-Sep-17	NULL	NULL	TOTAL PARENTERAL NUTRITION	NULL	NULL	NULL	NULL	NULL
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.089756703	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1154014752432845	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
SLC9A3	hgnc:11073	SLC9A3	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.057700738	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	SJ000111093	chembl:CHEMBL585045	CHEMBL:CHEMBL585045	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	NCI	14-Sep-17	NULL	0.358239472	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
SMOX	hgnc:15862	SMOX	NCI	14-Sep-17	NULL	7.001022831425934	AZASERINE	ncit:C289	AZASERINE	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	NCI	14-Sep-17	NULL	0.020048748	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.2476776945079929	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
SRI	hgnc:11292	SRI	NCI	14-Sep-17	NULL	5.250767123569449	ADM	ncit:C186783	ACELLULAR DERMAL MATRIX	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NSC-32984	chembl:CHEMBL1339015	CHEMBL:CHEMBL1339015	FALSE	FALSE	FALSE
SPINT1	hgnc:11246	SPINT1	NCI	14-Sep-17	NULL	2.763561643983921	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
SRY	hgnc:11311	SRY	NCI	14-Sep-17	NULL	6.563458904461812	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
STAB2	hgnc:18629	STAB2	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.029833904	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SULT2A1	hgnc:11458	SULT2A1	NCI	14-Sep-17	NULL	0.1875273972703374	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	0.6364566210387212	PROGESTOGENS	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
ST14	hgnc:11344	ST14	NCI	14-Sep-17	NULL	1.381780822	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.3889457128569963	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	7.001022831425932	AMG 334	rxcui:2045613	ERENUMAB	TRUE	FALSE	FALSE
TARP	ensembl:ENSG00000289746	TARP	NCI	14-Sep-17	NULL	4.039051633514962	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1848861663228679	TAS-115	chembl:CHEMBL3545144	TAS-115	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	NULL	CHONDROITIN	NULL	NULL	NULL	NULL	NULL
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.042880908	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.8899605294185507	SANDOSTATIN	chembl:CHEMBL408687	SANDOSTATIN	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1369170045259309	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
MAOA	hgnc:6833	MAOA	ChEMBL	33	activator	0.6731752722524935	PROXIBARBAL	rxcui:83885	PROXIBARBAL	TRUE	FALSE	FALSE
THRSP	hgnc:11800	THRSP	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.087732116	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	1.346350544504987	HALOFUGINONE	ncit:C1120	HALOFUGINONE	FALSE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.064824285	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
CDK12	hgnc:24224	CDK12	OncoKB	23-Jul-20	NULL	0.5000730593875666	Cemiplimab	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	OncoKB	23-Jul-20	NULL	0.066676408	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	OncoKB	23-Jul-20	NULL	1.184383561707394	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	OncoKB	23-Jul-20	NULL	1.831662950082366	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	OncoKB	23-Jul-20	NULL	0.1481697953740938	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
NCBIGENE:642	hgnc:1059	BLMH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7994	iuphar.ligand:7994	ANALOG 3 [VLATTAS ET AL., 1996]	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	OncoKB	23-Jul-20	NULL	NULL	Carboplatin-Taxol Regimen	NULL	NULL	NULL	NULL	NULL
FGFR1	hgnc:3688	FGFR1	OncoKB	23-Jul-20	NULL	0.3453256329104173	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	PharmGKB	4/5/24	NULL	NULL	chloroacetaldehyde	NULL	NULL	NULL	NULL	NULL
REN	hgnc:9958	REN	PharmGKB	4/5/24	NULL	NULL	vitamin d and analogues	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:8186	iuphar.ligand:8186	COMPOUND 19A [PMID: 21855335]	FALSE	FALSE	FALSE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	4.719790672871415	estrogens	rxcui:4100	ESTROGENS	FALSE	FALSE	FALSE
PARD3B	hgnc:14446	PARD3B	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
SLC28A1	hgnc:11001	SLC28A1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	0.7001022831425934	ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.2059124362184098	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	hydroxyamitriptyline	NULL	NULL	NULL	NULL	NULL
STK39	hgnc:17717	STK39	PharmGKB	4/5/24	NULL	9.546849315580818	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	PharmGKB	4/5/24	NULL	0.7326651800329465	ethosuximide	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
APOC3	hgnc:610	APOC3	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
STX11	hgnc:11429	STX11	PharmGKB	4/5/24	NULL	13.12691780892362	emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
UNC13D	hgnc:23147	UNC13D	PharmGKB	4/5/24	NULL	13.12691780892362	emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.020656047	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.2206204673768676	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	NULL	FOLFIRI	NULL	NULL	NULL	NULL	NULL
SLC28A3	hgnc:16484	SLC28A3	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	3.889457128569962	VELTUZUMAB	ncit:C48406	VELTUZUMAB	FALSE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	PharmGKB	4/5/24	NULL	0.077330885	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.1201548540862574	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
ADH7	hgnc:256	ADH7	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
COL26A1	hgnc:18038	COL26A1	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
MOCS1	hgnc:7190	MOCS1	PharmGKB	4/5/24	NULL	13.12691780892362	fosdenopterin	rxcui:2531288	FOSDENOPTERIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.034727296	avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.027781837	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1662	hgnc:2735	DDX10	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:6509	iuphar.ligand:6509	BMS-561392	FALSE	FALSE	FALSE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
PRSS3	hgnc:9486	PRSS3	DTC	9/2/20	NULL	5.834185692854944	CYANOPEPTOLIN SS	chembl:CHEMBL1076839	CYANOPEPTOLIN SS	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	1.875273972703375	2-(4-ISOPROPYLPHENYL)BENZOTHIAZOLE	chembl:CHEMBL1351908	CHEMBL:CHEMBL1351908	FALSE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
GABRA6	hgnc:4080	GABRA6	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
GABRP	hgnc:4089	GABRP	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
GAL	hgnc:4114	GAL	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.078369659	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
GRIA3	hgnc:4573	GRIA3	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
PLCB1	hgnc:15917	PLCB1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.042310775	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	VITAMIN B2	chembl:CHEMBL1397833	VITAMIN B2	FALSE	FALSE	FALSE
TPH1	hgnc:12008	TPH1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
SLC1A1	hgnc:10939	SLC1A1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
TXNRD2	hgnc:18155	TXNRD2	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1112450661773188	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	PharmGKB	4/5/24	NULL	0.036463661	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.6908904109959803	carbimazole	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.016916131	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
TCF7L2	hgnc:11641	TCF7L2	PharmGKB	4/5/24	NULL	NULL	Dipeptidyl peptidase 4 (DPP-4) inhibitors	NULL	NULL	NULL	NULL	NULL
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.1458546423213736	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1209854175937661	DAPHNORIN	chembl:CHEMBL1209491	DAPHNORIN	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	PharmGKB	4/5/24	NULL	NULL	antiarrhythmics, class i and iii	NULL	NULL	NULL	NULL	NULL
CHPT1	hgnc:17852	CHPT1	PharmGKB	4/5/24	NULL	2.187819634820604	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
ASIC2	hgnc:99	ASIC2	PharmGKB	4/5/24	NULL	0.108711535	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.2500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	GNF-PF-2298	chembl:CHEMBL578905	CHEMBL:CHEMBL578905	FALSE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.2273059360852575	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.023110771	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
REEP5	hgnc:30077	REEP5	PharmGKB	4/5/24	NULL	1.312691780892362	sertraline	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.071341945	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
ESYT2	hgnc:22211	ESYT2	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.021742307	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
ALDH1L1	hgnc:3978	ALDH1L1	PharmGKB	4/5/24	NULL	1.141471113819445	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
CHURC1	hgnc:20099	CHURC1	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.073954467	EMETINE	rxcui:3820	EMETINE	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	PharmGKB	4/5/24	NULL	0.02926849	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
PDIA2	hgnc:14180	PDIA2	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	NULL	selective beta-2-adrenoreceptor agonists	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	dextromethorphan hydrobromide / bupropion hydrochloride	NULL	NULL	NULL	NULL	NULL
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.09323095	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.092606122	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	1.166837138570989	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	OC144-093	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	XR9051	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.018699313	bepridil	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	highly active antiretroviral therapy (haart)	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	S-EDDP	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.023374141	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.008630452	carvedilol	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
CDH15	hgnc:1754	CDH15	PharmGKB	4/5/24	NULL	0.1241316104862754	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	NULL	vitamin d and analogues	NULL	NULL	NULL	NULL	NULL
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.069180068	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:8793	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
CASR	hgnc:1514	CASR	PharmGKB	4/5/24	NULL	NULL	Parathyroid Hormones And Analogues	NULL	NULL	NULL	NULL	NULL
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	NULL	ezetimibe / rosuvastatin	NULL	NULL	NULL	NULL	NULL
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.01143958	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.08572681	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	PharmGKB	4/5/24	NULL	0.1403266238077355	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.032572997	propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	0.081281225	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	PharmGKB	4/5/24	NULL	0.1567393171214761	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.182318303	mitotane	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.087512785	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.3281729452230906	ospemifene	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006909813	acalabrutinib	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.018521224	nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.060878459	nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	Ascorbic acid (vitamin C), plain	NULL	NULL	NULL	NULL	NULL
GLA	hgnc:4296	GLA	PharmGKB	4/5/24	NULL	4.039051633514961	migalastat	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2234368988752957	PIRENZEPINE	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
ATP2A3	hgnc:813	ATP2A3	PharmGKB	4/5/24	NULL	0.130616098	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CACNB1	hgnc:1401	CACNB1	PharmGKB	4/5/24	NULL	0.1119566550867686	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CACNA1D	hgnc:1391	CACNA1D	PharmGKB	4/5/24	NULL	0.036451004	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	PharmGKB	4/5/24	NULL	0.023748381	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:1614	hgnc:13557	ACE2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6555	iuphar.ligand:6555	COMPOUND 28 [PMID: 18324760]	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.033348791	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	PharmGKB	4/5/24	NULL	0.012539145	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
EYS	hgnc:21555	EYS	PharmGKB	4/5/24	NULL	NULL	HMG CoA reductase inhibitors, other combinations	NULL	NULL	NULL	NULL	NULL
TLR5	hgnc:11851	TLR5	PharmGKB	4/5/24	NULL	1.750255707856483	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:6170	iuphar.ligand:6170	MK-5046	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.095642388	ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.1012684112549556	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	PharmGKB	4/5/24	NULL	0.8751278539282416	tepotinib	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	noroxycodone	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	n-desmethyltramadol	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	n,o-didesmethyltramadol	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	desmethyl clomipramine	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.014757637	bepridil	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.035418328	upadacitinib	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	NULL	thioguanosine triphosphate	NULL	NULL	NULL	NULL	NULL
PRKCA	hgnc:9393	PRKCA	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
AGBL4	hgnc:25892	AGBL4	PharmGKB	4/5/24	NULL	2.625383561784725	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.095399112	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.026563746	n-desmethylclozapine	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
GRID2	hgnc:4576	GRID2	PharmGKB	4/5/24	NULL	NULL	6-hydroxy r-warfarin	NULL	NULL	NULL	NULL	NULL
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.1268301237577161	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:314	iuphar.ligand:314	MUSCARINIC TOXIN 7	FALSE	FALSE	FALSE
CHRNA6	hgnc:15963	CHRNA6	PharmGKB	4/5/24	NULL	0.9723642821424908	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.1689436011444482	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
HCP5	hgnc:21659	HCP5	PharmGKB	4/5/24	NULL	1.591141552596803	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	BGB3245	ncit:C173633	BRAF INHIBITOR BGB-3245	FALSE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	1.050153425	interferon alfa-n1	rxcui:202912	INTERFERON ALFA-N1	FALSE	TRUE	FALSE
ARG1	hgnc:663	ARG1	PharmGKB	4/5/24	NULL	NULL	selective beta-2-adrenoreceptor agonists	NULL	NULL	NULL	NULL	NULL
CYP24A1	hgnc:2602	CYP24A1	PharmGKB	4/5/24	NULL	2.917092846427472	tenofovir disoproxil fumarate	rxcui:322248	TENOFOVIR DISOPROXIL FUMARATE	TRUE	FALSE	FALSE
FMO2	hgnc:3770	FMO2	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	binder	2.282942227638891	COL-1	chembl:CHEMBL2109491	COL-1	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.05413162	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
BLVRB	hgnc:1063	BLVRB	PharmGKB	4/5/24	NULL	0.1973972602845657	methylene blue	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:2069	hgnc:3443	EREG	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:7836	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
ADAM33	hgnc:15478	ADAM33	PharmGKB	4/5/24	NULL	2.625383561784725	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
BCHE	hgnc:983	BCHE	PharmGKB	4/5/24	NULL	NULL	oxymetazoline and tetracaine	NULL	NULL	NULL	NULL	NULL
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	NULL	FOLFIRI	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	3.938075342677087	Maraviroc	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	NULL	FOLFIRI	NULL	NULL	NULL	NULL	NULL
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	NULL	FOLFIRI	NULL	NULL	NULL	NULL	NULL
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	NULL	FOLFIRI	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	MyCancerGenome	20-Jun-17	inhibitor	0.760980743	LY2784544	ncit:C116857	GANDOTINIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	desmethyl clomipramine	NULL	NULL	NULL	NULL	NULL
ALDH1A1	hgnc:402	ALDH1A1	PharmGKB	4/5/24	NULL	0.023598953	thiotepa	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.012043044	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
NUDT15	hgnc:23063	NUDT15	PharmGKB	4/5/24	NULL	4.375639269641208	acyclovir	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	0.5966780822238011	lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	NULL	antiinflammatory and antirheumatic products, non-steroids	NULL	NULL	NULL	NULL	NULL
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	NULL	Coxibs	NULL	NULL	NULL	NULL	NULL
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.9907107780319716	DEHYDROXYMETHYLEPOXYQUINOMICIN	chembl:CHEMBL169300	DEHYDROXYMETHYLEPOXYQUINOMICIN	FALSE	FALSE	FALSE
CHRNA5	hgnc:1959	CHRNA5	PharmGKB	4/5/24	NULL	0.9723642821424908	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	PharmGKB	4/5/24	NULL	0.2917092846427472	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
NT5C3A	hgnc:17820	NT5C3A	PharmGKB	4/5/24	NULL	1.093909817410302	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
CYP2C18	hgnc:2620	CYP2C18	PharmGKB	4/5/24	NULL	3.500511415712967	acenocoumarol	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	PharmGKB	4/5/24	NULL	0.084254928	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.037345428	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
FTO	hgnc:24678	FTO	PharmGKB	4/5/24	NULL	0.3454452054979901	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.073385984	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.1555782851427985	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.039068208	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
ERICH3	hgnc:25346	ERICH3	PharmGKB	4/5/24	NULL	1.000146118775133	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:12064	iuphar.ligand:12064	DANUGLIPRON	FALSE	FALSE	FALSE
ECT2L	hgnc:21118	ECT2L	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
CYP4X1	hgnc:20244	CYP4X1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
HNMT	hgnc:5028	HNMT	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
CBR1	hgnc:1548	CBR1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.7059854956059763	Bavencio	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
ABCB4	hgnc:45	ABCB4	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
GPR35	hgnc:4492	GPR35	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.6177373086552294	Anti-PD-L1	chembl:CHEMBL3707227	ATEZOLIZUMAB	FALSE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
SPG7	hgnc:11237	SPG7	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
SULT2B1	hgnc:11459	SULT2B1	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
CDK2	hgnc:1771	CDK2	CancerCommons	25-Jul-13	inhibitor	0.6819178082557726	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.4487835148349958	ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.9723642821424906	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.2917092846427472	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
POU5F1	hgnc:9221	POU5F1	PharmGKB	4/5/24	NULL	0.6250913242344582	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SLCO2A1	hgnc:10955	SLCO2A1	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	CancerCommons	25-Jul-13	inhibitor	0.1842374429322613	GSK1363089	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
CERS6	hgnc:23826	CERS6	PharmGKB	4/5/24	NULL	0.8468979231563629	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
RGL4	hgnc:31911	RGL4	PharmGKB	4/5/24	NULL	7.501095890813499	o-desmethyltramadol	chembl:CHEMBL4650315	DESMETRAMADOL	FALSE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.2344092465879218	spironolactone	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
HYKK	hgnc:34403	HYKK	PharmGKB	4/5/24	NULL	10.50153425	varenicline	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.012683012	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	CancerCommons	25-Jul-13	inhibitor	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.025795957	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TNFRSF1B	hgnc:11917	TNFRSF1B	PharmGKB	4/5/24	NULL	0.5250767123569451	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
SLC30A8	hgnc:20303	SLC30A8	PharmGKB	4/5/24	NULL	NULL	insulin recombinant	NULL	NULL	NULL	NULL	NULL
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	NULL	atazanavir / ritonavir	NULL	NULL	NULL	NULL	NULL
BRCA2	hgnc:1101	BRCA2	CGI	2/1/22	NULL	0.021301287	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
THRA	hgnc:11796	THRA	PharmGKB	4/5/24	NULL	0.1063985232739503	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	NULL	2-oxo-clopidogrel	NULL	NULL	NULL	NULL	NULL
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	NULL	S-EDDP	NULL	NULL	NULL	NULL	NULL
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	NULL	cotinine glucuronide	NULL	NULL	NULL	NULL	NULL
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.11707396	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.637458239	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.3125456621172291	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
SIK3	hgnc:29165	SIK3	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
SMAD7	hgnc:6773	SMAD7	PharmGKB	4/5/24	NULL	NULL	FOLFOX	NULL	NULL	NULL	NULL	NULL
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	NULL	FOLFOX	NULL	NULL	NULL	NULL	NULL
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.01402074	alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PSORS1C1	hgnc:17202	PSORS1C1	PharmGKB	4/5/24	NULL	0.5000730593875666	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	3.150460274	velpatasvir	rxcui:1799206	VELPATASVIR	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	3.500511415712966	velpatasvir	rxcui:1799206	VELPATASVIR	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	PharmGKB	4/5/24	NULL	0.005958317	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
F2R	hgnc:3537	F2R	PharmGKB	4/5/24	NULL	0.057291513	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.1766118064547324	dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
WDR24	hgnc:20852	WDR24	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.012413161	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CHEK2	hgnc:16627	CHEK2	CGI	2/1/22	NULL	0.1754935535952356	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
ST6GAL1	hgnc:10860	ST6GAL1	PharmGKB	4/5/24	NULL	11.66837138570989	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.4167275494896389	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	NULL	antiinflammatory and antirheumatic products, non-steroids	NULL	NULL	NULL	NULL	NULL
ADH1A	hgnc:249	ADH1A	PharmGKB	4/5/24	NULL	0.1367387271762877	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.062808219	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
SULT1A3	hgnc:11455	SULT1A3	PharmGKB	4/5/24	NULL	4.375639269641208	tapentadol	rxcui:787390	TAPENTADOL	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	CGI	2/1/22	NULL	0.088935758	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	PharmGKB	4/5/24	NULL	0.2567612285364034	olutasidenib	rxcui:2623641	OLUTASIDENIB	TRUE	FALSE	FALSE
LTC4S	hgnc:6719	LTC4S	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	CGI	2/1/22	NULL	0.025929714	Nintedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
GLCCI1	hgnc:18713	GLCCI1	PharmGKB	4/5/24	NULL	0.9131768910555564	triamcinolone	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
MOBP	hgnc:7189	MOBP	PharmGKB	4/5/24	NULL	105.0153424713889	creatine	rxcui:2907	CREATINE	TRUE	FALSE	FALSE
NME2	hgnc:7850	NME2	PharmGKB	4/5/24	NULL	0.7501095890813498	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
AK4	hgnc:363	AK4	PharmGKB	4/5/24	NULL	1.875273972703374	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.1298891063344329	dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PRKCH	hgnc:9403	PRKCH	CGI	2/1/22	NULL	0.095468493	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
EGLN2	hgnc:14660	EGLN2	PharmGKB	4/5/24	NULL	NULL	3-hydroxycotinine	NULL	NULL	NULL	NULL	NULL
PRORP	hgnc:19958	PRORP	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
MLLT3	hgnc:7136	MLLT3	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.01609924	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.1521961485092594	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.4327555321623172	ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	NULL	olanzapine 10-n-glucuronide	NULL	NULL	NULL	NULL	NULL
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.054695491	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
GLT1D1	hgnc:26483	GLT1D1	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	1.363835616511545	pamidronate	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
PML	hgnc:9113	PML	CGI	2/1/22	NULL	1.346350544504987	Arsenic Trioxide	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.09869863	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	TALC	12-May-16	inhibitor	0.1480131676834235	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.1123399042269886	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.1181009249565778	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.3059887601147698	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.1842374429322613	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
PML	hgnc:9113	PML	CGI	2/1/22	NULL	1.750255707856483	Volasertib	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	0.4245903334422736	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	NULL	ALN-VSP	NULL	NULL	NULL	NULL	NULL
UNIPROT:P02671	hgnc:3661	FGA	TdgClinicalTrial	Jan-14	NULL	3.182283105193605	ALFIMEPRASE	ncit:C79877	ALFIMEPRASE	FALSE	FALSE	FALSE
PTCH1	hgnc:9585	PTCH1	CGI	2/1/22	NULL	19.69037671338543	Vismodegib	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	NULL	ALN-VSP	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	NULL	ALN-VSP	NULL	NULL	NULL	NULL	NULL
UNIPROT:P52732	hgnc:6388	KIF11	TdgClinicalTrial	Jan-14	NULL	NULL	ALN-VSP	NULL	NULL	NULL	NULL	NULL
UNIPROT:O14788	hgnc:11926	TNFSF11	TdgClinicalTrial	Jan-14	NULL	NULL	ALX-0141	NULL	NULL	NULL	NULL	NULL
UNIPROT:P40933	hgnc:5977	IL15	TdgClinicalTrial	Jan-14	NULL	NULL	AMG0714	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	NULL	ALS 2-0426	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	NULL	AOD9604	NULL	NULL	NULL	NULL	NULL
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	PYRILAMINE MALEATE	rxcui:82091	PYRILAMINE MALEATE	TRUE	FALSE	FALSE
UNIPROT:Q01726	hgnc:6929	MC1R	TdgClinicalTrial	Jan-14	NULL	NULL	AP1030	NULL	NULL	NULL	NULL	NULL
UNIPROT:P32245	hgnc:6932	MC4R	TdgClinicalTrial	Jan-14	NULL	NULL	AP1030	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q92847	hgnc:4267	GHSR	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	ANAMORELIN	ncit:C52197	ANAMORELIN	FALSE	FALSE	FALSE
UNIPROT:P00740	hgnc:3551	F9	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	ANTIHEMOPHILIC FACTOR	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.068637479	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	TRIPELENNAMINE HYDROCHLORIDE	rxcui:91063	TRIPELENNAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P25103	hgnc:11526	TACR1	TdgClinicalTrial	Jan-14	NULL	2.838252499226729	APREPITANT	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	AZATADINE MALEATE	rxcui:58275	AZATADINE MALEATE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.061992528	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O00305	hgnc:1404	CACNB4	TdgClinicalTrial	Jan-14	NULL	0.4039051633514962	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.061197752	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P54284	hgnc:1403	CACNB3	TdgClinicalTrial	Jan-14	NULL	0.4039051633514962	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.058931169	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	BUCLIZINE HYDROCHLORIDE	rxcui:91070	BUCLIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.049337723	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.064505739	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P02686	hgnc:6925	MBP	TdgClinicalTrial	Jan-14	NULL	NULL	ATX-MS-1467	NULL	NULL	NULL	NULL	NULL
UNIPROT:P29474	hgnc:7876	NOS3	TdgClinicalTrial	Jan-14	NULL	NULL	ENOS PLASMID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	NULL	AVN-322	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q02750	hgnc:6840	MAP2K1	TdgClinicalTrial	Jan-14	NULL	NULL	AZD6244, ARRY-142886	NULL	NULL	NULL	NULL	NULL
INHA	hgnc:6065	INHA	ChEMBL	33	inhibitor	1.944728564284981	ISONIAZID	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
UNIPROT:P36507	hgnc:6842	MAP2K2	TdgClinicalTrial	Jan-14	NULL	NULL	AZD6244, ARRY-142886	NULL	NULL	NULL	NULL	NULL
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	BGG-492	chembl:CHEMBL3545042	SELURAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.3977853881492007	BGG-492	chembl:CHEMBL3545042	SELURAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P78380	hgnc:8133	OLR1	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	BI-204	chembl:CHEMBL2109533	ORTICUMAB	FALSE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	0.364636606	METHYSERGIDE MALEATE	rxcui:203190	METHYSERGIDE MALEATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	NULL	BIM23A760	NULL	NULL	NULL	NULL	NULL
UNIPROT:P30874	hgnc:11331	SSTR2	TdgClinicalTrial	Jan-14	NULL	NULL	BIM23A760	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35346	hgnc:11334	SSTR5	TdgClinicalTrial	Jan-14	NULL	NULL	BIM23A760	NULL	NULL	NULL	NULL	NULL
UNIPROT:P53779	hgnc:6872	MAPK10	TdgClinicalTrial	Jan-14	NULL	NULL	JNK-401	NULL	NULL	NULL	NULL	NULL
UNIPROT:P45983	hgnc:6881	MAPK8	TdgClinicalTrial	Jan-14	NULL	NULL	JNK-401	NULL	NULL	NULL	NULL	NULL
UNIPROT:P45984	hgnc:6886	MAPK9	TdgClinicalTrial	Jan-14	NULL	NULL	JNK-401	NULL	NULL	NULL	NULL	NULL
UNIPROT:P06731	hgnc:1817	CEACAM5	TdgClinicalTrial	Jan-14	NULL	NULL	CEA/MUC-1/VF/TRICOM	NULL	NULL	NULL	NULL	NULL
UNIPROT:P15941	hgnc:7508	MUC1	TdgClinicalTrial	Jan-14	NULL	NULL	CEA/MUC-1/VF/TRICOM	NULL	NULL	NULL	NULL	NULL
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	NULL	SYNTHETIC CONJUGATED ESTROGENS	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	NULL	SYNTHETIC CONJUGATED ESTROGENS	NULL	NULL	NULL	NULL	NULL
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.079798892	ETHOPROPAZINE HYDROCHLORIDE	rxcui:6541	ETHOPROPAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.364636606	CHIDAMIDE	hemonc:99	CHIDAMIDE	FALSE	FALSE	FALSE
UNIPROT:P63316	hgnc:11943	TNNC1	TdgClinicalTrial	Jan-14	NULL	NULL	TIRAMSETIV	NULL	NULL	NULL	NULL	NULL
UNIPROT:P02585	hgnc:11944	TNNC2	TdgClinicalTrial	Jan-14	NULL	NULL	TIRAMSETIV	NULL	NULL	NULL	NULL	NULL
UNIPROT:P19237	hgnc:11945	TNNI1	TdgClinicalTrial	Jan-14	NULL	NULL	TIRAMSETIV	NULL	NULL	NULL	NULL	NULL
PTGER2	hgnc:9594	PTGER2	ChEMBL	33	agonist	0.5707355569097228	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
UNIPROT:P48788	hgnc:11946	TNNI2	TdgClinicalTrial	Jan-14	NULL	NULL	TIRAMSETIV	NULL	NULL	NULL	NULL	NULL
UNIPROT:P45379	hgnc:11949	TNNT2	TdgClinicalTrial	Jan-14	NULL	NULL	TIRAMSETIV	NULL	NULL	NULL	NULL	NULL
UNIPROT:O60840	hgnc:1393	CACNA1F	TdgClinicalTrial	Jan-14	NULL	0.3571950424196904	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
UNIPROT:P08174	hgnc:2665	CD55	TdgClinicalTrial	Jan-14	NULL	NULL	COXSACKIEVIRUS TYPE A21	NULL	NULL	NULL	NULL	NULL
UNIPROT:P05362	hgnc:5344	ICAM1	TdgClinicalTrial	Jan-14	NULL	NULL	COXSACKIEVIRUS TYPE A21	NULL	NULL	NULL	NULL	NULL
UNIPROT:P29803	hgnc:8807	PDHA2	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
UNIPROT:P08559	hgnc:8806	PDHA1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141H	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141H	NULL	NULL	NULL	NULL	NULL
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141H	NULL	NULL	NULL	NULL	NULL
UNIPROT:P22455	hgnc:3691	FGFR4	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141H	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.1682938180631233	ESMIRTAZAPINE	ncit:C76963	ESMIRTAZAPINE	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.035890411	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.2365210416022274	METHYSERGIDE MALEATE	rxcui:203190	METHYSERGIDE MALEATE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.030368809	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.059297201	METOCLOPRAMIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.03140411	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.3804903712731485	DEXTROMETHORPHAN HYDROBROMIDE	rxcui:102490	DEXTROMETHORPHAN HYDROBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.033701971	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.035430277	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:Q99572	hgnc:8537	P2RX7	TdgClinicalTrial	Jan-14	NULL	NULL	EVT-401	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43405	hgnc:11491	SYK	TdgClinicalTrial	Jan-14	NULL	NULL	ACU-XSP-001	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01127	hgnc:8800	PDGFB	TdgClinicalTrial	Jan-14	NULL	NULL	ADENOVIRAL PDGF B	NULL	NULL	NULL	NULL	NULL
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	NULL	EXEBRYL-1	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10636	hgnc:6893	MAPT	TdgClinicalTrial	Jan-14	NULL	NULL	EXEBRYL-1	NULL	NULL	NULL	NULL	NULL
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.045898314	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.037345428	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	NULL	FK352B	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43405	hgnc:11491	SYK	TdgClinicalTrial	Jan-14	NULL	3.000438356	FOSTAMATINIB	rxcui:2044896	FOSTAMATINIB	TRUE	FALSE	TRUE
UNIPROT:Q9UNN8	hgnc:9452	PROCR	TdgClinicalTrial	Jan-14	NULL	NULL	GED-APC	NULL	NULL	NULL	NULL	NULL
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.064111931	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
UNIPROT:P35557	hgnc:4195	GCK	TdgClinicalTrial	Jan-14	NULL	NULL	LY-2599506	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00451	hgnc:3546	F8	TdgClinicalTrial	Jan-14	NULL	NULL	MAX-AD FACTOR VIII	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	NULL	MDX-214	NULL	NULL	NULL	NULL	NULL
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.026626608	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	NULL	MEM 63908	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9BYF1	hgnc:13557	ACE2	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	LISINOPRIL	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P04629	hgnc:8031	NTRK1	TdgClinicalTrial	Jan-14	NULL	2.157849503	MIM-D3	chembl:CHEMBL3544981	TAVILERMIDE	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	MK-6913	chembl:CHEMBL3545274	MK-6913	FALSE	FALSE	FALSE
UNIPROT:P13945	hgnc:288	ADRB3	TdgClinicalTrial	Jan-14	NULL	NULL	MN-246	NULL	NULL	NULL	NULL	NULL
UNIPROT:P15941	hgnc:7508	MUC1	TdgClinicalTrial	Jan-14	NULL	NULL	BREVAREX MAB	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21860	hgnc:3431	ERBB3	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	MM-111	drugbank:DB17983	MM-111	FALSE	TRUE	TRUE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.055740628	MN-201	chembl:CHEMBL4297361	1.ALPHA.-HYDROXYVITAMIN D5	FALSE	FALSE	FALSE
UNIPROT:Q9HCU0	hgnc:18219	CD248	TdgClinicalTrial	Jan-14	NULL	157.5230137070835	MORAB-004	ncit:C82406	ONTUXIZUMAB	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.035098711	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P29475	hgnc:7872	NOS1	TdgClinicalTrial	Jan-14	NULL	NULL	ISOTHIOUREA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35228	hgnc:7873	NOS2	TdgClinicalTrial	Jan-14	NULL	NULL	ISOTHIOUREA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P29474	hgnc:7876	NOS3	TdgClinicalTrial	Jan-14	NULL	NULL	ISOTHIOUREA	NULL	NULL	NULL	NULL	NULL
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	3.750547945	TAFLUPROST	rxcui:1244607	TAFLUPROST	TRUE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	NULL	MVA-BN-HER-2	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.036977233	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.04907259	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q15858	hgnc:10597	SCN9A	TdgClinicalTrial	Jan-14	NULL	NULL	NAV 1.7 BLOCKER	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	NULL	PEG-NALOXOL	NULL	NULL	NULL	NULL	NULL
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	NULL	17-BETA ESTRADIOL	NULL	NULL	NULL	NULL	NULL
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1204304386139782	LOPERAMIDE HYDROCHLORIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	NULL	17-BETA ESTRADIOL	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	NULL	NRX-5183	NULL	NULL	NULL	NULL	NULL
UNIPROT:P39086	hgnc:4579	GRIK1	TdgClinicalTrial	Jan-14	NULL	NULL	NS-1209	NULL	NULL	NULL	NULL	NULL
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.3241214273808302	DEXTROAMPHETAMINE ADIPATE	chembl:CHEMBL1200782	DEXTROAMPHETAMINE ADIPATE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	NULL	NSD-644	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	NULL	NSD-644	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	NULL	NSD-644	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	NULL	NSD-788	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	NULL	NSD-788	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	1.400204566285186	SOMATROPIN RECOMBINANT	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1111665587205952	HYDROMORPHONE	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.5738543304447485	NORELGESTROMIN	rxcui:326374	NORELGESTROMIN	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	1.615620653405984	NRM8499	chembl:CHEMBL4650301	VALILTRAMIPROSATE	FALSE	FALSE	FALSE
UNIPROT:P05019	hgnc:5464	IGF1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	NNZ-2566	rxcui:2632852	TROFINETIDE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	HYDROMORPHONE	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.5357925636295356	NONACOG ALFA	rxcui:1300488	NONACOG ALFA	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.1691068316769549	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.1480131676834235	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	PB1023	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q08334	hgnc:5965	IL10RB	TdgClinicalTrial	Jan-14	NULL	NULL	PEG-INTERFERON LAMBA	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8IU57	hgnc:18584	IFNLR1	TdgClinicalTrial	Jan-14	NULL	NULL	PEG-INTERFERON LAMBA	NULL	NULL	NULL	NULL	NULL
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.4861821410712453	AMPHETAMINE ASPARTATE	rxcui:221057	AMPHETAMINE ASPARTATE	TRUE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	0.9376369863516874	RECOMBINANT INTERFERON ALFA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P18858	hgnc:6598	LIG1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	ANILERIDINE HYDROCHLORIDE	rxcui:235413	ANILERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9NRA0	hgnc:18859	SPHK2	TdgClinicalTrial	Jan-14	NULL	1.875273972703374	PHENOXODIOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
UNIPROT:Q05397	hgnc:9611	PTK2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	PF-04554878	ncit:C79809	DEFACTINIB	FALSE	FALSE	FALSE
UNIPROT:P53350	hgnc:9077	PLK1	TdgClinicalTrial	Jan-14	NULL	NULL	PLK-1 INHIBITOR	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9HCN6	hgnc:14388	GP6	TdgClinicalTrial	Jan-14	NULL	NULL	PR-15	NULL	NULL	NULL	NULL	NULL
FSHR	hgnc:3969	FSHR	ChEMBL	33	agonist	18.37768493249307	FOLLITROPIN ALFA	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:P21453	hgnc:3165	S1PR1	TdgClinicalTrial	Jan-14	NULL	1.166837138570988	PONESIMOD	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.2778183663264258	PIRFENIDONE	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	NULL	PSD-506	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	NULL	PSD-506	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.2169738480813822	PROPAFENONE	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	DEXAMETHASONE ACETATE	rxcui:22690	DEXAMETHASONE ACETATE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	0.4434769530041765	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	0.1861974157294131	TEGAFUR	rxcui:10995	URACIL	TRUE	FALSE	TRUE
UNIPROT:P13612	hgnc:6140	ITGA4	TdgClinicalTrial	Jan-14	NULL	3.889457128569962	FIRATEGRAST	ncit:C76692	FIRATEGRAST	FALSE	FALSE	FALSE
UNIPROT:P30988	hgnc:1440	CALCR	TdgClinicalTrial	Jan-14	NULL	1.875273972703374	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.038173516	HYDROCORTISONE BUTYRATE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	TEPLIZUMAB	rxcui:2621880	TEPLIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	TONABERSAT	ncit:C97277	TONABERSAT	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.7119684235348407	TRANDOLAPRIL	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
NA	hgnc:12811	XK	ChEMBL	33	inhibitor	1.693795846312725	ZANAMIVIR	rxcui:69722	ZANAMIVIR	TRUE	FALSE	FALSE
UNIPROT:P32239	hgnc:1571	CCKBR	TdgClinicalTrial	Jan-14	NULL	NULL	TT-223	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01133	hgnc:3229	EGF	TdgClinicalTrial	Jan-14	NULL	NULL	TT-223	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	TT-223	NULL	NULL	NULL	NULL	NULL
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	1.186614039224734	VALSARTAN	rxcui:69749	VALSARTAN	TRUE	FALSE	FALSE
UNIPROT:P30874	hgnc:11331	SSTR2	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	VAPREOTIDE	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
UNIPROT:P35346	hgnc:11334	SSTR5	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	VAPREOTIDE	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
UNIPROT:P14555	hgnc:9031	PLA2G2A	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	VARESPLADIB	ncit:C152832	VARESPLADIB	FALSE	FALSE	FALSE
UNIPROT:P30926	hgnc:1964	CHRNB4	TdgClinicalTrial	Jan-14	NULL	0.4375639269641209	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	GLP1 AGONIST	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	NULL	VIROSOME-BASED BREAST CANCER VACCINE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	NULL	VR-147	NULL	NULL	NULL	NULL	NULL
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1752592497853621	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	NULL	VR-147	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NR97	hgnc:15632	TLR8	TdgClinicalTrial	Jan-14	NULL	NULL	VTX-1463	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.1280674908187671	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.092606122	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.094950581	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1282238613814273	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.089298761	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.096167896	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.091476779	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UGCG	hgnc:12524	UGCG	ChEMBL	33	inhibitor	7.001022831425932	MIGLUSTAT	rxcui:402316	MIGLUSTAT	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	CLIDINIUM	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	0.729273212	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
UNIPROT:P19235	hgnc:3416	EPOR	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	DARBEPOETIN ALFA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.8607814956671229	DESOGESTREL	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.1408971500063358	ERGOLOID MESYLATE	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.089756703	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.05309168	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.084553416	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.08780547	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.3006164383722967	FLUMETHASONE PIVALATE	rxcui:25113	FLUMETHASONE PIVALATE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	0.8334550989792778	FUROSEMIDE	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	GLICLAZIDE	rxcui:4816	GLICLAZIDE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.091583148	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	2.258394462	GOLIMUMAB	rxcui:819300	GOLIMUMAB	TRUE	TRUE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.061055432	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P23921	hgnc:10451	RRM1	TdgClinicalTrial	Jan-14	NULL	0.4412409347537352	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
UNIPROT:P06276	hgnc:983	BCHE	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	ISOFLUROPHATE	rxcui:6027	ISOFLUROPHATE	TRUE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	0.061791905	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.100976291	MESORIDAZINE	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.3804903712731485	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.053145416	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1017590527823536	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q14432	hgnc:8778	PDE3A	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	MILRINONE	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.28382525	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.7778914257139926	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.4118248724368196	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.9723642821424908	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.108711535	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	inhibitor	0.2044691247495891	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	0.3170753093942904	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1376347869874036	PENTAZOCINE	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
UNIPROT:P47872	hgnc:10608	SCTR	TdgClinicalTrial	Jan-14	NULL	15.75230137070834	SECRETIN	rxcui:9627	SECRETIN	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.1123158743009508	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P08514	hgnc:6138	ITGA2B	TdgClinicalTrial	Jan-14	NULL	3.500511415712967	TIROFIBAN	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.2763561643983921	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.201178817	DEXLANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	0.546954909	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
UNIPROT:P25021	hgnc:5183	HRH2	TEND	1-Aug-11	NULL	0.9376369863516874	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.2206204673768676	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TEND	1-Aug-11	NULL	1.988926940746003	ABARELIX	rxcui:301739	ABARELIX	TRUE	FALSE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1363127498330594	CONJUGATED ESTROGENS	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.375054795	OSPEMIFENE	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
UNIPROT:P43116	hgnc:9594	PTGER2	TEND	1-Aug-11	NULL	0.6563458904461813	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.8468979231563628	DIMENHYDRINATE	rxcui:3444	DIMENHYDRINATE	TRUE	FALSE	FALSE
DRD5	hgnc:3026	DRD5	ChEMBL	33	agonist	0.3750547945406749	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	2.100306849	DICHLORPHENAMIDE	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TEND	1-Aug-11	NULL	0.6177373086552295	EPOETIN ALFA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.080225625	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TEND	1-Aug-11	NULL	0.4526523382387456	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.3006164383722967	FLUMETHASONE PIVALATE	rxcui:25113	FLUMETHASONE PIVALATE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.1367387271762877	ALFUZOSIN HYDROCHLORIDE	rxcui:46043	ALFUZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.070197421	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.07182992	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.06757744	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.05814803	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.182318303	PHENYLEPHRINE BITARTRATE	rxcui:91167	PHENYLEPHRINE BITARTRATE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	0.5791287268642775	GALANTAMINE	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.2282942227638891	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.062139256	CARVEDILOL PHOSPHATE	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:P23921	hgnc:10451	RRM1	TEND	1-Aug-11	NULL	0.4412409347537352	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.2692701089009974	HYDROMORPHONE	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TEND	1-Aug-11	NULL	0.053038052	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.3088686543276147	ISOSORBIDE MONONITRATE	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.2616661357260523	LOFEXIDINE	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.4817217544559128	METHADYL ACETATE	rxcui:6814	METHADYL ACETATE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.100976291	MESORIDAZINE	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.2734774543525755	METHOXAMINE	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.060772768	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.3804903712731485	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1785975212098452	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.024241769	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.019929531	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.064111931	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1111665587205952	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2713574740862764	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.5427149481725528	PROCATEROL	rxcui:34530	PROCATEROL	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.015123177	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.2169738480813822	PROPAFENONE	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.2187819634820604	PROPERICIAZINE	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.09969811	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.093763699	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.2014360789093139	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	INNO-305	NULL	NULL	NULL	NULL	NULL
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.3409589041278863	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	BN-AA-003-NY	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	BN-CB-045	NULL	NULL	NULL	NULL	NULL
PROTEASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-2551	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	NULL	ASP-7035	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	DE-110	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.3889457128569962	OX-914	chembl:CHEMBL4297287	HT-0712	FALSE	FALSE	FALSE
ABAT	hgnc:23	ABAT	ChEMBL	33	inhibitor	0.6035364509849942	VIGABATRIN	rxcui:14851	VIGABATRIN	TRUE	FALSE	FALSE
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	NULL	BAX-817	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Research programme: peroxisome proliferator-activated receptor gamma agonist, Omeros	NULL	NULL	NULL	NULL	NULL
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	SCH-900978	NULL	NULL	NULL	NULL	NULL
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BI-847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
CD80	hgnc:1700	CD80	ChEMBL	33	inhibitor	1.750255707856483	BELATACEPT	rxcui:1112973	BELATACEPT	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	NULL	PD-200390	NULL	NULL	NULL	NULL	NULL
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	NULL	NKP-46	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	NULL	OTSGC-A24	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	OTSGC-A24	NULL	NULL	NULL	NULL	NULL
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	agonist	0.5000730593875667	DECAMETHONIUM BROMIDE	ncit:C65365	DECAMETHONIUM BROMIDE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CTP-298	NULL	NULL	NULL	NULL	NULL
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	DNA fusion vaccine	NULL	NULL	NULL	NULL	NULL
AROMATIC-L-AMINO-ACID DECARBOXYLASE	hgnc:2719	DDC	TTD	2020.06.01	NULL	NULL	AV-201	NULL	NULL	NULL	NULL	NULL
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	NULL	AMG 899	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aprocitentan	ncit:C174728	APROCITENTAN	TRUE	FALSE	FALSE
ANGIOGENESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABI-011	ncit:C116890	NANOPARTICLE ALBUMIN-BOUND THIOCOLCHICINE DIMER NAB-5404	FALSE	FALSE	FALSE
ADH1A	hgnc:249	ADH1A	ChEMBL	33	inhibitor	3.281729452230906	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
COAGULATION FACTOR XI	hgnc:3529	F11	TTD	2020.06.01	NULL	1.381780822	EP-7041	iuphar.ligand:11990	EP-7041	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	BGB-3113	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN CD47	hgnc:1682	CD47	TTD	2020.06.01	NULL	13.12691780892362	ALX148	ncit:C132851	EVORPACEPT	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	NULL	DS-1205	NULL	NULL	NULL	NULL	NULL
GLRB	hgnc:4329	GLRB	ChEMBL	33	positive modulator	0.1419126249613364	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
PROTEIN ARGININE METHYLTRANSFERASE 5	hgnc:10894	PRMT5	TTD	2020.06.01	NULL	11.66837138570988	GSK3326595	ncit:C142177	PEMRAMETOSTAT	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	0.4861821410712453	CYC065	ncit:C123902	FADRACICLIB	FALSE	FALSE	TRUE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.4039051633514961	KA2237	ncit:C126271	PI3K P110BETA/DELTA INHIBITOR KA2237	FALSE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	0.4795221117415022	LOXO-195	ncit:C138160	SELITRECTINIB	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	3.750547945	KHK2455	drugbank:DB17524	KHK2455	FALSE	FALSE	FALSE
EGFR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrotinib	ncit:C111895	PYROTINIB	FALSE	FALSE	FALSE
PDE7B	hgnc:8792	PDE7B	ChEMBL	33	inhibitor	0.375054795	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
CALCIUM-RELEASE ACTIVATED CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	RP4010	ncit:C136828	CALCIUM RELEASE-ACTIVATED CHANNELS INHIBITOR RP4010	FALSE	FALSE	FALSE
WNT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	SM08502	ncit:C142777	WNT SIGNALING PATHWAY INHIBITOR SM08502	FALSE	FALSE	FALSE
EGFR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CK-101	ncit:C132023	EGFR MUTANT-SPECIFIC INHIBITOR CK-101	FALSE	FALSE	FALSE
EXPORTIN-1	hgnc:12825	XPO1	TTD	2020.06.01	NULL	NULL	Eltanexor oral	NULL	NULL	NULL	NULL	NULL
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.029106248	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	GLG-801	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	1.458546423213736	CPI-1205	drugbank:DB14581	CPI-1205	FALSE	FALSE	FALSE
XIAP MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASTX660	ncit:C123913	TOLINAPANT	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	NULL	Bavencio avelumab	NULL	NULL	NULL	NULL	NULL
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.083257407	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	NULL	Bavencio avelumab	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.2500365296937833	Sym015	ncit:C127906	ANTI-MET MONOCLONAL ANTIBODY MIXTURE SYM015	FALSE	FALSE	FALSE
HIF1-ALPHA MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PT2385	iuphar.ligand:12707	PT2385	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NYX-2925	iuphar.ligand:11289	NYX-2925	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.028413242	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
HIF2-ALPHA MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PT2385	iuphar.ligand:12707	PT2385	FALSE	FALSE	FALSE
IMMUNOGLOBULIN FC RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.019695301	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
TRANSFORMING PROTEIN RHO	hgnc:10012	RHO	TTD	2020.06.01	NULL	NULL	VX-210	NULL	NULL	NULL	NULL	NULL
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.020164236	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	NULL	Application submitted	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	MD1003	NULL	NULL	NULL	NULL	NULL
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	NULL	JNJ-3534	NULL	NULL	NULL	NULL	NULL
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
TRANSCRIPTION FACTOR UNSPECIFIC	hgnc:11740	TF	TTD	2020.06.01	NULL	NULL	PF-06763809	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	SNA-125	NULL	NULL	NULL	NULL	NULL
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	NULL	ESR0114	NULL	NULL	NULL	NULL	NULL
CALGRANULIN D	hgnc:10489	S100A12	TTD	2020.06.01	NULL	5.250767123569449	MK-1602	rxcui:2268216	UBROGEPANT	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.093763699	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
PROTEIN SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Contezolid	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
PROTEIN SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Contezolid acefosamil	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	IFX-1	ncit:C172643	VILOBELIMAB	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	MM36 topical ointment	NULL	NULL	NULL	NULL	NULL
WNT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	SM04554	chembl:CHEMBL4650339	DALOSIRVAT	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-3/BETA-4	NULL	NULL	TTD	2020.06.01	NULL	NULL	TC-5214	chembl:CHEMBL2103881	DEXMECAMYLAMINE	FALSE	FALSE	FALSE
HEXOKINASE-2	hgnc:4923	HK2	TTD	2020.06.01	NULL	NULL	VDA-1102 topical ointment	NULL	NULL	NULL	NULL	NULL
VOLTAGE-DEPENDENT ANION-SELECTIVE CHANNEL 1	hgnc:12669	VDAC1	TTD	2020.06.01	NULL	NULL	VDA-1102 topical ointment	NULL	NULL	NULL	NULL	NULL
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
PROTEIN PHOSPHATASE 1A	hgnc:9275	PPM1A	TTD	2020.06.01	NULL	NULL	VP-102	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE PP2A-ALPHA	hgnc:9299	PPP2CA	TTD	2020.06.01	NULL	NULL	VP-102	NULL	NULL	NULL	NULL	NULL
VIRUS REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	CLS006	ncit:C153417	FUROSEMIDE TOPICAL GEL CLS006	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	JNJ-54728518	NULL	NULL	NULL	NULL	NULL
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.015768069	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
PYRUVATE DEHYDROGENASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	JTT-251	drugbank:DB18174	JTT-251	FALSE	FALSE	FALSE
MEMBRANE COPPER AMINE OXIDASE	hgnc:550	AOC3	TTD	2020.06.01	NULL	NULL	ASP8232	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	IONIS-GCCRRX	NULL	NULL	NULL	NULL	NULL
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
PROTEIN-TYROSINE PHOSPHATASE 1B	hgnc:9642	PTPN1	TTD	2020.06.01	NULL	NULL	IONIS-PTP1BRX	NULL	NULL	NULL	NULL	NULL
GLUCAGON	hgnc:4191	GCG	TTD	2020.06.01	NULL	NULL	MK-8521	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	MK-8521	NULL	NULL	NULL	NULL	NULL
GLUCAGON	hgnc:4191	GCG	TTD	2020.06.01	NULL	NULL	PB-1023	NULL	NULL	NULL	NULL	NULL
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	1.419126249613364	Serlopitant	ncit:C81499	SERLOPITANT	FALSE	FALSE	FALSE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	TT-401	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	TTP273	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	NULL	VPI-2690B	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	NULL	NGP 555	NULL	NULL	NULL	NULL	NULL
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.017306418	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
BETA-SECRETASE 1	hgnc:933	BACE1	TTD	2020.06.01	NULL	NULL	AMG520	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	ALZT-OP1	NULL	NULL	NULL	NULL	NULL
ALPHA-1-ANTITRYPSIN	hgnc:8941	SERPINA1	TTD	2020.06.01	NULL	NULL	Alpha1-proteinase inhibitor (human) modified process	NULL	NULL	NULL	NULL	NULL
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-02545920	ncit:C170150	MARDEPODECT	FALSE	FALSE	FALSE
BETA-SECRETASE 1	hgnc:933	BACE1	TTD	2020.06.01	NULL	1.346350544504987	verubecestat	ncit:C152868	VERUBECESTAT	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	PB-1023	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	CI-1012	NULL	NULL	NULL	NULL	NULL
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	IFN-alpha	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ED-1812	NULL	NULL	NULL	NULL	NULL
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER	NULL	NULL	TTD	2020.06.01	NULL	NULL	LIM-0705	chembl:CHEMBL4297397	QUERCETIN-3'-O-PHOSPHATE	FALSE	FALSE	FALSE
INTERLEUKIN 1 RECEPTOR TYPE 2	hgnc:5994	IL1R2	TTD	2020.06.01	NULL	NULL	GSK-1827771	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	VA-111913	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	NULL	RQ-00000007 (oral)	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	AZD1979	NULL	NULL	NULL	NULL	NULL
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	DSP-6952	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS CAPSID P24	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vacc-4x	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	BDD-10103	NULL	NULL	NULL	NULL	NULL
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.018193926	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS 791325	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BI 207127	chembl:CHEMBL2403318	DELEOBUVIR	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BI 201335	chembl:CHEMBL1241348	FALDAPREVIR	FALSE	FALSE	FALSE
BASIGIN	hgnc:1116	BSG	TTD	2020.06.01	NULL	13.12691780892362	Gavilimomab	ncit:C2621	GAVILIMOMAB	FALSE	FALSE	FALSE
HISTIDINE DECARBOXYLASE	hgnc:4855	HDC	TTD	2020.06.01	NULL	4.375639269641208	Lixivaptan	ncit:C74429	LIXIVAPTAN	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	MAL formulation	NULL	NULL	NULL	NULL	NULL
HISTAMINE RECEPTOR	hgnc:5172	HR	TTD	2020.06.01	NULL	NULL	ETX-9101	NULL	NULL	NULL	NULL	NULL
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.018193926	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
INTEGRIN BETA-8	hgnc:6163	ITGB8	TTD	2020.06.01	NULL	NULL	US10035778, Example 12	NULL	NULL	NULL	NULL	NULL
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.039598545	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US10040779, Example 1	NULL	NULL	NULL	NULL	NULL
KYNURENINE OXOGLUTARATE TRANSAMINASE II	hgnc:17929	AADAT	TTD	2020.06.01	NULL	NULL	US10065972, Example 560	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10100051, Compound 11	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10100051, Compound 2	NULL	NULL	NULL	NULL	NULL
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	67S	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	BDBM50177012	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10150740, Example 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	1190312-92-5	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US10179791, Compound 296	NULL	NULL	NULL	NULL	NULL
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.049256727	ZOLPIDEM TARTRATE	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	US8470836, 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	US8470836, 8	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US8524917, 10	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8536181, C35	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ZAP-70	hgnc:12858	ZAP70	TTD	2020.06.01	NULL	NULL	US8546370, 11	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ZAP-70	hgnc:12858	ZAP70	TTD	2020.06.01	NULL	NULL	US8546370, 17	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 2	hgnc:3169	S1PR2	TTD	2020.06.01	NULL	NULL	US8975409, Example 9(3)	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	US9006244, E1	NULL	NULL	NULL	NULL	NULL
SRD5A3	hgnc:25812	SRD5A3	ChEMBL	33	inhibitor	6.563458904461812	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9024044, 3	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9024044, 62	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	879325-11-8	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	US9040714, 7	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	SB19065	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	US9073931, E3	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	US9108950, 1	NULL	NULL	NULL	NULL	NULL
PC4 AND SFRS1-INTERACTING PROTEIN	hgnc:9527	PSIP1	TTD	2020.06.01	NULL	NULL	US9132129, Cpd023	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	ZNFTXQFGUIKQQE-UHFFFAOYSA-N	NULL	NULL	NULL	NULL	NULL
SRD5A1	hgnc:11284	SRD5A1	ChEMBL	33	inhibitor	6.563458904461812	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	AC1M1SP5	NULL	NULL	NULL	NULL	NULL
SERINE PROTEASE HEPSIN	hgnc:5155	HPN	TTD	2020.06.01	NULL	NULL	N-Methyl-D-aspartic acid	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9187437, 24	NULL	NULL	NULL	NULL	NULL
PLASMODIUM HYPOXANTHINE-GUANINE PHOSPHORIBOSYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9200020, Table 3 compound 8	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9024044, 1	NULL	NULL	NULL	NULL	NULL
DIBASIC-PROCESSING ENZYME	hgnc:8568	FURIN	TTD	2020.06.01	NULL	NULL	US9266828, C	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9340511, 6	NULL	NULL	NULL	NULL	NULL
AVPR1B	hgnc:896	AVPR1B	ChEMBL	33	agonist	1.666910197958555	DESMOPRESSIN ACETATE	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
PROTEIN-TYROSINE PHOSPHATASE ETA	hgnc:9668	PTPRD	TTD	2020.06.01	NULL	NULL	US9340574, 7	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	BDBM50434164	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	BDBM50434165	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9346821, B-13	NULL	NULL	NULL	NULL	NULL
PLASMODIUM PLASMEPSIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9353089, 135	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	US9359293, TA	NULL	NULL	NULL	NULL	NULL
IL2RG	hgnc:6010	IL2RG	ChEMBL	33	binder	1.750255707856483	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
RIBOSOMAL PROTEIN S6 KINASE ALPHA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9365572, 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 3B	hgnc:8779	PDE3B	TTD	2020.06.01	NULL	NULL	US9388139, 12	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9682991, 2	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	AC1LE05K	NULL	NULL	NULL	NULL	NULL
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	US9695118, 4	NULL	NULL	NULL	NULL	NULL
IFNGR2	hgnc:5440	IFNGR2	ChEMBL	33	agonist	105.0153424713889	INTERFERON GAMMA-1B	rxcui:5882	INTERFERON GAMMA-1B	TRUE	TRUE	FALSE
CHYMOTRYPSIN-C	hgnc:2523	CTRC	TTD	2020.06.01	NULL	NULL	AC1LCOK0	NULL	NULL	NULL	NULL	NULL
CHYMOTRYPSIN-C	hgnc:2523	CTRC	TTD	2020.06.01	NULL	NULL	Z223457004	NULL	NULL	NULL	NULL	NULL
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	NULL	US10053465, 12	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	AC1LFGWU	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	BK3	NULL	NULL	NULL	NULL	NULL
BUB1 MITOTIC CHECKPOINT SERINE/THREONINE KINASE	hgnc:1148	BUB1	TTD	2020.06.01	NULL	NULL	SCHEMBL17766424	NULL	NULL	NULL	NULL	NULL
PROTON-COUPLED FOLATE TRANSPORTER	hgnc:30521	SLC46A1	TTD	2020.06.01	NULL	NULL	PREMETREXED	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	SOTB07	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	NULL	SOTB07	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	NULL	SOTB07	NULL	NULL	NULL	NULL	NULL
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.043180651	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	NP-01	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	TAK-379	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	NN5401	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	NULL	VEGFR3 Monoclonal Antibody	NULL	NULL	NULL	NULL	NULL
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.052090944	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
B-RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	SPN-803	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	INCB039110	ncit:C116855	ITACITINIB	FALSE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	INCB039110	ncit:C116855	ITACITINIB	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	Novolimus	NULL	NULL	NULL	NULL	NULL
RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	SPN-803	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	Human prothrombin complex concentrate	NULL	NULL	NULL	NULL	NULL
LEGUMAIN	hgnc:9472	LGMN	TTD	2020.06.01	NULL	NULL	Legumain-cleavable doxorubicin prodrugs	NULL	NULL	NULL	NULL	NULL
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.044878351	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	AAB-002	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	LATIN T1D	NULL	NULL	NULL	NULL	NULL
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	NULL	OPK-0018	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	CPH-102	NULL	NULL	NULL	NULL	NULL
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	TTP-547	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	1.615620653405984	Crenezumab	ncit:C174789	CRENEZUMAB	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	1.166837138570988	ACT-128800	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	LY-2590443	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	FE-202767	NULL	NULL	NULL	NULL	NULL
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.099446347	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV1.5	hgnc:6224	KCNA5	TTD	2020.06.01	NULL	NULL	XEN-D0103	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Research programme: small molecule therapeutics, Boehringer Ingelheim	NULL	NULL	NULL	NULL	NULL
GASTRIC H(+)/K(+) ATPASE ALPHA	hgnc:819	ATP4A	TTD	2020.06.01	NULL	NULL	API-023	NULL	NULL	NULL	NULL	NULL
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.054243462	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	M-0004	NULL	NULL	NULL	NULL	NULL
SPECTRIN NON-ERYTHROID BETA CHAIN 1	hgnc:11275	SPTBN1	TTD	2020.06.01	NULL	NULL	ABT-413	NULL	NULL	NULL	NULL	NULL
HYALURONIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PEGylated hyaluronidase (human recombinant)	NULL	NULL	NULL	NULL	NULL
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.064111931	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	NULL	VG-101	NULL	NULL	NULL	NULL	NULL
NUCLEOSIDE DNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MBX-400/cyclopropavir	NULL	NULL	NULL	NULL	NULL
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valomaciclovir stearate	ncit:C152820	VALOMACICLOVIR STEARATE	FALSE	FALSE	FALSE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	7.501095891	APD-811	chembl:CHEMBL3301604	RALINEPAG	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	2.333674277141977	GSK3117391	drugbank:DB15440	GSK-3117391	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	2.059124362184098	TT-301	drugbank:DB12899	TT-301	FALSE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	6.848826682916673	YM-598	chembl:CHEMBL2107760	NEBENTAN	FALSE	FALSE	FALSE
INFLUENZA HEMAGGLUTININ	NULL	NULL	TTD	2020.06.01	NULL	NULL	A/Anhui/05	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	AVN 101	NULL	NULL	NULL	NULL	NULL
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.038382801	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS NON-STRUCTURAL 5	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDX-184	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AeroLEF	drugbank:DB05000	AEROLEF	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Apaziquone	ncit:C1087	APAZIQUONE	FALSE	FALSE	FALSE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7420	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.065145994	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	1.591141552596803	Romazarit	ncit:C73094	ROMAZARIT	FALSE	FALSE	FALSE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	AZ-01, PEGylated interferon-beta	NULL	NULL	NULL	NULL	NULL
CLOSTRIDIUM DIFFICILE TOXIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	ACAM-Cdiff	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	AVN 322	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	PCI-45292	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	GSK933776A	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	UB-311	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-12 BETA	hgnc:5970	IL12B	TTD	2020.06.01	NULL	NULL	Ad-RTS-IL-12	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	ACI-24	NULL	NULL	NULL	NULL	NULL
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.067317527	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
BACTERIAL PROTECTIVE ANTIGEN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVP-21D9	drugbank:DB17798	AVP-21D9	FALSE	FALSE	FALSE
HEPATITIS B VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MIV-210	ncit:C90784	LAGOCICLOVIR	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.068458502	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	0.2344092465879218	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ADCI	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	ADCI	NULL	NULL	NULL	NULL	NULL
GAR TRANSFORMYLASE	hgnc:4163	GART	TTD	2020.06.01	NULL	NULL	AG2034	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glitazone	chembl:CHEMBL1061	GLITAZONE	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	T-0128	NULL	NULL	NULL	NULL	NULL
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.020836377	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
CALCIUM RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	NPC-15199	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-33084	NULL	NULL	NULL	NULL	NULL
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.261046661	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.2027323213733378	SCH-442416	iuphar.ligand:3283	SCH442416	FALSE	FALSE	FALSE
FREE RADICAL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Disufenton sodium	ncit:C77600	DISUFENTON SODIUM	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Psoralen	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	CZ-48	NULL	NULL	NULL	NULL	NULL
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
KCNK2	hgnc:6277	KCNK2	ChEMBL	33	potentiator	0.6081969641200136	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Desflurane	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.4861821410712453	KF-17837	chembl:CHEMBL27508	CHEMBL:CHEMBL27508	FALSE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	Anti-MUC1 mab	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulphadoxine	chembl:CHEMBL244800	SULPHADOXINE	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aprobarbital	rxcui:17381	APROBARBITAL	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V4	hgnc:18083	TRPV4	TTD	2020.06.01	NULL	0.2592971419046642	phorbol 12-myristate 13-acetate	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cannabidiol	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
IMMUNOGLOBULIN G	NULL	NULL	TTD	2020.06.01	NULL	NULL	Protein A mimetics	NULL	NULL	NULL	NULL	NULL
KCNK3	hgnc:6278	KCNK3	ChEMBL	33	potentiator	0.6081969641200136	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
INTERLEUKIN 11 RECEPTOR ALPHA	hgnc:5967	IL11RA	TTD	2020.06.01	NULL	NULL	UNI-rhIL-11	NULL	NULL	NULL	NULL	NULL
FUNGAL CELL MEMBRANE ERGOSTEROL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amphotericin B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ciprofloxacin XR	NULL	NULL	NULL	NULL	NULL
CYTOMEGALOVIRUS GANCICLOVIR KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Maribavir	rxcui:2586068	MARIBAVIR	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Levorphanol	rxcui:6378	LEVORPHANOL	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aztreonam	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
NF-KAPPA-B MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oligonucleotide decoys (NFkappaB)	NULL	NULL	NULL	NULL	NULL
KCNK9	hgnc:6283	KCNK9	ChEMBL	33	potentiator	0.2365210416022274	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
CYCLIC NUCLEOTIDE-GATED CHANNEL ALPHA-1	hgnc:2148	CNGA1	TTD	2020.06.01	NULL	1.093909817410302	dequalinium	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR 2	hgnc:11848	TLR2	TTD	2020.06.01	NULL	NULL	Lipoteichoic acid	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	TA-270	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	MC-2001	NULL	NULL	NULL	NULL	NULL
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	2.143170254518142	SILTUXIMAB	rxcui:1535218	SILTUXIMAB	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	MC-2001	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ragaglitazar	ncit:C75192	RAGAGLITAZAR	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.2651902587661338	Ragaglitazar	ncit:C75192	RAGAGLITAZAR	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	SECTA belomycin	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acetylcholine	rxcui:194	ACETYLCHOLINE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Levorphanol	rxcui:6378	LEVORPHANOL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	NULL	Phenylephrine hydrochloride gel	NULL	NULL	NULL	NULL	NULL
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	LENVATINIB MESYLATE	rxcui:1604346	LENVATINIB MESYLATE	TRUE	FALSE	FALSE
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chloramphenicol	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
LACTOTRANSFERRIN	hgnc:6720	LTF	TTD	2020.06.01	NULL	NULL	HLF 1-11	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	NULL	BIBV 308	NULL	NULL	NULL	NULL	NULL
CD3E	hgnc:1674	CD3E	ChEMBL	33	modulator	0.2917092846427472	BLINATUMOMAB	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR	hgnc:2436	CSF2RB	TTD	2020.06.01	NULL	NULL	DT388IL-3	NULL	NULL	NULL	NULL	NULL
TGF-BETA RECEPTOR TYPE I	hgnc:11772	TGFBR1	TTD	2020.06.01	NULL	3.750547945	Metelimumab	ncit:C166745	METELIMUMAB	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	Elsamitrucin	ncit:C1080	ELSAMITRUCIN	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.013836014	ROXINDOLE	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Parthenolide	rxcui:32941	PARTHENOLIDE	FALSE	FALSE	FALSE
PIGMENT EPITHELIUM-DERIVED FACTOR	hgnc:8824	SERPINF1	TTD	2020.06.01	NULL	NULL	PEDF gene therapy	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	McN3377	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TPT-43	NULL	NULL	NULL	NULL	NULL
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.2083637747448194	LENVATINIB MESYLATE	rxcui:1604346	LENVATINIB MESYLATE	TRUE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD4	hgnc:1678	CD4	TTD	2020.06.01	NULL	3.281729452230906	TNX-355	rxcui:2043283	IBALIZUMAB	TRUE	FALSE	FALSE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	0.1562728310586145	FADROZOLE	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	Taxol/Paraplatin/Herceptin	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Taxol/Paraplatin/Herceptin	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Protexia	NULL	NULL	NULL	NULL	NULL
TYMP	hgnc:3148	TYMP	ChEMBL	33	inhibitor	3.281729452230906	TIPIRACIL HYDROCHLORIDE	rxcui:1670303	TIPIRACIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PREMETREXED	NULL	NULL	NULL	NULL	NULL
VEGFR1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	Ximelegatran	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	SRX-251	NULL	NULL	NULL	NULL	NULL
ADENINE SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-alanosine	ncit:C994	ALANOSINE	FALSE	FALSE	FALSE
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	1.400204566285186	Somatropin recombinant	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	MEM-1003	NULL	NULL	NULL	NULL	NULL
SLAMF7	hgnc:21394	SLAMF7	ChEMBL	33	inhibitor	26.25383561784724	ELOTUZUMAB	rxcui:1726104	ELOTUZUMAB	TRUE	FALSE	FALSE
TNF ALPHA CONVERTING ENZYME	hgnc:195	ADAM17	TTD	2020.06.01	NULL	NULL	GW-3333	NULL	NULL	NULL	NULL	NULL
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	2.838252499226729	ATL-313	ncit:C169974	EVODENOSON	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	0.2853677784548614	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	0.6563458904461812	Eptastigmine	ncit:C65525	EPTASTIGMINE	FALSE	FALSE	FALSE
BASIGIN	hgnc:1116	BSG	TTD	2020.06.01	NULL	NULL	[131I]-Metuximab injection	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Minocycline	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
EPSTEIN-BARR VIRUS LATENT MEMBRANE PROTEIN 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	LMP-1/LMP-2 CTLs	NULL	NULL	NULL	NULL	NULL
EPSTEIN-BARR VIRUS LATENT MEMBRANE PROTEIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	LMP-1/LMP-2 CTLs	NULL	NULL	NULL	NULL	NULL
PLASMODIUM ADENYLOSUCCINATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alanosine	ncit:C994	ALANOSINE	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Taxol/Paraplatin/Herceptin	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gemcitabine prodrug	NULL	NULL	NULL	NULL	NULL
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	NULL	Gemcitabine prodrug	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE COMMON ANTIGEN	hgnc:9666	PTPRC	TTD	2020.06.01	NULL	NULL	Anti-CD45 mabs	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-5/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATN-161	drugbank:DB05491	ATN-161	FALSE	FALSE	FALSE
INTEGRIN ALPHA-V/BETA-3	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATN-161	drugbank:DB05491	ATN-161	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	A-348441	chembl:CHEMBL219684	CHEMBL:CHEMBL219684	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefpiramide	ncit:C65303	CEFPIRAMIDE	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.1539814405738841	Phenacemide	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	NULL	TS-022	NULL	NULL	NULL	NULL	NULL
NR1H3	hgnc:7966	NR1H3	ChEMBL	33	agonist	1.250182648468916	CS-8080	chembl:CHEMBL3545238	CS-8080	FALSE	FALSE	FALSE
INTEGRIN ALPHA-L	hgnc:6148	ITGAL	TTD	2020.06.01	NULL	NULL	Cytolin	NULL	NULL	NULL	NULL	NULL
METHIONINE AMINOPEPTIDASE 2	hgnc:16672	METAP2	TTD	2020.06.01	NULL	6.563458904461812	D-Methionine	drugbank:DB02893	D-METHIONINE	FALSE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMG 386	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amitriptyline+ketamine	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	P-276	NULL	NULL	NULL	NULL	NULL
PORPHOBILINOGEN DEAMINASE	hgnc:4982	HMBS	TTD	2020.06.01	NULL	NULL	P-9808	NULL	NULL	NULL	NULL	NULL
TUMOR SUPPRESSOR CANDIDATE 2	hgnc:17034	TUSC2	TTD	2020.06.01	NULL	NULL	Fus-1 tumor suppressor gene therapy - nanoparticle formulation	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C BETA	hgnc:9395	PRKCB	TTD	2020.06.01	NULL	NULL	RUBOXISTAURIN HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
NR1H2	hgnc:7965	NR1H2	ChEMBL	33	modulator	2.019525817	BMS-852927	chembl:CHEMBL3545047	BMS-852927	FALSE	FALSE	FALSE
COMPLEMENT DECAY-ACCELERATING FACTOR	hgnc:2665	CD55	TTD	2020.06.01	NULL	10.50153424713889	Coxsackievirus A21	rxcui:2591813	COXSACKIEVIRUS A21	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Magnesium Sulfate	rxcui:1311625	MAGNESIUM SULFATE ANHYDROUS	TRUE	FALSE	FALSE
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	DNA vaccine, Memorial Sloan-Kettering Cancer Center	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	NULL	Pfizer 4	NULL	NULL	NULL	NULL	NULL
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.089298761	SU-014813	chembl:CHEMBL1721885	SU-014813	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-364735	chembl:CHEMBL1256978	GSK-364735	FALSE	FALSE	FALSE
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	NULL	PMID18163548C4	NULL	NULL	NULL	NULL	NULL
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	NULL	TRIDMAC	NULL	NULL	NULL	NULL	NULL
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	0.6035364509849942	Pyruvic acid	rxcui:35161	PYRUVIC ACID	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.037003292	Methoxyflurane	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE 1	hgnc:44465	RAB4B-EGLN2	TTD	2020.06.01	NULL	2.917092846427472	FG-4592	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinethazone	rxcui:59743	QUINETHAZONE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amdinocillin	rxcui:626	AMDINOCILLIN	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	1.521961485092594	TUROFEXORATE ISOPROPYL	ncit:C81536	TUROFEXORATE ISOPROPYL	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-9219	chembl:CHEMBL1823518	RABACFOSADINE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 22 MEMBER 8	hgnc:10972	SLC22A8	TTD	2020.06.01	NULL	NULL	Buproprion+zonisamide	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Pemirolast	rxcui:19551	PEMIROLAST	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.5016656487486736	Calcipotriol	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phentermine+topiramate	NULL	NULL	NULL	NULL	NULL
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.9907107780319716	AEW-541	chembl:CHEMBL551064	AEW-541	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phentermine+topiramate	NULL	NULL	NULL	NULL	NULL
CANDIDA MANNOSE-6-PHOSPHATE ISOMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfacetamide	rxcui:10169	SULFACETAMIDE	TRUE	FALSE	FALSE
CANDIDA MANNOSE-6-PHOSPHATE ISOMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfoxone	ncit:C72856	SULFOXONE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Salicyclic acid	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	NULL	BVT-A	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	NULL	Salicyclic acid	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	NULL	Salicyclic acid	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Salicyclic acid	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.047432404	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
CARBONIC ANHYDRASE VI	hgnc:1380	CA6	TTD	2020.06.01	NULL	NULL	Salicyclic acid	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE XII	hgnc:1371	CA12	TTD	2020.06.01	NULL	NULL	Salicyclic acid	NULL	NULL	NULL	NULL	NULL
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Trifluridine	rxcui:10803	TRIFLURIDINE	TRUE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.4102161815288632	TG-4010	chembl:CHEMBL4650517	MESMULOGENE ANCOVACIVEC	FALSE	FALSE	FALSE
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Levamlodipine	rxcui:2376944	LEVAMLODIPINE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Salicyclic acid	NULL	NULL	NULL	NULL	NULL
JAK-STAT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	CKD-712	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefoxitin	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	6.848826682916673	Felypressin	rxcui:4319	FELYPRESSIN	FALSE	FALSE	FALSE
PROSTATE SPECIFIC ANTIGEN	hgnc:6364	KLK3	TTD	2020.06.01	NULL	0.8751278539282416	Motexafin lutetium	ncit:C1651	MOTEXAFIN LUTETIUM	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.693795846312725	Mequitazine	rxcui:29528	MEQUITAZINE	TRUE	FALSE	FALSE
LUTEINIZING HORMONE RECEPTOR	hgnc:6585	LHCGR	TTD	2020.06.01	NULL	16.40864726115453	Lutropin alfa	rxcui:388084	LUTROPIN ALFA	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.055563673	CEP-32496	iuphar.ligand:7880	AGERAFENIB	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.1262203635473425	Vinorelbine	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Iron	rxcui:262150	IRON CARBONYL	TRUE	FALSE	FALSE
NF-KAPPA-B-P38 SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	VGX-1027	iuphar.ligand:11682	ZENUZOLAC	FALSE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	IDM-2101	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.2592971419046642	CEP-32496	iuphar.ligand:7880	AGERAFENIB	FALSE	FALSE	FALSE
MELANOMA-ASSOCIATED ANTIGEN 3	hgnc:6801	MAGEA3	TTD	2020.06.01	NULL	NULL	IDM-2101	NULL	NULL	NULL	NULL	NULL
BACTERIAL 16S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetracyclines	ncit:C1595	TETRACYCLINE ANTIBIOTIC	FALSE	FALSE	FALSE
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	AEB07	NULL	NULL	NULL	NULL	NULL
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.6250913242344582	CEP-5214	chembl:CHEMBL150894	CEP-5214	FALSE	FALSE	FALSE
SERINE PROTEASE UNSPECIFIC	hgnc:11756	TFF2	TTD	2020.06.01	NULL	NULL	VT-111	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	NULL	OrM3	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bimatoprost	rxcui:283810	BIMATOPROST	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sertaconazole	rxcui:36435	SERTACONAZOLE	TRUE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Foscavir	wikidata:Q47521633	FOSCAVIR	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.8899605294185507	MK-5108	drugbank:DB12556	MK-5108	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.8140724222588294	Carmoterol	ncit:C171749	CARMOTEROL	FALSE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	1.750255707856483	Atiprimod	ncit:C52184	ATIPRIMOD	FALSE	FALSE	FALSE
STREPTOCOCCUS ELONGATION FACTOR G	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fusidic Acid	rxcui:113608	FUSIDATE	TRUE	FALSE	FALSE
AMINOPEPTIDASE N	hgnc:500	ANPEP	TTD	2020.06.01	NULL	NULL	IP10 C8	NULL	NULL	NULL	NULL	NULL
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.3697723326457359	PALOMID-529	chembl:CHEMBL2141712	PALOMID-529	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	IP10 C8	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	INOC-005	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	INOC-005	NULL	NULL	NULL	NULL	NULL
BACTERIAL DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Proflavine	rxcui:8723	PROFLAVINE	TRUE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	MSH-1001	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	NULL	Alpha 1-PI	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	GCC-1290K	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED CALCIUM CHANNEL	hgnc:1527	CAV1	TTD	2020.06.01	NULL	NULL	GCC-1290K	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxacillin	rxcui:7773	OXACILLIN	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1495945049449985	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
MEASLES VIRUS FUSION GLYCOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	MLN1202	ncit:C88308	PLOZALIZUMAB	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	5.834185692854944	Ibritumomab	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.7119684235348407	Trandolapril	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
VACUOLAR-TYPE PROTON ATPASE CATALYTIC A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cruentaren	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indol-3-carbinol	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Insulin-glulisine	NULL	NULL	NULL	NULL	NULL
CDK3	hgnc:1772	CDK3	ChEMBL	33	inhibitor	0.4167275494896388	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	2.561349816375341	ABT-102	chembl:CHEMBL398338	ABT-102	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acamprosate	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefixime	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
SOMATOSTATIN	hgnc:11329	SST	TTD	2020.06.01	NULL	0.8078103267029924	Cysteamine	rxcui:1426886	CYSTEAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CARNITINE O-PALMITOYLTRANSFERASE I	hgnc:2329	CPT1B	TTD	2020.06.01	NULL	NULL	Levacecarnine hci	NULL	NULL	NULL	NULL	NULL
BACTERIAL PYRUVATE DECARBOXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vitamin B1	rxcui:10454	THIAMINE	TRUE	FALSE	FALSE
CDK15	hgnc:14434	CDK15	ChEMBL	33	inhibitor	0.6250913242344582	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ZK-93423	drugbank:DB17063	ZK-93423	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	exenatide suspension	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.2	hgnc:1389	CACNA1B	TTD	2020.06.01	NULL	NULL	CNSB-004	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	4.565884455277782	MK-0812	drugbank:DB11990	MK-0812	FALSE	FALSE	FALSE
ATM SERINE/THREONINE KINASE	hgnc:795	ATM	TTD	2020.06.01	NULL	0.1798207919030633	KU-60019	iuphar.ligand:8041	KU-60019	FALSE	FALSE	FALSE
TNF-ALPHA SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	ADVAX	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
VEGFR1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	E6201	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	NULL	PHA-568487	NULL	NULL	NULL	NULL	NULL
DYSTROPHIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Drisapersen	ncit:C166984	DRISAPERSEN	FALSE	FALSE	FALSE
G2/MITOTIC-SPECIFIC CYCLIN B1	hgnc:1579	CCNB1	TTD	2020.06.01	NULL	0.364636606	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.079376676	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
EPHRIN TYPE-A RECEPTOR 2	hgnc:3386	EPHA2	TTD	2020.06.01	NULL	NULL	MEDI-543	NULL	NULL	NULL	NULL	NULL
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	1.166837138570988	HBI-3000	chembl:CHEMBL4594410	SULCARDINE SULFATE	FALSE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	0.074797252	NITD609	ncit:C169853	CIPARGAMIN	FALSE	FALSE	FALSE
CDK17	hgnc:8750	CDK17	ChEMBL	33	inhibitor	0.6250913242344582	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	0.5527123287967842	(+)-JQ1	iuphar.ligand:7511	(+)-JQ1	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.6482428547616604	HBI-3000	chembl:CHEMBL4594410	SULCARDINE SULFATE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Carbenicillin	rxcui:2015	CARBENICILLIN	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	ORMD-0901	NULL	NULL	NULL	NULL	NULL
CHLORIDE CHANNEL UNSPECIFIC	hgnc:2014	CLC	TTD	2020.06.01	NULL	NULL	Lancovutide inhaled	NULL	NULL	NULL	NULL	NULL
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	NULL	BI-44370 TA	NULL	NULL	NULL	NULL	NULL
STROMAL CELL-DERIVED FACTOR 1	hgnc:10672	CXCL12	TTD	2020.06.01	NULL	NULL	MyoCell SDF-1	NULL	NULL	NULL	NULL	NULL
PROSTATE SPECIFIC ANTIGEN	hgnc:6364	KLK3	TTD	2020.06.01	NULL	1.750255707856483	PRX-302	chembl:CHEMBL2364656	TOPSALYSIN	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.8078103267029922	CAD-106	chembl:CHEMBL2108328	AMILOMOTIDE	FALSE	FALSE	FALSE
CDK18	hgnc:8751	CDK18	ChEMBL	33	inhibitor	0.5000730593875666	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
HISTAMINE H4 RECEPTOR	hgnc:17383	HRH4	TTD	2020.06.01	NULL	1.591141552596802	PF-3893787	iuphar.ligand:8985	ADRIFORANT	FALSE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-911543	drugbank:DB12591	BMS-911543	FALSE	FALSE	FALSE
MHC CLASS II ANTIGEN DR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IMMU-114	drugbank:DB18458	IMMU-114	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lobeglitazone	ncit:C91021	LOBEGLITAZONE	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 EPSILON	hgnc:1674	CD3E	TTD	2020.06.01	NULL	NULL	MT-110	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	NULL	MT-110	NULL	NULL	NULL	NULL	NULL
CDK12	hgnc:24224	CDK12	ChEMBL	33	inhibitor	0.1666910197958555	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	NULL	MT-110	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY 79-4620	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	ChEMBL	33	agonist	0.029235897	CR 1447	chembl:CHEMBL3545092	CR 1447	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS HELICASE-PRIMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASP-2151	chembl:CHEMBL4297592	AMENAMEVIR	FALSE	FALSE	FALSE
MYCOBACTERIUM MEMBRANE PROTEIN MMPL3	NULL	NULL	TTD	2020.06.01	NULL	NULL	SQ-109	drugbank:DB05186	SQ-109	FALSE	FALSE	FALSE
ENDOTHELIAL PLASMINOGEN ACTIVATOR INHIBITOR	hgnc:8583	SERPINE1	TTD	2020.06.01	NULL	1.544343271638073	THR-18	chembl:CHEMBL4802182	THR-18	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.9376369863516875	PRINABEREL	ncit:C76959	PRINABEREL	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	4.200613699	BSI-201	ncit:C62526	INIPARIB	FALSE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	4-aminosalicylate sodium (oral controlled release, ulcerative colitis), AGI Therapeutics	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP120	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-663068	rxcui:2380373	FOSTEMSAVIR	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	2.763561643983921	MT-3995	chembl:CHEMBL3545392	MT-3995	FALSE	FALSE	FALSE
APOLIPOPROTEIN(A)	hgnc:6667	LPA	TTD	2020.06.01	NULL	NULL	MG-1102	NULL	NULL	NULL	NULL	NULL
ERYTHROPOIETIN	hgnc:3415	EPO	TTD	2020.06.01	NULL	NULL	GC-1113	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	GW-409544	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	GW-409544	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Laquinimod	ncit:C76569	LAQUINIMOD	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.052824619	ANLOTINIB	ncit:C138997	ANLOTINIB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Ibrutinib companion diagnostic	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	E-2007	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	NULL	GS 9667	NULL	NULL	NULL	NULL	NULL
C-X-C MOTIF CHEMOKINE 10	hgnc:10637	CXCL10	TTD	2020.06.01	NULL	NULL	Anti-IP10	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	GW-870086-X	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE UNSPECIFIC	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	0.364636606	BMS-582949	drugbank:DB12696	BMS-582949	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	ChEMBL	33	inhibitor	0.546954909	BENTAMAPIMOD	ncit:C87441	BENTAMAPIMOD	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	NULL	GSK-1360707	NULL	NULL	NULL	NULL	NULL
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	GSK-1360707	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	GSK-1360707	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	J 591 Lu-177	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfamethizole	rxcui:10179	SULFAMETHIZOLE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	90Y-cG250	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	MUC1-Poly-ICLC	NULL	NULL	NULL	NULL	NULL
BACTERIAL PROTEIN SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	BC-3781 intravenous	NULL	NULL	NULL	NULL	NULL
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.1000146118775133	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V3	hgnc:18084	TRPV3	TTD	2020.06.01	NULL	NULL	SAR292833	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.8899605294185507	TRV027	drugbank:DB12199	TRV-120027	FALSE	FALSE	FALSE
MEMBRANE COPPER AMINE OXIDASE	hgnc:550	AOC3	TTD	2020.06.01	NULL	26.25383561784724	BTT-1023	ncit:C131541	TIMOLUMAB	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.108374966	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	ChEMBL	33	inhibitor	0.1250182648468916	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
INTERLEUKIN 4 RECEPTOR ALPHA	hgnc:6015	IL4R	TTD	2020.06.01	NULL	8.751278539282415	Dupilumab	rxcui:1876376	DUPILUMAB	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 3	hgnc:1772	CDK3	TTD	2020.06.01	NULL	0.4605936073306535	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
PLASMODIUM MEROZOITE SURFACE PROTEIN 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	AdCh63-MSP1	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	XP-21279	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	842166X	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR	hgnc:2436	CSF2RB	TTD	2020.06.01	NULL	8.751278539282415	CSL-362	chembl:CHEMBL4297837	TALACOTUZUMAB	FALSE	FALSE	FALSE
SIGNAL TRANSDUCTION UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	OMN-54	NULL	NULL	NULL	NULL	NULL
APOLIPOPROTEIN A-I	hgnc:600	APOA1	TTD	2020.06.01	NULL	NULL	CSL-112	NULL	NULL	NULL	NULL	NULL
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.2083637747448194	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dicycloplatin	ncit:C107676	DICYCLOPLATIN	FALSE	FALSE	FALSE
COMPLEMENT DECAY-ACCELERATING FACTOR	hgnc:2665	CD55	TTD	2020.06.01	NULL	NULL	PAT-SC1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	YSCMA	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.049302978	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	1.372749574789398	Patritumab	ncit:C78853	PATRITUMAB	FALSE	TRUE	TRUE
STERYL-SULFATASE	hgnc:11425	STS	TTD	2020.06.01	NULL	NULL	PGL-2	NULL	NULL	NULL	NULL	NULL
SOMATOSTATIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	177Lu-DOTA-octreotate (neuroendocrine tumors), Advanced Accelerator Applications	NULL	NULL	NULL	NULL	NULL
SOMATOSTATIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	177Lu-DOTATATE	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
B-CELL-SPECIFIC GLYCOPROTEIN B29	hgnc:1699	CD79B	TTD	2020.06.01	NULL	1.381780822	Polatuzumab vedotin	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,2,3-triazole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Amide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Azetidine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazole derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazole derivative 6	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	N-(arylalkyl)-1H-indole-2-sulfonic acid amide derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	PMID26161824-Compound-69	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrano[2,3-b]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrano[2,3-b]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 11	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 16	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 19	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 22	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 30	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 33	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 37	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 59	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazoline derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazoline derivative 10	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 10	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyridotriazolopyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Sulfonylated piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Sulfonylated piperazine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Tetra-hydro-1H-1,2,6-triazaazulene derivative 1	NULL	NULL	NULL	NULL	NULL
MARBURG VIRUS NP MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-7288	drugbank:DB17800	AVI-7288	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	NULL	SRT3025	NULL	NULL	NULL	NULL	NULL
CDK12	hgnc:24224	CDK12	ChEMBL	33	inhibitor	0.1250182648468916	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CALCIUM-DEPENDENT CHLORIDE CHANNEL ANOCTAMIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzbromarone	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 2 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PT2385	iuphar.ligand:12707	PT2385	FALSE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	3.182283105193605	Lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
P2X PURINOCEPTOR 3	hgnc:8534	P2RX3	TTD	2020.06.01	NULL	NULL	BAY-1817080a	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	BIIB095	NULL	NULL	NULL	NULL	NULL
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.1103102336884338	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	JNJ-55308942	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA 4	hgnc:4574	GRIA4	TTD	2020.06.01	NULL	1.790034246671403	E-2007	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2A	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.1017590527823536	MEDETOMIDINE	rxcui:52016	MEDETOMIDINE	FALSE	FALSE	FALSE
THYROID PEROXIDASE	hgnc:12015	TPO	TTD	2020.06.01	NULL	2.500365296937833	Methimazole	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cephapirin	rxcui:2238	CEPHAPIRIN	FALSE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	NULL	SSR-125047	NULL	NULL	NULL	NULL	NULL
CDK18	hgnc:8751	CDK18	ChEMBL	33	inhibitor	0.3750547945406749	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	NULL	Heparin low molecular weight	NULL	NULL	NULL	NULL	NULL
FK506-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ascrolimus	NULL	NULL	NULL	NULL	NULL
FK506-BINDING PROTEIN 1A	hgnc:3711	FKBP1A	TTD	2020.06.01	NULL	NULL	SDZ-281-240	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.1029562181092049	ACECLIDINE	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fialuridine	ncit:C73197	FIALURIDINE	FALSE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	NULL	CONTIGOSIDE B	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulopenem	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	NULL	Intranasal apomorphine	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Intranasal apomorphine	NULL	NULL	NULL	NULL	NULL
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	NULL	FK-070	NULL	NULL	NULL	NULL	NULL
CDK10	hgnc:1770	CDK10	ChEMBL	33	inhibitor	0.3750547945406749	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	NULL	FK-070	NULL	NULL	NULL	NULL	NULL
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heptabarbital	ncit:C76527	HEPTABARBITAL	FALSE	FALSE	FALSE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	0.3977853881492006	Spiroglumide	ncit:C73219	SPIROGLUMIDE	FALSE	FALSE	FALSE
ICAM1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS 1570	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	PT005	NULL	NULL	NULL	NULL	NULL
MART-1 MELANOMA ANTIGEN	hgnc:7124	MLANA	TTD	2020.06.01	NULL	NULL	Polynoma-1	NULL	NULL	NULL	NULL	NULL
MELANOMA-ASSOCIATED ANTIGEN 3	hgnc:6801	MAGEA3	TTD	2020.06.01	NULL	NULL	Polynoma-1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Polynoma-1	NULL	NULL	NULL	NULL	NULL
CDK16	hgnc:8749	CDK16	ChEMBL	33	inhibitor	0.3750547945406749	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	NP-500	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	PRX00933	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	KHK-6188	NULL	NULL	NULL	NULL	NULL
INFLUENZA HEMAGGLUTININ	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7745	chembl:CHEMBL4298040	GEDIVUMAB	FALSE	FALSE	FALSE
AROMATIC-L-AMINO-ACID DECARBOXYLASE	hgnc:2719	DDC	TTD	2020.06.01	NULL	3.500511415712966	ProSavin	wikidata:Q7246687	PROSAVIN	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	Bevacizumab + Erlotinib	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Bevacizumab + Erlotinib	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Bevacizumab + Rituximab	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Bevacizumab + Rituximab	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	EZN-4176	ncit:C96742	ANDROGEN RECEPTOR ANTISENSE OLIGONUCLEOTIDE EZN-4176	FALSE	FALSE	FALSE
APOLIPOPROTEIN B-100	hgnc:603	APOB	TTD	2020.06.01	NULL	NULL	SPC4955	NULL	NULL	NULL	NULL	NULL
PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9	hgnc:20001	PCSK9	TTD	2020.06.01	NULL	NULL	SPC5001	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	NULL	ONO-4053	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	5.834185692854944	RG7342	chembl:CHEMBL3545203	RG7342	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-500	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 2	hgnc:7957	NPY2R	TTD	2020.06.01	NULL	NULL	TM30338	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 4	hgnc:9329	NPY4R	TTD	2020.06.01	NULL	NULL	TM30338	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.1151484018326633	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	WT1-targeted autologous dendritic cell vaccine	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	CART33 cells	NULL	NULL	NULL	NULL	NULL
SYNDECAN-1	hgnc:10658	SDC1	TTD	2020.06.01	NULL	NULL	CART-138 cells	NULL	NULL	NULL	NULL	NULL
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ME1100	rxcui:26397	ARBEKACIN	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE I	hgnc:2528	CTSC	TTD	2020.06.01	NULL	NULL	GSK2793660	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.1842374429322613	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR Gene Transduced T Lymphocytes	NULL	NULL	NULL	NULL	NULL
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	5.250767123569449	Instiladrin	hemonc:111273	NADOFARAGENE FIRADENOVEC	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD20	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD30	NULL	NULL	NULL	NULL	NULL
CARBOHYDRATE ANTIGEN LEWIS-Y	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting Lewis-Y	NULL	NULL	NULL	NULL	NULL
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.4526523382387456	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting Mesothelin	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting MUC1	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19 and Anti-CD20 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Anti-CD19 and Anti-CD20 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD19/CD22 CAR T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19/CD22 CAR T cells	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting GD2	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Anti-CD22-CAR-transduced T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting Mesothelin	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting MUCI	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19 anti-CD20 Bispecific CAR-T	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Anti-CD19 anti-CD20 Bispecific CAR-T	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA CAR T cells	NULL	NULL	NULL	NULL	NULL
SYNDECAN-1	hgnc:10658	SDC1	TTD	2020.06.01	NULL	NULL	CD138 CAR T cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CD20-Specific CAR T Cells	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	EGFRvIII-CARs	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	P-BCMA-101 CAR-T cells	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	CART-123 cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CART-20 cells	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC PROGENITOR CELL ANTIGEN CD34	hgnc:1662	CD34	TTD	2020.06.01	NULL	NULL	CART-34 cells	NULL	NULL	NULL	NULL	NULL
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	NULL	CART-38 cells	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	CAR-BCMA T cell	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CAR-CD19 T cell	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA CAR-T	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	HuCART-meso cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Patient-derived CD19- and CD22 specific CAR	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Patient-derived CD19- and CD22 specific CAR	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD2	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting Muc1	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	MB-CART19.1	ncit:C172103	AUTOLOGOUS CD19 CAR-EXPRESSING CD4+/CD8+ T-CELLS MB-CART19.1	FALSE	FALSE	FALSE
NEUROTROPHIC TYROSINE KINASE ROR2	hgnc:10257	ROR2	TTD	2020.06.01	NULL	NULL	CCT301-59 (targeting ROR2)	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Dual Specificity CD19 and CD22 CAR-T Cell	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-EGFR V III CAR-T cells	NULL	NULL	NULL	NULL	NULL
CANCER/TESTIS ANTIGEN 1	hgnc:2491	CTAG1B	TTD	2020.06.01	NULL	NULL	Anti-NY-ESO-1 CAR-T cells	NULL	NULL	NULL	NULL	NULL
GP100[209-217] PEPTIDE	hgnc:10880	PMEL	TTD	2020.06.01	NULL	NULL	GPA-TriMAR-T cells	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA nanobody CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	SCRI-huCAR19v1	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	Anti-CD19/BCMA CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19/BCMA CAR-T cells	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	IC9.GD2.CAR.IL-15 T-cells	ncit:C158732	AUTOLOGOUS IC9-GD2CAR-CD28-CD3ZETA-IL-15-EXPRESSING T-LYMPHOCYTES	FALSE	FALSE	FALSE
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	NULL	CD38 CAR-T Cell	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	SAR-115740	NULL	NULL	NULL	NULL	NULL
TOXIC REACTIVE METABOLITE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amifostine	rxcui:1545987	AMIFOSTINE ANHYDROUS	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	CLIC-1901	ncit:C158604	AUTOLOGOUS ANTI-CD19 CAR-EXPRESSING T-LYMPHOCYTES CLIC-1901	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fospropofol disodium	rxcui:813021	FOSPROPOFOL DISODIUM	TRUE	FALSE	FALSE
ENDOTHELIUM OF BLOOD VESSELS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Polidocanol	rxcui:968170	POLIDOCANOL	TRUE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	DiabeCell	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.2234368988752957	Fesoterodine fumarate	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 9	NULL	NULL	TTD	2020.06.01	NULL	NULL	BI-409306	chembl:CHEMBL4206492	OSORESNONTRINE	FALSE	FALSE	FALSE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	0.172722603	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	DX-2802	NULL	NULL	NULL	NULL	NULL
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Abciximab	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aciclovir	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amcinonide	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminosalicylic Acid	rxcui:7833	AMINOSALICYLIC ACID	TRUE	FALSE	FALSE
HYALURONIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Asenapine	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	0.8204323630577265	Aminosalicylic Acid	rxcui:7833	AMINOSALICYLIC ACID	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Brinzolamide	rxcui:194881	BRINZOLAMIDE	TRUE	FALSE	FALSE
CANDIDA SQUALENE EPOXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Butenafine	rxcui:47461	BUTENAFINE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.045304289	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
BACTERIAL PENICILLIN BINDING PROTEIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefepime	rxcui:20481	CEFEPIME	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceftriaxone	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cephaloglycin	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cephalothin Sodium	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ciclopirox	rxcui:21090	CICLOPIROX	TRUE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cidofovir	rxcui:1546007	CIDOFOVIR ANHYDROUS	TRUE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	NULL	Clobazam - Lundbeck	NULL	NULL	NULL	NULL	NULL
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	1.944728564284981	Azimilide	ncit:C79923	AZIMILIDE	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.252440727	SR46349B	ncit:C95215	EPLIVANSERIN FUMARATE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.061055432	Clomethiazole	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	PENCLOMEDINE	ncit:C1188	PENCLOMEDINE	FALSE	FALSE	FALSE
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-tenatoprazole	NULL	NULL	NULL	NULL	NULL
FARNESYL PROTEIN TRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS214662	iuphar.ligand:8026	BMS-214662	FALSE	FALSE	FALSE
SOMATOTROPIN	hgnc:4261	GH1	TTD	2020.06.01	NULL	NULL	Somatropin intranasal rhGH	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.760980743	GANDOTINIB	ncit:C116857	GANDOTINIB	FALSE	FALSE	TRUE
VARICELLA-ZOSTER VIRUS DNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aciclovir	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	NULL	Autologous melanoma cell vaccine	NULL	NULL	NULL	NULL	NULL
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	NULL	CDNA vaccine	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.055859225	N-DESMETHYLCLOZAPINE	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	9.546849315580817	CR-3465	chembl:CHEMBL3545273	CR-3465	FALSE	FALSE	FALSE
THYROID HORMONE RECEPTOR ALPHA	hgnc:11796	THRA	TTD	2020.06.01	NULL	NULL	BCT303	NULL	NULL	NULL	NULL	NULL
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.6482428547616604	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	NULL	BCT303	NULL	NULL	NULL	NULL	NULL
SOMATOSTATIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Edotreotide	ncit:C2616	EDOTREOTIDE	FALSE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	Interferon beta 1a inhalation - Synairgen	NULL	NULL	NULL	NULL	NULL
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	NULL	KB002/003	NULL	NULL	NULL	NULL	NULL
SMALL-INDUCIBLE CYTOKINE A11	hgnc:10610	CCL11	TTD	2020.06.01	NULL	17.50255707856483	Bertilimumab	ncit:C166879	BERTILIMUMAB	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	2.100306849	E7016	ncit:C91387	PARP INHIBITOR E7016	FALSE	FALSE	FALSE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	6.563458904461812	LY2940680	ncit:C103826	TALADEGIB	FALSE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.2853677784548614	NEFLAMAPIMOD	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PDX-101	NULL	NULL	NULL	NULL	NULL
HYALURONIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PEGPH20	ncit:C82659	PEGVORHYALURONIDASE ALFA	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceftolozane sulfate	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Netoglitazone	ncit:C72822	NETOGLITAZONE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amdoxovir	ncit:C76927	AMDOXOVIR	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Metocurine Iodide	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	EMIVIRINE	ncit:C73147	EMIVIRINE	FALSE	FALSE	FALSE
FARNESYL PROTEIN TRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zarnestra	hemonc:496	TIPIFARNIB	FALSE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	0.3671865121377238	Donitriptan	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	NULL	CHF 5407	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GLYCOPROTEIN 41	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sifuvirtide	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
NEDD8-ACTIVATING ENZYME	NULL	NULL	TTD	2020.06.01	NULL	NULL	MLN4924	ncit:C77906	PEVONEDISTAT	FALSE	FALSE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	CIGB-128	NULL	NULL	NULL	NULL	NULL
INTERFERON-GAMMA	hgnc:5438	IFNG	TTD	2020.06.01	NULL	NULL	CIGB-128	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	1.750255707856483	SR-147778	ncit:C87598	SURINABANT	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2013059594(III)	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2014110399Splitomycin	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoline derivative 19	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo[4,3-b]pyridazine derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Ethinyl-pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Ethinyl-pyrazole derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	N-substituted pyrazole derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-15	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	1.500219178	CAPMATINIB	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-15	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-26	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 78	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 8	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 9	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Tetra-hydro-imidazo[1,5-d][1,4]oxazepin-3-yl derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Tetra-hydro-imidazo[1,5-d][1,4]oxazepin-3-yl derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	Disulfiram analog 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 6	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Hydroxyqunoline analog 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 7	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-oxalylglycine derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-oxalylglycine derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-oxalylglycine derivative 3	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.050246575	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-49	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-54	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-55	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-56	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridine-2,4-dicarboxylic acid derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Pyrido[1,2-a]indole-1.-carboxylic acid analog 4	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Azole derivative 7	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Lactam derivative 1	NULL	NULL	NULL	NULL	NULL
MANNOSIDE ACETYLGLUCOSAMINYLTRANSFERASE 2	hgnc:7045	MGAT2	TTD	2020.06.01	NULL	NULL	N-containing heterocyclic derivative 1	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-BAY744113	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-Figure4-1A	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL O-ACYLTRANSFERASE 2	hgnc:16940	DGAT2	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-Figure4-1A	NULL	NULL	NULL	NULL	NULL
GHRELIN O ACYLTRANSFERASE	hgnc:32311	MBOAT4	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-GO-CoA-Tat	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Pyridine-amide derivative 1	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Pyridine-carboximide derivative 2	NULL	NULL	NULL	NULL	NULL
MANNOSIDE ACETYLGLUCOSAMINYLTRANSFERASE 2	hgnc:7045	MGAT2	TTD	2020.06.01	NULL	NULL	Pyrimidine-4(3H)-one derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-phe compound 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydropyrrolopyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 44	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 45	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-11	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-16	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-21	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-69	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[1,2-f]triazine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 6	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-12	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-119	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-120	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-121	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-128	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-138	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-144	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-145	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-146	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-149	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-15	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-151	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-17	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-24	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-3	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-30	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-41	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-42	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-44	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-45	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-47	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-48	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-59	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-63	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-65	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-77	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-81	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-82	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-9	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-90	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-96	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-99	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzimidazole and imidazopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzonaphthyridine derivative 2	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-indolylmaleimide derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dibenzo [c,f]-[2,7]naphthyridine derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 6	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 8	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 11	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 14	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 4	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 6	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic-carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Biphenyl carboxamidopropanoic acid derivative 2	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Heterocycle-containing compound 2	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Heterocycle-containing compound 4	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	PMID25828189-Compound-21	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Quinolinyl compound 2	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Spiroimidazolone derivative 4	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-15	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-18	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-19	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-19	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-21	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-21	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-28	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-30	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-42	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-42	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-5	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-5	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A6	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A6	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-B1	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-B2	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-B3	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-C3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-D1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-D1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-Eb	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J5	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L	NULL	NULL	NULL	NULL	NULL
JNK-INTERACTING PROTEIN PEPTIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L2	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Phenylpyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Phenylpyridine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-10	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]-1,3,5-triazine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]-1,3,5-triazine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]-1,3,5-triazine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]-1,3,5-triazine derivative 1	NULL	NULL	NULL	NULL	NULL
MEK KINASE KINASE 2	hgnc:6864	MAP4K2	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 9	NULL	NULL	NULL	NULL	NULL
SPS1/STE20-RELATED PROTEIN KINASE YSK4	hgnc:26249	MAP3K19	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 9	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-12	hgnc:7158	MMP12	TTD	2020.06.01	NULL	NULL	FP-025	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 10	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	PMID26293650-Compound-34	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl compound 1	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl compound 5	NULL	NULL	NULL	NULL	NULL
ERBB4 TYROSINE KINASE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	JI-101	chembl:CHEMBL3545155	JI-101	FALSE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 6	NULL	NULL	NULL	NULL	NULL
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	4.039051633514961	VELUSETRAG	ncit:C84238	VELUSETRAG	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin analog 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Curcumin analog 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 4	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 5	hgnc:11366	STAT5A	TTD	2020.06.01	NULL	NULL	Indirubin derivative 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 2	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 3	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-21	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-42	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-44	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-52	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 5	hgnc:11366	STAT5A	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-56	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 5	hgnc:11366	STAT5A	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-57	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-Figure17	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 62	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Aryl urea derivative 4	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Aryl urea derivative 5	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azole derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azole derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azole derivative 5	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Boronic acid derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-4	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-48	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-6	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 9	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Triazole derivative 1	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 1	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 1	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 13	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 13	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 12	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 17	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 18	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 6	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 9	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 15	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 16	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 17	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 23	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 26	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 28	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 9	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 12	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 14	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 2	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 24	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 26	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 29	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 6	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 7	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	C-linked disaccharide biphenyl mannoside derivative 2	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	C-linked disaccharide biphenyl mannoside derivative 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-126b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-127	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-45	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-46	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5a	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-6d	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-6e	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-8c	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Aromatic hydrazine carboxyimidoamide derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzoic acid linked peptide analog 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 11	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 9	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 8	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Diamine derivative 2	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Benzanilide compound 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Benzanilide compound 2	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Cyclic octapeptide derivative 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-32	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-6	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-7	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1 ALPHA	hgnc:4910	HIF1A	TTD	2020.06.01	NULL	NULL	Pyrrolidine carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
VON HIPPEL-LINDAU DISEASE TUMOR SUPPRESSOR	hgnc:12687	VHL	TTD	2020.06.01	NULL	NULL	Pyrrolidine carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Steroid derivative 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Steroid derivative 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-51	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-55	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Pyrimido-indole derivative 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Pyrimido-indole derivative 3	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Amidine compound 1	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Amidine compound 4	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzothiazine-carboxamide compound 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-13	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-16	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-17	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-17	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-21a	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-28a	NULL	NULL	NULL	NULL	NULL
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.059532507	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-22	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-23	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-23	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-27	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-27	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-29	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-29	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-35	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-36	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-37	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-40	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-42	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-7	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-8	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-9	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 2	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 2	NULL	NULL	NULL	NULL	NULL
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.1356787370431382	BATEFENTEROL	ncit:C166503	BATEFENTEROL	FALSE	FALSE	FALSE
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Isoxazoles and isoxazoline derivative 5	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Pyrimidine benzenesulfonamide derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	1,3,5-triazine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Cyano(dimethyl)methyl isoxazoles and [1,3,4]-thiadiazoles derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Cyano(dimethyl)methyl isoxazoles and [1,3,4]-thiadiazoles derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Isoquinoline derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	N,N-methylenebis-2-phenylacetamide and benzenesulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	N,N-methylenebis-2-phenylacetamide and benzenesulfonamide derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	N,N-methylenebis-2-phenylacetamide and benzenesulfonamide derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-28	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [4,3-a]quinoxaline derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [4,3-a]quinoxaline derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Benzodiazepine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo triazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 7	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 7	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-9	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-asCEBP-1	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-asCEBP-2HPE	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Figure2aExample1	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3-LIKE	hgnc:2980	DNMT3L	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Figure2aExample1	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Figure3CM	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Figure3CN	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Table1Example16	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Table1Example5	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 14	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 3	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 5	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 8	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzoxazepine analog 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Bidentate pyrazolopyrimidine acetamide analog 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine acetamide derivative 6	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 8	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Phenylpyrrolidinone derivative 5	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Tricyclic isoxazoloquinazoline derivative 1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 2	NULL	NULL	NULL	NULL	NULL
RET G691S MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 2	NULL	NULL	NULL	NULL	NULL
RET M918T MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 2	NULL	NULL	NULL	NULL	NULL
RET S891A MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 2	NULL	NULL	NULL	NULL	NULL
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	1.544343271638073	GSK189254	iuphar.ligand:10736	GSK-189254	FALSE	FALSE	FALSE
RET V804L MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 2	NULL	NULL	NULL	NULL	NULL
RET V804M MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 2	NULL	NULL	NULL	NULL	NULL
RET Y791F MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 2	NULL	NULL	NULL	NULL	NULL
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.252440727	SB-773812	drugbank:DB16042	SB-773812	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Isothiazolidine derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Piperidinone derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Thiazole-fused cycloalkyl carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
CRHR1	hgnc:2357	CRHR1	ChEMBL	33	inhibitor	2.917092846427472	ONO-2333MS	iuphar.ligand:10376	ONO-2333MS	FALSE	FALSE	FALSE
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	Biphenyl carboxylic acid derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 4	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridone derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridone derivative 2	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Thiazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure12Example10	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure12Example10	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure6Example12	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure6Example12	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure6Example12	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure6Example12	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 11	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 11	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	Tetra-cyclic compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic compound 1	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-136	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-137	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-143	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Amidine oxime derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Egonol compound 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Egonol compound 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-13	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-14	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-neostenine	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-44	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-46	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-8	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Terpyridineplatinum(II) complexe 5	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Triazole gold complexe 3	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	Oxotetrahydro-2-H-furo[3.2-b]pyrrol-4(5-H)-yl derivative 1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	Oxotetrahydro-2-H-furo[3.2-b]pyrrol-4(5-H)-yl derivative 1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-15	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-15	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-22	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-7	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-7	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoquinoline derivative 5	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-19	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-19	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-21	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-3	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-3	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-5	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-5	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 3	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Bicyclo-heptan-2-amine derivative 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Bicyclo-heptan-2-amine derivative 4	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Phenylpropylamine derivative 1	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Piperazine derivative 7	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazine derivative 7	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	PMID28051882-Compound-XIV	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID28051882-Compound-XIV	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	2-(substituted ethynyl)quinoline derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Bicarboxylic and tricarboxylic ethynyl derivative 2	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33c	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33j	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33j	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-34	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-34a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-34a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-34c	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-34c	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Aminopyridine derivative 2	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Azaindazole derivative 4	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Bidentate ligands of Markush derivative 1	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bidentate ligands of Markush derivative 1	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 13	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-arylmethyl-N-phenyl cyclic urea derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure17-2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure17-3	NULL	NULL	NULL	NULL	NULL
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure21-b	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure21-b	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-1	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 14	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 15	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 17	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 20	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 22	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 24	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 6	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 9	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Ureido-phenyl-substituted triazine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 5	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 9	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Five membered heterocyclic benzamide derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Five membered heterocyclic benzamide derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpiperidine ether derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpyrrolidine ether derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2013161919Example85-117	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2014152663 701	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2015042088Example11	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2015042088Example12	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2016054807Example71	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2016054807Example82	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-d]pyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Six-membered heterocyclic benzamide derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Six-membered heterocyclic benzamide derivative 4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Six-membered heterocyclic benzamide derivative 6	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Tri-substituted urea derivative 2	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-1	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-12	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-15	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-16	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-22	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-23	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-12	NULL	NULL	NULL	NULL	NULL
EZH2 Y641F MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-12	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-14	NULL	NULL	NULL	NULL	NULL
EZH2 Y641F MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-14	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-22	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-24	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	P-toluenesulfonate derivative 1	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	Pyridopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	1,6-naphyridine-4-ketone fused heterocyclic derivative 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Antibodie derivative 10	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 4	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 21	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 15	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 17	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 18	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 20	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	PMID28621580-Compound-WO2013036866C66	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	PMID28621580-Compound-WO2013112959C68	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	PMID28621580-Compound-WO2015089220C70	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 10	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 11	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 13	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 5	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 6	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzamide derivative 15	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzamide derivative 16	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Imidazole benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 6	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Phthalazinone derivative 1	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Cyclohexane carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Cyclohexane carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Imidazole derivative 8	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl pyrazole derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 13	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 19	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 21	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 23	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 24	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 25	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 30	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme13INDY	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme15-1	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme16DMAT	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 2	hgnc:3093	DYRK2	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme16DMAT	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme1WO2011135259	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Left	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Left	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 2	hgnc:3093	DYRK2	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Left	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 3	hgnc:3094	DYRK3	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Left	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure13(4)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure13(4)	NULL	NULL	NULL	NULL	NULL
GELATINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure15(8)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure16(9c)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure16(9c)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-12	hgnc:7158	MMP12	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure17(11)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure17(11)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure18(14a)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure18(14a)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure18(14a)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure18(14a)	NULL	NULL	NULL	NULL	NULL
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzyl amine derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Coumarin/resveratrol hybrid derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lazabemide analog 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID29324067-Compound-25	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Secondary and tertiary (hetero)arylamide derivative 1	NULL	NULL	NULL	NULL	NULL
CASR	hgnc:1514	CASR	ChEMBL	33	positive modulator	6.563458904461812	ASP7991	chembl:CHEMBL3545100	ASP7991	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acrylamide compound 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acrylamide compound 2	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acrylamide compound 4	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl derivative 4	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	Citalopram derivative 1	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	Citalopram derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenoxypiperidine derivative 2	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-55	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-57	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-61	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-61	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-61	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-62	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-66	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-66	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-benzodiazepine derivative 2	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-26	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-29	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-31	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Aryl sulphoxide imine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Cyclohexyl-ethyl-substituted diaza and triaza-tricyclic compound 1	NULL	NULL	NULL	NULL	NULL
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	1.193356164447602	RELUGOLIX	rxcui:2472778	RELUGOLIX	TRUE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Five-membered heteroaromatic compound 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Imidazoleisoindoles derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Monoaryl-1,2-diamine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Monoaryl-1,2-diamine derivative 4	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-17	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-71b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-72a	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Indoline derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Indoline derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8a	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8a	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8c	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8c	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine heterodimer derivative 1	NULL	NULL	NULL	NULL	NULL
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.5585922471882393	AZD1446	chembl:CHEMBL2179529	AZD1446	FALSE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Tacrine heterodimer derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 3	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 3	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dipeptide analog 1	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dipeptide analog 1	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 11	NULL	NULL	NULL	NULL	NULL
GRIK5	hgnc:4583	GRIK5	ChEMBL	33	inhibitor	1.166837138570989	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 11	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 12	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 16	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 20	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 30	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 34	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 34	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-42	NULL	NULL	NULL	NULL	NULL
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	0.4773424657790409	DASOLAMPANEL	ncit:C166510	DASOLAMPANEL	FALSE	FALSE	FALSE
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-49	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-49	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-49	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-49	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-50	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-51	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-51	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-51	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-51	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-57	NULL	NULL	NULL	NULL	NULL
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	blocker	0.2419708351875322	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-60	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	Cyclic compound 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclic peptidomimetic derivative 1	NULL	NULL	NULL	NULL	NULL
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.2500365296937833	DASOLAMPANEL	ncit:C166510	DASOLAMPANEL	FALSE	FALSE	FALSE
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 1	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 2	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 4	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 4	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 5	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 5	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 6	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 6	NULL	NULL	NULL	NULL	NULL
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	blocker	0.577007376	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 7	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 7	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 8	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 8	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 9	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 9	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocyclic peptide analog 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 4	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylate derivative 1	NULL	NULL	NULL	NULL	NULL
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	2.663432598912039	OBETICHOLIC ACID	rxcui:1798288	OBETICHOLIC ACID	TRUE	FALSE	FALSE
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tobramycin	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	5.834185692854944	Pixykine	chembl:CHEMBL2108438	MILODISTIM	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	agonist	0.038159645	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	NULL	LYS-6KAKT1	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	NULL	LYS-6KAKT1	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Adenine	rxcui:290	ADENINE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.3777530304726222	FLUMATINIB	hemonc:38662	FLUMATINIB	FALSE	FALSE	FALSE
INFLUENZA M2 PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amantadine	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	0.31414846	Allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
LYMPHOID CELL ADHESION MOLECULE EXPRESSION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anapsos	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.066213961	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.3697723326457359	Amosulalol	rxcui:2667256	AMOSULALOL	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.4070362111294147	Barbiturate	ncit:C67084	BARBITURATE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.1795134059339983	Armodafinil	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beriplast-P	NULL	NULL	NULL	NULL	NULL
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.3314878234576672	COBIMETINIB	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bifonazole	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
PHOSPHOLIPASE A2 INHIBITORY PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Difluprednate	rxcui:23043	DIFLUPREDNATE	TRUE	FALSE	FALSE
DNA REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Elliptinium acetate	ncit:C1367	ELLIPTINIUM ACETATE	FALSE	FALSE	FALSE
IL1A	hgnc:5991	IL1A	ChEMBL	33	inhibitor	5.250767123569449	BERMEKIMAB	ncit:C95708	BERMEKIMAB	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.1535312024435511	Eszopiclone	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	H1N1 pandemic influenza A vaccine	NULL	NULL	NULL	NULL	NULL
HYALURONIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hyaluronidase (ovine)	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	NULL	Imidapril hci	NULL	NULL	NULL	NULL	NULL
CASP7	hgnc:1508	CASP7	ChEMBL	33	inhibitor	0.2375912725597036	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
ALPHA-GALACTOSIDASE A	hgnc:4296	GLA	TTD	2020.06.01	NULL	4.039051633514961	Migalastat	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
BACTERIAL FUMARATE REDUCTASE FLAVOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Morantel tartrate	rxcui:1368899	MORANTEL TARTRATE	FALSE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	1.750255707856483	Mizoribine	ncit:C66172	MIZORIBINE	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.9546849315580818	APRICOXIB	ncit:C74021	APRICOXIB	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.2917092846427472	Pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Quattvaxem	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION GENE 3 PROTEIN	hgnc:6476	LAG3	TTD	2020.06.01	NULL	NULL	IMP-321	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.2333674277141978	Sodium phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
C-C CHEMOKINE RECEPTOR TYPE 9	hgnc:1610	CCR9	TTD	2020.06.01	NULL	NULL	MLN-3126	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	MLN-576	NULL	NULL	NULL	NULL	NULL
CASP2	hgnc:1503	CASP2	ChEMBL	33	inhibitor	1.009762908	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	MLN-576	NULL	NULL	NULL	NULL	NULL
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NGD 94-1	iuphar.ligand:3297	[3H]NGD941	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	Nibentan	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 7 RECEPTOR ALPHA	hgnc:6024	IL7R	TTD	2020.06.01	NULL	NULL	PF-06342674	NULL	NULL	NULL	NULL	NULL
CASP12	hgnc:19004	CASP12	ChEMBL	33	inhibitor	4.039051633514962	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
SYNUCLEIN ALPHA	hgnc:11138	SNCA	TTD	2020.06.01	NULL	NULL	Posiphen R-phenserine	NULL	NULL	NULL	NULL	NULL
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	NULL	PTI-80	NULL	NULL	NULL	NULL	NULL
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	NULL	RG6100	NULL	NULL	NULL	NULL	NULL
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.3319450480417468	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	NULL	RG-7351	NULL	NULL	NULL	NULL	NULL
DIHYDROTHYMINE DEHYDROGENASE	hgnc:3012	DPYD	TTD	2020.06.01	NULL	NULL	RO-09-4889	NULL	NULL	NULL	NULL	NULL
NKG2-A/B-ACTIVATING NK RECEPTOR	hgnc:6374	KLRC1	TTD	2020.06.01	NULL	105.0153424713889	Monalizumab	ncit:C120208	MONALIZUMAB	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	1.357957014716237	ALDOXORUBICIN	ncit:C68921	ALDOXORUBICIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	SDZ-MKS-492	NULL	NULL	NULL	NULL	NULL
GLYCINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	UK-240455	chembl:CHEMBL539216	UK-240455	FALSE	FALSE	FALSE
TNNC2	hgnc:11944	TNNC2	ChEMBL	33	activator	5.834185692854944	TIRASEMTIV	ncit:C152657	TIRASEMTIV	FALSE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.07463777	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	CGS-15873A	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	CSP-1103	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	EVT302	NULL	NULL	NULL	NULL	NULL
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	K-201	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	Long-acting exenatide	NULL	NULL	NULL	NULL	NULL
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.036925226	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE LYASE 1	hgnc:10817	SGPL1	TTD	2020.06.01	NULL	26.25383561784724	LX2931	iuphar.ligand:9851	LX2931	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	MDL-27192	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PD-332991	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	PD-332991	NULL	NULL	NULL	NULL	NULL
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.067839369	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
RTP801 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-4523655	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	RA101495	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	4.773424657790408	CLEVUDINE	ncit:C95210	CLEVUDINE	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	Salvicine	NULL	NULL	NULL	NULL	NULL
VWF-DEPENDENT PLATELET-COLLAGEN CONVERSION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Saratin	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.07631929	SAGE-217	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	inhibitor	0.8204323630577265	ECOPIPAM	ncit:C74188	ECOPIPAM	FALSE	FALSE	FALSE
LEISHMANIA DNA TOPOISOMERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sodium stibogluconate	rxcui:8010	SODIUM STIBOGLUCONATE	FALSE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	NULL	SR-43845	NULL	NULL	NULL	NULL	NULL
B1 BRADYKININ RECEPTOR	hgnc:1029	BDKRB1	TTD	2020.06.01	NULL	NULL	SSR-240612	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	UNI-rE-4	NULL	NULL	NULL	NULL	NULL
POLA2	hgnc:30073	POLA2	ChEMBL	33	inhibitor	0.6250913242344582	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.2966535098061835	VX-680	ncit:C61319	TOZASERTIB LACTATE	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	3.088686543276147	ABT-761	ncit:C64176	ATRELEUTON	FALSE	FALSE	FALSE
T-CELL-SPECIFIC SURFACE GLYCOPROTEIN CD28	hgnc:1653	CD28	TTD	2020.06.01	NULL	3.500511415712966	AB-103	chembl:CHEMBL504088	BENZODEPA	FALSE	FALSE	FALSE
POLD2	hgnc:9176	POLD2	ChEMBL	33	inhibitor	0.729273212	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	6.058577450272442	Anacetrapib	ncit:C75251	ANACETRAPIB	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR	hgnc:2438	CSF3	TTD	2020.06.01	NULL	NULL	DA-3031	NULL	NULL	NULL	NULL	NULL
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	NULL	GASTRAZOLE	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	4.773424657790408	Candoxatril	ncit:C171870	CANDOXATRIL	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL	hgnc:1527	CAV1	TTD	2020.06.01	NULL	13.12691780892362	Eperisone	ncit:C83692	EPERISONE	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	1.693795846312725	Carisbamate	ncit:C75161	CARISBAMATE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	GSK642444	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	H1N1 influenza vaccine	NULL	NULL	NULL	NULL	NULL
MUC5AC	hgnc:7515	MUC5AC	ChEMBL	33	other/unknown	6.563458904461812	ENSITUXIMAB	ncit:C90532	ENSITUXIMAB	FALSE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Momelotinib	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:61	iuphar.ligand:61	(S)-UH 301	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:82	iuphar.ligand:82	[3H]ROBALZOTAN	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.6326225450083675	IUPHAR.LIGAND:114	iuphar.ligand:114	L-775,606	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.050781113	IUPHAR.LIGAND:85	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	inhibitor	2.019525817	STX-100	drugbank:DB16334	STX-100	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:151	iuphar.ligand:151	[3H]LY334370	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1346350544504987	IUPHAR.LIGAND:121	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:3928	iuphar.ligand:3928	LASMIDITAN	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.064111931	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.042516333	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.012454381	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
IL13RA2	hgnc:5975	IL13RA2	ChEMBL	33	binder	8.751278539282415	CINTREDEKIN BESUDOTOX	ncit:C2599	CINTREDEKIN BESUDOTOX	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.01678634	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.055155117	IUPHAR.LIGAND:192	iuphar.ligand:192	SB 228357	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.068458502	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:3235	iuphar.ligand:3235	SB357134	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:8435	iuphar.ligand:8435	LP-44	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.009496775	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.054187483	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
ENG	hgnc:3349	ENG	ChEMBL	33	inhibitor	26.25383561784724	CAROTUXIMAB	ncit:C74010	CAROTUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	modulator	1.322135606654178	IUPHAR.LIGAND:8962	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.029715717	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:1385	hgnc:2345	CREB1	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:11393	iuphar.ligand:11393	BW B70C	FALSE	FALSE	FALSE
NCBIGENE:779	hgnc:1397	CACNA1S	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:8762	iuphar.ligand:8762	WP814	FALSE	FALSE	FALSE
NCBIGENE:2436	hgnc:3834	FRA10F	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10150	iuphar.ligand:10150	K-604	FALSE	FALSE	FALSE
NCBIGENE:1924	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.056097939	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:10529	iuphar.ligand:10529	TL13-112	FALSE	FALSE	FALSE
NCBIGENE:2768	hgnc:4380	GNA12	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7415	ncit:C97357	SORBINIL	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:9698	iuphar.ligand:9698	CEP-37440	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:497	iuphar.ligand:497	RO-70-0004	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.055681518	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.07458476	IUPHAR.LIGAND:485	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:497	iuphar.ligand:497	RO-70-0004	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.037775303	IUPHAR.LIGAND:517	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.031555091	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:6947	rxcui:23678	DROMOSTANOLONE	TRUE	FALSE	TRUE
NCBIGENE:1560	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:8565	iuphar.ligand:8565	COMPOUND I3 [PMID: 23428964]	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3457	ncit:C166564	METRIBOLONE	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:11153	ncit:C148039	IMARADENANT	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:457	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:420	iuphar.ligand:420	CV-1808	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:3286	iuphar.ligand:3286	PSB1115	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.033832262	IUPHAR.LIGAND:2559	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.020048748	IUPHAR.LIGAND:413	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:471	iuphar.ligand:471	MRS1476	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:5930	iuphar.ligand:5930	AURORA KINASE INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.1539814405738841	IUPHAR.LIGAND:590	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
NCBIGENE:969	hgnc:1694	CD69	GuideToPharmacology	2024.1	inhibitor	0.4861821410712454	IUPHAR.LIGAND:4839	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:629	iuphar.ligand:629	[LEU14, &PSI; 13-14)]BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8503	iuphar.ligand:8503	COMPOUND 8A [PMID: 24900283]	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.1875273972703375	IUPHAR.LIGAND:570	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:537	ncit:C174691	PRENALTEROL	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:550	ncit:C72615	BUPRANOLOL	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:3465	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:550	ncit:C72615	BUPRANOLOL	FALSE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:11193	iuphar.ligand:11193	ZYBT1	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:5666	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:11791	iuphar.ligand:11791	BIIB091	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7525	iuphar.ligand:7525	XD1	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:7033	iuphar.ligand:7033	MOLIBRESIB	FALSE	FALSE	FALSE
NCBIGENE:2729	hgnc:4311	GCLC	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:12143	iuphar.ligand:12143	WNY0824	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:644	iuphar.ligand:644	[DES-ARG10]KALLIDIN	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:664	iuphar.ligand:664	CHROMAN 28	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:658	iuphar.ligand:658	NPC 18565	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:3841	iuphar.ligand:3841	[HYP3,TYR(ME)8]BK	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:3728	iuphar.ligand:3728	RIBOSOMAL PROTEIN S19	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:580	iuphar.ligand:580	RPR121154	FALSE	FALSE	FALSE
NCBIGENE:1597	hgnc:2312	CPN1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8675	iuphar.ligand:8675	COMPOUND 3 [PMID: 14640538]	FALSE	FALSE	FALSE
NCBIGENE:1594	hgnc:2606	CYP27B1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8656	iuphar.ligand:8656	SQ-24,798	FALSE	FALSE	FALSE
NCBIGENE:1617	hgnc:2682	DAZ1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:437	iuphar.ligand:437	AS101	FALSE	FALSE	FALSE
NCBIGENE:533	hgnc:861	ATP6V0B	GuideToPharmacology	2024.1	blocker	8.751278539282415	IUPHAR.LIGAND:2536	rxcui:68503	ZICONOTIDE	TRUE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	activator	0.1356787370431382	IUPHAR.LIGAND:2518	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	modulator	0.172722603	MDX-210	drugbank:DB17250	MDX-210	FALSE	FALSE	FALSE
NCBIGENE:2353	hgnc:3796	FOS	GuideToPharmacology	2024.1	inhibitor	0.42006137	IUPHAR.LIGAND:10746	iuphar.ligand:10746	VBY-825	FALSE	FALSE	FALSE
NCBIGENE:2348	hgnc:3791	FOLR1	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:8626	iuphar.ligand:8626	COMPOUND 4G [PMID: 22595175]	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:12208	iuphar.ligand:12208	COMPOUND 23 [PMID: 35944849]	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:765	iuphar.ligand:765	[125I]CCL7 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	3.580068493342807	IUPHAR.LIGAND:3477	iuphar.ligand:3477	[3H]L365260	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3492	iuphar.ligand:3492	BMS COMPOUND 87B	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:10653	ncit:C175807	LAZUCIRNON	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:775	iuphar.ligand:775	CCL24	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:3653	iuphar.ligand:3653	[125I]CCL27 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10317	ncit:C126641	SIMUROSERTIB	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	4.286340509036285	CLAZAKIZUMAB	ncit:C82359	CLAZAKIZUMAB	FALSE	FALSE	TRUE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	NULL	2.386712328895204	IUPHAR.LIGAND:10553	ncit:C171861	BAMOCAFTOR	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:7252	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.017036882	IUPHAR.LIGAND:2892	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.1187956362798518	IUPHAR.LIGAND:7273	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:7270	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:921	iuphar.ligand:921	UROCORTIN 2	FALSE	FALSE	FALSE
FCER2	hgnc:3612	FCER2	ChEMBL	33	inhibitor	31.50460274141669	LUMILIXIMAB	ncit:C26448	GOMILIXIMAB	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:844	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:5927	iuphar.ligand:5927	AMINOPURVALANOL A	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:7382	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:12076	iuphar.ligand:12076	CROZBACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:5951	iuphar.ligand:5951	CDK4 INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:9375	iuphar.ligand:9375	VTX-11E	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2381300282797936	IUPHAR.LIGAND:5707	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.048708415	IUPHAR.LIGAND:7380	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:11687	ncit:C121456	ATUVECICLIB	FALSE	FALSE	FALSE
NCBIGENE:1361	hgnc:2300	CPB2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:6745	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
NCBIGENE:1323	hgnc:2608	CYP2A13	GuideToPharmacology	2024.1	inhibitor	0.7292732116068681	IUPHAR.LIGAND:11052	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
NCBIGENE:1369	hgnc:2312	CPN1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8852	iuphar.ligand:8852	COMPOUND 4D [PMID: 20655626]	FALSE	FALSE	FALSE
NCBIGENE:1328	hgnc:2621	CYP2C19	GuideToPharmacology	2024.1	inhibitor	0.1084869240406911	IUPHAR.LIGAND:8749	iuphar.ligand:8749	COMPOUND 30 [PMID: 22239545]	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	ChEMBL	33	inhibitor	3.750547945	ORDESEKIMAB	ncit:C126841	ORDESEKIMAB	FALSE	FALSE	FALSE
NCBIGENE:1444	hgnc:2442	CSHL1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8860	iuphar.ligand:8860	AMINOETHOXYVINYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1548898856510162	IUPHAR.LIGAND:1634	iuphar.ligand:1634	BNTX	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.015488989	IUPHAR.LIGAND:1626	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1161674142382621	IUPHAR.LIGAND:9194	ncit:C170144	ATICAPRANT	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1623	iuphar.ligand:1623	ENDOMORPHIN-1	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1161674142382621	IUPHAR.LIGAND:9294	iuphar.ligand:9294	BU08028	FALSE	FALSE	FALSE
NCBIGENE:1396	hgnc:2360	CRIP1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10244	iuphar.ligand:10244	DH376	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11163	iuphar.ligand:11163	S312	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.050007306	IUPHAR.LIGAND:5501	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:955	iuphar.ligand:955	(+)-S-14297	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:937	iuphar.ligand:937	SKF-76783	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.093763699	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:2487	hgnc:3959	FRZB	GuideToPharmacology	2024.1	modulator	13.12691780892362	IUPHAR.LIGAND:11523	iuphar.ligand:11523	POCIREDIR	FALSE	FALSE	FALSE
NCBIGENE:2020	hgnc:3343	EN2	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8129	iuphar.ligand:8129	COMPOUND 34 [PMID: 24749861]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	modulator	0.5000730593875666	IUPHAR.LIGAND:12001	iuphar.ligand:12001	JBJ-09-063	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8240	iuphar.ligand:8240	GSK343	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:6017	iuphar.ligand:6017	PD 174265	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.062509132	IUPHAR.LIGAND:9922	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3165	iuphar.ligand:3165	NE10790	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3152	iuphar.ligand:3152	COMPOUND 31 [PMID: 17963374]	FALSE	FALSE	FALSE
NCBIGENE:1401	hgnc:2367	CRP	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8989	iuphar.ligand:8989	LY2077855	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:6484	ncit:C132780	FASIGLIFAM	FALSE	FALSE	FALSE
NCBIGENE:2985	hgnc:3621	FCGRT	GuideToPharmacology	2024.1	antibody	2.917092846427472	IUPHAR.LIGAND:11552	iuphar.ligand:11552	ZILTIVEKIMAB	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1055	rxcui:1370621	PALMITATE	TRUE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:3952	iuphar.ligand:3952	TUG-424	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1256164383629055	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:11887	iuphar.ligand:11887	TINENGOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:9039	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
NCBIGENE:2609	hgnc:4145	GAPDHP67	GuideToPharmacology	2024.1	inhibitor	0.3750547945406749	IUPHAR.LIGAND:6784	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:11414	iuphar.ligand:11414	TASURGRATINIB	FALSE	FALSE	FALSE
NCBIGENE:3175	hgnc:8138	ONECUT1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11480	iuphar.ligand:11480	SLF	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.015193192	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.045461187	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:1048	iuphar.ligand:1048	WKYMVM	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.027781837	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6246	iuphar.ligand:6246	N36	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1959	iuphar.ligand:1959	BIMATOPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4241	iuphar.ligand:4241	L838417	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:4192	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4347	iuphar.ligand:4347	ZK93426	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	blocker	0.062808219	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:11418	iuphar.ligand:11418	[125I]SPEXIN-1	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6101	iuphar.ligand:6101	M1145	FALSE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:4669	iuphar.ligand:4669	NNC-711	FALSE	FALSE	FALSE
NCBIGENE:2977	hgnc:4684	GUCY1A2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:9735	iuphar.ligand:9735	GROWTH DIFFERENTIATION FACTOR 15	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:4264	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.5250767123569451	IUPHAR.LIGAND:4288	rxcui:8351	PIRACETAM	FALSE	FALSE	FALSE
CLDN18	hgnc:2039	CLDN18	ChEMBL	33	binder	105.0153424713889	ZOLBETUXIMAB	ncit:C85475	ZOLBETUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:453	hgnc:771	ASS1P8	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:4181	drugbank:DB02852	DOMOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.1411496538593938	IUPHAR.LIGAND:4171	rxcui:1742747	SERINE, D-	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4243	iuphar.ligand:4243	LY233053	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.1346350544504987	IUPHAR.LIGAND:4216	iuphar.ligand:4216	HOMOQUINOLINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4088	iuphar.ligand:4088	[3H]MDL105519	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.3387591692625452	IUPHAR.LIGAND:4216	iuphar.ligand:4216	HOMOQUINOLINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:4869	iuphar.ligand:4869	ATRIAL NATRIURETIC PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1719	hgnc:2861	DHFR	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:11761	iuphar.ligand:11761	ANUMIGILIMAB	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:8391	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.074797252	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.112919723	IUPHAR.LIGAND:7495	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.112919723	IUPHAR.LIGAND:7502	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.081030357	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.1988926940746004	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
APP	hgnc:620	APP	ChEMBL	33	inhibitor	0.4039051633514961	LECANEMAB	rxcui:2626143	LECANEMAB	TRUE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:12804	iuphar.ligand:12804	J27644	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.1400204566285186	IUPHAR.LIGAND:7502	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2822	hgnc:4459	GPLD1	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8024	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1203	iuphar.ligand:1203	DIMETHYLHISTAPRODIFEN	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:1209	iuphar.ligand:1207	(&PLUSMN;)-TRANS-H2-PAT	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:8984	iuphar.ligand:8984	JNJ-39758979	FALSE	FALSE	FALSE
NCBIGENE:2763	ncbigene:2763	GMFA	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:10158	iuphar.ligand:10158	BMS-823778	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2987	iuphar.ligand:2987	COMPOUND 1A [PMID: 2153213]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2963	iuphar.ligand:2963	COMPOUND 6A [PATIL ET AL., 1989]	FALSE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	modulator	0.7001022831425933	EDRECOLOMAB	rxcui:80726	EDRECOLOMAB	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.030004384	IUPHAR.LIGAND:2955	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5737	iuphar.ligand:5737	COMPOUND 3A [PMID: 21444206]	FALSE	FALSE	FALSE
NCBIGENE:105	hgnc:227	ADARB2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:7803	iuphar.ligand:7803	COMPOUND 15 [PMID: 25313322]	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:741	iuphar.ligand:741	AM281	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:8224	iuphar.ligand:8224	TRYPTANTHRIN	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	0.8751278539282416	AMG-780	chembl:CHEMBL2109586	AMG-780	FALSE	FALSE	FALSE
NCBIGENE:1459	hgnc:2459	CSNK2A2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8878	iuphar.ligand:8878	AS1949490	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.201952582	ISOXSUPRINE HYDROCHLORIDE	rxcui:82033	ISOXSUPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1247	ncbigene:1247	CMR3A	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8830	iuphar.ligand:8830	COMPOUND 2E [PMID: 19013076]	FALSE	FALSE	FALSE
NCBIGENE:1398	hgnc:2362	CRK	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11055	iuphar.ligand:11055	ARN19874	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	BETAHISTINE	rxcui:1511	BETAHISTINE	TRUE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:5854	iuphar.ligand:5854	FR181157	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.1973972602845657	BEZAFIBRATE	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:2291	iuphar.ligand:2291	PICROTOXININ	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:7913	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:1655	iuphar.ligand:1655	U69593	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	agonist	4.118248724368195	CARBETOCIN	ncit:C96858	CARBETOCIN	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.008647508	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.009433646	IUPHAR.LIGAND:5887	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.001758815	IUPHAR.LIGAND:9927	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.069180068	IUPHAR.LIGAND:8245	iuphar.ligand:8245	ZM-306416	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.090064616	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.5966780822238011	CIPROFIBRATE	rxcui:21149	CIPROFIBRATE	TRUE	FALSE	FALSE
NCBIGENE:521	hgnc:846	ATP5ME	GuideToPharmacology	2024.1	activator	1.875273972703375	IUPHAR.LIGAND:2508	iuphar.ligand:2508	LYSOPHOSPHATIDYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.058277105	IUPHAR.LIGAND:5056	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	activator	1.093909817410302	IUPHAR.LIGAND:2324	iuphar.ligand:2324	DC-EBIO	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2320	iuphar.ligand:2320	UCL1684	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	modulator	0.5834185692854945	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
NCBIGENE:442	hgnc:755	ASNSP2	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:6848	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
CALM1	hgnc:1442	CALM1	ChEMBL	33	inhibitor	2.917092846427472	PRENYLAMINE	rxcui:8674	PRENYLAMINE	TRUE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	blocker	0.364636606	IUPHAR.LIGAND:2337	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2596	iuphar.ligand:2596	XE991	FALSE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6715	iuphar.ligand:6715	COMPOUND 5 [PMID: 22533316]	FALSE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:2596	iuphar.ligand:2596	XE991	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.108711535	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:3082	hgnc:4893	HGF	GuideToPharmacology	2024.1	NULL	0.9723642821424906	IUPHAR.LIGAND:10362	iuphar.ligand:10362	ABSCISIC ACID	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	agonist	0.4234489615781814	BETAHISTINE	rxcui:1511	BETAHISTINE	TRUE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:7910	iuphar.ligand:7910	DEFACTINIB	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.2778183663264259	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.2778183663264259	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
IGHE	hgnc:5522	IGHE	ChEMBL	33	inhibitor	17.50255707856483	MEDI-4212	chembl:CHEMBL2109452	MEDI-4212	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:8146	iuphar.ligand:8146	COMPOUND 23 [PMID: 17600705]	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:5995	iuphar.ligand:5995	JAK3 INHIBITOR VI	FALSE	FALSE	FALSE
NCBIGENE:2665	hgnc:4227	GDI2	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:12938	iuphar.ligand:12938	PF-9363	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11284	iuphar.ligand:11284	CC-90011	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.4773424657790409	TENOFOVIR ALAFENAMIDE	rxcui:1721603	TENOFOVIR ALAFENAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2095	ncbigene:2095	ERVT5	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8177	iuphar.ligand:8177	COMPOUND 16 [PMID: 17480064]	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1320	iuphar.ligand:1320	&ALPHA;-MSH	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	1.981421556063943	BIIB-022	chembl:CHEMBL2109356	BIIB-022	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1316	iuphar.ligand:1316	[125I](3-IODO-TYR13)-MCH	FALSE	FALSE	FALSE
NCBIGENE:283	hgnc:483	ANG	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:912	iuphar.ligand:912	CORTICOTROPHIN-RELEASING HORMONE	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1341	iuphar.ligand:1341	PG-901	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	2.500365296937833	IMC-3C5	chembl:CHEMBL2109602	IMC-3C5	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:11677	ncit:C129717	VEBRELTINIB	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6336	iuphar.ligand:1391	[3H]R214127	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:1399	iuphar.ligand:1399	[3H]LY341495	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:6224	iuphar.ligand:6224	COMPOUND 4 [PMID: 21105727]	FALSE	FALSE	FALSE
PGF	hgnc:8893	PGF	ChEMBL	33	inhibitor	52.50767123569449	TB-403	chembl:CHEMBL2109545	TB-403	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:10563	iuphar.ligand:10563	MS432	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:11679	iuphar.ligand:11679	ZAPNOMETINIB	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:296	drugbank:DB04365	ARECOLINE	FALSE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	F105	chembl:CHEMBL2109443	F105	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:7315	rxcui:10811	TRIHEXYPHENIDYL	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:8593	iuphar.ligand:8593	[3H]ACETYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:311	iuphar.ligand:311	MUSCARINIC TOXIN 1	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:318	iuphar.ligand:318	[3H]QNB	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:331	iuphar.ligand:331	SILAHEXOCYCLIUM	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:321	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:339	iuphar.ligand:339	WIN 51,708	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:306	ncit:C152278	SABCOMELINE	FALSE	FALSE	FALSE
CSF1	hgnc:2432	CSF1	ChEMBL	33	inhibitor	3.750547945	PD-360324	chembl:CHEMBL2109513	PD-360324	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:8593	iuphar.ligand:8593	[3H]ACETYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:309	iuphar.ligand:309	OTENZEPAD	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:9658	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:319	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.054243462	IUPHAR.LIGAND:359	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:11498	iuphar.ligand:11498	PD 102807	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:331	iuphar.ligand:331	SILAHEXOCYCLIUM	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:317	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:368	iuphar.ligand:3264	AFDX384	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:308	iuphar.ligand:308	P-F-HHSID	FALSE	FALSE	FALSE
TNFRSF4	hgnc:11918	TNFRSF4	ChEMBL	33	agonist	3.500511415712966	MEDI-6469	drugbank:DB15306	MEDI-6469	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:10665	iuphar.ligand:10665	UCSF3384	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	1.419126249613364	IUPHAR.LIGAND:7776	iuphar.ligand:7776	DIFLUOROAGOMELATINE	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:1361	iuphar.ligand:1361	S22153	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:9004	iuphar.ligand:9004	ADL5859	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:12730	iuphar.ligand:12730	EWB-3-14	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.016970805	IUPHAR.LIGAND:5458	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:2615	iuphar.ligand:2615	BC-III	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.5770073762164231	IUPHAR.LIGAND:12512	iuphar.ligand:12512	[3H]CTOP	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2615	iuphar.ligand:2615	BC-III	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2613	iuphar.ligand:2613	AFT-II	FALSE	FALSE	FALSE
TFRC	hgnc:11763	TFRC	ChEMBL	33	inhibitor	8.751278539282415	E2.3	chembl:CHEMBL2109495	E2.3	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:2613	iuphar.ligand:2613	AFT-II	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:10119	iuphar.ligand:10119	AM-6120	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:2615	iuphar.ligand:2615	BC-III	FALSE	FALSE	FALSE
NCBIGENE:1749	hgnc:2918	DLX5	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:9067	iuphar.ligand:9067	PL-3994	FALSE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	ChEMBL	33	binder	2.386712328895204	FARALIMOMAB	ncit:C188538	FARALIMOMAB	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.1419126249613365	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	modulator	0.6035364509849942	IUPHAR.LIGAND:3992	iuphar.ligand:3992	LY2087101	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.6886251965336985	AVAPRITINIB	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
NCBIGENE:2121	hgnc:3497	EVC	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8205	iuphar.ligand:8205	COMPOUND 22 [PMID: 20462760]	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2102	iuphar.ligand:2102	CP 99994	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	ChEMBL	33	inhibitor	0.1919140030544389	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:3763	iuphar.ligand:3763	[125I][MEPHE7]NKB	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12173	ncit:C184882	SELNOFLAST	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.128537751	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5772	iuphar.ligand:5772	SB 235375	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1476	iuphar.ligand:1476	[125I]NEUROMEDIN U-8 (PIG)	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1476	iuphar.ligand:1476	[125I]NEUROMEDIN U-8 (PIG)	FALSE	FALSE	FALSE
MTNR1A	hgnc:7463	MTNR1A	ChEMBL	33	agonist	1.034633915974276	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1689	iuphar.ligand:1689	[ARG14LYS15]N/OFQ	FALSE	FALSE	FALSE
NCBIGENE:310	hgnc:545	ANXA7	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1571	iuphar.ligand:1571	JMV457	FALSE	FALSE	FALSE
P2RY1	hgnc:8539	P2RY1	ChEMBL	33	agonist	4.375639269641208	DIQUAFOSOL TETRASODIUM	ncit:C65437	DIQUAFOSOL TETRASODIUM	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4688	rxcui:26143	GLYCYRRHIZIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1219	hgnc:10956	SLCO1A2	GuideToPharmacology	2024.1	NULL	0.8751278539282418	IUPHAR.LIGAND:4505	iuphar.ligand:4505	[3H]BSP	FALSE	FALSE	FALSE
NCBIGENE:1222	hgnc:13819	SLCO1C1	GuideToPharmacology	2024.1	NULL	1.312691780892362	IUPHAR.LIGAND:4505	iuphar.ligand:4505	[3H]BSP	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	inhibitor	0.040021091	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2253	iuphar.ligand:2253	L-372662	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.036718651	IUPHAR.LIGAND:2168	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:2221	iuphar.ligand:2221	D(CH2)5[TYR(ME)2,THR4,TYR-NH29]OVT	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1721	iuphar.ligand:1721	MRS2279	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	0.044573575	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	PHYSOSTIGMINE SALICYLATE	rxcui:33656	PHYSOSTIGMINE SALICYLATE	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	0.5645986154375752	IUPHAR.LIGAND:1714	iuphar.ligand:1714	ATP&GAMMA;S	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	inhibitor	0.03140411	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1858	iuphar.ligand:1839	RP-52770	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.2476776945079929	AMLODIPINE BENZOATE	rxcui:2184116	AMLODIPINE BENZOATE	TRUE	FALSE	FALSE
NCBIGENE:3253	ncbigene:3253	HPRTP1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12995	iuphar.ligand:12995	ATGLISTATIN	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:9486	iuphar.ligand:9486	LYS[Z(NO2)]-VAL	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:11137	ncit:C167015	SELADELPAR	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	ChEMBL	33	inhibitor	1.381780822	ANDEXANET ALFA	rxcui:2045114	ANDEXANET ALFA	TRUE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:2664	ncit:C75192	RAGAGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.089298761	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.028413242	IUPHAR.LIGAND:1056	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.9376369863516875	VONOPRAZAN FUMARATE	rxcui:2604576	VONOPRAZAN FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9379	iuphar.ligand:9379	PIK-III	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:12062	iuphar.ligand:12062	COMPOUND 27 [PMID: 35834807]	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:3443	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.5899738341089269	IUPHAR.LIGAND:11876	iuphar.ligand:11876	GILMELISIB	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:10163	iuphar.ligand:10163	RV6153	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2035181055647073	AZELNIDIPINE	ncit:C73023	AZELNIDIPINE	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.046303061	IUPHAR.LIGAND:6741	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	modulator	0.2083637747448194	IUPHAR.LIGAND:8968	iuphar.ligand:8968	PIK-108	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:10163	iuphar.ligand:10163	RV6153	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:5715	iuphar.ligand:5715	TG-100-115	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:6023	drugbank:DB04769	5-QUINOXALIN-6-YLMETHYLENE-THIAZOLIDINE-2,4-DIONE	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:11699	iuphar.ligand:11699	AMDIZALISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:10233	iuphar.ligand:10233	AZ2	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1651184630053286	AZELNIDIPINE	ncit:C73023	AZELNIDIPINE	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:9728	ncit:C107686	DEZAPELISIB	FALSE	FALSE	FALSE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:2347	iuphar.ligand:2347	CYCLIC GMP	FALSE	FALSE	FALSE
NCBIGENE:1310	hgnc:2196	COL19A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8758	iuphar.ligand:8758	COMPOUND 19 [PMID: 22142545]	FALSE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	ChEMBL	33	inhibitor	0.6731752722524935	ODEVIXIBAT	rxcui:2563966	ODEVIXIBAT	TRUE	FALSE	FALSE
NCBIGENE:1294	hgnc:2214	COL7A1	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:9151	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12725	iuphar.ligand:12725	LEO 239652	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:5258	iuphar.ligand:5258	RO20-1724	FALSE	FALSE	FALSE
GP	hgnc:18280	RNF130	ChEMBL	33	inhibitor	7.501095891	ODESIVIMAB	rxcui:2461340	ODESIVIMAB	TRUE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.078840347	IUPHAR.LIGAND:2330	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:2763	drugbank:DB04466	SR12813	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.052090944	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:2395	hgnc:3951	FXN	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8564	iuphar.ligand:8564	ARI-3531	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:2388	hgnc:3900	FRA4A	GuideToPharmacology	2024.1	antibody	2.500365296937833	IUPHAR.LIGAND:6744	rxcui:1659152	ALIROCUMAB	TRUE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:5576	iuphar.ligand:5576	[ALA1,12,AIB3,GLN10,HARG11,TRP14]PTH-(1-14)-NH2	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1808	iuphar.ligand:1808	[TRP23,TYR36]PTHRP-(1-36)-NH2 (HUMAN)	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:1814	iuphar.ligand:1814	PTHRP-(7-34) (HUMAN, RAT, MOUSE)	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:1814	iuphar.ligand:1814	PTHRP-(7-34) (HUMAN, RAT, MOUSE)	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9925	iuphar.ligand:9925	BALAMAPIMOD	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:5895	iuphar.ligand:5895	QRFP26 (26RFA)	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9129	iuphar.ligand:9129	L779450	FALSE	FALSE	FALSE
NCBIGENE:3006	hgnc:4716	H1-2	GuideToPharmacology	2024.1	modulator	7.501095891	IUPHAR.LIGAND:12399	iuphar.ligand:12399	COMPOUND 24 [PMID: 36723914]	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	ChEMBL	33	activator	1.810609352954982	SRT-2104	drugbank:DB12186	SRT-2104	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:9660	iuphar.ligand:9660	GNE-3500	FALSE	FALSE	FALSE
NCBIGENE:598	hgnc:992	BCL2L1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:8906	iuphar.ligand:8906	CD2314	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	BRANEBRUTINIB	ncit:C167033	BRANEBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12379	iuphar.ligand:12379	FLIZASERTIB	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10145	iuphar.ligand:10145	SR1555	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:2885	iuphar.ligand:2885	25-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:1293	hgnc:2213	COL6A3	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6556	iuphar.ligand:6556	HJC 0350	FALSE	FALSE	FALSE
NCBIGENE:1524	hgnc:2558	CX3CR1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12059	iuphar.ligand:12059	COMPOUND 23 [PMID: 35816678]	FALSE	FALSE	FALSE
NCBIGENE:1527	hgnc:2563	TEX28	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:8038	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
NCBIGENE:1529	ncbigene:1529	CYB5P1	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:8038	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	modulator	0.8078103267029922	IUPHAR.LIGAND:8322	iuphar.ligand:8322	ML290	FALSE	FALSE	FALSE
NCBIGENE:1866	ncbigene:1866	DYT7	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8850	iuphar.ligand:8850	COMPOUND 7B [HAFTCHENARY ET AL., 2013]	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.4039051633514961	IUPHAR.LIGAND:1995	iuphar.ligand:1995	INSL3	FALSE	FALSE	FALSE
NCBIGENE:1525	hgnc:2559	CXADR	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9355	iuphar.ligand:9355	GNE-3511	FALSE	FALSE	FALSE
NCBIGENE:1523	hgnc:2557	CUX1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12059	iuphar.ligand:12059	COMPOUND 23 [PMID: 35816678]	FALSE	FALSE	FALSE
NCBIGENE:1523	hgnc:2557	CUX1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8130	iuphar.ligand:8130	SB-747651A	FALSE	FALSE	FALSE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9223	iuphar.ligand:9223	COMPOUND 16 [PMID: 26794040]	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:2921	iuphar.ligand:2921	DIHYDROSPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:9495	iuphar.ligand:9495	COMPOUND 5C [PMID: 27894870]	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:9493	iuphar.ligand:9493	SPM-354	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:9569	iuphar.ligand:9569	ASP4058	FALSE	FALSE	FALSE
NCBIGENE:2197	hgnc:3597	FAU	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:2632	hgnc:4180	GBE1	GuideToPharmacology	2024.1	activator	5.250767123569449	IUPHAR.LIGAND:6804	rxcui:78484	DANAPAROID	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.043611023	IUPHAR.LIGAND:203	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1221108633388244	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2041	iuphar.ligand:2041	BIM 23197	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5638	iuphar.ligand:5638	EDOTREOTIDE	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.3659071166250487	DOSTARLIMAB	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	1.117184494376478	IUPHAR.LIGAND:2083	iuphar.ligand:2083	BIM 23268	FALSE	FALSE	FALSE
NCBIGENE:1758	hgnc:2932	DMP1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:9270	iuphar.ligand:9270	3M-002	FALSE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:5003	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
PSMB7	hgnc:9544	PSMB7	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:3196	hgnc:5057	TLX2	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:11772	iuphar.ligand:11772	PABINAFUSP ALFA	FALSE	FALSE	FALSE
NCBIGENE:3009	hgnc:4719	H1-5	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:9948	iuphar.ligand:9948	NAPTUMOMAB ESTAFENATOX	FALSE	FALSE	FALSE
PSMD4	hgnc:9561	PSMD4	ChEMBL	33	inhibitor	0.1785975212098452	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:363	hgnc:639	AQP6	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:2143	ncit:C77011	TALTIRELIN	FALSE	FALSE	FALSE
NCBIGENE:2421	hgnc:3931	FRA8C	GuideToPharmacology	2024.1	inhibitor	0.6819178082557728	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
PSMD12	hgnc:9557	PSMD12	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.5147810905460244	IUPHAR.LIGAND:10281	iuphar.ligand:10281	PYRAZOLOPYRIMIDINE 4N	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.3860858179095183	IUPHAR.LIGAND:2508	iuphar.ligand:2508	LYSOPHOSPHATIDYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:4132	iuphar.ligand:4132	AMTB	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.074690855	IUPHAR.LIGAND:2330	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	activator	0.09869863	IUPHAR.LIGAND:6784	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
PSMD1	hgnc:9554	PSMD1	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:498	hgnc:823	ATP5F1A	GuideToPharmacology	2024.1	activator	0.8078103267029924	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:498	hgnc:823	ATP5F1A	GuideToPharmacology	2024.1	blocker	0.8078103267029924	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4120	iuphar.ligand:4120	A778317	FALSE	FALSE	FALSE
PSMB8	hgnc:9545	PSMB8	ChEMBL	33	inhibitor	0.1136529680426287	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:1836	hgnc:10994	SLC26A2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8247	iuphar.ligand:8247	LDC1267	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2273	iuphar.ligand:2273	PHI	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2273	iuphar.ligand:2273	PHI	FALSE	FALSE	FALSE
PSMB1	hgnc:9537	PSMB1	ChEMBL	33	inhibitor	0.1785975212098452	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2778183663264258	IUPHAR.LIGAND:2172	iuphar.ligand:2172	LVP	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	3.889457128569962	TRU-015	drugbank:DB05580	TRU-015	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1561	iuphar.ligand:1561	[PP1-17,ALA31,AIB32]NPY (HUMAN)	FALSE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	ChEMBL	33	inhibitor	3.750547945	ONO-8539	drugbank:DB15325	ONO-8539	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.2944355396394084	LUCITANIB	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	0.1312691780892362	BAFETINIB	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
CCNE1	hgnc:1589	CCNE1	CIViC	10-Apr-24	NULL	0.3281729452230906	AKT INHIBITOR MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
FAAH	hgnc:3553	FAAH	ChEMBL	33	inhibitor	10.50153424713889	PF-04457845	drugbank:DB12012	PF-04457845	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.3453256329104173	INFIGRATINIB	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.013890918	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
MDM2	hgnc:6973	MDM2	CIViC	10-Apr-24	NULL	0.6563458904461812	HDM2 INHIBITOR MK-8242	ncit:C116867	HDM2 INHIBITOR MK-8242	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.3513393859865807	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ACACA	hgnc:84	ACACA	ChEMBL	33	inhibitor	1.141471113819445	PF-05175157	drugbank:DB12096	PF-05175157	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	CIViC	10-Apr-24	NULL	0.065634589	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
NPM1	hgnc:7910	NPM1	CIViC	10-Apr-24	NULL	NULL	NSC348884	NULL	NULL	NULL	NULL	NULL
APH1B	hgnc:24080	APH1B	ChEMBL	33	inhibitor	0.6731752722524935	RG-4733	drugbank:DB11870	RG-4733	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	CIViC	10-Apr-24	NULL	0.6105543166941221	ALK/TRK INHIBITOR TSR-011	ncit:C114287	ALK/TRK INHIBITOR TSR-011	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	4.702860988936115	ALECTINIB	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.010128795	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PSENEN	hgnc:30100	PSENEN	ChEMBL	33	inhibitor	0.729273212	RG-4733	drugbank:DB11870	RG-4733	FALSE	FALSE	FALSE
TSC1	hgnc:12362	TSC1	CIViC	10-Apr-24	NULL	2.625383561784725	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.3454452054979901	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
RPL15	hgnc:10306	RPL15	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	ARS-853	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.2734774543525755	ARS-1620	iuphar.ligand:10383	ARS-1620	FALSE	FALSE	TRUE
RPS20	hgnc:10405	RPS20	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.07330914	OSIMERTINIB	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	CIViC	10-Apr-24	NULL	NULL	FOLFOX REGIMEN	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	HEMATOPOIETIC CELL TRANSPLANTATION	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
RPL5	hgnc:10360	RPL5	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.2520944435184235	PACRITINIB	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.068985304	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
RPL10	hgnc:10298	RPL10	ChEMBL	33	inhibitor	0.108040476	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	CIViC	10-Apr-24	NULL	1.491695205559502	DURVALUMAB	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	NULL	JQ1 COMPOUND	NULL	NULL	NULL	NULL	NULL
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	CIViC	10-Apr-24	NULL	0.1363835616511545	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NF2	hgnc:7773	NF2	CIViC	10-Apr-24	NULL	0.1325951293830669	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
CIC	hgnc:14214	CIC	CIViC	10-Apr-24	NULL	0.3500511415712966	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	0.2075402025126264	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.005064397	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.1154860804304131	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	ChEMBL	33	binder	1.235474617310458	ENVAFOLIMAB	ncit:C129714	ENVAFOLIMAB	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	CIViC	10-Apr-24	NULL	0.020542907	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	CIViC	10-Apr-24	NULL	0.065226921	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.046303061	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	ncit:C69145	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	ZENOCUTUZUMAB	ncit:C152948	ZENOCUTUZUMAB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	NULL	CHMFL-KIT-031	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	NULL	CETUXIMAB/ENCORAFENIB REGIMEN	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	NULL	ADJUVANT CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
POLA1	hgnc:9173	POLA1	ChEMBL	33	inhibitor	0.5966780822238011	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
EZH2	hgnc:3527	EZH2	CIViC	10-Apr-24	NULL	2.917092846427472	JQEZ5	iuphar.ligand:9332	JQEZ5	FALSE	FALSE	TRUE
CD19	hgnc:1633	CD19	CIViC	10-Apr-24	NULL	1.921012362281506	TISAGENLECLEUCEL	rxcui:1986438	TISAGENLECLEUCEL	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	1.250182648468916	MAP855	iuphar.ligand:11940	MAP855	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.003219749	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
CDKN2A	hgnc:1787	CDKN2A	CIViC	10-Apr-24	NULL	0.100976291	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	DoCM	10-Apr-24	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	DoCM	10-Apr-24	NULL	0.1022876712383659	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	DoCM	10-Apr-24	NULL	0.179119736	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DoCM	10-Apr-24	NULL	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	DoCM	10-Apr-24	NULL	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	S63845	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	PKF115-584	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.070690956	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.5498185469706229	DT01	ncit:C99165	DNA-DEPENDENT PROTEIN KINASE-TARGETING SIDNA DT01	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	ASN003	ncit:C134967	BRAFV600/PI3K INHIBITOR ASN003	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.057700738	TENALISIB	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
POLD3	hgnc:20932	POLD3	ChEMBL	33	inhibitor	0.7955707762984016	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
E2F7	hgnc:23820	E2F7	ChEMBL	33	inhibitor	2.187819634820604	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	IHMT-RAF-128	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	SIJ777	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	IMM-6-415	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	S63845	NULL	NULL	NULL	NULL	NULL
AKR1B1	hgnc:381	AKR1B1	ChEMBL	33	inhibitor	4.039051633514961	CAFICRESTAT	ncit:C179076	CAFICRESTAT	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	A66	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2061819551139836	XL888	ncit:C79835	HSP90 INHIBITOR XL888	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	CC-91516	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	WNTinib	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	MAP855	iuphar.ligand:11940	MAP855	FALSE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.1121958787087489	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.2243917574174978	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.2991890098899971	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	GSK-1004723	drugbank:DB12806	GSK-1004723	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	ChEMBL	33	inhibitor	0.5707355569097228	PLB1003	chembl:CHEMBL4650298	PLB1003	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	2.059124362184098	CDX-3379	chembl:CHEMBL4650292	CDX-3379	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	NULL	X-376	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.04206222	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.4565884455277783	AZD3463	iuphar.ligand:7706	AZD3463	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	NULL	CYY292	NULL	NULL	NULL	NULL	NULL
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1635752997996713	HQP1351	ncit:C165549	OLVEREMBATINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.2035181055647073	HQP1351	ncit:C165549	OLVEREMBATINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	FIIN-3	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.034888818	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.07631929	Navitoclax	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	ChEMBL	33	inhibitor	0.060008767	KO-947	iuphar.ligand:9976	KO-947	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.065226921	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.2536602475154323	Pacritinib	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.047734247	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	WNTinib	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.1265245090016735	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.2108741816694558	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	1.518294108020081	Ripretinib	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.045187325	Adavosertib	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	NULL	WNTinib	NULL	NULL	NULL	NULL	NULL
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	NULL	unspecified MDM2 inhibitor	NULL	NULL	NULL	NULL	NULL
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	NULL	MX69	NULL	NULL	NULL	NULL	NULL
CA5A	hgnc:1377	CA5A	ChEMBL	33	inhibitor	2.187819634820604	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	NULL	KU60648	NULL	NULL	NULL	NULL	NULL
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	1.250182648468916	MAP855	iuphar.ligand:11940	MAP855	FALSE	FALSE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.9334697108567911	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.035719504	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.1312691780892362	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
MSH3	hgnc:7326	MSH3	JAX-CKB	10-Apr-24	NULL	NULL	KU60648	NULL	NULL	NULL	NULL	NULL
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	NULL	KU60648	NULL	NULL	NULL	NULL	NULL
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.066297565	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.07458476	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.9845188356692718	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	SBI-0640756	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	S63845	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.084689792	KO-947	iuphar.ligand:9976	KO-947	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.028229931	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.05293112	Navitoclax	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	BI-1347	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	IHMT-RAF-128	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	Sotorasib	rxcui:2550714	SOTORASIB	TRUE	FALSE	TRUE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	0.2187819634820604	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
CA5B	hgnc:1378	CA5B	ChEMBL	33	inhibitor	2.187819634820604	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
TACSTD2	hgnc:11530	TACSTD2	ChEMBL	33	binder	13.12691780892362	DS-1062	chembl:CHEMBL4297939	DS-1062	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	agonist	0.033701971	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.05293112	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
CHRM4	hgnc:1953	CHRM4	ChEMBL	33	agonist	0.1143957978991165	XANOMELINE	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	A66	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.018006746	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1458546423213736	Perifosine	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	AT-7867	NULL	NULL	NULL	NULL	NULL
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	2.187819634820604	EBDAROKIMAB	ncit:C179082	EBDAROKIMAB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	ASN003	ncit:C134967	BRAFV600/PI3K INHIBITOR ASN003	FALSE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	1.500219178	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
FTO	hgnc:24678	FTO	ChEMBL	33	inhibitor	3.281729452230906	BISANTRENE	ncit:C1019	BISANTRENE	FALSE	FALSE	FALSE
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	A66	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.04344264	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	S63845	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.020158043	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2365210416022274	Capmatinib	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1419126249613365	GDC0879	iuphar.ligand:5681	GDC-0879	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1182605208011137	ASN003	ncit:C134967	BRAFV600/PI3K INHIBITOR ASN003	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.044347695	Navitoclax	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.026280116	Infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.6035364509849942	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.1448487482363986	Topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	NULL	PT2399	NULL	NULL	NULL	NULL	NULL
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	NULL	BPTES	NULL	NULL	NULL	NULL	NULL
ITGA2B	hgnc:6138	ITGA2B	ChEMBL	33	inhibitor	2.187819634820604	TIROFIBAN HYDROCHLORIDE	rxcui:253202	TIROFIBAN HYDROCHLORIDE	TRUE	FALSE	FALSE
LAMC2	hgnc:6493	LAMC2	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
TNFRSF4	hgnc:11918	TNFRSF4	ChEMBL	33	agonist	3.500511415712966	GSK-3174998	chembl:CHEMBL4297968	GSK-3174998	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.207267123	AC-480	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	EFAROXAN	ncit:C72923	EFAROXAN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FENAMIDONE	chembl:CHEMBL1232792	FENAMIDONE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.2917092846427472	chlorpheniramine	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	ChEMBL	33	agonist	1.544343271638073	EMD-1201081	chembl:CHEMBL4297993	EMD-1201081	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	PharmGKB	4/5/24	NULL	0.048981037	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.021138354	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	6.563458904461812	LY2523355	ncit:C88328	LITRONESIB	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	ChEMBL	33	inhibitor	2.187819634820604	VORASIDENIB	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.2616661357260523	Lofexidine	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:12459	iuphar.ligand:12459	AMAROGENTIN	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	TEBOTELIMAB	ncit:C143957	TEBOTELIMAB	FALSE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.5357925636295356	MOSAPRIDE	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:562	hgnc:6297	KCNQ3	GuideToPharmacology	2024.1	blocker	0.2083637747448194	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:2615	iuphar.ligand:2615	BC-III	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	CIViC	10-Apr-24	NULL	0.0136917	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.5357925636295356	MOSAPRIDE	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	4.773424657790408	IUPHAR.LIGAND:12548	iuphar.ligand:12548	ISOCHLOROGENIC ACID A	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	CIViC	10-Apr-24	NULL	0.2243917574174978	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.5834185692854944	AZD-7268	iuphar.ligand:7824	AZD7268	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1363835616511545	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	0.2047082699247349	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.4546118721705151	MEDROXYPROGESTERONE	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.064505739	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	VIRULIZIN	ncit:C26677	VIRULIZIN	FALSE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	1.400204566285186	MORAb-022	ncit:C172615	GIMSILUMAB	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.045032308	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2104	hgnc:3474	ESRRG	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:6010	iuphar.ligand:6010	MNK1 INHIBITOR	FALSE	FALSE	FALSE
MMP14	hgnc:7160	MMP14	ChEMBL	33	inhibitor	1.250182648468916	REBIMASTAT	ncit:C1875	REBIMASTAT	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	CancerCommons	25-Jul-13	antibody	0.6471533709721451	RG7446	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	inhibitor	0.029301156	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.5048814541893701	ALLOXAN	rxcui:2466730	ALLOXAN	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.182318303	ACETOPHENAZINE	rxcui:16735	ACETOPHENAZINE	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	ChEMBL	33	inhibitor	0.4375639269641208	REBIMASTAT	ncit:C1875	REBIMASTAT	FALSE	FALSE	FALSE
NCBIGENE:466	hgnc:783	ATF1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:4009	iuphar.ligand:4009	&ALPHA;-CONOTOXIN-GIC	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:10751	iuphar.ligand:10751	(R)-16 [PMID: 32267688]	FALSE	FALSE	FALSE
PDE9A	hgnc:8795	PDE9A	ChEMBL	33	inhibitor	6.563458904461812	OSORESNONTRINE	ncit:C174793	OSORESNONTRINE	FALSE	FALSE	FALSE
NCBIGENE:2993	hgnc:4702	GYPA	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9842	iuphar.ligand:9842	COMPOUND 19A [PMID: 26506089]	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	Tipifarnib	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	GNF-PF-4786	chembl:CHEMBL602363	CHEMBL:CHEMBL602363	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.084553416	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.5000730593875667	REVAMILAST	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
UNIPROT:P17787	hgnc:1962	CHRNB2	TEND	1-Aug-11	NULL	0.3170753093942904	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	PharmGKB	4/5/24	NULL	0.055839424	propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.063858524	Loxapine	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	ChEMBL	33	inhibitor	17.50255707856483	INCOBOTULINUMTOXINA	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	NSC-49789	chembl:CHEMBL469309	CHEMBL:CHEMBL469309	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.2318219480604613	IMIDAZOLE-CALIXARENE	chembl:CHEMBL1801219	CHEMBL:CHEMBL1801219	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	1.166837138570988	2,2',4,4',5,5'-HEXACHLOROBIPHENYL	chembl:CHEMBL14377	2,2',4,4',5,5'-HEXACHLOROBIPHENYL	FALSE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.5834185692854945	SOMATOSTATIN	rxcui:9939	SOMATOSTATIN	FALSE	FALSE	FALSE
MAMMALIAN DISINTEGRIN-METALLOPROTEASE	hgnc:188	ADAM10	TTD	2020.06.01	NULL	1.640864726115453	Aderbasib	ncit:C76115	ADERBASIB	FALSE	FALSE	FALSE
FGB	hgnc:3662	FGB	ChEMBL	33	cleavage	0.8751278539282416	ANCROD	rxcui:772	ANCROD	FALSE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	2.386712328895204	SALACINOL	chembl:CHEMBL1208974	SALACINOL	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.093721859	Infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
GPR84	hgnc:4535	GPR84	ChEMBL	33	inhibitor	13.12691780892362	SETOGEPRAM	drugbank:DB15447	SETOGEPRAM	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1223955040459079	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
SMO	hgnc:11119	SMO	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	6.563458904461812	LY2940680	ncit:C103826	TALADEGIB	FALSE	FALSE	TRUE
UNIPROT:Q9Y243	hgnc:393	AKT3	TdgClinicalTrial	Jan-14	NULL	1.230648544586589	XL418	drugbank:DB05204	XL418	FALSE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	1.458546423213736	Unfractionated heparin	hemonc:521	UNFRACTIONATED HEPARIN	TRUE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:1053	iuphar.ligand:1053	MEDICA 16	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	NSC-371682	chembl:CHEMBL1288106	CHEMBL:CHEMBL1288106	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.041672755	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004176557	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.044878351	zolpidem	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	0.1904575128526865	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	DIHYDROERGOCRISTINE	rxcui:3416	DIHYDROERGOCRISTINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.2169738480813822	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.066297565	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.5125748858722557	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.087512785	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.6863747873946994	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2983390411119005	MEK165	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
UNIPROT:P28702	hgnc:10478	RXRB	TdgClinicalTrial	Jan-14	NULL	0.1282238613814273	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.007699637	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	0.096123883	RXDX 101	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1193356164447602	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:11782	iuphar.ligand:11782	ZEMIRCICLIB	FALSE	FALSE	FALSE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2983390411119005	MEK163	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:2137	hgnc:3518	EXTL3	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1250182648468916	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.025390557	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.025567767	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.062509132	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1041818873724097	PKI-588	ncit:C84837	PI3K/MTOR KINASE INHIBITOR PF-04691502	FALSE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.062065805	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TANNIN PYROGALLOL	chembl:CHEMBL491582	TANNIN PYROGALLOL	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.017114626	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	TRAZODONE HYDROCHLORIDE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	1,2,3,5-TETRACHLOROBENZENE	chembl:CHEMBL44011	CHEMBL:CHEMBL44011	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.012582715	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	TALC	12-May-16	inhibitor	3.281729452230906	PF04449913	rxcui:2105845	GLASDEGIB	TRUE	FALSE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.099446347	NSC-695801	chembl:CHEMBL461193	CHEMBL:CHEMBL461193	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.1508841127462485	Aclarubicin	rxcui:239	ACLARUBICIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003559601	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:6988	iuphar.ligand:6988	AM095	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
NCBIGENE:2106	hgnc:26617	MLKL	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9513	iuphar.ligand:9513	MLKL COMPOUND 1	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2214	iuphar.ligand:2214	D(CH2)5[D-ILE2,ILE4,ALA-NH29]AVP	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.016281448	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.05073205	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.2375912725597036	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.032982206	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	2-ARACHIDONOYLGLYCEROL	iuphar.ligand:729	2-ARACHIDONOYLGLYCEROL	FALSE	FALSE	FALSE
DCK	hgnc:2704	DCK	PharmGKB	4/5/24	NULL	0.095122593	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.072424374	BROXYQUINOLINE	ncit:C73253	BROXYQUINOLINE	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	CGI	2/1/22	NULL	0.1275696580070323	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	modulator	0.1215455352678113	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.5427149481725528	Arformoterol	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9662	iuphar.ligand:9662	PYROTINIB	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GITOXIGENIN	chembl:CHEMBL464658	GITOXIGENIN	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	negative modulator	0.026680727	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	DIPYRONE SODIUM	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	NSC-636948	chembl:CHEMBL1998001	CHEMBL:CHEMBL1998001	FALSE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.060146244	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.042293734	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.008245551	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.02321294	RACEMETIROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.4375639269641208	3-FLUOROEVODIAMINE	chembl:CHEMBL2171781	CHEMBL:CHEMBL2171781	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.42006137	TIOXOLONE	rxcui:2059173	TIOXOLONE	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.046303061	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
F8	hgnc:3546	F8	NCI	14-Sep-17	NULL	0.3860858179095183	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.010148371	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.150021918	IUPHAR.LIGAND:730	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DoCM	10-Apr-24	NULL	0.3513393859865807	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.045579576	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	SJ000202381	chembl:CHEMBL591598	CHEMBL:CHEMBL591598	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002423506	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NCBIGENE:2646	hgnc:4196	GCKR	GuideToPharmacology	2024.1	inhibitor	0.5770073762164232	IUPHAR.LIGAND:6817	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	CCT196969	iuphar.ligand:9815	CCT196969	FALSE	FALSE	FALSE
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	0.6177373086552295	Epoetin zeta	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:7782	iuphar.ligand:7782	2-(INDOLIN-1YL)-MELATONIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	ESCULETIN	iuphar.ligand:5180	ESCULETIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.03070624	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	PERAZINE	rxcui:8042	PERAZINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.069824031	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.012070729	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.026136223	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
NCBIGENE:148	hgnc:277	ADRA1A	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:3699	iuphar.ligand:3699	R-SPONDIN-3	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	GLOFITAMAB	rxcui:2639782	GLOFITAMAB	TRUE	FALSE	FALSE
UNIPROT:P16871	hgnc:6024	IL7R	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	CYT-107	ncit:C77879	GLYCOSYLATED RECOMBINANT HUMAN INTERLEUKIN-7	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.067317527	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:1007	ncit:C74027	SOVATELTIDE	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:11583	iuphar.ligand:11583	RETIFANLIMAB	FALSE	FALSE	FALSE
COL27A1	hgnc:22986	COL27A1	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001012879	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
CCDC148	hgnc:25191	CCDC148	PharmGKB	4/5/24	NULL	3.088686543276147	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.004916449	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
UNIPROT:P62942	hgnc:3711	FKBP1A	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	GPI-1485	drugbank:DB05814	GPI-1485	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	1.211715490054488	Dorzolamide	rxcui:60207	DORZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.07631929	IUPHAR.LIGAND:9916	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.095642388	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	DNDI1383301	chembl:CHEMBL1509103	CHEMBL:CHEMBL1509103	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	OncoKB	23-Jul-20	NULL	0.272767123	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.3697723326457359	CP-547632	ncit:C93263	CP-547632	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:752	iuphar.ligand:752	BP-CCL3	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.2616661357260523	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.1766118064547324	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.138178082	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
NCBIGENE:80	hgnc:153	ACTG1P8	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:2902	iuphar.ligand:2902	TC14012	FALSE	FALSE	FALSE
NCBIGENE:1617	hgnc:2682	DAZ1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:5302	iuphar.ligand:5302	Z-YVAD-FMK	FALSE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:822	iuphar.ligand:822	[125I]CXCL8 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2838	hgnc:4469	GPR15	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:8254	iuphar.ligand:8254	OZANEZUMAB	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.068191781	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:9367	iuphar.ligand:9367	LGB321	FALSE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.036463661	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.4795221117415022	RADICICOL	ncit:C1462	RADICICOL	FALSE	FALSE	FALSE
ANGIOPOIETIN-1	hgnc:484	ANGPT1	TTD	2020.06.01	NULL	1.312691780892362	AMG 386	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1495945049449985	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.015019357	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.1363835616511545	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.020836377	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.6482428547616604	D-ALPHA-TOCOPHEROL ACETATE	ncit:C74962	D-ALPHA-TOCOPHEROL ACETATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003614115	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.2853677784548614	SULINDAC SULFIDE	ncit:C29854	SULINDAC SULFIDE	FALSE	FALSE	FALSE
SRI	hgnc:11292	SRI	NCI	14-Sep-17	NULL	0.2592971419046642	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NCBIGENE:1720	hgnc:52354	DHFRP3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7485	rxcui:278739	PEGVISOMANT	TRUE	FALSE	FALSE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	0.2187819634820604	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.039068208	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	1.009762908	NSC-106547	chembl:CHEMBL223575	CHEMBL:CHEMBL223575	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.05309168	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:5145	ncit:C1529	BATIMASTAT	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.7001022831425934	IUPHAR.LIGAND:1365	iuphar.ligand:1365	(1S,3R)-ACPD	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8209	iuphar.ligand:8209	COMPOUND 35 [PMID: 20684608]	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.1620607136904151	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	modulator	2.763561643983921	IUPHAR.LIGAND:9694	iuphar.ligand:9694	LY2389575	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.078136416	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.9010915075351876	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004191225	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.07631929	PROSTAGLANDIN B1	chembl:CHEMBL1561148	PROSTAGLANDIN B1	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.01036472	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	DEMETHOXYCURCUMIN	chembl:CHEMBL179512	DEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.02832129	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:570	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.3182283105193605	IUPHAR.LIGAND:8529	iuphar.ligand:8529	RO5028442	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.1084869240406911	ANABASINE	chembl:CHEMBL1526229	ANABASINE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013192882	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.039361073	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	NSC-628113	chembl:CHEMBL176599	CHEMBL:CHEMBL176599	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.043756393	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.3365876361262467	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007179391	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NSC-117079	chembl:CHEMBL471225	CHEMBL:CHEMBL471225	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE	iuphar.ligand:4512	NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	DTC	9/2/20	NULL	0.2273059360852575	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
NCBIGENE:630	hgnc:7981	NR4A2	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:9860	iuphar.ligand:9860	VIDOFLUDIMUS	FALSE	FALSE	FALSE
UNIPROT:Q15303	hgnc:3432	ERBB4	TdgClinicalTrial	Jan-14	NULL	0.2263261691193728	AC480	ncit:C48380	PAN-HER KINASE INHIBITOR AC480	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.068985304	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.013964806	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.1605739181519709	SAMIDORPHAN L-MALATE	rxcui:2570387	SAMIDORPHAN L-MALATE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.1054370908347279	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.059667808	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:11215	rxcui:2474340	CLASCOTERONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:5927	iuphar.ligand:5927	AMINOPURVALANOL A	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:2010	hgnc:3331	EMD	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8165	iuphar.ligand:8165	COMPOUND 68 [PMID: 24900699]	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:8211	iuphar.ligand:8211	COMPOUND 4G [PMID: 21316219]	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1291	iuphar.ligand:1291	C3	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3665	iuphar.ligand:3665	QRFP43 (43RFA)	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3846715841442821	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.074690855	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.1094923635591405	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	activator	0.6482428547616605	IUPHAR.LIGAND:2518	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.042073455	REBASTINIB	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.049256727	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP1	hgnc:9593	PTGER1	TTD	2020.06.01	NULL	0.7501095890813501	BUTAPROST	ncit:C74369	BUTAPROST	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00808059	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
CCL22	hgnc:10621	CCL22	NCI	14-Sep-17	NULL	17.50255707856483	FRACTALKINE	ncit:C2257	RECOMBINANT FRACTALKINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
CGA	hgnc:1885	CGA	NCI	14-Sep-17	NULL	4.375639269641208	IL-18	iuphar.ligand:4983	IL-18	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.2536602475154323	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	CILOMILAST	ncit:C95232	CILOMILAST	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	(20S,21S)-FLUOROCAMPTOTHECIN	chembl:CHEMBL2435327	(20S,21S)-FLUOROCAMPTOTHECIN	FALSE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	HISTRELIN	rxcui:1294622	HISTRELIN ACETATE	TRUE	FALSE	FALSE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9527	iuphar.ligand:9527	LLY-283	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1808	iuphar.ligand:1808	[TRP23,TYR36]PTHRP-(1-36)-NH2 (HUMAN)	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	CIViC	10-Apr-24	NULL	0.017835486	PEGINTERFERON ALFA-2B	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IVB	chembl:CHEMBL1094681	AESCULIOSIDE IVB	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.007308974	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	(S)-ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.091583148	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.3271505995993426	Endoxifen	iuphar.ligand:10203	ENDOXIFEN	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	NITROBENZENE	chembl:CHEMBL15750	NITROBENZENE	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR-GAMMA	hgnc:10479	RXRG	TTD	2020.06.01	NULL	0.9092237443410301	Alitretinoin	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.09741683	DIHYDREXIDINE	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	Anti-BCMA CAR-T cells	ncit:C176023	ANTI-BCMA CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.064944553	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MMP9	hgnc:7176	MMP9	DTC	9/2/20	NULL	1.050153425	CURCUMIN PYRAZOLE	chembl:CHEMBL180239	CURCUMIN PYRAZOLE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	PF-05230907	drugbank:DB18417	PF-05230907	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	2,4,6-TRIBROMOPHENOL	drugbank:DB02417	2,4,6-TRIBROMOPHENOL	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.2035181055647073	OXATOMIDE	rxcui:54236	OXATOMIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	SJ000120449	chembl:CHEMBL609027	CHEMBL:CHEMBL609027	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008345148	TICLOPIDINE	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	0.6563458904461813	BUTAPROST	ncit:C74369	BUTAPROST	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	1,3-DIPHENYLTHIOUREA	chembl:CHEMBL275260	CHEMBL:CHEMBL275260	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.1829535583125243	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.007479725	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CYP24A1	hgnc:2602	CYP24A1	PharmGKB	4/5/24	NULL	0.082754407	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	CGP-13501	iuphar.ligand:7848	CGP13501	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.016992774	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.053854022	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.1084869240406911	(R)-ZOLPICLONE	chembl:CHEMBL250053	CHEMBL:CHEMBL250053	FALSE	FALSE	FALSE
ALDH5A1	hgnc:408	ALDH5A1	PharmGKB	4/5/24	NULL	2.500365296937833	sodium oxybate	rxcui:9899	SODIUM OXYBATE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.2408608772279564	METHYLNALTREXONE BROMIDE	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.031555091	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:664	hgnc:1084	BNIP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:10901	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.081030357	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10672	iuphar.ligand:10672	COMPOUND 5 [TOMASSI ET AL., 2020]	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124634	chembl:CHEMBL587923	CHEMBL:CHEMBL587923	FALSE	FALSE	FALSE
NCBIGENE:2526	hgnc:4015	FUT4	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:6649	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:1634	iuphar.ligand:1634	BNTX	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	FLUOROSALAN	ncit:C82318	FLUOROSALAN	FALSE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	ChEMBL	33	inhibitor	2.917092846427472	PEXACERFONT	ncit:C76508	PEXACERFONT	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:143	iuphar.ligand:143	SB 277011-A	FALSE	FALSE	FALSE
MSTN	hgnc:4223	MSTN	ChEMBL	33	inhibitor	2.187819634820604	APITEGROMAB	ncit:C174923	APITEGROMAB	FALSE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.7501095890813501	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	AMORFRUTIN A	chembl:CHEMBL491820	AMORFRUTIN A	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.058931169	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012112496	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.044498026	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.009242681	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	(R)-2,3-BIS(OCTYLOXY)PROPYL DIHYDROGEN PHOSPHATE	chembl:CHEMBL202243	CHEMBL:CHEMBL202243	FALSE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.057796006	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007866318	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
MICB	hgnc:7091	MICB	PharmGKB	4/5/24	NULL	0.921187215	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.02302968	IUPHAR.LIGAND:1626	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.027010119	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.039126432	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	2.917092846427472	AAD-2004	drugbank:DB18405	CRISDESALAZINE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2A	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.2616661357260523	Lofexidine	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006397133	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:7298	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	8-FLUOROTRYPTANTHRIN	chembl:CHEMBL1098875	CHEMBL:CHEMBL1098875	FALSE	FALSE	FALSE
NCBIGENE:247	hgnc:434	ALOX15B	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:9114	iuphar.ligand:9114	JMR-132	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:2220	iuphar.ligand:2220	D(CH2)5[TYR(ME)2,THR4,TYR(3125I)-NH29]OVT	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	DNDI1417195	chembl:CHEMBL1303948	CHEMBL:CHEMBL1303948	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	activator	0.760980743	IUPHAR.LIGAND:10281	iuphar.ligand:10281	PYRAZOLOPYRIMIDINE 4N	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	COSMIC	4-Sep-20	NULL	0.1935766681500258	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	BUTINOLINE	ncit:C78064	BUTINOLINE	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 EPSILON	hgnc:1674	CD3E	TTD	2020.06.01	NULL	1.458546423213736	Resimmune	chembl:CHEMBL4297555	RESIMMUNE	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.060077427	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:4449	iuphar.ligand:4449	PTH-(1-34) (RAT)	FALSE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.4579157375205915	ARQ 087	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.5427149481725528	ARFORMOTEROL	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.023823807	IUPHAR.LIGAND:34	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.019059046	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.6482428547616604	MK-2201	chembl:CHEMBL3545000	MK-2201	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.030176823	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1875273972703375	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007866318	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	MyCancerGenome	20-Jun-17	inhibitor	1.312691780892362	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1875273972703375	ISOORIENTIN	chembl:CHEMBL239559	ISOORIENTIN	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.03043923	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.1795134059339983	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.2734774543525755	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
RAMP1	hgnc:9843	RAMP1	ChEMBL	33	agonist	3.281729452230906	PRAMLINTIDE ACETATE	rxcui:356773	PRAMLINTIDE ACETATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	GNF-PF-3515	iuphar.ligand:4203	GMQ	FALSE	FALSE	FALSE
NCBIGENE:1310	hgnc:2196	COL19A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11625	iuphar.ligand:11625	TC-E 5005	FALSE	FALSE	FALSE
NCBIGENE:1257	ncbigene:1257	CNC2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9243	iuphar.ligand:9243	EPZ020411	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.035418328	ENDO-ATROPINE	chembl:CHEMBL2449003	ENDO-ATROPINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	OXYCARBOXIN	chembl:CHEMBL1712057	OXYCARBOXIN	FALSE	FALSE	FALSE
NCBIGENE:990	hgnc:1744	CDC6	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10605	iuphar.ligand:10605	AZD3965	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:5258	iuphar.ligand:5258	RO20-1724	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.073089743	FLUOXYMESTERONE	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.078136416	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
NCBIGENE:511	hgnc:3145	TRPV5	GuideToPharmacology	2024.1	blocker	0.5770073762164232	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.039531467	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.082950507	GNF-PF-2936	chembl:CHEMBL582503	CHEMBL:CHEMBL582503	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1033615575505797	AVOBENZONE	rxcui:45045	AVOBENZONE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.031301145	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:P00915	hgnc:1368	CA1	TdgClinicalTrial	Jan-14	NULL	0.7501095890813498	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	modulator	0.5000730593875666	IUPHAR.LIGAND:12278	iuphar.ligand:12278	EGFR INHIBITOR 57	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.029698909	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.023440925	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
RAC1	hgnc:9801	RAC1	DTC	9/2/20	NULL	5.834185692854944	ZU-0073945	chembl:CHEMBL563777	CHEMBL:CHEMBL563777	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	TALC	12-May-16	inhibitor	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.091476779	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	ChEMBL	33	binder	0.8751278539282418	LUTETIUM DOTATATE LU-177	chembl:CHEMBL3989924	LUTETIUM DOTATATE LU-177	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	NSC-145669	chembl:CHEMBL191611	CHEMBL:CHEMBL191611	FALSE	FALSE	FALSE
TGFBR1	hgnc:11772	TGFBR1	DTC	9/2/20	inhibitor	3.000438356	HTS-466284	drugbank:DB03921	4-(3-PYRIDIN-2-YL-1H-PYRAZOL-4-YL)QUINOLINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.075010959	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CHRM1	hgnc:1950	CHRM1	DTC	9/2/20	NULL	0.1117184494376478	PIPERTRAMINE AMIDE	chembl:CHEMBL130835	PIPERTRAMINE AMIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	SJ000147784	chembl:CHEMBL590186	CHEMBL:CHEMBL590186	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	OncoKB	23-Jul-20	NULL	1.040600372117402	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.6731752722524935	ALPHA-ADRENERGIC AGONIST	ncit:C29709	ALPHA-ADRENERGIC AGONIST	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	blocker	0.4039051633514962	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007378818	SB-224289	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	0.2651902587661338	IUPHAR.LIGAND:2608	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.6050266644442165	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	TIBOLONE	rxcui:38260	TIBOLONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013299815	WIN-552122	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	NCI	14-Sep-17	NULL	0.1182605208011137	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.1268301237577161	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	1.135300999690692	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
NCBIGENE:2140	hgnc:3521	EYA3	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:7813	iuphar.ligand:7813	OTS964	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:9814	iuphar.ligand:9814	CCT241161	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.3302369260106572	OPHIOBOLIN O	chembl:CHEMBL1934283	OPHIOBOLIN O	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.077217164	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
PROC	hgnc:9451	PROC	FDA	10-Apr-24	NULL	1.500219178162699	Avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:374	iuphar.ligand:374	CCPA	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:7953	iuphar.ligand:7953	BMS-777607	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000541406	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
COL1A2	hgnc:2198	COL1A2	ChEMBL	33	cleavage	0.1535312024435511	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	ZUCAPSAICIN	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
KCND2	hgnc:6238	KCND2	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.070860555	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1615620653405984	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:2094	ncbigene:2094	ERVT4	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8177	iuphar.ligand:8177	COMPOUND 16 [PMID: 17480064]	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.1000146118775133	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.07458476	IUPHAR.LIGAND:6287	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:2454	iuphar.ligand:2454	NN-DIMETHYL-D-ERYTHROSPHINGOSINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	ECADOTRIL	ncit:C75238	ECADOTRIL	FALSE	FALSE	FALSE
ATXN1L	hgnc:33279	ATXN1L	CIViC	10-Apr-24	NULL	0.4861821410712454	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1141471113819445	ENDOSULFAN	chembl:CHEMBL194399	ENDOSULFAN	FALSE	FALSE	FALSE
PROTEIN KINASE C ALPHA	hgnc:9393	PRKCA	TTD	2020.06.01	NULL	0.1093909817410302	Sodium phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.050222545	ANTIBIOTICS	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	TALC	12-May-16	inhibitor	15.31473744374422	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DIPHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER	iuphar.ligand:4093	&ALPHA;&BETA;-MEATP	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	S-NITROSOGLUTATHIONE	drugbank:DB17877	S-NITROSOGLUTATHIONE	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.4526523382387456	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.019346968	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:12575	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:827	iuphar.ligand:827	CXCL2	FALSE	FALSE	FALSE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:3542	iuphar.ligand:3542	GASTRIC INHIBITORY POLYPEPTIDE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.021240967	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TEND	1-Aug-11	NULL	0.5016656487486736	CALCIPOTRIOL	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
GATA2	hgnc:4171	GATA2	NCI	14-Sep-17	NULL	0.5791287268642776	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.026830696	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	NCI	14-Sep-17	NULL	0.055711057	CISPLATINUM	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.057700738	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	CIViC	10-Apr-24	NULL	0.010388507	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
NTNG1	hgnc:23319	NTNG1	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:5830	iuphar.ligand:5830	DIAMIDE 7	FALSE	FALSE	FALSE
NCBIGENE:596	hgnc:990	BCL2	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:4349	iuphar.ligand:4349	HEME	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.031707531	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	PAXILLINE	iuphar.ligand:2309	PAXILLINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GABACULINE HYDROCHLORIDE	chembl:CHEMBL1256019	GABACULINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 1	hgnc:11330	SSTR1	TTD	2020.06.01	NULL	1.750255707856483	Lutetium Lu 177 dotatate	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:11438	iuphar.ligand:11438	DS37001789	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.2014360789093139	SUMATRIPTAN SUCCINATE	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	blocker	0.1553481397505754	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:8434	iuphar.ligand:8434	LP-12	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1889	iuphar.ligand:1889	ZK110841	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.1505380482674727	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011746683	flutamide	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	TOREMIFENE CITRATE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.3254607721220733	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1790034246671403	Vilazodone	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009170044	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
CA9	hgnc:1383	CA9	CGI	2/1/22	NULL	0.076541795	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:3469	ncit:C75036	DABUZALGRON	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.2365210416022274	IUPHAR.LIGAND:1347	iuphar.ligand:1347	6-HYDROXYMELATONIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	TCMDC-124506	chembl:CHEMBL579640	CHEMBL:CHEMBL579640	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.2408608772279564	METHYLNALTREXONE BROMIDE	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.1234748294784115	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-3125	chembl:CHEMBL534288	CHEMBL:CHEMBL534288	FALSE	FALSE	FALSE
FZD7	hgnc:4045	FZD7	ChEMBL	33	inhibitor	3.000438356325399	VANTICTUMAB	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	ChEMBL	33	agonist	2.187819634820604	LARAZOTIDE ACETATE	ncit:C81670	LARAZOTIDE ACETATE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.020164236	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.02804897	IUPHAR.LIGAND:548	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	1.944728564284981	Macimorelin	rxcui:1999420	MACIMORELIN	TRUE	FALSE	FALSE
ARAF	hgnc:646	ARAF	MyCancerGenome	20-Jun-17	inhibitor	0.028929846	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
SULT1A3	hgnc:11455	SULT1A3	PharmGKB	4/5/24	NULL	1.093909817410302	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2083637747448194	CEP-7055	chembl:CHEMBL346631	CEP-7055	FALSE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.2206204673768676	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:10351	iuphar.ligand:10351	LUF7602	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	PharmGKB	4/5/24	NULL	0.027855529	dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TEND	1-Aug-11	NULL	1.750255707856483	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.142490288	BI-847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
ASPARAGINASE	hgnc:16448	ASRGL1	TTD	2020.06.01	NULL	26.25383561784724	GRASPA	ncit:C99767	ERYASPASE	FALSE	FALSE	FALSE
ANGIOPOIETIN 1 RECEPTOR	hgnc:11724	TEK	TTD	2020.06.01	NULL	0.546954909	DCC-2036	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	PIMETHIXENE	rxcui:33712	PIMETHIXENE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.04321619	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.009972967	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.1209854175937661	MECLIZINE	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.051731696	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
UNIPROT:P23921	hgnc:10451	RRM1	TdgClinicalTrial	Jan-14	NULL	0.2324817828272369	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.596678082	BEVANTOLOL	ncit:C79556	BEVANTOLOL	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:547	iuphar.ligand:547	SR59230A	FALSE	FALSE	FALSE
CCL7	hgnc:10634	CCL7	NCI	14-Sep-17	NULL	1.250182648468916	RU 486	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.026680727	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.038187397	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.2447910080918158	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1178056726441863	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.596678082	KC706	drugbank:DB05157	KC706	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.3977853881492007	12-HYDROXY-OCTADECANOIC ACID	chembl:CHEMBL292352	CHEMBL:CHEMBL292352	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.1881995384791917	HALOFUGINONE	ncit:C1120	HALOFUGINONE	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.038159645	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.2169738480813822	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.046221542	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
LTC4S	hgnc:6719	LTC4S	PharmGKB	4/5/24	NULL	0.2482632209725508	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
THY1	hgnc:11801	THY1	NCI	14-Sep-17	NULL	17.50255707856483	THYMOSIN FRACTION 5	ncit:C2700	HUMAN THYMOSIN-FRACTION 5	FALSE	FALSE	FALSE
GSTA1	hgnc:4626	GSTA1	DTC	9/2/20	NULL	2.100306849	BROMOSULFOPHTHALEIN	iuphar.ligand:4505	[3H]BSP	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	HEXADECYLTRIMETHYLAMMONIUM CHLORIDE	chembl:CHEMBL1895807	HEXADECYLTRIMETHYLAMMONIUM CHLORIDE	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	0.6471533709721451	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1280674908187671	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	DINALINE	ncit:C79870	DINALINE	FALSE	FALSE	FALSE
CAST	hgnc:1515	CAST	NCI	14-Sep-17	NULL	0.5357925636295356	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.1244257612220248	4-BENZAMIDOPHENYLSTIBONIC ACID	chembl:CHEMBL1726814	CHEMBL:CHEMBL1726814	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	CORONOPILIN	chembl:CHEMBL248564	CORONOPILIN	FALSE	FALSE	FALSE
NFIB	hgnc:7785	NFIB	PharmGKB	4/5/24	NULL	0.5707355569097228	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	(-)-ESEROLINE	chembl:CHEMBL310934	CHEMBL:CHEMBL310934	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005412046	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-4102	chembl:CHEMBL596836	CHEMBL:CHEMBL596836	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.1101559536413171	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.029301156	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:1108	hgnc:1919	CHD4	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8801	iuphar.ligand:8801	COMPOUND 5K [PMID: 23528296]	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.006222025	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	inhibitor	0.035598421	IUPHAR.LIGAND:4920	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1017590527823536	Methylphenobarbital	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2651902587661338	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	ELINAFIDE	ncit:C1615	ELINAFIDE	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	CGI	2/1/22	NULL	0.087512785	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002450766	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
NCBIGENE:1816	hgnc:3026	DRD5	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	0.078252863	IUPHAR.LIGAND:7946	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	GNF-PF-4012	chembl:CHEMBL584269	CHEMBL:CHEMBL584269	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	DTC	9/2/20	NULL	1.842374429322613	NAPHMETHONIUM	chembl:CHEMBL274413	NAPHMETHONIUM	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.034318739	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.014206621	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.032016873	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
PSMC4	hgnc:9551	PSMC4	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.431569901	E7449	ncit:C102746	PARP/TANKYRASE INHIBITOR 2X-121	FALSE	FALSE	TRUE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.2734774543525755	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1346350544504987	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:1593	iuphar.ligand:1593	&BETA;-D-HYDROXYBUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:7428	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:297	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	PRASTERONE	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2044691247495891	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:2613	iuphar.ligand:2613	AFT-II	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11184	ncit:C175871	VENADAPARIB	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	CIViC	10-Apr-24	NULL	0.007268504	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	MANUMYCIN A	chembl:CHEMBL285848	MANUMYCIN A	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.1296485709523321	SELINEXOR	rxcui:2178390	SELINEXOR	TRUE	FALSE	TRUE
PTGDR2	hgnc:4502	PTGDR2	DTC	9/2/20	NULL	2.072671233	VIDUPIPRANT	ncit:C152874	VIDUPIPRANT	FALSE	FALSE	FALSE
PARP3	hgnc:273	PARP3	ChEMBL	33	inhibitor	0.1988926940746004	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.046303061	FEDRATINIB	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1657439117288336	BCP9000383	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.159436249	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11855	iuphar.ligand:11855	SG-005	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.4234489615781814	5-FLUOROINDOLE-2-CARBOXYLIC ACID	chembl:CHEMBL23507	5-FLUOROINDOLE-2-CARBOXYLIC ACID	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	ESFLURBIPROFEN	ncit:C80544	ESFLURBIPROFEN	FALSE	FALSE	FALSE
SSTR3	hgnc:11332	SSTR3	ChEMBL	33	binder	1.166837138570989	LUTETIUM DOTATATE LU-177	chembl:CHEMBL3989924	LUTETIUM DOTATATE LU-177	TRUE	FALSE	FALSE
TNFSF12	hgnc:11927	TNFSF12	ChEMBL	33	inhibitor	26.25383561784724	BIIB-023	chembl:CHEMBL2109598	BIIB-023	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1621	iuphar.ligand:1621	DYNORPHIN A-(1-8)	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.006623484	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.2333674277141977	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.006948216	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
UNIPROT:O15379	hgnc:4854	HDAC3	TEND	1-Aug-11	NULL	0.1829535583125243	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.053854022	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.046840028	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	OncoKB	23-Jul-20	NULL	0.1166837138570988	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	NCI-13239	chembl:CHEMBL187216	CHEMBL:CHEMBL187216	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.8975670296699914	IBANDRONATE	rxcui:115264	IBANDRONATE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.084146909	NEFAZODONE HYDROCHLORIDE	rxcui:236082	NEFAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	0.7001022831425934	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1166837138570988	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	ARQ-197	ncit:C62437	TIVANTINIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004216468	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.1725334213659184	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
NCBIGENE:1466	hgnc:2470	CSRP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8143	iuphar.ligand:8143	COMPOUND 1O [PMID: 24210504]	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	5.834185692854944	ADX10059	drugbank:DB05070	ADX10059	FALSE	FALSE	FALSE
ACYL-COA DESATURASE	hgnc:10571	SCD	TTD	2020.06.01	NULL	7.501095891	Aramchol	drugbank:DB11860	ARAMCHOL	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.2397610558707511	PYRIDOXINE	rxcui:42954	VITAMIN B6	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001218162	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	NSC-292213	chembl:CHEMBL222808	CHEMBL:CHEMBL222808	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.005310242	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.210030685	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	0.3394892536790592	INTERFERON ALFA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
POLD4	hgnc:14106	POLD4	ChEMBL	33	inhibitor	0.2573905452730122	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	LEVOMILNACIPRAN HYDROCHLORIDE	rxcui:1433211	LEVOMILNACIPRAN HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
RAF-1	hgnc:9829	RAF1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.159436249	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.042344896	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	1.184383561707394	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.2187819634820604	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.1535312024435511	trastuzumab emtansine	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.039479452	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
UNIPROT:P28908	hgnc:11923	TNFRSF8	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	AFM13	iuphar.ligand:10067	AFM13	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:9294	iuphar.ligand:9294	BU08028	FALSE	FALSE	FALSE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	modulator	6.563458904461812	IUPHAR.LIGAND:12539	iuphar.ligand:12539	APV207010A	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.094608417	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.088248187	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	modulator	0.1944728564284981	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	NSC-747270	chembl:CHEMBL594772	CHEMBL:CHEMBL594772	FALSE	FALSE	FALSE
NCBIGENE:1360	hgnc:2299	CPB1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:8311	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:12439	iuphar.ligand:12439	RTOXA-43	FALSE	FALSE	FALSE
CASP2	hgnc:1503	CASP2	DTC	9/2/20	NULL	26.25383561784724	N-DECYLBUTYRAMIDE	chembl:CHEMBL265439	CHEMBL:CHEMBL265439	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:9486	iuphar.ligand:9486	LYS[Z(NO2)]-VAL	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.036062961	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.1875273972703375	ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
MMP9	hgnc:7176	MMP9	TALC	12-May-16	vaccine	0.3000438356325399	PRINOMASTAT	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	1.944728564284981	4SCAR-PSMA	ncit:C150699	AUTOLOGOUS PSMA-4SCAR-EXPRESSING T-CELLS 4SCAR-PSMA	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	BOSENTAN	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:5598	iuphar.ligand:5598	CP608,039	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	AMINOPTERIN	rxcui:1440264	AMINOPTERIN	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	1.591141552596802	NSC-87877	chembl:CHEMBL472004	CHEMBL:CHEMBL472004	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	0.5834185692854944	AMG 386	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.072927321	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.055563673	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
NCBIGENE:1282	hgnc:2202	COL4A1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:5233	iuphar.ligand:5233	NKY80	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
NCBIGENE:939	hgnc:11922	CD27	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:7601	rxcui:1424	BENZTROPINE	TRUE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:10566	iuphar.ligand:10566	AMCENESTRANT	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.064111931	IUPHAR.LIGAND:7591	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
NCBIGENE:2150	hgnc:3538	F2RL1	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:8839	iuphar.ligand:8839	TORIN 2	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1325951293830669	TEGASEROD MALEATE	rxcui:339270	TEGASEROD MALEATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	PHENINDIONE	rxcui:8130	PHENINDIONE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.032899543	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.5048814541893701	Begacestat	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.1481697953740938	OSIMERTINIB	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1495945049449985	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.9814517987980279	GUANETHIDINE	rxcui:5036	GUANETHIDINE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.013990853	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:3280	iuphar.ligand:3280	VUF5574	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.018488617	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011762471	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.017561094	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
IL23R	hgnc:19100	IL23R	PharmGKB	4/5/24	NULL	1.129197231	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.064624826	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR BETA-2	hgnc:1962	CHRNB2	TTD	2020.06.01	NULL	2.917092846427472	TC-5214	chembl:CHEMBL2103881	DEXMECAMYLAMINE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2580229544751573	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.006199253	Citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.044878351	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
NOTCH1	hgnc:7881	NOTCH1	CGI	2/1/22	NULL	1.312691780892362	Mk-0752	drugbank:DB12852	MK-0752	FALSE	FALSE	TRUE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	ChEMBL	33	inhibitor	7.778914257139925	RILOTUMUMAB	ncit:C67079	RILOTUMUMAB	FALSE	TRUE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1296485709523321	ENDOSULFAN	chembl:CHEMBL194399	ENDOSULFAN	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1259176768242074	OLVEREMBATINIB	ncit:C165549	OLVEREMBATINIB	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:6500	iuphar.ligand:6500	1-METHYLCYCLOPROPANECARBOXYLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	activator	0.8334550989792776	IUPHAR.LIGAND:2324	iuphar.ligand:2324	DC-EBIO	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	2.423430980108977	Tramiprosate	rxcui:1374845	TRAMIPROSATE	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.030142176	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	CYCLOPHOSPHAMIDE HYDRATE	chembl:CHEMBL1200796	CYCLOPHOSPHAMIDE	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	DTC	9/2/20	NULL	0.1017590527823536	ISONIPECOTIC ACID	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.055271233	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.2047082699247349	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
NCBIGENE:2213	hgnc:3618	FCGR2B	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:11895	iuphar.ligand:11895	COMPOUND 13 [PMID: 34333981]	FALSE	FALSE	FALSE
DDC	hgnc:2719	DDC	NCI	14-Sep-17	NULL	0.3684748858645227	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
CHST1	hgnc:1969	CHST1	PharmGKB	4/5/24	NULL	1.400204566285186	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.150021918	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.022730594	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CANNABINOL	rxcui:1976	CANNABINOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	TEBUFENOZIDE	chembl:CHEMBL226968	TEBUFENOZIDE	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.1323722804261206	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.09969811	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:871	hgnc:1546	SERPINH1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:4631	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:9559	iuphar.ligand:9559	RITLECITINIB	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1262203635473425	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
NCBIGENE:1488	hgnc:2495	CTBP2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	PharmGKB	4/5/24	NULL	1.262203635473425	ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BENODANIL	chembl:CHEMBL1357627	BENODANIL	FALSE	FALSE	FALSE
PSMB3P	hgnc:20633	PSMB3P1	PharmGKB	4/5/24	NULL	0.8824818695074705	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P14618	hgnc:9021	PKM	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	TLN-232	chembl:CHEMBL539934	TT-232	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:5527	iuphar.ligand:5527	LL-37	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FUDOSTEINE	ncit:C65777	FUDOSTEINE	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	blocker	0.070860555	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:9461	iuphar.ligand:9461	L-732,138	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.013890918	ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
ERBB3	hgnc:3431	ERBB3	TALC	12-May-16	inhibitor	1.372749574789398	U3-1287	ncit:C78853	PATRITUMAB	FALSE	TRUE	TRUE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.064268875	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.024141458	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
RARB	hgnc:9865	RARB	ChEMBL	33	inhibitor	1.029562181092048	IRX4310	chembl:CHEMBL3545173	IRX4310	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	2.019525817	FERRUGINENE C	chembl:CHEMBL1775033	FERRUGINENE C	FALSE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TEND	1-Aug-11	NULL	6.848826682916673	FELYPRESSIN	rxcui:4319	FELYPRESSIN	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	AMILORIDE HYDROCHLORIDE	rxcui:142424	AMILORIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TEND	1-Aug-11	NULL	0.1000146118775133	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1111665587205952	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	inhibitor	0.028850369	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.012683012	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
SLC30A9	hgnc:1329	SLC30A9	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.075768645	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	4.375639269641208	Fotemustine	ncit:C1106	FOTEMUSTINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.02706581	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00626658	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.037693949	NSC-638080	chembl:CHEMBL136344	CHEMBL:CHEMBL136344	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.095904422	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.4667348554283955	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
RORA	hgnc:10258	RORA	DTC	9/2/20	NULL	0.8204323630577265	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.3017682254924971	ROFLUMILAST	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.076840494	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:11666	iuphar.ligand:11666	ATUZABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3175	iuphar.ligand:3175	GERANYL BIPHOSPHONATE	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.1172046232939609	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	0.1470803115845784	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.082171629	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	SYM-004	chembl:CHEMBL2109388	FUTUXIMAB	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.033487035	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.083279415	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
MACROPHAGE INFLAMMATORY PROTEIN 1-ALPHA	hgnc:10627	CCL3	TTD	2020.06.01	NULL	17.50255707856483	Nagrestipen	ncit:C98294	NAGRESTIPEN	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	negative modulator	0.067839369	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1000146118775133	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.1693795846312726	UPADACITINIB	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	2.442217266776488	VALPROPYLHYDROXAMIC ACID	chembl:CHEMBL186311	VALPROPYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:524	iuphar.ligand:524	ARC-239	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:9787	drugbank:DB12903	DEBIO-1347	FALSE	FALSE	FALSE
NCBIGENE:311	hgnc:535	ANXA11	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:2932	iuphar.ligand:2932	L-LACTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:1612	iuphar.ligand:1612	[3H]DIPRENORPHINE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.061628722	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.006908904	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	TALC	12-May-16	vaccine	0.1159109740302306	AD.P53-DC	ncit:C148241	AUTOLOGOUS DENDRITIC CELLS TRANSDUCED WITH WILD-TYPE P53 ADENOVIRUS VACCINE	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1250182648468916	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	PROGABIDE	rxcui:34568	PROGABIDE	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.4688184931758437	VITAMIN B12	rxcui:11248	VITAMIN B12	TRUE	FALSE	FALSE
PRKG1	hgnc:9414	PRKG1	DTC	9/2/20	NULL	0.072324616	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.2273059360852575	GNF-PF-5061	chembl:CHEMBL601385	CHEMBL:CHEMBL601385	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	TALC	12-May-16	inhibitor	7.778914257139925	RILOTUMUMAB	ncit:C67079	RILOTUMUMAB	FALSE	TRUE	TRUE
ERBB3	hgnc:3431	ERBB3	DTC	9/2/20	NULL	0.5147810905460245	METHYLCURCUMIN	chembl:CHEMBL494826	METHYLCURCUMIN	FALSE	FALSE	FALSE
PSMB8	hgnc:9545	PSMB8	DTC	9/2/20	NULL	4.773424657790408	BELACTOSIN A	chembl:CHEMBL491636	BELACTOSIN A	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.2067231151011594	METHOXYARACHIDONOYL FLUOROPHOSPHONATE	chembl:CHEMBL113262	METHOXYARACHIDONOYL FLUOROPHOSPHONATE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.010388507	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.1666910197958555	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2835	iuphar.ligand:2835	GSK4716	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:10382	drugbank:DB11968	MK-7145	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:7870	iuphar.ligand:7870	COMPOUND 1 [PMID: 24900526]	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.6105543166941221	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.7955707762984014	GYROPHORIC ACID	chembl:CHEMBL470648	GYROPHORIC ACID	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.061340737	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.1396480617970598	APTIGANEL	ncit:C79861	APTIGANEL	FALSE	FALSE	FALSE
NCBIGENE:669	hgnc:1093	BPGM	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:12456	iuphar.ligand:12456	SINIGRIN	FALSE	FALSE	FALSE
DUSP6	hgnc:3072	DUSP6	CIViC	10-Apr-24	NULL	0.3500511415712966	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1312691780892362	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.085796848	IUPHAR.LIGAND:6741	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	DoCM	10-Apr-24	NULL	1.040600372117402	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
FASLG	hgnc:11936	FASLG	NCI	14-Sep-17	NULL	0.1973972602845657	ANGIOTENSIN CONVERTING ENZYME INHIBITOR	ncit:C247	ACE INHIBITOR	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.029970132	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.2678962818147678	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.4795221117415022	SELITRECTINIB	ncit:C138160	SELITRECTINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.831662950082366	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.145753425	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	NSC-11437	chembl:CHEMBL1814509	CHEMBL:CHEMBL1814509	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:6194	iuphar.ligand:6194	N-METHYL LTC4	FALSE	FALSE	FALSE
MYELOPEROXIDASE	hgnc:7218	MPO	TTD	2020.06.01	NULL	1.750255707856483	E-101	ncit:C114986	E-101 SOLUTION	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BENFURACARB	ncit:C163590	BENFURACARB	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	0.1682938180631233	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.017679351	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	MyCancerGenome	20-Jun-17	inhibitor	1.312691780892362	DANUSERTIB	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	NCI	14-Sep-17	NULL	0.4070362111294147	BRONCHODILATOR	ncit:C319	BRONCHODILATOR	FALSE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.062509132	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	FLUORESCEIN DIACETATE	chembl:CHEMBL1492044	FLUORESCEIN DIACETATE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.2453629496995069	HORMONE THERAPY	ncit:C147908	HORMONE THERAPY AGENT	FALSE	FALSE	TRUE
AR	hgnc:644	AR	CGI	2/1/22	NULL	NULL	Orterone	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	CGI	2/1/22	NULL	2.212697851403848	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	CGI	2/1/22	NULL	4.702860988936115	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.1108075556053025	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	2,4,6-TRIBROMOPHENOL	drugbank:DB02417	2,4,6-TRIBROMOPHENOL	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.1535312024435511	Ado-Trastuzumab Emtansine	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.6482428547616605	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
PALB2	hgnc:26144	PALB2	CGI	2/1/22	NULL	NULL	Platinum Agent	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004172574	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
NOTCH2	hgnc:7882	NOTCH2	CGI	2/1/22	NULL	1.500219178	Mk-0752	drugbank:DB12852	MK-0752	FALSE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CGI	2/1/22	NULL	0.5527123287967842	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.2075402025126264	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.1562728310586145	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	CGI	2/1/22	NULL	0.055329474	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.1750255707856483	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RAD50	hgnc:9816	RAD50	CGI	2/1/22	NULL	NULL	2 inhibitor	NULL	NULL	NULL	NULL	NULL
ATM	hgnc:795	ATM	CGI	2/1/22	NULL	NULL	2 inhibitor	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	PROPARACAINE	rxcui:34905	PROPARACAINE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	CGI	2/1/22	NULL	0.3513393859865807	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.1250182648468916	Rociletinib	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.086361301	Rociletinib	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	DNDI1416934	chembl:CHEMBL1989750	CHEMBL:CHEMBL1989750	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.1535312024435511	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	FLUPHENAZINE ENANTHATE	rxcui:30129	FLUPHENAZINE ENANTHATE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	2.258394462	GOLIMUMAB	rxcui:819300	GOLIMUMAB	TRUE	TRUE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.031929262	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
TPO	hgnc:12015	TPO	ChEMBL	33	inhibitor	2.500365296937833	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	0.7955707762984014	GONADORELIN ACETATE	rxcui:204193	GONADORELIN ACETATE	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	ChEMBL	33	inhibitor	0.31414846	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.2224901323546377	DNDI1417147	chembl:CHEMBL2094484	CHEMBL:CHEMBL2094484	FALSE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	0.9376369863516874	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.5016656487486736	CALCIPOTRIENE	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.019929531	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.072125922	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
FAS	hgnc:11920	FAS	ChEMBL	33	inhibitor	0.069638821	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
PPPK-DHPS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFADOXINE	rxcui:10173	SULFADOXINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	4-(7-METHYLOCTYL)PHENOL	chembl:CHEMBL503990	CHEMBL:CHEMBL503990	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.4861821410712453	AMPHETAMINE ADIPATE	ncit:C87425	AMPHETAMINE ADIPATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.080164384	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.145753425	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
M	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIMANTADINE HYDROCHLORIDE	rxcui:82093	RIMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.04339477	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.596678082	ROFLUMILAST	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	0.4321619031744403	PRAVASTATIN SODIUM	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.1223004764806549	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.08334551	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.729273212	ESOMEPRAZOLE SODIUM	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.192335792	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
CA13	hgnc:14914	CA13	ChEMBL	33	inhibitor	1.750255707856483	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.038894571	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.042174836	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.1810609352954983	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.1620607136904151	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.091583148	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.046881849	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.2051080907644316	MIDODRINE HYDROCHLORIDE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.036718651	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.02926849	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.050488145	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.023274677	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.3106962795011509	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.2243917574174979	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.5834185692854945	SODIUM NITROPRUSSIDE	rxcui:9895	SODIUM NITROPRUSSIDE	TRUE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.3671865121377238	ISOSORBIDE DINITRATE	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.6177373086552295	SODIUM NITROPRUSSIDE	rxcui:9895	SODIUM NITROPRUSSIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.108711535	NAPHAZOLINE HYDROCHLORIDE	rxcui:82054	NAPHAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.056888051	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.2586584789935689	TOLAZAMIDE	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.3750547945406749	GLIPIZIDE	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	1.750255707856483	ACETOHEXAMIDE	rxcui:173	ACETOHEXAMIDE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.078136416	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELAPREVIR	rxcui:1102261	TELAPREVIR	TRUE	FALSE	FALSE
M	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	ChEMBL	33	inhibitor	2.573905452730122	CANAKINUMAB	rxcui:853491	CANAKINUMAB	TRUE	TRUE	TRUE
FABI	NULL	NULL	ChEMBL	33	inhibitor	NULL	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
FABI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TRICLOSAN	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	PALIVIZUMAB	rxcui:194279	PALIVIZUMAB	TRUE	FALSE	FALSE
PBPB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZLOCILLIN SODIUM	rxcui:203836	AZLOCILLIN SODIUM	TRUE	FALSE	FALSE
PBPA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZLOCILLIN SODIUM	rxcui:203836	AZLOCILLIN SODIUM	TRUE	FALSE	FALSE
PONB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZLOCILLIN SODIUM	rxcui:203836	AZLOCILLIN SODIUM	TRUE	FALSE	FALSE
PBPC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZLOCILLIN SODIUM	rxcui:203836	AZLOCILLIN SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZLOCILLIN SODIUM	rxcui:203836	AZLOCILLIN SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZLOCILLIN SODIUM	rxcui:203836	AZLOCILLIN SODIUM	TRUE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	ChEMBL	33	inhibitor	17.50255707856483	ABOBOTULINUMTOXINA	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
COL4A6	hgnc:2208	COL4A6	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
COL11A1	hgnc:2186	COL11A1	ChEMBL	33	cleavage	0.086361301	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	VORICONAZOLE	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	TERCONAZOLE	rxcui:37806	TERCONAZOLE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULCONAZOLE NITRATE	rxcui:56798	SULCONAZOLE NITRATE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIOCONAZOLE	rxcui:38298	TIOCONAZOLE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	POSACONAZOLE	rxcui:282446	POSACONAZOLE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXICONAZOLE NITRATE	rxcui:32638	OXICONAZOLE	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	agonist	0.3409589041278864	SUCCINYLCHOLINE CHLORIDE	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	negative modulator	0.026680727	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	negative modulator	0.025439763	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	negative modulator	0.026045472	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	negative modulator	0.028413242	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	negative modulator	0.026045472	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.092606122	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	negative modulator	0.027010119	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.094950581	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.060169218	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.081407242	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.032412143	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.025003653	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.027276712	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.026927011	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.050879526	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.056097939	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.052090944	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.048618214	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.053361455	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.049723174	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.033658764	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.031254566	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.032016873	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.034318739	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.03591496	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.041739007	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.038131933	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.040112812	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.037666909	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.079557078	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.039390601	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.020164236	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.018613141	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.021715331	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.020656047	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROVAFLOXACIN MESYLATE	rxcui:221177	TROVAFLOXACIN MESYLATE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	MAFENIDE ACETATE	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFISOXAZOLE DIOLAMINE	rxcui:10208	SULFISOXAZOLE DIOLAMINE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFADIAZINE SODIUM	rxcui:220087	SULFADIAZINE SODIUM	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFACETAMIDE	rxcui:10169	SULFACETAMIDE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAMETHIZOLE	rxcui:10179	SULFAMETHIZOLE	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	agonist	0.7955707762984013	LYPRESSIN	rxcui:6531	LYPRESSIN	TRUE	FALSE	FALSE
BLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TAZOBACTAM SODIUM	rxcui:221167	TAZOBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-3	NULL	NULL	ChEMBL	33	inhibitor	NULL	TAZOBACTAM SODIUM	rxcui:221167	TAZOBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-4	NULL	NULL	ChEMBL	33	inhibitor	NULL	TAZOBACTAM SODIUM	rxcui:221167	TAZOBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-5	NULL	NULL	ChEMBL	33	inhibitor	NULL	TAZOBACTAM SODIUM	rxcui:221167	TAZOBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-6	NULL	NULL	ChEMBL	33	inhibitor	NULL	TAZOBACTAM SODIUM	rxcui:221167	TAZOBACTAM SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERTAPENEM SODIUM	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.040051618	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERTAPENEM SODIUM	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERTAPENEM SODIUM	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERTAPENEM SODIUM	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	NSC-11437	chembl:CHEMBL1814509	CHEMBL:CHEMBL1814509	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.1319288222002374	PROPIDIUM	drugbank:DB02166	PROPIDIUM	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.3409589041278863	SB-242235	chembl:CHEMBL95692	SB-242235	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014160645	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	GNF-PF-3286	chembl:CHEMBL581880	CHEMBL:CHEMBL581880	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.1174668260306364	TCMDC-135909	chembl:CHEMBL453384	CHEMBL:CHEMBL453384	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.012794267	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIMETHOMORPH	chembl:CHEMBL3138617	DIMETHOMORPH	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	2-(METHYLSULFONAMIDO)BENZOIC ACID	chembl:CHEMBL491550	CHEMBL:CHEMBL491550	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.054243462	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.009553798	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	METIZOLINE	ncit:C99577	METIZOLINE	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.3017682254924971	INTERFERON ALFA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
IL2RG	hgnc:6010	IL2RG	ChEMBL	33	inhibitor	1.750255707856483	BASILIXIMAB	rxcui:196102	BASILIXIMAB	TRUE	TRUE	FALSE
RPSZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPME2	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMG1	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMG2	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
RPMG3	NULL	NULL	ChEMBL	33	inhibitor	NULL	RETAPAMULIN	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROVAFLOXACIN MESYLATE	rxcui:221177	TROVAFLOXACIN MESYLATE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROVAFLOXACIN MESYLATE	rxcui:221177	TROVAFLOXACIN MESYLATE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LOMEFLOXACIN HYDROCHLORIDE	rxcui:235762	LOMEFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LOMEFLOXACIN HYDROCHLORIDE	rxcui:235762	LOMEFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GREPAFLOXACIN HYDROCHLORIDE	rxcui:236862	GREPAFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GREPAFLOXACIN HYDROCHLORIDE	rxcui:236862	GREPAFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
PRIM1	hgnc:9369	PRIM1	ChEMBL	33	inhibitor	0.2206204673768676	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLD3	hgnc:20932	POLD3	ChEMBL	33	inhibitor	0.2573905452730122	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLE2	hgnc:9178	POLE2	ChEMBL	33	inhibitor	0.2573905452730122	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLD4	hgnc:14106	POLD4	ChEMBL	33	inhibitor	0.108040476	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.062808219	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.05293112	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.2386712328895204	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.057574201	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.076765601	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.057700738	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.074163377	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.068369364	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.057574201	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	GREPAFLOXACIN HYDROCHLORIDE	rxcui:236862	GREPAFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNK3	hgnc:6278	KCNK3	ChEMBL	33	potentiator	0.2419708351875322	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	GREPAFLOXACIN HYDROCHLORIDE	rxcui:236862	GREPAFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSR1	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSR2	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	SIMEPREVIR SODIUM	rxcui:1484518	SIMEPREVIR SODIUM	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	DESVENLAFAXINE FUMARATE	chembl:CHEMBL3989861	DESVENLAFAXINE FUMARATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	LEVOMILNACIPRAN HYDROCHLORIDE	rxcui:1433211	LEVOMILNACIPRAN HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.1374032518317239	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	PARITAPREVIR	rxcui:1597373	PARITAPREVIR	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.1810609352954983	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
HCN4	hgnc:16882	HCN4	ChEMBL	33	blocker	1.093909817410302	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.1250182648468916	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	inhibitor	3.281729452230906	CANGRELOR TETRASODIUM	rxcui:1656051	CANGRELOR TETRASODIUM	TRUE	FALSE	FALSE
KCNJ2	hgnc:6263	KCNJ2	ChEMBL	33	blocker	3.281729452230906	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PSMB9	hgnc:9546	PSMB9	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	5.104912481248077	SONIDEGIB PHOSPHATE	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.4375639269641209	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
PSMD1	hgnc:9554	PSMD1	ChEMBL	33	inhibitor	0.5385402178019948	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	inhibitor	0.2763561643983921	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
PSMA1	hgnc:9530	PSMA1	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMB11	hgnc:31963	PSMB11	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMD7	hgnc:9565	PSMD7	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.058471794	VK5211	chembl:CHEMBL3545356	VK5211	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	ChEMBL	33	modulator	0.2083637747448194	MOFAROTENE	ncit:C63667	MOFAROTENE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	inhibitor	0.801643836	RELACORILANT	ncit:C127838	RELACORILANT	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.3621218705909966	AC-480	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.546954909	MIRANSERTIB	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1666910197958555	AC-480	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.4070362111294147	AZD-7451	chembl:CHEMBL3545179	AZD-7451	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	0.8078103267029924	TOVORAFENIB	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1223955040459079	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.092606122	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	ChEMBL	33	inhibitor	0.062808219	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.3697723326457359	HENATINIB	drugbank:DB13019	HENATINIB	FALSE	FALSE	FALSE
TRPM8	hgnc:17961	TRPM8	ChEMBL	33	agonist	8.290684931951763	D-3263	chembl:CHEMBL3707315	D-3263	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	positive modulator	0.3125456621172291	PESAMPATOR	ncit:C186393	PESAMPATOR	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.6250913242344582	MK-6913	chembl:CHEMBL3545274	MK-6913	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.037160418	LUNACALCIPOL	iuphar.ligand:11382	LUNACALCIPOL	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	modulator	0.42006137	INT131	chembl:CHEMBL1236924	INT131	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	FX-005	chembl:CHEMBL3545216	FX-005	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1584738568481725	FRUQUINTINIB	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	inhibitor	0.375054795	KW-2450	chembl:CHEMBL3545156	KW-2450	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.4953553890159858	KW-2450	chembl:CHEMBL3545156	KW-2450	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	0.1438566335224506	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.069454592	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
TGFBR1	hgnc:11772	TGFBR1	ChEMBL	33	inhibitor	2.500365296937833	GALUNISERTIB	ncit:C116891	GALUNISERTIB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.064413418	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1250182648468916	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.1374546367426557	RAF-265	drugbank:DB05984	RAF-265	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.073540156	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.095036509	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	ChEMBL	33	inhibitor	0.082043236	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	ChEMBL	33	inhibitor	0.1193356164447602	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.023110771	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.8751278539282416	TEPOTINIB	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	BAVISANT	ncit:C171762	BAVISANT	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	2.838252499226729	EVODENOSON	ncit:C169974	EVODENOSON	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	3.281729452230906	GLASDEGIB	rxcui:2105845	GLASDEGIB	TRUE	FALSE	TRUE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	1.419126249613364	SERLOPITANT	ncit:C81499	SERLOPITANT	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	4.375639269641208	PATIDEGIB	ncit:C80063	PATIDEGIB	FALSE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.1605739181519709	SAMIDORPHAN	rxcui:2559612	SAMIDORPHAN	TRUE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	inhibitor	5.834185692854944	MAVOGLURANT	ncit:C170154	MAVOGLURANT	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	1.458546423213736	NAXIFYLLINE	ncit:C83991	NAXIFYLLINE	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	2.763561643983921	AZD1981	iuphar.ligand:7680	AZD1981	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	3.500511415712966	MK3207	chembl:CHEMBL1910936	MK3207	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	1.458546423213736	PBF-680	chembl:CHEMBL3545162	PBF-680	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	inhibitor	1.141471113819445	SRX246	iuphar.ligand:12262	SRX246	FALSE	FALSE	FALSE
KCNH1	hgnc:6250	KCNH1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1339481409073839	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	ChEMBL	33	blocker	0.070010228	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.079798892	ASM-024	chembl:CHEMBL3707249	ASM-024	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1013661606866689	ASM-024	chembl:CHEMBL3707249	ASM-024	FALSE	FALSE	FALSE
PMP22	hgnc:9118	PMP22	DTC	9/2/20	NULL	3.750547945406749	KETOPROFEN	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	ChEMBL	33	inhibitor	0.3125456621172291	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	ChEMBL	33	inhibitor	0.023609564	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	TESAGLITAZAR	ncit:C75985	TESAGLITAZAR	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	3.500511415712966	TIVANTINIB	ncit:C62437	TIVANTINIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.2634164108814105	MOMELOTINIB	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	ELBASVIR	rxcui:1734628	ELBASVIR	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	ChEMBL	33	inhibitor	0.5609793935437446	TARIQUIDAR	ncit:C2246	TARIQUIDAR	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.035719504	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	2-AMINO-ANTHRAQUINONE	chembl:CHEMBL84685	CHEMBL:CHEMBL84685	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	ChEMBL	33	inhibitor	3.088686543276147	ALEPLASININ	ncit:C76071	ALEPLASININ	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	ChEMBL	33	modulator	0.729273212	DUVOGLUSTAT HYDROCHLORIDE	ncit:C87374	DUVOGLUSTAT HYDROCHLORIDE	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	0.8204323630577265	ERTUGLIFLOZIN	rxcui:1992672	ERTUGLIFLOZIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000236197	chembl:CHEMBL582496	CHEMBL:CHEMBL582496	FALSE	FALSE	FALSE
MYL4	hgnc:7585	MYL4	ChEMBL	33	activator	2.187819634820604	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
GBA1	hgnc:4177	GBA1	ChEMBL	33	modulator	1.500219178	AFEGOSTAT TARTRATE	ncit:C83521	AFEGOSTAT TARTRATE	FALSE	FALSE	FALSE
PNP	hgnc:7892	PNP	ChEMBL	33	inhibitor	35.00511415712966	FORODESINE HYDROCHLORIDE	ncit:C26655	FORODESINE HYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE	chembl:CHEMBL1255936	CHEMBL:CHEMBL1255936	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	ChEMBL	33	inhibitor	0.1067229090156392	OBATOCLAX MESYLATE	ncit:C62771	OBATOCLAX MESYLATE	FALSE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	ChEMBL	33	inhibitor	1.406455479527531	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	ChEMBL	33	inhibitor	1.790034246671403	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
BIRC2	hgnc:590	BIRC2	ChEMBL	33	inhibitor	1.312691780892362	BIRINAPANT	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.4375639269641208	IRINOTECAN SUCROSOFATE	ncit:C82676	IRINOTECAN SUCROSOFATE	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	ChEMBL	33	inhibitor	0.1562728310586145	OBATOCLAX MESYLATE	ncit:C62771	OBATOCLAX MESYLATE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.5427149481725528	ALPRENOLOL	rxcui:597	ALPRENOLOL	FALSE	FALSE	FALSE
BCL2A1	hgnc:991	BCL2A1	ChEMBL	33	inhibitor	1.458546423213736	OBATOCLAX MESYLATE	ncit:C62771	OBATOCLAX MESYLATE	FALSE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMINOSALICYLIC ACID	rxcui:7833	AMINOSALICYLIC ACID	TRUE	FALSE	FALSE
UL97	NULL	NULL	ChEMBL	33	inhibitor	NULL	MARIBAVIR	rxcui:2586068	MARIBAVIR	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	1.875273972703375	GUSELKUMAB	rxcui:1928588	GUSELKUMAB	TRUE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	0.900131507	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
CALCB	hgnc:1438	CALCB	ChEMBL	33	inhibitor	5.834185692854944	EPTINEZUMAB	rxcui:2282660	EPTINEZUMAB	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	TCMDC-123868	chembl:CHEMBL548615	CHEMBL:CHEMBL548615	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	inhibitor	0.071928317	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
TGFB3	hgnc:11769	TGFB3	ChEMBL	33	inhibitor	4.375639269641208	FRESOLIMUMAB	ncit:C63546	FRESOLIMUMAB	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.8140724222588294	ICI-118551	chembl:CHEMBL513389	ICI-118551	FALSE	FALSE	FALSE
AOC3	hgnc:550	AOC3	ChEMBL	33	inhibitor	13.12691780892362	VEPALIMOMAB	ncit:C152854	VEPALIMOMAB	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	MAB-425	chembl:CHEMBL2109390	MAB-425	FALSE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	ChEMBL	33	inhibitor	6.177373086552294	NI-0801	chembl:CHEMBL2109379	NI-0801	FALSE	FALSE	FALSE
TNFRSF8	hgnc:11923	TNFRSF8	ChEMBL	33	other/unknown	9.845188356692718	IRATUMUMAB	ncit:C26441	IRATUMUMAB	FALSE	FALSE	FALSE
S1PR2	hgnc:3169	S1PR2	ChEMBL	33	modulator	1.500219178	AMISELIMOD HYDROCHLORIDE	ncit:C142922	AMISELIMOD HYDROCHLORIDE	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.1105424657593568	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
LINGO1	hgnc:21205	LINGO1	ChEMBL	33	inhibitor	26.25383561784724	OPICINUMAB	ncit:C170259	OPICINUMAB	FALSE	FALSE	FALSE
FN1	hgnc:3778	FN1	ChEMBL	33	binder	8.078103267029922	L19IL2	chembl:CHEMBL2109608	L19IL2	FALSE	FALSE	TRUE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
ICOSLG	hgnc:17087	ICOSLG	ChEMBL	33	inhibitor	52.50767123569449	AMG-557	chembl:CHEMBL2109249	AMG-557	FALSE	FALSE	FALSE
IFNA10	hgnc:5418	IFNA10	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
IFNA13	hgnc:5419	IFNA13	ChEMBL	33	inhibitor	1.346350544504987	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
MUC5AC	hgnc:7515	MUC5AC	ChEMBL	33	binder	13.12691780892362	YTTRIUM Y 90 CLIVATUZUMAB TETRAXETAN	chembl:CHEMBL2108708	YTTRIUM Y 90 CLIVATUZUMAB TETRAXETAN	FALSE	FALSE	FALSE
NCAM1	hgnc:7656	NCAM1	ChEMBL	33	binder	13.12691780892362	BB-10901	chembl:CHEMBL2109484	BB-10901	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	2.000292237550266	EMIBETUZUMAB	ncit:C95732	EMIBETUZUMAB	FALSE	TRUE	TRUE
IFNA1	hgnc:5417	IFNA1	ChEMBL	33	inhibitor	0.3671865121377238	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
IFNA14	hgnc:5420	IFNA14	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
CSF2RA	hgnc:2435	CSF2RA	ChEMBL	33	inhibitor	5.834185692854944	MAVRILIMUMAB	ncit:C95788	MAVRILIMUMAB	FALSE	FALSE	FALSE
STXB	NULL	NULL	ChEMBL	33	inhibitor	NULL	URTOXAZUMAB	ncit:C152808	URTOXAZUMAB	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	BENZYDAMINE HYDROCHLORIDE	rxcui:81963	BENZYDAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	inhibitor	0.07767407	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.1187956362798518	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	BENZYDAMINE HYDROCHLORIDE	rxcui:81963	BENZYDAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFODIZIME	rxcui:20485	CEFODIZIME	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFODIZIME	rxcui:20485	CEFODIZIME	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFODIZIME	rxcui:20485	CEFODIZIME	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFODIZIME	rxcui:20485	CEFODIZIME	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFODIZIME	rxcui:20485	CEFODIZIME	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFODIZIME	rxcui:20485	CEFODIZIME	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFODIZIME	rxcui:20485	CEFODIZIME	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.8468979231563628	DIMETHINDENE	rxcui:3449	DIMETHINDENE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	agonist	0.8899605294185507	ANGIOTENSIN II ACETATE	ncit:C142924	ANGIOTENSIN II ACETATE	TRUE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	binder	0.5834185692854945	LUTETIUM DOTATATE LU-177	chembl:CHEMBL3989924	LUTETIUM DOTATATE LU-177	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	1.944728564284981	TOSITUMOMAB 131I	chembl:CHEMBL3833304	TOSITUMOMAB 131I	FALSE	FALSE	FALSE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	8.751278539282415	CNTO-5825	chembl:CHEMBL2109464	CNTO-5825	FALSE	FALSE	FALSE
ICOS	hgnc:5351	ICOS	ChEMBL	33	inhibitor	35.00511415712966	MEDI-570	chembl:CHEMBL2109449	MEDI-570	FALSE	FALSE	FALSE
MPL	hgnc:7217	MPL	ChEMBL	33	agonist	4.773424657790408	AVATROMBOPAG MALEATE	rxcui:2045727	AVATROMBOPAG MALEATE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.027781837	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE	chembl:CHEMBL1255936	CHEMBL:CHEMBL1255936	FALSE	FALSE	FALSE
OPG057	NULL	NULL	ChEMBL	33	inhibitor	NULL	TECOVIRIMAT	rxcui:2055104	TECOVIRIMAT	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.4070362111294147	LAROTRECTINIB SULFATE	rxcui:2104548	LAROTRECTINIB SULFATE	TRUE	FALSE	FALSE
BLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RELEBACTAM	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
GLA	hgnc:4296	GLA	ChEMBL	33	modulator	4.039051633514961	MIGALASTAT HYDROCHLORIDE	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
AMPC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RELEBACTAM	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
BLAUOE-1	NULL	NULL	ChEMBL	33	inhibitor	NULL	RELEBACTAM	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	RAFOXANIDE	ncit:C152146	RAFOXANIDE	FALSE	FALSE	FALSE
ITK	hgnc:6171	ITK	ChEMBL	33	inhibitor	0.5147810905460244	PF-06651600	chembl:CHEMBL4085457	PF-06651600	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.022869195	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	inhibitor	0.032899543	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	inhibitor	0.024674658	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.02232469	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.021805511	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.024041974	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.021805511	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.022869195	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.5147810905460245	ZANUBRUTINIB	rxcui:2262435	ZANUBRUTINIB	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	SOVAPREVIR	ncit:C152411	SOVAPREVIR	FALSE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	FURAPREVIR	ncit:C166437	FURAPREVIR	FALSE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	NARLAPREVIR	ncit:C166554	NARLAPREVIR	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAZUFLOXACIN	ncit:C66331	PAZUFLOXACIN	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PAZUFLOXACIN	ncit:C66331	PAZUFLOXACIN	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SITAFLOXACIN	ncit:C76922	SITAFLOXACIN	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SITAFLOXACIN	ncit:C76922	SITAFLOXACIN	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SITAFLOXACIN	ncit:C76922	SITAFLOXACIN	FALSE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	FOSRAVUCONAZOLE	ncit:C175721	FOSRAVUCONAZOLE	FALSE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	ChEMBL	33	inhibitor	1.909369863116163	VADADUSTAT	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
LY6E	hgnc:6727	LY6E	ChEMBL	33	binder	3.281729452230906	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2442217266776488	NITRENDIPINE	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	ChEMBL	33	inhibitor	0.5834185692854944	CADONILIMAB	ncit:C153379	CADONILIMAB	FALSE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	SETROBUVIR	ncit:C152351	SETROBUVIR	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	ChEMBL	33	inhibitor	1.105424657593568	PELABRESIB	ncit:C188265	PELABRESIB	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	negative modulator	NULL	LOMIBUVIR	ncit:C166650	LOMIBUVIR	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOXACILLIN	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOXACILLIN	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOXACILLIN	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOXACILLIN	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOXACILLIN	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOXACILLIN	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	RADEZOLID	ncit:C81442	RADEZOLID	FALSE	FALSE	FALSE
LTB4R2	hgnc:19260	LTB4R2	ChEMBL	33	inhibitor	6.563458904461812	CP-195543	drugbank:DB13053	CP-195543	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEMONOXACIN	ncit:C174838	NEMONOXACIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.042174836	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEMONOXACIN	ncit:C174838	NEMONOXACIN	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.042174836	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.035719504	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.038894571	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
DPRE1	NULL	NULL	ChEMBL	33	inhibitor	NULL	TBA-7371	drugbank:DB16243	TBA-7371	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.064033745	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	negative modulator	0.1389091831632129	BDTX189	chembl:CHEMBL4650279	BDTX189	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	SERDEXMETHYLPHENIDATE CHLORIDE	rxcui:2562177	SERDEXMETHYLPHENIDATE CHLORIDE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.1646008502686348	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	0.9723642821424908	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	inhibitor	0.7095631248066824	DU 125530	chembl:CHEMBL79261	DU 125530	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	ZIRESOVIR	ncit:C170395	ZIRESOVIR	FALSE	FALSE	FALSE
TOPB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ZOLIFLODACIN	ncit:C152962	ZOLIFLODACIN	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.2365210416022274	TALSACLIDINE	ncit:C96885	TALSACLIDINE	FALSE	FALSE	FALSE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	0.4167275494896388	OLVEREMBATINIB	ncit:C165549	OLVEREMBATINIB	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	ELRANATAMAB	rxcui:2644880	ELRANATAMAB	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
FABI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CG-400549	drugbank:DB12347	CG-400549	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
ECE1	hgnc:3146	ECE1	ChEMBL	33	inhibitor	5.250767123569449	DAGLUTRIL	ncit:C73039	DAGLUTRIL	FALSE	FALSE	FALSE
PIKFYVE	hgnc:23785	PIKFYVE	ChEMBL	33	inhibitor	52.50767123569449	APILIMOD MESYLATE	ncit:C90809	APILIMOD MESYLATE	FALSE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	agonist	1.093909817410302	CD40 LIGAND	iuphar.ligand:5077	CD40 LIGAND	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	ChEMBL	33	inhibitor	1.750255707856483	VERDIPERSTAT	ncit:C152861	VERDIPERSTAT	FALSE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	ChEMBL	33	inhibitor	1.544343271638073	BMS-823778	iuphar.ligand:10158	BMS-823778	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.088945801	LEVOSULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	SAMIDORPHAN L-MALATE	rxcui:2570387	SAMIDORPHAN L-MALATE	TRUE	FALSE	FALSE
ALOX5AP	hgnc:436	ALOX5AP	ChEMBL	33	inhibitor	7.501095891	VELIFLAPON	ncit:C152848	VELIFLAPON	FALSE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	ChEMBL	33	inhibitor	0.8751278539282416	ERFONRILIMAB	ncit:C157632	ERFONRILIMAB	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	PSI-352938	drugbank:DB12896	PSI-352938	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	VALOPICITABINE	ncit:C66649	VALOPICITABINE	FALSE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFALAZIL	ncit:C152213	RIFALAZIL	FALSE	FALSE	FALSE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFALAZIL	ncit:C152213	RIFALAZIL	FALSE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFALAZIL	ncit:C152213	RIFALAZIL	FALSE	FALSE	FALSE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFALAZIL	ncit:C152213	RIFALAZIL	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	2.282942227638891	PF-4136309	drugbank:DB17200	PF-4136309	FALSE	FALSE	FALSE
HA	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIS-410	chembl:CHEMBL4594613	VIS-410	FALSE	FALSE	FALSE
EEF2	hgnc:3214	EEF2	ChEMBL	33	negative modulator	0.9723642821424906	LMB-100	drugbank:DB18591	LMB-100	FALSE	FALSE	FALSE
ACE-1	NULL	NULL	ChEMBL	33	inhibitor	NULL	TRICHLORFON	rxcui:1000581	TRICHLORFON	TRUE	FALSE	FALSE
KLH1	NULL	NULL	ChEMBL	33	vaccine	NULL	ADAGLOXAD SIMOLENIN	ncit:C99766	ADAGLOXAD SIMOLENIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	ChEMBL	33	inhibitor	0.2318219480604613	SIREMADLIN	ncit:C116325	SIREMADLIN	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.2500365296937833	TRAZPIROBEN	ncit:C171664	TRAZPIROBEN	FALSE	FALSE	FALSE
DPRE1	NULL	NULL	ChEMBL	33	inhibitor	NULL	MACOZINONE	ncit:C174599	MACOZINONE	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	1.458546423213736	RESIMMUNE	chembl:CHEMBL4297555	RESIMMUNE	FALSE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	blocker	0.1442518440541058	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
TACR3	hgnc:11528	TACR3	ChEMBL	33	inhibitor	2.917092846427472	ELINZANETANT	ncit:C174774	ELINZANETANT	FALSE	FALSE	FALSE
CD47	hgnc:1682	CD47	ChEMBL	33	inhibitor	13.12691780892362	EVORPACEPT	ncit:C132851	EVORPACEPT	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.042968634	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
TUF1	NULL	NULL	ChEMBL	33	inhibitor	NULL	LFF-571	drugbank:DB13013	LFF-571	FALSE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	blocker	0.2243917574174979	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	ChEMBL	33	inhibitor	0.2151953739167807	BIRICODAR	ncit:C71621	BIRICODAR	FALSE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	blocker	0.2019525816757481	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	blocker	0.2243917574174979	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
ADAMTS5	hgnc:221	ADAMTS5	ChEMBL	33	inhibitor	8.751278539282415	ALDUMASTAT	ncit:C175739	ALDUMASTAT	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	OTESECONAZOLE	rxcui:2602577	OTESECONAZOLE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFILAVANCIN	ncit:C169833	CEFILAVANCIN	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFILAVANCIN	ncit:C169833	CEFILAVANCIN	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFILAVANCIN	ncit:C169833	CEFILAVANCIN	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFILAVANCIN	ncit:C169833	CEFILAVANCIN	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFILAVANCIN	ncit:C169833	CEFILAVANCIN	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFILAVANCIN	ncit:C169833	CEFILAVANCIN	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFILAVANCIN	ncit:C169833	CEFILAVANCIN	FALSE	FALSE	FALSE
RIPK1	hgnc:10019	RIPK1	ChEMBL	33	inhibitor	26.25383561784724	GSK2982772	iuphar.ligand:9554	GSK2982772	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1312691780892362	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
PRKAA1	hgnc:9376	PRKAA1	ClearityFoundationClinicalTrial	15-Jun-13	activator	0.029301156	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	COSMIC	4-Sep-20	NULL	4.702860988936115	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	COSMIC	4-Sep-20	NULL	0.4735540335109532	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	COSMIC	4-Sep-20	NULL	0.065226921	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NR1H2	hgnc:7965	NR1H2	DTC	9/2/20	NULL	1.262203635473425	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.6806549974997433	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.078252863	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.023609564	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
HSF1	hgnc:5224	HSF1	DTC	9/2/20	NULL	0.138178082	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.004043095	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.546954909	GNF-PF-4068	chembl:CHEMBL584668	CHEMBL:CHEMBL584668	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.006049271	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.4234489615781814	DIMETHYL YELLOW	chembl:CHEMBL263116	DIMETHYL YELLOW	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.080781033	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00393537	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	(R)-PINOCEMBRIN	chembl:CHEMBL399249	(R)-PINOCEMBRIN	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.2651902587661338	DNDI1417599	chembl:CHEMBL2094833	CHEMBL:CHEMBL2094833	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	NCG-C00094300-01	chembl:CHEMBL1256754	CHEMBL:CHEMBL1256754	FALSE	FALSE	FALSE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.072324616	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.033875917	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	NSC-81747	chembl:CHEMBL1371696	CHEMBL:CHEMBL1371696	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.2476776945079929	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.030176823	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	4-AMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL60824	4-AMINO-[1,2]NAPHTHOQUINONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	ESCULETIN	iuphar.ligand:5180	ESCULETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	SULFISOXAZOLE	rxcui:10207	SULFISOXAZOLE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.040452751	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	TCMDC-123781	chembl:CHEMBL581194	CHEMBL:CHEMBL581194	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.008143249	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.023943307	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	(R,S)-IFENPRODIL	chembl:CHEMBL49623	(R,S)-IFENPRODIL	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	CRYPTOCHINONE B	chembl:CHEMBL1223741	CRYPTOCHINONE B	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	BISANHYDRORUTILANTINONE	chembl:CHEMBL1436035	BISANHYDRORUTILANTINONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	MECLOFENAMATE SODIUM	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01823183	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.2917092846427472	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.072826174	ROSE BENGAL	rxcui:9471	ROSE BENGAL	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1981421556063943	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.1438566335224507	PERMETHRIN	rxcui:33199	PERMETHRIN	TRUE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.28382525	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	TCMDC-123992	chembl:CHEMBL530149	CHEMBL:CHEMBL530149	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.036718651	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	1.693795846312725	NSC-88915	chembl:CHEMBL387152	CHEMBL:CHEMBL387152	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	ANTIMYCIN A	chembl:CHEMBL211501	ANTIMYCIN A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TETRABUTYLAMMONIUM BROMIDE	chembl:CHEMBL60696	TETRABUTYLAMMONIUM BROMIDE	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.067403943	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007813642	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2328499833068492	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2580229544751573	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	PIRFENIDONE	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	ALACHLOR	chembl:CHEMBL1414154	ALACHLOR	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.0135995	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL199592	CHEMBL:CHEMBL199592	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	GNF-PF-1295	chembl:CHEMBL579837	CHEMBL:CHEMBL579837	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	IOXYNIL	chembl:CHEMBL509523	IOXYNIL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00195778	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	U-0124	chembl:CHEMBL97858	CHEMBL:CHEMBL97858	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	TCMDC-125298	chembl:CHEMBL581152	CHEMBL:CHEMBL581152	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.01823183	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.072125922	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	DNDI1417484	chembl:CHEMBL1308677	CHEMBL:CHEMBL1308677	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.019607047	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.4526523382387456	TENONITROZOLE	rxcui:236186	TENONITROZOLE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	RIBOFLAVIN	rxcui:9346	RIBOFLAVIN	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.4102161815288632	OLSALAZINE	rxcui:32385	OLSALAZINE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	DTC	9/2/20	NULL	1.158257453728555	PRALIDOXIME	rxcui:1546365	PRALIDOXIME CATION	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	CAFFEIC ACID	rxcui:1311397	CAFFEIC ACID	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1250182648468916	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	chembl:CHEMBL1226	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004458114	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.040390516	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.072424374	DIBENZ[A,H]ANTHRACENE	chembl:CHEMBL1346946	DIBENZ[A,H]ANTHRACENE	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	1.750255707856483	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1325951293830669	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.015429818	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.052455216	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	0.2027323213733378	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.061773731	INDOCYANINE GREEN SODIUM	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.1526385791735305	RAUWOLSCINE	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.5357925636295356	IB-MECA	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.059667808	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.087952548	AMPICILLIN TRIHYDRATE	rxcui:203115	AMPICILLIN TRIHYDRATE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	ANGUIDIN	chembl:CHEMBL433680	ANGUIDIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.012713722	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	2.442217266776488	4-CHLOROBENZOHYDROXAMIC ACID	chembl:CHEMBL569419	CHEMBL:CHEMBL569419	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	ETICLOPRIDE	ncit:C65572	ETICLOPRIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006570029	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.1041818873724097	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	DIMETHYLPHENYLPIPERAZINIUM IODIDE	chembl:CHEMBL47814	DIMETHYLPHENYLPIPERAZINIUM IODIDE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	INDOCYANINE GREEN SODIUM	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	DNDI1417759	chembl:CHEMBL1446254	CHEMBL:CHEMBL1446254	FALSE	FALSE	FALSE
NCOR2	hgnc:7673	NCOR2	DTC	9/2/20	NULL	1.093909817410302	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.9293393139060973	THEONELLASTEROL H	chembl:CHEMBL1782603	THEONELLASTEROL H	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	SCOULERINE	chembl:CHEMBL1235966	SCOULERINE	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.04321619	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.030004384	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	N-ACETYLCOLCHINOL	chembl:CHEMBL486504	N-ACETYLCOLCHINOL	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.3182283105193606	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.044763573	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1861974157294131	DAIDZIN	drugbank:DB02115	DAIDZIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	BROMHEXINE HYDROCHLORIDE	rxcui:1601	BROMHEXINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	QUERCITRIN	chembl:CHEMBL82242	QUERCITRIN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	NSC-7387	chembl:CHEMBL119878	CHEMBL:CHEMBL119878	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001432522	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2051080907644316	TCMDC-125603	chembl:CHEMBL528734	CHEMBL:CHEMBL528734	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ANGUIDIN	chembl:CHEMBL433680	ANGUIDIN	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.1275696580070323	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV008455	chembl:CHEMBL584655	CHEMBL:CHEMBL584655	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	CID 1540545	chembl:CHEMBL259784	CHEMBL:CHEMBL259784	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NSC-176327	chembl:CHEMBL363332	CHEMBL:CHEMBL363332	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.009213489	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.07148764	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	FEPRAZONE	rxcui:8673	FEPRAZONE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.017951341	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW631581B	chembl:CHEMBL176553	GW631581B	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	SJ000281118	chembl:CHEMBL592561	CHEMBL:CHEMBL592561	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.022632617	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.004865425	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
CDC42	hgnc:1736	CDC42	DTC	9/2/20	NULL	8.751278539282415	ZU-3594419	chembl:CHEMBL562095	CHEMBL:CHEMBL562095	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010093747	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.080781033	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DNDI1417457	chembl:CHEMBL1530911	CHEMBL:CHEMBL1530911	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.1470803115845784	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1136529680426287	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	GNF-PF-2755	chembl:CHEMBL600738	CHEMBL:CHEMBL600738	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.031861451	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	PAXILLINE	iuphar.ligand:2309	PAXILLINE	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.097236428	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.00574545	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.024309107	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.025390557	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.014405397	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	BRONOPOL	rxcui:1114345	BRONOPOL	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2660861718025059	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.3906820776465364	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	DIPHYLLIN	chembl:CHEMBL221190	DIPHYLLIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.061701141	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011810092	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-735465	chembl:CHEMBL261440	CHEMBL:CHEMBL261440	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005284588	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.8140724222588294	CARTEOLOL	rxcui:2116	CARTEOLOL	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.026372512	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.027855529	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.015777545	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	VU0080241	iuphar.ligand:6227	VU0080241	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	2.333674277141977	1,4-DICHLOROBENZENE	chembl:CHEMBL190982	1,4-DICHLOROBENZENE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	TCMDC-123598	chembl:CHEMBL547269	CHEMBL:CHEMBL547269	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.005085489	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.011540148	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
DGAT1	hgnc:2843	DGAT1	DTC	9/2/20	NULL	21.00306849427779	PF-04620110	drugbank:DB14887	PF-04620110	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.1400204566285186	PROCHLORAZ	chembl:CHEMBL522782	PROCHLORAZ	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	GNF-PF-1134	chembl:CHEMBL600694	CHEMBL:CHEMBL600694	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GR-4661	chembl:CHEMBL344127	CHEMBL:CHEMBL344127	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.2917092846427472	FEPRAZONE	rxcui:8673	FEPRAZONE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	GNF-PF-516	chembl:CHEMBL602970	CHEMBL:CHEMBL602970	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.041872146	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.019724895	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.053038052	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1207072901969988	DNDI1417388	chembl:CHEMBL1528359	CHEMBL:CHEMBL1528359	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	MORICIZINE	rxcui:40169	MORICIZINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	PD-0118057	iuphar.ligand:7676	PD-118057	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.375054795	ALOSETRON HYDROCHLORIDE	rxcui:85247	ALOSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.068637479	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV000621	chembl:CHEMBL601743	CHEMBL:CHEMBL601743	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.043466615	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	UCCF-029	iuphar.ligand:4335	UCCF-029	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.058341857	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	TCMDC-124336	chembl:CHEMBL527271	CHEMBL:CHEMBL527271	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.003883703	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002088278	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.019318496	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.03729238	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.064824285	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.039778539	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	1,7-O-DIACETYLMETHYLGEOPYXIN A	chembl:CHEMBL1889303	CHEMBL:CHEMBL1889303	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.006868237	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.049723174	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
FPR2	hgnc:3827	FPR2	DTC	9/2/20	NULL	8.751278539282415	AG-09/96	chembl:CHEMBL1290139	CHEMBL:CHEMBL1290139	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.005592467	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	NSC-145669	chembl:CHEMBL191611	CHEMBL:CHEMBL191611	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	SJ000111875	chembl:CHEMBL590949	CHEMBL:CHEMBL590949	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	GNF-PF-4012	chembl:CHEMBL584269	CHEMBL:CHEMBL584269	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	TCMDC-123927	chembl:CHEMBL531268	CHEMBL:CHEMBL531268	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	FEPRAZONE	rxcui:8673	FEPRAZONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	SB-431542	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.012573676	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	THIOINOSINE	ncit:C877	THIOINOSINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	TCMDC-125134	chembl:CHEMBL546975	CHEMBL:CHEMBL546975	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.072524408	CHELERYTHRINE CHLORIDE	chembl:CHEMBL258893	CHELERYTHRINE CHLORIDE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.008481291	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.030004384	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	BREFELDIN A	drugbank:DB07348	BREFELDIN A	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	SJ000111875	chembl:CHEMBL590949	CHEMBL:CHEMBL590949	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.3889457128569963	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.024721126	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.3889457128569963	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1715936968486748	DIMETHYLPINOCEMBRIN	chembl:CHEMBL107131	DIMETHYLPINOCEMBRIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	BROMOCRIPTINE MESYLATE	rxcui:142426	BROMOCRIPTINE MESYLATE	TRUE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	DTC	9/2/20	NULL	6.563458904461812	S-TRITYL-L-CYSTEINE	chembl:CHEMBL392695	S-TRITYL-L-CYSTEINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	OCTADEC-17-YNOIC ACID	iuphar.ligand:8851	17-OCTADECYNOIC ACID	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.2386712328895204	DNDI1417165	chembl:CHEMBL1406948	CHEMBL:CHEMBL1406948	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.3302369260106572	GAMBOGIC AMIDE	chembl:CHEMBL444109	GAMBOGIC AMIDE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.046221542	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006439499	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	GNF-PF-3343	chembl:CHEMBL599943	CHEMBL:CHEMBL599943	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	HYDROXYLAMMONIUM CHLORIDE	chembl:CHEMBL542448	HYDROXYLAMMONIUM CHLORIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	DEXMEDETOMIDINE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	SJ000114961	chembl:CHEMBL590168	CHEMBL:CHEMBL590168	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	DTC	9/2/20	NULL	0.3281729452230906	GALANTAMINE	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	6-AZAURIDINE	ncit:C291	6-AZAURIDINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001770916	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.069824031	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.072927321	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	DTC	9/2/20	NULL	0.072324616	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005563432	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.012026494	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.055504938	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.018131102	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.4303907478335614	EMTRICITABINE	rxcui:276237	EMTRICITABINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	NSC-102030	chembl:CHEMBL406834	CHEMBL:CHEMBL406834	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009875432	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006705961	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	GNF-PF-5149	chembl:CHEMBL600309	CHEMBL:CHEMBL600309	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	SB-224289	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.084012274	PROPYLPARABEN	rxcui:34706	PROPYLPARABEN	TRUE	FALSE	FALSE
CHRM5	hgnc:1954	CHRM5	DTC	9/2/20	NULL	0.2059124362184098	PIPERTRAMINE AMIDE	chembl:CHEMBL130835	PIPERTRAMINE AMIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	1-HEXYLPYRIDINIUM IODIDE	chembl:CHEMBL555242	CHEMBL:CHEMBL555242	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	PROPANTHELINE BROMIDE	rxcui:8762	PROPANTHELINE BROMIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.022789788	CYPROHEPTADINE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001144706	ATORVASTATIN CALCIUM	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.2476776945079929	TCMDC-124063	chembl:CHEMBL534535	CHEMBL:CHEMBL534535	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	NSC-636948	chembl:CHEMBL1998001	CHEMBL:CHEMBL1998001	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.6863747873946993	CARDAMOMIN	chembl:CHEMBL378104	CARDAMOMIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	FLUOCINOLONE ACETONIDE	rxcui:4461	FLUOCINOLONE ACETONIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.008599357	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.1600843635234588	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.094608417	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CYSTEINE	rxcui:3024	CYSTEINE	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2536602475154323	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	NSC-49789	chembl:CHEMBL469309	CHEMBL:CHEMBL469309	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.085378327	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.052090944	ARTEMISININ	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.3017682254924971	CID 4970947	chembl:CHEMBL1451921	CHEMBL:CHEMBL1451921	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1562728310586145	VU0080241	iuphar.ligand:6227	VU0080241	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	IMETIT DIHYDROBROMIDE	chembl:CHEMBL544911	IMETIT DIHYDROBROMIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.02339914	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	1.810609352954982	FORMETOREX	ncit:C65752	FORMETOREX	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.081030357	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.014832675	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.020778659	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.1235474617310458	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001678098	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CID 2093195	chembl:CHEMBL411085	CHEMBL:CHEMBL411085	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	SJ000119988	chembl:CHEMBL589694	CHEMBL:CHEMBL589694	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.042516333	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	AMINOQUINURIDE	rxcui:17747	AMINOQUINURIDE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.032982206	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.09745299	NANDROLONE PHENPROPIONATE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.009481342	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.058341857	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	GNF-PF-3343	chembl:CHEMBL599943	CHEMBL:CHEMBL599943	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	NSC-116702	chembl:CHEMBL1477383	CHEMBL:CHEMBL1477383	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	PHENACETIN	rxcui:8113	PHENACETIN	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	DTC	9/2/20	NULL	0.5791287268642775	GALANTAMINE	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.050781113	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	TOSYL-L-LYSINE CHLOROMETHYL KETONE	chembl:CHEMBL466465	CHEMBL:CHEMBL466465	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	TAMSULOSIN HYDROCHLORIDE	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.046059361	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.5073204950308646	ISOSILYBIN B	chembl:CHEMBL3542340	ISOSILYBIN B	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	ITRAZOLE	chembl:CHEMBL64391	ITRACONAZOLE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	PROPYLPARABEN	rxcui:34706	PROPYLPARABEN	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.020778659	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	CGS-12066A MALEATE	chembl:CHEMBL1256689	CHEMBL:CHEMBL1256689	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	GNF-PF-5392	chembl:CHEMBL576809	CHEMBL:CHEMBL576809	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.076208521	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.3387591692625452	FLUAZINAM	chembl:CHEMBL1878267	FLUAZINAM	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	MMV007396	chembl:CHEMBL582286	CHEMBL:CHEMBL582286	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.045898314	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	TCMDC-123781	chembl:CHEMBL581194	CHEMBL:CHEMBL581194	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.037884323	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	CUDRAFLAVONE B	chembl:CHEMBL221907	CUDRAFLAVONE B	FALSE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	DTC	9/2/20	NULL	8.078103267029922	20S-HYDROXYVITAMIN D3	chembl:CHEMBL2036072	CHEMBL:CHEMBL2036072	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.070574827	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	IMETIT	iuphar.ligand:1250	IMETIT	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.026385764	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	GW775608X	chembl:CHEMBL476351	GW775608X	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.03292017	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-4291	chembl:CHEMBL585462	CHEMBL:CHEMBL585462	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.046881849	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	DEMETHOXYCURCUMIN	chembl:CHEMBL179512	DEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00301197	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
MARK4	hgnc:13538	MARK4	DTC	9/2/20	NULL	0.1198805279353755	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
FZD1	hgnc:4038	FZD1	DTC	9/2/20	NULL	0.9723642821424907	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.021933029	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-4945	chembl:CHEMBL585628	CHEMBL:CHEMBL585628	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.084146909	MP-412	chembl:CHEMBL5095024	MP-412	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.084012274	2-PHENYLPHENOL	rxcui:236677	2-PHENYLPHENOL	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	RO-106-9920	chembl:CHEMBL271023	CHEMBL:CHEMBL271023	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.016027983	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.1339481409073839	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.6250913242344582	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	8-CYCLOPENTYLTHEOPHYLLINE	iuphar.ligand:385	8-CYCLOPENTYLTHEOPHYLLINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.01214331	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	U-50488 METHANE SULFONATE	iuphar.ligand:1652	U50488	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.100589408	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.092851762	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	PARBENDAZOLE	ncit:C96752	PARBENDAZOLE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	N-(3-PHENYLPROPYL)BENZAMIDE	chembl:CHEMBL1404865	CHEMBL:CHEMBL1404865	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	METHYLISOTHIOCYANATE	chembl:CHEMBL396000	METHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.1268301237577161	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.1553481397505754	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	GITOXIN	chembl:CHEMBL109317	GITOXIN	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1325951293830669	TCMDC-123927	chembl:CHEMBL531268	CHEMBL:CHEMBL531268	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.2853677784548614	HTS-05058	chembl:CHEMBL261692	CHEMBL:CHEMBL261692	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.077444943	SCOULERINE	chembl:CHEMBL1235966	SCOULERINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	NSC-106547	chembl:CHEMBL223575	CHEMBL:CHEMBL223575	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.1875273972703375	WIN-62577	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.020737627	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	N,N'-DIPHENYL-GUANIDINE	chembl:CHEMBL77675	CHEMBL:CHEMBL77675	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.3763990769583835	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	U-101958	iuphar.ligand:5781	U101958	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.315046027	FENOFIBRIC ACID	rxcui:24852	FENOFIBRIC ACID	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2'-HYDROXY-2,3,4',6',TETRAMETHOXYCHALCONE	chembl:CHEMBL1254091	CHEMBL:CHEMBL1254091	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	N-(4-(CYANO(PHENYL)METHYL)PHENYL)ACETAMIDE	chembl:CHEMBL1580175	CHEMBL:CHEMBL1580175	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-2414	chembl:CHEMBL601353	CHEMBL:CHEMBL601353	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.011176601	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.003105125	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.013781541	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.023110771	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.4375639269641209	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.017295017	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	(S)-5-IODOWILLARDIINE	drugbank:DB02818	IODO-WILLARDIINE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.05853698	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.088396753	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	5-NITRO-[1,10]PHENANTHROLINE	chembl:CHEMBL101815	CHEMBL:CHEMBL101815	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	NIZOFENONE	ncit:C76783	NIZOFENONE	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.4930297768609811	NALTREXONE HYDROCHLORIDE	rxcui:105069	NALTREXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010588359	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.091159151	TYRAMINE	rxcui:10958	TYRAMINE	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.2323348284765243	SJ000244621	chembl:CHEMBL600175	CHEMBL:CHEMBL600175	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.062808219	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	3,5-DIMETHOXYISONAPHTHOIC ACID	chembl:CHEMBL1608067	CHEMBL:CHEMBL1608067	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.182318303	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BROMCRESOL GREEN	iuphar.ligand:4530	BROMOCRESOL GREEN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	DIETHYLSTILBESTROL DIPROPIONATE	ncit:C74557	DIETHYLSTILBESTROL DIPROPIONATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	MECHLORETHAMINE HYDROCHLORIDE	rxcui:155036	MECHLORETHAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	RELCOVAPTAN	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	DTC	9/2/20	NULL	6.563458904461812	CLASTO-LACTACYSTIN BETA-LACTONE	chembl:CHEMBL490829	CHEMBL:CHEMBL490829	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	REL-CARINATIN C	chembl:CHEMBL2332127	CHEMBL:CHEMBL2332127	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	ISOETHARINE MESYLATE	rxcui:6024	ISOETHARINE MESYLATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.044535769	E-GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.033985548	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV008160	chembl:CHEMBL586026	CHEMBL:CHEMBL586026	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	DTC	9/2/20	NULL	0.7095631248066824	VU0365137	chembl:CHEMBL1084941	CHEMBL:CHEMBL1084941	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00506733	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	4.039051633514961	BYAKANGELICIN	chembl:CHEMBL508648	BYAKANGELICIN	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.3017682254924971	GNF-PF-4665	chembl:CHEMBL601744	CHEMBL:CHEMBL601744	FALSE	FALSE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	0.3535870116881784	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.1458546423213736	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.016574391	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.3977853881492006	DEMETHOXYCURCUMIN	chembl:CHEMBL179512	DEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.2465148884304905	ABIETIC ACID	chembl:CHEMBL71893	ABIETIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NSC-99550	chembl:CHEMBL1288014	CHEMBL:CHEMBL1288014	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.2586584789935689	IB-MECA	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	MMV007396	chembl:CHEMBL582286	CHEMBL:CHEMBL582286	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.058602312	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	DIPICOLINIC ACID	drugbank:DB04267	DIPICOLINIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	6-CHLOROMELATONIN	iuphar.ligand:1346	6-CL-MLT	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	DICLAZURIL	rxcui:1368201	DICLAZURIL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CHLOROXURON	chembl:CHEMBL1568699	CHLOROXURON	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.046798281	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	GNF-PF-4068	chembl:CHEMBL584668	CHEMBL:CHEMBL584668	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.4339476961627644	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	CARBAZOLE	drugbank:DB07301	CARBAZOLE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.062065805	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	MESORIDAZINE	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	LOMATIN	chembl:CHEMBL1414353	LOMATIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005903055	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003027077	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.027333509	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TRIBROMOACETIC ACID	chembl:CHEMBL502627	TRIBROMOACETIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	ISOCONAZOLE	rxcui:27901	ISOCONAZOLE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	2-PHENYLPHENOL	rxcui:236677	2-PHENYLPHENOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	METHANESULFONIC ACID METHYL ESTER	chembl:CHEMBL313493	METHANESULFONIC ACID METHYL ESTER	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	SJ000024553	chembl:CHEMBL589238	CHEMBL:CHEMBL589238	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.045265234	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	ANTHRALIN	rxcui:873	ANTHRALIN	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.5469549087051511	DUVOGLUSTAT	ncit:C87373	DUVOGLUSTAT	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	2-(2-AMINOETHYL)ISOTHIOUREA DIHYDROBROMIDE	chembl:CHEMBL1256025	CHEMBL:CHEMBL1256025	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	NSC-106547	chembl:CHEMBL223575	CHEMBL:CHEMBL223575	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.017543492	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MERCURIC IODIDE	rxcui:1426941	MERCURIC IODIDE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.015097088	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	DILTIAZEM	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00411841	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.011219588	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.055681518	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
CYP1B1	hgnc:2597	CYP1B1	DTC	9/2/20	NULL	3.182283105193606	2'H,4H-[2,8'-BICHROMEN]-4-ONE	chembl:CHEMBL2347757	2'H,4H-[2,8'-BICHROMEN]-4-ONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	GNF-PF-4012	chembl:CHEMBL584269	CHEMBL:CHEMBL584269	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004708786	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.1084869240406911	MONO-N-ACETYL DAPSONE	chembl:CHEMBL1246	MONO-N-ACETYL DAPSONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	LEUCINE	rxcui:6308	LEUCINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SALICYLHYDROXAMIC ACID	drugbank:DB03819	SALICYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.031555091	PD-173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	(-)-LEPTOCLINIDAMINE B	chembl:CHEMBL2208197	CHEMBL:CHEMBL2208197	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	20(S)-PROTOPANAXATRIOL	chembl:CHEMBL255683	CHEMBL:CHEMBL255683	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.028199609	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
CAMK2A	hgnc:1460	CAMK2A	DTC	9/2/20	NULL	0.4412409347537353	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	NSC-23217	chembl:CHEMBL1367935	CHEMBL:CHEMBL1367935	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	CGP-7930	iuphar.ligand:1079	CGP7930	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.008224886	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
TLR9	hgnc:15633	TLR9	DTC	9/2/20	NULL	0.2573905452730122	DEMETHOXYCURCUMIN	chembl:CHEMBL179512	DEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	GNF-PF-4945	chembl:CHEMBL585628	CHEMBL:CHEMBL585628	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	OMEPRAZOLE MAGNESIUM	rxcui:236486	OMEPRAZOLE MAGNESIUM	TRUE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.2524407270946851	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.015791781	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIIB	chembl:CHEMBL1094683	AESCULIOSIDE IIIB	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011188509	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.280789686	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	RADANAMYCIN	chembl:CHEMBL383015	RADANAMYCIN	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.062509132	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PICONOL	chembl:CHEMBL2103981	PICONOL	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	PIMETHIXENE MALEATE	ncit:C97703	PIMETHIXENE MALEATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	PRIDINOL METHANESULFONATE	chembl:CHEMBL1528011	PRIDINOL METHANESULFONATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009433646	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	BMS-182874	chembl:CHEMBL267458	BMS-182874	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	SB-242084	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00626658	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.027121731	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007813642	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.005585922	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.011741429	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
LDHA	hgnc:6535	LDHA	DTC	9/2/20	NULL	52.50767123569449	TETRAHYDRO-NAD	chembl:CHEMBL2058994	CHEMBL:CHEMBL2058994	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00808059	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	DTC	9/2/20	NULL	0.4895820161836317	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	INDOCYANINE GREEN SODIUM	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.1232574442152452	NSC-22225	chembl:CHEMBL462314	CHEMBL:CHEMBL462314	FALSE	FALSE	FALSE
PRKAB1	hgnc:9378	PRKAB1	DTC	9/2/20	NULL	1.875273972703374	SAPONARIN	chembl:CHEMBL538921	SAPONARIN	FALSE	FALSE	FALSE
PRKAG2	hgnc:9386	PRKAG2	DTC	9/2/20	NULL	3.750547945406749	SAPONARIN	chembl:CHEMBL538921	SAPONARIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	AMPEROZIDE	ncit:C74191	AMPEROZIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.014638325	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	SULFADIAZINE, SILVER	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00808059	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.0135995	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	METHOXSALEN	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.012683012	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	MICONAZOLE NITRATE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.2917092846427472	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	DTC	9/2/20	NULL	3.182283105193606	2'H,4H-[2,5'-BICHROMEN]-4-ONE	chembl:CHEMBL2347758	2'H,4H-[2,5'-BICHROMEN]-4-ONE	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.2983390411119005	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	FENOLDOPAM BROMIDE	chembl:CHEMBL1256646	FENOLDOPAM BROMIDE	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.3409589041278864	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.1704794520639432	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.043039075	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	SJ000260249	chembl:CHEMBL601311	CHEMBL:CHEMBL601311	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.018206543	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	DNDI1417739	chembl:CHEMBL487356	CHEMBL:CHEMBL487356	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007946076	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DESERPIDINE	rxcui:62174	DESERPIDINE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.090530468	ISOETHARINE MESYLATE	rxcui:6024	ISOETHARINE MESYLATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001399085	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.03409589	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.9376369863516875	CEFUROXIME	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004961042	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	SJ000113372	chembl:CHEMBL589912	CHEMBL:CHEMBL589912	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-125810	chembl:CHEMBL528119	CHEMBL:CHEMBL528119	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.1037701012563132	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.172722603	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.022439176	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00218782	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	N,N'-DIPHENYL-GUANIDINE	chembl:CHEMBL77675	CHEMBL:CHEMBL77675	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005527705	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.099446347	TEGASEROD MALEATE	rxcui:339270	TEGASEROD MALEATE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	FORMONONETIN	drugbank:DB15335	FORMONONETIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	ISOBOLDINE	chembl:CHEMBL462880	ISOBOLDINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001886051	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.024309107	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	SJ000276790	chembl:CHEMBL602922	CHEMBL:CHEMBL602922	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.008288504	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.078958904	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	INDOCYANINE GREEN SODIUM	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	4.375639269641208	AZELAIC ACID	rxcui:18602	AZELAIC ACID	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	TCMDC-124416	chembl:CHEMBL530664	CHEMBL:CHEMBL530664	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000721874	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.027781837	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00389812	CANDESARTAN CILEXETIL	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	DTC	9/2/20	NULL	0.6819178082557728	HU-210	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.032899543	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	GNF-PF-1654	chembl:CHEMBL602776	CHEMBL:CHEMBL602776	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1944728564284981	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	chembl:CHEMBL1226	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	2.561349816375341	NOBILAMIDE B	chembl:CHEMBL1784750	NOBILAMIDE B	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012112496	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	SPIRAMIDE	ncit:C66559	SPIRAMIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.034118045	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.013415348	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.1835932560688619	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.061701141	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	DICHLORODIPHENYLDICHLOROETHYLENE	chembl:CHEMBL363207	DICHLORODIPHENYLDICHLOROETHYLENE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	NSC-62406	chembl:CHEMBL1332182	CHEMBL:CHEMBL1332182	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1944728564284981	GNF-PF-4068	chembl:CHEMBL584668	CHEMBL:CHEMBL584668	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	VANIPREVIR	ncit:C152828	VANIPREVIR	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.3977853881492007	ABT-702	iuphar.ligand:5131	ABT702	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	ISOCONAZOLE	rxcui:27901	ISOCONAZOLE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	SULOCHRIN	chembl:CHEMBL61133	SULOCHRIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CID 1540951	chembl:CHEMBL259421	CHEMBL:CHEMBL259421	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.1187956362798518	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DIBENZ[A,H]ANTHRACENE	chembl:CHEMBL1346946	DIBENZ[A,H]ANTHRACENE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-108	chembl:CHEMBL578929	CHEMBL:CHEMBL578929	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	CYSTAMINE HYDROCHLORIDE	chembl:CHEMBL1256388	CYSTAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2744303374687866	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.088945801	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	PIROCTONE	rxcui:2058907	PIROCTONE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.012354746	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.1682938180631234	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-2755	chembl:CHEMBL600738	CHEMBL:CHEMBL600738	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.05814803	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.1178056726441863	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.057700738	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
SIRT5	hgnc:14933	SIRT5	DTC	9/2/20	NULL	6.563458904461812	GNF-PF-1720	chembl:CHEMBL578329	CHEMBL:CHEMBL578329	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.2638576444004749	DCMU	chembl:CHEMBL278489	DCMU	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.036718651	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	CIS-RESVERATROL	chembl:CHEMBL87333	CIS-RESVERATROL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	GNF-PF-3125	chembl:CHEMBL534288	CHEMBL:CHEMBL534288	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.039361073	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.9460841664089098	ISORHAMNETIN	drugbank:DB16767	ISORHAMNETIN	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.047518255	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	FDA	10-Apr-24	NULL	0.6471533709721451	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.003405608	Carvedilol	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.034727296	Avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.002529881	Citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	3.150460274	Daclatasvir	rxcui:1606218	DACLATASVIR	FALSE	FALSE	FALSE
GALNS	hgnc:4122	GALNS	FDA	10-Apr-24	NULL	NULL	Elosulfase	NULL	NULL	NULL	NULL	NULL
NTRK	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
GLA	hgnc:4296	GLA	FDA	10-Apr-24	NULL	4.039051633514961	Migalastat	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Ramucirumab	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.04427291	Palonosetron	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.029443554	Raloxifene	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.007749066	Phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
CYB5R	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Rasburicase	rxcui:283821	RASBURICASE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.210030685	Ropivacaine	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	FDA	10-Apr-24	NULL	0.031707531	Rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Trifluridine	rxcui:10803	TRIFLURIDINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.2917092846427472	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.061737415	Vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.01090502	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.038256955	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	NULL	TAK901	NULL	NULL	NULL	NULL	NULL
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.3236220106976548	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.009603891	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	1.175544878411071	PF-03814735	drugbank:DB13059	PF-03814735	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	MyCancerGenome	20-Jun-17	inhibitor	0.297662535	PD0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
BTK	hgnc:1133	BTK	MyCancerGenome	20-Jun-17	inhibitor	0.02617531	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.1715936968486748	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.1172046232939609	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.049026771	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.1607377690888607	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.04464938	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.057700738	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	MyCancerGenome	20-Jun-17	inhibitor	0.1835932560688619	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
SYK	hgnc:11491	SYK	MyCancerGenome	20-Jun-17	inhibitor	3.000438356	FOSTAMATINIB	rxcui:2044896	FOSTAMATINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenome	20-Jun-17	inhibitor	0.1375060601009582	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.070129236	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
CTLA4	hgnc:2505	CTLA4	MyCancerGenome	20-Jun-17	immunotherapy	0.7001022831425934	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
CTLA4	hgnc:2505	CTLA4	MyCancerGenome	20-Jun-17	antibody	0.7001022831425934	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
IL1B	hgnc:5992	IL1B	MyCancerGenome	20-Jun-17	immunotherapy	2.573905452730122	CANAKINUMAB	rxcui:853491	CANAKINUMAB	TRUE	TRUE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	antibody	2.000292237550266	LY2875358	ncit:C95732	EMIBETUZUMAB	FALSE	TRUE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.179119736	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1704794520639432	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.0287871	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1229687850953032	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
ADK	hgnc:257	ADK	NCI	14-Sep-17	NULL	0.7001022831425934	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	4.565884455277782	6-METHYLMERCAPTOPURINE RIBOSIDE	ncit:C2352	METHYLMERCAPTOPURINE RIBOSIDE	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	2.282942227638891	ANTIMALARIALS	ncit:C271	ANTIMALARIAL AGENT	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.040766825	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	NCI	14-Sep-17	NULL	0.2308029504865691	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.4150804050252529	DIFFERENTIATING AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
ADAMTS5	hgnc:221	ADAMTS5	NCI	14-Sep-17	NULL	2.333674277141977	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
ADK	hgnc:257	ADK	NCI	14-Sep-17	NULL	0.7501095890813498	2&APOS;,3&APOS;-DIDEOXYINOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	NULL	LIGNANS	NULL	NULL	NULL	NULL	NULL
ALDH3A1	hgnc:405	ALDH3A1	NCI	14-Sep-17	NULL	0.075960465	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	NULL	CHONDROITIN	NULL	NULL	NULL	NULL	NULL
APEX1	hgnc:587	APEX1	NCI	14-Sep-17	NULL	0.1319288222002374	OLTIPRAZ	ncit:C1177	OLTIPRAZ	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.093346971	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1400204566285186	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	0.062509132	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.024564992	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.4268916360625568	ENDOTHELIN RECEPTOR ANTAGONIST	ncit:C28313	ENDOTHELIN RECEPTOR ANTAGONIST	FALSE	FALSE	FALSE
CBS	hgnc:1550	CBS	NCI	14-Sep-17	NULL	3.500511415712966	VITAMIN B6	rxcui:42954	VITAMIN B6	TRUE	FALSE	FALSE
CCL4	hgnc:10630	CCL4	NCI	14-Sep-17	NULL	1.029562181092049	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.02232469	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.011162345	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CD1A	hgnc:1634	CD1A	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	1.750255707856483	PI3-KINASE INHIBITORS	ncit:C2152	PHOSPHATIDYLINOSITIDE 3-KINASE INHIBITOR	FALSE	FALSE	TRUE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	0.2258394461750301	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	0.7001022831425934	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
CD58	hgnc:1688	CD58	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	0.7001022831425934	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.7242437411819932	TUMOR VACCINES	ncit:C1663	ANTINEOPLASTIC VACCINE	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	inhibitor	0.044955198	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	1.458546423213736	TETANUS TOXOID	chembl:CHEMBL2108875	TETANUS TOXOID	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.09741683	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	1.221108633388244	PROPIONIBACTERIUM ACNES	rxcui:1310910	PROPIONIBACTERIUM ACNES	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.064111931	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.042700736	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.073643298	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
CKM	hgnc:1994	CKM	NCI	14-Sep-17	NULL	2.763561643983921	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
CHAT	hgnc:1912	CHAT	NCI	14-Sep-17	NULL	0.2215513554248712	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	0.4861821410712453	MITOMYCIN C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
CGA	hgnc:1885	CGA	NCI	14-Sep-17	NULL	1.312691780892362	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
CHUK	hgnc:1974	CHUK	NCI	14-Sep-17	NULL	0.2885036881082116	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.4321619031744403	IL-1RA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.9723642821424906	CLOMIPHENE CITRATE	rxcui:142431	CLOMIPHENE CITRATE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.017724108	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CRH	hgnc:2355	CRH	NCI	14-Sep-17	NULL	3.281729452230906	MEDICATION	ncit:C459	MEDICATION	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	NULL	RV-GM-CSF	NULL	NULL	NULL	NULL	NULL
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	NULL	SURGICAL ADJUVANT	NULL	NULL	NULL	NULL	NULL
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	0.364636606	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.2243917574174978	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.1682938180631233	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.1223955040459079	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
CX3CL1	hgnc:10647	CX3CL1	NCI	14-Sep-17	NULL	2.917092846427472	COMPLETE FREUND&APOS;S ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005059761	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	NULL	TOTAL PARENTERAL NUTRITION	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.000987116	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.208916464	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
EPHA8	hgnc:3391	EPHA8	NCI	14-Sep-17	NULL	0.577007376	CHEMOTHERAPEUTIC AGENT	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	IRBESARTAN	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
F8	hgnc:3546	F8	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.093652208	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	NCI	14-Sep-17	NULL	0.3088686543276147	TETRAHYDROCANNABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.1539814405738841	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1651184630053286	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.2476776945079929	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	1.000146118775133	HEREGULIN	ncit:C1426	RECOMBINANT HEREGULIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.038894571	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.4118248724368196	ANTIBIOTICS	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.4667348554283955	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.2625383561784725	PENICILLIN	wikidata:Q12190	PENICILLIN	FALSE	FALSE	FALSE
NTSR1	hgnc:8039	NTSR1	DTC	9/2/20	NULL	0.076765601	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	1.29648571	ANABOLIC STEROID	ncit:C2360	ANABOLIC STEROID	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.054355767	NDGA	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.2047082699247349	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.2287915957982331	ANTIBIOTICS	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.061055432	PRED	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
GUCA2A	hgnc:4682	GUCA2A	NCI	14-Sep-17	NULL	2.059124362184098	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.8751278539282416	SELENOMETHIONINE	rxcui:9644	SELENOMETHIONINE	TRUE	FALSE	FALSE
HIST3H2A	hgnc:20507	H2AC25	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
HK1	hgnc:4922	HK1	NCI	14-Sep-17	NULL	7.501095890813499	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.1215455352678113	SODIUM HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.9723642821424906	PROTEOLYTIC ENZYMES	ncit:C38728	PANCREATIC PROTEOLYTIC ENZYMES	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	0.6563458904461813	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	1.640864726115453	MEDICATION	ncit:C459	MEDICATION	FALSE	FALSE	FALSE
HMOX1	hgnc:5013	HMOX1	NCI	14-Sep-17	NULL	2.333674277141978	ZNCL2	rxcui:39937	ZINC CHLORIDE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.1973972602845657	HEXAMETHYLENE BISACETAMIDE	ncit:C1125	HEXAMETHYLENE BISACETAMIDE	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.8751278539282416	BETA-NAPHTHOFLAVONE	ncit:C29812	BETA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.093931433	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.6105543166941221	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.3977853881492008	DIFFERENTIATION AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	NCI	14-Sep-17	NULL	0.041639708	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.016807833	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
IBSP	hgnc:5341	IBSP	NCI	14-Sep-17	NULL	1.400204566285186	ZOLEDRONIC ACID	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	MEPIVACAINE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	NULL	IP-10	NULL	NULL	NULL	NULL	NULL
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.1842374429322613	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	0.9376369863516874	ETIDRONATE	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.8334550989792778	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	BENZTHIAZIDE	rxcui:19008	BENZTHIAZIDE	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005618798	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1930429089547591	ETRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.3241214273808302	RO 31-8220	ncit:C1310	RO 31-8220	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.108040476	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
LGALS2	hgnc:6562	LGALS2	NCI	14-Sep-17	NULL	4.375639269641208	MITOMYCIN C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.051177067	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
MAOB	hgnc:6834	MAOB	NCI	14-Sep-17	NULL	0.054581779	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	NCI	14-Sep-17	NULL	0.1182605208011137	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.050007306	COMPLETE FREUND&APOS;S ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.1100789753368857	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006419031	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.030281241	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.1630673019742065	HEREGULIN	ncit:C1426	RECOMBINANT HEREGULIN	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.093763699	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.167488584	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	NCI	14-Sep-17	NULL	0.070956312	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	NULL	CHONDROITIN	NULL	NULL	NULL	NULL	NULL
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.09972967	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	ICRF-193	chembl:CHEMBL275665	ICRF-193	FALSE	FALSE	FALSE
MT2A	hgnc:7406	MT2A	NCI	14-Sep-17	NULL	0.6646540662746139	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	0.4054646427466756	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.08334551	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.300043836	NOVOBIOCIN	rxcui:7538	NOVOBIOCIN	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.4500657534488099	THYROTROPIN	rxcui:10579	THYROTROPIN	TRUE	FALSE	FALSE
NCOA3	hgnc:7670	NCOA3	NCI	14-Sep-17	NULL	0.1615620653405984	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.01798824	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	ncit:C2149	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	NULL	PHOSPHOROTHIOATE OLIGONUCLEOTIDE	NULL	NULL	NULL	NULL	NULL
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1848861663228679	DIURETIC	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.052090944	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	1.166837138570989	STEEL FACTOR	ncit:C1410	RECOMBINANT HUMAN STEM CELL FACTOR	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1056492378987816	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.3697723326457359	PENICILLIN	wikidata:Q12190	PENICILLIN	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.1773907812016706	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	1.166837138570988	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1112450661773188	SKF-83565 HYDROBROMIDE	chembl:CHEMBL541585	CHEMBL:CHEMBL541585	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.2917092846427472	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.1438566335224507	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.212581665	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	NCI	14-Sep-17	NULL	0.025147352	CYCLOSPORIN	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NTRK2	hgnc:8032	NTRK2	NCI	14-Sep-17	NULL	0.1151484018326633	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PHB2	hgnc:30306	PHB2	NCI	14-Sep-17	NULL	13.12691780892362	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.015683295	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.027010119	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.201952582	BPDE	ncit:C196	BENZO(A)PYRENE-7,8-DIOL 9,10-EPOXIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	DNDI1417165	chembl:CHEMBL1406948	CHEMBL:CHEMBL1406948	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	FLUOROSALAN	ncit:C82318	FLUOROSALAN	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.1666910197958555	ACTIVIN	ncit:C2689	IH636 GRAPE SEED PROANTHOCYANIDIN EXTRACT	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.032899543	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.041672755	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	NULL	IP-10	NULL	NULL	NULL	NULL	NULL
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1250182648468916	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1666910197958555	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	0.2734774543525755	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	NULL	HYPOTENSIVE AGENT	NULL	NULL	NULL	NULL	NULL
PTHLH	hgnc:9607	PTHLH	NCI	14-Sep-17	NULL	4.375639269641208	PROTEOLYTIC ENZYMES	ncit:C38728	PANCREATIC PROTEOLYTIC ENZYMES	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.192335792	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.3365876361262467	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	1.346350544504987	PAMIDRONATE DISODIUM	rxcui:105443	PAMIDRONATE DISODIUM	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	4-METHYL-[1,10]PHENANTHROLINE	chembl:CHEMBL316589	CHEMBL:CHEMBL316589	FALSE	FALSE	FALSE
SDF4	hgnc:24188	SDF4	NCI	14-Sep-17	NULL	1.329308132549227	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	NCI	14-Sep-17	NULL	0.094950581	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
SLAMF1	hgnc:10903	SLAMF1	NCI	14-Sep-17	NULL	0.9376369863516874	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	1.810609352954982	GINGER	rxcui:899420	GINGER ALLERGENIC EXTRACT	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.2586584789935689	ETIDRONATE	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.3621218705909966	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	NULL	ALBUMIN	NULL	NULL	NULL	NULL	NULL
TERT	hgnc:11730	TERT	NCI	14-Sep-17	NULL	0.1154014752432846	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1271372184883643	IFN ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.027383401	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.04724037	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.062733179	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	1.129197231	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
TNFRSF1A	hgnc:11916	TNFRSF1A	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.037666909	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
TNFRSF1B	hgnc:11917	TNFRSF1B	NCI	14-Sep-17	NULL	0.8078103267029924	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.060772768	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.047647615	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.019318496	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.023182195	TRIETHYLENETHIOPHOSPHORAMIDE	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.8678953923255289	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.015627283	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.028977744	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.1178623372293928	ARABINOFURANOSYLCYTOSINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	NULL	CREAM	NULL	NULL	NULL	NULL	NULL
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.5527123287967842	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.1707566544250227	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
TSPYL2	hgnc:24358	TSPYL2	NCI	14-Sep-17	NULL	1.875273972703374	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00575742	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	NCI	14-Sep-17	NULL	0.6364566210387212	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	NCI	14-Sep-17	NULL	0.3590268118679965	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.066465407	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	NULL	UVB	NULL	NULL	NULL	NULL	NULL
USP9Y	hgnc:12633	USP9Y	NCI	14-Sep-17	NULL	2.692701089009974	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.009368006	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	2.625383561784725	AZASERINE	ncit:C289	AZASERINE	FALSE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.9211872146613068	VITAMIN B6	rxcui:42954	VITAMIN B6	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	NULL	POLYPHENOL	NULL	NULL	NULL	NULL	NULL
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.375054795	7-HYDROXYCHLORPROMAZINE	chembl:CHEMBL909	7-HYDROXYCHLORPROMAZINE	FALSE	FALSE	FALSE
RPP30	hgnc:17688	RPP30	PharmGKB	4/5/24	NULL	1.400204566285186	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.028078969	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
SULT1A1	hgnc:11453	SULT1A1	PharmGKB	4/5/24	NULL	43.75639269641208	estrogens	rxcui:4100	ESTROGENS	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.039155609	benzphetamine	rxcui:1422	BENZPHETAMINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.038382801	ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
MDGA2	hgnc:19835	MDGA2	PharmGKB	4/5/24	NULL	1.400204566285186	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.024838066	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
ZMPSTE24	hgnc:12877	ZMPSTE24	PharmGKB	4/5/24	NULL	5.834185692854945	lonafarnib	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
ADRB3	hgnc:288	ADRB3	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	XANTHYLETIN	chembl:CHEMBL303846	XANTHYLETIN	FALSE	FALSE	FALSE
TPH2	hgnc:20692	TPH2	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.596678082	evodiamine	rxcui:2199291	EVODIAMINE	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	NULL	morphine-3-glucuronide	NULL	NULL	NULL	NULL	NULL
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.063160791	dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
NELFCD	hgnc:15934	NELFCD	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	ANTAZOLINE	rxcui:865	ANTAZOLINE	FALSE	FALSE	FALSE
PCYT2	hgnc:8756	PCYT2	PharmGKB	4/5/24	NULL	2.187819634820604	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
FGF22	hgnc:3679	FGF22	DTC	9/2/20	NULL	2.500365296937833	NSC-135810	chembl:CHEMBL1605629	CHEMBL:CHEMBL1605629	FALSE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	PharmGKB	4/5/24	NULL	0.07463777	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1548898856510162	dicloxacillin	rxcui:3356	DICLOXACILLIN	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1548898856510162	rifapentine	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.011063563	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.01787191	reserpine	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.007841647	propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.192335792	fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.005524797	rosiglitazone	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.016574391	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	NULL	Selective serotonin reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	NULL	thioguanosine diphosphate	NULL	NULL	NULL	NULL	NULL
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
ZDHHC3	hgnc:18470	ZDHHC3	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	PharmGKB	4/5/24	NULL	0.008740353	vitamin a	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	NULL	Opioid anesthetics	NULL	NULL	NULL	NULL	NULL
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	NULL	ezetimibe / rosuvastatin	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
METTL3	hgnc:17563	METTL3	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
RIPOR2	hgnc:13872	RIPOR2	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
METTL14	hgnc:29330	METTL14	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
HMOX1	hgnc:5013	HMOX1	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
HPX	hgnc:5171	HPX	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	NULL	Drugs For Treatment Of Tuberculosis	NULL	NULL	NULL	NULL	NULL
NT5C	hgnc:17144	NT5C	PharmGKB	4/5/24	NULL	1.093909817410302	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	NULL	Anticholinergics	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	Actinomycines	NULL	NULL	NULL	NULL	NULL
ATP5F1E	hgnc:838	ATP5F1E	PharmGKB	4/5/24	NULL	0.2419708351875322	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	0.4039051633514962	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
CREB1	hgnc:2345	CREB1	PharmGKB	4/5/24	NULL	0.2273059360852575	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
ADCY1	hgnc:232	ADCY1	PharmGKB	4/5/24	NULL	0.8334550989792776	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.4861821410712454	bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
ICA1	hgnc:5343	ICA1	PharmGKB	4/5/24	NULL	2.187819634820604	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.004520289	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
OR52J3	hgnc:14799	OR52J3	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	PharmGKB	4/5/24	NULL	0.151537291	lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	0.2344092465879218	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.091159151	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.2386712328895204	tranilast	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	NULL	oxymetazoline and tetracaine	NULL	NULL	NULL	NULL	NULL
CYCSP5	hgnc:24416	CYCSP5	PharmGKB	4/5/24	NULL	0.8334550989792776	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
TRIB3	hgnc:16228	TRIB3	PharmGKB	4/5/24	NULL	0.760980743	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
PEBP4	hgnc:28319	PEBP4	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
CMTM8	hgnc:19179	CMTM8	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
PSEN1	hgnc:9508	PSEN1	DTC	9/2/20	NULL	1.514644363	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
AMPD1	hgnc:468	AMPD1	PharmGKB	4/5/24	NULL	0.9723642821424906	regadenoson	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
PURA	hgnc:9701	PURA	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
TSPYL1	hgnc:12382	TSPYL1	PharmGKB	4/5/24	NULL	4.375639269641208	abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
MMP9	hgnc:7176	MMP9	PharmGKB	4/5/24	NULL	0.135503668	Methyldopa	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.2016939996249468	motesanib	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.070197421	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.064724402	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1750255707856483	sulfamethazine	rxcui:10178	SULFAMETHAZINE	TRUE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.1272913242077442	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CYP3A7	hgnc:2640	CYP3A7	PharmGKB	4/5/24	NULL	0.1363835616511545	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.1123158743009508	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.1272913242077442	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.030796288	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	NULL	elexacaftor / tezacaftor / ivacaftor	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	phenothiazines with aliphatic side-chain	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.023493365	ripretinib	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	TCMDC-123868	chembl:CHEMBL548615	CHEMBL:CHEMBL548615	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.068191781	nimesulide	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.3043922970185188	dacarbazine	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.2375912725597036	digoxin	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.1103102336884338	digoxin	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	NULL	atazanavir / ritonavir	NULL	NULL	NULL	NULL	NULL
ENOSF1	hgnc:30365	ENOSF1	PharmGKB	4/5/24	NULL	0.1764963739014941	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IGF2BP2	hgnc:28867	IGF2BP2	PharmGKB	4/5/24	NULL	0.2206204673768676	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
TPH1	hgnc:12008	TPH1	PharmGKB	4/5/24	NULL	0.9376369863516874	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	NULL	thioguanosine monophosphate	NULL	NULL	NULL	NULL	NULL
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	0.31414846	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	0.059837802	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
MMADHC	hgnc:25221	MMADHC	PharmGKB	4/5/24	NULL	10.50153425	betaine	rxcui:1512	BETAINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	SB-224289	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
NEDD4L	hgnc:7728	NEDD4L	PharmGKB	4/5/24	NULL	NULL	Aldosterone antagonists	NULL	NULL	NULL	NULL	NULL
POU5F1	hgnc:9221	POU5F1	PharmGKB	4/5/24	NULL	0.8751278539282417	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
TBL1XR1	hgnc:29529	TBL1XR1	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
APOC1	hgnc:607	APOC1	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.1521961485092594	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.7955707762984013	rilonacept	rxcui:763450	RILONACEPT	TRUE	FALSE	FALSE
TNFRSF11B	hgnc:11909	TNFRSF11B	PharmGKB	4/5/24	NULL	1.363835616511545	pamidronate	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
FNTB	hgnc:3785	FNTB	PharmGKB	4/5/24	NULL	3.500511415712966	lonafarnib	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.040235763	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
CYSLTR2	hgnc:18274	CYSLTR2	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
ASS1	hgnc:758	ASS1	PharmGKB	4/5/24	NULL	0.1785975212098452	hydroxyurea	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	NULL	selective beta-2-adrenoreceptor agonists	NULL	NULL	NULL	NULL	NULL
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	NULL	vitamin d and analogues	NULL	NULL	NULL	NULL	NULL
KLC1	hgnc:6387	KLC1	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	FLAVANONE	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.1082632396612257	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003454907	ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006182465	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006525935	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.023867123	mesalazine	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.1186614039224734	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	NULL	Thiazides, plain	NULL	NULL	NULL	NULL	NULL
IL23R	hgnc:19100	IL23R	PharmGKB	4/5/24	NULL	0.5224643904049203	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	drospirenone / ethinyl estradiol	NULL	NULL	NULL	NULL	NULL
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	NULL	drospirenone / ethinyl estradiol	NULL	NULL	NULL	NULL	NULL
PROC	hgnc:9451	PROC	PharmGKB	4/5/24	NULL	NULL	drospirenone / ethinyl estradiol	NULL	NULL	NULL	NULL	NULL
PROS1	hgnc:9456	PROS1	PharmGKB	4/5/24	NULL	NULL	drospirenone / ethinyl estradiol	NULL	NULL	NULL	NULL	NULL
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.035800685	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	NULL	drospirenone / ethinyl estradiol	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	NULL	topoisomerase I inhibitors	NULL	NULL	NULL	NULL	NULL
TOMM40	hgnc:18001	TOMM40	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	2.333674277141977	asunaprevir	rxcui:1652103	ASUNAPREVIR	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	NULL	zidovudine / lamivudine / abacavir	NULL	NULL	NULL	NULL	NULL
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.5527123287967842	clindamycin	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.051277023	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2344092465879218	levonorgestrel	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
ADCY2	hgnc:233	ADCY2	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
CDX2	hgnc:1806	CDX2	PharmGKB	4/5/24	NULL	NULL	FOLFOX	NULL	NULL	NULL	NULL	NULL
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.326134604	rivastigmine	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.1111273465305703	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
PRKCE	hgnc:9401	PRKCE	PharmGKB	4/5/24	NULL	0.7501095890813498	rivastigmine	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
SOCS3	hgnc:19391	SOCS3	PharmGKB	4/5/24	NULL	0.6908904109959803	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1154860804304131	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
IL11	hgnc:5966	IL11	PharmGKB	4/5/24	NULL	0.5625821918110125	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	NULL	Calcineurin inhibitors	NULL	NULL	NULL	NULL	NULL
SLFN11	hgnc:26633	SLFN11	PharmGKB	4/5/24	NULL	NULL	topoisomerase I inhibitors	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	U-74389G MALEATE	chembl:CHEMBL1256186	CHEMBL:CHEMBL1256186	FALSE	FALSE	FALSE
CDKAL1	hgnc:21050	CDKAL1	PharmGKB	4/5/24	NULL	NULL	Dipeptidyl peptidase 4 (DPP-4) inhibitors	NULL	NULL	NULL	NULL	NULL
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	NULL	highly active antiretroviral therapy (haart)	NULL	NULL	NULL	NULL	NULL
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	NULL	highly active antiretroviral therapy (haart)	NULL	NULL	NULL	NULL	NULL
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	NULL	highly active antiretroviral therapy (haart)	NULL	NULL	NULL	NULL	NULL
SCNN1B	hgnc:10600	SCNN1B	PharmGKB	4/5/24	NULL	NULL	insulin recombinant	NULL	NULL	NULL	NULL	NULL
RARG	hgnc:9866	RARG	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	1.250182648468916	DESMOSTEROL	iuphar.ligand:2748	DESMOSTEROL	FALSE	FALSE	FALSE
PML	hgnc:9113	PML	PharmGKB	4/5/24	NULL	0.384671584	tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.030386384	CYCLOBENZAPRINE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	PharmGKB	4/5/24	NULL	0.082754407	talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
ADAMTS1	hgnc:217	ADAMTS1	PharmGKB	4/5/24	NULL	3.889457128569963	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
SLC7A5	hgnc:11063	SLC7A5	PharmGKB	4/5/24	NULL	1.312691780892362	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.1077080435603989	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	PharmGKB	4/5/24	NULL	0.065634589	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
SPP1	hgnc:11255	SPP1	PharmGKB	4/5/24	NULL	0.6364566210387212	pamidronate	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
ADAM33	hgnc:15478	ADAM33	PharmGKB	4/5/24	NULL	NULL	selective beta-2-adrenoreceptor agonists	NULL	NULL	NULL	NULL	NULL
ABCB4	hgnc:45	ABCB4	PharmGKB	4/5/24	NULL	0.2800409132570373	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.015475294	thioridazine	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.021697385	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.1108075556053025	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CES2	hgnc:1864	CES2	PharmGKB	4/5/24	NULL	1.193356164447602	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	NULL	Opioid anesthetics	NULL	NULL	NULL	NULL	NULL
FOLH1	hgnc:3788	FOLH1	PharmGKB	4/5/24	NULL	0.086432381	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CXCL8	hgnc:6025	CXCL8	PharmGKB	4/5/24	NULL	0.010894838	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
MUTYH	hgnc:7527	MUTYH	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2A13	hgnc:2608	CYP2A13	PharmGKB	4/5/24	NULL	NULL	nnk	NULL	NULL	NULL	NULL	NULL
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.044198376	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
SLC10A1	hgnc:10905	SLC10A1	PharmGKB	4/5/24	NULL	0.6482428547616604	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	PharmGKB	4/5/24	NULL	0.2419708351875322	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1312691780892362	tolbutamide	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
C3	hgnc:1318	C3	PharmGKB	4/5/24	NULL	0.120292489	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	10-HYDROXYEVODIAMINE	chembl:CHEMBL2171812	CHEMBL:CHEMBL2171812	FALSE	FALSE	FALSE
UGT2B10	hgnc:12544	UGT2B10	PharmGKB	4/5/24	NULL	0.3608774655374192	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.017748072	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
HLA-DRB5	hgnc:4953	HLA-DRB5	PharmGKB	4/5/24	NULL	0.2165264793224515	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	PharmGKB	4/5/24	NULL	0.013879903	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP2C18	hgnc:2620	CYP2C18	PharmGKB	4/5/24	NULL	0.1804387327687096	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.041639708	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.040598715	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	NULL	ledipasvir / sofosbuvir	NULL	NULL	NULL	NULL	NULL
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	NULL	ledipasvir / sofosbuvir	NULL	NULL	NULL	NULL	NULL
XRCC1	hgnc:12828	XRCC1	PharmGKB	4/5/24	NULL	0.2386712328895204	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	1.944728564284981	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
SLC22A2	hgnc:10966	SLC22A2	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
HAS3	hgnc:4820	HAS3	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	NULL	vitamin d and analogues	NULL	NULL	NULL	NULL	NULL
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.008180039	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
GNL3	hgnc:29931	GNL3	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.040112812	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.014466916	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PROC	hgnc:9451	PROC	PharmGKB	4/5/24	NULL	1.500219178162699	avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
CXCL12	hgnc:10672	CXCL12	PharmGKB	4/5/24	NULL	4.375639269641208	alemtuzumab	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
CBR3	hgnc:1549	CBR3	PharmGKB	4/5/24	NULL	0.098053541	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.2258394461750301	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
ALDH3A1	hgnc:405	ALDH3A1	PharmGKB	4/5/24	NULL	0.025213768	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
FOXO1	hgnc:3819	FOXO1	PharmGKB	4/5/24	NULL	0.1764963739014941	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.021484317	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.6731752722524935	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
SELE	hgnc:10718	SELE	PharmGKB	4/5/24	NULL	0.080225625	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.1141471113819445	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	PharmGKB	4/5/24	NULL	0.2763561643983921	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	CLORGYLINE HYDROCHLORIDE	chembl:CHEMBL539507	CLORGYLINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.073540156	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	PharmGKB	4/5/24	NULL	NULL	XELOX	NULL	NULL	NULL	NULL	NULL
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	NULL	Arsenic compounds	NULL	NULL	NULL	NULL	NULL
CBS	hgnc:1550	CBS	PharmGKB	4/5/24	NULL	NULL	Arsenic compounds	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	insulin recombinant	NULL	NULL	NULL	NULL	NULL
HTR3A	hgnc:5297	HTR3A	DTC	9/2/20	NULL	0.1111273465305703	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	oxymetazoline and tetracaine	NULL	NULL	NULL	NULL	NULL
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	NULL	anthracyclines and related substances	NULL	NULL	NULL	NULL	NULL
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	NULL	XELOX	NULL	NULL	NULL	NULL	NULL
LTA4H	hgnc:6710	LTA4H	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
HLA-DRB5	hgnc:4953	HLA-DRB5	PharmGKB	4/5/24	NULL	2.333674277141978	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.3281729452230906	desvenlafaxine	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
APOA5	hgnc:17288	APOA5	PharmGKB	4/5/24	NULL	NULL	Antivirals for treatment of HIV infections, combinations	NULL	NULL	NULL	NULL	NULL
TLR3	hgnc:11849	TLR3	PharmGKB	4/5/24	NULL	0.074478966	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.4102161815288633	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.003869394	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	PharmGKB	4/5/24	NULL	NULL	antiinflammatory and antirheumatic products, non-steroids	NULL	NULL	NULL	NULL	NULL
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.2876257097512176	enflurane	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	PharmGKB	4/5/24	NULL	0.1178056726441863	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	NULL	S-EDDP	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	NULL	atazanavir / ritonavir	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	NULL	3,4-dehydrocilostazol	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.01495945	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.1750255707856483	thiotepa	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
DYNC2H1	hgnc:2962	DYNC2H1	PharmGKB	4/5/24	NULL	1.779921058837101	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	NULL	Leukotriene receptor antagonists	NULL	NULL	NULL	NULL	NULL
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	NULL	3,5-dimethyl-2-(3-pyridyl)thiazolidin-4-one	NULL	NULL	NULL	NULL	NULL
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	NULL	3-hydroxycotinine	NULL	NULL	NULL	NULL	NULL
IKBKG	hgnc:5961	IKBKG	PharmGKB	4/5/24	NULL	4.375639269641208	sulfadoxine	rxcui:10173	SULFADOXINE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.5000730593875667	blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
HCG22	hgnc:27780	HCG22	PharmGKB	4/5/24	NULL	4.565884455277782	triamcinolone	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.2917092846427472	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.093931433	TSU-68	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.1096651446025365	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.2910624791335615	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.081597003	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.2016939996249468	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.08334551	BMS777607	iuphar.ligand:7953	BMS-777607	FALSE	FALSE	TRUE
NAIP	hgnc:7634	NAIP	TALC	12-May-16	inhibitor	NULL	GDC0917	NULL	NULL	NULL	NULL	NULL
NTRK1	hgnc:8031	NTRK1	TALC	12-May-16	inhibitor	NULL	AZD 6918	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PYRAZOPHOS	chembl:CHEMBL1537719	PYRAZOPHOS	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.151464436	TSU-68	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
PARP1	hgnc:270	PARP1	TALC	12-May-16	inhibitor	2.100306849	AG014699	ncit:C78186	RUCAPARIB PHOSPHATE	FALSE	FALSE	TRUE
PARP1	hgnc:270	PARP1	TALC	12-May-16	inhibitor	0.900131507	MK4827	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.026748686	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.2357246744587856	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
PSMC2	hgnc:9548	PSMC2	TALC	12-May-16	inhibitor	0.5087952639117684	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	TALC	12-May-16	inhibitor	4.375639269641208	IPI-926	ncit:C80063	PATIDEGIB	FALSE	FALSE	TRUE
SIRT7	hgnc:14935	SIRT7	TALC	12-May-16	inhibitor	1.591141552596803	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
XIAP	hgnc:592	XIAP	TALC	12-May-16	inhibitor	NULL	GDC0917	NULL	NULL	NULL	NULL	NULL
BIRC2	hgnc:590	BIRC2	TALC	12-May-16	inhibitor	NULL	GDC0917	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
BIRC3	hgnc:591	BIRC3	TALC	12-May-16	inhibitor	NULL	GDC0917	NULL	NULL	NULL	NULL	NULL
BIRC6	hgnc:13516	BIRC6	TALC	12-May-16	inhibitor	NULL	GDC0917	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	NULL	MM151	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	1.184383561707394	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.012347483	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.1984416902331613	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
UNIPROT:P06746	hgnc:9174	POLB	TdgClinicalTrial	Jan-14	NULL	NULL	MBO7133 (CYTARABINE PRODRUG)	NULL	NULL	NULL	NULL	NULL
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.008460791	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
UNIPROT:Q03431	hgnc:9608	PTH1R	TdgClinicalTrial	Jan-14	NULL	NULL	768974	NULL	NULL	NULL	NULL	NULL
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.054020238	4SC-202	drugbank:DB13101	4SC-202	FALSE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	NULL	NAVITOCLAX, ABT-263	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q07817	hgnc:992	BCL2L1	TdgClinicalTrial	Jan-14	NULL	NULL	NAVITOCLAX, ABT-263	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q92843	hgnc:42959	BCL2L2-PABPN1	TdgClinicalTrial	Jan-14	NULL	NULL	NAVITOCLAX, ABT-263	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21860	hgnc:3431	ERBB3	TdgClinicalTrial	Jan-14	NULL	0.2573905452730122	AC480	ncit:C48380	PAN-HER KINASE INHIBITOR AC480	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	NULL	ACP-104	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	NULL	ACP-104	NULL	NULL	NULL	NULL	NULL
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.024309107	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	NULL	ACP-104	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	NULL	ACP-104	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	NULL	ACTB1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	NULL	ACTB1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	NULL	ACTB1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:P22455	hgnc:3691	FGFR4	TdgClinicalTrial	Jan-14	NULL	NULL	ACTB1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23443	hgnc:10436	RPS6KB1	TdgClinicalTrial	Jan-14	NULL	NULL	ACTB1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:P29459	hgnc:5969	IL12A	TdgClinicalTrial	Jan-14	NULL	NULL	AD-RTS-IL-12	NULL	NULL	NULL	NULL	NULL
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	NULL	AD-RTS-IL-12	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14432	hgnc:8778	PDE3A	TdgClinicalTrial	Jan-14	NULL	0.2651902587661338	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P24394	hgnc:6015	IL4R	TdgClinicalTrial	Jan-14	NULL	NULL	AER001,AEROVANT	NULL	NULL	NULL	NULL	NULL
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.089756703	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
UNIPROT:P78552	hgnc:5974	IL13RA1	TdgClinicalTrial	Jan-14	NULL	NULL	AER001,AEROVANT	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14627	hgnc:5975	IL13RA2	TdgClinicalTrial	Jan-14	NULL	NULL	AER001,AEROVANT	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	NULL	AEZS-112, ZEN-012	NULL	NULL	NULL	NULL	NULL
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	NULL	AEZS-112, ZEN-012	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	NULL	AEZS-112, ZEN-012	NULL	NULL	NULL	NULL	NULL
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.01678634	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	NULL	AIKO-150	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.1017590527823536	AGN-214868	chembl:CHEMBL3137348	SENREBOTASE	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.1562728310586145	AGN-214868	chembl:CHEMBL3137348	SENREBOTASE	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1704794520639432	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.6908904109959803	ZALEPLON	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
UNIPROT:P60880	hgnc:11132	SNAP25	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	BOTULINUM TOXIN TYPE A	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
UNIPROT:P30872	hgnc:11330	SSTR1	TdgClinicalTrial	Jan-14	NULL	1.215455352678113	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.2476776945079929	CHIDAMIDE	hemonc:99	CHIDAMIDE	FALSE	FALSE	FALSE
UNIPROT:Q15274	hgnc:9755	QPRT	TdgClinicalTrial	Jan-14	NULL	3.750547945406749	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
UNIPROT:P78552	hgnc:5974	IL13RA1	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	CINTREDEKIN BESUDOTOX	ncit:C2599	CINTREDEKIN BESUDOTOX	FALSE	FALSE	FALSE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.31919557	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	2.692701089009974	1-PHENETHYLPIPERIDINE	chembl:CHEMBL75228	1-PHENETHYLPIPERIDINE	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	2.258394462	CNTO 148	rxcui:819300	GOLIMUMAB	TRUE	TRUE	FALSE
UNIPROT:P08138	hgnc:7809	NGFR	TdgClinicalTrial	Jan-14	NULL	NULL	CXB909	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04629	hgnc:8031	NTRK1	TdgClinicalTrial	Jan-14	NULL	NULL	CXB909	NULL	NULL	NULL	NULL	NULL
UNIPROT:CYSTINE	NULL	NULL	TdgClinicalTrial	Jan-14	NULL	NULL	CYSTEAMINE	rxcui:1426886	CYSTEAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9UBU3	hgnc:18129	GHRL	TdgClinicalTrial	Jan-14	NULL	NULL	CYT-009-GHRQB	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01584	hgnc:5992	IL1B	TdgClinicalTrial	Jan-14	NULL	NULL	CYT013-IL1BQB	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	DAC:GLP-1	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q02643	hgnc:4266	GHRHR	TdgClinicalTrial	Jan-14	NULL	NULL	DAC:GRF	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.014299475	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
UNIPROT:P31785	hgnc:6010	IL2RG	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	CYT-107	ncit:C77879	GLYCOSYLATED RECOMBINANT HUMAN INTERLEUKIN-7	FALSE	FALSE	FALSE
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	NULL	DEBIO-9902 SR	NULL	NULL	NULL	NULL	NULL
UNIPROT:P06239	hgnc:6524	LCK	TdgClinicalTrial	Jan-14	NULL	0.05348375	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.073403082	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.059690418	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	NULL	DOV 102,677	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	NULL	DOV 102,677	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	NULL	DOV 102,677	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.080164384	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
UNIPROT:P20711	hgnc:2719	DDC	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.482607272	DONEPEZIL	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005953251	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	NULL	E75	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	GLP	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.2628669398532891	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
UNIPROT:Q08289	hgnc:1402	CACNB2	TdgClinicalTrial	Jan-14	NULL	0.1930429089547592	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	NULL	EV-077-3201-2TBS	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	0.060388351	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.064111931	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.067839369	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005208578	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
UNIPROT:P16109	hgnc:10721	SELP	TdgClinicalTrial	Jan-14	NULL	8.751278539282417	GMI-1070	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
UNIPROT:P16581	hgnc:10718	SELE	TdgClinicalTrial	Jan-14	NULL	6.364566210387211	GMI-1070	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.057700738	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
UNIPROT:Q8WXA8	hgnc:24003	HTR3C	TdgClinicalTrial	Jan-14	NULL	0.3409589041278864	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	NULL	GTF505	NULL	NULL	NULL	NULL	NULL
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW827102X	chembl:CHEMBL362155	GW827102X	FALSE	FALSE	FALSE
UNIPROT:Q03181	hgnc:9235	PPARD	TdgClinicalTrial	Jan-14	NULL	NULL	GTF505	NULL	NULL	NULL	NULL	NULL
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	NULL	GTF505	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	NULL	PX 104.1	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q03181	hgnc:9235	PPARD	TdgClinicalTrial	Jan-14	NULL	0.4934931507114145	GW501516	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.001998465	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	GSK-1004723	drugbank:DB12806	GSK-1004723	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.315046027	GW501516	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
UNIPROT:O60760	hgnc:17890	HPGDS	TdgClinicalTrial	Jan-14	NULL	NULL	HF0220	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	NULL	AMG 0001	NULL	NULL	NULL	NULL	NULL
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.1715936968486748	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
UNIPROT:Q16665	hgnc:4910	HIF1A	TdgClinicalTrial	Jan-14	NULL	NULL	HIF-1ALPHA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P19835	hgnc:1848	CEL	TdgClinicalTrial	Jan-14	NULL	NULL	BILE SALT STIMULATED LIPASE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	0.7343730242754476	ISOSORBIDE DINITRATE	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	NULL	IDRABIOTAPARINUX	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.1108075556053025	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P04629	hgnc:8031	NTRK1	TdgClinicalTrial	Jan-14	NULL	0.019180884	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	TICLOPIDINE	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TdgClinicalTrial	Jan-14	NULL	NULL	INS-20	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.1252170220247087	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:Q9NZ20	hgnc:17934	PLA2G3	TdgClinicalTrial	Jan-14	NULL	NULL	MRX-6	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	LIRANAFTATE	ncit:C66019	LIRANAFTATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	TCMDC-124571	chembl:CHEMBL533542	CHEMBL:CHEMBL533542	FALSE	FALSE	FALSE
UNIPROT:P41231	hgnc:8541	P2RY2	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	INS37217	ncit:C78118	DENUFOSOL	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.1816874437221263	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P15260	hgnc:5439	IFNGR1	TdgClinicalTrial	Jan-14	NULL	NULL	IFN-GAMMA	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	TCMDC-125286	chembl:CHEMBL533965	CHEMBL:CHEMBL533965	FALSE	FALSE	FALSE
UNIPROT:P38484	hgnc:5440	IFNGR2	TdgClinicalTrial	Jan-14	NULL	NULL	IFN-GAMMA	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004636439	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
UNIPROT:P25942	hgnc:11919	CD40	TdgClinicalTrial	Jan-14	NULL	NULL	ISF35	NULL	NULL	NULL	NULL	NULL
CHUK	hgnc:1974	CHUK	DTC	9/2/20	NULL	3.750547945	PEPEROMIN E	chembl:CHEMBL521941	PEPEROMIN E	FALSE	FALSE	FALSE
UNIPROT:P02741	hgnc:2367	CRP	TdgClinicalTrial	Jan-14	NULL	NULL	ISIS 353512	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
UNIPROT:P16410	hgnc:2505	CTLA4	TdgClinicalTrial	Jan-14	NULL	0.7001022831425934	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
UNIPROT:P02741	hgnc:2367	CRP	TdgClinicalTrial	Jan-14	NULL	NULL	ISIS-CRPRX	NULL	NULL	NULL	NULL	NULL
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV006861	chembl:CHEMBL582666	CHEMBL:CHEMBL582666	FALSE	FALSE	FALSE
UNIPROT:P03951	hgnc:3529	F11	TdgClinicalTrial	Jan-14	NULL	NULL	ISIS-FXIRX	NULL	NULL	NULL	NULL	NULL
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	RO-256981	chembl:CHEMBL1256726	CHEMBL:CHEMBL1256726	FALSE	FALSE	FALSE
UNIPROT:P31639	hgnc:11037	SLC5A2	TdgClinicalTrial	Jan-14	NULL	NULL	ISIS-SGLT2RX	NULL	NULL	NULL	NULL	NULL
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.073266518	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.4953553890159858	(+)-CATECHIN HYDRATE	chembl:CHEMBL1256783	CHEMBL:CHEMBL1256783	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.069240885	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.076840494	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	NULL	KN38-7271	NULL	NULL	NULL	NULL	NULL
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.060772768	DOXAZOSIN MESYLATE	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1750255707856483	TCMDC-125813	chembl:CHEMBL580076	CHEMBL:CHEMBL580076	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
PRKG1	hgnc:9414	PRKG1	DTC	9/2/20	NULL	0.1223955040459079	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
UNIPROT:P34972	hgnc:2160	CNR2	TdgClinicalTrial	Jan-14	NULL	NULL	KN38-7271	NULL	NULL	NULL	NULL	NULL
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.059667808	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:O43193	hgnc:4495	MLNR	TdgClinicalTrial	Jan-14	NULL	NULL	KOS-2187	NULL	NULL	NULL	NULL	NULL
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	KC706	drugbank:DB05157	KC706	FALSE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.1426838892274307	KC706	drugbank:DB05157	KC706	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	3,5-DIPHENYLISOXAZOLE	chembl:CHEMBL1374535	3,5-DIPHENYLISOXAZOLE	FALSE	FALSE	FALSE
UNIPROT:Q05655	hgnc:9399	PRKCD	TdgClinicalTrial	Jan-14	NULL	4.922594178346359	KAI-9803	ncit:C101384	DELCASERTIB	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.073266518	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	NULL	LU AE04621	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	NULL	LU AE04621	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	NULL	LU AE04621	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	NULL	LU AE04621	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	NULL	LU AE04621	NULL	NULL	NULL	NULL	NULL
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.045226246	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	LU-AE58054	ncit:C166835	IDALOPIRDINE	FALSE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.028009071	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.011219588	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.025739055	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	0.026572708	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	0.046059361	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.024241769	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.008033609	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:Q14626	hgnc:5967	IL11RA	TdgClinicalTrial	Jan-14	NULL	10.50153425	OPRELVEKIN	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.034544521	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.233887177	ENOBOSARM	rxcui:2168587	ENOBOSARM	FALSE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	1.117184494376478	ONX 0801	ncit:C120550	IDETREXED	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	7.001022831425932	PRX-07034	drugbank:DB05993	PRX-07034	FALSE	FALSE	FALSE
UNIPROT:Q9H015	hgnc:10968	SLC22A4	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
UNIPROT:P42336	hgnc:8975	PIK3CA	TdgClinicalTrial	Jan-14	NULL	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.1458546423213736	HYDROCODONE	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.053038052	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1505380482674727	HYDROCODONE	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	PTC299	drugbank:DB05173	PTC299	FALSE	FALSE	FALSE
UNIPROT:P12319	hgnc:3609	FCER1A	TdgClinicalTrial	Jan-14	NULL	NULL	R112	NULL	NULL	NULL	NULL	NULL
UNIPROT:P30273	hgnc:3611	FCER1G	TdgClinicalTrial	Jan-14	NULL	NULL	R112	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	GNF-PF-4832	chembl:CHEMBL601137	CHEMBL:CHEMBL601137	FALSE	FALSE	FALSE
UNIPROT:Q01362	hgnc:7316	MS4A2	TdgClinicalTrial	Jan-14	NULL	NULL	R112	NULL	NULL	NULL	NULL	NULL
UNIPROT:P52333	hgnc:6193	JAK3	TdgClinicalTrial	Jan-14	NULL	NULL	R348	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	SDZ-205557	iuphar.ligand:258	SDZ 205557	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	R667	iuphar.ligand:8276	PALOVAROTENE	FALSE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	R667	iuphar.ligand:8276	PALOVAROTENE	FALSE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	R667	iuphar.ligand:8276	PALOVAROTENE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	CITRONELLYL ACETATE	rxcui:2056062	CITRONELLYL ACETATE	TRUE	FALSE	FALSE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.9460841664089098	REGADENOSON	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.041021618	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:Q9NR82	hgnc:6299	KCNQ5	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	RETIGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
UNIPROT:P33681	hgnc:1700	CD80	TdgClinicalTrial	Jan-14	NULL	NULL	AV1142742	NULL	NULL	NULL	NULL	NULL
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.2864054794674245	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.305277158	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	ARISTOLOCHIC ACID	iuphar.ligand:12438	ARISTOLOCHIC ACID	FALSE	FALSE	FALSE
UNIPROT:O00329	hgnc:8977	PIK3CD	TdgClinicalTrial	Jan-14	NULL	0.092606122	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
UNIPROT:P48736	hgnc:8978	PIK3CG	TdgClinicalTrial	Jan-14	NULL	0.067317527	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
UNIPROT:Q8NEB9	hgnc:8974	PIK3C3	TdgClinicalTrial	Jan-14	NULL	0.364636606	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.049723174	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.03849536	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1988926940746003	SIBUTRAMINE	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
UNIPROT:P28908	hgnc:11923	TNFRSF8	TdgClinicalTrial	Jan-14	NULL	1.276228120312019	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.041182487	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
UNIPROT:P50613	hgnc:1778	CDK7	TdgClinicalTrial	Jan-14	NULL	2.100306849	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	NULL	SPC-2996	NULL	NULL	NULL	NULL	NULL
UNIPROT:P78363	hgnc:34	ABCA4	TdgClinicalTrial	Jan-14	NULL	NULL	STARGEN	NULL	NULL	NULL	NULL	NULL
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.025147352	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	NULL	TC-2403-12	NULL	NULL	NULL	NULL	NULL
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	NULL	TC-2403-12	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	2.333674277141977	TARANABANT	ncit:C81420	TARANABANT	FALSE	FALSE	FALSE
UNIPROT:P01857	hgnc:5525	IGHG1	TdgClinicalTrial	Jan-14	NULL	NULL	IGG1 ANTIBODY	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-125495	chembl:CHEMBL532412	CHEMBL:CHEMBL532412	FALSE	FALSE	FALSE
UNIPROT:O00519	hgnc:3553	FAAH	TdgClinicalTrial	Jan-14	NULL	NULL	V158866	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.3409589041278863	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	1.400204566285186	RECOMBINANT HUMAN GROWTH HORMONE	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1215455352678113	TERAZOSIN HYDROCHLORIDE	rxcui:235224	TERAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.364636606	ALPHA-TERTHIENYL	chembl:CHEMBL90017	ALPHA-TERTHIENYL	FALSE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	HISTRELIN	rxcui:1294622	HISTRELIN ACETATE	TRUE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.1630673019742065	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	0.8751278539282416	NRP104	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.3163112725041837	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.04907259	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	NS-2028	iuphar.ligand:6554	NS 2028	FALSE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.1232574442152452	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.062509132	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.062509132	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TdgClinicalTrial	Jan-14	NULL	NULL	R-BACLOFEN	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	METHYLBENZETHONIUM CHLORIDE	rxcui:1796444	METHYLBENZETHONIUM CHLORIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005677733	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O75899	hgnc:4507	GABBR2	TdgClinicalTrial	Jan-14	NULL	NULL	R-BACLOFEN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P30872	hgnc:11330	SSTR1	TdgClinicalTrial	Jan-14	NULL	NULL	YTTRIUM-90 EDOTREOTIDE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P30874	hgnc:11331	SSTR2	TdgClinicalTrial	Jan-14	NULL	NULL	YTTRIUM-90 EDOTREOTIDE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35346	hgnc:11334	SSTR5	TdgClinicalTrial	Jan-14	NULL	NULL	YTTRIUM-90 EDOTREOTIDE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P02766	hgnc:12405	TTR	TdgClinicalTrial	Jan-14	NULL	NULL	ALN-TTR	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.048859496	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	ACEBUTOLOL	rxcui:149	ACEBUTOLOL	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.182318303	ACETOPHENAZINE	rxcui:16735	ACETOPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TdgClinicalTrial	Jan-14	NULL	0.4327555321623173	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.078958904	TRIBUTYLTIN-OXIDE	chembl:CHEMBL511667	TRIBUTYLTIN-OXIDE	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	ATRACURIUM	rxcui:1218	ATRACURIUM	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	BENZPHETAMINE	rxcui:1422	BENZPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.4605936073306534	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.5321723436050118	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1221108633388244	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.025757994	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.8140724222588294	CLENBUTEROL	rxcui:2580	CLENBUTEROL	TRUE	FALSE	FALSE
UNIPROT:P41180	hgnc:1514	CASR	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	CINACALCET	rxcui:407990	CINACALCET	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	TDR77578	chembl:CHEMBL1364172	CHEMBL:CHEMBL1364172	FALSE	FALSE	FALSE
UNIPROT:Q14432	hgnc:8778	PDE3A	TdgClinicalTrial	Jan-14	NULL	0.6819178082557726	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	CHORIOGONADOTROPIN ALFA	rxcui:283550	CHORIOGONADOTROPIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	DEXBROMPHENIRAMINE	rxcui:1767	BROMPHENIRAMINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1595977849109255	DIPHENIDOL	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.2631963470460877	DIPHENIDOL	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	NODAKENIN	chembl:CHEMBL459825	NODAKENIN	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1185944014357865	DOMPERIDONE	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.03729238	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.4526523382387456	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.1682938180631233	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.031929262	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.1014640990061729	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TEND	1-Aug-11	NULL	0.023716202	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	8-FLUOROTRYPTANTHRIN	chembl:CHEMBL1098875	CHEMBL:CHEMBL1098875	FALSE	FALSE	FALSE
UNIPROT:P16444	hgnc:3002	DPEP1	TEND	1-Aug-11	NULL	17.50255707856483	CILASTATIN	rxcui:2540	CILASTATIN	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.2302968036653267	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TEND	1-Aug-11	NULL	0.6177373086552295	DARBEPOETIN ALFA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	BROMPHENIRAMINE	rxcui:1767	BROMPHENIRAMINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	HARMAN	chembl:CHEMBL12014	HARMAN	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1595977849109255	CEVIMELINE	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.251232877	GS 6201	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.9546849315580818	CARPROFEN	rxcui:20343	CARPROFEN	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.079197091	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	0.7501095890813498	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.080225625	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.058341857	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.040703621	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.059667808	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.041508041	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:Q05586	hgnc:4584	GRIN1	TEND	1-Aug-11	NULL	0.4286340509036286	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1848861663228679	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	NALIDIXIC ACID	rxcui:7240	NALIDIXIC ACID	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TEND	1-Aug-11	NULL	0.112919723	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TEND	1-Aug-11	NULL	0.192335792	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TEND	1-Aug-11	NULL	0.1682938180631233	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TEND	1-Aug-11	NULL	0.2500365296937833	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
EIF4A1	hgnc:3282	EIF4A1	DTC	9/2/20	NULL	2.019525817	SILVESTROL	chembl:CHEMBL555196	SILVESTROL	FALSE	FALSE	FALSE
UNIPROT:Q14626	hgnc:5967	IL11RA	TEND	1-Aug-11	NULL	10.50153425	OPRELVEKIN	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.7143900848393808	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TEND	1-Aug-11	NULL	0.033243223	DRONEDARONE	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	1.750255707856483	GLICLAZIDE	rxcui:4816	GLICLAZIDE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.046881849	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1111665587205952	HYDROMORPHONE	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.039531467	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TEND	1-Aug-11	NULL	0.060388351	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.3211478363039418	LEVORPHANOL	rxcui:6378	LEVORPHANOL	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.02232469	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TEND	1-Aug-11	NULL	0.2112984757975633	LOFEXIDINE	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1479089330582944	MEPERIDINE	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.003805731	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
UNIPROT:P22888	hgnc:6585	LHCGR	TEND	1-Aug-11	NULL	16.40864726115453	LUTROPIN ALFA	rxcui:388084	LUTROPIN ALFA	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007596596	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
UNIPROT:P07202	hgnc:12015	TPO	TEND	1-Aug-11	NULL	2.500365296937833	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.546954909	MEPHENTERMINE	rxcui:6756	MEPHENTERMINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1396480617970598	METHYLSCOPOLAMINE	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1017590527823536	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.011306561	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
UNIPROT:P00519	hgnc:76	ABL1	TEND	1-Aug-11	NULL	0.637458239	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.061737415	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TEND	1-Aug-11	NULL	0.089298761	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.108711535	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.055563673	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.064944553	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.1591141552596803	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
UNIPROT:P19793	hgnc:10477	RXRA	TEND	1-Aug-11	NULL	0.1166837138570988	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1376347869874036	PENTAZOCINE	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
UNIPROT:P21453	hgnc:3165	S1PR1	TEND	1-Aug-11	NULL	1.458546423213736	FINGOLIMOD	rxcui:1012892	FINGOLIMOD	TRUE	TRUE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.014245163	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.087512785	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	SJ000114740	chembl:CHEMBL592068	CHEMBL:CHEMBL592068	FALSE	FALSE	FALSE
UNIPROT:P48443	hgnc:10479	RXRG	TEND	1-Aug-11	NULL	0.7955707762984013	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.4070362111294147	PENBUTOLOL	rxcui:7973	PENBUTOLOL	TRUE	FALSE	FALSE
UNIPROT:P35499	hgnc:10591	SCN4A	TEND	1-Aug-11	NULL	0.201952582	FOSPROPOFOL	rxcui:828682	FOSPROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TEND	1-Aug-11	NULL	0.1022876712383659	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.05913026	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.061055432	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.2631963470460877	ROCURONIUM	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
UNIPROT:P35346	hgnc:11334	SSTR5	TEND	1-Aug-11	NULL	3.125456621172291	LANREOTIDE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.088945801	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.086551106	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.061055432	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.083257407	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1704794520639432	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.079557078	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.078682824	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TEND	1-Aug-11	NULL	0.048708415	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
UNIPROT:Q7Z2W7	hgnc:17961	TRPM8	TEND	1-Aug-11	NULL	4.836232876971861	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.2442217266776488	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TEND	1-Aug-11	NULL	1.262203635473425	TICLOPIDINE	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.100976291	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.049337723	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.7119684235348407	TRANDOLAPRIL	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TEND	1-Aug-11	NULL	0.093346971	TREPROSTINIL	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.03271506	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TEND	1-Aug-11	NULL	0.012347483	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.9460841664089098	CHRYSOERIOL	drugbank:DB17283	CHRYSOERIOL	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.061197752	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	TROSPIUM	rxcui:236778	TROSPIUM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.061992528	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1396480617970598	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	NYLIDRIN HYDROCHLORIDE	rxcui:82060	NYLIDRIN HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P23763	hgnc:12642	VAMP1	TEND	1-Aug-11	NULL	35.00511415712966	BOTULINUM TOXIN TYPE B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	1.186614039224734	VALSARTAN	rxcui:69749	VALSARTAN	TRUE	FALSE	FALSE
LEUKOCYTE COMMON ANTIGEN	hgnc:9666	PTPRC	TTD	2020.06.01	NULL	NULL	LM-CD45	NULL	NULL	NULL	NULL	NULL
ESTROGEN-RELATED RECEPTOR-ALPHA	hgnc:3471	ESRRA	TTD	2020.06.01	NULL	NULL	D-5519	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	MCP-202	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 2 RECEPTOR	hgnc:4325	GLP2R	TTD	2020.06.01	NULL	NULL	SAN-134	NULL	NULL	NULL	NULL	NULL
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	CLP-1004	NULL	NULL	NULL	NULL	NULL
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	PENT-1-ENE	chembl:CHEMBL295337	CHEMBL:CHEMBL295337	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS MATURATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK2838232	iuphar.ligand:12680	GSK2838232	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	NULL	Drug 2881078	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	NULL	MP-157	NULL	NULL	NULL	NULL	NULL
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	0.7955707762984014	ASP-1707	chembl:CHEMBL3989969	OPIGOLIX	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	AVE0897	NULL	NULL	NULL	NULL	NULL
GAP JUNCTION ALPHA-1 PROTEIN	hgnc:4274	GJA1	TTD	2020.06.01	NULL	NULL	Act1	NULL	NULL	NULL	NULL	NULL
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.1339481409073839	ABI-011	ncit:C116890	NANOPARTICLE ALBUMIN-BOUND THIOCOLCHICINE DIMER NAB-5404	FALSE	FALSE	FALSE
DNA-DIRECTED RNA POLYMERASE II	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lurbinectedin	rxcui:2374729	LURBINECTEDIN	TRUE	FALSE	FALSE
STAT3 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Napabucasin	ncit:C96429	NAPABUCASIN	FALSE	FALSE	FALSE
TNF RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ETX201	NULL	NULL	NULL	NULL	NULL
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.01712579	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
IMMUNOGLOBULIN GAMMA-1 HEAVY NIE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MORAb-022	ncit:C172615	GIMSILUMAB	FALSE	FALSE	FALSE
OSTEOBLAST CADHERIN	hgnc:1750	CDH11	TTD	2020.06.01	NULL	NULL	RG6125	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	SGM-1019	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	TYrosine kinase 2 inhibitor	NULL	NULL	NULL	NULL	NULL
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
BETA-CATENIN	hgnc:2514	CTNNB1	TTD	2020.06.01	NULL	NULL	C 82	NULL	NULL	NULL	NULL	NULL
CREB-BINDING PROTEIN	hgnc:2348	CREBBP	TTD	2020.06.01	NULL	NULL	C 82	NULL	NULL	NULL	NULL	NULL
LYSOSPHINGOLIPID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cenerimod	ncit:C169837	CENERIMOD	FALSE	FALSE	FALSE
C-X-C MOTIF CHEMOKINE 10	hgnc:10637	CXCL10	TTD	2020.06.01	NULL	NULL	JT02	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C1S COMPONENT	hgnc:1247	C1S	TTD	2020.06.01	NULL	10.50153424713889	TNT009	rxcui:2591404	SUTIMLIMAB	TRUE	FALSE	FALSE
DNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifaximin DR	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	Actimab-M	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	Duvortuxizumab	ncit:C122406	DUVORTUXIZUMAB	FALSE	FALSE	FALSE
CYTOTOXIC T-LYMPHOCYTE PROTEIN 4	hgnc:2505	CTLA4	TTD	2020.06.01	NULL	NULL	TRemelimumab + MEDI0562	NULL	NULL	NULL	NULL	NULL
OX40L RECEPTOR	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	NULL	TRemelimumab + MEDI0562	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hu3F8 mAb	NULL	NULL	NULL	NULL	NULL
ACTIVATION-INDUCIBLE TNFR FAMILY RECEPTOR	hgnc:11914	TNFRSF18	TTD	2020.06.01	NULL	NULL	INCAGN1876	NULL	NULL	NULL	NULL	NULL
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	NULL	MAGE-A10 TCR	NULL	NULL	NULL	NULL	NULL
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-3/BETA-4	NULL	NULL	TTD	2020.06.01	NULL	NULL	18-MC	chembl:CHEMBL5095410	ZOLUNICANT	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	NULL	EVT100	NULL	NULL	NULL	NULL	NULL
SEROTONINNOREPINEPHRINEDOPAMINE REUPTAKE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Centanafadine	ncit:C171666	CENTANAFADINE	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	FKB01MD	NULL	NULL	NULL	NULL	NULL
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	NULL	FKB01MD	NULL	NULL	NULL	NULL	NULL
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	PHOSMET	drugbank:DB11448	PHOSMET	FALSE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	FKB01MD	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	FKW00GA	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	FKW00GA	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
5-HT 7 RECEPTOR	hgnc:5302	HTR7	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
SEROTONINNOREPINEPHRINEDOPAMINE REUPTAKE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RP5063	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	26.25383561784724	MIN-101	chembl:CHEMBL4298043	ROLUPERIDONE HYDROCHLORIDE	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	2.000292237550266	Emibetuzumab	ncit:C95732	EMIBETUZUMAB	FALSE	TRUE	TRUE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GLYX-13	chembl:CHEMBL3544917	RAPASTINEL	FALSE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ITI-007	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	GTP-004	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	chembl:CHEMBL1322879	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	FALSE	FALSE	FALSE
BETA-N-ACETYLHEXOSAMINIDASE	hgnc:7056	OGA	TTD	2020.06.01	NULL	26.25383561784724	MK 8719	drugbank:DB16989	MK-8719	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	TRV734	NULL	NULL	NULL	NULL	NULL
PACAP TYPE I RECEPTOR	hgnc:242	ADCYAP1R1	TTD	2020.06.01	NULL	NULL	AMG 301	NULL	NULL	NULL	NULL	NULL
EARLY GROWTH RESPONSE PROTEIN 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	AYX-1	chembl:CHEMBL4297228	BRIVOLIGIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.023493365	ENDO-ATROPINE	chembl:CHEMBL2449003	ENDO-ATROPINE	FALSE	FALSE	FALSE
QUINONE REDUCTASE 1	hgnc:2874	NQO1	TTD	2020.06.01	NULL	NULL	BioE-743	NULL	NULL	NULL	NULL	NULL
OXIDOREDUCTASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	EPX-200	NULL	NULL	NULL	NULL	NULL
HELPER-INDUCER T-LYMPHOCYTE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AE-H vaccine	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005669763	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 1	hgnc:6877	MAPK3	TTD	2020.06.01	NULL	NULL	VAN-10-4-eluting stent	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR SIGNAL-REGULATED KINASE 2	hgnc:6871	MAPK1	TTD	2020.06.01	NULL	NULL	VAN-10-4-eluting stent	NULL	NULL	NULL	NULL	NULL
TUFTSIN RECEPTOR	hgnc:11727	TERC	TTD	2020.06.01	NULL	NULL	99MTC-RP-128	NULL	NULL	NULL	NULL	NULL
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	NULL	KD-7040	NULL	NULL	NULL	NULL	NULL
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.02706581	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	VM-206	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY 86-8050	NULL	NULL	NULL	NULL	NULL
OSTEOCLAST DIFFERENTIATION FACTOR	hgnc:11926	TNFSF11	TTD	2020.06.01	NULL	NULL	ALX-0141	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.002927502	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ACH-1625	NULL	NULL	NULL	NULL	NULL
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	NULL	OPA-6566	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	NULL	AEZS-123	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Targeted ranpirnase conjugates	NULL	NULL	NULL	NULL	NULL
TRANSTHYRETIN	hgnc:12405	TTR	TTD	2020.06.01	NULL	NULL	ALN-TTRsc	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
HUNTINGTIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALN-HTT	NULL	NULL	NULL	NULL	NULL
COLLAGEN I	hgnc:2198	COL1A2	TTD	2020.06.01	NULL	NULL	Solubilized type 1 native bovine collagen	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD7325	iuphar.ligand:7712	AZD7325	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	TCMDC-125617	chembl:CHEMBL545900	CHEMBL:CHEMBL545900	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.7955707762984013	Ronomilast	ncit:C97274	RONOMILAST	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	Lexibulin iv infusion	NULL	NULL	NULL	NULL	NULL
APOPTOSIS INHIBITOR SURVIVIN	hgnc:593	BIRC5	TTD	2020.06.01	NULL	NULL	CV-9201	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006397133	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
CANCER/TESTIS ANTIGEN 1	hgnc:2491	CTAG1B	TTD	2020.06.01	NULL	NULL	CV-9201	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	5-(4-PHENYLBUTOXY)PSORALEN	iuphar.ligand:9583	PSORA-4	FALSE	FALSE	FALSE
CANCER/TESTIS ANTIGEN MAGE-C1/CT7	hgnc:6812	MAGEC1	TTD	2020.06.01	NULL	NULL	CV-9201	NULL	NULL	NULL	NULL	NULL
MELANOMA-ASSOCIATED ANTIGEN C2	hgnc:13574	MAGEC2	TTD	2020.06.01	NULL	NULL	CV-9201	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
ONCOTROPHOBLAST GLYCOPROTEIN 5T4	hgnc:12004	TPBG	TTD	2020.06.01	NULL	NULL	CV-9201	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	PLX-3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	L19-IL-2 fusion protein	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR C	hgnc:12682	VEGFC	TTD	2020.06.01	NULL	5.834185692854944	VGX-100	chembl:CHEMBL4297847	VGX-100	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.3947945205691315	NSC-74859	chembl:CHEMBL477936	CHEMBL:CHEMBL477936	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	1.166837138570988	SHP-141	ncit:C97513	REMETINOSTAT	FALSE	FALSE	FALSE
NOTCH-1 RECEPTOR	hgnc:7881	NOTCH1	TTD	2020.06.01	NULL	19.69037671338543	OMP-52M51	ncit:C103274	BRONTICTUZUMAB	FALSE	FALSE	TRUE
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	ABT-RTA-408	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	IOPAMIDOL	rxcui:5966	IOPAMIDOL	TRUE	FALSE	FALSE
MYCBP MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	DCR-MYC	ncit:C115108	MYC-TARGETING SIRNA DCR-MYC	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	NULL	SRT2379	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CB-01-16	NULL	NULL	NULL	NULL	NULL
CCNB1	hgnc:1579	CCNB1	DTC	9/2/20	NULL	2.500365296937833	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
PARATHYROID HORMONE	hgnc:9606	PTH	TTD	2020.06.01	NULL	NULL	KUR-111	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	MAL formulation	NULL	NULL	NULL	NULL	NULL
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	5.250767123569449	CVX-060	chembl:CHEMBL4594470	CVX-060	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
SUPPRESSOR OF TUMORIGENICITY 14 PROTEIN	hgnc:11344	ST14	TTD	2020.06.01	NULL	NULL	US8569313, Inhibitor 15	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US8586571, 6	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
ACETYL-COA TRANSPORTER	hgnc:95	SLC33A1	TTD	2020.06.01	NULL	NULL	US8592431, 185	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8592455, 3	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	T8361	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	EEC	NULL	NULL	NULL	NULL	NULL
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	TOTAROL	rxcui:1600439	TOTAROL	TRUE	FALSE	FALSE
GALECTIN-1	hgnc:6561	LGALS1	TTD	2020.06.01	NULL	NULL	US8703720, Reference Compound 2	NULL	NULL	NULL	NULL	NULL
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.039420174	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
CARBOXYPEPTIDASE B1	hgnc:2299	CPB1	TTD	2020.06.01	NULL	NULL	US8710232, 7	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8759338, 2	NULL	NULL	NULL	NULL	NULL
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	NG7	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
ADAM METALLOPEPTIDASE 33	hgnc:15478	ADAM33	TTD	2020.06.01	NULL	NULL	US8772478, 1	NULL	NULL	NULL	NULL	NULL
ADAM METALLOPEPTIDASE 33	hgnc:15478	ADAM33	TTD	2020.06.01	NULL	NULL	US8772478, 5	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8536181, C17	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	LEVDOBUTAMINE	ncit:C166431	LEVDOBUTAMINE	FALSE	FALSE	FALSE
BACTERIAL NICOTINATE-NUCLEOTIDE ADENYLYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	STK696827	NULL	NULL	NULL	NULL	NULL
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.006978691	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CASEIN KINASE II ALPHA PRIME	hgnc:2459	CSNK2A2	TTD	2020.06.01	NULL	NULL	US8791257, 38	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8829193, 1	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8829193, 2	NULL	NULL	NULL	NULL	NULL
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.006722273	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PRKACA MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	VFEDEOUBYBLDKN-AAFJCEBUSA-N	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US8853215, 3	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US8877733, 28	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C ZETA	hgnc:9412	PRKCZ	TTD	2020.06.01	NULL	NULL	US8889696, 39	NULL	NULL	NULL	NULL	NULL
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.1704794520639432	GS 6201	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
ROTAMASE D	hgnc:9257	PPID	TTD	2020.06.01	NULL	NULL	1313212-89-3	NULL	NULL	NULL	NULL	NULL
ROTAMASE D	hgnc:9257	PPID	TTD	2020.06.01	NULL	NULL	US8901295, F609	NULL	NULL	NULL	NULL	NULL
KYNURENINE OXOGLUTARATE TRANSAMINASE II	hgnc:17929	AADAT	TTD	2020.06.01	NULL	NULL	US8933095, 1	NULL	NULL	NULL	NULL	NULL
BCL-2-RELATED PROTEIN A1	hgnc:991	BCL2A1	TTD	2020.06.01	NULL	NULL	Apogossypolone	NULL	NULL	NULL	NULL	NULL
CASEIN KINASE II ALPHA PRIME	hgnc:2459	CSNK2A2	TTD	2020.06.01	NULL	NULL	US8940736, 6	NULL	NULL	NULL	NULL	NULL
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.2273059360852575	RAMATROBAN	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9409892, 59	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9434725, 113	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	US8614253, 29-19	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	US8614253, 32-4	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	US9241942, 32-12	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8669361, 102	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9586942, 16	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	4-PHENOXYPHENOL	chembl:CHEMBL224318	CHEMBL:CHEMBL224318	FALSE	FALSE	FALSE
MEK KINASE KINASE 4	hgnc:6866	MAP4K4	TTD	2020.06.01	NULL	NULL	6-Phenylquinazolin-4-amine	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8598210, Table XV, 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4C	hgnc:8782	PDE4C	TTD	2020.06.01	NULL	NULL	US10077269, Example 6	NULL	NULL	NULL	NULL	NULL
ABCB11	hgnc:42	ABCB11	DTC	9/2/20	NULL	2.386712328895204	GS-9256	drugbank:DB12876	GS-9256	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4C	hgnc:8782	PDE4C	TTD	2020.06.01	NULL	NULL	ZINC584606052	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US9073936, 3	NULL	NULL	NULL	NULL	NULL
RAR-RELATED ORPHAN RECEPTOR-BETA	hgnc:10259	RORB	TTD	2020.06.01	NULL	NULL	US9598431, 1	NULL	NULL	NULL	NULL	NULL
RAR-RELATED ORPHAN RECEPTOR-BETA	hgnc:10259	RORB	TTD	2020.06.01	NULL	NULL	US9598431, 2	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.005284588	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NUCLEAR RECEPTOR ROR-ALPHA	hgnc:10258	RORA	TTD	2020.06.01	NULL	NULL	US9598431, 3	NULL	NULL	NULL	NULL	NULL
RAR-RELATED ORPHAN RECEPTOR-BETA	hgnc:10259	RORB	TTD	2020.06.01	NULL	NULL	US9598431, 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US9714230, 46	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	BDBM50080559	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9617250, Example 1 Example 204 of D1	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001193302	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CALMODULIN-DEPENDENT KINASE II	hgnc:1470	CAMKK2	TTD	2020.06.01	NULL	NULL	CQ7	NULL	NULL	NULL	NULL	NULL
CALMODULIN-DEPENDENT KINASE II	hgnc:1470	CAMKK2	TTD	2020.06.01	NULL	NULL	US9623028, Compound 79	NULL	NULL	NULL	NULL	NULL
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.5147810905460245	LEUKOTRIENE D4	drugbank:DB11858	LEUKOTRIENE D4	FALSE	FALSE	FALSE
ACTIVIN RECEPTOR TYPE IB	hgnc:172	ACVR1B	TTD	2020.06.01	NULL	NULL	BDBM108945	NULL	NULL	NULL	NULL	NULL
ACTIVIN RECEPTOR TYPE IB	hgnc:172	ACVR1B	TTD	2020.06.01	NULL	NULL	US9682983, 33	NULL	NULL	NULL	NULL	NULL
LYMPHOTOXIN-ALPHA	hgnc:6709	LTA	TTD	2020.06.01	NULL	NULL	Anti-LT alpha	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	L-765314	iuphar.ligand:506	L-765314	FALSE	FALSE	FALSE
INTERFERON-GAMMA	hgnc:5438	IFNG	TTD	2020.06.01	NULL	NULL	VIR-201	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	CM-2236	NULL	NULL	NULL	NULL	NULL
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.2187819634820604	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	NULL	CM-2236	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-7268	iuphar.ligand:7824	AZD7268	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	NULL	BMS-954561	NULL	NULL	NULL	NULL	NULL
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	NULL	EC20	NULL	NULL	NULL	NULL	NULL
JNK SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	REN-1654	NULL	NULL	NULL	NULL	NULL
HTR7	hgnc:5302	HTR7	DTC	9/2/20	NULL	3.500511415712966	FUKINOLIC ACID	chembl:CHEMBL487192	FUKINOLIC ACID	FALSE	FALSE	FALSE
MAPK/ERK SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	REN-1654	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	1.312691780892362	GDC-0623	drugbank:DB11982	GDC-0623	FALSE	FALSE	TRUE
PLASMINOGEN ACTIVATOR INHIBITOR	hgnc:8583	SERPINE1	TTD	2020.06.01	NULL	3.088686543276147	Aleplasinin	ncit:C76071	ALEPLASININ	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	CMS-024-02	NULL	NULL	NULL	NULL	NULL
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.032412143	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	NULL	AGN-XX/YY	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	Topetecan	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK618334	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK239512	chembl:CHEMBL3092650	GSK239512	FALSE	FALSE	FALSE
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK598809	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	Pazopanib + Tyverb/Tykerb	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Pazopanib + Tyverb/Tykerb	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	NULL	Dutasteride + tamsulosin	NULL	NULL	NULL	NULL	NULL
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1620607136904151	DICHLORVOS	drugbank:DB11397	DICHLORVOS	FALSE	FALSE	FALSE
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dutasteride + tamsulosin	NULL	NULL	NULL	NULL	NULL
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	GM-CSF cancer vaccine	NULL	NULL	NULL	NULL	NULL
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	Myeloma cancer vaccine	NULL	NULL	NULL	NULL	NULL
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.0053937	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
PROLACTIN RECEPTOR	hgnc:9446	PRLR	TTD	2020.06.01	NULL	NULL	LFA-102	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Ryzodeq	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ALVOCIDIB HYDROCHLORIDE	ncit:C1571	ALVOCIDIB HYDROCHLORIDE	FALSE	FALSE	FALSE
FACILITATES CHROMATIN TRANSCRIPTION COMPLEX	hgnc:11465	SUPT16H	TTD	2020.06.01	NULL	NULL	CBL0102	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.047626006	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	NULL	INCB15050	NULL	NULL	NULL	NULL	NULL
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.024479101	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	VRX496	chembl:CHEMBL2107847	LEXGENLEUCEL-T	FALSE	FALSE	FALSE
ITGAV MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TV-1102	NULL	NULL	NULL	NULL	NULL
HUNTINGTIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Huntingtin gene antisense	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP160	NULL	NULL	TTD	2020.06.01	NULL	NULL	PENNVAX-6	NULL	NULL	NULL	NULL	NULL
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Danoprevir	ncit:C171872	DANOPREVIR	FALSE	FALSE	FALSE
FACTOR XI MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-FXI	NULL	NULL	NULL	NULL	NULL
NCOA1	hgnc:7668	NCOA1	DTC	9/2/20	NULL	1.009762908	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
CTGF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	EXC 001	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-GCGR	NULL	NULL	NULL	NULL	NULL
PTPN1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-PTP1B	NULL	NULL	NULL	NULL	NULL
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	KUR-212	NULL	NULL	NULL	NULL	NULL
HEPATITIS B VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	LB80380	chembl:CHEMBL1652128	LB80380	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.01274458	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TMC649128	chembl:CHEMBL4297499	TMC-649128	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-3281	chembl:CHEMBL1233524	MK-3281	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	MK-1293	NULL	NULL	NULL	NULL	NULL
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	5.834185692854944	Mavrilimumab	ncit:C95788	MAVRILIMUMAB	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR	hgnc:2438	CSF3	TTD	2020.06.01	NULL	NULL	MK-4214	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004458114	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	Insulin determir	NULL	NULL	NULL	NULL	NULL
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	RX-01-423	NULL	NULL	NULL	NULL	NULL
OSTEOCLAST DIFFERENTIATION FACTOR	hgnc:11926	TNFSF11	TTD	2020.06.01	NULL	NULL	CEP-37251	NULL	NULL	NULL	NULL	NULL
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BF-1	iuphar.ligand:8424	BF-1	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	NAN-190	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	DS-7309	NULL	NULL	NULL	NULL	NULL
FUNGAL CELL MEMBRANE ERGOSTEROL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nystatin	rxcui:7597	NYSTATIN	TRUE	FALSE	FALSE
SINUS NODE I(F) CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ivabradine	rxcui:1649480	IVABRADINE	TRUE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.053854022	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
PARATHYROID HORMONE RECEPTOR	hgnc:9609	PTH2R	TTD	2020.06.01	NULL	NULL	UNI-PH (1-34)	NULL	NULL	NULL	NULL	NULL
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	HARMAN-3-CARBOXYLIC ACID	chembl:CHEMBL504850	HARMAN-3-CARBOXYLIC ACID	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II BETA	hgnc:11990	TOP2B	TTD	2020.06.01	NULL	NULL	XB-947	NULL	NULL	NULL	NULL	NULL
INFLUENZA NA MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALN-FLU01	NULL	NULL	NULL	NULL	NULL
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	FENBUTATIN OXIDE	chembl:CHEMBL1472895	FENBUTATIN OXIDE	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anagliptin	ncit:C96202	ANAGLIPTIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Midismase	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	NULL	OPL-CCL2-LPM	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV7	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flupirtine	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	Pentacea	NULL	NULL	NULL	NULL	NULL
IL6ST	hgnc:6021	IL6ST	DTC	9/2/20	NULL	7.001022831425934	BAZEDOXIFENE	rxcui:1441386	BAZEDOXIFENE	TRUE	FALSE	FALSE
COMPLEMENT C3	hgnc:7422	MT-CO3	TTD	2020.06.01	NULL	26.25383561784724	POT-4	iuphar.ligand:9219	AL-78898A	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	3.088686543276147	JVRS-100	ncit:C82353	TLR-DIRECTED CATIONIC LIPID-DNA COMPLEX JVRS-100	FALSE	FALSE	FALSE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	3.580068493342807	Itriglumide	ncit:C65992	ITRIGLUMIDE	FALSE	FALSE	FALSE
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	LC-1	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	NULL	Recombinant von Willebrand factor/recombinant Factor VIII complex	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CHAETOCIN	iuphar.ligand:8388	CHAETOCIN	FALSE	FALSE	FALSE
VON WILLEBRAND FACTOR	hgnc:12726	VWF	TTD	2020.06.01	NULL	NULL	Recombinant von Willebrand factor/recombinant Factor VIII complex	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	GlyT1 PET radiotracers	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002088278	FLUOXETINE HYDROCHLORIDE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GROWTH/DIFFERENTIATION FACTOR 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMG 745	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	NN-1218	NULL	NULL	NULL	NULL	NULL
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.1101559536413171	GDC-0084	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BC-3205	iuphar.ligand:10998	BC-3205	FALSE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	IL-2/gene-modified lymphocytes	NULL	NULL	NULL	NULL	NULL
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.016161179	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
NADPH OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GKT-137831	ncit:C166721	SETANAXIB	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.087512785	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
EBOLA VIRUS VP24 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-7537	drugbank:DB15433	AVI-7537	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	NULL	NIC-002	NULL	NULL	NULL	NULL	NULL
SERINE PROTEASE UNSPECIFIC	hgnc:11756	TFF2	TTD	2020.06.01	NULL	NULL	VT-111a	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.6471533709721451	RG-7446	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	NULL	SB-728-T	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	MINOCYCLINE	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
FREE FATTY ACID RECEPTOR 1	hgnc:4498	FFAR1	TTD	2020.06.01	NULL	NULL	P11187	NULL	NULL	NULL	NULL	NULL
FREE FATTY ACID RECEPTOR 1	hgnc:4498	FFAR1	TTD	2020.06.01	NULL	NULL	JTT-851	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	GNF-PF-3537	chembl:CHEMBL601110	CHEMBL:CHEMBL601110	FALSE	FALSE	FALSE
STAPHYLOCOCCUS ALPHA-HEMOLYSIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AR-301	chembl:CHEMBL4594526	TOSATOXUMAB	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.015892152	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
REGENERATING HUMAN PRO-ISLET PEPTIDE	hgnc:8601	REG3A	TTD	2020.06.01	NULL	NULL	ALF-5755	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	AZD-3199	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	HEPTANE	rxcui:2472186	HEPTANE	TRUE	FALSE	FALSE
LYSOPHOSPHATIDIC ACID RECEPTOR 1	hgnc:3166	LPAR1	TTD	2020.06.01	NULL	8.751278539282415	SAR-100842	iuphar.ligand:11315	SAR100842	FALSE	FALSE	FALSE
SOMATOTROPIN	hgnc:4261	GH1	TTD	2020.06.01	NULL	5.834185692854944	HGH-CTP	iuphar.ligand:12013	SOMATROGON	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	CYCLOPIAZONIC ACID	iuphar.ligand:5350	CYCLOPIAZONIC ACID	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	NULL	SAR351034	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	NIGULDIPINE	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
PLATELET ACTIVATING FACTOR	hgnc:28961	PCLAF	TTD	2020.06.01	NULL	NULL	Indol-3-carbinol	NULL	NULL	NULL	NULL	NULL
GASTRIC H(+)/K(+) ATPASE ALPHA	hgnc:819	ATP4A	TTD	2020.06.01	NULL	NULL	AG-SPT201	NULL	NULL	NULL	NULL	NULL
BACTERIAL 16S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxazolidinones	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.09323095	Norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxazolidinones	NULL	NULL	NULL	NULL	NULL
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	DNDI1417195	chembl:CHEMBL1303948	CHEMBL:CHEMBL1303948	FALSE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Colistimethate	rxcui:2708	COLISTIMETHATE	TRUE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Polymyxin B Sulfate	rxcui:388	POLYMYXIN B SULFATE	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HER2p63-71 peptide vaccine	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	Falecalcitrol	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Enflurane	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.2083637747448194	SCH-442416	iuphar.ligand:3283	SCH442416	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
CHOLESTEROL DESMOLASE	hgnc:2590	CYP11A1	TTD	2020.06.01	NULL	4.375639269641208	Aminoglutethimide	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.031555091	ZOTEPINE	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	BEMA buprenorphine transmucosal	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ZK-200775	ncit:C65617	FANAPANEL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	DISULFOTON	ncit:C163652	DISULFOTON	FALSE	FALSE	FALSE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	NULL	PREMETREXED	NULL	NULL	NULL	NULL	NULL
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.009532983	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
AMILORIDE-SENSITIVE SODIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triamterene	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
BACTERIAL CYSTATHIONINE GAMMA-SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GW-3333	NULL	NULL	NULL	NULL	NULL
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2328499833068492	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	NULL	RWJ-51204	NULL	NULL	NULL	NULL	NULL
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	2.917092846427472	Xanthine	rxcui:1311085	XANTHINE	FALSE	FALSE	FALSE
BACTERIAL INTEGRAL MEMBRANE LMRP	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinupristin	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2273059360852575	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
TRYPTOPHAN 5-HYDROXYLASE 1	hgnc:12008	TPH1	TTD	2020.06.01	NULL	NULL	AGN-2979	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	NULL	DL-017	NULL	NULL	NULL	NULL	NULL
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2220197515251353	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
PANCREATIC ELASTASE 1	hgnc:3308	CELA1	TTD	2020.06.01	NULL	NULL	Alpha 1-PI	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	1.093909817410302	NGD 94-1	iuphar.ligand:3297	[3H]NGD941	FALSE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR	hgnc:2436	CSF2RB	TTD	2020.06.01	NULL	4.375639269641208	Leridistim	ncit:C1846	LERIDISTIM	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2580229544751573	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
CYP3A4 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-4557	drugbank:DB05447	AVI-4557	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Inamrinone Lactate	rxcui:91236	INAMRINONE LACTATE	TRUE	FALSE	FALSE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	FR167653	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	NULL	LU302146	NULL	NULL	NULL	NULL	NULL
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.007733089	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CATECHOL-O-METHYL-TRANSFERASE	hgnc:2228	COMT	TTD	2020.06.01	NULL	NULL	BIA 3-202	NULL	NULL	NULL	NULL	NULL
STEROID 5-ALPHA-REDUCTASE 1	hgnc:11284	SRD5A1	TTD	2020.06.01	NULL	NULL	FR-146687	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	Lomefloxacin	rxcui:28872	LOMEFLOXACIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	6.563458904461812	SGN-30	drugbank:DB05471	SGN-30	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	2.316514907	Huperzine A	rxcui:2267703	HUPERZINE A	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	NULL	LT-1951	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceforanide	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.048618214	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
PLASMODIUM APICAL MEMBRANE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PfAMA-1	NULL	NULL	NULL	NULL	NULL
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	DMP-444	NULL	NULL	NULL	NULL	NULL
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	0.5303805175322677	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
5-HT 1E RECEPTOR	hgnc:5291	HTR1E	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	S32504	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	S32504	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	0.049723174	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Demeclocycline	rxcui:3154	DEMECLOCYCLINE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Capravirine	ncit:C81612	CAPRAVIRINE	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS HELICASE-PRIMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY 57-1293	ncit:C136516	PRITELIVIR	FALSE	FALSE	FALSE
MYCOBACTERIUM D-ALANINE-D-ALANINE LIGASE A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloserine	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
PLASMODIUM CDK PFMRK	NULL	NULL	TTD	2020.06.01	NULL	NULL	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
PIGMENT EPITHELIUM-DERIVED FACTOR	hgnc:8824	SERPINF1	TTD	2020.06.01	NULL	NULL	AdPEDR	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Neramexane	ncit:C76781	NERAMEXANE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	Quinolones	NULL	NULL	NULL	NULL	NULL
AURORA B MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PHA-739358	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Balofloxacin	ncit:C72631	BALOFLOXACIN	FALSE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefozopran	ncit:C76172	CEFOZOPRAN	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ciprofloxacin XR	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-944	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALO-02 Oxycodone- naltrexone core	NULL	NULL	NULL	NULL	NULL
INTERFERON ALPHA/BETA RECEPTOR 1	hgnc:5432	IFNAR1	TTD	2020.06.01	NULL	NULL	Zadaxin/lamivudine	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	Zadaxin/lamivudine	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	FFC-14A	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	GW-427353	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	LY-362884	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	N-5984	NULL	NULL	NULL	NULL	NULL
CHOLECYSTOKININ RECEPTOR TYPE A	hgnc:1570	CCKAR	TTD	2020.06.01	NULL	NULL	A-74498	NULL	NULL	NULL	NULL	NULL
CHOLECYSTOKININ RECEPTOR TYPE A	hgnc:1570	CCKAR	TTD	2020.06.01	NULL	NULL	GG-8573	NULL	NULL	NULL	NULL	NULL
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	NULL	GG-8573	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 5	hgnc:7958	NPY5R	TTD	2020.06.01	NULL	NULL	GW-594884A	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDDB-41331	NULL	NULL	NULL	NULL	NULL
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	NULL	Ro-27-3225	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	Golnerminogene pradenovac	NULL	NULL	NULL	NULL	NULL
TRYPANOSOMA TRYPANOTHIONE REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vitamin A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	NULL	GW-796406	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	NULL	GW-796406	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	NULL	Liproca Depot	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 5	hgnc:7958	NPY5R	TTD	2020.06.01	NULL	7.501095891	FR-79620	chembl:CHEMBL6893	FR-79620	FALSE	FALSE	FALSE
VIRUS MAJOR ENVELOPE P37	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tecovirimat	rxcui:2055104	TECOVIRIMAT	TRUE	FALSE	FALSE
STREPTOCOCCUS METHIONYL-TRNA SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	REP8839	drugbank:DB05224	REP8839	FALSE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	IL-2/CD40L-expressing leukemia vaccine	NULL	NULL	NULL	NULL	NULL
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	NULL	IL-2/CD40L-expressing leukemia vaccine	NULL	NULL	NULL	NULL	NULL
RECEPTOR UNSPECIFIC	hgnc:16147	MCM8	TTD	2020.06.01	NULL	NULL	Lactermin	NULL	NULL	NULL	NULL	NULL
CORTICOSTEROID-BINDING GLOBULIN	hgnc:1540	SERPINA6	TTD	2020.06.01	NULL	NULL	I-vation	NULL	NULL	NULL	NULL	NULL
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA4.1	hgnc:18865	KCNT1	TTD	2020.06.01	NULL	0.7001022831425934	phorbol 12-myristate 13-acetate	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	NULL	ErepoXen	NULL	NULL	NULL	NULL	NULL
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATN-224	ncit:C62514	TIOMOLIBDATE CHOLINE	FALSE	FALSE	FALSE
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Coprexa	ncit:C74001	TIOMOLIBDATE DIAMMONIUM	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefpodoxime	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Loracarbef	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	FAD-104	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Barbiturate	ncit:C67084	BARBITURATE	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nitrous oxide	rxcui:7486	NITROUS OXIDE	TRUE	FALSE	FALSE
LAMININ BETA-3 CHAIN	hgnc:6490	LAMB3	TTD	2020.06.01	NULL	NULL	LAMB3-transduced autologous epidermal stem cells	NULL	NULL	NULL	NULL	NULL
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	UK-66914	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	NULL	KP-496	NULL	NULL	NULL	NULL	NULL
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	NULL	KP-496	NULL	NULL	NULL	NULL	NULL
MYCOBACTERIUM BIOSYNTHETIC ALANINE RACEMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloserine	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
PLASMODIUM ELONGATION FACTOR 1-ALPHA 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ge2270a	NULL	NULL	NULL	NULL	NULL
RAS-RELATED PROTEIN RAB-9A	hgnc:9792	RAB9A	TTD	2020.06.01	NULL	0.182318303	Benzoic Acid	rxcui:18989	BENZOIC ACID	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.012208247	Ephedrine	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
RIBOSOME A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Arbekacin	rxcui:26397	ARBEKACIN	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Neocarzinostatin	chembl:CHEMBL454708	NEOCARZINOSTATIN	FALSE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ramosetron	ncit:C61921	RAMOSETRON	FALSE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tandospirone	ncit:C87208	TANDOSPIRONE	FALSE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	NULL	CB-10-01	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Darunavir	rxcui:460132	DARUNAVIR	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2B	hgnc:282	ADRA2B	TTD	2020.06.01	NULL	NULL	AGN-199981	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	INDAZOLE-3-CARBOXYLICACID	chembl:CHEMBL502057	CHEMBL:CHEMBL502057	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	CHF-3381	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	CHF-3381	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CHF-3381	NULL	NULL	NULL	NULL	NULL
BACTERIAL 70S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Capreomycin	rxcui:78903	CAPREOMYCIN	TRUE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	NULL	Cyclolignan picropodophyllin	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	SSR-125047	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	4.150804050252529	Nemonapride	ncit:C73036	NEMONAPRIDE	FALSE	FALSE	FALSE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	0.9376369863516875	Aminoglutethimide	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-332991	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PD-332991	NULL	NULL	NULL	NULL	NULL
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-332991	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ADX-2 series	NULL	NULL	NULL	NULL	NULL
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	NULL	BSF-78438	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxytrex	wikidata:Q7116185	OXYTREX	FALSE	FALSE	FALSE
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	99mTc-rBitistatin	NULL	NULL	NULL	NULL	NULL
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	NULL	GSK-326416	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	GPD-1116	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	NULL	GPD-1116	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	NULL	GPD-1116	NULL	NULL	NULL	NULL	NULL
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	NULL	ADR-851	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	NULL	Clobazam - Lundbeck	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	0.2983390411119005	ATOSIBAN	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1221108633388244	Butethal	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Recoflavone eye drops	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM CHAPERONE BIP	hgnc:5238	HSPA5	TTD	2020.06.01	NULL	NULL	SAM-6	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Altretamine	rxcui:5296	ALTRETAMINE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceftazidime	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	Desvenalfaxine succinate	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 1	hgnc:1602	CCR1	TTD	2020.06.01	NULL	NULL	AVE1701	NULL	NULL	NULL	NULL	NULL
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	NULL	PU3	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-Glutamic Acid	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	N-0923	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF9601N	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	GYKI-47261	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Huperzine A	rxcui:2267703	HUPERZINE A	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Saquinavir	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	NULL	AVE-2268	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Denagliptin	ncit:C76909	DENAGLIPTIN	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	DIFLOMOTECAN	ncit:C90824	DIFLOMOTECAN	FALSE	FALSE	FALSE
SERINE PROTEASE UNSPECIFIC	hgnc:11756	TFF2	TTD	2020.06.01	NULL	2.917092846427472	Camostat	ncit:C73213	CAMOSTAT	FALSE	FALSE	FALSE
THIOREDOXIN REDUCTASE	hgnc:9355	PRDX5	TTD	2020.06.01	NULL	3.750547945406749	Motexafin gadolinium	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.4375639269641208	Dolasetron	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indinavir	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
INFLUENZA M2 PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rimantadine	rxcui:9386	RIMANTADINE	TRUE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Finasteride	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	XL019	drugbank:DB05243	XL019	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.1835932560688619	Fosphenytoin	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	2.625383561784724	Vicriviroc	ncit:C73589	VICRIVIROC	FALSE	FALSE	FALSE
RESPIRATORY SYNCYTIAL VIRUS PROTEIN F	NULL	NULL	TTD	2020.06.01	NULL	NULL	TMC-353121	NULL	NULL	NULL	NULL	NULL
HIF-1 RESPONSIVE PROTEIN RTP801	hgnc:24944	DDIT4	TTD	2020.06.01	NULL	NULL	PF-04523655	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfapyridine	rxcui:10188	SULFAPYRIDINE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.023716202	Taxol	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
GABA(A) RECEPTOR GAMMA-2	hgnc:4087	GABRG2	TTD	2020.06.01	NULL	0.1562728310586145	ZK-93423	drugbank:DB17063	ZK-93423	FALSE	FALSE	FALSE
GUANYLATE CYCLASE	hgnc:4187	GC	TTD	2020.06.01	NULL	0.4375639269641209	Nitric Oxide	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
INTERLEUKIN-10	hgnc:5962	IL10	TTD	2020.06.01	NULL	NULL	F-8-IL-10 fusion protein	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	BERBAMINE	ncit:C162341	BERBAMINE	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.019304291	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CYTOMEGALOVIRUS DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASP0113	ncit:C111903	CMVPP65/GB PLASMID VACCINE ASP0113	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.013429072	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID MINOR GROOVE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Brostallicin	ncit:C1889	BROSTALLICIN	FALSE	FALSE	FALSE
PROSTATE SPECIFIC ANTIGEN	hgnc:6364	KLK3	TTD	2020.06.01	NULL	0.8751278539282416	Rilimogene galvacirepvec	ncit:C38681	RILIMOGENE GALVACIREPVEC	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.013905633	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
STEROID 11-BETA-HYDROXYLASE	hgnc:2591	CYP11B1	TTD	2020.06.01	NULL	1.093909817410302	FADROZOLE	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
VARIOLA VIRUS ENVELOPE PHOSPHOLIPASE F13	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tecovirimat	rxcui:2055104	TECOVIRIMAT	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	ThermoProfen	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	ThermoProfen	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	S-ETOMIDATE	chembl:CHEMBL279678	S-ETOMIDATE	FALSE	FALSE	FALSE
SECOND PHASE INSULIN SECRETION	NULL	NULL	TTD	2020.06.01	NULL	NULL	AGI-1067	chembl:CHEMBL83626	SUCCINOBUCOL	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAL-30072	iuphar.ligand:11004	BAL30072	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	NULL	INGN-225	NULL	NULL	NULL	NULL	NULL
TRYPANOSOMA CRUZIPAIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	MANIDIPINE	rxcui:29275	MANIDIPINE	FALSE	FALSE	FALSE
PLACENTA GROWTH FACTOR	hgnc:8893	PGF	TTD	2020.06.01	NULL	NULL	SFLT-01	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	SFLT-01	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	P-276	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	INOC-005	NULL	NULL	NULL	NULL	NULL
IMMUNOGLOBULIN G	NULL	NULL	TTD	2020.06.01	NULL	NULL	Immune globulin subcutaneous, 20% liquid	NULL	NULL	NULL	NULL	NULL
CARBAMOYL-PHOSPHATE SYNTHETASE I	hgnc:2323	CPS1	TTD	2020.06.01	NULL	NULL	Polidocanol - BioForm Medical/Chemische Fabrik Kreussler & Co	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cethrin	NULL	NULL	NULL	NULL	NULL
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	IODOMELATONIN	drugbank:DB08190	N-[2-(2-IODO-5-METHOXY-1H-INDOL-3-YL)ETHYL]ACETAMIDE	FALSE	FALSE	FALSE
OVARIAN CARCINOMA ANTIGEN CA125	hgnc:15582	MUC16	TTD	2020.06.01	NULL	11.25164383622025	Abagovomab	ncit:C26449	ABAGOVOMAB	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	ISOORIENTIN	chembl:CHEMBL239559	ISOORIENTIN	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.052090944	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.064944553	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.007072693	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.008874036	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
HEPARANASE	hgnc:5164	HPSE	TTD	2020.06.01	NULL	2.917092846427472	PG-545	ncit:C95202	PIXATIMOD	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.040515178	MGCD516	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002170994	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.8607814956671229	Estradiol valerate/dienogest	wikidata:Q60218116	ESTRADIOL VALERATE/DIENOGEST	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	EUGENOL	rxcui:4186	EUGENOL	TRUE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	AZD-2327	NULL	NULL	NULL	NULL	NULL
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	CLANFENUR	ncit:C78082	CLANFENUR	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1363835616511545	DAPHNORIN	chembl:CHEMBL1209491	DAPHNORIN	FALSE	FALSE	FALSE
ACTIVATION B7-1 ANTIGEN	hgnc:1700	CD80	TTD	2020.06.01	NULL	NULL	RhuDex	NULL	NULL	NULL	NULL	NULL
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.012719882	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	Adjustable basal insulin	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
BACTERIAL PROTEIN SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Radezolid iv	NULL	NULL	NULL	NULL	NULL
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.3059887601147698	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.027276712	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	1.944728564284981	RP-49356	chembl:CHEMBL1563246	CHEMBL:CHEMBL1563246	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HM-78136B	NULL	NULL	NULL	NULL	NULL
CELL SURFACE A33 ANTIGEN	hgnc:4445	GPA33	TTD	2020.06.01	NULL	NULL	Radiolabelled-huA33	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	DULOXETINE HYDROCHLORIDE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 70	hgnc:5232	HSPA1A	TTD	2020.06.01	NULL	NULL	AG-707	NULL	NULL	NULL	NULL	NULL
BACTERIAL NADH-DEPENDENT ENOYL-ACP REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MUT-056399	iuphar.ligand:11000	MUT056399	FALSE	FALSE	FALSE
STAPHYLOCOCCUS ENOYL ACP REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MUT-056399	iuphar.ligand:11000	MUT056399	FALSE	FALSE	FALSE
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	NULL	BAY-60-5521	NULL	NULL	NULL	NULL	NULL
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Butoconazole	rxcui:19884	BUTOCONAZOLE	TRUE	FALSE	FALSE
RHINOVIRUS CAPSID PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	BTA-798	chembl:CHEMBL2062774	VAPENDAVIR	FALSE	FALSE	FALSE
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	WT1 peptide vaccine	NULL	NULL	NULL	NULL	NULL
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	NULL	Tau-binding PET tracer	NULL	NULL	NULL	NULL	NULL
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	NULL	Davunetide intranasal spray	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CX-717	drugbank:DB05047	CX-717	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS GAG PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	RVSVIN HIV-1 gag vaccine	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.7955707762984014	Lobeglitazone	ncit:C91021	LOBEGLITAZONE	FALSE	FALSE	FALSE
B2 BRADYKININ RECEPTOR	hgnc:1030	BDKRB2	TTD	2020.06.01	NULL	2.187819634820604	Fasitibant chloride	ncit:C167030	FASITIBANT CHLORIDE	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	0.3125456621172291	XEN-402	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ladostigil	ncit:C77584	LADOSTIGIL	FALSE	FALSE	FALSE
HEPATITIS C VIRUS SERINE PROTEASE NS3/4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Telaprevir	rxcui:1102261	TELAPREVIR	TRUE	FALSE	FALSE
S-NITROSOGLUTATHIONE REDUCTASE	hgnc:1548	CBR1	TTD	2020.06.01	NULL	4.375639269641208	N6022	chembl:CHEMBL1738699	N6022	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.073954467	KH-902	ncit:C162879	CONBERCEPT	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	NULL	VCH-286	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP160	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN/ENV	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GAG PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN/ENV	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS NEGATIVE FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN/ENV	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REV PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN/ENV	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN/ENV	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	Merestinib, LY2801653	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	HuM195/rGel	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lurbinectedin	rxcui:2374729	LURBINECTEDIN	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	NULL	COR-1	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	NULL	SCH-900117	NULL	NULL	NULL	NULL	NULL
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE BETA	hgnc:5960	IKBKB	TTD	2020.06.01	NULL	5.000730593875666	IMD-1041	chembl:CHEMBL3545168	IMD-1041	FALSE	FALSE	FALSE
INTERLEUKIN-13	hgnc:5973	IL13	TTD	2020.06.01	NULL	8.751278539282415	CNTO-5825	chembl:CHEMBL2109464	CNTO-5825	FALSE	FALSE	FALSE
NEURAL CELL ADHESION MOLECULE	hgnc:7656	NCAM1	TTD	2020.06.01	NULL	NULL	FGLL	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	CNTO-3649	NULL	NULL	NULL	NULL	NULL
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	NULL	SD-6010	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	SAR-114137	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	SAR-114137	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	PSMA-VRP	NULL	NULL	NULL	NULL	NULL
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	1.050153425	BMS-936564	iuphar.ligand:9161	ULOCUPLUMAB	FALSE	FALSE	FALSE
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	1.750255707856483	REGN-910	iuphar.ligand:8457	NESVACUMAB	FALSE	FALSE	FALSE
LIPOPROTEIN LIPASE	hgnc:6677	LPL	TTD	2020.06.01	NULL	NULL	AMT-011	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS IRON-REGULATED SURFACE DETERMINANT B	NULL	NULL	TTD	2020.06.01	NULL	NULL	V-710	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	LY2784544	ncit:C116857	GANDOTINIB	FALSE	FALSE	TRUE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ARRY-300	chembl:CHEMBL3545359	ARRY-300	FALSE	FALSE	FALSE
DYSTROPHIN	hgnc:2928	DMD	TTD	2020.06.01	NULL	NULL	Biostrophin	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	AN-2898	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	NULL	AN-2898	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	NULL	AN-2898	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	4.039051633514961	E-2212	chembl:CHEMBL2151205	E-2212	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	DABIS MALEATE	NULL	NULL	NULL	NULL	NULL
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	NULL	PMID23981898C11d	NULL	NULL	NULL	NULL	NULL
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY-35-3377	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Odelepran	chembl:CHEMBL2103878	ODELEPRAN	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	ZYH-1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ZYH-1	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	TT-401	NULL	NULL	NULL	NULL	NULL
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	2.059124362184098	LJM716	ncit:C101895	ELGEMTUMAB	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-7288	drugbank:DB17094	MK-7288	FALSE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	NULL	RQ-00000005	NULL	NULL	NULL	NULL	NULL
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	NULL	RG7201	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-12 BETA	hgnc:5970	IL12B	TTD	2020.06.01	NULL	NULL	NHS-IL 12	NULL	NULL	NULL	NULL	NULL
PHENYLALANINE HYDROXYLASE	hgnc:8582	PAH	TTD	2020.06.01	NULL	NULL	Phenylalanine hydroxylase	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	Girentuximab	ncit:C1960	GIRENTUXIMAB	FALSE	FALSE	FALSE
INTEGRIN BETA-1	hgnc:6153	ITGB1	TTD	2020.06.01	NULL	NULL	131I-radretumab	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 9	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-4447943	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.2	hgnc:1395	CACNA1H	TTD	2020.06.01	NULL	NULL	TTA-A8	NULL	NULL	NULL	NULL	NULL
PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9	hgnc:20001	PCSK9	TTD	2020.06.01	NULL	NULL	PCSK9 Adnectin	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ADX-71943	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	Nelipepimut S	ncit:C117985	NELIPEPIMUT-S	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	PF-05280014	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	FRM-6308	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	AV4025	NULL	NULL	NULL	NULL	NULL
HEPATITIS B VIRUS LARGE ENVELOPE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	NASVAC	NULL	NULL	NULL	NULL	NULL
NATURAL KILLER CELL RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NASVAC	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMG-139	ncit:C166795	BRAZIKUMAB	FALSE	FALSE	FALSE
DYSTROPHIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PRO-044	NULL	NULL	NULL	NULL	NULL
CORTICOSTEROID-BINDING GLOBULIN	hgnc:1540	SERPINA6	TTD	2020.06.01	NULL	3.281729452230906	Alclometasone	rxcui:108088	ALCLOMETASONE	TRUE	FALSE	FALSE
PLASMODIUM APICAL MEMBRANE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	DNA-Ad	NULL	NULL	NULL	NULL	NULL
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	U300	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gemigliptin	ncit:C118446	GEMIGLIPTIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	MEM-1414	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	NULL	MEM-1414	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	NULL	MEM-1414	NULL	NULL	NULL	NULL	NULL
SOMATOSTATIN RECEPTOR TYPE 2	hgnc:11331	SSTR2	TTD	2020.06.01	NULL	NULL	Re-188-P-2045	NULL	NULL	NULL	NULL	NULL
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	NULL	ISF35	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-13	hgnc:5973	IL13	TTD	2020.06.01	NULL	8.751278539282415	QAX-576	chembl:CHEMBL2109465	QAX-576	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.3236220106976548	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
FUNGAL 1,3-BETA-GLUCAN SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	SCY-078	rxcui:2560213	IBREXAFUNGERP	TRUE	FALSE	FALSE
APOPTOSIS SIGNAL-REGULATING KINASE 1	hgnc:6857	MAP3K5	TTD	2020.06.01	NULL	NULL	GS-4977	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 3	hgnc:8534	P2RX3	TTD	2020.06.01	NULL	26.25383561784724	AF-219	ncit:C166945	GEFAPIXANT	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN 4F2	hgnc:11026	SLC3A2	TTD	2020.06.01	NULL	26.25383561784724	IGN523	iuphar.ligand:8737	IGN523	FALSE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DL2	hgnc:6330	KIR2DL2	TTD	2020.06.01	NULL	4.375639269641208	IPH-2102	chembl:CHEMBL2109500	LIRILUMAB	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.09869863	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.000146118775133	SAR-125844	drugbank:DB15382	SAR-125844	FALSE	FALSE	FALSE
RESPIRATORY SYNCYTIAL VIRUS PROTEIN F	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-5806	ncit:C118505	PRESATOVIR	FALSE	FALSE	FALSE
BCL-2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beclanorsen	ncit:C171736	BECLANORSEN	FALSE	FALSE	FALSE
INTEGRIN ALPHA-4/BETA-7	NULL	NULL	TTD	2020.06.01	NULL	NULL	MLN0002	rxcui:1538097	VEDOLIZUMAB	TRUE	FALSE	FALSE
BACILLUS ANTHRACIS PROTECTIVE ANTIGEN	NULL	NULL	TTD	2020.06.01	NULL	NULL	ETI-204	chembl:CHEMBL3544926	OBILTOXAXIMAB	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	1.346350544504987	verubecestat	ncit:C152868	VERUBECESTAT	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	1.009762908	ALG-1001	chembl:CHEMBL4297529	RISUTEGANIB	FALSE	FALSE	FALSE
GATA4	hgnc:4173	GATA4	DTC	9/2/20	NULL	17.50255707856483	NSC-140905	chembl:CHEMBL1684097	CHEMBL:CHEMBL1684097	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	2.972132334095915	Cixutumumab	ncit:C79828	CIXUTUMUMAB	FALSE	TRUE	TRUE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	1.280674908	JNJ-39439335	ncit:C170153	MAVATREP	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.057700738	PF-05212384	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	CHLORIDE	drugbank:DB14547	CHLORIDE ION	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BIS(PIPERIDINYLTHIOCARBONYL)DISULFIDE	chembl:CHEMBL121516	BIS(PIPERIDINYLTHIOCARBONYL)DISULFIDE	FALSE	FALSE	FALSE
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	GSK618334	NULL	NULL	NULL	NULL	NULL
KRUPPEL LIKE FACTOR 4	hgnc:6348	KLF4	TTD	2020.06.01	NULL	26.25383561784724	APTO-253	drugbank:DB17143	APTO-253	FALSE	FALSE	FALSE
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	0.3889457128569963	Daratumumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	0.596678082	CC-486	ncit:C118288	ORAL AZACITIDINE	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Radium-223-Dichloride	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	ICI 118,551	NULL	NULL	NULL	NULL	NULL
PLASMODIUM DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Delafloxacin Meglumine	rxcui:1927662	DELAFLOXACIN MEGLUMINE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Delafloxacin Meglumine	rxcui:1927662	DELAFLOXACIN MEGLUMINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	AZOXYSTROBIN	drugbank:DB07401	AZOXYSTROBIN	FALSE	FALSE	FALSE
INFLUENZA POLYMERASE ACIDIC ENDONUCLEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Baloxavir marboxil	rxcui:2099995	BALOXAVIR MARBOXIL	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Moxidectin	rxcui:1047072	MOXIDECTIN	TRUE	FALSE	FALSE
ONCHOCERCA GLUTAMATE-GATED CHLORIDE CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Moxidectin	rxcui:1047072	MOXIDECTIN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Revefenacin	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.6908904109959803	NAKIJIQUINONES G	chembl:CHEMBL502529	NAKIJIQUINONES G	FALSE	FALSE	FALSE
HYPERPOLARIZATION CYCLIC NUCLEOTIDE-GATED CHANNEL	hgnc:29665	MALAT1	TTD	2020.06.01	NULL	2.917092846427472	Ivabradine	rxcui:1649480	IVABRADINE	TRUE	FALSE	FALSE
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	BIL010t	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BIIB104	chembl:CHEMBL5095022	PESAMPATOR	FALSE	FALSE	FALSE
GAP JUNCTION ALPHA-1 PROTEIN	hgnc:4274	GJA1	TTD	2020.06.01	NULL	NULL	Granexin gel	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	NULL	CONTIGOSIDE B	NULL	NULL	NULL	NULL	NULL
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	3,4-DIMETHOXYBENZALDEHYDE	chembl:CHEMBL1088937	3,4-DIMETHOXYBENZALDEHYDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	VITAMIN K3H2	chembl:CHEMBL1405447	VITAMIN K3H2	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	1,3-DINITRO-NAPHTHALENE	chembl:CHEMBL163970	CHEMBL:CHEMBL163970	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.1400204566285186	TRIFLOXYSTROBIN	chembl:CHEMBL1897483	TRIFLOXYSTROBIN	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	1.419126249613364	RO-4603325	chembl:CHEMBL2203705	CHEMBL:CHEMBL2203705	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.2488515224440497	SJ000117911	chembl:CHEMBL589915	CHEMBL:CHEMBL589915	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	(+)-ALPHA-TOCOPHERYL SUCCINATE	chembl:CHEMBL81421	(+)-ALPHA-TOCOPHERYL SUCCINATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.014024485	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.036951211	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.020257589	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	0.4688184931758437	ADENOSINE DIPHOSPHATE	iuphar.ligand:1712	ADP	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.054695491	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	ADIPHENINE	rxcui:333	ADIPHENINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
ADRENERGIC NEURON	NULL	NULL	TTD	2020.06.01	NULL	NULL	Debrisoquin	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	Anisodamine	drugbank:DB11785	ANISODAMINE	FALSE	FALSE	FALSE
P2X PURINOCEPTOR 3	hgnc:8534	P2RX3	TTD	2020.06.01	NULL	26.25383561784724	Gefapixant	ncit:C166945	GEFAPIXANT	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.5645986154375752	HBI-3000	chembl:CHEMBL4594410	SULCARDINE SULFATE	FALSE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Troleandomycin	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1620607136904151	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,3,3',4',5'-PENTAMETHOXYCHALCONE	chembl:CHEMBL608862	CHEMBL:CHEMBL608862	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	L-CYSTEINESULPHINIC ACID	iuphar.ligand:5447	L-CYSTEINE SULPHINIC ACID	FALSE	FALSE	FALSE
IMMUNOGLOBULIN EPSILON FC RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzylpenicilloyl Polylysine	rxcui:19079	BENZYLPENICILLOYL POLYLYSINE	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	YM-934	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Seebri	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	SJ000147784	chembl:CHEMBL590186	CHEMBL:CHEMBL590186	FALSE	FALSE	FALSE
ESTRAMUSTINE BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Estramustine	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
RNA SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Plicamycin	rxcui:6995	PLICAMYCIN	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flufenamic Acid	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	8-[METHYL(4-PHENYLBUTYL)AMINO]CAFFEINE	chembl:CHEMBL1927684	CHEMBL:CHEMBL1927684	FALSE	FALSE	FALSE
5-HT 5A RECEPTOR	hgnc:5300	HTR5A	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
HISTAMINE RECEPTOR	hgnc:5172	HR	TTD	2020.06.01	NULL	NULL	LCB-2183	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	NDDP	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	YM-430	NULL	NULL	NULL	NULL	NULL
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vancomycin inhalation powder	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ontazolast	ncit:C79123	ONTAZOLAST	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	0.5048814541893701	2-ARACHIDONOYLGLYCEROL	iuphar.ligand:729	2-ARACHIDONOYLGLYCEROL	FALSE	FALSE	FALSE
MYOSIN LIGHT KINASE	hgnc:7590	MYLK	TTD	2020.06.01	NULL	NULL	ME-3407	NULL	NULL	NULL	NULL	NULL
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.4773424657790409	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
5-HT 1F RECEPTOR	hgnc:5292	HTR1F	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	NULL	DT-TX-30	NULL	NULL	NULL	NULL	NULL
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	NULL	MPL-S	NULL	NULL	NULL	NULL	NULL
LIVER CARBOXYLESTERASE	hgnc:1863	CES1	TTD	2020.06.01	NULL	NULL	HL-004	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefamandole	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PD-143188	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.1286952726365061	Hyoscine	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
HISTAMINE RECEPTOR	hgnc:5172	HR	TTD	2020.06.01	NULL	17.50255707856483	Levomequitazine	ncit:C90859	LEVOMEQUITAZINE	FALSE	FALSE	FALSE
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Intranasal apomorphine	NULL	NULL	NULL	NULL	NULL
CHOLESTENOL DELTA-ISOMERASE	hgnc:3133	EBP	TTD	2020.06.01	NULL	NULL	SR-31747	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY-Y-5959	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	GNF-PF-4832	chembl:CHEMBL601137	CHEMBL:CHEMBL601137	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.105015342	CHLORFENAPYR	chembl:CHEMBL1869551	CHLORFENAPYR	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.063110182	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.1704794520639431	DAPHNORIN	chembl:CHEMBL1209491	DAPHNORIN	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.1902451856365742	N-(3-OXODODECANOYL)HOMOSERINELACTONE	chembl:CHEMBL8483	CHEMBL:CHEMBL8483	FALSE	FALSE	FALSE
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hydroquinone	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	RHODAMINE	chembl:CHEMBL428971	RHODAMINE	FALSE	FALSE	FALSE
IRON	hgnc:4650	GTF2E1	TTD	2020.06.01	NULL	NULL	Monohydroxyethylrutoside	NULL	NULL	NULL	NULL	NULL
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	2.187819634820604	Rilapladib	ncit:C76401	RILAPLADIB	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.0296486	Metaraminol	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PHOSALONE	chembl:CHEMBL1528531	PHOSALONE	FALSE	FALSE	FALSE
G1/S-SPECIFIC CYCLIN-D1	hgnc:1582	CCND1	TTD	2020.06.01	NULL	1.250182648468916	Briciclib	ncit:C141431	BRICICLIB	FALSE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	2.187819634820604	ONT-10	ncit:C101262	LIPOSOMAL MUC1/PET-LIPID A VACCINE ONT-10	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.8751278539282416	TLC-388	chembl:CHEMBL4594352	TLC-388	FALSE	FALSE	FALSE
RECEPTOR UNSPECIFIC	hgnc:16147	MCM8	TTD	2020.06.01	NULL	NULL	Prosaptide TX14(A)	NULL	NULL	NULL	NULL	NULL
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.050007306	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
CYTOKINE RECEPTOR UNSPECIFIC	hgnc:2355	CRH	TTD	2020.06.01	NULL	NULL	AD-452	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Anti-CD22	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-297995	rxcui:1876597	NALDEMEDINE	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAND-26	ncit:C125608	BEGELOMAB	FALSE	FALSE	FALSE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	ADX N05	NULL	NULL	NULL	NULL	NULL
RIBONUCLEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MazF gene therapy, HIV	NULL	NULL	NULL	NULL	NULL
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-466317A	chembl:CHEMBL427058	GSK-466317A	FALSE	FALSE	FALSE
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	NULL	Vedolizmab	NULL	NULL	NULL	NULL	NULL
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.3977853881492007	2-(4-ISOPROPYLPHENYL)BENZOTHIAZOLE	chembl:CHEMBL1351908	CHEMBL:CHEMBL1351908	FALSE	FALSE	FALSE
INTEGRIN BETA-7	hgnc:6162	ITGB7	TTD	2020.06.01	NULL	NULL	Vedolizmab	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	TH-302	ncit:C71722	EVOFOSFAMIDE	FALSE	FALSE	FALSE
RETINAL PIGMENT EPITHELIUM PROTEIN	hgnc:10294	RPE65	TTD	2020.06.01	NULL	NULL	Leber's congenital amaurosis gene therapy	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-04776548	chembl:CHEMBL3219143	PF-04776548	FALSE	FALSE	FALSE
PLASMODIUM APICAL MEMBRANE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AdCh63 AMA1	NULL	NULL	NULL	NULL	NULL
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.08334551	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	CAR CD30 T cells	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	INO-3401	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	Anti-GPC3 CAR T	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART-meso-19 T cells	NULL	NULL	NULL	NULL	NULL
CSNK1G3	hgnc:2456	CSNK1G3	DTC	9/2/20	NULL	0.4375639269641208	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	CART-meso-19 T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19+ CAR T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-directed CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19-CAR T	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	Autologous Anti-CD 123 CAR TCR/4-1BB-expressing T-lymphocytes	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CART22 cells expressing anti-CD22 scFv TCRz:41BB	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19.CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Retroviral vector-transduced autologous T cells to express CD22-specific CARs	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	Mesothelin-targeted T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Allogeneic CART-19	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	Allogeneic CART-33	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-EGFRvIII CAR T cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CD20 CAR T cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD22-Targeted CAR-T cells	NULL	NULL	NULL	NULL	NULL
EPSTEIN-BARR VIRUS LATENT MEMBRANE PROTEIN 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	LMP1-CAR-T cells	ncit:C136986	LMP1-SPECIFIC CHIMERIC ANTIGEN RECEPTOR-EXPRESSING T LYMPHOCYTES	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 Redirected Autologous T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR-T cells	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	Retroviral vector-transduced autologous T cells to express anti-GPC3 CARs	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD19	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR20	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR20	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Anti-CD19/22-CAR vector-transduced T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19/22-CAR vector-transduced T cells	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	NULL	CD10-CART	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	CART-19/BCMA	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART-19/BCMA	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR-T lymphocytes	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC PROGENITOR CELL ANTIGEN CD34	hgnc:1662	CD34	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD34	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA-CART	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CARTmeso/19	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	CARTmeso/19	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CAR19 T cells carrying cytoplasmic activated PD-1	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA CART and huCART19	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	BCMA CART and huCART19	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-targeted CAR-T cells	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TMB-607	chembl:CHEMBL168640	PPL-100	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cabotegravir LA	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Dual Specificity CD19 and CD22 CAR-T Cell	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Delavirdine	rxcui:83816	DELAVIRDINE	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Desoximetasone	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
EPSTEIN-BARR VIRUS ENVELOPE GLYCOPROTEIN GP340	NULL	NULL	TTD	2020.06.01	NULL	NULL	Docosanol	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
CALCIUM	NULL	NULL	TTD	2020.06.01	NULL	NULL	Etidronate Disodium	rxcui:9872	ETIDRONATE DISODIUM	TRUE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gatifloxacin	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gatifloxacin	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Halcinonide	rxcui:5084	HALCINONIDE	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Halobetasol Propionate	rxcui:41208	HALOBETASOL	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	Insulin-detemir	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Milrinone	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxtriphylline	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penicillin V Potassium	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
DNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifabutin	rxcui:55672	RIFABUTIN	TRUE	FALSE	FALSE
CANDIDA SQUALENE EPOXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Terbinafine	rxcui:37801	TERBINAFINE	TRUE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	NN-9926	NULL	NULL	NULL	NULL	NULL
ADENOSINE DEAMINASE	hgnc:186	ADA	TTD	2020.06.01	NULL	NULL	Ex vivo adenosine deaminase-transduced hematopoietic stem cell therapy	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005349192	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
ANGPTL3 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-ANGPTL3	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-AR	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	RH 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penicillin G Sodium	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.086861325	Enbrel	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
PHOSPHOINOSITIDE DEPENDENT PROTEIN KINASE-1	hgnc:8816	PDPK1	TTD	2020.06.01	NULL	1.591141552596802	AR-12	iuphar.ligand:8005	OSU-03012	FALSE	FALSE	FALSE
PRO-NEUREGULIN-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	GGF-2	chembl:CHEMBL3039542	CIMAGLERMIN ALFA	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.032412143	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
SARCOGLYCAN ALPHA	hgnc:10805	SGCA	TTD	2020.06.01	NULL	NULL	rAAV1.tMCK.human-alpha-sarcoglycan	NULL	NULL	NULL	NULL	NULL
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	NULL	TeloB-Vax	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-4/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	CDP323	drugbank:DB05092	CDP323	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hetacillin	rxcui:26797	HETACILLIN	TRUE	FALSE	FALSE
HEPATITIS C VIRUS MICRORNA MIR-122	NULL	NULL	TTD	2020.06.01	NULL	NULL	Miravirsen	ncit:C174858	MIRAVIRSEN	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.5000730593875666	N-(3,4-DICHLOROPHENYL)BENZAMIDE	chembl:CHEMBL560296	CHEMBL:CHEMBL560296	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	RPL-554	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD0914	ncit:C152962	ZOLIFLODACIN	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.8514757497680189	KW-6002	rxcui:2199015	ISTRADEFYLLINE	TRUE	FALSE	FALSE
PROTEIN TYROSINE PHOSPHATASE BETA	hgnc:9665	PTPRB	TTD	2020.06.01	NULL	19.69037671338543	AKB-9778	ncit:C152161	RAZUPROTAFIB	FALSE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	8.751278539282417	Farletuzumab	ncit:C61503	FARLETUZUMAB	FALSE	FALSE	FALSE
ITGA4 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATL1102	drugbank:DB04997	ATL1102	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.6908904109959803	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 6	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 8	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 1	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 10	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 3	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 7	NULL	NULL	NULL	NULL	NULL
SERUM AMYLOID P-COMPONENT	hgnc:584	APCS	TTD	2020.06.01	NULL	13.12691780892362	CPHPC	ncit:C153209	MIRIDESAP	FALSE	FALSE	FALSE
INTERLEUKIN-25	hgnc:13765	IL25	TTD	2020.06.01	NULL	8.751278539282415	ALX-0761	chembl:CHEMBL4298023	M-1095	FALSE	FALSE	FALSE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	1.346350544504987	ALX-0761	chembl:CHEMBL4298023	M-1095	FALSE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Moclobemide	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	2-Methoxyphenol	rxcui:5031	GUAIACOL	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	3,4-Dihydroxybenzaldehyde	drugbank:DB11268	PROTOCATECHUALDEHYDE	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	4-Hydroxy-2,5-dimethyl-3(2H)-furanone	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	4-Hydroxybenzoicacid	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	4-Hydroxybenzylalcohol	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ethylvanillin	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	GypensapogeninA	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	GypensapogeninB	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	IncarviatoneA	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperonal	rxcui:33753	PIPERONAL	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure1-Neonectrolide A	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure3-Lycojaponicumin A	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-11	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-11	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-14	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-14	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-9	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-9	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 7-Veratraldehyde	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C14	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C19	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C21	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C24	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C25	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C9	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	NULL	1-(biphenyl-4-yl-methyl)-1H-imidazole derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-(biphenyl-4-yl-methyl)-1H-imidazole derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	A-substituted phenylpropionic acid derivative 2	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cannabinoid quinone derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Crystalline anhydrous toluene derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure2-K	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure2-N	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-C	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-C	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazolidine dione crystalline derivative 1	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2012006391H3K9TSu	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2012106509Tenovin-6	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2012149608USYDS1	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-20	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-21	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-25	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-28	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-30	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-41	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-43	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-5	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-51	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-6	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Cyclopropyl-spiro piperidine derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 1	NULL	NULL	NULL	NULL	NULL
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydrothieno [2,3-e]indazole derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-EP20132578214 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2011000295210	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2011801300410	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2011803494010	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2012819831110	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US20138552206 5	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2011127048 32	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2011127048 34	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoxaline derivative 4	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoxaline derivative 6	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	6,6-fused nitrogenous heterocyclic compound 3	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-16a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-23b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-29a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-30a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-30b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36d	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36d	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-40	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Pyridoindole derivative 1	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Pyridoindole derivative 2	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl pyrazolamine derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-100	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-103	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-106	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20120277229 40(1.2)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20120277229 45(1.5)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20130053382 35(1-11)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2004087707	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2008079988	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2008107444	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2009153313	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2011137219 36(3-5)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2011137219 37(4-6)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2011137219 38(5-7)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 13	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 16	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 21	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 26	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 27	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 28	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 5	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 7	NULL	NULL	NULL	NULL	NULL
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAK-438	rxcui:2604576	VONOPRAZAN FUMARATE	TRUE	FALSE	FALSE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 3	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-10	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-18	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-20	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-23	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-29	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-30	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-31	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-45	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-59	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-60	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 21	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-EP20082149552C9	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-EP2149552diaminopyrimidines	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750M3	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750TG6-10-1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-WO2012177618M6	NULL	NULL	NULL	NULL	NULL
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	1.193356164447602	PF-04971729	rxcui:1992672	ERTUGLIFLOZIN	TRUE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	Tetra-azabenzo[e]azulene derivative 2	NULL	NULL	NULL	NULL	NULL
JNK-INTERACTING PROTEIN PEPTIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L3	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L3	NULL	NULL	NULL	NULL	NULL
JUN N TERMINAL KINASE	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-O1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-O3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-O3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-O3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P4	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P4	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P4	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P6	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P6	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P6	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140031349D	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140142115A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140309213B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2010129379A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2010129379B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2012058134B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013028474C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013039802A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013039802C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014099633D	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014150132A	NULL	NULL	NULL	NULL	NULL
ZINC FINGER-CONTAINING UBIQUITIN PEPTIDASE 1	hgnc:21224	ZUP1	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 3	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN TRANSPORTER	hgnc:10955	SLCO2A1	TTD	2020.06.01	NULL	NULL	PMID26099857-Compound-WO2011037610Formula(I)	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 60	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 60	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 64	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 67	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Pyrimidinone derivative 4	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	4-amino-3,5-di-substituted-thiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Alkyl sulfone derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Alkyl sulfone derivative 1	NULL	NULL	NULL	NULL	NULL
AURORA KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Diamidothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	NULL	Diamidothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Diamidothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE 1	hgnc:6840	MAP2K1	TTD	2020.06.01	NULL	NULL	Diamidothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 7	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indole-based analog 12	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Isosteric imidazolyl pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	Isosteric imidazolyl pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 4	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 5	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 7	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Ethylaminopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Ethylaminopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Isoxazoline derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Ketoheterocycle derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Spirocyclic diamine urea derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL SHIGA TOXIN 2 SUBUNIT B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Shigamabs	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	Imidazole derivative 10	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	Isothiazolone derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	3-acylidene-2-oxoindole derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Acyl piperidine derivative 3	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Azachalcone derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Benzotriazole derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Chloroacetyl ester derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Isothiocyanate derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Peptide analog 52	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-12	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-23	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-25	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-31	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-32	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 25	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 25	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 26	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 26	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 30	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 30	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 31	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 31	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 34	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 34	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 9	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 9	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Benzazepine derivative 3	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 13	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 6	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	L-piperazino-3-phenyl-indane derivative 1	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	L-piperazino-3-phenyl-indane derivative 1	NULL	NULL	NULL	NULL	NULL
DOPAMINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-piperazino-3-phenyl-indane derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 69	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 70	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 71	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 23	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 23	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 23	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 24	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 24	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 24	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 27	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 27	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 27	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 11	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 8	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	C-linked disaccharide biphenyl mannoside derivative 5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 12	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-105	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-106	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-107	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-108	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-10d	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-110	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-112	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-115	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-116	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-119	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-122	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-124	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-126a	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 9	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 9	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	PMID26666870-Compound-16	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure11Ala down	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9left02	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle03	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle04	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle06	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle07	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	3-(phenoxymethyl) benzylamine derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	3-(phenoxymethyl) benzylamine derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Dihydroxyfumaric acid derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Monoamine derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Nicotinyl hydroxamic acid derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	P-coumaric acid derivative 6	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-116	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-121	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-124	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-49	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-52	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-93	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 11	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 27	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 29	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 30	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 7	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 9	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Thiazolidine derivative 3	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	2,2-dimethylbenzopyran derivative 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 15	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 16	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 17	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 18	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 4	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 7	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 9	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN TESTIS-SPECIFIC PROTEIN	hgnc:1105	BRDT	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-102	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-102	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 3	hgnc:1104	BRD3	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-102	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-102	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-20	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-22	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-33	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR SIGNAL-REGULATED KINASE 5	hgnc:6880	MAPK7	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-33	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Piperazine urea derivative 3	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	PMID26936077-Compound-13	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Aryl cyclopropylamine derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Benzenamine derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Benzenamine derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 11	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 11	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 12	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 12	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-47	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1B	hgnc:21577	KDM1B	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-47	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-48	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1B	hgnc:21577	KDM1B	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-48	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-49	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-50	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-12	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-12	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-18	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-18	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-22	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 2	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 3	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 10	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Isoxazoles and isoxazoline derivative 2	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Amidopyrazole derivative 3	NULL	NULL	NULL	NULL	NULL
IL-1 RECEPTOR-ASSOCIATED KINASE 1	hgnc:6112	IRAK1	TTD	2020.06.01	NULL	NULL	Indazoletriazolephenyl derivative 1	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Indazoletriazolephenyl derivative 1	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Macrolactam derivative 1	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Macrolactam derivative 2	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Macrolactam derivative 3	NULL	NULL	NULL	NULL	NULL
IL-1 RECEPTOR-ASSOCIATED KINASE 1	hgnc:6112	IRAK1	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine and thienopyrimidine amide derivative 1	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine and thienopyrimidine amide derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [1,5-a]pyrimidin-7-yl derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [1,5-a]pyrimidin-7-yl derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27321640-Compound-59	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	PMID27321640-Compound-59	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	PMID27321640-Compound-75	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Purin-6-one derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-11	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-13	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-15	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR ALPHA	hgnc:9864	RARA	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-5	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 16	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Benzoic acid derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Cycloalkyl acid derivative 2	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 12	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 11	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Tetrazole acetic acid derivative 1	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-100	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-97	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	PMID27537201-Compound-Figure13b	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Poly-substituted miazine derivative 1	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-10	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-11	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-14	NULL	NULL	NULL	NULL	NULL
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	4.375639269641208	PEPEROMIN E	chembl:CHEMBL521941	PEPEROMIN E	FALSE	FALSE	FALSE
SPHINGOSINE KINASE	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-4	NULL	NULL	NULL	NULL	NULL
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	PMID27551786-Compound-IV	NULL	NULL	NULL	NULL	NULL
RECEPTOR-INTERACTING PROTEIN 1	hgnc:10019	RIPK1	TTD	2020.06.01	NULL	NULL	Tricyclic compound 10	NULL	NULL	NULL	NULL	NULL
RECEPTOR-INTERACTING PROTEIN 1	hgnc:10019	RIPK1	TTD	2020.06.01	NULL	NULL	Tricyclic compound 8	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Indole-based analog 10	NULL	NULL	NULL	NULL	NULL
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.048083948	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Indole-based analog 9	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine acetamide analog 4	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Isoquinoline carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-59	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-60	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-62	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-65	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine acetamide analog 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 5	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 7	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 10	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	FANGCHINOLINE	chembl:CHEMBL504256	FANGCHINOLINE	FALSE	FALSE	FALSE
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 10	NULL	NULL	NULL	NULL	NULL
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Pyridine derivative 18	NULL	NULL	NULL	NULL	NULL
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	NULL	Pyridine derivative 20	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 20	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyridine derivative 20	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	Pyridine derivative 20	NULL	NULL	NULL	NULL	NULL
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	NULL	Pyridine derivative 21	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 21	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyridine derivative 21	NULL	NULL	NULL	NULL	NULL
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.015286076	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	Pyridine derivative 21	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 4	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 16	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 16	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Aminobenzoxazole analog 1	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-3	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-Fomula2	NULL	NULL	NULL	NULL	NULL
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1250182648468916	6-HYDROXYMELATONIN	iuphar.ligand:1347	6-HYDROXYMELATONIN	FALSE	FALSE	FALSE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminooxazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminooxazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Aminooxazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Aminooxazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Aminopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclic cyanoethypypazole derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclic cyanoethypypazole derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-methylmethanesulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	N-methylmethanesulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	N-methylmethanesulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Example1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Example1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Example1	NULL	NULL	NULL	NULL	NULL
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.019889269	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Tricyclic compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic compound 3	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Imidazo pyridine derivative 4	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Oxazolo[3,4-a]pyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Oxazolo[3,4-a]pyrazine derivative 3	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Oxazolo[3,4-a]pyrazine derivative 4	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-6a	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002349337	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-20	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolodihydropyridine derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinolinyl pyrazinyl urea derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiadiazolidindione derivative 2	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiadiazolidindione derivative 3	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007727398	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	3-phenyl isoquinolin-1(2H) derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 2	hgnc:272	PARP2	TTD	2020.06.01	NULL	NULL	3-phenyl isoquinolin-1(2H) derivative 1	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	VINORELBIN DITARTRATE	chembl:CHEMBL538943	VINORELBINE TARTRATE	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 3	hgnc:273	PARP3	TTD	2020.06.01	NULL	NULL	3-phenyl isoquinolin-1(2H) derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	4-Carboxamido-isoindolinone derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	4-Carboxamido-isoindolinone derivative 4	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Dihydropyrido phthalazinone derivative 3	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Dihydropyrido phthalazinone derivative 4	NULL	NULL	NULL	NULL	NULL
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	ONONIN	chembl:CHEMBL465980	ONONIN	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Quinazolinedione derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Quinazolinedione derivative 3	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Tetra-hydro-quinoline derivative 1	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azaindole derivative 6	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azaindole derivative 7	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azole benzene derivative 3	NULL	NULL	NULL	NULL	NULL
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.030386384	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 10	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 11	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 4	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 7	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-129	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-131	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	4-aryl quinol derivative 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	4-aryl quinol derivative 4	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Acyl oxymethyl acrylamide ester derivative 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Binuclear gold(I) compound 3	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Golden phosphorous acetyletic compound 1	NULL	NULL	NULL	NULL	NULL
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.017751072	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
GLUTATHIONE REDUCTASE	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	Golden phosphorous acetyletic compound 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Golden phosphorous acetyletic compound 2	NULL	NULL	NULL	NULL	NULL
GLUTATHIONE REDUCTASE	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	Golden phosphorous acetyletic compound 2	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	PYRAZINOIC ACID	chembl:CHEMBL613	PYRAZINOIC ACID	FALSE	FALSE	FALSE
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Golden phosphorous acetyletic compound 3	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Metal complex derivative 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Metal complex derivative 3	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Palmarumycin derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Palmarumycin derivative 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-17	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Central azetidine derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Diazepinone derivative 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Diazepinone derivative 5	NULL	NULL	NULL	NULL	NULL
PBK	hgnc:18282	PBK	DTC	9/2/20	NULL	0.1312691780892362	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Ethynyl compound 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Ethynyl compound 7	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Imidazopyridine and triazolopyridine compound 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Imidazopyridine and triazolopyridine compound 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	N-alkylamide derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	PMID28067079-Compound-95	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyridine derivative 15	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyridine derivative 17	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-pyrazolopyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-pyrazolopyrazine derivative 5	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 7	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 11	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 3	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 4	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 7	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20100022547C83	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20100022547C86	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-WO2009018344C79	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	ZOMEPIRAC SODIUM	rxcui:58331	ZOMEPIRAC SODIUM	TRUE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	VX-944	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32f	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32f	NULL	NULL	NULL	NULL	NULL
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.049723174	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32h	NULL	NULL	NULL	NULL	NULL
PRKCB	hgnc:9395	PRKCB	DTC	9/2/20	NULL	0.8204323630577265	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.010170977	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32h	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32j	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32j	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32t	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32t	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33c	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	PMID28117607-Compound-21	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	PMID28117607-Compound-5	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	PMID28117607-Compound-6	NULL	NULL	NULL	NULL	NULL
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004972317	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 6	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 6	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	Cyclopenta[d]pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	Cyclopenta[d]pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 4	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-36	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-39	NULL	NULL	NULL	NULL	NULL
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.2692701089009974	PH-797804	drugbank:DB07941	PH-797804	FALSE	FALSE	FALSE
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-40	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-42	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-43	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-50	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-51	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-53	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-20	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-23	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-24	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-27	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 87	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridine and pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrido/pyrrolo-fused pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	4-(2-cyclohexylethoxy) aniline derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	4-(2-cyclohexylethoxy) aniline derivative 4	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazole derivative 2	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	CHLORFENAPYR	chembl:CHEMBL1869551	CHLORFENAPYR	FALSE	FALSE	FALSE
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazole derivative 3	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-3	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-37	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-37	NULL	NULL	NULL	NULL	NULL
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.010614043	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-40	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-40	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-41	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-41	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DUAL DLG AND ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-57	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-57	NULL	NULL	NULL	NULL	NULL
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.024861587	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
KEAP1-NRF2[DUAL DLG AND ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-58	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-58	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-8	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-8	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 1	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 3	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridyl compound 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Pyridyl compound 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Thiazole derivative 2	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	PMID28460551-Compound-6	NULL	NULL	NULL	NULL	NULL
ALOX5	hgnc:435	ALOX5	DTC	9/2/20	NULL	3.088686543276147	6-PENTYLSALICYLIC ACID	chembl:CHEMBL502496	CHEMBL:CHEMBL502496	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	NULL	PMID28460551-Compound-6	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	Benzoimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	Benzoimidazole derivative 2	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	PMID28594589-Compound-TABLE3C12	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme27LeucettamineB	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme8NCGC-00010037	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme8NCGC-00185981	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT9851	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT9851	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-37	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-39	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-46	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-53	NULL	NULL	NULL	NULL	NULL
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.04339477	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-55	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-58	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-64	NULL	NULL	NULL	NULL	NULL
CASPASE-1	hgnc:1499	CASP1	TTD	2020.06.01	NULL	NULL	Ac-YVAD-cmk	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	Isoquinolone derivative 1	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	N-(benzimidazole/indole) benzoic acid derivative 2	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	N-(indolylcarbonyl)-piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	Nitrogen/sulfur-substituted estrene derivative 1	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 10	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 13	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 13	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Triazole derivative 5	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidine-benzoxazin-3(4H)-one derivative 1	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidinyl-piperazine derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 9	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 9	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 1	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 1	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 2	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 2	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 2	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 4	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 4	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL LIPASE ALPHA	hgnc:1165	DAGLA	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-15	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-15	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-15	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-4	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-5	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-7c	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-76	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-76	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Pyridino tricyclic compound 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Sulfamic acid ester derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Sulfamoylamide derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 8	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Thieno[2,3-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-11	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-14	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-18	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-2	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-20	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-24	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-25	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-32	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-33	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-42	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-8	NULL	NULL	NULL	NULL	NULL
G-PROTEIN COUPLED BILE ACID RECEPTOR 1	hgnc:19680	GPBAR1	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-8	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-INT767	NULL	NULL	NULL	NULL	NULL
G-PROTEIN COUPLED BILE ACID RECEPTOR 1	hgnc:19680	GPBAR1	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-INT767	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-13	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-13	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-13	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-19	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-19	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 10	hgnc:18128	HDAC10	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 11	hgnc:19086	HDAC11	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.028771327	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 9	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-22	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-22	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 11	hgnc:19086	HDAC11	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 5	hgnc:14068	HDAC5	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 5	hgnc:14068	HDAC5	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 9	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-31	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 10	hgnc:18128	HDAC10	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 11	hgnc:19086	HDAC11	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-47b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-52	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 10	hgnc:18128	HDAC10	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 11	hgnc:19086	HDAC11	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 5	hgnc:14068	HDAC5	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 9	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-62	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-71a	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 17	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30074415-Compound-19	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30074415-Compound-GS3	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfonamide-thiadiazole derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-oxadiazole derivative 6	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-oxadiazole derivative 7	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3,4-oxadiazole derivative 5	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example43	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example47	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example52	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example60	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-LDT8	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-LDT8	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-LDT8	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-LDT8	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Fused aryl carbocycle derivative 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Fused aryl carbocycle derivative 2	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Fused aryl carbocycle derivative 9	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 4	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazinyl methyl quinazolinone derivative 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazinyl methyl quinazolinone derivative 2	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazinyl norbenzomorphane compound 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazinyl norbenzomorphane compound 4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-28	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-53	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-56	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-1	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-22a	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-40	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-US20170128558	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-US20179642901	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2009082440	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2013148426	NULL	NULL	NULL	NULL	NULL
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ciprofloxacin XR	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ciprofloxacin XR	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clonazepam	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloserine	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
RIBONUCLEOTIDE REDUCTASE	hgnc:581	APBB1	TTD	2020.06.01	NULL	NULL	G-207 virus construct	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	Dobutamine	rxcui:3616	DOBUTAMINE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Emtricitabine	rxcui:276237	EMTRICITABINE	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Felbamate	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.116943588	Hydroxyflutamide	ncit:C63948	HYDROXYFLUTAMIDE	FALSE	FALSE	FALSE
BACTERIAL FATTY ACID SYNTHETASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoniazid	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ketobemidone	ncit:C80583	KETOBEMIDONE	FALSE	FALSE	FALSE
PHOSPHATE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lanthanum carbonate	rxcui:234416	LANTHANUM CARBONATE	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Linagliptin	rxcui:1100699	LINAGLIPTIN	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Memantine	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Metergolin	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	Pachycarpine	NULL	NULL	NULL	NULL	NULL
INFLUENZA NEURAMINIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peramivir	rxcui:1598096	PERAMIVIR ANHYDROUS	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Prinomastat	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.022730594	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NEUROPILIN-1	hgnc:8004	NRP1	TTD	2020.06.01	NULL	17.50255707856483	Pegaptanib	rxcui:498509	PEGAPTANIB	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-7	hgnc:7174	MMP7	TTD	2020.06.01	NULL	1.071585127259071	Prinomastat	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.7395446652914718	Propylhexedrine	rxcui:8792	PROPYLHEXEDRINE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
PI3K/AKT/MTOR PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulphadoxine	chembl:CHEMBL244800	SULPHADOXINE	FALSE	FALSE	FALSE
PLASMODIUM DIHYDROOROTATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Teriflunomide	rxcui:1310520	TERIFLUNOMIDE	TRUE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ximelegatran	NULL	NULL	NULL	NULL	NULL
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	NULL	ABT-110	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-239	iuphar.ligand:1218	ABT-239	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	FLAVANONE	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
CD40L RECEPTOR	hgnc:11919	CD40	TTD	2020.06.01	NULL	4.375639269641208	APX005M	ncit:C123734	SOTIGALIMAB	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	0.097236428	Verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	BI-11634	NULL	NULL	NULL	NULL	NULL
FGFR4 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BLU-554	ncit:C123826	FISOGATINIB	FALSE	FALSE	TRUE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	NULL	Drug 2849330	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 9	NULL	NULL	TTD	2020.06.01	NULL	NULL	E2027	chembl:CHEMBL4650368	IRSENONTRINE	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Englitazone sodium	ncit:C72759	ENGLITAZONE SODIUM	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.006682916	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	ITI-214	ncit:C177065	LENRISPODUN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	KUL-7211	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	KUL-7211	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C DELTA	hgnc:9399	PRKCD	TTD	2020.06.01	NULL	4.922594178346359	KAI-9803	ncit:C101384	DELCASERTIB	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BILR-355	NULL	NULL	NULL	NULL	NULL
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	FK-143	chembl:CHEMBL25083	CHEMBL:CHEMBL25083	FALSE	FALSE	FALSE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	GLPG-0634	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	HM-78136B	NULL	NULL	NULL	NULL	NULL
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	Interferon-alpha lozenge	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.1930429089547591	Vabicaserin	ncit:C132725	VABICASERIN	FALSE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	4.039051633514961	Tonabersat	ncit:C97277	TONABERSAT	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	NLG8189	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.3029288725136221	M100907	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	0.9546849315580819	LX-4211	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.6226206075378794	Pridopidine	ncit:C170349	PRIDOPIDINE	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Remacemide	ncit:C152183	REMACEMIDE	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SUVN-G3031	drugbank:DB14835	SUVN-G3031	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Synthetic conjugated estrogen	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	TG101348	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
SODIUM/HYDROGEN EXCHANGER 1	hgnc:11071	SLC9A1	TTD	2020.06.01	NULL	NULL	Zoniporide hydrochloride	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	CART-EGFRvIII T cells	NULL	NULL	NULL	NULL	NULL
C-X-C CHEMOKINE RECEPTOR TYPE 1	hgnc:6026	CXCR1	TTD	2020.06.01	NULL	5.000730593875666	Reparixin	ncit:C66515	REPARIXIN	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	CS-3030	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	FR167653	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	CILOSTAMIDE	ncit:C76315	CILOSTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2464	hgnc:3861	FRA16E	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8284	iuphar.ligand:8284	CPP-115	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.015608701	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:1878	ncbigene:1878	E11S	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:9244	iuphar.ligand:9244	UTOMILUMAB	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:8436	iuphar.ligand:8436	LP-211	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.045265234	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.004666519	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.014601688	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:95	ncit:C74388	REPINOTAN	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.00644424	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.3163112725041837	IUPHAR.LIGAND:131	iuphar.ligand:131	[3H]GR 125,743	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.048083948	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.020164236	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:131	iuphar.ligand:131	[3H]GR 125,743	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.2524407270946851	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.029766254	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:8422	iuphar.ligand:8422	5-BODMT	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1117184494376478	IUPHAR.LIGAND:121	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.020836377	IUPHAR.LIGAND:7241	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:165	iuphar.ligand:165	MK-212	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.024130364	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:188	iuphar.ligand:188	RS-127445	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.073540156	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:9444	ncit:C166572	INTEPIRDINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.009174851	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.076765601	IUPHAR.LIGAND:277	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.043866058	IUPHAR.LIGAND:87	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:122	iuphar.ligand:122	DIPROPYL-5-CT	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.005297384	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:1264	hgnc:2155	CNN1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10670	iuphar.ligand:10670	COMPOUND 2E [PMID: 31900320]	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:8009	iuphar.ligand:8009	PHT-427	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.024767769	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.032694689	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:493	rxcui:720825	SILODOSIN	TRUE	FALSE	FALSE
NCBIGENE:1921	hgnc:19679	AAK1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11895	iuphar.ligand:11895	COMPOUND 13 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:6374	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	PYRAZINOIC ACID	chembl:CHEMBL613	PYRAZINOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:10061	iuphar.ligand:10061	AZELAPRAG	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:6312	iuphar.ligand:6312	CYCLOUREA APELIN-12 (1-7)	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.028078969	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:12564	iuphar.ligand:12564	ASC06-IGG1	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.078136416	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NCBIGENE:1245	ncbigene:1245	CMR1A	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:5107	iuphar.ligand:5107	2(S)-AMINO-6-BORONOHEXANOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1244	hgnc:53	ABCC2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5107	iuphar.ligand:5107	2(S)-AMINO-6-BORONOHEXANOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.251232877	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.04339477	BRADANICLINE	ncit:C169814	BRADANICLINE	FALSE	FALSE	FALSE
NCBIGENE:685	hgnc:1121	BTC	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:4116	iuphar.ligand:4116	A-317567	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:11472	iuphar.ligand:11472	JNJ-799760	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:10443	iuphar.ligand:10443	COMPOUND 10 [PMID: 31306001]	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:10443	iuphar.ligand:10443	COMPOUND 10 [PMID: 31306001]	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001827244	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:398	iuphar.ligand:398	MRS1086	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:437	iuphar.ligand:437	AS101	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:427	iuphar.ligand:427	CPX	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:5616	iuphar.ligand:5616	ATL802	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.5413161983061289	IUPHAR.LIGAND:11706	iuphar.ligand:11706	COMPOUND 6C [PMID: 34435786]	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1804387327687096	IUPHAR.LIGAND:10351	iuphar.ligand:10351	LUF7602	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:5616	iuphar.ligand:5616	ATL802	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1804387327687096	IUPHAR.LIGAND:423	iuphar.ligand:423	N(6)-CYCLOHEXYLADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:386	iuphar.ligand:386	DPCPX	FALSE	FALSE	FALSE
MMP12	hgnc:7158	MMP12	DTC	9/2/20	NULL	1.296485709523321	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.013087655	IUPHAR.LIGAND:9927	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:8863	ncit:C127116	DUBERMATINIB	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:7455	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:560	rxcui:10368	TERBUTALINE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.025244073	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:7543	rxcui:1546059	OLODATEROL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:7353	rxcui:1424884	VILANTEROL	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.05293112	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	SULMAZOLE	ncit:C84188	SULMAZOLE	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:6159	iuphar.ligand:6159	12-HYDROXYHEPTADECATRIENOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:571	ncit:C81654	TERTATOLOL	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	0.026045472	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
NCBIGENE:1941	hgnc:18041	BMP2K	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:11893	iuphar.ligand:11893	COMPOUND 6 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9129	iuphar.ligand:9129	L779450	FALSE	FALSE	FALSE
NCBIGENE:3210	hgnc:5110	HOXB@	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12232	iuphar.ligand:12232	BAY-069	FALSE	FALSE	FALSE
C3AR1	hgnc:1319	C3AR1	DTC	9/2/20	NULL	10.50153424713889	SB-290157	iuphar.ligand:3529	SB290157	FALSE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:7147	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
NCBIGENE:2599	hgnc:1375	CA4	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:6792	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.03505185	PROPACHLOR	chembl:CHEMBL1394829	PROPACHLOR	FALSE	FALSE	FALSE
NCBIGENE:1624	hgnc:2692	DBIP1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8628	iuphar.ligand:8628	COMPOUND 4 [PMID: 12408711]	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE	chembl:CHEMBL1371413	2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:9473	iuphar.ligand:9473	RONACALERET	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	DTC	9/2/20	NULL	0.3547815624033412	ZAMIFENACIN	ncit:C66682	ZAMIFENACIN	FALSE	FALSE	FALSE
NCBIGENE:2343	ncbigene:2343	FNTBL1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:10746	iuphar.ligand:10746	VBY-825	FALSE	FALSE	FALSE
NCBIGENE:2344	hgnc:2528	CTSC	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11179	iuphar.ligand:11179	ICATCXPZ-01	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
NCBIGENE:2346	hgnc:3788	FOLH1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:8634	iuphar.ligand:8634	COMPOUND 3 [PMID: 8410973]	FALSE	FALSE	FALSE
NCBIGENE:2472	hgnc:3882	FRA20B	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8988	rxcui:2362167	OPICAPONE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.018081154	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:10272	iuphar.ligand:10272	GAT211	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:10690	iuphar.ligand:10690	JD5037	FALSE	FALSE	FALSE
SIRT5	hgnc:14933	SIRT5	DTC	9/2/20	NULL	0.364636606	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:864	rxcui:9800	SINCALIDE	TRUE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:9233	ncit:C87598	SURINABANT	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:860	iuphar.ligand:860	CCK-33	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	0.4039051633514962	IUPHAR.LIGAND:759	iuphar.ligand:759	CCL7	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:3536	iuphar.ligand:3536	UCB35625	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	N-PHENETHYLCINNAMAMIDE	chembl:CHEMBL1305393	CHEMBL:CHEMBL1305393	FALSE	FALSE	FALSE
NCBIGENE:63	hgnc:136	ACTBP3	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12765	iuphar.ligand:12765	PF-07054894	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:11597	iuphar.ligand:11597	BMS-753426	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.053253216	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
NCBIGENE:3010	hgnc:4720	H1-6	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:9950	iuphar.ligand:9950	LILOTOMAB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	OSAJIN	chembl:CHEMBL238188	OSAJIN	FALSE	FALSE	FALSE
NCBIGENE:2786	hgnc:4407	GNG4	GuideToPharmacology	2024.1	antibody	6.563458904461812	IUPHAR.LIGAND:8266	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.011810092	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
NCBIGENE:2995	hgnc:4704	GYPC	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:10208	rxcui:2043283	IBALIZUMAB	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002258977	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
NCBIGENE:2340	hgnc:2097	CMA1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:6563	iuphar.ligand:6563	JNJ-10311795	FALSE	FALSE	FALSE
NCBIGENE:2338	hgnc:3308	CELA1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:7871	rxcui:1102261	TELAPREVIR	TRUE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.4861821410712454	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
NCBIGENE:1255	ncbigene:1255	CNA1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9259	iuphar.ligand:9259	SGC2085	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	antibody	0.9907107780319716	IUPHAR.LIGAND:9107	iuphar.ligand:9107	CABIRALIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:5689	iuphar.ligand:5689	JNJ-28312141	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:9000	iuphar.ligand:9000	(R)-ARN2508	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:4820	rxcui:4331	FENOPROFEN	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.2206204673768676	IUPHAR.LIGAND:4795	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:7185	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10335	iuphar.ligand:10335	ASTRESSIN 2B	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:912	iuphar.ligand:912	CORTICOTROPHIN-RELEASING HORMONE	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5955	drugbank:DB08325	2-({6-[(3-CHLOROPHENYL)AMINO]-9-ISOPROPYL-9H-PURIN-2-YL}AMINO)ETHANOL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.007479725	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	N-(2-PYRIDYLMETHYL)PHENYLAMINE	chembl:CHEMBL402456	CHEMBL:CHEMBL402456	FALSE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8733	iuphar.ligand:8733	COMPOUND 4 [PMID: 26191369]	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
NCBIGENE:2636	hgnc:4185	GBX1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8261	iuphar.ligand:8261	(S)-DRF-1042	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.002354393	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.05853698	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	ALPHA-TERTHIENYL	chembl:CHEMBL90017	ALPHA-TERTHIENYL	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:937	iuphar.ligand:937	SKF-76783	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:9216	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	modulator	1.346350544504987	IUPHAR.LIGAND:11938	iuphar.ligand:11938	LY3154885	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.087512785	IUPHAR.LIGAND:7124	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:8436	iuphar.ligand:8436	LP-211	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:8435	iuphar.ligand:8435	LP-44	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.026927011	IUPHAR.LIGAND:963	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.050007306	IUPHAR.LIGAND:958	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.033338204	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.071341945	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:944	iuphar.ligand:944	SKF-83566	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.058341857	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8165	iuphar.ligand:8165	COMPOUND 68 [PMID: 24900699]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:5917	iuphar.ligand:5917	AG 9	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:11580	iuphar.ligand:11580	AZ5104	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12952	iuphar.ligand:12952	EXAMPLE 10 [CN110740999A]	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.066047385	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:10124	iuphar.ligand:10124	DUAL SEH/FAAH INHIBITOR 11	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012325744	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.2625383561784725	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	NULL	0.5000730593875666	IUPHAR.LIGAND:5059	iuphar.ligand:5059	TGF&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.2430910705356226	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NONIVAMIDE	rxcui:31945	NONIVAMIDE	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.4773424657790409	IUPHAR.LIGAND:1894	ncit:C79571	CLOPROSTENOL	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	0.4546118721705151	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.05293112	IUPHAR.LIGAND:5692	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:6011	ncit:C66212	MUBRITINIB	FALSE	FALSE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:12612	iuphar.ligand:12612	PIROTINIB	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9662	iuphar.ligand:9662	PYROTINIB	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:9922	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	NULL	0.4526523382387456	IUPHAR.LIGAND:4873	iuphar.ligand:4873	BETACELLULIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.005753635	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:6700	ncit:C76959	PRINABEREL	FALSE	FALSE	FALSE
NCBIGENE:622	hgnc:1027	BDH1	GuideToPharmacology	2024.1	agonist	0.1810609352954982	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIDODECYL-DIMETHYL-AMMONIUM BROMIDE	chembl:CHEMBL332670	CHEMBL:CHEMBL332670	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12286	ncit:C79486	CLAZOSENTAN	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:10070	ncit:C174728	APROCITENTAN	TRUE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:12286	ncit:C79486	CLAZOSENTAN	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.022062047	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:10644	ncit:C169848	CILOFEXOR	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:2742	iuphar.ligand:2742	22R-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	NULL	0.5834185692854945	IUPHAR.LIGAND:4534	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
NCBIGENE:871	hgnc:1546	SERPINH1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4573	iuphar.ligand:4573	THREO-3-METHYLGLUTAMATE	FALSE	FALSE	FALSE
NCBIGENE:868	hgnc:1542	CBLB	GuideToPharmacology	2024.1	NULL	0.9546849315580819	IUPHAR.LIGAND:4698	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	PROPACHLOR	chembl:CHEMBL1394829	PROPACHLOR	FALSE	FALSE	FALSE
NCBIGENE:2826	hgnc:4474	CCR10	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8028	iuphar.ligand:8028	LB42908	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:3164	drugbank:DB06548	MINODRONIC ACID	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	8-FLUOROTRYPTANTHRIN	chembl:CHEMBL1098875	CHEMBL:CHEMBL1098875	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:4083	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4327	iuphar.ligand:4327	TPA023	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	agonist	0.078722146	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	3,5-DIPHENYLISOXAZOLE	chembl:CHEMBL1374535	3,5-DIPHENYLISOXAZOLE	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:4301	iuphar.ligand:4301	RY024	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4094	iuphar.ligand:4094	&ALPHA;3IA	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
NCBIGENE:416	hgnc:721	ARSF	GuideToPharmacology	2024.1	blocker	0.5527123287967842	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.075442056	IUPHAR.LIGAND:4192	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.3017682254924971	IUPHAR.LIGAND:4366	iuphar.ligand:4366	[3H]CGS8216	FALSE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.056622219	Anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
NCBIGENE:415	hgnc:719	ARSL	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6074	iuphar.ligand:6074	M1160	FALSE	FALSE	FALSE
NCBIGENE:1268	hgnc:2159	CNR1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:6960	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
NCBIGENE:247	hgnc:434	ALOX15B	GuideToPharmacology	2024.1	agonist	0.3804903712731485	IUPHAR.LIGAND:2270	rxcui:236901	SOMATORELIN	FALSE	FALSE	FALSE
NCBIGENE:247	hgnc:434	ALOX15B	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:3857	iuphar.ligand:3857	BIM28011	FALSE	FALSE	FALSE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:9135	iuphar.ligand:9135	MK-0893	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:4070	drugbank:DB02966	FLUORO-WILLARDIINE	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:4070	drugbank:DB02966	FLUORO-WILLARDIINE	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.375054795	IUPHAR.LIGAND:4288	rxcui:8351	PIRACETAM	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:9649	ncit:C170007	FOSDAGROCORAT	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4089	iuphar.ligand:4089	[3H]DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4243	iuphar.ligand:4243	LY233053	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:4080	iuphar.ligand:4080	[3H]CGS19755	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.065145994	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	blocker	0.130291988	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4088	iuphar.ligand:4088	[3H]MDL105519	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1165	iuphar.ligand:1165	[125I][TYR5,DALA6,NMELEU7,PRO9-NET]GNRH	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:5797	drugbank:DB02556	D-PHENYLALANINE	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.07699072	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.027276712	IUPHAR.LIGAND:2949	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5720	iuphar.ligand:5720	(R)-N-OLEOYLTYROSINOL	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:4028	iuphar.ligand:4028	LYSOPHOSPHATIDYLINOSITOL	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:4029	iuphar.ligand:4029	2-ARACHIDONOYLGLYCEROLPHOSPHOINOSITOL	FALSE	FALSE	FALSE
NCBIGENE:112	hgnc:237	ADCY6	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:114	hgnc:239	ADCY8	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:10571	iuphar.ligand:10571	CARTPT (76-96)	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	modulator	2.763561643983921	IUPHAR.LIGAND:11208	iuphar.ligand:11208	DIM	FALSE	FALSE	FALSE
NCBIGENE:122	ncbigene:122	ADFN	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:2907	iuphar.ligand:2907	KI16425	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.1172046232939609	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11415	iuphar.ligand:11415	ZABEDOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12510	iuphar.ligand:12510	GLPG2534	FALSE	FALSE	FALSE
NCBIGENE:1723	hgnc:2867	DHODH	GuideToPharmacology	2024.1	antibody	1.381780822	IUPHAR.LIGAND:8258	iuphar.ligand:8258	ANIFROLUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	0.4948366922735607	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:1695	hgnc:6008	IL2RA	GuideToPharmacology	2024.1	antibody	1.029562181092049	IUPHAR.LIGAND:6880	rxcui:190353	DACLIZUMAB	TRUE	TRUE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:12466	iuphar.ligand:12466	6-METHYLFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:682	hgnc:1116	BSG	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:12456	iuphar.ligand:12456	SINIGRIN	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:10298	iuphar.ligand:10298	NARINGENIN	FALSE	FALSE	FALSE
NCBIGENE:682	hgnc:1116	BSG	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:6649	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:12471	iuphar.ligand:12471	3-METHYLHEXANAL	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:12498	rxcui:17354	ALLOIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.1084869240406911	Brivaracetam	rxcui:1739745	BRIVARACETAM	TRUE	FALSE	FALSE
NCBIGENE:677	hgnc:1107	ZFP36L1	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:12459	iuphar.ligand:12459	AMAROGENTIN	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:12459	iuphar.ligand:12459	AMAROGENTIN	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:11410	ncit:C175770	DEURUXOLITINIB	FALSE	FALSE	FALSE
NCBIGENE:664	hgnc:1084	BNIP3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12429	iuphar.ligand:12429	S6821	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:8476	iuphar.ligand:8476	AZ960	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:7971	iuphar.ligand:7971	XL019	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:9432	iuphar.ligand:9432	PF-06263276	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:9697	ncit:C152385	SOLCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.076765601	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:9803	iuphar.ligand:9803	SAR-20347	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:11878	drugbank:DB16756	IVARMACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:10148	iuphar.ligand:10148	JAK INHIBITOR 17B	FALSE	FALSE	FALSE
NCBIGENE:2866	hgnc:4500	GPR42	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8488	iuphar.ligand:8488	COMPOUND 3 [PMID: 23849879]	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:9803	iuphar.ligand:9803	SAR-20347	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:9559	iuphar.ligand:9559	RITLECITINIB	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:1652	iuphar.ligand:1652	U50488	FALSE	FALSE	FALSE
NCBIGENE:968	hgnc:1693	CD68	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:4742	rxcui:33770	PIRETANIDE	FALSE	FALSE	FALSE
NCBIGENE:2849	hgnc:4481	GPR26	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:8323	iuphar.ligand:8323	MONALIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.018012923	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	modulator	3.281729452230906	IUPHAR.LIGAND:11978	iuphar.ligand:11978	AZD4625	FALSE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	activator	0.9376369863516875	IUPHAR.LIGAND:2503	rxcui:1362698	CHLOROFORM	TRUE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	activator	0.101562227	IUPHAR.LIGAND:1013	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	blocker	0.8334550989792776	IUPHAR.LIGAND:2316	iuphar.ligand:2316	LEIUROTOXIN I	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:2325	iuphar.ligand:2325	P05	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	0.06757744	IUPHAR.LIGAND:2330	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	0.2386712328895204	IUPHAR.LIGAND:357	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:441	hgnc:6269	KCNJ8	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:6848	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.008854582	Quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:573	hgnc:937	BAG1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7689	iuphar.ligand:7689	&GAMMA;-KTX1.7	FALSE	FALSE	FALSE
NCBIGENE:543	hgnc:880	ALDH7A1P3	GuideToPharmacology	2024.1	blocker	0.7292732116068681	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.020257589	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
NCBIGENE:547	hgnc:888	KIF1A	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7759	iuphar.ligand:7759	RY796	FALSE	FALSE	FALSE
NCBIGENE:545	hgnc:882	ATR	GuideToPharmacology	2024.1	blocker	0.097236428	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:11207	iuphar.ligand:11207	DPO-1	FALSE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2911	iuphar.ligand:2911	FARNESYL MONOPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:5704	iuphar.ligand:5704	PP-242	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:8839	iuphar.ligand:8839	TORIN 2	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.081407242	IUPHAR.LIGAND:12616	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8108	iuphar.ligand:8108	DENFIVONTINIB	FALSE	FALSE	FALSE
NCBIGENE:1572	hgnc:2632	CYP2F1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8557	iuphar.ligand:8557	COMPOUND 14 [PMID: 23634668]	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12320	iuphar.ligand:12320	SLC-391	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6231	iuphar.ligand:6231	COMPOUND 22A [PMID: 21688779]	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:3956	iuphar.ligand:3956	VU0361737	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:1417	iuphar.ligand:1417	CHPG	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.2625383561784725	Sulfisoxazole	rxcui:10207	SULFISOXAZOLE	TRUE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	0.5000730593875667	IUPHAR.LIGAND:1365	iuphar.ligand:1365	(1S,3R)-ACPD	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	FDA	10-Apr-24	NULL	10.74020548002842	Tezacaftor	rxcui:1999382	TEZACAFTOR	TRUE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1407	iuphar.ligand:1407	(S)-3,4-DCPG	FALSE	FALSE	FALSE
NCBIGENE:2099	hgnc:3467	ESR1	GuideToPharmacology	2024.1	inhibitor	0.1226814748497534	IUPHAR.LIGAND:11896	iuphar.ligand:11896	COMPOUND 14 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:2100	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:12937	iuphar.ligand:12937	PCC0208017	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:1415	iuphar.ligand:1415	MPPG	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:1399	iuphar.ligand:1399	[3H]LY341495	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2869	iuphar.ligand:2869	CORTICOSTERONE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	FDA	10-Apr-24	NULL	0.096264064	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:2103	hgnc:3473	ESRRB	GuideToPharmacology	2024.1	inhibitor	0.9723642821424908	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:3024	hgnc:4715	H1-1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:12601	ncit:C1146	LONIDAMINE	FALSE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:9375	iuphar.ligand:9375	VTX-11E	FALSE	FALSE	FALSE
DMD	hgnc:2928	DMD	FDA	10-Apr-24	NULL	15.00219178	Eteplirsen	rxcui:1810569	ETEPLIRSEN	TRUE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5997	iuphar.ligand:5997	JNK INHIBITOR V	FALSE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:9210	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:2072	hgnc:3436	ERCC4	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9355	iuphar.ligand:9355	GNE-3511	FALSE	FALSE	FALSE
NCBIGENE:2072	hgnc:3436	ERCC4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9990	iuphar.ligand:9990	GNE-8505	FALSE	FALSE	FALSE
NCBIGENE:1634	hgnc:2705	DCN	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8259	iuphar.ligand:8259	CM-352	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.2224901323546377	IUPHAR.LIGAND:7823	iuphar.ligand:7823	AZD6605	FALSE	FALSE	FALSE
NCBIGENE:3183	hgnc:5035	HNRNPC	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11541	iuphar.ligand:11541	SR-0813	FALSE	FALSE	FALSE
NCBIGENE:1631	hgnc:7174	MMP7	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8636	iuphar.ligand:8636	COMPOUND 15 [PMID: 22017539]	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:12057	iuphar.ligand:12057	TP0556351	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:6526	drugbank:DB08388	5-(2-ETHOXYETHYL)-5-[4-(4-FLUOROPHENOXY)PHENOXY]PYRIMIDINE-2,4,6(1H,3H,5H)-TRIONE	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8291	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.1262203635473425	IUPHAR.LIGAND:339	iuphar.ligand:339	WIN 51,708	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.055271233	IUPHAR.LIGAND:288	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.078958904	IUPHAR.LIGAND:297	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.1105424657593568	IUPHAR.LIGAND:342	iuphar.ligand:342	BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:3274	iuphar.ligand:3274	VU0255035	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:321	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.1944728564284981	IUPHAR.LIGAND:1347	iuphar.ligand:1347	6-HYDROXYMELATONIN	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:7783	iuphar.ligand:7783	UCM 454	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1348	iuphar.ligand:1348	GR 128107	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1362	iuphar.ligand:1362	S26131	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:11196	iuphar.ligand:11196	ICOA-13	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1351	iuphar.ligand:1351	LY 156735	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.096167896	IUPHAR.LIGAND:7563	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	modulator	0.5770073762164231	IUPHAR.LIGAND:9160	iuphar.ligand:9160	BMS-986124	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:1641	iuphar.ligand:1641	NALTRINDOLE	FALSE	FALSE	FALSE
NCBIGENE:3112	hgnc:4937	HLA-DOB	GuideToPharmacology	2024.1	antibody	1.544343271638073	IUPHAR.LIGAND:10738	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.1182605208011137	IUPHAR.LIGAND:7321	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10314	iuphar.ligand:10314	SELITRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:5685	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
NCBIGENE:463	hgnc:777	ZFHX3	GuideToPharmacology	2024.1	modulator	2.917092846427472	IUPHAR.LIGAND:3992	iuphar.ligand:3992	LY2087101	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:3979	iuphar.ligand:3979	[3H]CYTISINE	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:3490	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:2118	iuphar.ligand:2118	R396	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:2123	ncit:C84001	NEPADUTANT	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2105	iuphar.ligand:2105	R-486	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1492	iuphar.ligand:1492	NEUROPEPTIDE S	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:1580	iuphar.ligand:1580	SR142948A	FALSE	FALSE	FALSE
NCBIGENE:1873	hgnc:11918	TNFRSF4	GuideToPharmacology	2024.1	antibody	3.500511415712966	IUPHAR.LIGAND:9245	iuphar.ligand:9245	VONLEROLIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	modulator	2.625383561784724	IUPHAR.LIGAND:8936	iuphar.ligand:8936	COMPOUND 3 [PMID: 26191365]	FALSE	FALSE	FALSE
NCBIGENE:2136	hgnc:16059	PAK4	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:8938	iuphar.ligand:8938	FRAX486	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8938	iuphar.ligand:8938	FRAX486	FALSE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.2044691247495891	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	modulator	3.281729452230906	IUPHAR.LIGAND:8936	iuphar.ligand:8936	COMPOUND 3 [PMID: 26191365]	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:1703	iuphar.ligand:1703	SB-334867	FALSE	FALSE	FALSE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:8938	iuphar.ligand:8938	FRAX486	FALSE	FALSE	FALSE
NCBIGENE:2135	hgnc:3516	EXTL2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8938	iuphar.ligand:8938	FRAX486	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	agonist	0.5527123287967842	IUPHAR.LIGAND:1757	iuphar.ligand:1757	BZATP	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	0.5147810905460244	IUPHAR.LIGAND:1711	iuphar.ligand:1711	2MESATP	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	1.093909817410302	IUPHAR.LIGAND:5527	iuphar.ligand:5527	LL-37	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	agonist	0.065964411	IUPHAR.LIGAND:1755	iuphar.ligand:1755	ADP&BETA;S	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1711	iuphar.ligand:1711	2MESATP	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:1767	iuphar.ligand:1767	BX 667	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1714	iuphar.ligand:1714	ATP&GAMMA;S	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1736	ncit:C65436	DIQUAFOSOL	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1747	iuphar.ligand:1747	MRS2693	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:2260	iuphar.ligand:2260	[125I][AC-HIS1]PACAP-27	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:2668	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:2679	iuphar.ligand:2679	8S-HETE	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	3.088686543276147	IUPHAR.LIGAND:11369	iuphar.ligand:11369	[3H]-LKP	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:12616	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:9563	ncit:C125471	EGANELISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:6023	drugbank:DB04769	5-QUINOXALIN-6-YLMETHYLENE-THIAZOLIDINE-2,4-DIONE	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:10163	iuphar.ligand:10163	RV6153	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:6557	iuphar.ligand:6557	RS-25344	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11950	iuphar.ligand:11950	PF-07038124	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:7372	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
NCBIGENE:2394	hgnc:3906	FRA5B	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:6574	rxcui:99	6-AMINOCAPROIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2394	hgnc:3906	FRA5B	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:6573	rxcui:10691	TRANEXAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:11192	iuphar.ligand:11192	IACS-9439	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.095468493	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.070010228	IUPHAR.LIGAND:7649	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.070010228	IUPHAR.LIGAND:7649	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.095468493	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.019093699	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:5658	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:6021	iuphar.ligand:6021	PDGF RTK INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:8094	iuphar.ligand:8094	AG14361	FALSE	FALSE	FALSE
NCBIGENE:3145	hgnc:4982	HMBS	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11168	iuphar.ligand:11168	ETC-1922159	FALSE	FALSE	FALSE
NCBIGENE:1721	hgnc:9446	PRLR	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:4893	iuphar.ligand:4893	CHORIOMAMMOTROPIN	FALSE	FALSE	FALSE
NCBIGENE:2386	hgnc:3898	FRA3C	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8658	iuphar.ligand:8658	PEPTIDE 18 [PMID: 24350995]	FALSE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	0.07631929	IUPHAR.LIGAND:6391	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1258	hgnc:2151	CNGB1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8395	iuphar.ligand:8395	DS-437	FALSE	FALSE	FALSE
NCBIGENE:2401	hgnc:3912	FRA6A	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8626	iuphar.ligand:8626	COMPOUND 4G [PMID: 22595175]	FALSE	FALSE	FALSE
NCBIGENE:1477	hgnc:2483	CSTF1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:1488	hgnc:2495	CTBP2	GuideToPharmacology	2024.1	inhibitor	0.1434635826111871	IUPHAR.LIGAND:7946	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
NCBIGENE:2182	hgnc:3571	ACSL4	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9051	iuphar.ligand:9051	TILFRINIB	FALSE	FALSE	FALSE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12884	iuphar.ligand:12884	TEGEPROTAFIB	FALSE	FALSE	FALSE
NCBIGENE:3084	hgnc:7997	NRG1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:8856	iuphar.ligand:8856	COMPOUND 8A [PMID: 23713581]	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10419	iuphar.ligand:10419	RIPK2 INHIBITOR 5	FALSE	FALSE	FALSE
NCBIGENE:1014	hgnc:1755	CDH16	GuideToPharmacology	2024.1	NULL	0.729273212	IUPHAR.LIGAND:4562	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:8727	iuphar.ligand:8727	(5Z)-1-(2-FLUOROPHENYL)-2-SULFANYLIDENE-5-(THIOPHEN-2-YLMETHYLIDENE)-1,3-DIAZINANE-4,6-DIONE	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8033	iuphar.ligand:8033	RGS4 INHIBITOR 11B	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:2652	iuphar.ligand:2652	CD666	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:7784	iuphar.ligand:7784	CCG-50014	FALSE	FALSE	FALSE
NCBIGENE:2813	hgnc:4441	GP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7784	iuphar.ligand:7784	CCG-50014	FALSE	FALSE	FALSE
NCBIGENE:596	hgnc:990	BCL2	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:2904	iuphar.ligand:2904	SR8278	FALSE	FALSE	FALSE
NCBIGENE:1528	hgnc:2570	CYB5A	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8205	iuphar.ligand:8205	COMPOUND 22 [PMID: 20462760]	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1995	iuphar.ligand:1995	INSL3	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:4374	iuphar.ligand:4374	EUROPIUM-LABELLED RELAXIN-3-B/INSL5 A CHIMERA	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:11458	iuphar.ligand:11458	JK1	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:9493	iuphar.ligand:9493	SPM-354	FALSE	FALSE	FALSE
NCBIGENE:1172	hgnc:18044	SLC38A3	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:4634	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:10356	iuphar.ligand:10356	PURMORPHAMINE	FALSE	FALSE	FALSE
NCBIGENE:960	hgnc:1681	CD44	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:11708	iuphar.ligand:11708	MARALIXIBAT	FALSE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:10332	iuphar.ligand:10332	MRT-92	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:11730	iuphar.ligand:11730	TAK-020	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.034727296	Flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.00804962	Propafenone	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2040	iuphar.ligand:2040	BIM 23068	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2041	iuphar.ligand:2041	BIM 23197	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2023	iuphar.ligand:2023	[125I]LTT-SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:2007	iuphar.ligand:2007	CORTISTATIN-14	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2019	iuphar.ligand:2019	SRIF-14	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2023	iuphar.ligand:2023	[125I]LTT-SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11779	iuphar.ligand:11779	AZ6102	FALSE	FALSE	FALSE
NCBIGENE:3242	hgnc:5147	HPD	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:12814	iuphar.ligand:12814	GNE-7883	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5862	iuphar.ligand:5862	RO5166017	FALSE	FALSE	FALSE
NCBIGENE:2233	ncbigene:2233	FEB1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8191	iuphar.ligand:8191	COMPOUND 18 [PMID: 20873740]	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.013622434	Quinine Sulfate	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:11193	iuphar.ligand:11193	ZYBT1	FALSE	FALSE	FALSE
NCBIGENE:1722	hgnc:7217	MPL	GuideToPharmacology	2024.1	agonist	2.983390411119005	IUPHAR.LIGAND:6974	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.4375639269641208	Raltegravir	rxcui:1235585	RALTEGRAVIR POTASSIUM	TRUE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:1940	ncit:C76900	FLUPROSTENOL	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:6072	iuphar.ligand:6072	ICI 192605	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:6280	iuphar.ligand:6280	A-967079	FALSE	FALSE	FALSE
NCBIGENE:486	hgnc:4026	FXYD2	GuideToPharmacology	2024.1	blocker	0.729273212	IUPHAR.LIGAND:2441	iuphar.ligand:2441	SKF96365	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:10289	iuphar.ligand:10289	BTD	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.172722603	IUPHAR.LIGAND:2449	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	modulator	1.500219178	IUPHAR.LIGAND:12546	iuphar.ligand:12546	S-RHTX	FALSE	FALSE	FALSE
NCBIGENE:2424	ncbigene:2424	FRA8F	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7863	ncit:C76960	GABEXATE	FALSE	FALSE	FALSE
CPS1	hgnc:2323	CPS1	FDA	10-Apr-24	NULL	0.7501095890813501	Sodium Phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
NCBIGENE:511	hgnc:3145	TRPV5	GuideToPharmacology	2024.1	blocker	0.5357925636295356	IUPHAR.LIGAND:2446	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:9697	ncit:C152385	SOLCITINIB	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2159	iuphar.ligand:2159	[BZ-PHE6]U-II (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:2789	iuphar.ligand:2789	ZK159222	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:2171	iuphar.ligand:2171	F180	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:8529	iuphar.ligand:8529	RO5028442	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2201	iuphar.ligand:2201	SSR126768A	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:3869	iuphar.ligand:3869	D[VAL4,DARG8]VP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2228	iuphar.ligand:2228	[3H]DDAVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.097236428	IUPHAR.LIGAND:2182	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2195	iuphar.ligand:2195	OH-LVA	FALSE	FALSE	FALSE
NCBIGENE:812	hgnc:854	ATP6V1B2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8882	rxcui:3925	ENOXACIN	TRUE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.6482428547616604	IUPHAR.LIGAND:1507	iuphar.ligand:1507	NPY-(13-36) (PIG)	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	NULL	CHZ868	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
MS4A1	hgnc:7315	MS4A1	FDA	10-Apr-24	NULL	0.3025133322221082	Rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
KDR	hgnc:6307	KDR	CIViC	10-Apr-24	NULL	0.09055649	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	NULL	AKTI-1/2	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.2917092846427472	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.0095957	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
MAP2K2	hgnc:6842	MAP2K2	CIViC	10-Apr-24	NULL	0.033148782	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	NULL	DS-6501B	NULL	NULL	NULL	NULL	NULL
ASS1	hgnc:758	ASS1	FDA	10-Apr-24	NULL	0.1875273972703375	Sodium Phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.2187819634820604	ALK INHIBITOR TAE684	ncit:C171615	ALK INHIBITOR TAE684	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.2357246744587856	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
SMO	hgnc:11119	SMO	CIViC	10-Apr-24	NULL	4.375639269641208	PATIDEGIB	ncit:C80063	PATIDEGIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	JQ-1	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.2749092734853114	PAN-RAF INHIBITOR LY3009120	ncit:C116861	PAN-RAF INHIBITOR LY3009120	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.003566492	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
HSPA5	hgnc:5238	HSPA5	CIViC	10-Apr-24	NULL	0.027577558	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1875273972703375	Sulfamethoxazole	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
PDCD4	hgnc:8763	PDCD4	CIViC	10-Apr-24	NULL	0.4861821410712453	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	FDA	10-Apr-24	NULL	0.00804962	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
HLA-DRA	hgnc:4947	HLA-DRA	CIViC	10-Apr-24	NULL	0.2143170254518142	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
GATA2	hgnc:4171	GATA2	CIViC	10-Apr-24	NULL	0.2263261691193728	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
VKORC1	hgnc:23663	VKORC1	FDA	10-Apr-24	NULL	0.6364566210387212	Warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	CIViC	10-Apr-24	NULL	0.042700736	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
PTPRB	hgnc:9665	PTPRB	CIViC	10-Apr-24	NULL	0.2678962818147678	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.007378818	Tolterodine	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
PTPRB	hgnc:9665	PTPRB	CIViC	10-Apr-24	NULL	0.7292732116068681	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
APC	hgnc:583	APC	CIViC	10-Apr-24	NULL	NULL	G007-LK	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	MyCancerGenome	20-Jun-17	inhibitor	2.080014029626545	LDK378	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.010537361	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	CIViC	10-Apr-24	NULL	0.1256164383629055	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.5527123287967842	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
SMO	hgnc:11119	SMO	CIViC	10-Apr-24	NULL	NULL	PSI	NULL	NULL	NULL	NULL	NULL
AKT1	hgnc:391	AKT1	MyCancerGenome	20-Jun-17	inhibitor	0.3697723326457359	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	NULL	CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	NULL	CYTOREDUCTIVE SURGERY	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	1.518294108020081	RIPRETINIB	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	0.2536602475154323	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CEBPA	hgnc:1833	CEBPA	CIViC	10-Apr-24	NULL	13.12691780892362	OICR-9429	iuphar.ligand:8231	OICR-9429	FALSE	FALSE	TRUE
ARAF	hgnc:646	ARAF	CIViC	10-Apr-24	NULL	0.1060761035064535	COBIMETINIB	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.039688338	AEE788	iuphar.ligand:7643	AEE788	FALSE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	CIViC	10-Apr-24	NULL	0.1411496538593938	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.5164688974002737	RIPRETINIB	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
NT5E	hgnc:8021	NT5E	CIViC	10-Apr-24	NULL	0.076765601	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.020591244	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.031198854	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	MyCancerGenome	20-Jun-17	inhibitor	0.02077044	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
MITF	hgnc:7105	MITF	CIViC	10-Apr-24	NULL	0.030021539	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
ABCC10	hgnc:52	ABCC10	CIViC	10-Apr-24	NULL	0.081030357	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	CIViC	10-Apr-24	NULL	NULL	JQ-1	NULL	NULL	NULL	NULL	NULL
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.1682938180631233	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
ETV1	hgnc:3490	ETV1	CIViC	10-Apr-24	NULL	1.050153425	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	CIViC	10-Apr-24	NULL	0.1446492320542548	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
RAC1	hgnc:9801	RAC1	CIViC	10-Apr-24	NULL	0.1620607136904151	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	CIViC	10-Apr-24	NULL	0.014569276	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.2991890098899972	GDC-0032	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.060878459	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.072092912	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.052181537	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.021307461	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	4.702860988936115	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	X-376	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	MF tricyclic	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	CCT036477	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	CCT031374	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	iCRT-3	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	NC043	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	JW55	NULL	NULL	NULL	NULL	NULL
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.036925226	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	iCRT-14	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	G-631	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.596678082	BMS-906024	ncit:C116872	OSUGACESTAT	FALSE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.048708415	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.2273059360852575	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.2892984641085096	Buthionine sulfoximine	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	1.591141552596803	APR-246	ncit:C85465	EPRENETAPOPT	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.039272753	Gedatolisib	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.070690956	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.049983504	BI-847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.2051080907644316	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.021146867	Rabeprazole	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	SBI-0640756	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	SBI-755199	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	ARCC4	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	BDTX-4933	ncit:C200038	RAF INHIBITOR BDTX-4933	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.5498185469706229	BCA101	ncit:C173165	FICERAFUSP ALFA	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	NULL	CD19-PD-1/CD28-CAR T cells	NULL	NULL	NULL	NULL	NULL
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	CDX-527	ncit:C176983	ANTI-PD-L1/CD27 BISPECIFIC ANTIBODY CDX-527	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.042118453	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.864832232	Toripalimab-tpzi	rxcui:2669407	TORIPALIMAB-TPZI	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
PRKD2	hgnc:17293	PRKD2	MyCancerGenome	20-Jun-17	inhibitor	0.019548649	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.853211925965688	ZKAB001	ncit:C162504	SOCAZOLIMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.091516638	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	NULL	SBI-0640756	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	WNTinib	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	CC-91516	NULL	NULL	NULL	NULL	NULL
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.1000146118775133	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.2282942227638891	Taletrectinib	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	0.025929714	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.1579178082276526	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.3453256329104173	Infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
CCR4	hgnc:1605	CCR4	MyCancerGenome	20-Jun-17	antibody	12.35474617310458	MOGAMULIZUMAB	rxcui:2054068	MOGAMULIZUMAB	TRUE	TRUE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	M-COPA	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.016256245	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	1.040600372117402	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.022559687	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	NMS-P088	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	A-419259	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.014405397	Alisertib	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	antibody	0.3454452054979901	ADO-TRASTUZUMABEMTANSINE	wikidata:Q29006063	KADCYLA	FALSE	TRUE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2520944435184235	Pacritinib	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	NVP-BSK805	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	NVP-BVB808	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	FLT3/CD3 Fabsc antibody	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	CCT137690	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	APG-2575	chembl:CHEMBL4650374	APG-2575	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.108040476	Sonidegib	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	antibody	0.3081436105381133	RAMUCIRUMAB	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	WM-8014	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.172722603	Rigosertib	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.038382801	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	IHMT-RAF-128	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	NULL	BPTES	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	NULL	IDH1 R132H peptide vaccine	NULL	NULL	NULL	NULL	NULL
NOTCH1	hgnc:7881	NOTCH1	MyCancerGenome	20-Jun-17	other/unknown	1.312691780892362	REGN421	ncit:C82367	ENOTICUMAB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.036680176	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.9842513760562132	Ivosidenib	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.021396769	Veliparib	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	NULL	TQ05310	NULL	NULL	NULL	NULL	NULL
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	NULL	AGI-6780	NULL	NULL	NULL	NULL	NULL
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	NULL	SHP099	NULL	NULL	NULL	NULL	NULL
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.094099769	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	NULL	NVP-BSK805	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	NULL	NVP-BVB808	NULL	NULL	NULL	NULL	NULL
APH1B	hgnc:24080	APH1B	MyCancerGenome	20-Jun-17	other/unknown	0.4039051633514962	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.5645986154375752	Pyridone 6	drugbank:DB04716	2-TERT-BUTYL-9-FLUORO-1,6-DIHYDROBENZO[H]IMIDAZO[4,5-F]ISOQUINOLIN-7-ONE	FALSE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.3763990769583835	Pacritinib	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2853677784548614	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.1935766681500258	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	SAR405838	ncit:C106120	P53-HDM2 INTERACTION INHIBITOR MI-773	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.03136659	Infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	OKI-219	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.054020238	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
PARP1	hgnc:270	PARP1	MyCancerGenome	20-Jun-17	other/unknown	0.4296082192011368	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.5173169579871378	Trilaciclib	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	ALW-II-41-27	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	XMD15-44	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	LOX-18228	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	Y078-DM1	NULL	NULL	NULL	NULL	NULL
HSP90AA1	hgnc:5253	HSP90AA1	MyCancerGenome	20-Jun-17	other/unknown	0.3621218705909965	RETASPIMYCIN	ncit:C80378	RETASPIMYCIN	FALSE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	2.187819634820604	NUV-520	ncit:C185422	ZIDESAMTINIB	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.3281729452230906	Taletrectinib	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.024861587	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.1293292394967844	Gedatolisib	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.013246968	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	unspecified ERBB3 antibody	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.038636991	AZD1390	iuphar.ligand:11277	AZD1390	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.011591097	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PSME1	hgnc:9568	PSME1	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.006623484	Camptothecin	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	unspecified immune checkpoint inhibitor	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	ReACp53	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	MK-8745	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.04636439	CEP1347	iuphar.ligand:8173	CEP-1347	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.4636438961209227	APR-246	ncit:C85465	EPRENETAPOPT	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.077273983	Trifluridine	rxcui:10803	TRIFLURIDINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	MX69	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	PT2399	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	HLA-A2 p53:264-272 vaccine	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	YW3-56	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	M8891	iuphar.ligand:12714	M8891	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.011591097	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.004189553	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	NULL	STF-62247	NULL	NULL	NULL	NULL	NULL
PSMD14	hgnc:16889	PSMD14	MyCancerGenome	20-Jun-17	other/unknown	0.1878628666751144	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1238388472539964	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.038159645	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	NIFURALDEZONE	ncit:C77051	NIFURALDEZONE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
PSMB6	hgnc:9543	PSMB6	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1875273972703375	3-(PHENYLAMINO)PHENOL	chembl:CHEMBL1523215	CHEMBL:CHEMBL1523215	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TRIS(4-ISOPROPYLPHENYL) PHOSPHATE	chembl:CHEMBL458602	CHEMBL:CHEMBL458602	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00202529	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
PSMD8	hgnc:9566	PSMD8	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.042516333	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-123457	chembl:CHEMBL285157	CHEMBL:CHEMBL285157	FALSE	FALSE	FALSE
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	0.6335767268258763	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
PSMB9	hgnc:9546	PSMB9	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:Q13698	hgnc:1397	CACNA1S	TdgClinicalTrial	Jan-14	NULL	0.283060222	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.060492709	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
NCBIGENE:2842	hgnc:4473	GPR19	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8296	iuphar.ligand:8296	EXAMPLE 373 [WO2012093101]	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:12612	iuphar.ligand:12612	PIROTINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.014916952	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PSMB4	hgnc:9541	PSMB4	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4347	iuphar.ligand:4347	ZK93426	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.023151531	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.068191781	IGURATIMOD	ncit:C65886	IGURATIMOD	FALSE	FALSE	FALSE
PSMB7	hgnc:9544	PSMB7	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CGI	2/1/22	NULL	0.1999620096341412	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	DICLOFENAC EPOLAMINE	rxcui:40968	DICLOFENAC EPOLAMINE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.023482858	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
UNIPROT:O43772	hgnc:1421	SLC25A20	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
PSME2P2	hgnc:30160	PSME2P2	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	N-(PHENETHYLCARBAMOTHIOYL)BENZAMIDE	chembl:CHEMBL1448292	CHEMBL:CHEMBL1448292	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1548898856510162	IUPHAR.LIGAND:10452	iuphar.ligand:10452	NMRA-140	FALSE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR BETA	hgnc:6009	IL2RB	TTD	2020.06.01	NULL	4.039051633514961	NKTR 214	chembl:CHEMBL4298058	BEMPEGALDESLEUKIN	FALSE	FALSE	FALSE
PSMD5	hgnc:9563	PSMD5	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
S1PR2	hgnc:3169	S1PR2	DTC	9/2/20	NULL	0.3125456621172291	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2311077079035849	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.2763561643983921	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	0.2885036881082115	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	TCMDC-123480	chembl:CHEMBL588683	CHEMBL:CHEMBL588683	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:10306	iuphar.ligand:10306	PI-HEXATOXIN-HI1A	FALSE	FALSE	FALSE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1767935058440892	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:374	iuphar.ligand:374	CCPA	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:11879	iuphar.ligand:11879	NARAZACICLIB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Tislelizumab	rxcui:2677426	TISLELIZUMAB	TRUE	FALSE	FALSE
ICMT	hgnc:5350	ICMT	DTC	9/2/20	NULL	1.050153425	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	PALMITOYL-DL-CARNITINE CHLORIDE	chembl:CHEMBL1256761	CHEMBL:CHEMBL1256761	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.1988926940746004	DIFFERENTIATING AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1988926940746004	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
GCKR	hgnc:4196	GCKR	PharmGKB	4/5/24	NULL	0.1260688385010672	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	PharmGKB	4/5/24	NULL	0.006561408	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.08607815	FLAVOPIRIDOL	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.1715936968486748	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.4243044140258141	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1434635826111871	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
PROTEINASE ACTIVATED RECEPTOR 1	hgnc:3537	F2R	TTD	2020.06.01	NULL	1.009762908	Vorapaxar	rxcui:1537034	VORAPAXAR	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.4234489615781814	IUPHAR.LIGAND:9326	ncit:C132738	ABEDITEROL	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.00897567	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:1251	iuphar.ligand:1251	IMMEPIP	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.049442252	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.038837035	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.059532507	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.2711239478607289	PLX-3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-1241	chembl:CHEMBL528724	CHEMBL:CHEMBL528724	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2062	iuphar.ligand:2062	[125I]TYR3 SMS 201-995	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1704794520639431	MILNACIPRAN	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.027781837	IUPHAR.LIGAND:213	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:7461	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:660	hgnc:1079	BMX	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:5535	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.037666909	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.077789143	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006419031	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	2.940429589198891	Rasburicase	rxcui:283821	RASBURICASE	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.08334551	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	0.760980743	RS-504393	iuphar.ligand:781	RS-504393	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.028708404	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2160809515872201	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
MIF	hgnc:7097	MIF	ChEMBL	33	inhibitor	1.250182648468916	IGURATIMOD	ncit:C65886	IGURATIMOD	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004821641	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.021608095	1-BETA-D-ARABINOFURANOSYLCYTOSINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.2408608772279564	levomethadone	rxcui:236913	LEVOMETHADONE	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.3017682254924971	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.011157601	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.028929846	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.1182605208011137	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.3889457128569963	INFIGRATINIB	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.088996053	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
THYMIDINE PHOSPHORYLASE	hgnc:3148	TYMP	TTD	2020.06.01	NULL	0.8204323630577265	Uridine	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.151537291	ALPHA-DIFLUOROMETHYLORNITHINE	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:12442	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
EREG	hgnc:3443	EREG	CIViC	10-Apr-24	NULL	0.2430910705356227	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	INTERFERON ALFA-N1	rxcui:202912	INTERFERON ALFA-N1	FALSE	TRUE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	Genz-644282	chembl:CHEMBL191958	GENZ-644282	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	CGP-7930	iuphar.ligand:1079	CGP7930	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	1.166837138570988	Z160	iuphar.ligand:7765	NP118809	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.074163377	IUPHAR.LIGAND:277	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:8391	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.2734774543525755	IUPHAR.LIGAND:2441	iuphar.ligand:2441	SKF96365	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR BETA	hgnc:9865	RARB	TTD	2020.06.01	NULL	0.4412409347537352	Alitretinoin	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.060772768	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
CSF2RB	hgnc:2436	CSF2RB	ChEMBL	33	inhibitor	2.917092846427472	MAVRILIMUMAB	ncit:C95788	MAVRILIMUMAB	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.064824285	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q99250	hgnc:10588	SCN2A	TEND	1-Aug-11	NULL	0.2083637747448194	FOSPROPOFOL	rxcui:828682	FOSPROPOFOL	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.7425327245451747	Atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	negative modulator	0.097236428	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.1881995384791917	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	RO-194603	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.1254663589861278	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P55157	hgnc:7467	MTTP	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	LOMITAPIDE	rxcui:1364478	LOMITAPIDE MESYLATE	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.029041854	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.019739726	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1143957978991165	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
CASR	hgnc:1514	CASR	ChEMBL	33	agonist	3.281729452230906	VELCALCETIDE	rxcui:1876119	ETELCALCETIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.4052907728312611	methoxyflurane	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.078194596	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.5645986154375752	AN0128	drugbank:DB05054	AN0128	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:7252	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
NCBIGENE:310	hgnc:545	ANXA7	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1579	iuphar.ligand:1579	NEUROTENSIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.042174836	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
THYROID HORMONE RECEPTOR ALPHA	hgnc:11796	THRA	TTD	2020.06.01	NULL	1.875273972703375	Levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.025588534	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.1591141552596803	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.035574303	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	1.500219178	PRT-2607	chembl:CHEMBL3545138	PRT-2607	FALSE	FALSE	FALSE
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	7.001022831425932	PF-05212377	drugbank:DB16044	PF-05212377	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.009787078	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.2243917574174978	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
UNIPROT:P33402	hgnc:4684	GUCY1A2	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	NITRIC OXIDE	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:1359	iuphar.ligand:1359	K185	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-3832	chembl:CHEMBL261693	CHEMBL:CHEMBL261693	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1526385791735305	GNF-PF-3725	chembl:CHEMBL598695	CHEMBL:CHEMBL598695	FALSE	FALSE	FALSE
PRKAG3	hgnc:9387	PRKAG3	DTC	9/2/20	NULL	1.795134059339982	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
UNIPROT:Q13421	hgnc:7371	MSLN	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	AMATUXIMAB	ncit:C62483	AMATUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.3125456621172291	IUPHAR.LIGAND:12002	iuphar.ligand:12002	ABBV-318	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.013673873	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
NCBIGENE:1560	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9668	iuphar.ligand:9668	JFD00064	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.068369364	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2428	hgnc:3938	FRA9D	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12225	iuphar.ligand:12225	SJB2-043	FALSE	FALSE	FALSE
NCBIGENE:1623	hgnc:2691	DBIP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8628	iuphar.ligand:8628	COMPOUND 4 [PMID: 12408711]	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.201178817	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	1.944728564284981	Reparixin	ncit:C66515	REPARIXIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	negative modulator	0.172722603	BDTX189	chembl:CHEMBL4650279	BDTX189	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1434635826111871	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	PharmGKB	4/5/24	NULL	0.218327115	fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	NCI	14-Sep-17	NULL	1.848379561100067	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TEND	1-Aug-11	NULL	0.8078103267029924	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	Bambuterol	rxcui:18751	BAMBUTEROL	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	NCI	14-Sep-17	NULL	0.037748146	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.013879903	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
CD33	hgnc:1659	CD33	ChEMBL	33	binder	4.039051633514961	ONCOLYSIN M	chembl:CHEMBL2109520	ONCOLYSIN M	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	SB-203186	iuphar.ligand:255	SB 203186	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	2-((4-(DIMETHYLAMINO)PHENYL)DIAZENYL)BENZOIC ACID	chembl:CHEMBL375971	CHEMBL:CHEMBL375971	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.024861587	PROPAFENONE	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.038104261	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	6-AZAURIDINE	ncit:C291	6-AZAURIDINE	FALSE	FALSE	FALSE
ADCYAP1R1	hgnc:242	ADCYAP1R1	NCI	14-Sep-17	NULL	0.2631963470460877	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.02804897	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NOTCH1	hgnc:7881	NOTCH1	CIViC	10-Apr-24	NULL	1.406455479527531	NIROGACESTAT	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.027248402	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	0.325124899	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.014385663	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
SLC22A6	hgnc:10970	SLC22A6	PharmGKB	4/5/24	NULL	13.12691780892362	cidofovir	rxcui:1546007	CIDOFOVIR ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.073954467	PTC299	drugbank:DB05173	PTC299	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.1491695205559502	Propranolol	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4327	iuphar.ligand:4327	TPA023	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1620607136904151	CORONOPILIN	chembl:CHEMBL248564	CORONOPILIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	POLIDOCANOL	rxcui:968170	POLIDOCANOL	TRUE	FALSE	FALSE
NAPEPLD	hgnc:21683	NAPEPLD	NCI	14-Sep-17	NULL	1.329308132549227	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	BD-1008	chembl:CHEMBL20377	CHEMBL:CHEMBL20377	FALSE	FALSE	FALSE
ABI1	hgnc:11320	ABI1	PharmGKB	4/5/24	NULL	0.1750255707856483	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2931	iuphar.ligand:2931	W146	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.1988926940746003	IUPHAR.LIGAND:4366	iuphar.ligand:4366	[3H]CGS8216	FALSE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.041628703	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	0.1241316104862754	IUPHAR.LIGAND:1013	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:4125	iuphar.ligand:4125	AF353	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6473	iuphar.ligand:6473	MORPHANTHRIDINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.022062047	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	INCSHR1210	iuphar.ligand:9758	CAMRELIZUMAB	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	0.6731752722524935	Ladostigil	ncit:C77584	LADOSTIGIL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	ENDRIN	chembl:CHEMBL44072	ENDRIN	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.212152207	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.1363835616511545	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
NR5A2	hgnc:7984	NR5A2	DTC	9/2/20	NULL	52.50767123569449	GSK8470	chembl:CHEMBL385911	CHEMBL:CHEMBL385911	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.038894571	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	DIPROTIN A	chembl:CHEMBL214381	DIPROTIN A	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8146	iuphar.ligand:8146	COMPOUND 23 [PMID: 17600705]	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DoCM	10-Apr-24	NULL	0.1331836936859721	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.098053541	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	negative modulator	0.02956513	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:822	iuphar.ligand:822	[125I]CXCL8 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12386	iuphar.ligand:12386	ZELASUDIL	FALSE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.001814112	Celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	MRS-1220	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.1295419520617463	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	1.607377690888607	BETRIXABAN	rxcui:1927851	BETRIXABAN	TRUE	FALSE	FALSE
IFNA17	hgnc:5422	IFNA17	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.033295923	IUPHAR.LIGAND:34	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	activator	0.7721716358190367	IUPHAR.LIGAND:2508	iuphar.ligand:2508	LYSOPHOSPHATIDYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:132	hgnc:257	ADK	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:8791	iuphar.ligand:8791	COMPOUND 33 [TODA ET AL., 2013]	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:6657	iuphar.ligand:6657	GB110	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.038636991	Alemtuzumab	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
CD2	hgnc:1639	CD2	NCI	14-Sep-17	NULL	2.333674277141978	ZNCL2	rxcui:39937	ZINC CHLORIDE	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.082429625	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011049594	DEXMEDETOMIDINE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.009656583	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.073540156	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.2344092465879218	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.061737415	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
RYR3	hgnc:10485	RYR3	ChEMBL	33	inhibitor	1.458546423213736	DANTROLENE SODIUM	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
BLK	hgnc:1057	BLK	ChEMBL	33	inhibitor	0.078136416	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.073694977	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
NCBIGENE:1385	hgnc:2345	CREB1	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:5169	iuphar.ligand:5169	CJ13610	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3119	iuphar.ligand:3119	COMPOUND 21 [PMID: 19191557]	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	1.117184494376478	IUPHAR.LIGAND:2084	iuphar.ligand:2084	BIM 23313	FALSE	FALSE	FALSE
PROMININ-1	hgnc:9454	PROM1	TTD	2020.06.01	NULL	105.0153424713889	ICT-121	ncit:C124652	ICT-121 DENDRITIC CELL VACCINE	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:5913	iuphar.ligand:5913	AG 112	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.076024621	LY3023414	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.4039051633514961	IUPHAR.LIGAND:11462	iuphar.ligand:11462	TAMRLX	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	ChEMBL	33	inhibitor	3.000438356	IMETELSTAT	ncit:C49084	IMETELSTAT	FALSE	FALSE	TRUE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.050294704	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1909369863116163	NITROGEN MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.045898314	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	P-CYANOCHALCONE	chembl:CHEMBL445153	CHEMBL:CHEMBL445153	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.1944728564284981	IUPHAR.LIGAND:1343	drugbank:DB08190	N-[2-(2-IODO-5-METHOXY-1H-INDOL-3-YL)ETHYL]ACETAMIDE	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.07182992	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	blocker	0.2822993077187876	IUPHAR.LIGAND:2403	ncit:C65450	DIZOCILPINE	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inverse agonist	1.514644363	NELOTANSERIN	ncit:C83996	NELOTANSERIN	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.5707355569097228	ZEARALANONE	chembl:CHEMBL491499	ZEARALANONE	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.064268875	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
VITAMIN K-DEPENDENT GAMMA-CARBOXYLASE	hgnc:4247	GGCX	TTD	2020.06.01	NULL	3.500511415712966	Phytonadione	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	CGI	2/1/22	NULL	0.4167275494896388	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.014073351	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
IGHE	hgnc:5522	IGHE	ChEMBL	33	inhibitor	8.751278539282415	LIGELIZUMAB	ncit:C175809	LIGELIZUMAB	FALSE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	2.019525817	PERAKIZUMAB	ncit:C175189	PERAKIZUMAB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DODECYL-TRIMETHYL-AMMONIUM BROMIDE	chembl:CHEMBL109873	CHEMBL:CHEMBL109873	FALSE	FALSE	FALSE
NCBIGENE:2147	hgnc:3535	F2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.080042182	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TEND	1-Aug-11	NULL	0.6364566210387211	EXENATIDE	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	0.02302968	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
DDR2	hgnc:2731	DDR2	DoCM	10-Apr-24	NULL	0.9546849315580819	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.034727296	Acalisib	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.2430910705356227	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	1.280674908	DOLASTATIN 10	ncit:C1300	DOLASTATIN 10	FALSE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	DTC	9/2/20	NULL	1.591141552596803	(12E,20Z,18S)-8-HYDROXYVARIABILIN	iuphar.ligand:4072	(12E,20Z,18S)-8-HYDROXYVARIABILIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013281873	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	GNF-PF-4218	chembl:CHEMBL585269	CHEMBL:CHEMBL585269	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.092118721	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	Autologous Anti-CD19CAR-4-1BB-CD3zeta-EGFRt-expressing T Lymphocytes	ncit:C116914	AUTOLOGOUS ANTI-CD19CAR-4-1BB-CD3ZETA-EGFRT-EXPRESSING T LYMPHOCYTES	FALSE	FALSE	FALSE
TMEM196	hgnc:22431	TMEM196	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.2397610558707511	NU7441	iuphar.ligand:8010	NU-7441	FALSE	FALSE	TRUE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	3.141484604	IL-1RA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:562	hgnc:6297	KCNQ3	GuideToPharmacology	2024.1	activator	0.093763699	IUPHAR.LIGAND:5483	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:4046	iuphar.ligand:4046	NF546	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:9787	drugbank:DB12903	DEBIO-1347	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2045	iuphar.ligand:2045	[111IN]DOTA-NOC	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.05068308	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
UNIPROT:O76074	hgnc:8784	PDE5A	TEND	1-Aug-11	NULL	0.1406455479527531	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.052455216	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:736	iuphar.ligand:736	[3H]WIN55212-2	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.3387591692625452	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CD40	hgnc:11919	CD40	ChEMBL	33	agonist	2.187819634820604	TENELIXIMAB	ncit:C87768	TENELIXIMAB	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	1.346350544504987	PRX-03140	drugbank:DB05596	PRX-03140	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.016669102	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.013920379	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.2386712328895204	FLECAINIDE ACETATE	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	DALFOPRISTIN	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2047	iuphar.ligand:2047	L-363,301	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.085587076	Elimusertib	ncit:C146807	ELIMUSERTIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
SULT2A1	hgnc:11458	SULT2A1	DTC	9/2/20	NULL	10.50153424713889	EMATE	chembl:CHEMBL122708	EMATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	NCI	14-Sep-17	NULL	0.022530646	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.4268916360625568	HEN EGG LYSOZYME	ncit:C1925	LYSOZYME	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	TALC	12-May-16	vaccine	0.384671584	PRINOMASTAT	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
PYROXD2	hgnc:23517	PYROXD2	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.2323348284765243	penicillin v	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.081407242	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
AVPR1B	hgnc:896	AVPR1B	ChEMBL	33	binder	3.750547945	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.6563458904461812	Rubitecan	ncit:C1485	RUBITECAN	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	ChEMBL	33	inhibitor	2.386712328895204	SLX-4090	drugbank:DB05678	SLX-4090	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006141248	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.026319635	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	DTC	9/2/20	NULL	0.7778914257139925	TYRAMINE	rxcui:10958	TYRAMINE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	6-HYDROXYFLAVONE	chembl:CHEMBL138649	6-HYDROXYFLAVONE	FALSE	FALSE	FALSE
S1PR4	hgnc:3170	S1PR4	ChEMBL	33	modulator	1.166837138570989	AMISELIMOD HYDROCHLORIDE	ncit:C142922	AMISELIMOD HYDROCHLORIDE	FALSE	FALSE	FALSE
CBL	hgnc:1541	CBL	NCI	14-Sep-17	NULL	0.210030685	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
SLIT AND NTRK-LIKE FAMILY MEMBER 6	hgnc:23503	SLITRK6	TTD	2020.06.01	NULL	52.50767123569449	ASG-15ME	ncit:C152370	SIRTRATUMAB VEDOTIN	FALSE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.1262203635473425	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
DLG4	hgnc:2903	DLG4	NCI	14-Sep-17	NULL	0.9723642821424908	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
GFRA2	hgnc:4244	GFRA2	PharmGKB	4/5/24	NULL	0.2706580991530644	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.055504938	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.051731696	ZERANOL	rxcui:1368476	ZERANOL	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	DNDI1417623	chembl:CHEMBL2002849	CHEMBL:CHEMBL2002849	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	OXYBENZONE	rxcui:32673	OXYBENZONE	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.2500365296937833	NORETHINDRONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.7458476027797514	BISOPROLOL	rxcui:19484	BISOPROLOL	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.2333674277141977	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004427291	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.3040984820600068	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	PharmGKB	4/5/24	NULL	0.1111273465305703	somatropin recombinant	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
CCL14	hgnc:10612	CCL14	NCI	14-Sep-17	NULL	8.751278539282415	RANTES	ncit:C1211	RECOMBINANT RANTES	FALSE	FALSE	FALSE
SODIUM PUMP	hgnc:15879	CTNNBL1	TTD	2020.06.01	NULL	26.25383561784724	Alpha-acetyldigoxin	drugbank:DB13691	ACETYLDIGOXIN	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	Exarafenib	ncit:C180835	EXARAFENIB	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.040275444	AMIODARONE HYDROCHLORIDE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	modulator	0.041377203	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002356506	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.089501712	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	SAVIRIN	chembl:CHEMBL1494499	SAVIRIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.013021444	pimozide	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.5834185692854944	4-HYDROXYBENZOHYDRAZIDE	chembl:CHEMBL124267	CHEMBL:CHEMBL124267	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	DTC	9/2/20	NULL	0.6908904109959803	N6-CYCLOPENTYLADENOSINE	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	CEAROIN	chembl:CHEMBL1613209	CEAROIN	FALSE	FALSE	FALSE
LOXL2	hgnc:6666	LOXL2	ChEMBL	33	inhibitor	52.50767123569449	SIMTUZUMAB	ncit:C91735	SIMTUZUMAB	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.1166837138570989	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	1.009762908	TAK-070	iuphar.ligand:6940	TAK-070	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	2.187819634820604	GNF-PF-5149	chembl:CHEMBL600309	CHEMBL:CHEMBL600309	FALSE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:5278	drugbank:DB08626	THIORPHAN	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.2069267831948551	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.093680056	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
SIN3A	hgnc:19353	SIN3A	PharmGKB	4/5/24	NULL	5.000730593875666	hydroxyurea	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	1.544343271638073	DEMECARIUM BROMIDE	rxcui:22482	DEMECARIUM BROMIDE	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	2.019525817	AFASEVIKUMAB	ncit:C169767	AFASEVIKUMAB	FALSE	FALSE	FALSE
UNIPROT:P05093	hgnc:2593	CYP17A1	TdgClinicalTrial	Jan-14	NULL	30.00438356	ORTERONEL	ncit:C90582	ORTERONEL	FALSE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.06466462	IUPHAR.LIGAND:15	iuphar.ligand:15	L-694,247	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:12153	iuphar.ligand:12153	FLX475	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:12089	iuphar.ligand:12089	RUSERONTINIB	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1176247115494948	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.3562257207306275	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
ELP5	hgnc:30617	ELP5	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.1553481397505754	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	FDA	10-Apr-24	NULL	0.8579684842433742	Denileukin Diftitox	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	NSC-753576	chembl:CHEMBL2088731	CHEMBL:CHEMBL2088731	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	PARBENDAZOLE	ncit:C96752	PARBENDAZOLE	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.2453629496995069	PHENYLPROPANOLAMINE POLISTIREX	chembl:CHEMBL1201535	PHENYLPROPANOLAMINE POLISTIREX	TRUE	FALSE	FALSE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	inhibitor	1.346350544504987	BASILIXIMAB	rxcui:196102	BASILIXIMAB	TRUE	TRUE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.076098074	IUPHAR.LIGAND:7649	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.014708031	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
CCL8	hgnc:10635	CCL8	NCI	14-Sep-17	NULL	1.944728564284981	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.013415348	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.018430211	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	ABM-1310	ncit:C170951	BRAF(V600E) KINASE INHIBITOR ABM-1310	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	CYSTEINE	rxcui:3024	CYSTEINE	TRUE	FALSE	FALSE
CYCLIC NUCLEOTIDE-GATED CHANNEL ALPHA-2	hgnc:2149	CNGA2	TTD	2020.06.01	NULL	3.281729452230906	dequalinium	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1056492378987816	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
SLC22A3	hgnc:10967	SLC22A3	NCI	14-Sep-17	NULL	0.5048814541893702	ANTIDEPRESSANT DRUGS	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	IMIPENEM	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
CCNA2	hgnc:1578	CCNA2	NCI	14-Sep-17	NULL	6.563458904461812	3-DEOXYADENOSINE	ncit:C1057	CORDYCEPIN	FALSE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	0.9376369863516875	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.072927321	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9979	iuphar.ligand:9979	PF-04634817	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.058997383	IUPHAR.LIGAND:955	iuphar.ligand:955	(+)-S-14297	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2853677784548614	Go6976	iuphar.ligand:5973	G&OUML; 6976	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	L-GLUTAMATE	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003716042	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	3.842024724563012	COLTUXIMAB RAVTANSINE	ncit:C71009	COLTUXIMAB RAVTANSINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1077080435603989	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	NCI	14-Sep-17	NULL	0.8078103267029924	INTERFERON GAMMA	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.6819178082557728	DIFFERENTIATING AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.021440454	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.5339763176511304	SPARSENTAN	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	1.193356164447602	OZARELIX	ncit:C95214	OZARELIX	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.066297565	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:1757	iuphar.ligand:1757	BZATP	FALSE	FALSE	FALSE
CCL22	hgnc:10621	CCL22	NCI	14-Sep-17	NULL	4.375639269641208	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:9728	ncit:C107686	DEZAPELISIB	FALSE	FALSE	FALSE
EIF2S1	hgnc:3265	EIF2S1	NCI	14-Sep-17	NULL	1.250182648468916	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	0.2954018072331617	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
UNIPROT:P30872	hgnc:11330	SSTR1	TEND	1-Aug-11	NULL	1.250182648468916	LANREOTIDE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.084146909	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.2592971419046642	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.5000730593875666	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	3-(PHENYLAMINO)PHENOL	chembl:CHEMBL1523215	CHEMBL:CHEMBL1523215	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.061041236	pergolide	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	PharmGKB	4/5/24	NULL	0.075732218	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:1359	hgnc:2298	CPA3	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:8311	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	antibody	0.036463661	IUPHAR.LIGAND:5082	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
STAT5B	hgnc:11367	STAT5B	NCI	14-Sep-17	NULL	0.6177373086552295	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	TCMDC-123634	chembl:CHEMBL530499	CHEMBL:CHEMBL530499	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	ISOBOLDINE	chembl:CHEMBL462880	ISOBOLDINE	FALSE	FALSE	FALSE
UNIPROT:O60896	hgnc:9845	RAMP3	TdgClinicalTrial	Jan-14	NULL	5.000730593875666	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
ADORA1	hgnc:262	ADORA1	PharmGKB	4/5/24	NULL	0.020688602	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	2.386712328895204	YM-543	chembl:CHEMBL2397450	YM-543	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.092443083	Rivoceranib	ncit:C152237	RIVOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.033658764	IUPHAR.LIGAND:2168	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.066860362	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.9907107780319716	RG-2833	drugbank:DB16955	RG-2833	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	3.842024724563012	Coltuximab ravtansine	ncit:C71009	COLTUXIMAB RAVTANSINE	FALSE	FALSE	FALSE
PIK3C2A	hgnc:8971	PIK3C2A	NCI	14-Sep-17	NULL	0.7721716358190367	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003405608	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.021240967	RU-24969	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003541833	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.037345428	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
UNIPROT:P33151	hgnc:1764	CDH5	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	FX06	drugbank:DB05685	FX06	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.052455216	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	modulator	0.8334550989792776	IUPHAR.LIGAND:8498	ncit:C66515	REPARIXIN	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.083279415	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
ICA1	hgnc:5343	ICA1	PharmGKB	4/5/24	NULL	7.501095890813499	o-desmethyltramadol	chembl:CHEMBL4650315	DESMETRAMADOL	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	ERYTHROMYCIN STEARATE	rxcui:24351	ERYTHROMYCIN STEARATE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:2907	iuphar.ligand:2907	KI16425	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:317	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.2333674277141978	clindamycin	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.049723174	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.1141471113819445	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
AK2	hgnc:362	AK2	PharmGKB	4/5/24	NULL	1.875273972703374	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.100976291	ANTI-VEGF	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
TNFRSF1B	hgnc:11917	TNFRSF1B	NCI	14-Sep-17	NULL	0.7501095890813498	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.064033745	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.2027323213733378	Flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	ChEMBL	33	inhibitor	0.760980743	TIDEGLUSIB	ncit:C97364	TIDEGLUSIB	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.3201687270469177	IUPHAR.LIGAND:493	rxcui:720825	SILODOSIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.5385402178019949	acetylcysteine	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	DTC	9/2/20	NULL	0.030886865	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.6364566210387211	Exenatide	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.043890503	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1473	iuphar.ligand:1473	NEUROMEDIN U-8	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:1755	iuphar.ligand:1755	ADP&BETA;S	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.026927011	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.007416338	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
SULT1A2	hgnc:11454	SULT1A2	PharmGKB	4/5/24	NULL	11.66837138570988	endoxifen	iuphar.ligand:10203	ENDOXIFEN	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	ChEMBL	33	inhibitor	0.1190650141398968	POSDINEMAB	ncit:C188522	POSDINEMAB	FALSE	FALSE	FALSE
SLC10A1	hgnc:10905	SLC10A1	ChEMBL	33	inhibitor	8.751278539282415	MYRCLUDEX B	drugbank:DB14853	MYRCLUDEX B	FALSE	FALSE	FALSE
NCBIGENE:1264	hgnc:2155	CNN1	GuideToPharmacology	2024.1	modulator	1.875273972703375	IUPHAR.LIGAND:10645	ncit:C169983	FIRSOCOSTAT	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:1039	iuphar.ligand:1039	QUIN-C7	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:8827	iuphar.ligand:8827	COMPOUND 11J [PMID: 23021994]	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.008558708	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.034018575	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.347732922	N-(3,4-DIMETHOXYPHENETHYL)BENZENESULFONAMIDE	chembl:CHEMBL258316	CHEMBL:CHEMBL258316	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007551801	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	DICLAZURIL	rxcui:1368201	DICLAZURIL	TRUE	FALSE	FALSE
NCBIGENE:2609	hgnc:4145	GAPDHP67	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:11480	iuphar.ligand:11480	SLF	FALSE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:12663	iuphar.ligand:12663	TRULI	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:11526	iuphar.ligand:11526	SARUPARIB	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.035418328	NEOSTIGMINE BROMIDE	rxcui:82055	NEOSTIGMINE BROMIDE	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.079197091	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
FOLH1	hgnc:3788	FOLH1	PharmGKB	4/5/24	NULL	3.889457128569962	lutetium (177lu) vipivotide tetraxetan	rxcui:2597053	LUTETIUM LU 177 VIPIVOTIDE TETRAXETAN	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	1.050153425	GLICLAZIDE	rxcui:4816	GLICLAZIDE	TRUE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:660	iuphar.ligand:660	PS020990	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:3520	iuphar.ligand:3520	R121919	FALSE	FALSE	FALSE
NCBIGENE:1344	hgnc:2645	CYP4F2	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:8851	iuphar.ligand:8851	17-OCTADECYNOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	blocker	0.067403943	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.007549629	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.091159151	AGN-214868	chembl:CHEMBL3137348	SENREBOTASE	FALSE	FALSE	FALSE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	MPC-3100	ncit:C84836	HSP90 INHIBITOR LAM-003A	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:7241	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.0136917	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	modulator	0.8204323630577265	SOLITOMAB	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6298	iuphar.ligand:6298	1'-ACETOXYCHAVICOL ACETATE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	GW405833	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.014092236	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
UNIPROT:P35568	hgnc:6125	IRS1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	GS-101	ncit:C148131	AGANIRSEN	FALSE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:7338	iuphar.ligand:7338	RO4929097	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.046303061	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.005984462	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
GART	hgnc:4163	GART	ChEMBL	33	inhibitor	0.1536809889825205	PEMETREXED DISODIUM	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.063160791	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.004370177	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.084553416	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.048394167	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.2536602475154323	N-(PHENETHYLCARBAMOTHIOYL)BENZAMIDE	chembl:CHEMBL1448292	CHEMBL:CHEMBL1448292	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.003566128	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.6482428547616604	JAK2 INHIBITOR AZD1480	ncit:C91394	JAK2 INHIBITOR AZD1480	FALSE	FALSE	TRUE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.1684738114514262	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	SJ000295151	chembl:CHEMBL590660	CHEMBL:CHEMBL590660	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	CGI	2/1/22	NULL	0.1621858570986702	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
RPS6KB2	hgnc:10437	RPS6KB2	ChEMBL	33	inhibitor	2.625383561784725	LY-2780301	chembl:CHEMBL3545134	LY-2780301	FALSE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TdgClinicalTrial	Jan-14	NULL	1.014640990061729	DESMOPRESSIN	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:1787	hgnc:2977	TRDMT1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7797	ncit:C116891	GALUNISERTIB	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5651	iuphar.ligand:5651	1-STEAROYL-LYSOPHOSPHATIDYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:5526	iuphar.ligand:5526	ABNORMAL CANNABIDIOL	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.032342267	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	TCMDC-123927	chembl:CHEMBL531268	CHEMBL:CHEMBL531268	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.08178765	HYDROXYPROGESTERONE	ncit:C87242	HYDROXYPROGESTERONE	FALSE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	PharmGKB	4/5/24	NULL	0.2778183663264259	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.007184958	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	1.790034246671403	Practolol	rxcui:8620	PRACTOLOL	TRUE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.038159645	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.055859225	ACECLIDINE	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.3977853881492007	OLEOYLETHANOLAMIDE	iuphar.ligand:2661	N-OLEOYLETHANOLAMIDE	FALSE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	0.3500511415712966	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	ISONIAZID	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.057260274	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.040235763	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.042073455	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	MECLOFENAMATE SODIUM	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:7707	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:1489	iuphar.ligand:1489	DNPA	FALSE	FALSE	FALSE
CD14	hgnc:1628	CD14	NCI	14-Sep-17	NULL	0.2447910080918158	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
SOMATOSTATIN RECEPTOR TYPE 3	hgnc:11332	SSTR3	TTD	2020.06.01	NULL	3.500511415712966	ODT-8	chembl:CHEMBL452157	CHEMBL:CHEMBL452157	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.025123288	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.010205573	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	P-CYANOCHALCONE	chembl:CHEMBL445153	CHEMBL:CHEMBL445153	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.018962684	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002236844	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.3017682254924971	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.023493365	ethosuximide	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.03729238	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TACR2	hgnc:11527	TACR2	ChEMBL	33	inhibitor	10.50153424713889	NEPADUTANT	ncit:C84001	NEPADUTANT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TCMDC-125788	chembl:CHEMBL529986	CHEMBL:CHEMBL529986	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	NCI	14-Sep-17	NULL	0.729273212	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.1143957978991165	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.1346350544504987	Urapidil	rxcui:39230	URAPIDIL	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.0296486	Prochlorperazine	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1623	iuphar.ligand:1623	ENDOMORPHIN-1	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	antibody	0.525076712	IUPHAR.LIGAND:9172	rxcui:1855735	OLARATUMAB	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.099220845	NVP-BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.2386712328895204	FLECAINIDE	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.1875273972703375	IUPHAR.LIGAND:565	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.069454592	Taxol	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	0.525076712	IMCgp100	rxcui:2590743	TEBENTAFUSP	TRUE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.066297565	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CancerCommons	25-Jul-13	inhibitor	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CD44	hgnc:1681	CD44	NCI	14-Sep-17	NULL	0.6141248097742047	MOMETASONE FUROATE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
PARP2	hgnc:272	PARP2	CancerCommons	25-Jul-13	inhibitor	2.187819634820604	ABT-888	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.082115757	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	CGI	2/1/22	NULL	0.1438566335224507	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
DDR2	hgnc:2731	DDR2	CGI	2/1/22	NULL	0.9546849315580819	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.038741518	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CGI	2/1/22	NULL	0.087782887	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.013286354	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MKI67	hgnc:7107	MKI67	CGI	2/1/22	NULL	0.5357925636295356	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	1.750255707856483	CANCER VACCINE	ncit:C1663	ANTINEOPLASTIC VACCINE	FALSE	FALSE	FALSE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	0.7501095890813498	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	CGI	2/1/22	NULL	0.2234869519440402	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.2365210416022274	OXYPHENCYCLIMINE HYDROCHLORIDE	rxcui:91164	OXYPHENCYCLIMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	1.381780822	ARGATROBAN	rxcui:15202	ARGATROBAN	TRUE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.1392776425349987	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.2966535098061835	QUINAPRIL HYDROCHLORIDE	rxcui:235759	QUINAPRIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	BIPERIDEN HYDROCHLORIDE	rxcui:91154	BIPERIDEN HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC12A1	hgnc:10910	SLC12A1	ChEMBL	33	inhibitor	0.9376369863516875	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.042619863	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CD82	hgnc:6210	CD82	NCI	14-Sep-17	NULL	8.751278539282415	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.661861402	RIZATRIPTAN BENZOATE	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	3.281729452230906	METHANTHELINE BROMIDE	rxcui:91163	METHANTHELINE BROMIDE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	ChEMBL	33	inhibitor	0.7693431682885642	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN LISPRO PROTAMINE RECOMBINANT	chembl:CHEMBL1201611	INSULIN LISPRO PROTAMINE RECOMBINANT	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.032003863	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
CD86	hgnc:1705	CD86	NCI	14-Sep-17	NULL	0.1356787370431382	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.6543011991986852	PHENTERMINE HYDROCHLORIDE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.4293851619741372	ATOMOXETINE HYDROCHLORIDE	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.032003863	METHYLPHENIDATE HYDROCHLORIDE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.3271505995993426	TAPENTADOL HYDROCHLORIDE	rxcui:857492	TAPENTADOL HYDROCHLORIDE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	1.032937794800547	ETONOGESTREL	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	CODEINE PHOSPHATE	rxcui:2672	CODEINE PHOSPHATE	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.1881995384791917	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.035145697	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.02875557	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.1591141552596803	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.067897851	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.034970144	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.035719504	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.1521961485092594	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.033875917	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.1209854175937661	DEPSIPEPTIDE	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.2019525816757481	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.070574827	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.2375912725597036	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.2333674277141977	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.1154014752432845	NAPHAZOLINE HYDROCHLORIDE	rxcui:82054	NAPHAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1339481409073839	NAPHAZOLINE HYDROCHLORIDE	rxcui:82054	NAPHAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.087222045	NAPHAZOLINE HYDROCHLORIDE	rxcui:82054	NAPHAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.2586584789935689	GLIPIZIDE	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
COIL	hgnc:2184	COIL	NCI	14-Sep-17	NULL	35.00511415712966	ANTI-P80	ncit:C2000	TP3 IMMUNOTOXIN	FALSE	FALSE	FALSE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	0.1544343271638073	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.020465128	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.014617949	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
ODC1	hgnc:8109	ODC1	ChEMBL	33	inhibitor	10.50153424713889	EFLORNITHINE HYDROCHLORIDE	rxcui:81945	EFLORNITHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1077080435603989	D4T	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
LAMB2	hgnc:6487	LAMB2	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
LAMC1	hgnc:6492	LAMC1	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.026418954	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
COL4A5	hgnc:2207	COL4A5	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.076208521	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
COL24A1	hgnc:20821	COL24A1	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
COL4A2	hgnc:2203	COL4A2	ChEMBL	33	cleavage	0.4605936073306535	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
COL6A2	hgnc:2212	COL6A2	ChEMBL	33	cleavage	0.4605936073306535	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.212581665	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
COL1A1	hgnc:2197	COL1A1	ChEMBL	33	cleavage	0.1973972602845657	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.8751278539282416	FAS-LIGAND	ncit:C1538	RECOMBINANT FAS LIGAND	FALSE	FALSE	FALSE
COL11A2	hgnc:2187	COL11A2	ChEMBL	33	cleavage	0.138178082	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.251232877	OXYBUTYNIN CHLORIDE	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.085239726	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.055155117	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	NCI	14-Sep-17	NULL	0.7001022831425933	RANTES	ncit:C1211	RECOMBINANT RANTES	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.033919684	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.056097939	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.091583148	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.100976291	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
CTSG	hgnc:2532	CTSG	NCI	14-Sep-17	NULL	6.563458904461812	SULFONE	ncit:C849	SULFONE ANTI-INFECTIVE AGENT	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.1022876712383659	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.036770078	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
KCNK18	hgnc:19439	KCNK18	ChEMBL	33	potentiator	0.3387591692625452	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	NCI	14-Sep-17	NULL	0.1704794520639431	RIFAMPIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	0.5303805175322677	ADEFOVIR DIPIVOXIL	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	modulator	0.1143957978991165	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.048083948	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.052090944	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.019577804	8-MOP	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.057574201	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.076765601	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.070574827	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.3431873936973497	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.074163377	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.1988926940746003	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.05293112	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.055622533	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.070010228	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.035598421	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.032173818	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.066676408	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.013515488	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	1.458546423213736	METHSUXIMIDE	rxcui:47858	METHSUXIMIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1183271464466354	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1000146118775133	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.283060222	BESTATIN	ncit:C1015	UBENIMEX	FALSE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	6.058577450272442	EVOLOCUMAB	rxcui:1665684	EVOLOCUMAB	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.028413242	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.043902735	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.064824285	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	ChEMBL	33	inhibitor	0.7925686224255775	RAVOXERTINIB	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.037398626	PTK INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	ChEMBL	33	inhibitor	0.077217164	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	ChEMBL	33	inhibitor	0.1544343271638073	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	ChEMBL	33	inhibitor	0.096521454	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.078136416	GSK-2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
RPS6KB1	hgnc:10436	RPS6KB1	ChEMBL	33	inhibitor	0.28382525	LY-2780301	chembl:CHEMBL3545134	LY-2780301	FALSE	FALSE	FALSE
FGF4	hgnc:3682	FGF4	NCI	14-Sep-17	NULL	0.6563458904461812	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.1479089330582944	LY-2780301	chembl:CHEMBL3545134	LY-2780301	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.2465148884304905	MK-2201	chembl:CHEMBL3545000	MK-2201	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.022099188	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.041085815	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
GABPA	hgnc:4071	GABPA	NCI	14-Sep-17	NULL	0.2215513554248712	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	4.109296009750004	ENSARTINIB	ncit:C102754	ENSARTINIB	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	inhibitor	6.300920548	MSX-122	drugbank:DB12715	MSX-122	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.006649908	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.006896201	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GAL	hgnc:4114	GAL	NCI	14-Sep-17	NULL	1.640864726115453	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
TRPV4	hgnc:18083	TRPV4	ChEMBL	33	inhibitor	3.889457128569962	GSK2798745	drugbank:DB16033	GSK2798745	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1143957978991165	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
HCK	hgnc:4840	HCK	ChEMBL	33	inhibitor	0.1562728310586145	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	1.419126249613364	BURAPITANT	ncit:C90718	BURAPITANT	FALSE	FALSE	FALSE
GATA2	hgnc:4171	GATA2	NCI	14-Sep-17	NULL	0.3281729452230906	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
HRH4	hgnc:17383	HRH4	ChEMBL	33	inhibitor	7.160136986685614	TOREFORANT	ncit:C152698	TOREFORANT	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	1.591141552596803	SUFUGOLIX	ncit:C97486	SUFUGOLIX	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.4449802647092754	PRATOSARTAN	ncit:C72935	PRATOSARTAN	FALSE	FALSE	FALSE
SLC22A6	hgnc:10970	SLC22A6	ChEMBL	33	inhibitor	1.640864726115453	PRATOSARTAN	ncit:C72935	PRATOSARTAN	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.1209854175937661	AFACIFENACIN	ncit:C90741	AFACIFENACIN	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.175610941	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
LTB4R	hgnc:6713	LTB4R	ChEMBL	33	inhibitor	6.563458904461812	AMELUBANT	ncit:C73299	AMELUBANT	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	0.1583941817064691	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	0.5048814541893701	NONABINE	ncit:C72950	NONABINE	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	0.6403374540938354	AZD1386	iuphar.ligand:7820	AZD1386	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.2778183663264258	GW468816	chembl:CHEMBL1207366	GW468816	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.8975670296699915	AMINOGLYCOSIDES	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	2.917092846427472	ISPRONICLINE	ncit:C65986	ISPRONICLINE	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.099446347	AZD1305	chembl:CHEMBL3545169	AZD1305	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.6731752722524935	TRAXOPRODIL	ncit:C87769	TRAXOPRODIL	FALSE	FALSE	FALSE
CHRNA6	hgnc:15963	CHRNA6	ChEMBL	33	agonist	2.187819634820604	POZANICLINE	ncit:C81045	POZANICLINE	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.5000730593875667	PERMETHRIN	rxcui:33199	PERMETHRIN	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.5357925636295356	RADIPRODIL	ncit:C152143	RADIPRODIL	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.013817808	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNG1	hgnc:6248	KCNG1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
GTF2B	hgnc:4648	GTF2B	NCI	14-Sep-17	NULL	8.751278539282415	PC4	ncit:C2651	SILICON PHTHALOCYANINE 4	FALSE	FALSE	FALSE
KCNV1	hgnc:18861	KCNV1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNH5	hgnc:6254	KCNH5	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
HES1	hgnc:5192	HES1	NCI	14-Sep-17	NULL	1.154014752432846	ALL-TRANS-RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
KCNF1	hgnc:6246	KCNF1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNH7	hgnc:18863	KCNH7	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	1.944728564284981	CA19-9	ncit:C327	CA19-9 ANTIGEN	FALSE	FALSE	FALSE
KCNC2	hgnc:6234	KCNC2	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.012501826	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNG4	hgnc:19697	KCNG4	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.2160809515872201	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
KCNH6	hgnc:18862	KCNH6	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNA10	hgnc:6219	KCNA10	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	1.944728564284981	EQUINE CHORIONIC GONADOTROPIN	chembl:CHEMBL1201509	GONADOTROPIN, CHORIONIC	TRUE	FALSE	FALSE
KCNS2	hgnc:6301	KCNS2	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.057177137	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	positive modulator	0.4234489615781814	MK-8777	chembl:CHEMBL3707401	MK-8777	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	positive modulator	0.596678082	MK-8777	chembl:CHEMBL3707401	MK-8777	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	1.842374429322613	GP100	ncit:C2386	GP100 ANTIGEN	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	positive modulator	0.3977853881492007	MK-8777	chembl:CHEMBL3707401	MK-8777	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.42006137	ALEGLITAZAR	ncit:C72687	ALEGLITAZAR	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.1752592497853621	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.106290832	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1584738568481725	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.04464938	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.1434635826111871	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.652269208	FEDRATINIB	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.2536602475154323	PACRITINIB	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1405827877796372	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.1773907812016706	SARIZOTAN HYDROCHLORIDE	ncit:C76654	SARIZOTAN HYDROCHLORIDE	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.1017590527823536	ESMIRTAZAPINE MALEATE	ncit:C76940	ESMIRTAZAPINE MALEATE	FALSE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	3.750547945	LATANOPROSTENE BUNOD	rxcui:1988390	LATANOPROSTENE BUNOD	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.4817217544559128	BEVENOPRAN	ncit:C169810	BEVENOPRAN	FALSE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	inhibitor	2.386712328895204	LIXIVAPTAN	ncit:C74429	LIXIVAPTAN	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.053579256	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
IL17RA	hgnc:5985	IL17RA	ChEMBL	33	inhibitor	35.00511415712966	BRODALUMAB	rxcui:1872251	BRODALUMAB	TRUE	FALSE	FALSE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	activator	0.4688184931758437	FLINDOKALNER	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
IL5RA	hgnc:6017	IL5RA	ChEMBL	33	inhibitor	52.50767123569449	BENRALIZUMAB	rxcui:1989100	BENRALIZUMAB	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.8334550989792777	ZALUTUMUMAB	ncit:C64620	ZALUTUMUMAB	FALSE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	modulator	1.721562991334245	ULIPRISTAL	rxcui:1005920	ULIPRISTAL ACETATE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	inhibitor	4.039051633514961	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.034318739	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	negative modulator	0.035719504	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
MYL3	hgnc:7584	MYL3	ChEMBL	33	activator	2.187819634820604	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
NAMPT	hgnc:30092	NAMPT	ChEMBL	33	inhibitor	10.50153424713889	TEGLARINAD CHLORIDE	ncit:C68931	TEGLARINAD CHLORIDE	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	ChEMBL	33	inhibitor	3.750547945	FONTOLIZUMAB	ncit:C87765	FONTOLIZUMAB	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	NCI	14-Sep-17	NULL	0.010857666	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	inhibitor	4.200613699	ADECATUMUMAB	ncit:C82358	ADECATUMUMAB	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	ONCOLYSIN B	chembl:CHEMBL2109308	ONCOLYSIN B	FALSE	FALSE	FALSE
F8	hgnc:3546	F8	ChEMBL	33	inhibitor	9.26605963	TB-402	drugbank:DB06050	TB-402	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.072725306	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	ChEMBL	33	inhibitor	1.29648571	ABX-IL8	chembl:CHEMBL2109616	ABX-IL8	FALSE	FALSE	FALSE
BACE1	hgnc:933	BACE1	ChEMBL	33	inhibitor	2.019525817	ELENBECESTAT	ncit:C169934	ELENBECESTAT	FALSE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.6731752722524935	FENFLURAMINE HYDROCHLORIDE	rxcui:82018	FENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.032134438	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	blocker	0.1262203635473425	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.042968634	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	blocker	0.2019525816757481	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	blocker	0.1346350544504987	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	0.1286952726365061	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	inhibitor	0.041739007	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.4070362111294147	DDC	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
AKR1B1	hgnc:381	AKR1B1	ChEMBL	33	inhibitor	1.346350544504987	TOLRESTAT	rxcui:38386	TOLRESTAT	TRUE	FALSE	FALSE
HTR1F	hgnc:5292	HTR1F	ChEMBL	33	inhibitor	0.280789686	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR6	hgnc:5301	HTR6	ChEMBL	33	inhibitor	0.2059124362184098	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.054271495	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
IFNG	hgnc:5438	IFNG	ChEMBL	33	inhibitor	1.875273972703375	AMG-811	chembl:CHEMBL2109450	AMG-811	FALSE	FALSE	FALSE
IFNA21	hgnc:5424	IFNA21	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.6105543166941221	PHOSPHODIESTERASE INHIBITOR	ncit:C744	PHOSPHODIESTERASE INHIBITOR	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.044878351	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	inhibitor	0.051782713	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	NCI	14-Sep-17	NULL	0.072125922	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
HTR1E	hgnc:5291	HTR1E	ChEMBL	33	inhibitor	0.4039051633514962	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	ChEMBL	33	binder	0.2344092465879218	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	modulator	0.4861821410712453	MEDI-565	chembl:CHEMBL2109372	MEDI-565	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	NCI	14-Sep-17	NULL	0.040703621	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.640864726115453	DAPAGLIFLOZIN	rxcui:1486966	DAPAGLIFLOZIN PROPANEDIOL	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.031650194	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.3125456621172291	LOFEXIDINE HYDROCHLORIDE	rxcui:235853	LOFEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.032055965	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	0.525076712	ANAGLIPTIN	ncit:C96202	ANAGLIPTIN	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.1117184494376478	NITRENDIPINE	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	NCI	14-Sep-17	NULL	0.2853677784548614	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
MGAM2	hgnc:28101	MGAM2	ChEMBL	33	inhibitor	6.563458904461812	CELGOSIVIR	ncit:C79567	CELGOSIVIR	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	ChEMBL	33	inhibitor	0.182318303	CELGOSIVIR	ncit:C79567	CELGOSIVIR	FALSE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	positive modulator	0.7721716358190367	OLINCIGUAT	ncit:C153148	OLINCIGUAT	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	1.432027397337122	CIMICOXIB	ncit:C77551	CIMICOXIB	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.3431873936973497	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.3387591692625452	BREPOCITINIB	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.3125456621172291	CILOMILAST	ncit:C95232	CILOMILAST	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2983390411119005	TETOMILAST	ncit:C90922	TETOMILAST	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.3977853881492007	MK-0767	drugbank:DB12055	MK-0767	FALSE	FALSE	FALSE
C5AR1	hgnc:1338	C5AR1	ChEMBL	33	inhibitor	6.563458904461812	AVDORALIMAB	ncit:C163020	AVDORALIMAB	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.1630673019742065	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.8140724222588294	PF-00610355	drugbank:DB11871	PF-00610355	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	ChEMBL	33	inhibitor	2.763561643983921	BAY-1093884	chembl:CHEMBL4297904	BAY-1093884	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.1944728564284981	AZT	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	ChEMBL	33	inhibitor	1.810609352954982	DAZODALIBEP	ncit:C175714	DAZODALIBEP	FALSE	FALSE	FALSE
INPP5D	hgnc:6079	INPP5D	ChEMBL	33	activator	26.25383561784724	ROSIPTOR	ncit:C152258	ROSIPTOR	FALSE	FALSE	FALSE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.251232877	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.5707355569097228	SNX 5422	ncit:C141504	SNX 5422	FALSE	FALSE	FALSE
PPP3CA	hgnc:9314	PPP3CA	ChEMBL	33	inhibitor	6.563458904461812	VOCLOSPORIN	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.789589041	PPD	rxcui:1362740	4-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.3061671792168775	GALLIUM NITRATE	rxcui:25544	GALLIUM NITRATE	TRUE	FALSE	FALSE
LGALS3	hgnc:6563	LGALS3	ChEMBL	33	inhibitor	6.563458904461812	DAVANAT	drugbank:DB15311	DAVANAT	FALSE	FALSE	FALSE
IFNB1	hgnc:5434	IFNB1	ChEMBL	33	inhibitor	26.25383561784724	PF-06823859	chembl:CHEMBL4297808	PF-06823859	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.3241214273808302	FLYSYN	chembl:CHEMBL4650288	FLYSYN	FALSE	FALSE	FALSE
IL7	hgnc:6023	IL7	NCI	14-Sep-17	NULL	1.591141552596803	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	2.333674277141977	ADL-5747	chembl:CHEMBL4297345	ADL-5747	FALSE	FALSE	FALSE
IL8RB	hgnc:6027	CXCR2	NCI	14-Sep-17	NULL	0.5303805175322677	NITROGEN MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
IL1RAP	hgnc:5995	IL1RAP	ChEMBL	33	inhibitor	8.751278539282415	SPESOLIMAB	rxcui:2610417	SPESOLIMAB	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	agonist	0.2500365296937833	TEREVALEFIM	ncit:C175863	TEREVALEFIM	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	1.458546423213736	PARNAPARIN SODIUM	ncit:C132777	PARNAPARIN SODIUM	FALSE	FALSE	FALSE
F8	hgnc:3546	F8	ChEMBL	33	positive modulator	0.7721716358190367	ANTIHEMOPHILIC FACTOR, HUMAN RECOMBINANT	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.8751278539282416	AR-67	iuphar.ligand:8919	AR-67	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.1296485709523321	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
F11	hgnc:3529	F11	ChEMBL	33	inhibitor	2.763561643983921	ABELACIMAB	ncit:C169755	ABELACIMAB	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.04321619	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	agonist	1.969037671338543	RESIQUIMOD	ncit:C63958	RESIQUIMOD	FALSE	FALSE	FALSE
LIPC	hgnc:6619	LIPC	NCI	14-Sep-17	NULL	0.8204323630577265	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
IL18RAP	hgnc:5989	IL18RAP	ChEMBL	33	agonist	17.50255707856483	IBOCTADEKIN	ncit:C1680	IBOCTADEKIN	FALSE	FALSE	FALSE
CTSK	hgnc:2536	CTSK	ChEMBL	33	inhibitor	5.834185692854944	ONO-5334	iuphar.ligand:10747	ONO-5334	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.4363518385237769	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
PDE9A	hgnc:8795	PDE9A	ChEMBL	33	inhibitor	6.563458904461812	IRSENONTRINE	ncit:C179092	IRSENONTRINE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.055563673	LAZERTINIB	ncit:C148147	LAZERTINIB	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.5834185692854944	ADL-5859	iuphar.ligand:9004	ADL5859	FALSE	FALSE	FALSE
LPAR2	hgnc:3168	LPAR2	NCI	14-Sep-17	NULL	0.9460841664089098	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	ChEMBL	33	inhibitor	15.75230137070834	TECARFARIN	ncit:C152523	TECARFARIN	FALSE	FALSE	FALSE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	1.750255707856483	MYCOPHENOLATE SODIUM	rxcui:408142	MYCOPHENOLATE SODIUM	TRUE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.064268875	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.3365876361262467	RELENOPRIDE	ncit:C152177	RELENOPRIDE	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.046965717	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.046965717	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1061475833605683	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
NOX4	hgnc:7891	NOX4	ChEMBL	33	inhibitor	78.76150685354175	SETANAXIB	ncit:C166721	SETANAXIB	FALSE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	ChEMBL	33	agonist	2.019525817	ROVAZOLAC	ncit:C152263	ROVAZOLAC	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1562728310586145	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	ChEMBL	33	inhibitor	5.527123287967842	BREQUINAR	ncit:C1560	BREQUINAR	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.082364974	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.3947945205691315	FONADELPAR	ncit:C170003	FONADELPAR	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	binder	0.3889457128569963	FINGOLIMOD LAURYL SULFATE	rxcui:2610292	FINGOLIMOD LAURYL SULFATE	TRUE	FALSE	FALSE
ME3	hgnc:6985	ME3	NCI	14-Sep-17	NULL	0.921187215	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.2419708351875322	NEZULCITINIB	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1215455352678113	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.064824285	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.023652104	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.053217234	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
MT1F	hgnc:7398	MT1F	NCI	14-Sep-17	NULL	0.6105543166941221	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1520492410300034	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2059124362184098	MGAH22	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.08334551	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1183271464466354	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.047712559	ENMD 2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	ADOZELESIN	ncit:C1270	ADOZELESIN	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1000146118775133	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
IL-12B	hgnc:5970	IL12B	ClearityFoundationClinicalTrial	15-Jun-13	other/unknown	3.750547945	CID 446414	drugbank:DB05953	EGEN-001	FALSE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.03261346	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.5903640284436551	XL518	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.054953083	ALL-TRANS-RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6250913242344583	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
PRKAB1	hgnc:9378	PRKAB1	ClearityFoundationClinicalTrial	15-Jun-13	activator	0.1172046232939609	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.054953083	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.030176823	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.6250913242344583	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	PLICAMYCIN	rxcui:6995	PLICAMYCIN	TRUE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.034487797	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.252440727	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.6731752722524936	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003632492	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	EDARAVONE	rxcui:1921877	EDARAVONE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.201178817	CARBOFENOTION	chembl:CHEMBL452866	CARBOFENOTION	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.015858554	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.5966780822238011	CLODRONATE	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ISOQUINE	chembl:CHEMBL147587	ISOQUINE	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.1342907192728759	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.030996264	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1136529680426287	PHENAMIL METHANESULFONATE	chembl:CHEMBL1256775	PHENAMIL METHANESULFONATE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	LASSBIO-123	chembl:CHEMBL573111	CHEMBL:CHEMBL573111	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	1.479089330582943	ANTI-ULCER AGENT	ncit:C29701	ANTI-ULCER AGENT	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	FUROXAN	chembl:CHEMBL336467	FUROXAN	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.05309168	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1041818873724097	ESCULETIN	iuphar.ligand:5180	ESCULETIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.011812749	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.0095957	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.201178817	FLAVANOMAREIN	chembl:CHEMBL1405715	FLAVANOMAREIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	BREFELDIN A	drugbank:DB07348	BREFELDIN A	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	5.834185692854944	TOPOISOMERASE-I INHIBITOR	ncit:C1904	TOPOISOMERASE-I INHIBITOR	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.4070362111294147	GAMBOGIC AMIDE	chembl:CHEMBL444109	GAMBOGIC AMIDE	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.040235763	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.064033745	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.2488515224440497	SJ000291458	chembl:CHEMBL592598	CHEMBL:CHEMBL592598	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.1100789753368857	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	SJ000124275	chembl:CHEMBL602150	CHEMBL:CHEMBL602150	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.01795748	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	TCMDC-123598	chembl:CHEMBL547269	CHEMBL:CHEMBL547269	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.077846807	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	NSC-699479	chembl:CHEMBL1701915	CHEMBL:CHEMBL1701915	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.218327115	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.1750255707856483	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	TDR81525	chembl:CHEMBL1422704	CHEMBL:CHEMBL1422704	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.030670369	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	0.6563458904461812	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.002827097	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.4449802647092754	DNDI1417478	chembl:CHEMBL1972216	CHEMBL:CHEMBL1972216	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	4.375639269641208	TRISMETHOXYRESVERATROL	chembl:CHEMBL296411	TRISMETHOXYRESVERATROL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	TCMDC-123598	chembl:CHEMBL547269	CHEMBL:CHEMBL547269	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	NEOCUPROINE	chembl:CHEMBL375781	NEOCUPROINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	NSC-116702	chembl:CHEMBL1477383	CHEMBL:CHEMBL1477383	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	GNF-PF-2755	chembl:CHEMBL600738	CHEMBL:CHEMBL600738	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.7721716358190367	DIMETHYLPHENYLPIPERAZINIUM IODIDE	chembl:CHEMBL47814	DIMETHYLPHENYLPIPERAZINIUM IODIDE	FALSE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.8078103267029922	REL-3,4-DICAFFEOYLQUINIC ACID	iuphar.ligand:12549	ISOCHLOROGENIC ACID B	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.016590101	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.018860514	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.065964411	EQUILIN	ncit:C29020	EQUILIN	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.315361389	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004557958	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	SESAMIN	rxcui:2593413	SESAMIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	TCMDC-123927	chembl:CHEMBL531268	CHEMBL:CHEMBL531268	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NARASIN	rxcui:1314370	NARASIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.1521961485092594	FLUAZINAM	chembl:CHEMBL1878267	FLUAZINAM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.014537008	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.043430663	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	FENOLDOPAM BROMIDE	chembl:CHEMBL1256646	FENOLDOPAM BROMIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.2900976311364336	NSC-22357	chembl:CHEMBL327209	CHEMBL:CHEMBL327209	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	WAY-629	chembl:CHEMBL258465	CHEMBL:CHEMBL258465	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.018962684	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	ISOBOLDINE	chembl:CHEMBL462880	ISOBOLDINE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.078958904	TYRPHOSTIN 1	iuphar.ligand:5917	AG 9	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	TCMDC-124416	chembl:CHEMBL530664	CHEMBL:CHEMBL530664	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-109483	chembl:CHEMBL507159	CHEMBL:CHEMBL507159	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.013415348	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.1798207919030633	SJ000047241	chembl:CHEMBL601933	CHEMBL:CHEMBL601933	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002269228	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2822993077187876	IRETOL	chembl:CHEMBL1606248	IRETOL	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.083744292	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	METHYL 3-(2,5-DIHYDROXYPHENYL)ACRYLATE	chembl:CHEMBL17329	CHEMBL:CHEMBL17329	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1400204566285186	2-PHENYLPHENOL	rxcui:236677	2-PHENYLPHENOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE	chembl:CHEMBL1513686	12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE	FALSE	FALSE	FALSE
ERAP1	hgnc:18173	ERAP1	DTC	9/2/20	NULL	4.375639269641208	UMBELLIFERONE	chembl:CHEMBL51628	UMBELLIFERONE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.075442056	HELIOMYCIN	ncit:C75147	HELIOMYCIN	FALSE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	1.193356164447602	TCMDC-125603	chembl:CHEMBL528734	CHEMBL:CHEMBL528734	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	TRICLOSAN	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.1405827877796372	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.011316308	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.011585982	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.056826484	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.047561296	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.020470827	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	OXATOMIDE	rxcui:54236	OXATOMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.018354192	DILTIAZEM	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	2.838252499226729	RO-4858154	chembl:CHEMBL2203708	CHEMBL:CHEMBL2203708	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.028536778	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.046303061	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.010564924	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	GNF-PF-4945	chembl:CHEMBL585628	CHEMBL:CHEMBL585628	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.014114965	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.091159151	PIRARUBICIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	GNF-PF-3237	chembl:CHEMBL602206	CHEMBL:CHEMBL602206	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.029918901	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.017751072	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.016408647	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.002904025	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.012211086	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	CYSTEINE METHYL-ESTER HCL	chembl:CHEMBL1426508	CHEMBL:CHEMBL1426508	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.04321619	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.2386712328895204	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.006162872	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TROVAFLOXACIN MESYLATE	rxcui:221177	TROVAFLOXACIN MESYLATE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	GNF-PF-4012	chembl:CHEMBL584269	CHEMBL:CHEMBL584269	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.053854022	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.085239726	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.033948925	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.020696756	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2289578687602957	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.214025834	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.088396753	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	GNF-PF-516	chembl:CHEMBL602970	CHEMBL:CHEMBL602970	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	TCMDC-124336	chembl:CHEMBL527271	CHEMBL:CHEMBL527271	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ANCITABINE	ncit:C80636	ANCITABINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.003349772	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	SJ000001516	chembl:CHEMBL592316	CHEMBL:CHEMBL592316	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	CGP-7930	iuphar.ligand:1079	CGP7930	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.375054795	TCMDC-125319	chembl:CHEMBL527586	CHEMBL:CHEMBL527586	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	2.282942227638891	RO-3201195	chembl:CHEMBL203567	RO-3201195	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	NSC-81747	chembl:CHEMBL1371696	CHEMBL:CHEMBL1371696	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	METHOXYVONE	chembl:CHEMBL1591080	METHOXYVONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	DTC	9/2/20	NULL	1.973972602845657	IB-MECA	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.015839418	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	NSC-102045	chembl:CHEMBL483633	CHEMBL:CHEMBL483633	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MONATEPIL	ncit:C83970	MONATEPIL	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.1121958787087489	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.3500511415712966	GNF-PF-4102	chembl:CHEMBL596836	CHEMBL:CHEMBL596836	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	PIMPINELLIN	chembl:CHEMBL1491809	PIMPINELLIN	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.038187397	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003789252	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007003824	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	RO-106-9920	chembl:CHEMBL271023	CHEMBL:CHEMBL271023	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.025244073	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.000662725	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	SJ000111875	chembl:CHEMBL590949	CHEMBL:CHEMBL590949	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004237907	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	SIB-1893	iuphar.ligand:1432	SIB-1893	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.027563082	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002529881	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.021215221	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	CLOFAZIMINE	rxcui:2592	CLOFAZIMINE	TRUE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.2117244807890907	DIPYRONE SODIUM	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.5048814541893701	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	CYSTAMINE DIHYDROCHLORIDE	ncit:C97356	CYSTAMINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.1235474617310458	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	EVANS BLUE	rxcui:4191	EVANS BLUE	FALSE	FALSE	FALSE
PRNP	hgnc:9449	PRNP	DTC	9/2/20	NULL	7.501095890813499	BREFELDIN A	drugbank:DB07348	BREFELDIN A	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	OCTADEC-17-YNOIC ACID	iuphar.ligand:8851	17-OCTADECYNOIC ACID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	CID 3238892	chembl:CHEMBL261118	CHEMBL:CHEMBL261118	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	TCMDC-123598	chembl:CHEMBL547269	CHEMBL:CHEMBL547269	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.08334551	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	ANGUIDIN	chembl:CHEMBL433680	ANGUIDIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.034521809	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.036718651	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	NSC-81747	chembl:CHEMBL1371696	CHEMBL:CHEMBL1371696	FALSE	FALSE	FALSE
TACR3	hgnc:11528	TACR3	DTC	9/2/20	NULL	5.834185692854944	RO-4861497	chembl:CHEMBL2203707	CHEMBL:CHEMBL2203707	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.040390516	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.013624201	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	CGP-7930	iuphar.ligand:1079	CGP7930	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.2051080907644316	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.081407242	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-125149	chembl:CHEMBL547175	CHEMBL:CHEMBL547175	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	TCMDC-123516	chembl:CHEMBL547304	CHEMBL:CHEMBL547304	FALSE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	DTC	9/2/20	NULL	5.250767123569449	CLASTO-LACTACYSTIN BETA-LACTONE	chembl:CHEMBL490829	CHEMBL:CHEMBL490829	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-742865	chembl:CHEMBL102936	CHEMBL:CHEMBL102936	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.5645986154375752	N-(PHENETHYLCARBAMOTHIOYL)BENZAMIDE	chembl:CHEMBL1448292	CHEMBL:CHEMBL1448292	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	VU0080241	iuphar.ligand:6227	VU0080241	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	2.282942227638891	SERGEOLIDE	chembl:CHEMBL521373	SERGEOLIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	DNDI1417759	chembl:CHEMBL1446254	CHEMBL:CHEMBL1446254	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007873395	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.010295622	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	NSC-49789	chembl:CHEMBL469309	CHEMBL:CHEMBL469309	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008432935	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.038467158	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1071585127259071	NSC-699479	chembl:CHEMBL1701915	CHEMBL:CHEMBL1701915	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.035502144	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.061055432	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	DTC	9/2/20	NULL	0.1419126249613365	PIPERTRAMINE AMIDE	chembl:CHEMBL130835	PIPERTRAMINE AMIDE	FALSE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	2.500365296937833	22(S)-HYDROXYCHOLESTEROL	chembl:CHEMBL1243244	CHEMBL:CHEMBL1243244	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	CEPHARANTHINE	ncit:C83611	CEPHARANTHINE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.091159151	UH-301	iuphar.ligand:61	(S)-UH 301	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.01644462	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DEMETHOXYCURCUMIN	chembl:CHEMBL179512	DEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	RIMSULFURON	chembl:CHEMBL1867091	RIMSULFURON	FALSE	FALSE	FALSE
P2RY1	hgnc:8539	P2RY1	DTC	9/2/20	NULL	11.66837138570988	ISO-IANTHERAN A	chembl:CHEMBL240681	ISO-IANTHERAN A	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.210030685	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.020721259	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002175312	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	CAFFEIC ACID	rxcui:1311397	CAFFEIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	WARFARIN POTASSIUM	rxcui:82118	WARFARIN POTASSIUM	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.021484317	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW612286X	chembl:CHEMBL479079	GW612286X	FALSE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	0.100976291	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.025256215	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.072324616	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.364636606	SB-431542	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	ARBIDOL	ncit:C152799	UMIFENOVIR	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-718429A	chembl:CHEMBL505187	GSK-718429A	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.3977853881492008	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	RS-67506	iuphar.ligand:3230	RS67506	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	RILMENIDINE	rxcui:55679	RILMENIDINE	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.041672755	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	NSC-102045	chembl:CHEMBL483633	CHEMBL:CHEMBL483633	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.7395446652914718	THIOURACIL	ncit:C29856	THIOURACIL	FALSE	FALSE	FALSE
GPBAR1	hgnc:19680	GPBAR1	DTC	9/2/20	NULL	17.50255707856483	23(S)-METHYL-CHENODEOXYCHOLIC ACID	chembl:CHEMBL583611	CHEMBL:CHEMBL583611	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	BISPHENOL A	rxcui:1433347	BISPHENOL A	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.022315202	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.07631929	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CAMK1D	hgnc:19341	CAMK1D	DTC	9/2/20	NULL	0.1491695205559502	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.073954467	TCMDC-125575	chembl:CHEMBL587620	CHEMBL:CHEMBL587620	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	XANTHOPTERIN	chembl:CHEMBL1236854	XANTHOPTERIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	TCMDC-124336	chembl:CHEMBL527271	CHEMBL:CHEMBL527271	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007551801	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	GNF-PF-5029	chembl:CHEMBL1198140	CHEMBL:CHEMBL1198140	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009922085	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	SALICYLHYDROXAMIC ACID	drugbank:DB03819	SALICYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.010491043	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.05073205	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.092118721	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	FURAMIDINE	chembl:CHEMBL24057	FURAMIDINE	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.016829382	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
SUMO2	hgnc:11125	SUMO2	DTC	9/2/20	NULL	0.6403374540938354	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.4487835148349957	AMINOGLYCOSIDE ANTIBIOTIC	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW856804X	chembl:CHEMBL241517	GW856804X	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	UH-232	chembl:CHEMBL278751	CHEMBL:CHEMBL278751	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.028929846	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005712634	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.088322407	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	1.419126249613364	RO-4861497	chembl:CHEMBL2203707	CHEMBL:CHEMBL2203707	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	WAY-629	chembl:CHEMBL258465	CHEMBL:CHEMBL258465	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	ZERANOL	rxcui:1368476	ZERANOL	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008857569	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	5-NITRO-[1,10]PHENANTHROLINE	chembl:CHEMBL101815	CHEMBL:CHEMBL101815	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.060284353	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	FIDUXOSIN	ncit:C65682	FIDUXOSIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	IMETIT	iuphar.ligand:1250	IMETIT	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	PADIMATE O	rxcui:32786	PADIMATE-O	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.015839418	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	NIFLUMIC ACID	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.210030685	GNF-PF-3343	chembl:CHEMBL599943	CHEMBL:CHEMBL599943	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.003038638	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.075714018	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	JTC-801	iuphar.ligand:1692	JTC-801	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003131234	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
GPR12	hgnc:4466	GPR12	DTC	9/2/20	NULL	15.00219178	NEOCYCLOCITRINOL C	chembl:CHEMBL524981	NEOCYCLOCITRINOL C	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.012932924	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	LAVENDUSTIN A	ncit:C1142	LAVENDUSTIN A	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.014500876	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.016727516	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.013920379	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.015002192	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	SALMETEROL	rxcui:36117	SALMETEROL	TRUE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.072324616	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	ANISALDEHYDE	chembl:CHEMBL161598	ANISALDEHYDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.003371279	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.027855529	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	ACRIDIN-1-YLAMINE	chembl:CHEMBL146525	CHEMBL:CHEMBL146525	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.010346339	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.007012242	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.092118721	PHENAMIL METHANESULFONATE	chembl:CHEMBL1256775	PHENAMIL METHANESULFONATE	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1458546423213736	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.8204323630577265	TARIQUIDAR	ncit:C2246	TARIQUIDAR	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.044198376	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.051731696	GNF-PF-1134	chembl:CHEMBL600694	CHEMBL:CHEMBL600694	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2778183663264259	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.031310478	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.015744429	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	6-3'-DIMETHYLFLAVONE	chembl:CHEMBL137498	CHEMBL:CHEMBL137498	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	NSC-74429	chembl:CHEMBL1269022	CHEMBL:CHEMBL1269022	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	TRIPELENNAMINE HYDROCHLORIDE	rxcui:91063	TRIPELENNAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.046840028	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.041672755	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.02109589	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.010554306	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
PNMT	hgnc:9160	PNMT	NCI	14-Sep-17	NULL	8.751278539282415	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	(Z)-PIPLARTINE	chembl:CHEMBL1456697	(Z)-PIPLARTINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.015791781	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006381584	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.04464938	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	VANIPREVIR	ncit:C152828	VANIPREVIR	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	1.250182648468916	BOVINE CARTILAGE	ncit:C2418	BOVINE CARTILAGE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	BENZOTHIAZOL-2-YLAMINE	chembl:CHEMBL329785	CHEMBL:CHEMBL329785	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	RAC-NUTLIN-3	chembl:CHEMBL211045	CHEMBL:CHEMBL211045	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.009293393	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	QUINOLINIC ACID	drugbank:DB01796	QUINOLINIC ACID	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	PIRENOXINE	rxcui:228080	PIRENOXINE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.018860514	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ALTHIAZIDE	rxcui:17599	ALTHIAZIDE	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1801292323694494	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2220197515251353	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.017150962	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
PPP1R1A	hgnc:9286	PPP1R1A	NCI	14-Sep-17	NULL	1.981421556063943	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2580229544751573	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2328499833068492	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	NIHYDRAZONE	ncit:C175162	NIHYDRAZONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GITOXIGENIN	chembl:CHEMBL464658	GITOXIGENIN	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1944728564284981	TCMDC-124307	chembl:CHEMBL546865	CHEMBL:CHEMBL546865	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	INDOCYANINE GREEN SODIUM	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.015791781	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.017114626	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.035005114	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001750547	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	TENONITROZOLE	rxcui:236186	TENONITROZOLE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	4-BENZAMIDOPHENYLSTIBONIC ACID	chembl:CHEMBL1726814	CHEMBL:CHEMBL1726814	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.048618214	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	ERGOCRISTINE	chembl:CHEMBL446315	ERGOCRISTINE	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1458546423213736	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006488837	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.024467694	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	SJ000047241	chembl:CHEMBL601933	CHEMBL:CHEMBL601933	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.04464938	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
RHOA	hgnc:667	RHOA	DTC	9/2/20	NULL	1.154014752432846	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002436325	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.016910683	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
PASK	hgnc:17270	PASK	DTC	9/2/20	NULL	0.3977853881492008	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	1.141471113819445	RADANAMYCIN	chembl:CHEMBL383015	RADANAMYCIN	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	NCI	14-Sep-17	NULL	0.086789539	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.017047945	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.182318303	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	KAINIC ACID	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.014369915	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.019404165	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.1215455352678113	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	2.838252499226729	RO-4908594	chembl:CHEMBL2203704	CHEMBL:CHEMBL2203704	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	SJ000113107	chembl:CHEMBL589245	CHEMBL:CHEMBL589245	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.108711535	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.2651902587661338	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	2.692701089009974	131-IODINE	ncit:C1639	IODINE I-131	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.087512785	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.011540148	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.019483366	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.047518255	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
AKR1B10	hgnc:382	AKR1B10	DTC	9/2/20	NULL	8.751278539282415	TOLRESTAT	rxcui:38386	TOLRESTAT	TRUE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.024309107	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.1682938180631233	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.01037701	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.1750255707856483	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
RALA	hgnc:9839	RALA	NCI	14-Sep-17	NULL	6.563458904461812	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
RBP4	hgnc:9922	RBP4	DTC	9/2/20	NULL	4.039051633514962	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.006596441	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CHLORPYRIFOS-METHYL	ncit:C163642	CHLORPYRIFOS-METHYL	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	DTC	9/2/20	NULL	1.842374429322613	L-655708	chembl:CHEMBL52030	CHEMBL:CHEMBL52030	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DECYLUBIQUINONE	chembl:CHEMBL217894	DECYLUBIQUINONE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	2-ACETYLPYRIDINE N4(ETHYL)THIOSEMICARBAZONE	chembl:CHEMBL507986	CHEMBL:CHEMBL507986	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	DNDI1417268	chembl:CHEMBL1517542	CHEMBL:CHEMBL1517542	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	TCMDC-124640	chembl:CHEMBL547161	CHEMBL:CHEMBL547161	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
SDC1	hgnc:10658	SDC1	NCI	14-Sep-17	NULL	1.640864726115453	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	CYCLOHEXANONE OXIME	chembl:CHEMBL137035	CYCLOHEXANONE OXIME	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	4-NONYLPHENOL	rxcui:1788868	4-NONYLPHENOL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.016116535	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	CANDESARTAN CILEXETIL	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.1628144844517658	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.1944728564284981	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.02832129	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	DTC	9/2/20	NULL	3.621218705909965	CASEARINONE A	chembl:CHEMBL525043	CASEARINONE A	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.8204323630577265	RECOMBINANT HUMAN KERATINOCYTE GROWTH FACTOR	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	SCOULERINE	chembl:CHEMBL1235966	SCOULERINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	NSC-720622	chembl:CHEMBL1287980	CHEMBL:CHEMBL1287980	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.004251633	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.1400204566285186	FLUORODIFEN	chembl:CHEMBL1892429	FLUORODIFEN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	NSC-720622	chembl:CHEMBL1287980	CHEMBL:CHEMBL1287980	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	BISPHENOL A	rxcui:1433347	BISPHENOL A	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004051518	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	SJ000113107	chembl:CHEMBL589245	CHEMBL:CHEMBL589245	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.009423487	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	MOCLOBEMIDE	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005905046	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.043137707	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	TCMDC-125298	chembl:CHEMBL581152	CHEMBL:CHEMBL581152	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-638080	chembl:CHEMBL136344	CHEMBL:CHEMBL136344	FALSE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	2.625383561784724	IL-7	iuphar.ligand:4999	IL-7	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GR-4661	chembl:CHEMBL344127	CHEMBL:CHEMBL344127	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	E-GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	2.692701089009974	Y-27632	drugbank:DB08756	Y-27632	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	RO-194603	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.05073205	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.4773424657790409	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.4773424657790409	DNDI1417457	chembl:CHEMBL1530911	CHEMBL:CHEMBL1530911	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	GNF-PF-3832	chembl:CHEMBL261693	CHEMBL:CHEMBL261693	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.021484317	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.023493365	NEOSTIGMINE BROMIDE	rxcui:82055	NEOSTIGMINE BROMIDE	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.095468493	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	1.810609352954982	NIZATIDINE	rxcui:42319	NIZATIDINE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW679410X	chembl:CHEMBL202891	GW679410X	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	16-DEHYDROPREGNENOLONE ACETATE	chembl:CHEMBL1761683	CHEMBL:CHEMBL1761683	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.9053046764774912	MEXILETINE	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
HCAR2	hgnc:24827	HCAR2	DTC	9/2/20	NULL	5.834185692854944	ACIFRAN	ncit:C81534	ACIFRAN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.025147352	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
CCR6	hgnc:1607	CCR6	DTC	9/2/20	NULL	2.187819634820604	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1000146118775133	SL-327	iuphar.ligand:6008	MEK1/2 INHIBITOR	FALSE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	0.1553481397505754	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PENDIMETHALIN	chembl:CHEMBL1256630	PENDIMETHALIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.055839424	ALL-TRANS-RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PTGER4	hgnc:9596	PTGER4	DTC	9/2/20	NULL	0.7721716358190367	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	1.129197231	ACEBUTOLOL	rxcui:149	ACEBUTOLOL	TRUE	FALSE	FALSE
SENP1	hgnc:17927	SENP1	DTC	9/2/20	NULL	3.500511415712967	NOMIFENSINE MALEATE	rxcui:262302	NOMIFENSINE MALEATE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.050978322	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	QUINOLINIC ACID	drugbank:DB01796	QUINOLINIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TCMDC-123730	chembl:CHEMBL530280	CHEMBL:CHEMBL530280	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.067231333	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.020470827	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.6908904109959803	TCMDC-125603	chembl:CHEMBL528734	CHEMBL:CHEMBL528734	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.025147352	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	TCMDC-123634	chembl:CHEMBL530499	CHEMBL:CHEMBL530499	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	6-CHLOROMELATONIN	iuphar.ligand:1346	6-CL-MLT	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	DILTIAZEM	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	DNDI1417623	chembl:CHEMBL2002849	CHEMBL:CHEMBL2002849	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.049349315	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	ETIDRONIC ACID	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.3079628811477683	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	ISOBAVACHALCONE	chembl:CHEMBL253467	ISOBAVACHALCONE	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.182318303	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	GNF-PF-4864	chembl:CHEMBL583558	CHEMBL:CHEMBL583558	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.029301156	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	ANTIMYCIN A	chembl:CHEMBL211501	ANTIMYCIN A	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.3125456621172291	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
CASP9	hgnc:1511	CASP9	DTC	9/2/20	NULL	6.563458904461812	AICAR	drugbank:DB01700	AICA RIBONUCLEOTIDE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.4102161815288632	SINENSETIN	chembl:CHEMBL226507	SINENSETIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	MECLOFENOXATE	rxcui:2228	MECLOFENOXATE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2822993077187876	AMPICILLIN TRIHYDRATE	rxcui:203115	AMPICILLIN TRIHYDRATE	TRUE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.108711535	STREPTOZOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.1591141552596802	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.024309107	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.192335792	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.061197752	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NIRIDAZOLE	ncit:C90757	NIRIDAZOLE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.034612835	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	4-(4-HYDROXYPHENYLSULFONYL)PHENOL	chembl:CHEMBL384441	CHEMBL:CHEMBL384441	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.3409589041278864	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	TIOXOLONE	rxcui:2059173	TIOXOLONE	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.041247189	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.8334550989792778	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.2083637747448194	RG-7304	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.03136659	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
SMPD1	hgnc:11120	SMPD1	DTC	9/2/20	NULL	0.9376369863516874	ETIDRONIC ACID	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	NCI	14-Sep-17	NULL	0.006035365	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	PIRFENIDONE	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124127	chembl:CHEMBL1237255	CHEMBL:CHEMBL1237255	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
TNFRSF8	hgnc:11923	TNFRSF8	NCI	14-Sep-17	NULL	0.3454452054979901	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.596678082	BUPRANOLOL	rxcui:1817	BUPRANOLOL	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.003050289	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.06525008	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	PD-173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	AMCINAFIDE	ncit:C80807	AMCINAFIDE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.100589408	PAC-1	drugbank:DB13048	PAC-1	FALSE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.596678082	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	NEFAZODONE HYDROCHLORIDE	rxcui:236082	NEFAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	ZEARALANONE	chembl:CHEMBL491499	ZEARALANONE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.007075552	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	FLUORODIFEN	chembl:CHEMBL1892429	FLUORODIFEN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	SULINDAC SULFIDE	ncit:C29854	SULINDAC SULFIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	TETROQUINONE	chembl:CHEMBL1329029	TETROQUINONE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.347732922	GNF-PF-77	chembl:CHEMBL602987	CHEMBL:CHEMBL602987	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DOXYLAMINE	rxcui:3642	DOXYLAMINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	6-HYDROXYFLAVONE	chembl:CHEMBL138649	6-HYDROXYFLAVONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002331809	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	4-HYDROXYBENZOHYDRAZIDE	chembl:CHEMBL124267	CHEMBL:CHEMBL124267	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.012201155	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	FDA	10-Apr-24	NULL	0.074927706	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.7955707762984013	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.052507671	Flutamide	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.007244436	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.044198376	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	MyCancerGenome	20-Jun-17	inhibitor	0.2117244807890907	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.3642372228836055	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
TPSD1	hgnc:14118	TPSD1	NCI	14-Sep-17	NULL	1.810609352954982	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.5000730593875666	AMG208	chembl:CHEMBL496102	AMG-208	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.06697407	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.067897851	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.091850154	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.3938075342677087	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.068037151	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
TPSB2	hgnc:14120	TPSB2	NCI	14-Sep-17	NULL	1.640864726115453	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.091850154	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.099220845	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1816874437221263	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.075442056	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1479089330582944	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	1.381780822	LACTOSE	rxcui:6211	LACTOSE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.091636424	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.066297565	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.3454452054979901	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	NCI	14-Sep-17	NULL	0.069824031	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.092443083	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
AKT3	hgnc:393	AKT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2051080907644316	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
UCP2	hgnc:12518	UCP2	NCI	14-Sep-17	NULL	0.546954909	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.165474011072658	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1591141552596803	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2430910705356226	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
UGT1A10	hgnc:12531	UGT1A10	NCI	14-Sep-17	NULL	0.3947945205691315	ANTINEOPLASTIC AGENT	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
VEGFB	hgnc:12681	VEGFB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.076765601	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.005099813	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.00377129	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.035430277	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.016621612	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.009899636	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.1121958787087489	RO 31-8220	ncit:C1310	RO 31-8220	FALSE	FALSE	FALSE
UCP1	hgnc:12517	UCP1	NCI	14-Sep-17	NULL	0.9907107780319716	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
AGER	hgnc:320	AGER	NCI	14-Sep-17	NULL	3.000438356325399	VITAMIN B12	rxcui:11248	VITAMIN B12	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.08780547	NDGA	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	0.3070624048871023	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
UGDH	hgnc:12525	UGDH	NCI	14-Sep-17	NULL	0.7447896629176524	ACETYLSALICYLIC ACID	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
AKR1B1	hgnc:381	AKR1B1	NCI	14-Sep-17	NULL	8.078103267029922	TECTORIGENIN	ncit:C1205	TECTORIGENIN	FALSE	FALSE	FALSE
AKR1C1	hgnc:384	AKR1C1	NCI	14-Sep-17	NULL	1.591141552596803	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.3621218705909966	INTRALIPID	rxcui:1309980	SOYBEAN SEED OIL	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.3017682254924971	NORETHISTERONE ACETATE	rxcui:31983	NORETHINDRONE ACETATE	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.4526523382387456	BPDE	ncit:C196	BENZO(A)PYRENE-7,8-DIOL 9,10-EPOXIDE	FALSE	FALSE	FALSE
VDAC2	hgnc:12672	VDAC2	NCI	14-Sep-17	NULL	2.100306849	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.036590712	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1200632726425941	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.085378327	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.2845944240417045	NYSTATIN	rxcui:7597	NYSTATIN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.056918885	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.023716202	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.011734869	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.010540534	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.013560866	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.068847471	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.010028203	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.2983390411119005	ADM	ncit:C186783	ACELLULAR DERMAL MATRIX	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.042619863	FR901228	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.059667808	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.1988926940746003	ROFECOXIB	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	NCI	14-Sep-17	NULL	0.8751278539282416	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	2.763561643983921	TNP-470	drugbank:DB08633	TNP-470	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	NCI	14-Sep-17	NULL	0.021608095	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	NCI	14-Sep-17	NULL	0.2778183663264258	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
CALR	hgnc:1455	CALR	NCI	14-Sep-17	NULL	3.281729452230906	OLTIPRAZ	ncit:C1177	OLTIPRAZ	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	NCI	14-Sep-17	NULL	1.250182648468916	MEDICATION	ncit:C459	MEDICATION	FALSE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	PharmGKB	4/5/24	NULL	0.1446492320542548	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
CDX2	hgnc:1806	CDX2	NCI	14-Sep-17	NULL	3.889457128569963	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.2573905452730123	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.084553416	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.2430910705356226	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.2333674277141977	HEXADECYLPHOSPHOCHOLINE	rxcui:1494066	MILTEFOSINE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.2333674277141977	4-HC	ncit:C1423	PERFOSFAMIDE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.2000292237550266	CETIRIZINE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	0.049864835	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CREB1	hgnc:2345	CREB1	NCI	14-Sep-17	NULL	0.2075402025126264	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.158394182	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.8334550989792776	ISOPROPANOL	rxcui:797541	ISOPROPYL ALCOHOL	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.7693431682885642	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.075768645	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
CRHBP	hgnc:2356	CRHBP	PharmGKB	4/5/24	NULL	3.088686543276147	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.2447910080918158	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.2447910080918158	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.010804048	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.032055965	pentazocine	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
DCN	hgnc:2705	DCN	NCI	14-Sep-17	NULL	0.2631963470460877	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
DBH	hgnc:2689	DBH	NCI	14-Sep-17	NULL	0.1795134059339982	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.087222045	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
REN	hgnc:9958	REN	PharmGKB	4/5/24	NULL	1.750255707856483	muraglitazar	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
DNAJB1	hgnc:5270	DNAJB1	NCI	14-Sep-17	NULL	21.00306849	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.1256164383629055	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.074927706	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IRF6	hgnc:6121	IRF6	PharmGKB	4/5/24	NULL	3.500511415712966	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
DSG1	hgnc:3048	DSG1	NCI	14-Sep-17	NULL	0.7095631248066824	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
EIF4E	hgnc:3287	EIF4E	NCI	14-Sep-17	NULL	0.2223555345734189	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.2125816649218401	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.2263261691193728	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.038382801	sacituzumab govitecan	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.4953553890159858	PENICILLIN	wikidata:Q12190	PENICILLIN	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	1.009762908	RHIGF-1	rxcui:274403	MECASERMIN	TRUE	FALSE	FALSE
GDF15	hgnc:30142	GDF15	NCI	14-Sep-17	NULL	3.750547945	SULINDAC SULFIDE	ncit:C29854	SULINDAC SULFIDE	FALSE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.3671865121377238	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.2590839041234926	tucatinib	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.6482428547616604	MANNITOL	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.3633748874442526	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.4773424657790409	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	2.059124362184097	PSYLLIUM	rxcui:104129	ISPAGHULA HUSK	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.1178623372293928	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	NCI	14-Sep-17	NULL	0.3387591692625452	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
GRB2	hgnc:4566	GRB2	NCI	14-Sep-17	NULL	2.143170254518142	HEREGULIN	ncit:C1426	RECOMBINANT HEREGULIN	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	NCI	14-Sep-17	NULL	0.073850452	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
GRM1	hgnc:4593	GRM1	NCI	14-Sep-17	NULL	0.8751278539282417	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.6863747873946993	THYROGLOBULIN	rxcui:10565	THYROGLOBULIN	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.058832125	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.2734774543525755	HALOFUGINONE	ncit:C1120	HALOFUGINONE	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.8204323630577265	MISTLETOE LECTIN	ncit:C2703	MISTLETOE EXTRACT	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.072927321	isotretinoin	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.082043236	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.2941606231691568	CETIRIZINE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.082429625	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.2287915957982331	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
IRF2	hgnc:6117	IRF2	NCI	14-Sep-17	NULL	5.250767124	INTERFERON GAMMA	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.4375639269641208	midazolam	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1065064325267637	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.729273212	CYCLOOXYGENASE INHIBITOR	ncit:C1323	CYCLOOXYGENASE INHIBITOR	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1944728564284981	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.8751278539282416	SELENOMETHIONINE	rxcui:9644	SELENOMETHIONINE	TRUE	FALSE	FALSE
KRT10	hgnc:6413	KRT10	NCI	14-Sep-17	NULL	11.66837138570989	EGFR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.3088686543276147	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	1.693795846312725	HEPARIN CALCIUM	rxcui:20044	HEPARIN CALCIUM	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.5645986154375752	ACTH	iuphar.ligand:1331	ACTH	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.1035654265003836	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.3431873936973496	EOTAXIN	ncit:C1531	RECOMBINANT EOTAXIN	FALSE	FALSE	FALSE
MBL2	hgnc:6922	MBL2	NCI	14-Sep-17	NULL	6.563458904461812	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
MAPKAPK2	hgnc:6887	MAPKAPK2	NCI	14-Sep-17	NULL	0.6482428547616604	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.2282942227638891	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
MARCKSL1	hgnc:7142	MARCKSL1	NCI	14-Sep-17	NULL	0.6250913242344582	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.092118721	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.5834185692854944	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1161674142382621	bosentan	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.024932417	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.2500365296937833	LEUKOCYTE INTERFERON	ncit:C225	RECOMBINANT INTERFERON ALFA	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.00449706	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.044820889	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.192335792	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.2187819634820604	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.056980652	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	NCI	14-Sep-17	NULL	0.1324279224103266	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.013666755	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PC	hgnc:8636	PC	NCI	14-Sep-17	NULL	4.039051633514962	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.03319069	ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
PCNA	hgnc:8729	PCNA	NCI	14-Sep-17	NULL	21.00306849427779	SUNSCREEN	ncit:C851	SUNSCREEN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.100976291	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
PIP	hgnc:8993	PIP	NCI	14-Sep-17	NULL	0.8078103267029924	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	NCI	14-Sep-17	NULL	0.009994798	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
PLD1	hgnc:9067	PLD1	NCI	14-Sep-17	NULL	0.5385402178019949	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.4646696569530486	nafcillin	rxcui:7233	NAFCILLIN	TRUE	FALSE	FALSE
RBL2	hgnc:9894	RBL2	NCI	14-Sep-17	NULL	1.842374429322613	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.4773424657790409	lumiracoxib	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
RBP4	hgnc:9922	RBP4	NCI	14-Sep-17	NULL	4.039051633514962	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.3968833804663227	SU11248	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	3.088686543276147	THROMBOLYTIC AGENT	ncit:C29750	THROMBOLYTIC AGENT	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.5385402178019948	PSYLLIUM	rxcui:104129	ISPAGHULA HUSK	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	NCI	14-Sep-17	NULL	0.042276708	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.052116795	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1548898856510162	terbinafine	rxcui:37801	TERBINAFINE	TRUE	FALSE	FALSE
SLCO1A2	hgnc:10956	SLCO1A2	NCI	14-Sep-17	NULL	0.2243917574174978	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
SLPI	hgnc:11092	SLPI	NCI	14-Sep-17	NULL	2.625383561784725	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
SMOX	hgnc:15862	SMOX	NCI	14-Sep-17	NULL	3.182283105193606	DFMO	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	NCI	14-Sep-17	NULL	0.088396753	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	1.750255707856483	lumiracoxib	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.6731752722524935	FREUND&APOS;S ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
CYB5R2	hgnc:24376	CYB5R2	PharmGKB	4/5/24	NULL	0.7501095890813498	metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	NCI	14-Sep-17	NULL	1.166837138570988	EOTAXIN	ncit:C1531	RECOMBINANT EOTAXIN	FALSE	FALSE	FALSE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	0.9546849315580819	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	3.500511415712966	BENZNIDAZOLE	rxcui:18994	BENZNIDAZOLE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.317586721	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.038693936	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.068458502	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.034084824	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	NCI	14-Sep-17	NULL	1.363835616511545	PROMEGAPOIETIN	ncit:C2475	PROMEGAPOIETIN	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	3.750547945	METHYLCELLULOSE	rxcui:6873	METHYLCELLULOSE	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.018317694	ALL TRANS-RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	1.615620653405984	ACTIVIN	ncit:C2689	IH636 GRAPE SEED PROANTHOCYANIDIN EXTRACT	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.1250182648468916	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.151537291	DIFFERENTIATING AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	OncoKB	23-Jul-20	NULL	1.078924751	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
CYP24A1	hgnc:2602	CYP24A1	PharmGKB	4/5/24	NULL	2.917092846427472	daclatasvir	rxcui:1606218	DACLATASVIR	FALSE	FALSE	FALSE
FLI1	hgnc:3749	FLI1	OncoKB	23-Jul-20	NULL	26.25383561784724	TK216	drugbank:DB17414	TK216	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	OncoKB	23-Jul-20	NULL	4.699760697022038	LOXO-292	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	OncoKB	23-Jul-20	NULL	0.8008364246019593	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	OncoKB	23-Jul-20	NULL	1.165474011072658	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	0.8247278204559345	PLX8394	drugbank:DB16038	PLX8394	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	OncoKB	23-Jul-20	NULL	0.3889457128569963	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.2586584789935689	rivastigmine	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.2414145803939976	thioridazine	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.056097939	pyrilamine	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.014299475	pioglitazone	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRCP	hgnc:9344	PRCP	PharmGKB	4/5/24	NULL	17.50255707856483	benazepril	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.077789143	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.050048162	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
SULT1A4	hgnc:30004	SULT1A4	PharmGKB	4/5/24	NULL	1.141471113819445	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.020399251	propafenone	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.034184682	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.8204323630577265	rhodamine 123	iuphar.ligand:4607	RHODAMINE123	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	PharmGKB	4/5/24	NULL	0.014906788	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.054020238	nateglinide	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
GADL1	hgnc:27949	GADL1	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.1190650141398968	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	PharmGKB	4/5/24	NULL	0.4861821410712453	bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
ADD1	hgnc:243	ADD1	PharmGKB	4/5/24	NULL	1.458546423213736	bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
KCNE1	hgnc:6240	KCNE1	PharmGKB	4/5/24	NULL	0.8824818695074707	Antibiotics	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
RFPL4B	hgnc:33264	RFPL4B	PharmGKB	4/5/24	NULL	2.187819634820604	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.003689409	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
MT-ND1	hgnc:7455	MT-ND1	PharmGKB	4/5/24	NULL	5.250767123569449	isepamicin	ncit:C83838	ISEPAMICIN	FALSE	FALSE	FALSE
UST	hgnc:17223	UST	PharmGKB	4/5/24	NULL	4.922594178346359	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.026680727	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
ATP5F1E	hgnc:838	ATP5F1E	PharmGKB	4/5/24	NULL	0.2885036881082116	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
SLC39A14	hgnc:20858	SLC39A14	PharmGKB	4/5/24	NULL	3.281729452230906	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
PPM1A	hgnc:9275	PPM1A	PharmGKB	4/5/24	NULL	3.281729452230906	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	PharmGKB	4/5/24	NULL	0.017835486	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
ARHGEF28	hgnc:30322	ARHGEF28	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.030996264	flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.042073455	spironolactone	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.034521809	reserpine	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
IRS1	hgnc:6125	IRS1	PharmGKB	4/5/24	NULL	0.1103102336884338	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ATP5F1E	hgnc:838	ATP5F1E	PharmGKB	4/5/24	NULL	0.2273059360852576	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
REV3L	hgnc:9968	REV3L	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.029260335	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.03394161	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
FCER1G	hgnc:3611	FCER1G	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ARG2	hgnc:664	ARG2	PharmGKB	4/5/24	NULL	0.1613138901250215	Methyldopa	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
IL4R	hgnc:6015	IL4R	PharmGKB	4/5/24	NULL	0.3571950424196904	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.1530835896084387	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	1.521961485092594	raltegravir	rxcui:1235585	RALTEGRAVIR POTASSIUM	TRUE	FALSE	FALSE
MACROD2	hgnc:16126	MACROD2	PharmGKB	4/5/24	NULL	3.281729452230906	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	PharmGKB	4/5/24	NULL	0.028283152	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NAGS	hgnc:17996	NAGS	PharmGKB	4/5/24	NULL	26.25383561784724	carglumic acid	rxcui:401713	CARGLUMIC ACID	TRUE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	PharmGKB	4/5/24	NULL	0.1223955040459079	lenalidomide	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	1.250182648468916	pyridoxal phosphate	rxcui:1599827	PYRIDOXAL PHOSPHATE ANHYDROUS	FALSE	FALSE	FALSE
NFIB	hgnc:7785	NFIB	PharmGKB	4/5/24	NULL	0.4059871487295966	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	PharmGKB	4/5/24	NULL	0.07463777	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.071245144	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PDK1	hgnc:8809	PDK1	PharmGKB	4/5/24	NULL	0.2239133101735373	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
ALOX12	hgnc:429	ALOX12	PharmGKB	4/5/24	NULL	0.05056107	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
IGFBP3	hgnc:5472	IGFBP3	PharmGKB	4/5/24	NULL	0.7836965856073805	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	PharmGKB	4/5/24	NULL	0.088866948	olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
CASP9	hgnc:1511	CASP9	PharmGKB	4/5/24	NULL	0.1959241464018451	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
DDIT3	hgnc:2726	DDIT3	PharmGKB	4/5/24	NULL	0.1275785139360852	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.014622019	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
MAP3K5	hgnc:6857	MAP3K5	PharmGKB	4/5/24	NULL	0.8334550989792776	hydroxyurea	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.039688338	cemiplimab-rwlc	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.069454592	tepotinib	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.900646162	succinylcholine	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.022136455	ketorolac	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.025298806	lofexidine	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.004216468	sertindole	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.035418328	cariprazine	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.04427291	acetaminophen / codeine	wikidata:Q48566735	ACETAMINOPHEN / CODEINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.017709164	amoxapine	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.5250767123569451	n-desmethylclozapine	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.3182283105193606	dapsone	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.1795134059339982	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	PharmGKB	4/5/24	NULL	0.012623554	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
SULT1A1	hgnc:11453	SULT1A1	PharmGKB	4/5/24	NULL	3.889457128569963	conjugated estrogens	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
HPRT1	hgnc:5157	HPRT1	PharmGKB	4/5/24	NULL	1.193356164447602	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
F2	hgnc:3535	F2	PharmGKB	4/5/24	NULL	0.3947945205691315	avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	0.1685639526025505	avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.1754935535952356	lidocaine	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
HLA-DPB1	hgnc:4940	HLA-DPB1	PharmGKB	4/5/24	NULL	0.8468979231563629	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
HLA-DRB3	hgnc:4951	HLA-DRB3	PharmGKB	4/5/24	NULL	0.2706580991530644	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.092199598	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	PharmGKB	4/5/24	NULL	0.2051080907644316	risdiplam	rxcui:2390935	RISDIPLAM	TRUE	FALSE	FALSE
ADAMTS10	hgnc:13201	ADAMTS10	PharmGKB	4/5/24	NULL	15.00219178162699	levonorgestrel	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
WFS1	hgnc:12762	WFS1	PharmGKB	4/5/24	NULL	0.7242437411819931	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PGK1	hgnc:8896	PGK1	PharmGKB	4/5/24	NULL	2.187819634820604	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.006780433	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
ADAMTSL2	hgnc:14631	ADAMTSL2	PharmGKB	4/5/24	NULL	8.751278539282415	buprenorphine	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1944728564284981	dabigatran	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	PharmGKB	4/5/24	NULL	0.2333674277141977	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
NT5C2	hgnc:8022	NT5C2	PharmGKB	4/5/24	NULL	0.7778914257139925	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	1.071585127259071	rocuronium	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
UPB1	hgnc:16297	UPB1	PharmGKB	4/5/24	NULL	0.661861402	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	PharmGKB	4/5/24	NULL	0.011031023	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.08854582	valbenazine	rxcui:1918219	VALBENAZINE	TRUE	FALSE	FALSE
IL21R	hgnc:6006	IL21R	PharmGKB	4/5/24	NULL	0.921187215	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
KLRK1	hgnc:18788	KLRK1	PharmGKB	4/5/24	NULL	0.6908904109959803	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.021357605	selegiline	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.2625383561784725	articaine / epinephrine	wikidata:Q48566634	ARTICAINE / EPINEPHRINE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.2827336143460473	nitrofurantoin	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	PharmGKB	4/5/24	NULL	0.087903467	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	PharmGKB	4/5/24	NULL	2.625383561784724	tenofovir disoproxil fumarate	rxcui:322248	TENOFOVIR DISOPROXIL FUMARATE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.1141471113819445	tepotinib	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
ITGA2B	hgnc:6138	ITGA2B	PharmGKB	4/5/24	NULL	3.500511415712967	eptifibatide	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
SLCO1C1	hgnc:13819	SLCO1C1	PharmGKB	4/5/24	NULL	0.6351734423672721	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
SLC9A8	hgnc:20728	SLC9A8	PharmGKB	4/5/24	NULL	1.693795846312725	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	0.4167275494896388	avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.034727296	ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.014585464	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	PharmGKB	4/5/24	NULL	1.500219178	capmatinib	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.2500365296937833	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.02726255	ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.037870661	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
IL12A	hgnc:5969	IL12A	PharmGKB	4/5/24	NULL	1.050153425	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
NME1	hgnc:7849	NME1	PharmGKB	4/5/24	NULL	0.7501095890813498	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2237542808339254	selegiline	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.031707531	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.08780547	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.053199262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
WBP2NL	hgnc:28389	WBP2NL	PharmGKB	4/5/24	NULL	1.640864726115453	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.065226921	cemiplimab-rwlc	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
MYOM2	hgnc:7614	MYOM2	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NEDD4L	hgnc:7728	NEDD4L	PharmGKB	4/5/24	NULL	1.000146118775133	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NECAB1	hgnc:20983	NECAB1	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	PharmGKB	4/5/24	NULL	0.020405196	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.012623554	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NEDD4L	hgnc:7728	NEDD4L	PharmGKB	4/5/24	NULL	5.834185692854944	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	PharmGKB	4/5/24	NULL	0.1682938180631233	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.280789686	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.005534114	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	PharmGKB	4/5/24	NULL	0.031254566	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.1521961485092594	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
TCF19	hgnc:11629	TCF19	PharmGKB	4/5/24	NULL	4.773424657790409	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	PharmGKB	4/5/24	NULL	0.1363835616511545	vildagliptin	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	3.750547945	tetanus antitoxin	chembl:CHEMBL2108107	TETANUS ANTITOXIN	FALSE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.2500365296937833	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.021370644	MOMELOTINIB	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.8334550989792777	ZALUTUMUMAB	ncit:C64620	ZALUTUMUMAB	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.1552333222045661	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.1244847587380144	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.1060761035064535	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.1346350544504987	AGN-214868	chembl:CHEMBL3137348	SENREBOTASE	FALSE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.067403943	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q15858	hgnc:10597	SCN9A	TdgClinicalTrial	Jan-14	NULL	0.1103102336884338	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
UNIPROT:P02679	hgnc:3694	FGG	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	ALFIMEPRASE	ncit:C79877	ALFIMEPRASE	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	PharmGKB	4/5/24	NULL	0.283060222	certolizumab pegol	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.1219218372345847	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.032154116	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
UNIPROT:P02671	hgnc:3661	FGA	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	ALTEPLASE	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.2678962818147678	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	ALTEPLASE	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
UNIPROT:P14210	hgnc:4893	HGF	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	AMG-102	hemonc:443	RILOTUMUMAB	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1840222122746302	CLOMIFENE	rxcui:2596	CLOMIPHENE	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.1567393171214761	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.546954909	ANTI-CD3 MONOCLONAL ANTIBODY	ncit:C112883	ANTI-CD3 MONOCLONAL ANTIBODY	FALSE	FALSE	FALSE
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	ANTI-CD3 MONOCLONAL ANTIBODY	ncit:C112883	ANTI-CD3 MONOCLONAL ANTIBODY	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.024773612	conjugated estrogens	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	ANA773	chembl:CHEMBL4650440	RG-7795	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.030746697	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
UNIPROT:P04275	hgnc:12726	VWF	TdgClinicalTrial	Jan-14	NULL	0.6908904109959803	ANTIHEMOPHILIC FACTOR	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.014683353	arteether	ncit:C73002	ARTEMOTIL	TRUE	FALSE	FALSE
UNIPROT:O75116	hgnc:10252	ROCK2	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	AR-12286	ncit:C152866	VEROSUDIL	FALSE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.1017590527823536	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.1461794856227575	ARN-509	rxcui:1999574	APALUTAMIDE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.016018204	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.4167275494896388	ARRY-334543	ncit:C62530	VARLITINIB	FALSE	FALSE	FALSE
UNIPROT:Q13464	hgnc:10251	ROCK1	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	AR-12286	ncit:C152866	VEROSUDIL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.021357605	sildenafil	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.1067229090156392	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.039155609	proguanil	rxcui:2382	PROGUANIL	TRUE	FALSE	FALSE
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.1325951293830669	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.1215455352678113	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.055504938	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.055504938	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.1725162436059257	dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.056826484	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.1117184494376478	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.058212496	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
DDX53	hgnc:20083	DDX53	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:P01106	hgnc:7553	MYC	TdgClinicalTrial	Jan-14	NULL	0.750109589	AVI-4126	ncit:C62518	PHOSPHORODIAMIDATE MORPHOLINO OLIGOMER AVI-4126	FALSE	FALSE	FALSE
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	ATL1102	drugbank:DB04997	ATL1102	FALSE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.3889457128569963	hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.2778183663264259	AV-412	drugbank:DB06021	AV-412	FALSE	FALSE	TRUE
UNIPROT:P13612	hgnc:6140	ITGA4	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	ATL1102	drugbank:DB04997	ATL1102	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.4293851619741372	ATOMOXETINE	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	0.9907107780319716	AXL1717	ncit:C87736	PICROPODOPHYLLIN	FALSE	FALSE	FALSE
UNIPROT:Q92542	hgnc:17091	NCSTN	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	BMS-299897	chembl:CHEMBL247471	CHEMBL:CHEMBL247471	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.078545507	atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	3.231241306811969	BIIB037	rxcui:2557217	ADUCANUMAB	TRUE	FALSE	FALSE
UNIPROT:P35225	hgnc:5973	IL13	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	TRALOKINUMAB	rxcui:2589225	TRALOKINUMAB	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.2332563532602643	selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
UNIPROT:P01138	hgnc:7808	NGF	TdgClinicalTrial	Jan-14	NULL	15.00219178	CERE-110	drugbank:DB05898	CERE-110	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.068191781	ESCITALOPRAM	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	0.2651902587661338	phenprocoumon	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.8607814956671229	GESTODENE	rxcui:25734	GESTODENE	TRUE	FALSE	FALSE
UNIPROT:Q15119	hgnc:8810	PDK2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.081281225	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P42081	hgnc:1705	CD86	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	RG-2077	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.030670369	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	CVT-3619	iuphar.ligand:5593	GS9667	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.09869863	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.039899446	METOCLOPRAMIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.068369364	tucatinib	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.03070624	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.034118045	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.6105543166941221	FIPAMEZOLE	ncit:C65684	FIPAMEZOLE	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.034981793	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1842374429322614	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
UNIPROT:P30411	hgnc:1030	BDKRB2	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	ICATIBANT	rxcui:1148138	ICATIBANT	TRUE	FALSE	FALSE
UNIPROT:P30988	hgnc:1440	CALCR	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	SALMON CALCITONIN	rxcui:36118	SALMON CALCITONIN	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.064824285	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
UNIPROT:Q16555	hgnc:3014	DPYSL2	TdgClinicalTrial	Jan-14	NULL	0.2125816649218401	LACOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.042845917	enalapril	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	KETOTIFEN	rxcui:11404	KETOTIFEN FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.150021918	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	LERCANIDIPINE	rxcui:135056	LERCANIDIPINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1835932560688619	VORTIOXETINE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
CRP	hgnc:2367	CRP	PharmGKB	4/5/24	NULL	0.3977853881492008	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:P23458	hgnc:6190	JAK1	TdgClinicalTrial	Jan-14	NULL	0.6159257622955366	LY3009104	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	0.9907107780319716	MECASERMIN	rxcui:274403	MECASERMIN	TRUE	FALSE	FALSE
UNIPROT:Q8TBC4	hgnc:12470	UBA3	TdgClinicalTrial	Jan-14	NULL	21.00306849	MLN-4924	ncit:C77906	PEVONEDISTAT	FALSE	FALSE	FALSE
CASP9	hgnc:1511	CASP9	PharmGKB	4/5/24	NULL	0.3977853881492008	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:P43235	hgnc:2536	CTSK	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	MIV-701	drugbank:DB05736	MIV-701	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1704794520639431	MILNACIPRAN	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.6908904109959803	MM-111	drugbank:DB17983	MM-111	FALSE	TRUE	TRUE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.8751278539282416	PEG-IRINOTECAN	ncit:C74069	ETIRINOTECAN PEGOL	FALSE	FALSE	TRUE
HFE	hgnc:4886	HFE	PharmGKB	4/5/24	NULL	0.7955707762984016	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.096432821	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.086007651	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.6364566210387211	EXENDIN-4	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	16.15620653405984	PL-3994	drugbank:DB15355	PL-3994	FALSE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.081533651	PIRFENIDONE	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	0.5339763176511304	PS433540	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.072324616	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:O00264	hgnc:16090	PGRMC1	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	OPC-14523	drugbank:DB05422	OPC-14523	FALSE	FALSE	FALSE
UNIPROT:Q9NY47	hgnc:1400	CACNA2D2	TdgClinicalTrial	Jan-14	NULL	0.2344092465879218	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	SUFENTANIL	rxcui:56795	SUFENTANIL	TRUE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	PharmGKB	4/5/24	NULL	0.1097339001790898	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:O60894	hgnc:9843	RAMP1	TdgClinicalTrial	Jan-14	NULL	3.750547945406749	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	SYL040012	chembl:CHEMBL4298113	BAMOSIRAN	FALSE	FALSE	FALSE
UNIPROT:Q02643	hgnc:4266	GHRHR	TdgClinicalTrial	Jan-14	NULL	19.69037671338543	TESAMORELIN	rxcui:1044584	TESAMORELIN	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.061197752	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TdgClinicalTrial	Jan-14	NULL	15.75230137070834	TECARFARIN	ncit:C152523	TECARFARIN	FALSE	FALSE	FALSE
HLA-E	hgnc:4962	HLA-E	PharmGKB	4/5/24	NULL	0.5303805175322677	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:P24530	hgnc:3180	EDNRB	TdgClinicalTrial	Jan-14	NULL	3.750547945	BOSENTAN	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P32297	hgnc:1957	CHRNA3	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.3351553483129436	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.3443125982668492	NORETHINDRONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
UNIPROT:P16298	hgnc:9315	PPP3CB	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	VOCLOSPORIN	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
DOCK8	hgnc:19191	DOCK8	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:Q08209	hgnc:9314	PPP3CA	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	VOCLOSPORIN	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	0.046303061	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1221108633388244	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.09741683	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
PRRC2A	hgnc:13918	PRRC2A	PharmGKB	4/5/24	NULL	0.3977853881492008	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.1013661606866689	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TdgClinicalTrial	Jan-14	NULL	0.8655110643246346	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.068191781	CITALOPRAM	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.07963752	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	1.158257453728555	EDROPHONIUM	rxcui:1546421	EDROPHONIUM CATION	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.086694009	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.083522277	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.054695491	FLUPENTHIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.055344054	FLUPENTHIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.093763699	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.1022876712383659	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.100976291	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.087512785	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.096050618	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.075010959	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.048844345	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.1658136986390352	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.073266518	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	LEVOBUNOLOL	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
TRIM5	hgnc:16276	TRIM5	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1363835616511545	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.062262061	MESORIDAZINE	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P49019	hgnc:16824	HCAR3	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	MEPENZOLATE	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.097236428	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	0.016574391	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.1067229090156392	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.096167896	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.3351553483129436	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.091159151	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.2386712328895204	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.1286952726365061	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	NAFARELIN	rxcui:28656	NAFARELIN	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.8950171233357017	OXPRENOLOL	rxcui:7801	OXPRENOLOL	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.091796628	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.101562227	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.070197421	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P22748	hgnc:1375	CA4	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	TOLAZAMIDE	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TdgClinicalTrial	Jan-14	NULL	0.8751278539282416	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TEND	1-Aug-11	NULL	0.8655110643246346	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TEND	1-Aug-11	NULL	0.1902451856365742	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.3889457128569962	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TEND	1-Aug-11	NULL	0.1769126389342806	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:P32754	hgnc:5147	HPD	TEND	1-Aug-11	NULL	70.01022831425932	NITISINONE	rxcui:61805	NITISINONE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.3938075342677087	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	0.4487835148349958	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.3818739726232327	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
UNIPROT:Q15842	hgnc:6269	KCNJ8	TEND	1-Aug-11	NULL	3.281729452230906	THIAMYLAL	rxcui:10464	THIAMYLAL	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TEND	1-Aug-11	NULL	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.068191781	ESCITALOPRAM	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.07182992	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.064944553	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.2983390411119005	FLUMETHASONE PIVALATE	rxcui:25113	FLUMETHASONE PIVALATE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1282238613814273	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.063300387	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.079197091	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.055563673	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.064111931	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.3241214273808302	FOSPROPOFOL	rxcui:828682	FOSPROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.060984519	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P03886	hgnc:7455	MT-ND1	TEND	1-Aug-11	NULL	0.3500511415712967	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P26358	hgnc:2976	DNMT1	TEND	1-Aug-11	NULL	0.1704794520639431	IFOSFAMIDE	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.596678082	HYDROCORTAMATE	ncit:C65862	HYDROCORTAMATE	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TEND	1-Aug-11	NULL	0.046549354	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.096167896	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.1067229090156392	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P43115	hgnc:9595	PTGER3	TEND	1-Aug-11	NULL	1.458546423213736	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.192335792	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.007196775	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.064111931	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.019739726	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.024384367	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.060984519	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.8950171233357017	OXPRENOLOL	rxcui:7801	OXPRENOLOL	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1137761023525341	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.06525008	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.0296486	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.009767052	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TEND	1-Aug-11	NULL	0.054398002	PROPAFENONE	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.5834185692854944	PROPOXYPHENE	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.4565884455277782	PROPERICIAZINE	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.086551106	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P30939	hgnc:5292	HTR1F	TEND	1-Aug-11	NULL	0.4150804050252529	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.068191781	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
UNIPROT:P27815	hgnc:8780	PDE4A	TEND	1-Aug-11	NULL	0.2983390411119005	TADALAFIL	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	0.6908904109959803	GDC-0425	drugbank:DB14791	GDC-0425	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	2.128689374420047	Xaliproden	ncit:C152924	XALIPRODEN	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.3088686543276147	CA-170	drugbank:DB15772	CA-170	FALSE	FALSE	FALSE
PROTEIN-SERINE O-PALMITOLEOYLTRANSFERASE PORCUPINE	hgnc:17652	PORCN	TTD	2020.06.01	NULL	13.12691780892362	ETC-1922159	iuphar.ligand:11168	ETC-1922159	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	IT-141	ncit:C148511	NANOPARTICLE SN-38-ENCAPSULATED MICELLE FORMULATION IT-141	FALSE	FALSE	FALSE
EPHRIN TYPE-B RECEPTOR 2	hgnc:3393	EPHB2	TTD	2020.06.01	NULL	0.138178082	KO-947	iuphar.ligand:9976	KO-947	FALSE	FALSE	FALSE
GPX5	hgnc:4557	GPX5	PharmGKB	4/5/24	NULL	0.3977853881492008	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	1.166837138570988	EDO-S101	ncit:C126105	TINOSTAMUSTINE	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	TAS3681	ncit:C137818	ANDROGEN RECEPTOR ANTAGONIST TAS3681	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	2.100306849	USL311	ncit:C131534	CXCR4 ANTAGONIST USL311	FALSE	FALSE	FALSE
STEROID 5-ALPHA-REDUCTASE 2	hgnc:11285	SRD5A2	TTD	2020.06.01	NULL	3.750547945	Finasteride	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	5.250767123569449	ANA773	chembl:CHEMBL4650440	RG-7795	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	PharmGKB	4/5/24	NULL	0.002681699	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.8204323630577265	APN-301	ncit:C162537	LORUKAFUSP ALFA	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	3.150460274	BL-8040	rxcui:2664896	MOTIXAFORTIDE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.1211249624814175	ACP-196	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.3977853881492006	carbimazole	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
PROTEIN-TYROSINE PHOSPHATASE SHP-1	hgnc:9658	PTPN6	TTD	2020.06.01	NULL	2.917092846427472	NSC-87877	chembl:CHEMBL472004	CHEMBL:CHEMBL472004	FALSE	FALSE	FALSE
PI3-KINASE BETA	hgnc:8976	PIK3CB	TTD	2020.06.01	NULL	0.078136416	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
VEGFB	hgnc:12681	VEGFB	PharmGKB	4/5/24	NULL	7.001022831425934	aflibercept	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	0.1151484018326633	RXDX 101	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.4861821410712453	KX2-361	iuphar.ligand:10004	KX2-361	FALSE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	9.26605963	TB-402	drugbank:DB06050	TB-402	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.2187819634820604	(S)-DRF-1042	iuphar.ligand:8261	(S)-DRF-1042	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	3.889457128569962	Obinutuzumab	rxcui:974779	OBINUTUZUMAB	TRUE	FALSE	FALSE
CYB5R4	hgnc:20147	CYB5R4	PharmGKB	4/5/24	NULL	2.100306849	rasburicase	rxcui:283821	RASBURICASE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-2	hgnc:4076	GABRA2	TTD	2020.06.01	NULL	0.096167896	Flumazenil	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-3	hgnc:4077	GABRA3	TTD	2020.06.01	NULL	0.097236428	Flumazenil	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
ENDOPLASMIC RETICULUM CHAPERONE BIP	hgnc:5238	HSPA5	TTD	2020.06.01	NULL	1.640864726115453	NKP-1339	ncit:C97948	RUTHENIUM-BASED TRANSFERRIN TARGETING AGENT NKP-1339	FALSE	FALSE	FALSE
GLUTAMINYL CYCLASE	hgnc:9753	QPCT	TTD	2020.06.01	NULL	105.0153424713889	PQ-912	chembl:CHEMBL3659477	VAROGLUTAMSTAT	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.070574827	mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
ANNEXIN A5	hgnc:543	ANXA5	TTD	2020.06.01	NULL	2.625383561784724	Diannexin	ncit:C169905	DIANEXIN	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	PharmGKB	4/5/24	NULL	0.2044691247495891	venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
FOLATE RECEPTOR	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	2.917092846427472	Tetrahydrofolic acid	drugbank:DB00116	TETRAHYDROFOLIC ACID	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.3818739726232327	Diflunisal	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.2734774543525755	DAS-431 IV	drugbank:DB05432	DAS-431 IV	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.1861974157294131	Cotinine	ncit:C70941	COTININE	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.3889457128569962	DENBUFYLLINE	ncit:C76316	DENBUFYLLINE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1805819381121768	ABX-EGF	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.1302919881779019	pyrazinamide	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M2	hgnc:1951	CHRM2	TTD	2020.06.01	NULL	0.083744292	Gallamine Triethiodide	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.060077427	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	1.050153425	CC-486	ncit:C118288	ORAL AZACITIDINE	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Buclizine	rxcui:59636	BUCLIZINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.8950171233357017	Oxprenolol	rxcui:7801	OXPRENOLOL	TRUE	FALSE	FALSE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	0.7721716358190367	ATOSIBAN	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	1.458546423213736	Teriflunomide	rxcui:1310520	TERIFLUNOMIDE	TRUE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	Lerisetron	ncit:C30143	LERISETRON	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3040984820600068	Buspirone	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.1600843635234588	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
FERROCHELATASE	hgnc:3647	FECH	TTD	2020.06.01	NULL	0.8751278539282416	Cholic Acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
LIVER CARBOXYLESTERASE	hgnc:1863	CES1	TTD	2020.06.01	NULL	0.1902451856365742	Cholic Acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
EPB41	hgnc:3377	EPB41	PharmGKB	4/5/24	NULL	0.760980743	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 1	hgnc:4584	GRIN1	TTD	2020.06.01	NULL	0.2678962818147678	Cycloserine	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE	hgnc:877	ALDH7A1	TTD	2020.06.01	NULL	1.093909817410302	NM-702	drugbank:DB05505	NM-702	FALSE	FALSE	FALSE
ZNF697	hgnc:32034	ZNF697	PharmGKB	4/5/24	NULL	5.250767124	interferon beta-1b	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	0.064347636	Ibudilast	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	2.386712328895204	Lixivaptan	ncit:C74429	LIXIVAPTAN	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1232574442152452	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.073437302	Niflumic Acid	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	0.6731752722524935	RGH-896	chembl:CHEMBL182066	RADIPRODIL	FALSE	FALSE	FALSE
FATTY ACID SYNTHASE	hgnc:3594	FASN	TTD	2020.06.01	NULL	1.944728564284981	PA-824	rxcui:2198359	PRETOMANID	TRUE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	0.2853677784548614	ATOSIBAN	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
MUTYH	hgnc:7527	MUTYH	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE	hgnc:30092	NAMPT	TTD	2020.06.01	NULL	21.00306849427779	Daporinad	ncit:C67043	DAPORINAD	FALSE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.5770073762164231	Mosapride	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	1.093909817410302	TG-4010	chembl:CHEMBL4650517	MESMULOGENE ANCOVACIVEC	FALSE	FALSE	FALSE
LYSOSOMAL ALPHA-GLUCOSIDASE	hgnc:4065	GAA	TTD	2020.06.01	NULL	0.364636606	SALACINOL	chembl:CHEMBL1208974	SALACINOL	FALSE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.1119566550867686	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	7.501095891	Pipecuronium	rxcui:33742	PIPECURONIUM	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.068147529	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.2	hgnc:1395	CACNA1H	TTD	2020.06.01	NULL	0.6105543166941221	Sodium bicarbonate	rxcui:36676	SODIUM BICARBONATE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.5147810905460245	Cyclopentolate	rxcui:3001	CYCLOPENTOLATE	TRUE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	0.2853677784548614	SSR149415	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	0.3860858179095183	SSR149415	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	PharmGKB	4/5/24	NULL	0.020094784	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
CARBOXYPEPTIDASE B2	hgnc:2300	CPB2	TTD	2020.06.01	NULL	3.750547945	UK-396082	iuphar.ligand:8657	UK-396,082	FALSE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	0.5469549087051511	IMGN-853	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1635752997996713	Levomilnacipran	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	15.00219178	CERE-110	drugbank:DB05898	CERE-110	FALSE	FALSE	FALSE
GRID2	hgnc:4576	GRID2	PharmGKB	4/5/24	NULL	0.7836965856073805	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
PROTEASOME	hgnc:9338	PRB2	TTD	2020.06.01	NULL	7.501095891	ONX-0912	hemonc:373	OPROZOMIB	FALSE	FALSE	FALSE
CELL SURFACE A33 ANTIGEN	hgnc:4445	GPA33	TTD	2020.06.01	NULL	26.25383561784724	HuA33	chembl:CHEMBL2109435	HUA33	FALSE	FALSE	FALSE
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	3.500511415712966	SAM-531	ncit:C169839	CERLAPIRDINE	FALSE	FALSE	FALSE
HISTIDINE DECARBOXYLASE	hgnc:4855	HDC	TTD	2020.06.01	NULL	26.25383561784724	ALPHA-FMH	iuphar.ligand:5189	FMH	FALSE	FALSE	FALSE
GRM7	hgnc:4599	GRM7	PharmGKB	4/5/24	NULL	0.7836965856073805	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
LEUKOCYTE ANTIGEN CD37	hgnc:1666	CD37	TTD	2020.06.01	NULL	35.00511415712966	BI-836826	drugbank:DB17322	BI-836826	FALSE	FALSE	FALSE
ACTIVATION-INDUCIBLE TNFR FAMILY RECEPTOR	hgnc:11914	TNFRSF18	TTD	2020.06.01	NULL	13.12691780892362	MK-4166	ncit:C116065	ANTI-GITR MONOCLONAL ANTIBODY MK-4166	FALSE	FALSE	FALSE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.1422972120208523	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
MONOCYTE CHEMOTACTIC AND ACTIVATING FACTOR	hgnc:10618	CCL2	TTD	2020.06.01	NULL	17.50255707856483	NOX-E36	ncit:C171710	EMAPTICAP PEGOL	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.1211249624814175	Acalabrutinib	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	TESTOSTERONE BUCICLATE	ncit:C87245	TESTOSTERONE BUCYCLATE	FALSE	FALSE	FALSE
TRANSTHYRETIN	hgnc:12405	TTR	TTD	2020.06.01	NULL	17.50255707856483	Inotersen	rxcui:2099289	INOTERSEN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M2	hgnc:1951	CHRM2	TTD	2020.06.01	NULL	0.092118721	ACECLIDINE	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	0.2328499833068492	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR-ALPHA	hgnc:10477	RXRA	TTD	2020.06.01	NULL	0.2333674277141977	Alitretinoin	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.4730420832044549	KF-17837	chembl:CHEMBL27508	CHEMBL:CHEMBL27508	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR-BETA	hgnc:10478	RXRB	TTD	2020.06.01	NULL	0.8334550989792776	Alitretinoin	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.070956312	ACECLIDINE	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
GNL3	hgnc:29931	GNL3	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	0.1902451856365742	AMG 386	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	0.3977853881492007	Leuprorelin acetate	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.3697723326457359	ASP-8477	chembl:CHEMBL5095212	ASP-8477	FALSE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	Anti-CD33 CAR-T cells	ncit:C191739	ANTI-CD33 CAR T-CELLS	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.8008364246019593	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	PharmGKB	4/5/24	NULL	0.019404165	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.595325071	Rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.8751278539282416	Becaplermin	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
CARDIOTROPHIN-1	hgnc:2499	CTF1	TTD	2020.06.01	NULL	7.501095891	Cardiotrophin-1	iuphar.ligand:4906	CARDIOTROPHIN-1	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.6134073742487676	elacestrant	rxcui:2628469	ELACESTRANT	TRUE	FALSE	TRUE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	1.312691780892362	LY2944876	chembl:CHEMBL3990012	PEGAPAMODUTIDE	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.4953553890159858	HBI-8000	ncit:C97263	TUCIDINOSTAT	FALSE	FALSE	FALSE
GABA(A) RECEPTOR DELTA	hgnc:4084	GABRD	TTD	2020.06.01	NULL	0.0296486	Gaboxadol	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.1600843635234588	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	2.386712328895204	SLV-334	drugbank:DB15356	SLV-334	FALSE	FALSE	FALSE
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	0.3621218705909966	Hydroxyamphetamine Hydrobromide	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.2983390411119005	LITOXETINE	ncit:C66021	LITOXETINE	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.5834185692854944	LITOXETINE	ncit:C66021	LITOXETINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.004919212	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.7955707762984013	Aceclofenac	rxcui:16689	ACECLOFENAC	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.061340737	Cenestin	rxcui:253166	SYNTHETIC CONJUGATED ESTROGENS, A	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Doxylamine	rxcui:3642	DOXYLAMINE	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	1.032937794800547	Etonogestrel	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	0.8334550989792776	Heparin Sodium	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	0.5000730593875666	sulindac	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	0.084689792	Propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
HISTAMINE H2 RECEPTOR	hgnc:5183	HRH2	TTD	2020.06.01	NULL	0.8204323630577265	Ranitidine	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.034590034	Quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	1.250182648468916	Torasemide	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.7395446652914718	Tetrahydrozoline	rxcui:37935	TETRAHYDROZOLINE	TRUE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.105947682	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	1.050153425	Igmesine	ncit:C170052	IGMESINE	FALSE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DS1	hgnc:6333	KIR2DS1	TTD	2020.06.01	NULL	21.00306849	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
LIPOPROTEIN LIPASE	hgnc:6677	LPL	TTD	2020.06.01	NULL	1.875273972703375	Ibrolipim	ncit:C75256	IBROLIPIM	FALSE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	17.50255707856483	MORAb-009	ncit:C62483	AMATUXIMAB	FALSE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR ACETYLHYDROLASE	hgnc:9040	PLA2G7	TTD	2020.06.01	NULL	6.563458904461812	Rilapladib	ncit:C76401	RILAPLADIB	FALSE	FALSE	FALSE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	2.386712328895204	Z 360	iuphar.ligand:907	Z-360	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.6250913242344583	Camptothecin	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
FAST SKELETAL MUSCLE TROPONIN COMPLEX	hgnc:11944	TNNC2	TTD	2020.06.01	NULL	17.50255707856483	CK-2017357	iuphar.ligand:8280	TIRASEMTIV	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.1581556362520918	IUPHAR.LIGAND:122	iuphar.ligand:122	DIPROPYL-5-CT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.027505328	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:182	iuphar.ligand:182	LY320954	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.021933029	IUPHAR.LIGAND:34	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.015434354	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:199	ncit:C169779	AMESERGIDE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.037363144	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:174	iuphar.ligand:174	AC-90179	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:8430	iuphar.ligand:8430	[11C]GSK215083	FALSE	FALSE	FALSE
NCBIGENE:3060	hgnc:4847	HCRT	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:10184	iuphar.ligand:10184	TH5487	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.3777530304726222	IUPHAR.LIGAND:10526	iuphar.ligand:10526	SIAIS178	FALSE	FALSE	FALSE
NCBIGENE:1263	hgnc:2154	PLK3	GuideToPharmacology	2024.1	modulator	0.8751278539282416	IUPHAR.LIGAND:10645	ncit:C169983	FIRSOCOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.8008364246019593	IUPHAR.LIGAND:5890	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:1264	hgnc:2155	CNN1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:12243	iuphar.ligand:12243	CP-640186	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:12092	iuphar.ligand:12092	UNECRITINIB	FALSE	FALSE	FALSE
NCBIGENE:2768	hgnc:4380	GNA12	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7411	ncit:C81356	LIDORESTAT ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:482	iuphar.ligand:482	HEAT (BE2254)	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.2134458180312784	IUPHAR.LIGAND:483	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:496	ncit:C75061	UPIDOSIN	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.080042182	IUPHAR.LIGAND:485	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:493	rxcui:720825	SILODOSIN	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.012302641	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1084869240406911	IUPHAR.LIGAND:7268	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.1259176768242074	IUPHAR.LIGAND:523	ncit:C75049	XYLAZINE	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.012185582	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.018887652	IUPHAR.LIGAND:7241	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.031479419	IUPHAR.LIGAND:520	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	modulator	0.075550606	IUPHAR.LIGAND:4186	iuphar.ligand:4186	ETHYLISOPROPYLAMILORIDE	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.099446347	IUPHAR.LIGAND:520	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.032572997	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:523	ncit:C75049	XYLAZINE	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:7117	rxcui:14845	APRACLONIDINE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:2861	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:428	iuphar.ligand:428	KF 17837S	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:427	iuphar.ligand:427	CPX	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:393	iuphar.ligand:393	MRS1042	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:472	iuphar.ligand:472	MRS1486	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:2504	rxcui:1999003	ANGIOTENSIN II	TRUE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:6902	drugbank:DB12199	TRV-120027	FALSE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7710	iuphar.ligand:7710	AZD5582	FALSE	FALSE	FALSE
NCBIGENE:2957	hgnc:4646	GTF2A1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:11778	iuphar.ligand:11778	BCL6 PROTAC 15	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8509	iuphar.ligand:8509	COMPOUND 9G [PMID: 24412111]	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:632	iuphar.ligand:632	[D-PHE6,&BETA;-ALA11,PHE13,NLE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:7455	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.1875273972703375	IUPHAR.LIGAND:3465	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:560	rxcui:10368	TERBUTALINE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:9326	ncit:C132738	ABEDITEROL	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:547	iuphar.ligand:547	SR59230A	FALSE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:11413	iuphar.ligand:11413	NEMTABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1941	hgnc:18041	BMP2K	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11895	iuphar.ligand:11895	COMPOUND 13 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:2730	hgnc:4312	GCLM	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:7810	iuphar.ligand:7810	COMPOUND 2 [PMID: 25408830]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:10728	iuphar.ligand:10728	MZ1	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:10743	iuphar.ligand:10743	NHWD-870	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:7837	ncit:C97037	SPEBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:9265	ncit:C102876	TIRABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:9752	ncit:C141427	EVOBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8066	iuphar.ligand:8066	CGI1746	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:11413	iuphar.ligand:11413	NEMTABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:665	iuphar.ligand:665	COMPOUND 11 [PMID: 12812482]	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:646	iuphar.ligand:646	[DES-ARG9]BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:11252	iuphar.ligand:11252	C3A RECEPTOR AGONIST	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:677	iuphar.ligand:677	WIN 64338	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:667	rxcui:1148138	ICATIBANT	TRUE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8379	iuphar.ligand:8379	SQ007-5	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.089756703	IUPHAR.LIGAND:6814	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:6810	rxcui:60207	DORZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.096167896	IUPHAR.LIGAND:6792	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1995	hgnc:3314	ELAVL3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:5985	iuphar.ligand:5985	IC261	FALSE	FALSE	FALSE
NCBIGENE:1594	hgnc:2606	CYP27B1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8657	iuphar.ligand:8657	UK-396,082	FALSE	FALSE	FALSE
NCBIGENE:1594	hgnc:2606	CYP27B1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8675	iuphar.ligand:8675	COMPOUND 3 [PMID: 14640538]	FALSE	FALSE	FALSE
NCBIGENE:2000	hgnc:3319	ELF4	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8154	iuphar.ligand:8154	COMPOUND 14 [PMID: 24900428]	FALSE	FALSE	FALSE
NCBIGENE:1618	hgnc:2685	DAZL	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8628	iuphar.ligand:8628	COMPOUND 4 [PMID: 12408711]	FALSE	FALSE	FALSE
NCBIGENE:1997	hgnc:3316	ELF1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8154	iuphar.ligand:8154	COMPOUND 14 [PMID: 24900428]	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	1.009762908	IUPHAR.LIGAND:716	iuphar.ligand:716	NPS 2143	FALSE	FALSE	FALSE
NCBIGENE:534	hgnc:862	ATP6V1G2	GuideToPharmacology	2024.1	blocker	2.625383561784725	IUPHAR.LIGAND:2525	iuphar.ligand:2525	PB2+	FALSE	FALSE	FALSE
SMDT1	hgnc:25055	SMDT1	PharmGKB	4/5/24	NULL	6.563458904461812	dextromethorphan	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7720	iuphar.ligand:7720	ML218	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10883	iuphar.ligand:10883	GC-376	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.3182283105193606	IUPHAR.LIGAND:759	iuphar.ligand:759	CCL7	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:3696	iuphar.ligand:3696	COMPOUND 2B-1 [PMID: 12614873]	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:756	iuphar.ligand:756	CCL3	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9032	iuphar.ligand:9032	INCB8761	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:775	iuphar.ligand:775	CCL24	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:756	iuphar.ligand:756	CCL3	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:770	iuphar.ligand:770	CCL13	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.081533651	IUPHAR.LIGAND:7401	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1426838892274307	IUPHAR.LIGAND:6661	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.08780547	IUPHAR.LIGAND:7273	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:8530	iuphar.ligand:8530	CXCL12&GAMMA;	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:851	iuphar.ligand:851	SDF-1, 1-9[P2G] DIMER	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:8580	ncit:C126660	MAVORIXAFOR	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:853	iuphar.ligand:853	T140	FALSE	FALSE	FALSE
NCBIGENE:74	hgnc:147	ACTG1P2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:856	iuphar.ligand:856	CX3CL1	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:8160	iuphar.ligand:8160	COMPOUND 9B [PMID: 18986805]	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2041114528112516	IUPHAR.LIGAND:7380	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:11662	iuphar.ligand:11662	CP-10	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12076	iuphar.ligand:12076	CROZBACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1321	ncbigene:1321	CORD4	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:5180	iuphar.ligand:5180	ESCULETIN	FALSE	FALSE	FALSE
NCBIGENE:1319	ncbigene:1319	CORD1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11351	iuphar.ligand:11351	5H78PF	FALSE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.2075402025126264	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:6197	iuphar.ligand:6197	HAMI3379	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:6194	iuphar.ligand:6194	N-METHYL LTC4	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:1607	iuphar.ligand:1607	DADLE	FALSE	FALSE	FALSE
NCBIGENE:2603	hgnc:2861	DHFR	GuideToPharmacology	2024.1	inhibitor	2.734774543525755	IUPHAR.LIGAND:6840	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.3182283105193606	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	5.527123287967842	IUPHAR.LIGAND:7406	ncit:C1560	BREQUINAR	FALSE	FALSE	FALSE
NCBIGENE:2821	hgnc:4458	GPI	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7831	iuphar.ligand:7831	COMPOUND 5B [PMID: 25349648]	FALSE	FALSE	FALSE
XPO1	hgnc:12825	XPO1	PharmGKB	4/5/24	NULL	0.6250913242344582	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.007217549	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.058997383	IUPHAR.LIGAND:3296	iuphar.ligand:3296	[3H]7-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.007374673	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.003806283	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.039331589	IUPHAR.LIGAND:143	iuphar.ligand:143	SB 277011-A	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.011767743	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.008428198	IUPHAR.LIGAND:5501	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.036821649	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8956	iuphar.ligand:8956	BAY-678	FALSE	FALSE	FALSE
CA12	hgnc:1371	CA12	PharmGKB	4/5/24	NULL	0.300043836	zonisamide	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2895	hgnc:4576	GRID2	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:9098	iuphar.ligand:9098	CAROTUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6694	iuphar.ligand:6694	PF-04457845	FALSE	FALSE	FALSE
NCBIGENE:1401	hgnc:2367	CRP	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:5235	iuphar.ligand:5235	OL135	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1500219178162699	tolazamide	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:2806	drugbank:DB08231	MYRISTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:1050	iuphar.ligand:1050	GW9508	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	0.1256164383629055	IUPHAR.LIGAND:1056	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
CCL11	hgnc:10610	CCL11	PharmGKB	4/5/24	NULL	0.5147810905460245	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:3420	iuphar.ligand:3420	(S)-4-CMTB	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:9787	drugbank:DB12903	DEBIO-1347	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:7707	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:9039	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:11414	iuphar.ligand:11414	TASURGRATINIB	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:9039	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:9787	drugbank:DB12903	DEBIO-1347	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:9767	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:11887	iuphar.ligand:11887	TINENGOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:12370	ncit:C174208	LIRAFUGRATINIB	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.060878459	lorazepam	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:9767	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:9039	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.024861587	IUPHAR.LIGAND:5660	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.024861587	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.032173818	IUPHAR.LIGAND:5056	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.082043236	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:9921	iuphar.ligand:9921	TAFETINIB	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.045461187	IUPHAR.LIGAND:5660	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:9921	iuphar.ligand:9921	TAFETINIB	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:5835	iuphar.ligand:5835	AG-14	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:1027	iuphar.ligand:1027	[125I]CHIPS	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:6268	iuphar.ligand:6268	AG-26	FALSE	FALSE	FALSE
NPY1R	hgnc:7956	NPY1R	PharmGKB	4/5/24	NULL	0.3088686543276147	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:9875	ncit:C152337	SEPETAPROST	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:1940	ncit:C76900	FLUPROSTENOL	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:6264	iuphar.ligand:6264	FPRL1-INHIBITOR PROTEIN	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4327	iuphar.ligand:4327	TPA023	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.01123399	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:2366	hgnc:3874	FRA1G	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8658	iuphar.ligand:8658	PEPTIDE 18 [PMID: 24350995]	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	blocker	0.021422958	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6087	iuphar.ligand:6087	GALANIN(1-16) (RAT/MOUSE/PIG)	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.021891879	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:6125	iuphar.ligand:6125	SNAP 398299	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6091	iuphar.ligand:6091	GALANIN(3-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6087	iuphar.ligand:6087	GALANIN(1-16) (RAT/MOUSE/PIG)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6104	iuphar.ligand:6104	M1153	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:3593	iuphar.ligand:3593	GALANIN	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:3593	iuphar.ligand:3593	GALANIN	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3200	iuphar.ligand:3065	COMPOUND 1 [OVERHAND ET AL., 1997]	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.2500365296937833	IUPHAR.LIGAND:4288	rxcui:8351	PIRACETAM	FALSE	FALSE	FALSE
SEPTIN3	hgnc:10750	SEPTIN3	PharmGKB	4/5/24	NULL	1.615620653405984	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:9653	iuphar.ligand:9653	GSK866	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4080	iuphar.ligand:4080	[3H]CGS19755	FALSE	FALSE	FALSE
NCBIGENE:451	hgnc:769	ASS1P6	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:4317	iuphar.ligand:4317	SYM2081	FALSE	FALSE	FALSE
NCBIGENE:453	hgnc:771	ASS1P8	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:4317	iuphar.ligand:4317	SYM2081	FALSE	FALSE	FALSE
NCBIGENE:454	hgnc:772	ASS1P9	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:4181	drugbank:DB02852	DOMOIC ACID	FALSE	FALSE	FALSE
SULT2B1	hgnc:11459	SULT2B1	PharmGKB	4/5/24	NULL	0.3241214273808302	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:453	hgnc:771	ASS1P8	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:4085	iuphar.ligand:4085	[3H]KAINATE	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:4250	iuphar.ligand:4250	LY466195	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:4080	iuphar.ligand:4080	[3H]CGS19755	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1173	iuphar.ligand:1173	[TYR8]GNRH	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:1175	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:12058	drugbank:DB02342	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	PharmGKB	4/5/24	NULL	0.1103102336884338	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1469	hgnc:2473	CST1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8143	iuphar.ligand:8143	COMPOUND 1O [PMID: 24210504]	FALSE	FALSE	FALSE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9163	iuphar.ligand:9163	PEPTIDE P19 [PMID: 15652659]	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:9067	iuphar.ligand:9067	PL-3994	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	0.1250182648468916	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:723	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:1590	iuphar.ligand:1590	3-PYRIDINE-ACETIC ACID	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	0.1630673019742065	IUPHAR.LIGAND:1588	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
METTL21A	hgnc:30476	METTL21A	PharmGKB	4/5/24	NULL	2.250328767	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:2032	ncbigene:2032	ENUR2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:7495	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.1268301237577161	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.047432404	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:11119	iuphar.ligand:11119	BAVAROSTAT	FALSE	FALSE	FALSE
CFH	hgnc:4883	CFH	PharmGKB	4/5/24	NULL	4.773424657790409	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.077789143	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.095468493	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:1200	iuphar.ligand:1200	UR-PG146	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.028739831	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:212	rxcui:10510	THIOTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:207	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.033529803	IUPHAR.LIGAND:2608	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
GPX5	hgnc:4557	GPX5	PharmGKB	4/5/24	NULL	0.2414145803939976	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.019468918	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:1214	rxcui:356887	LEVOCETIRIZINE	TRUE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3015	iuphar.ligand:3015	COMPOUND 11JJ [PMID: 1656041]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	0.1944728564284981	IUPHAR.LIGAND:2488	ncit:C166774	OLVANIL	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.069454592	sacituzumab govitecan	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
NCBIGENE:84	ncbigene:84	ACTL4	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10206	iuphar.ligand:10206	NE 52-QQ57	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:10539	iuphar.ligand:10539	MANSC (415-431)	FALSE	FALSE	FALSE
NCBIGENE:2371	hgnc:3879	FRA1L	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8599	iuphar.ligand:8599	QUINOLINE 2	FALSE	FALSE	FALSE
ZMAT4	hgnc:25844	ZMAT4	PharmGKB	4/5/24	NULL	4.039051633514962	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
NCBIGENE:2375	hgnc:3887	FRA2C	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8488	iuphar.ligand:8488	COMPOUND 3 [PMID: 23849879]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1630	ncit:C170234	NORMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.076765601	IUPHAR.LIGAND:1663	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.1037701012563132	IUPHAR.LIGAND:12905	iuphar.ligand:12905	DUAL VEGFR/PARP INHIBITOR 14B	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	PharmGKB	4/5/24	NULL	1.346350544504987	crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.005061956	IUPHAR.LIGAND:5661	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0296486	IUPHAR.LIGAND:11887	iuphar.ligand:11887	TINENGOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:11510	iuphar.ligand:11510	M4205	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	antibody	0.9907107780319716	IUPHAR.LIGAND:11607	iuphar.ligand:11607	BARZOLVOLIMAB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:5689	iuphar.ligand:5689	JNJ-28312141	FALSE	FALSE	FALSE
NCBIGENE:525	hgnc:853	ATP6V1B1	GuideToPharmacology	2024.1	blocker	2.625383561784724	IUPHAR.LIGAND:2503	rxcui:1362698	CHLOROFORM	TRUE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	blocker	0.8334550989792776	IUPHAR.LIGAND:2315	iuphar.ligand:2315	LEI-DAB7	FALSE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.106290832	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2311	iuphar.ligand:2311	APAMIN	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:2314	iuphar.ligand:2314	EBIO	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	blocker	0.182318303	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:437	hgnc:6266	KCNJ5	GuideToPharmacology	2024.1	blocker	2.917092846427472	IUPHAR.LIGAND:7704	iuphar.ligand:7704	AZD2927	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.1037701012563132	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:7661	iuphar.ligand:7661	A-935142	FALSE	FALSE	FALSE
NCBIGENE:545	hgnc:882	ATR	GuideToPharmacology	2024.1	blocker	0.079557078	IUPHAR.LIGAND:2568	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
NCBIGENE:547	hgnc:888	KIF1A	GuideToPharmacology	2024.1	blocker	0.6731752722524936	IUPHAR.LIGAND:2510	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	1.346350544504987	IUPHAR.LIGAND:2600	iuphar.ligand:2600	(S)-N-[1-(3-MORPHOLIN-4-YL-PHENYL)-ETHYL]-3-PHENYL-ACRYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:2599	ncit:C82306	LINOPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	blocker	0.2430910705356227	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	blocker	0.1620607136904151	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6710	iuphar.ligand:6710	RO 48-8071	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:11730	iuphar.ligand:11730	TAK-020	FALSE	FALSE	FALSE
GCKR	hgnc:4196	GCKR	PharmGKB	4/5/24	NULL	0.1899011617927468	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:1838	hgnc:3058	DTNB	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.028283152	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:5151	ncit:C1015	UBENIMEX	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9396	iuphar.ligand:9396	LRRK2-IN-1	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12908	iuphar.ligand:12908	JH-XII-03-02	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12009	iuphar.ligand:12009	XL01126	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	PharmGKB	4/5/24	NULL	0.088248187	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8690	iuphar.ligand:8690	GSK2033	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.1852122442176172	AEE 788	ncit:C48369	MULTIKINASE INHIBITOR AEE788	FALSE	FALSE	TRUE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	modulator	1.166837138570988	IUPHAR.LIGAND:8693	iuphar.ligand:8693	GSK9772	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:2905	iuphar.ligand:2905	AM966	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:6983	iuphar.ligand:6983	OLEOYL-THIOPHOSPHATE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.043866058	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2677	hgnc:4247	GGCX	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:12807	iuphar.ligand:12807	ZAVONDEMSTAT	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	activator	5.250767123569449	IUPHAR.LIGAND:8390	iuphar.ligand:8390	ORY-1001	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9116	iuphar.ligand:9116	GSK2879552	FALSE	FALSE	FALSE
NCBIGENE:2668	hgnc:4232	GDNF	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:12938	iuphar.ligand:12938	PF-9363	FALSE	FALSE	FALSE
NCBIGENE:2718	hgnc:28405	KMT5C	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8949	iuphar.ligand:8949	A-196	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	0.8751278539282418	IUPHAR.LIGAND:9272	iuphar.ligand:9272	SETMELANOTIDE	FALSE	FALSE	FALSE
NCBIGENE:283	hgnc:483	ANG	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:1332	iuphar.ligand:1332	ACTH-(11-24)	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1308	iuphar.ligand:1308	S36539	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1315	iuphar.ligand:1315	TPI 1361-17	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	0.6403374540938354	IUPHAR.LIGAND:1416	iuphar.ligand:1416	PHCCC	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6338	iuphar.ligand:6338	COMPOUND 23H [PMID: 17929793]	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.3860858179095183	IUPHAR.LIGAND:6224	iuphar.ligand:6224	COMPOUND 4 [PMID: 21105727]	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6362	iuphar.ligand:6362	COMPOUND 9N [PMID: 23084894]	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	TALC	12-May-16	inhibitor	0.076765601	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6321	iuphar.ligand:6321	COMPOUND 34 [PMID: 20409708]	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6320	iuphar.ligand:6320	COMPOUND 48 [PMID: 22364337]	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:5676	iuphar.ligand:5676	CI-1040	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:306	ncit:C152278	SABCOMELINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:309	iuphar.ligand:309	OTENZEPAD	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:296	drugbank:DB04365	ARECOLINE	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.074690855	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:296	drugbank:DB04365	ARECOLINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:297	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:331	iuphar.ligand:331	SILAHEXOCYCLIUM	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:3274	iuphar.ligand:3274	VU0255035	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:299	ncit:C76041	FURTRETHONIUM IODIDE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1988926940746003	IUPHAR.LIGAND:306	ncit:C152278	SABCOMELINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:296	drugbank:DB04365	ARECOLINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:8593	iuphar.ligand:8593	[3H]ACETYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.054243462	IUPHAR.LIGAND:359	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:318	iuphar.ligand:318	[3H]QNB	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:331	iuphar.ligand:331	SILAHEXOCYCLIUM	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1351	iuphar.ligand:1351	LY 156735	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:10666	iuphar.ligand:10666	UCSF7447	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:2615	iuphar.ligand:2615	BC-III	FALSE	FALSE	FALSE
NCBIGENE:585	hgnc:969	BBS4	GuideToPharmacology	2024.1	blocker	3.750547945	IUPHAR.LIGAND:12002	iuphar.ligand:12002	ABBV-318	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:10119	iuphar.ligand:10119	AM-6120	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3971	iuphar.ligand:3971	[3H]AZ11637326	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:2132	ncit:C76464	TALNETANT	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5752	ncit:C72949	VOFOPITANT	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:2106	iuphar.ligand:2106	SCH 206272	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:5775	ncit:C166698	PAVINETANT	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:2130	iuphar.ligand:2130	N',2-DIPHENYLQUINOLINE-4-CARBOHYDRAZIDE 8M	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:2132	ncit:C76464	TALNETANT	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8228	iuphar.ligand:8228	MCC950	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:10057	iuphar.ligand:10057	CY-09	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:10380	iuphar.ligand:10380	CPN-267	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:9009	iuphar.ligand:9009	NM4-C16	FALSE	FALSE	FALSE
NCBIGENE:2129	hgnc:14311	NUAK1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:11879	iuphar.ligand:11879	NARAZACICLIB	FALSE	FALSE	FALSE
NCBIGENE:2129	hgnc:14311	NUAK1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:8977	iuphar.ligand:8977	HTH-01-015	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	inhibitor	0.1268301237577161	IUPHAR.LIGAND:4749	ncit:C47521	ESTROPIPATE	FALSE	FALSE	FALSE
NCBIGENE:2130	hgnc:3508	EWSR1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11085	iuphar.ligand:11085	HTH-02-006	FALSE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	NULL	0.42006137	IUPHAR.LIGAND:4505	iuphar.ligand:4505	[3H]BSP	FALSE	FALSE	FALSE
NCBIGENE:2965	hgnc:4655	GTF2H1	GuideToPharmacology	2024.1	blocker	13.12691780892362	IUPHAR.LIGAND:10088	iuphar.ligand:10088	GSK-7975A	FALSE	FALSE	FALSE
NCBIGENE:2964	hgnc:4654	GTF2F2P1	GuideToPharmacology	2024.1	blocker	5.250767123569449	IUPHAR.LIGAND:10088	iuphar.ligand:10088	GSK-7975A	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2245	iuphar.ligand:2245	L-366,948	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2251	iuphar.ligand:2251	L-369,020	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:2223	iuphar.ligand:2223	D(CH2)5[TYR(ME)2]AVP	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	0.5645986154375752	IUPHAR.LIGAND:1710	iuphar.ligand:1710	2MESADP	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9470	iuphar.ligand:9470	MRS4174	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1727	iuphar.ligand:1727	[3H]MRS2279	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:9135	iuphar.ligand:9135	MK-0893	FALSE	FALSE	FALSE
NCBIGENE:347	hgnc:612	APOD	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:3823	iuphar.ligand:3823	[3H]HATRAP	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:4702	iuphar.ligand:4702	4-AMBA	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	0.044385183	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2658	iuphar.ligand:2658	LY-518674	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:10751	iuphar.ligand:10751	(R)-16 [PMID: 32267688]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:10601	iuphar.ligand:10601	AZD7648	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.039331589	IUPHAR.LIGAND:12616	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:9800	iuphar.ligand:9800	SELETALISIB	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.098328972	IUPHAR.LIGAND:10627	ncit:C123925	ZANDELISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:9997	iuphar.ligand:9997	AZD3458	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:9997	iuphar.ligand:9997	AZD3458	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:9916	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:10441	iuphar.ligand:10441	COMPOUND 5D [PMID: 31335136]	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:12062	iuphar.ligand:12062	COMPOUND 27 [PMID: 35834807]	FALSE	FALSE	FALSE
NCBIGENE:2858	ncbigene:2858	GPR34P	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11794	iuphar.ligand:11794	BAY-297	FALSE	FALSE	FALSE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:6557	iuphar.ligand:6557	RS-25344	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:12099	iuphar.ligand:12099	TUNODAFIL	FALSE	FALSE	FALSE
NCBIGENE:1308	hgnc:2194	COL17A1	GuideToPharmacology	2024.1	inhibitor	0.3723948314588262	IUPHAR.LIGAND:4807	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11099	iuphar.ligand:11099	COMPOUND 3M [PMID: 32603117]	FALSE	FALSE	FALSE
NCBIGENE:1306	hgnc:2192	COL15A1	GuideToPharmacology	2024.1	inhibitor	0.074478966	IUPHAR.LIGAND:4807	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:2773	iuphar.ligand:2773	S20	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.007235451	IUPHAR.LIGAND:2377	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:2391	hgnc:3903	FRA4D	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8634	iuphar.ligand:8634	COMPOUND 3 [PMID: 8410973]	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.062065805	IUPHAR.LIGAND:1013	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:1161	hgnc:3439	ERCC8	GuideToPharmacology	2024.1	inhibitor	0.4375639269641209	IUPHAR.LIGAND:7071	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
NCBIGENE:1161	hgnc:3439	ERCC8	GuideToPharmacology	2024.1	inhibitor	0.1861974157294131	IUPHAR.LIGAND:1013	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	0.5834185692854945	IUPHAR.LIGAND:3738	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
NCBIGENE:3007	hgnc:4717	H1-3	GuideToPharmacology	2024.1	modulator	13.12691780892362	IUPHAR.LIGAND:11975	ncit:C176893	ETAVOPIVAT	FALSE	FALSE	FALSE
NCBIGENE:3006	hgnc:4716	H1-2	GuideToPharmacology	2024.1	activator	7.501095891	IUPHAR.LIGAND:10556	iuphar.ligand:10556	DASA-58	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8187	iuphar.ligand:8187	COMPOUND 21 [PMID: 24900635]	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:9554	iuphar.ligand:9554	GSK2982772	FALSE	FALSE	FALSE
NCBIGENE:1524	hgnc:2558	CX3CR1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8763	iuphar.ligand:8763	COMPOUND 8 [PMID: 17480064]	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:2924	iuphar.ligand:2924	FINGOLIMOD-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:11312	iuphar.ligand:11312	CYM5520	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	TALC	12-May-16	inhibitor	9.723642821424907	FICLATUZUMAB	ncit:C78844	FICLATUZUMAB	FALSE	TRUE	TRUE
NCBIGENE:3103	hgnc:10721	SELP	GuideToPharmacology	2024.1	antibody	2.625383561784724	IUPHAR.LIGAND:12312	iuphar.ligand:12312	INCLACUMAB	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:9889	iuphar.ligand:9889	RP-101075	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2221	ncbigene:2221	FCP1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8190	iuphar.ligand:8190	COMPOUND 1 [PMID: 21742770]	FALSE	FALSE	FALSE
NCBIGENE:2397	hgnc:3908	FRA5D	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2214	hgnc:3619	FCGR3A	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:11894	iuphar.ligand:11894	COMPOUND 7 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7537	iuphar.ligand:7537	NORZOTEPINE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.074690855	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:1534	hgnc:2571	CYB561	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9407	iuphar.ligand:9407	EMD638683	FALSE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	modulator	1.693795846312725	IUPHAR.LIGAND:10326	iuphar.ligand:10326	GSA-10	FALSE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:7716	iuphar.ligand:7716	AZD8542	FALSE	FALSE	FALSE
NCBIGENE:2521	hgnc:4010	FUS	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10054	iuphar.ligand:10054	SPHINGOMYELIN SYNTHASE 2 INHIBITOR 15W	FALSE	FALSE	FALSE
NCBIGENE:2521	hgnc:4010	FUS	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8834	iuphar.ligand:8834	COMPOUND D24 [PMID: 24374347]	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9925	iuphar.ligand:9925	BALAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3108	iuphar.ligand:3108	COMPOUND 4Q [PMID: 7650673]	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:11886	ncit:C123912	SOVLEPLENIB	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:2030	iuphar.ligand:2030	SRA880	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:5645	iuphar.ligand:5645	DOTA-BASS	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2036	iuphar.ligand:2036	BIM 23056	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	0.3723948314588262	IUPHAR.LIGAND:2036	iuphar.ligand:2036	BIM 23056	FALSE	FALSE	FALSE
NCBIGENE:2418	hgnc:3929	FRA8A	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8488	iuphar.ligand:8488	COMPOUND 3 [PMID: 23849879]	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.2488515224440497	IUPHAR.LIGAND:11661	iuphar.ligand:11661	TBK1 PROTAC 3I	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	0.3281729452230906	IUPHAR.LIGAND:2635	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:5051	ncit:C63958	RESIQUIMOD	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6293	iuphar.ligand:6293	BROMOACETONE	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.066297565	IUPHAR.LIGAND:1056	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
NCBIGENE:502	hgnc:13357	MCOLN2	GuideToPharmacology	2024.1	activator	8.751278539282415	IUPHAR.LIGAND:10301	iuphar.ligand:10301	ML2-SA1	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.6908904109959803	IUPHAR.LIGAND:2443	iuphar.ligand:2443	ACAA	FALSE	FALSE	FALSE
NCBIGENE:2752	hgnc:4341	GLUL	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:8854	iuphar.ligand:8854	COMBRETASTATIN A4	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	3.962843112127886	FIGITUMUMAB	ncit:C52187	FIGITUMUMAB	FALSE	TRUE	TRUE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:10148	iuphar.ligand:10148	JAK INHIBITOR 17B	FALSE	FALSE	FALSE
NCBIGENE:1841	hgnc:3061	DTYMK	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11791	iuphar.ligand:11791	BIIB091	FALSE	FALSE	FALSE
NCBIGENE:3063	ncbigene:3063	HCVS	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11718	iuphar.ligand:11718	VANIN-1 INHIBITOR [PMID: 33196323]	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:2223	iuphar.ligand:2223	D(CH2)5[TYR(ME)2]AVP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:2221	iuphar.ligand:2221	D(CH2)5[TYR(ME)2,THR4,TYR-NH29]OVT	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:3800	iuphar.ligand:3800	[125I]PP (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1544	iuphar.ligand:1544	[D-TRP32]NPY	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	1.374546367426557	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
BRD4	hgnc:13575	BRD4	CIViC	10-Apr-24	NULL	0.3454452054979901	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.087782887	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
KIF11	hgnc:6388	KIF11	TALC	12-May-16	inhibitor	9.845188356692718	ARRY-520	ncit:C68937	FILANESIB	FALSE	FALSE	TRUE
EWSR1	hgnc:3508	EWSR1	CIViC	10-Apr-24	NULL	0.2678962818147678	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HMOX1	hgnc:5013	HMOX1	CIViC	10-Apr-24	NULL	0.1190650141398968	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.364636606	PATRITUMAB	ncit:C78853	PATRITUMAB	FALSE	TRUE	TRUE
NTRK3	hgnc:8033	NTRK3	CIViC	10-Apr-24	NULL	0.1110098757625676	REPOTRECTINIB	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.016086909	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.6961244292611014	REPOTRECTINIB	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.2734774543525755	SHP2 INHIBITOR RMC-4630	ncit:C155850	VOCIPROTAFIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.1999620096341412	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.023151531	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1135300999690691	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.053217234	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
RAD50	hgnc:9816	RAD50	CIViC	10-Apr-24	NULL	0.8334550989792777	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SMARCA4	hgnc:11100	SMARCA4	CIViC	10-Apr-24	NULL	0.3454452054979901	ABEMACICLIB	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.092443083	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
TF	hgnc:11740	TF	CIViC	10-Apr-24	NULL	0.364636606	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.057574201	ABEMACICLIB	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	0.2739530673166669	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.3517260274161354	FUTIBATINIB	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.021172448	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
B2M	hgnc:914	B2M	CIViC	10-Apr-24	NULL	0.750109589	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MAGEA3	hgnc:6801	MAGEA3	TALC	12-May-16	vaccine	35.00511415712966	GSK1572932A	ncit:C78478	ASTUPROTIMUT-R	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.046059361	OSIMERTINIB	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
ERRFI1	hgnc:18185	ERRFI1	CIViC	10-Apr-24	NULL	2.917092846427472	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	CIViC	10-Apr-24	NULL	0.3922986931402463	4'-(9-ACRIDINYLAMINO)METHANESULFON-M-ANISIDIDE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	CIViC	10-Apr-24	NULL	0.652269208	FEDRATINIB	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.001347802	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
EPHA2	hgnc:3386	EPHA2	DoCM	10-Apr-24	NULL	0.4167275494896388	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	DoCM	10-Apr-24	NULL	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
MAGEA2	hgnc:6800	MAGEA2	TALC	12-May-16	vaccine	13.12691780892362	EP-2101	ncit:C26645	MULTI-NEO-EPITOPE VACCINE OSE 2101	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	0.091636424	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	DoCM	10-Apr-24	NULL	0.6326225450083675	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
ARAF	hgnc:646	ARAF	DoCM	10-Apr-24	NULL	0.075369863	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	0.082115757	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	DoCM	10-Apr-24	NULL	0.3968833804663227	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.060878459	Zoledronic acid	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2290910612377596	CCT196969	iuphar.ligand:9815	CCT196969	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2061819551139836	Nab-paclitaxel	ncit:C2688	NAB-PACLITAXEL	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.1842374429322613	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.034363659	Mocetinostat	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	AZD0364	ncit:C176765	TIZATERKIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	CFT1946	iuphar.ligand:12623	CFT1946	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.078545507	Sapitinib	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.027454991	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.5048814541893701	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	1.141471113819445	APG-2449	chembl:CHEMBL5095166	APG-2449	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.138178082	Cetrelimab	ncit:C129448	CETRELIMAB	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.3889457128569963	Infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.1200175342530159	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.3818739726232327	Buthionine sulfoximine	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.1201548540862574	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.6326225450083675	IDRX-42	drugbank:DB18087	IDRX-42	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.6326225450083675	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.7143900848393808	Refametinib	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.8751278539282416	RG7112	drugbank:DB14793	RO-5045337	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.078136416	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	1.750255707856483	Idasanutlin	ncit:C99131	IDASANUTLIN	FALSE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	1.218928082257193	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2234869519440402	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.096264064	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1999620096341412	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.045369532	Adavosertib	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	Anti-CD19 CAR-T cells	ncit:C176018	ANTI-CD19 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.087782887	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	BAY1082439	ncit:C103861	PI3K ALPHA/BETA INHIBITOR BAY1082439	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.064824285	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	Onatasertib	ncit:C92575	ONATASERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.4861821410712453	Inavolisib	ncit:C132166	INAVOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	TOS-358	ncit:C198692	PI3K-ALPHA INHIBITOR TOS-358	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	PKI-179	drugbank:DB13109	PKI-179	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	TALC	12-May-16	inhibitor	1.225178995499538	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	Ridaforolimus	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	1.077080435603989	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.019447286	Topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	0.600087671	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	0.3500511415712967	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	0.1458546423213736	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1520492410300034	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.05068308	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.4688184931758437	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.044347695	Voxtalisib	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.088695391	Abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.06335385	Gedatolisib	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.062608511	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.052560231	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.039420174	Tipifarnib	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1182605208011137	Ganitumab	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
RAF1	hgnc:9829	RAF1	TALC	12-May-16	antisense oligonucleotide	2.019525817	ISIS 5132	ncit:C2721	C-RAF ANTISENSE OLIGONUCLEOTIDE ISIS 5132	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.9723642821424906	M8891	iuphar.ligand:12714	M8891	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.007292732	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE	chembl:CHEMBL1569494	CHEMBL:CHEMBL1569494	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.076765601	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	TALC	12-May-16	inhibitor	0.07699072	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.024932417	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
OR10AE3P	hgnc:31235	OR10AE3P	PharmGKB	4/5/24	NULL	0.8824818695074705	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.252440727	ABI-011	ncit:C116890	NANOPARTICLE ALBUMIN-BOUND THIOCOLCHICINE DIMER NAB-5404	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.1060761035064535	JNJ-26481585	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.098053541	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
BIRC6	hgnc:13516	BIRC6	TALC	12-May-16	inhibitor	3.281729452230906	TL 32711	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:6040	iuphar.ligand:6040	SKF-86002	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9355	iuphar.ligand:9355	GNE-3511	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:9658	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:311	iuphar.ligand:311	MUSCARINIC TOXIN 1	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.1060761035064535	IUPHAR.LIGAND:2182	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.1093909817410302	IUPHAR.LIGAND:5429	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.2234869519440402	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.4565884455277782	APG-2449	chembl:CHEMBL5095166	APG-2449	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	CGP-13501	iuphar.ligand:7848	CGP13501	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.092933931	clindamycin	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	TALC	12-May-16	inhibitor	1.826353782111112	X-396	drugbank:DB13104	X-396	FALSE	FALSE	TRUE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	modulator	1.575230137070835	SOLITOMAB	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
OCRL	hgnc:8108	OCRL	PharmGKB	4/5/24	NULL	7.501095890813499	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
PERP	hgnc:17637	PERP	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.012079059	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.079718124	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	15.00219178	Latanoprost	rxcui:43611	LATANOPROST	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	0.750109589	Amosulalol	rxcui:2667256	AMOSULALOL	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	3.231241306811969	BIIB037	rxcui:2557217	ADUCANUMAB	TRUE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	0.2083637747448194	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.5125748858722557	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:9061	iuphar.ligand:9061	PF-03882845	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	ChEMBL	33	inhibitor	3.424413341458336	LORLATINIB	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.3977853881492007	SAROGLITAZAR	ncit:C152303	SAROGLITAZAR	FALSE	FALSE	FALSE
UNIPROT:P24821	hgnc:5318	TNC	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	NEURADIAB	ncit:C2488	IODINE I 131 MONOCLONAL ANTIBODY 81C6	FALSE	FALSE	FALSE
CCNB1	hgnc:1579	CCNB1	DTC	9/2/20	NULL	1.250182648468916	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.1562728310586145	TENOFOVIR	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	TALC	12-May-16	inhibitor	0.4167275494896388	SALINOSPORAMIDE A	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
UNIPROT:P29317	hgnc:3386	EPHA2	TdgClinicalTrial	Jan-14	NULL	0.4167275494896388	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P49146	hgnc:7957	NPY2R	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	PEPTIDE YY	iuphar.ligand:1514	PEPTIDE YY	FALSE	FALSE	FALSE
UNIPROT:Q9Y251	hgnc:5164	HPSE	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.099446347	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P14410	hgnc:10856	SI	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:835	iuphar.ligand:835	CXCL10	FALSE	FALSE	FALSE
NCBIGENE:623	hgnc:1029	BDKRB1	GuideToPharmacology	2024.1	agonist	0.100589408	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
UNIPROT:P37023	hgnc:175	ACVRL1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	DALANTERCEPT	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:10347	iuphar.ligand:10347	K-80003	FALSE	FALSE	FALSE
NCBIGENE:1233	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:5115	iuphar.ligand:5115	3-DEAZAADENOSINE	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.546954909	MUC1-TARGETED PEPTIDE GO-203-2C	ncit:C95722	MUC1-TARGETED PEPTIDE GO-203-2C	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.02956513	Veliparib	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.7955707762984014	CYCLIRAMINE MALEATE	ncit:C65355	CYCLIRAMINE MALEATE	FALSE	FALSE	FALSE
UNIPROT:P04746	hgnc:477	AMY2A	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:11694	iuphar.ligand:11694	SRI22141	FALSE	FALSE	FALSE
CYP2C18	hgnc:2620	CYP2C18	PharmGKB	4/5/24	NULL	0.5000730593875666	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.7955707762984014	CWP232291	ncit:C97663	SAM68 MODULATOR CWP232291	FALSE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.2573905452730122	IUPHAR.LIGAND:2397	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.1419126249613365	ACLIDINIUM	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.1041818873724097	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12372	iuphar.ligand:12372	ODITRASERTIB	FALSE	FALSE	FALSE
NCBIGENE:2252	hgnc:3685	FGF7	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8396	iuphar.ligand:8396	COMPOUND 34 [PMID: 25974391]	FALSE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	inhibitor	2.386712328895204	TOLVAPTAN	rxcui:358257	TOLVAPTAN	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	ANTHRACENE-9-CARBOXYLIC ACID	iuphar.ligand:4113	9-ANTHROIC ACID	FALSE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	INTERFERON BETA-1A	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	CV-1808	iuphar.ligand:420	CV-1808	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	NIFUROXAZIDE	rxcui:31782	NIFUROXAZIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000615493	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.060353645	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.9546849315580818	Valdecoxib	rxcui:278567	VALDECOXIB	TRUE	FALSE	FALSE
UNIPROT:P12268	hgnc:6053	IMPDH2	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	AVN-944	drugbank:DB05500	AVN-944	FALSE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 2	hgnc:6053	IMPDH2	TTD	2020.06.01	NULL	1.312691780892362	Mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	ESMOLOL HYDROCHLORIDE	rxcui:203222	ESMOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.029074015	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.1881995384791917	HEXADECYLPHOSPHOCHOLINE	rxcui:1494066	MILTEFOSINE	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	1.334940794127826	AZILSARTAN	rxcui:1091642	AZILSARTAN MEDOXOMIL	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	PharmGKB	4/5/24	NULL	0.012429322	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:674	iuphar.ligand:674	FR173657	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.7292732116068681	IL-1RA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.4605936073306534	Dacomitinib	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.2456499239096818	ONDANSETRON	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.1842374429322613	HMPL-453	chembl:CHEMBL4650297	HMPL-453	FALSE	FALSE	FALSE
IL18	hgnc:5986	IL18	ChEMBL	33	inhibitor	2.763561643983921	TADEKINIG ALFA	ncit:C152488	TADEKINIG ALFA	FALSE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	ChEMBL	33	inhibitor	2.386712328895204	PRI-724	drugbank:DB15034	PRI-724	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.525076712	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011575765	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.6563458904461812	E163	chembl:CHEMBL443095	E163	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	TCMDC-124307	chembl:CHEMBL546865	CHEMBL:CHEMBL546865	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.064347636	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	0.2333674277141977	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.099446347	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.05387244	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:2055	hgnc:2079	CLN8	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8118	iuphar.ligand:8118	COMPOUND 30 [PMID: 22902653]	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1136529680426288	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.1000146118775133	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:390	hgnc:671	RND3	GuideToPharmacology	2024.1	activator	0.1483267549030918	IUPHAR.LIGAND:2377	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:4366	iuphar.ligand:4366	[3H]CGS8216	FALSE	FALSE	FALSE
NCBIGENE:1768	hgnc:2951	DNAH6	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:5024	iuphar.ligand:5024	MURAMYL DIPEPTIDE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.3889457128569962	ISOPROPANOL	rxcui:797541	ISOPROPYL ALCOHOL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.062645859	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	ChEMBL	33	inhibitor	0.1190650141398968	SEMORINEMAB	ncit:C174790	SEMORINEMAB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.021805511	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	THEONELLASTEROL F	chembl:CHEMBL1782581	THEONELLASTEROL F	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.003324322	VERAPAMIL HYDROCHLORIDE	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P12931	hgnc:11283	SRC	TdgClinicalTrial	Jan-14	NULL	0.1691068316769549	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
FZD5	hgnc:4043	FZD5	ChEMBL	33	inhibitor	7.501095890813499	VANTICTUMAB	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	0.1260688385010672	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.3561566847382379	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.4487835148349957	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q8WW43	hgnc:24080	APH1B	TdgClinicalTrial	Jan-14	NULL	1.009762908	BMS-708163	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
PPA1	hgnc:9226	PPA1	NCI	14-Sep-17	NULL	0.6646540662746139	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.5933070196123671	SILYMARIN	rxcui:9794	SILYMARIN	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	4.039051633514961	PLX51107	drugbank:DB17543	PLX51107	FALSE	FALSE	FALSE
UNIPROT:Q96LZ3	hgnc:9318	PPP3R2	TdgClinicalTrial	Jan-14	NULL	1.207072901969988	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:2042	hgnc:3387	EPHA3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:5990	iuphar.ligand:5990	IRAK-1/4 INHIBITOR	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.060878459	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.079557078	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:643	iuphar.ligand:643	[SAR,D-PHE8,DES-ARG9]BRADYKININ	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.2419708351875322	CETIRIZINE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ZBTB22	hgnc:13085	ZBTB22	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:10408	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1472	iuphar.ligand:1472	NEUROMEDIN U-8	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.014287802	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.081407242	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.095122593	MECHLORETHAMINE HYDROCHLORIDE	rxcui:155036	MECHLORETHAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.033117421	levonorgestrel	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.079557078	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.8204323630577265	ADAGRASIB	rxcui:2625882	ADAGRASIB	TRUE	FALSE	TRUE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.2206204673768676	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.085239726	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.030176823	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.036162308	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
NFE2	hgnc:7780	NFE2	NCI	14-Sep-17	NULL	0.9723642821424907	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:P08253	hgnc:7166	MMP2	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	COL-3	ncit:C2454	INCYCLINIDE	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:7657	iuphar.ligand:7657	RPR260243	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:3274	iuphar.ligand:3274	VU0255035	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	N-PHENETHYL-NICOTINAMIDE	chembl:CHEMBL309848	CHEMBL:CHEMBL309848	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.5556367326528517	IUPHAR.LIGAND:10313	ncit:C138165	LEROCICLIB	FALSE	FALSE	FALSE
INTERLEUKIN-12 BETA	hgnc:5970	IL12B	TTD	2020.06.01	NULL	3.750547945	EGEN-001	drugbank:DB05953	EGEN-001	FALSE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.2453629496995069	AMPHETAMINE ADIPATE	ncit:C87425	AMPHETAMINE ADIPATE	TRUE	FALSE	FALSE
UNIPROT:P30874	hgnc:11331	SSTR2	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	DG3173	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
PSMD8	hgnc:9566	PSMD8	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	INDOTECAN	ncit:C95907	INDOTECAN	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	4.039051633514961	CTX	ncit:C400	CROTOXIN	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.2344092465879218	PENTAMIDINE ISETHIONATE	rxcui:7995	PENTAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.2059124362184097	DEXPRAMIPEXOLE	ncit:C169899	DEXPRAMIPEXOLE	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.046425881	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.011394894	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
UNIPROT:P31391	hgnc:11333	SSTR4	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	DG3173	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
TPO	hgnc:12015	TPO	ChEMBL	33	inhibitor	2.625383561784725	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
CASR	hgnc:1514	CASR	NCI	14-Sep-17	NULL	0.5966780822238011	PAMIDRONATE	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
UNIPROT:P35346	hgnc:11334	SSTR5	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	DG3173	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	0.021011473	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.045461187	IUPHAR.LIGAND:7741	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12018	iuphar.ligand:12018	COMPOUND A34 [PMID: 35635004]	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:496	ncit:C75061	UPIDOSIN	FALSE	FALSE	FALSE
UNIPROT:O95264	hgnc:5298	HTR3B	TdgClinicalTrial	Jan-14	NULL	0.3860858179095183	DOLASETRON	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	CGI	2/1/22	NULL	0.3968833804663227	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.016418909	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.073266518	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.591141552596803	ACYLINE	drugbank:DB11906	ACYLINE	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.3804903712731485	IUPHAR.LIGAND:2441	iuphar.ligand:2441	SKF96365	FALSE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TdgClinicalTrial	Jan-14	NULL	0.1182605208011137	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
ALDH2	hgnc:404	ALDH2	ChEMBL	33	inhibitor	0.07963752	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	7.001022831425932	DDD	chemidplus:72-54-8	TDE	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.022789788	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
UNIPROT:O14763	hgnc:11905	TNFRSF10B	TdgClinicalTrial	Jan-14	NULL	29.17092846427472	LEXATUMUMAB	ncit:C64621	LEXATUMUMAB	FALSE	TRUE	TRUE
UNIPROT:P13631	hgnc:9866	RARG	TEND	1-Aug-11	NULL	0.7721716358190367	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
POLE	hgnc:9177	POLE	CIViC	10-Apr-24	NULL	0.600087671	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	NSC-747267	chembl:CHEMBL610767	CHEMBL:CHEMBL610767	FALSE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	DTC	9/2/20	NULL	6.563458904461812	DIMETHYLENASTRON	chembl:CHEMBL394880	DIMETHYLENASTRON	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	DTC	9/2/20	NULL	0.789589041	GSK1210151A	iuphar.ligand:7518	I-BET151	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1193356164447602	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2404931506978374	FLUOCINOLONE ACETONIDE	rxcui:4461	FLUOCINOLONE ACETONIDE	TRUE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	DTC	9/2/20	NULL	0.4688184931758437	N6-CYCLOPENTYLADENOSINE	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.030176823	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
EPO	hgnc:3415	EPO	NCI	14-Sep-17	NULL	1.666910197958555	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	CGI	2/1/22	NULL	0.2957715794844315	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:5707	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9707	iuphar.ligand:9707	LINRODOSTAT	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.729273212	IUPHAR.LIGAND:8899	iuphar.ligand:8899	(S)-LIQUIRITIGENIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	QUINOLINIC ACID	drugbank:DB01796	QUINOLINIC ACID	FALSE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	0.072927321	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.1988926940746003	Mephenytoin	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.001593895	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	4.039051633514961	Filgrastim-SNDZ	rxcui:1433764	TBO-FILGRASTIM	TRUE	FALSE	FALSE
UNIPROT:O60664	hgnc:16893	PLIN3	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	GALSULFASE	rxcui:578033	GALSULFASE	TRUE	FALSE	FALSE
CD86	hgnc:1705	CD86	NCI	14-Sep-17	NULL	1.060761035064535	PAMIDRONATE	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	ChEMBL	33	inhibitor	0.2273059360852575	ASM-024	chembl:CHEMBL3707249	ASM-024	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.072125922	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	ChEMBL	33	inhibitor	1.381780822	RO-6870810	drugbank:DB15151	RO-6870810	FALSE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	1.591141552596803	GFT14	drugbank:DB05061	GFT14	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	ALIZAPRIDE	rxcui:17311	ALIZAPRIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	8-CYCLOPENTYLTHEOPHYLLINE	iuphar.ligand:385	8-CYCLOPENTYLTHEOPHYLLINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	PIMETHIXENE MALEATE	ncit:C97703	PIMETHIXENE MALEATE	FALSE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.1296485709523321	IUPHAR.LIGAND:2406	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:Q09428	hgnc:59	ABCC8	TdgClinicalTrial	Jan-14	NULL	0.2715914029432474	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TdgClinicalTrial	Jan-14	NULL	0.1795134059339982	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1B	hgnc:278	ADRA1B	TTD	2020.06.01	NULL	0.063415062	Methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:10408	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.018071819	budesonide	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
UNIPROT:Q9BYF1	hgnc:13557	ACE2	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	GL1001	iuphar.ligand:7866	MLN-4760	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.3271505995993426	Tapentadol hydrochloride	rxcui:857492	TAPENTADOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:9811	iuphar.ligand:9811	GSK-3&BETA; INHIBITOR 3 [PMID: 25845281]	FALSE	FALSE	FALSE
NCBIGENE:255	hgnc:12373	TSHR	GuideToPharmacology	2024.1	agonist	0.9309870786470656	IUPHAR.LIGAND:3920	rxcui:4952	THYROTROPIN ALFA	TRUE	FALSE	FALSE
UNIPROT:Q09428	hgnc:59	ABCC8	TdgClinicalTrial	Jan-14	NULL	0.9845188356692718	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-2260	chembl:CHEMBL601351	CHEMBL:CHEMBL601351	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.023813003	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
CTSG	hgnc:2532	CTSG	NCI	14-Sep-17	NULL	2.187819634820604	MANNITOL	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.2287915957982331	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.013022736	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
UNIPROT:O76082	hgnc:10969	SLC22A5	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.150021918	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.026045472	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	blocker	0.4605936073306534	IUPHAR.LIGAND:2291	iuphar.ligand:2291	PICROTOXININ	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4018	iuphar.ligand:4018	AC262970	FALSE	FALSE	FALSE
UNIPROT:O14672	hgnc:188	ADAM10	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	INCB7839	drugbank:DB05033	INCB7839	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	PIDILIZUMAB	ncit:C71014	PIDILIZUMAB	FALSE	TRUE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00393537	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.027347745	DIHYDROERGOTAMINE	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	modulator	0.1389091831632129	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	INO-8875	chembl:CHEMBL3545407	TRABODENOSON	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.064111931	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.059397818	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.1495945049449985	IUPHAR.LIGAND:7147	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:11418	iuphar.ligand:11418	[125I]SPEXIN-1	FALSE	FALSE	FALSE
UNIPROT:P14778	hgnc:5993	IL1R1	TdgClinicalTrial	Jan-14	NULL	1.570742301922485	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
POLE3	hgnc:13546	POLE3	ChEMBL	33	inhibitor	0.2573905452730122	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:9389	iuphar.ligand:9389	SB590885	FALSE	FALSE	FALSE
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	8.751278539282415	GSK1482160	iuphar.ligand:10504	GSK1482160	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1666910197958555	ROPINIROLE	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:682	iuphar.ligand:682	&BETA;-CGRP	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9465	iuphar.ligand:9465	[3H]-ALMOREXANT	FALSE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.1029562181092048	ROPINIROLE	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1084869240406911	lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TdgClinicalTrial	Jan-14	NULL	0.201178817	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P28482	hgnc:6871	MAPK1	TdgClinicalTrial	Jan-14	NULL	0.042863405	RDEA119	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.091796628	DULOXETINE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.055504938	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:5243	iuphar.ligand:5243	PF3845	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.596678082	LICARBAZEPINE	ncit:C81475	LICARBAZEPINE	FALSE	FALSE	FALSE
S1PR5	hgnc:14299	S1PR5	ChEMBL	33	binder	2.625383561784725	FINGOLIMOD LAURYL SULFATE	rxcui:2610292	FINGOLIMOD LAURYL SULFATE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	GNF-PF-4945	chembl:CHEMBL585628	CHEMBL:CHEMBL585628	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	LIPOTECAN	drugbank:DB17385	LIPOTECAN	FALSE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	NCI	14-Sep-17	NULL	1.887530665335423	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.2408608772279564	SUFENTANIL	rxcui:56795	SUFENTANIL	TRUE	FALSE	FALSE
UNIPROT:Q99250	hgnc:10588	SCN2A	TdgClinicalTrial	Jan-14	NULL	0.052090944	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	LURASIDONE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TEND	1-Aug-11	NULL	4.039051633514961	FILGRASTIM	rxcui:1433764	TBO-FILGRASTIM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.7160136986685613	TIAPROFENIC ACID	rxcui:38253	TIAPROFENIC ACID	FALSE	FALSE	FALSE
UNIPROT:P51788	hgnc:2020	CLCN2	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	OGX-011	ncit:C1055	CUSTIRSEN SODIUM	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CID 1540545	chembl:CHEMBL259784	CHEMBL:CHEMBL259784	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2917092846427472	BENZOFURAN	drugbank:DB04179	BENZOFURAN	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.087222045	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.016083624	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ARSA	hgnc:713	ARSA	PharmGKB	4/5/24	NULL	0.095122593	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003740928	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	OCRELIZUMAB	rxcui:1876366	OCRELIZUMAB	TRUE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.055504938	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	MECHLORETHAMINE HYDROCHLORIDE	rxcui:155036	MECHLORETHAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.187193124	clodronate	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
INTERLEUKIN-10	hgnc:5962	IL10	TTD	2020.06.01	NULL	0.6563458904461812	AM0010	ncit:C113295	PEGILODECAKIN	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.027347745	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.546954909	OTELIXIZUMAB	ncit:C95790	OTELIXIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:860	iuphar.ligand:860	CCK-33	FALSE	FALSE	FALSE
NCBIGENE:2929	ncbigene:2929	GSK1	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:9483	iuphar.ligand:9483	GLCC14C18	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.022606632	RISPERDAL	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	1.544343271638073	YM443	ncit:C72222	ACOTIAMIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
UNIPROT:P43405	hgnc:11491	SYK	TdgClinicalTrial	Jan-14	NULL	0.750109589	PRT062607	iuphar.ligand:8070	P505-15	FALSE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	PharmGKB	4/5/24	NULL	0.3409589041278864	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
UNIPROT:P29459	hgnc:5969	IL12A	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	DC-RTS-IL-12	ncit:C101789	ADENOVIRAL TRANSDUCED HIL-12-EXPRESSING AUTOLOGOUS DENDRITIC CELLS INXN-3001 PLUS ACTIVATOR LIGAND INXN-1001	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1215455352678113	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.3314878234576672	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
TLR7	hgnc:15631	TLR7	ChEMBL	33	agonist	2.625383561784724	GSK-2245035	chembl:CHEMBL4297492	GSK-2245035	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:9212	iuphar.ligand:9212	RAPALINK-1	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.1406455479527531	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.2302968036653267	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.090608578	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
UNIPROT:P49146	hgnc:7957	NPY2R	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	PYY3-36	drugbank:DB05004	PEPTIDE YY (3-36)	FALSE	FALSE	FALSE
NCBIGENE:2789	hgnc:4409	GNG5P1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10051	iuphar.ligand:10051	AMINOPYRIDINE 2	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.4688184931758437	Afuresertib	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.057574201	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124003	chembl:CHEMBL535730	CHEMBL:CHEMBL535730	FALSE	FALSE	FALSE
UNIPROT:P50391	hgnc:9329	NPY4R	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	PYY3-36	drugbank:DB05004	PEPTIDE YY (3-36)	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2660861718025059	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.3302369260106572	EOTAXIN	ncit:C1531	RECOMBINANT EOTAXIN	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.018031481	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
UNIPROT:Q16665	hgnc:4910	HIF1A	TdgClinicalTrial	Jan-14	NULL	1.086365611772989	PX-478	drugbank:DB06082	PX-478	FALSE	FALSE	TRUE
NCBIGENE:1620	hgnc:2687	BRINP1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8635	iuphar.ligand:8635	CASP 4 INHIB	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.2251615404618117	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
FAAH	hgnc:3553	FAAH	ChEMBL	33	inhibitor	5.250767123569449	JNJ-42165279	drugbank:DB15173	JNJ-42165279	FALSE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	1.117184494376478	RALTITREXED	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
NCBIGENE:2066	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:8064	iuphar.ligand:8064	BIX02188	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.030598876	IUPHAR.LIGAND:2566	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
DDX43	hgnc:18677	DDX43	CIViC	10-Apr-24	NULL	0.5303805175322677	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	TRICLOSAN	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.066241806	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	OZARELIX	ncit:C95214	OZARELIX	FALSE	FALSE	FALSE
GGH	hgnc:4248	GGH	PharmGKB	4/5/24	NULL	0.5707355569097228	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1595977849109255	BETHANECHOL	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	4.200613699	Andecaliximab	ncit:C105803	ANDECALIXIMAB	FALSE	FALSE	FALSE
NCBIGENE:1385	hgnc:2345	CREB1	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:10079	iuphar.ligand:10079	5-LOX INHIBITOR 2M [PMID: 30199704]	FALSE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.3621218705909965	SNX-5422	drugbank:DB06070	SNX-5422	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.048083948	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02804897	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	1.640864726115453	USTEKINUMAB	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
UNIPROT:O14920	hgnc:5960	IKBKB	TdgClinicalTrial	Jan-14	NULL	0.1136529680426287	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	ChEMBL	33	inhibitor	6.563458904461812	BRIOBACEPT	ncit:C97707	BRIOBACEPT	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.092118721	SOLIFENACIN	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
PSCA	hgnc:9500	PSCA	ChEMBL	33	inhibitor	13.12691780892362	MK-4721	drugbank:DB05933	MK-4721	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	GNF-PF-516	chembl:CHEMBL602970	CHEMBL:CHEMBL602970	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.034888818	IUPHAR.LIGAND:7177	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.086361301	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	1.300189954407673	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	DIETHYLPROPION HYDROCHLORIDE	rxcui:81998	DIETHYLPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TdgClinicalTrial	Jan-14	NULL	1.060761035064535	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	ChEMBL	33	inhibitor	0.729273212	AME-133V	chembl:CHEMBL2109346	AME-133V	FALSE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.089756703	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	TICAGRELOR	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
CBS	hgnc:1550	CBS	PharmGKB	4/5/24	NULL	2.100306849	betaine	rxcui:1512	BETAINE	TRUE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:9625	iuphar.ligand:9625	ROVAZOLAC	FALSE	FALSE	FALSE
UNIPROT:P43088	hgnc:9600	PTGFR	TdgClinicalTrial	Jan-14	NULL	15.00219178	TRAVOPROST	rxcui:283809	TRAVOPROST	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.6848826682916673	UPADACITINIB	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
UNIPROT:P17813	hgnc:3349	ENG	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	TRC105	ncit:C74010	CAROTUXIMAB	FALSE	FALSE	FALSE
CYSLTR1	hgnc:17451	CYSLTR1	ChEMBL	33	inhibitor	7.955707762984016	PRANLUKAST	ncit:C96712	PRANLUKAST	FALSE	FALSE	FALSE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.095122593	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:10751	iuphar.ligand:10751	(R)-16 [PMID: 32267688]	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:5829	iuphar.ligand:5829	METHIONINE BENZIMIDAZOLE 6	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1262	iuphar.ligand:1262	JB 98064	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.025298806	ketoprofen	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.070322774	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
PROTEIN KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	0.2187819634820604	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1041818873724097	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	1.555782851427985	Acetyldigitoxin	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
UNIPROT:Q96RI0	hgnc:3540	F2RL3	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	VORAPAXAR	rxcui:1537034	VORAPAXAR	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	CIViC	10-Apr-24	NULL	0.1591141552596802	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.049442252	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	1.790034246671403	ARBUTAMINE	rxcui:61609	ARBUTAMINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001244081	ESTRADIOL ACETATE	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:9563	ncit:C125471	EGANELISIB	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.021846337	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	antibody	0.7955707762984014	IUPHAR.LIGAND:8921	iuphar.ligand:8921	PLOZALIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.066297565	IUPHAR.LIGAND:1015	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5774	iuphar.ligand:5774	GSK 256471	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9337	iuphar.ligand:9337	COMPOUND 3 [PMID: 27347366]	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.1434635826111871	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	1.666910197958555	AMINOCAPROIC ACID	rxcui:99	6-AMINOCAPROIC ACID	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.6789785073581185	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
UNIPROT:P63316	hgnc:11943	TNNC1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:P09884	hgnc:9173	POLA1	TdgClinicalTrial	Jan-14	NULL	0.5791287268642776	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.019695301	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.054695491	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:10524	iuphar.ligand:10524	MW150	FALSE	FALSE	FALSE
UNIPROT:P12319	hgnc:3609	FCER1A	TdgClinicalTrial	Jan-14	NULL	3.750547945	BENZYLPENICILLOYL POLYLYSINE	rxcui:19079	BENZYLPENICILLOYL POLYLYSINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	NCI	14-Sep-17	NULL	0.009651258	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.061412481	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P30273	hgnc:3611	FCER1G	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	BENZYLPENICILLOYL POLYLYSINE	rxcui:19079	BENZYLPENICILLOYL POLYLYSINE	TRUE	FALSE	FALSE
ULK3	hgnc:19703	ULK3	PharmGKB	4/5/24	NULL	0.7001022831425933	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	0.4339476961627644	ketoconazole	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	TRIFLUPERIDOL	rxcui:10804	TRIFLUPERIDOL	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.008496387	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
UNIPROT:P35408	hgnc:9596	PTGER4	TEND	1-Aug-11	NULL	0.7721716358190367	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:Q9H2X9	hgnc:13818	SLC12A5	TdgClinicalTrial	Jan-14	NULL	5.834185692854945	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
GRM2	hgnc:4594	GRM2	ChEMBL	33	agonist	1.875273972703375	POMAGLUMETAD METHIONIL	ncit:C170541	POMAGLUMETAD METHIONIL	FALSE	FALSE	FALSE
UNIPROT:P33765	hgnc:268	ADORA3	TdgClinicalTrial	Jan-14	NULL	1.973972602845657	CF-101	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	1.491695205559502	CARTEOLOL	rxcui:2116	CARTEOLOL	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1392776425349986	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:8628	iuphar.ligand:8628	COMPOUND 4 [PMID: 12408711]	FALSE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	0.7955707762984016	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	0.1930429089547592	ADENOSINE TRIPHOSPHATE	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.012213217	thioridazine	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.4375639269641209	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
ATP7A	hgnc:869	ATP7A	NCI	14-Sep-17	NULL	0.1325951293830669	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.026680727	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.013411921	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CID 670282	chembl:CHEMBL260213	CHEMBL:CHEMBL260213	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	2.282942227638891	BRUCEANTIN	ncit:C1025	BRUCEANTIN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DoCM	10-Apr-24	NULL	0.8643238063488805	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	DIPHENYLPYRALINE	rxcui:23386	DIPHENYLPYRALINE	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.1842374429322614	DAROTROPIUM BROMIDE	ncit:C76000	DAROTROPIUM BROMIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	DAPSONE	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1367387271762877	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
UMPS	hgnc:12563	UMPS	DTC	9/2/20	NULL	26.25383561784724	5-FLUORO-6-AMIDO-UMP	chembl:CHEMBL1164954	CHEMBL:CHEMBL1164954	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	1-AMINOBENZOTRIAZOLE	chembl:CHEMBL101168	CHEMBL:CHEMBL101168	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.068637479	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	blocker	0.212581665	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	activator	0.2983390411119005	IUPHAR.LIGAND:7443	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1041818873724097	LY3023414	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.073540156	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P42701	hgnc:5971	IL12RB1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	ETHYNODIOL DIACETATE	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
UNIPROT:P20273	hgnc:1643	CD22	TEND	1-Aug-11	NULL	8.751278539282417	OSPA LIPOPROTEIN	rxcui:54214	OSPA PROTEIN	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.047886613	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.056097939	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1909369863116163	FENOPROFEN	rxcui:4331	FENOPROFEN	TRUE	FALSE	FALSE
UNIPROT:Q13698	hgnc:1397	CACNA1S	TdgClinicalTrial	Jan-14	NULL	0.099071078	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:Q7Z2W7	hgnc:17961	TRPM8	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	D3263	ncit:C162345	TRPM8 AGONIST D-3263	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.047219129	IUPHAR.LIGAND:7461	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.067883221	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	antibody	1.381780822	IUPHAR.LIGAND:8930	iuphar.ligand:8930	ISTIRATUMAB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.048260727	IUPHAR.LIGAND:9916	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	TEGASEROD MALEATE	rxcui:339270	TEGASEROD MALEATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	DIPHYLLIN	chembl:CHEMBL221190	DIPHYLLIN	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	PharmGKB	4/5/24	NULL	0.087077398	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	OXYBUPROCAINE	rxcui:18889	BENOXINATE	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.1389091831632129	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.801643836	REL-BENDIGOLE D	chembl:CHEMBL1915269	CHEMBL:CHEMBL1915269	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	PharmGKB	4/5/24	NULL	0.2447910080918158	pamidronate	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.093763699	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:3303	iuphar.ligand:3303	L745870	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.069180068	IUPHAR.LIGAND:9513	iuphar.ligand:9513	MLKL COMPOUND 1	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:9294	iuphar.ligand:9294	BU08028	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:8827	iuphar.ligand:8827	COMPOUND 11J [PMID: 23021994]	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.076098074	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2713574740862764	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.2045753424767318	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1785975212098452	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
FN1	hgnc:3778	FN1	ChEMBL	33	cleavage	0.212581665	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	PROCYCLIDINE	rxcui:8718	PROCYCLIDINE	TRUE	FALSE	FALSE
UNIPROT:P16422	hgnc:11529	EPCAM	TdgClinicalTrial	Jan-14	NULL	4.200613699	ADECATUMUMAB	ncit:C82358	ADECATUMUMAB	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.050781113	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.1060761035064535	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.019318496	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.064505739	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	NCI	14-Sep-17	NULL	0.036212187	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.01689436	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.074690855	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.7395446652914718	5-METHOXYCANTHINONE	chembl:CHEMBL508649	5-METHOXYCANTHINONE	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2393966773663883	PROPANTHELINE	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	ChEMBL	33	inhibitor	2.100306849	NAMILUMAB	ncit:C97943	NAMILUMAB	FALSE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.085032666	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P32754	hgnc:5147	HPD	TdgClinicalTrial	Jan-14	NULL	70.01022831425932	NITISINONE	rxcui:61805	NITISINONE	TRUE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.020010545	IUPHAR.LIGAND:5661	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.099446347	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.101562227	SUCCINYLCHOLINE	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
NADPH OXIDASE 4	hgnc:7891	NOX4	TTD	2020.06.01	NULL	78.76150685354175	GKT-137831	ncit:C166721	SETANAXIB	FALSE	FALSE	FALSE
UNIPROT:P29275	hgnc:264	ADORA2B	TEND	1-Aug-11	NULL	0.3241214273808303	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.2397610558707511	NSC-319994	chembl:CHEMBL1329443	CHEMBL:CHEMBL1329443	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	SEIMATOPOLIDE A	chembl:CHEMBL2036277	SEIMATOPOLIDE A	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.030386384	ketorolac	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	CIViC	10-Apr-24	NULL	0.076934317	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.8204323630577265	O6-BENZYLGUANINE	ncit:C1306	O6-BENZYLGUANINE	FALSE	FALSE	FALSE
VAV1	hgnc:12657	VAV1	NCI	14-Sep-17	NULL	1.029562181092049	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.004037499	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	modulator	0.6177373086552295	IUPHAR.LIGAND:10908	iuphar.ligand:10908	BAY1125976	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.010277485	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.058212496	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.8643238063488805	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	IMIDAZOLE-4-ACETIC ACID HCL	chembl:CHEMBL1256325	CHEMBL:CHEMBL1256325	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:12469	iuphar.ligand:12469	BENGALENSOL	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:309	iuphar.ligand:309	OTENZEPAD	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	N-DESMETHYLCLOZAPINE	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
HIST3H2A	hgnc:20507	H2AC25	NCI	14-Sep-17	NULL	1.050153425	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1193356164447602	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TEND	1-Aug-11	NULL	0.4412409347537352	MECLOFENAMIC ACID	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.3409589041278864	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.4375639269641208	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	ChEMBL	33	inhibitor	1.093909817410302	AVAGACESTAT	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.2344092465879218	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.8899605294185507	ALISERTIB SODIUM	ncit:C142912	ALISERTIB SODIUM	FALSE	FALSE	TRUE
NCBIGENE:1821	hgnc:3032	DRP2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8124	iuphar.ligand:8124	COMPOUND 20 [PMID: 23489211]	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	modulator	0.5707355569097228	IUPHAR.LIGAND:8098	ncit:C74080	TASQUINIMOD	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.032134438	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:10281	iuphar.ligand:10281	PYRAZOLOPYRIMIDINE 4N	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	AZ628	iuphar.ligand:8475	AZ628	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.06714536	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.1691068316769549	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
RUNX3	hgnc:10473	RUNX3	NCI	14-Sep-17	NULL	0.8334550989792777	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.9546849315580818	valdecoxib	rxcui:278567	VALDECOXIB	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	CID 1540951	chembl:CHEMBL259421	CHEMBL:CHEMBL259421	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.4039051633514962	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.023620185	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.8643238063488805	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:3932	iuphar.ligand:3932	L-748337	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:3932	iuphar.ligand:3932	L-748337	FALSE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:10519	iuphar.ligand:10519	NF-56-EJ40	FALSE	FALSE	FALSE
UNIPROT:P51788	hgnc:2020	CLCN2	TEND	1-Aug-11	NULL	35.00511415712966	LUBIPROSTONE	rxcui:623033	LUBIPROSTONE	TRUE	FALSE	FALSE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	3.750547945	plazomicin	rxcui:2049549	PLAZOMICIN	TRUE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.039778539	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.0287871	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	2-MERCAPTONICOTINIC ACID	chembl:CHEMBL1521174	2-MERCAPTONICOTINIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	CI-218872	chembl:CHEMBL13662	CI-218872	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.061919424	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.6105543166941221	APRACLONIDINE	rxcui:14845	APRACLONIDINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.3251536612259921	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7720	iuphar.ligand:7720	ML218	FALSE	FALSE	FALSE
UNIPROT:P32927	hgnc:2436	CSF2RB	TEND	1-Aug-11	NULL	13.12691780892362	SARGRAMOSTIM	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:3274	iuphar.ligand:3274	VU0255035	FALSE	FALSE	FALSE
NCBIGENE:2240	hgnc:11732	TESK2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8118	iuphar.ligand:8118	COMPOUND 30 [PMID: 22902653]	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.003198567	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.8899605294185507	tipiracil hydrochloride	rxcui:1670303	TIPIRACIL HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.016603216	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.2059124362184098	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
UNIPROT:Q8TDV5	hgnc:19060	GPR119	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	APD668	drugbank:DB05166	APD668	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:309	iuphar.ligand:309	OTENZEPAD	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1364544470782081	Taselisib	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	CIViC	10-Apr-24	NULL	0.2069267831948551	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	LICOAGRODIN	chembl:CHEMBL2437368	LICOAGRODIN	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.5834185692854944	GNF-PF-4068	chembl:CHEMBL584668	CHEMBL:CHEMBL584668	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	ISOCONAZOLE	rxcui:27901	ISOCONAZOLE	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.096167896	GW468816	chembl:CHEMBL1207366	GW468816	FALSE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	ChEMBL	33	blocker	0.075010959	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	blocker	0.1187956362798518	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	0.750109589	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.3454452054979901	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SJ000119988	chembl:CHEMBL589694	CHEMBL:CHEMBL589694	FALSE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	TALC	12-May-16	antibody	1.260184109656668	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.023284998	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.035145697	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.085239726	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
CRTC1	hgnc:16062	CRTC1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2678962818147678	NVP-BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.016342257	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	0.6563458904461812	IUPHAR.LIGAND:2314	iuphar.ligand:2314	EBIO	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	BUPRANOLOL	rxcui:1817	BUPRANOLOL	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	RS-67506	iuphar.ligand:3230	RS67506	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.1141471113819445	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UCP2	hgnc:12518	UCP2	NCI	14-Sep-17	NULL	17.50255707856483	BRL49653	ncit:C2583	ROSIGLITAZONE MALEATE	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	PharmGKB	4/5/24	NULL	0.036087747	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
RPS6KA5	hgnc:10434	RPS6KA5	DTC	9/2/20	NULL	0.1136529680426288	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	GNF-PF-3832	chembl:CHEMBL261693	CHEMBL:CHEMBL261693	FALSE	FALSE	FALSE
SLC26A9	hgnc:14469	SLC26A9	PharmGKB	4/5/24	NULL	26.25383561784724	ivacaftor	rxcui:1243041	IVACAFTOR	TRUE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	agonist	1.400204566285186	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003174779	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:Q9NYX4	hgnc:17938	CALY	TEND	1-Aug-11	NULL	0.9723642821424907	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.057197899	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.037213091	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.1346350544504987	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.034318739	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.011517366	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:4083	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:2937	iuphar.ligand:2937	AFD(R)	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.011715232	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
AGAP3	hgnc:16923	AGAP3	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PTGIR	hgnc:9602	PTGIR	PharmGKB	4/5/24	NULL	0.053199262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
RPA1	hgnc:10289	RPA1	DTC	9/2/20	NULL	105.0153424713889	NSC-15520	chembl:CHEMBL1765371	CHEMBL:CHEMBL1765371	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	CIViC	10-Apr-24	NULL	0.013890918	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
DAGLB	hgnc:28923	DAGLB	DTC	9/2/20	NULL	8.078103267029924	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.032055965	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.062262061	MESORIDAZINE	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.1988926940746003	Abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
TOP1MT	hgnc:29787	TOP1MT	ChEMBL	33	inhibitor	0.84012274	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2035181055647073	AZD1305	chembl:CHEMBL3545169	AZD1305	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.056826484	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.1666910197958555	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
LPA	hgnc:6667	LPA	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P26439	hgnc:5218	HSD3B2	TEND	1-Aug-11	NULL	13.12691780892362	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:11193	iuphar.ligand:11193	ZYBT1	FALSE	FALSE	FALSE
UNIPROT:P08185	hgnc:1540	SERPINA6	TEND	1-Aug-11	NULL	0.546954909	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
NCBIGENE:544	hgnc:881	ALDH7A1P4	GuideToPharmacology	2024.1	blocker	0.4039051633514962	IUPHAR.LIGAND:2566	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CancerCommons	25-Jul-13	inhibitor	0.364636606	ASP3026	ncit:C116727	ALK INHIBITOR ASP3026	FALSE	FALSE	TRUE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.09741683	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.096050618	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2100	iuphar.ligand:2100	SUBSTANCE P-(6-11)	FALSE	FALSE	FALSE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8395	iuphar.ligand:8395	DS-437	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	1.346350544504987	BETHANECHOL CHLORIDE	rxcui:47088	BETHANECHOL CHLORIDE	TRUE	FALSE	FALSE
HAVCR2	hgnc:18437	HAVCR2	CIViC	10-Apr-24	NULL	8.751278539282415	ANTI-TIM-3 MONOCLONAL ANTIBODY	ncit:C141146	ANTI-TIM-3 MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	1.944728564284981	Iodine-131-tositumomab	rxcui:234449	IODINE-131-TOSITUMOMAB	TRUE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	ChEMBL	33	inhibitor	3.141484604	ANAKINRA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.3561566847382379	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
KCND3	hgnc:6239	KCND3	ChEMBL	33	blocker	0.1312691780892362	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
UNIPROT:O75899	hgnc:4507	GABBR2	TEND	1-Aug-11	NULL	1.750255707856483	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
DLL4	hgnc:2910	DLL4	ChEMBL	33	inhibitor	4.200613698855561	ENOTICUMAB	ncit:C82367	ENOTICUMAB	FALSE	FALSE	TRUE
CXCL10	hgnc:10637	CXCL10	ChEMBL	33	inhibitor	3.088686543276147	ELDELUMAB	ncit:C166466	ELDELUMAB	FALSE	FALSE	FALSE
UNIPROT:Q8N8R3	hgnc:20116	SLC25A29	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.175610941	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.052350619	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.014683353	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:2593	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.00767656	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	2.493675356344019	LORLATINIB	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.2778183663264258	PIRFENIDONE	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	PLICAMYCIN	rxcui:6995	PLICAMYCIN	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2035181055647073	ISOETHARINE MESYLATE	rxcui:6024	ISOETHARINE MESYLATE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	1.166837138570988	AICAR	drugbank:DB01700	AICA RIBONUCLEOTIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	CANDIDIN	chembl:CHEMBL454843	CANDIDIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006324701	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	2.187819634820604	Trimethadione	rxcui:10827	TRIMETHADIONE	TRUE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	agonist	0.7778914257139926	ETRASIMOD	rxcui:2668045	ETRASIMOD	TRUE	FALSE	FALSE
IL4	hgnc:6014	IL4	ChEMBL	33	inhibitor	5.250767123569449	ROMILKIMAB	ncit:C174791	ROMILKIMAB	FALSE	FALSE	FALSE
UNIPROT:Q01668	hgnc:1391	CACNA1D	TdgClinicalTrial	Jan-14	NULL	0.1436598392221464	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.099446347	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
NCBIGENE:2348	hgnc:3791	FOLR1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10714	ncit:C76907	ALOXISTATIN	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.061919424	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	CIViC	10-Apr-24	NULL	0.1646008502686348	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	0.5357925636295356	MEDI5117	iuphar.ligand:11552	ZILTIVEKIMAB	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.1141471113819445	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.032837818	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
SENP3	hgnc:17862	SENP3	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.092933931	permethrin	rxcui:33199	PERMETHRIN	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	FDA	10-Apr-24	NULL	0.4167275494896388	Avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.1058622403945453	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	2.500365296937833	Tenecteplase	rxcui:259280	TENECTEPLASE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004292999	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.096050618	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.024384367	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.1154014752432846	AZD7325	iuphar.ligand:7712	AZD7325	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:4028	iuphar.ligand:4028	LYSOPHOSPHATIDYLINOSITOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	PURVALANOLA	chembl:CHEMBL23327	PURVALANOLA	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	0.3547815624033412	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	DNDI1417260	chembl:CHEMBL2094573	CHEMBL:CHEMBL2094573	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001350506	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NCBIGENE:544	hgnc:881	ALDH7A1P4	GuideToPharmacology	2024.1	blocker	1.050153425	IUPHAR.LIGAND:2560	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9459	iuphar.ligand:9459	ML354	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	MyCancerGenome	20-Jun-17	inhibitor	0.2041114528112516	PD0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.1193356164447602	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
ODC1	hgnc:8109	ODC1	DTC	9/2/20	NULL	0.2592971419046642	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.043109746	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.049723174	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.2500365296937833	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.020994671	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.07699072	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:2719	hgnc:4451	GPC3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8732	iuphar.ligand:8732	COMPOUND 33 [PMID: 26230603]	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:3794	iuphar.ligand:3794	[125I]MOTILIN (HUMAN)	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.067883221	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.7095631248066824	PICLOZOTAN	ncit:C90944	PICLOZOTAN	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.08334551	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	PharmGKB	4/5/24	NULL	0.1205687054780585	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	TALC	12-May-16	inhibitor	0.1750255707856483	NMS1286937	ncit:C143162	ONVANSERTIB	FALSE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.03729238	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	2.187819634820604	BENZTHIAZIDE	rxcui:19008	BENZTHIAZIDE	TRUE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.5000730593875666	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.037693949	TETROQUINONE	chembl:CHEMBL1329029	TETROQUINONE	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.054355767	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V4	hgnc:18083	TRPV4	TTD	2020.06.01	NULL	3.889457128569962	GSK2798745	drugbank:DB16033	GSK2798745	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:8976	iuphar.ligand:8976	NS-398	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.03409589	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.046059361	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	3.454452054979901	Eplerenone	rxcui:298869	EPLERENONE	TRUE	FALSE	FALSE
TRAF3IP2	hgnc:1343	TRAF3IP2	PharmGKB	4/5/24	NULL	2.386712328895204	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	0.8423690572571311	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.012337329	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.5000730593875667	IUPHAR.LIGAND:4288	rxcui:8351	PIRACETAM	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.096167896	IUPHAR.LIGAND:7472	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.070197421	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	1.491695205559502	CARTEOLOL	rxcui:2116	CARTEOLOL	TRUE	FALSE	FALSE
NCBIGENE:938	hgnc:1649	CD24P4	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:4576	iuphar.ligand:4576	LP-403812	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.035982643	ENZALUTAMIDE	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	1.500219178	Nipradilol	ncit:C76555	NIPRADILOL	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.045265234	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.006002249	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1875273972703375	EQUILIN	ncit:C29020	EQUILIN	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.07182992	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.032899543	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.034590034	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.2134458180312784	IUPHAR.LIGAND:4366	iuphar.ligand:4366	[3H]CGS8216	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	modulator	3.500511415712966	IUPHAR.LIGAND:6216	iuphar.ligand:6216	AZ12216052	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.048083948	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.039778539	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	PharmGKB	4/5/24	NULL	0.3070624048871023	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013281873	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	1.693795846312725	ALCAFTADINE	rxcui:1000082	ALCAFTADINE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	BROMOPRIDE	rxcui:19768	BROMOPRIDE	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.079758488	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:2352	hgnc:3795	FOLR3	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:10746	iuphar.ligand:10746	VBY-825	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007699637	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	2.625383561784724	SP-54	chembl:CHEMBL1201516	PENTOSAN POLYSULFATE SODIUM	FALSE	FALSE	FALSE
TXN2	hgnc:17772	TXN2	DTC	9/2/20	NULL	3.889457128569963	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01715937	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.750109589	CETIRIZINE DIHYDROCHLORIDE	chembl:CHEMBL1607273	CETIRIZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
HBB	hgnc:4827	HBB	PharmGKB	4/5/24	NULL	0.9053046764774912	voxelotor	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.073540156	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TEND	1-Aug-11	NULL	0.8334550989792776	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:185	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
NCBIGENE:1758	hgnc:2932	DMP1	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:9690	iuphar.ligand:9690	COMPOUND 12P [LARSON ET AL., 2017]	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.1973972602845657	Adavosertib	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	ARQ 751	ncit:C128250	PAN-AKT INHIBITOR ARQ751	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.032412143	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.082364974	CA4P	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TPH1	hgnc:12008	TPH1	PharmGKB	4/5/24	NULL	0.3125456621172291	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.3542686252046857	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	1.250182648468916	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.022173848	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	1.250182648468916	CHLORTHALIDONE	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
GUANYLYL CYCLASE C	hgnc:4688	GUCY2C	TTD	2020.06.01	NULL	1.640864726115453	MLN0264	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.192335792	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	1-NAPHTHYLISOTHIOCYANATE	chembl:CHEMBL1381098	1-NAPHTHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.047070974	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	1.093909817410302	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	blocker	0.096167896	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	NSC-16211	chembl:CHEMBL1162521	CHEMBL:CHEMBL1162521	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	CGI	2/1/22	NULL	2.493675356344019	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.066297565	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.3472729579080324	Rociletinib	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	CGI	2/1/22	NULL	0.089103927	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CSF3R	hgnc:2439	CSF3R	CGI	2/1/22	NULL	0.1049104320393496	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1583941817064691	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	CHLORPHENIRAMINE POLISTIREX	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.072851434	INFLIXIMAB	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.028300937	FLUPHENAZINE HYDROCHLORIDE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	EMEDASTINE DIFUMARATE	rxcui:221094	EMEDASTINE DIFUMARATE	TRUE	FALSE	FALSE
CD33	hgnc:1659	CD33	ChEMBL	33	binder	2.423430980108977	GEMTUZUMAB OZOGAMICIN	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.4449802647092754	IRBESARTAN	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.2734774543525755	PHENYLPROPANOLAMINE POLISTIREX	chembl:CHEMBL1201535	PHENYLPROPANOLAMINE POLISTIREX	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.8899605294185507	EPROSARTAN MESYLATE	rxcui:236878	EPROSARTAN MESYLATE	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	0.7955707762984014	GONADORELIN HYDROCHLORIDE	rxcui:204194	GONADORELIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.096937239	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	ChEMBL	33	inhibitor	2.625383561784724	WARFARIN POTASSIUM	rxcui:82118	WARFARIN POTASSIUM	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	0.8334550989792776	HEPARIN SODIUM	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	0.8334550989792776	TINZAPARIN SODIUM	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.055740628	CALCIFEDIOL	rxcui:1855064	CALCIFEDIOL ANHYDROUS	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.080550887	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.077217164	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
REN	hgnc:9958	REN	ChEMBL	33	inhibitor	5.250767123569449	ALISKIREN FUMARATE	chembl:CHEMBL1667	ALISKIREN FUMARATE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.042898424	CYCLOBENZAPRINE HYDROCHLORIDE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.048172175	MEPERIDINE HYDROCHLORIDE	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	DIFENOXIN HYDROCHLORIDE	rxcui:235373	DIFENOXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.3006164383722967	DIFLUPREDNATE	rxcui:23043	DIFLUPREDNATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	MEDRYSONE	rxcui:29439	MEDRYSONE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.091796628	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
CYP11A1	hgnc:2590	CYP11A1	ChEMBL	33	inhibitor	1.944728564284981	MITOTANE	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.06525008	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.057260274	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	ACEPROMETAZINE	rxcui:161203	ACEPROMETAZINE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	ChEMBL	33	inhibitor	0.035502144	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.3889457128569962	ROFLUMILAST	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.1013661606866689	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.6674703970639131	DESERPIDINE	rxcui:62174	DESERPIDINE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.1769126389342806	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.1250182648468916	QUINESTROL	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.2243917574174979	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1962903597596056	QUINESTROL	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.08178765	DIETHYLSTILBESTROL DIPHOSPHATE	chembl:CHEMBL1200598	DIETHYLSTILBESTROL DIPHOSPHATE	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.041628703	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CA5A	hgnc:1377	CA5A	ChEMBL	33	inhibitor	1.750255707856483	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	CODEINE PHOSPHATE	rxcui:2672	CODEINE PHOSPHATE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.029170928	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.041672755	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.2692701089009974	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.1448487482363986	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.1693795846312726	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.1902451856365742	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UNIPROT:P08887	hgnc:6019	IL6R	TEND	1-Aug-11	NULL	4.039051633514961	TOCILIZUMAB	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
CALCR	hgnc:1440	CALCR	ChEMBL	33	agonist	1.640864726115453	PRAMLINTIDE ACETATE	rxcui:356773	PRAMLINTIDE ACETATE	TRUE	FALSE	FALSE
RAMP3	hgnc:9845	RAMP3	ChEMBL	33	agonist	4.375639269641208	PRAMLINTIDE ACETATE	rxcui:356773	PRAMLINTIDE ACETATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	DICLOFENAC POTASSIUM	rxcui:81997	DICLOFENAC POTASSIUM	TRUE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.280789686	ISOSORBIDE DINITRATE	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.2917092846427472	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	inhibitor	0.2763561643983921	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.089501712	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.2692701089009974	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.1419126249613365	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.2651902587661338	ISOSORBIDE DINITRATE	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.062139256	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TEND	1-Aug-11	NULL	0.06697407	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.6035364509849942	ACETOHEXAMIDE	rxcui:173	ACETOHEXAMIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.05853698	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.075442056	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
HPD	hgnc:5147	HPD	ChEMBL	33	inhibitor	70.01022831425932	NITISINONE	rxcui:61805	NITISINONE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.09969811	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	2.625383561784724	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	ChEMBL	33	inhibitor	32.81729452230906	BELIMUMAB	rxcui:1092437	BELIMUMAB	TRUE	TRUE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.1411496538593938	HYDROXYZINE	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
CD86	hgnc:1705	CD86	ChEMBL	33	inhibitor	3.500511415712966	ABATACEPT	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
LAMA1	hgnc:6481	LAMA1	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.098451884	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
COL15A1	hgnc:2192	COL15A1	ChEMBL	33	cleavage	0.2763561643983921	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.1535312024435511	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
COL6A5	hgnc:26674	COL6A5	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.6563458904461812	DESERPIDINE	rxcui:62174	DESERPIDINE	TRUE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	inhibitor	3.281729452230906	CLOPIDOGREL BISULFATE	rxcui:236991	CLOPIDOGREL BISULFATE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	negative modulator	0.096167896	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.1013661606866689	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.1118771404169627	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.9376369863516875	ESOMEPRAZOLE STRONTIUM	rxcui:1435522	ESOMEPRAZOLE STRONTIUM	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.054243462	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.3017682254924971	AFATINIB DIMALEATE	rxcui:1430441	AFATINIB DIMALEATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	OLODATEROL HYDROCHLORIDE	rxcui:1546396	OLODATEROL HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	0.3750547945406749	LEVETIRACETAM	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
PSMC6	hgnc:9553	PSMC6	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMD4	hgnc:9561	PSMD4	ChEMBL	33	inhibitor	0.192335792	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
UNIPROT:P10827	hgnc:11796	THRA	TEND	1-Aug-11	NULL	0.9092237443410304	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
SEM1	hgnc:10845	SEM1	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMB3	hgnc:9540	PSMB3	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TEND	1-Aug-11	NULL	0.4227670791923872	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	ChEMBL	33	inhibitor	0.4487835148349957	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
ADRM1	hgnc:15759	ADRM1	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.596678082	RG-7167	chembl:CHEMBL3545383	RG-7167	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TEND	1-Aug-11	NULL	0.6035364509849942	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	ChEMBL	33	inhibitor	0.4167275494896388	IRX4310	chembl:CHEMBL3545173	IRX4310	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.3125456621172291	RG-7167	chembl:CHEMBL3545383	RG-7167	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	inhibitor	0.801643836	CORT 108297	chembl:CHEMBL271220	CORT 108297	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.3241214273808302	MIRANSERTIB	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	1.166837138570988	AMG-900	drugbank:DB17197	AMG-900	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.364636606	AZD-7451	chembl:CHEMBL3545179	AZD-7451	FALSE	FALSE	FALSE
UNIPROT:P06746	hgnc:9174	POLB	TEND	1-Aug-11	NULL	0.007162904	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ARAF	hgnc:646	ARAF	ChEMBL	33	inhibitor	0.3818739726232327	TOVORAFENIB	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1363835616511545	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	positive modulator	2.282942227638891	AVL-3288	drugbank:DB18707	AVL-3288	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	2.561349816375341	MR-1817	chembl:CHEMBL3707397	MR-1817	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	positive modulator	0.596678082	PESAMPATOR	ncit:C186393	PESAMPATOR	FALSE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TEND	1-Aug-11	NULL	18.37768493249307	MENOTROPINS	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	positive modulator	0.3977853881492007	PESAMPATOR	ncit:C186393	PESAMPATOR	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	positive modulator	0.4234489615781814	PESAMPATOR	ncit:C186393	PESAMPATOR	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	1.875273972703375	AUS-131	chembl:CHEMBL198877	AUS-131	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	inhibitor	0.801643836	ORG-34517	drugbank:DB05423	ORG-34517	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.061340737	IDOXIFENE	ncit:C1406	IDOXIFENE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.111481255	BECOCALCIDIOL	ncit:C77083	BECOCALCIDIOL	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1121958787087489	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.034727296	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.061628722	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.0545251	MEGESTROL	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.050879526	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.056826484	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.151537291	MILCICLIB	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.2479701120930082	MILCICLIB	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.052090944	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	1.500219178	R-343	chembl:CHEMBL2170582	R-343	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.2375912725597036	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.030670369	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.1682938180631233	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
FRK	hgnc:3955	FRK	ChEMBL	33	inhibitor	0.1172046232939609	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.041021618	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
CHRM4	hgnc:1953	CHRM4	ChEMBL	33	inhibitor	0.3889457128569963	DAROTROPIUM BROMIDE	ncit:C76000	DAROTROPIUM BROMIDE	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1419126249613365	DAROTROPIUM BROMIDE	ncit:C76000	DAROTROPIUM BROMIDE	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	1.458546423213736	BAY1067197	chembl:CHEMBL3545405	BAY1067197	FALSE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TEND	1-Aug-11	NULL	0.2681242786503549	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
HTR6	hgnc:5301	HTR6	ChEMBL	33	inhibitor	7.001022831425932	PF-05212377	drugbank:DB16044	PF-05212377	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	agonist	1.944728564284981	KRP203	chembl:CHEMBL3545101	KRP203	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.2465148884304905	ODELEPRAN	chembl:CHEMBL2103878	ODELEPRAN	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	2.838252499226729	BVT.115959	chembl:CHEMBL3545409	BVT.115959	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1013661606866689	AFACIFENACIN	ncit:C90741	AFACIFENACIN	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	2.019525817	PRS-211375	chembl:CHEMBL3545290	PRS-211375	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.00598378	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.083744292	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.1058622403945453	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.252440727	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
KCNC1	hgnc:6233	KCNC1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNA6	hgnc:6225	KCNA6	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.021422958	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
KCNA7	hgnc:6226	KCNA7	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	ALEGLITAZAR	ncit:C72687	ALEGLITAZAR	FALSE	FALSE	FALSE
UNIPROT:P37088	hgnc:10599	SCNN1A	TEND	1-Aug-11	NULL	2.470949234620918	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.210030685	TESAGLITAZAR	ncit:C75985	TESAGLITAZAR	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.3125456621172291	ACOLBIFENE	ncit:C64183	ACOLBIFENE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	inhibitor	0.052507671	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.2333674277141978	VOLASERTIB	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.1201548540862574	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.2035181055647073	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	ChEMBL	33	inhibitor	0.8204323630577265	RUBOXISTAURIN	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.1591141552596802	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	1.093909817410302	ALBINTERFERON ALFA-2B	ncit:C87296	ALBINTERFERON ALFA-2B	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	negative modulator	0.2885036881082115	ESKETAMINE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	negative modulator	0.108711535	ESKETAMINE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	negative modulator	0.1209854175937661	ESKETAMINE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	GOSOGLIPTIN	ncit:C90616	GOSOGLIPTIN	FALSE	FALSE	FALSE
TTR	hgnc:12405	TTR	ChEMBL	33	modulator	17.50255707856483	TAFAMIDIS	rxcui:1545063	TAFAMIDIS	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	0.3125456621172291	REPAGLINIDE	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
CYP26A1	hgnc:2603	CYP26A1	ChEMBL	33	inhibitor	15.75230137070834	TALAROZOLE	ncit:C90792	TALAROZOLE	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.2430910705356227	TAMSULOSIN	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.2536602475154323	TAMSULOSIN	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TLR4	hgnc:11850	TLR4	ChEMBL	33	inhibitor	1.141471113819445	ERITORAN TETRASODIUM	ncit:C91759	ERITORAN TETRASODIUM	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.03049226	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.05814803	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.030868707	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	ChEMBL	33	cleavage	8.751278539282415	PRABOTULINUMTOXIN A	chembl:CHEMBL4297229	PRABOTULINUMTOXIN A	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	1.779921058837101	TASOSARTAN	ncit:C152517	TASOSARTAN	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	ChEMBL	33	inhibitor	1.009762908	RO-6870810	drugbank:DB15151	RO-6870810	FALSE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TEND	1-Aug-11	NULL	0.1620607136904151	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	ChEMBL	33	inhibitor	0.596678082	RO-6870810	drugbank:DB15151	RO-6870810	FALSE	FALSE	FALSE
BRDT	hgnc:1105	BRDT	ChEMBL	33	inhibitor	0.9376369863516875	RO-6870810	drugbank:DB15151	RO-6870810	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.1715936968486748	PF-06651600	chembl:CHEMBL4085457	PF-06651600	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.049723174	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
TXK	hgnc:12434	TXK	ChEMBL	33	inhibitor	4.375639269641208	PF-06651600	chembl:CHEMBL4085457	PF-06651600	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	inhibitor	0.031254566	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TEND	1-Aug-11	NULL	0.1215455352678113	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
HBB	hgnc:4827	HBB	ChEMBL	33	positive modulator	0.9053046764774912	VOXELOTOR	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.020836377	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.024354207	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	2.100306849	DUTOGLIPTIN	ncit:C87492	DUTOGLIPTIN	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	1.544343271638073	ACOTIAMIDE HYDROCHLORIDE	ncit:C72222	ACOTIAMIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	BAMBUTEROL	rxcui:18751	BAMBUTEROL	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.1458546423213736	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.093098708	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	1.640864726115453	PAZUFLOXACIN	ncit:C66331	PAZUFLOXACIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	2.187819634820604	CALCIUM OXYBATE	rxcui:2387307	CALCIUM OXYBATE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1132444383228493	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
GHR	hgnc:4263	GHR	ChEMBL	33	agonist	5.250767123569449	SOMAPACITAN	rxcui:2557373	SOMAPACITAN	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.099071078	NITRENDIPINE	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
UNIPROT:Q9GZZ6	hgnc:13800	CHRNA10	TEND	1-Aug-11	NULL	10.50153424713889	TRIMETHAPHAN	rxcui:10828	TRIMETHAPHAN	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2234368988752957	NILVADIPINE	rxcui:53692	NILVADIPINE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1383601350084176	ITOPRIDE	ncit:C65991	ITOPRIDE	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	ChEMBL	33	binder	0.3559842117674203	BINTRAFUSP ALFA	ncit:C124229	BINTRAFUSP ALFA	FALSE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TEND	1-Aug-11	NULL	0.082429625	VINORELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TLR9	hgnc:15633	TLR9	ChEMBL	33	agonist	4.633029815	LEFITOLIMOD	ncit:C94207	LEFITOLIMOD	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	MAVELERTINIB	ncit:C120307	MAVELERTINIB	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.4268916360625568	CADONILIMAB	ncit:C153379	CADONILIMAB	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.5147810905460244	ITOPRIDE	ncit:C65991	ITOPRIDE	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.4468737977505915	CYTISINICLINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.5081387538938177	BREPOCITINIB	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	0.105015342	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
CCR1	hgnc:1602	CCR1	ChEMBL	33	inhibitor	11.66837138570988	BMS-817399	drugbank:DB14941	BMS-817399	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.3500511415712967	Arverapamil	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
CD37	hgnc:1666	CD37	ChEMBL	33	inhibitor	35.00511415712966	BI-836826	drugbank:DB17322	BI-836826	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	ChEMBL	33	inhibitor	0.8078103267029924	PELABRESIB	ncit:C188265	PELABRESIB	FALSE	FALSE	FALSE
TACR3	hgnc:11528	TACR3	ChEMBL	33	inhibitor	2.917092846427472	FEZOLINETANT	rxcui:2637134	FEZOLINETANT	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	ChEMBL	33	inhibitor	0.1190650141398968	TILAVONEMAB	ncit:C174727	TILAVONEMAB	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	ChEMBL	33	inhibitor	1.312691780892362	SIREMADLIN	ncit:C116325	SIREMADLIN	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.9158314750411831	BEMARITUZUMAB	ncit:C120040	BEMARITUZUMAB	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	2.100306849	AMELPARIB DIHYDROCHLORIDE DIHYDRATE	chembl:CHEMBL4298003	AMELPARIB DIHYDROCHLORIDE DIHYDRATE	FALSE	FALSE	FALSE
CSF2RB	hgnc:2436	CSF2RB	ChEMBL	33	agonist	2.187819634820604	CIBINETIDE	ncit:C171683	CIBINETIDE	FALSE	FALSE	FALSE
LOXL2	hgnc:6666	LOXL2	ChEMBL	33	inhibitor	26.25383561784724	PAT-1251	drugbank:DB16735	PAT-1251	FALSE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	blocker	0.2243917574174979	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
MMP12	hgnc:7158	MMP12	ChEMBL	33	inhibitor	0.8334550989792776	CTS-1027	drugbank:DB08490	CTS-1027	FALSE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	blocker	0.1187956362798518	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.063110182	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	blocker	0.2019525816757481	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.8751278539282416	EDOTECARIN	ncit:C2665	EDOTECARIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CRTC2	hgnc:27301	CRTC2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2678962818147678	NVP-BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1805819381121768	AKOS004227608	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
FLT4	hgnc:3767	FLT4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.060492709	ENMD 2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1894216134043813	BCP9000383	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	1.129197231	AVX-470	drugbank:DB18455	AVX-470	FALSE	FALSE	FALSE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.099220845	NVP-BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.034018575	NVP-BEZ240	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.075768645	BCP9000383	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
P-SELECTIN GLYCOPROTEIN LIGAND 1	hgnc:10722	SELPLG	TTD	2020.06.01	NULL	52.50767123569449	Neihulizumab	ncit:C121711	NEIHULIZUMAB	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.021878196	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.7395446652914718	PSOROMIC ACID	chembl:CHEMBL176570	PSOROMIC ACID	FALSE	FALSE	FALSE
PHOSPHODIESTERASE	hgnc:877	ALDH7A1	TTD	2020.06.01	NULL	4.375639269641208	M-518101	chembl:CHEMBL3989862	PEFCALCITOL	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.034773292	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
PTGER3	hgnc:9595	PTGER3	DTC	9/2/20	NULL	1.458546423213736	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
GUANYLYL CYCLASE C	hgnc:4688	GUCY2C	TTD	2020.06.01	NULL	13.12691780892362	SP-333	ncit:C153478	DOLCANATIDE	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	DTC	9/2/20	NULL	0.4167275494896388	SM-122	iuphar.ligand:8855	SM-122	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003401858	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	TCMDC-123781	chembl:CHEMBL581194	CHEMBL:CHEMBL581194	FALSE	FALSE	FALSE
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	10.50153424713889	Codrituzumab	ncit:C80043	CODRITUZUMAB	FALSE	FALSE	FALSE
PABPC1	hgnc:8554	PABPC1	DTC	9/2/20	NULL	4.375639269641208	DITOLYLGUANIDINE	iuphar.ligand:6684	1,3-DITOLYLGUANIDINE	FALSE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	DTC	9/2/20	NULL	0.5373592085524291	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	MRS-1220	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
PLACENTA GROWTH FACTOR	hgnc:8893	PGF	TTD	2020.06.01	NULL	52.50767123569449	TB-403	chembl:CHEMBL2109545	TB-403	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	TCMDC-124381	chembl:CHEMBL579919	CHEMBL:CHEMBL579919	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.023609564	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.013920379	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TCMDC-125298	chembl:CHEMBL581152	CHEMBL:CHEMBL581152	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.023482858	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	DNDI1417701	chembl:CHEMBL1326164	CHEMBL:CHEMBL1326164	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.4565884455277783	BETULINIC ACID	ncit:C38126	BETULINIC ACID	FALSE	FALSE	FALSE
ADAPTOR-ASSOCIATED KINASE 1	hgnc:19679	AAK1	TTD	2020.06.01	NULL	17.50255707856483	LX9211	iuphar.ligand:11957	PILAVAPADIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	WISTIN	chembl:CHEMBL464707	WISTIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	GNF-PF-52	chembl:CHEMBL601142	CHEMBL:CHEMBL601142	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.012869527	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.019949723	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.012020987	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.3697723326457359	BI 860585	ncit:C122836	MTORC1/2 KINASE INHIBITOR BI 860585	FALSE	FALSE	FALSE
DELTA-LIKE PROTEIN 3	hgnc:2909	DLL3	TTD	2020.06.01	NULL	78.76150685354175	Rova-T	ncit:C107678	ROVALPITUZUMAB TESIRINE	FALSE	FALSE	TRUE
XPO1	hgnc:12825	XPO1	DTC	9/2/20	NULL	8.751278539282415	GONIOTHALAMIN	chembl:CHEMBL464443	GONIOTHALAMIN	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	1.000146118775133	EUCALYPTIN A	chembl:CHEMBL2171206	EUCALYPTIN A	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.007952093	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TRIDECAN-1-OL	chembl:CHEMBL24832	TRIDECAN-1-OL	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.031032903	FPL-64176	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.033148782	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.022949157	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1426838892274307	ENDRIN	chembl:CHEMBL44072	ENDRIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.007445784	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
P-SELECTIN GLYCOPROTEIN LIGAND 1	hgnc:10722	SELPLG	TTD	2020.06.01	NULL	52.50767123569449	AbGn-168	ncit:C121711	NEIHULIZUMAB	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	7.501095891	2,4-DIISOVALERYL PHLOROGLUCINOL	chembl:CHEMBL277845	CHEMBL:CHEMBL277845	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.032899543	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1801292323694494	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.2363572458670459	BIBW 2992	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
TNNI3	hgnc:11947	TNNI3	DTC	9/2/20	NULL	0.525076712	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	TRELANSERIN	ncit:C90946	TRELANSERIN	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.063415062	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	SR 16234	ncit:C61494	SELECTIVE ESTROGEN RECEPTOR MODULATOR TAS-108	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	DTC	9/2/20	NULL	0.035478156	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007374673	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	FORMONONETIN	drugbank:DB15335	FORMONONETIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
MELANOCYTES LINEAGE-SPECIFIC ANTIGEN GP100	hgnc:10880	PMEL	TTD	2020.06.01	NULL	2.187819634820604	Melanoma vaccine	ncit:C2517	MELANOMA VACCINE	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.106290832	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	DEHYDROVARIABILIN	chembl:CHEMBL1520512	DEHYDROVARIABILIN	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.008403917	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.08780547	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	ALLOXAN	rxcui:2466730	ALLOXAN	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	2.561349816375341	AMP-224	drugbank:DB15767	AMP-224	FALSE	TRUE	TRUE
NOS3	hgnc:7876	NOS3	DTC	9/2/20	NULL	0.1530835896084387	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	2.917092846427472	AMODIAQUINE HYDROCHLORIDE	rxcui:314495	AMODIAQUINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.500219178	INCB28060	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007179391	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	MECLOFENAMATE SODIUM	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL199592	CHEMBL:CHEMBL199592	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	SCOULERINE	chembl:CHEMBL1235966	SCOULERINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.023223207	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	WR-159412	chembl:CHEMBL268089	WR-159412	FALSE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	2.983390411119005	PROMACTA	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004172574	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.06697407	STILONIUM IODIDE	ncit:C73168	STILONIUM IODIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.026927011	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.011124507	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	(S)-ONDANSETRON	chembl:CHEMBL399705	(S)-ONDANSETRON	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.093763699	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	DOCUSATE	rxcui:82003	DOCUSATE	TRUE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.6482428547616604	Amitifadine	ncit:C169780	AMITIFADINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DYDROGESTERONE	rxcui:3706	DYDROGESTERONE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.2900976311364336	SJ000059272	chembl:CHEMBL592369	CHEMBL:CHEMBL592369	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1875273972703375	ORTHOTOLIDINE	chembl:CHEMBL85109	ORTHOTOLIDINE	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	1.363835616511545	FR-901464	chembl:CHEMBL494107	CHEMBL:CHEMBL494107	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.1562728310586145	Sulfatinib	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.1151484018326633	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	SPIRAMIDE	ncit:C66559	SPIRAMIDE	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.9907107780319716	GNF-PF-3951	chembl:CHEMBL597649	CHEMBL:CHEMBL597649	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.030038714	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	NSC-62406	chembl:CHEMBL1332182	CHEMBL:CHEMBL1332182	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	CYSTEINE METHYL-ESTER HCL	chembl:CHEMBL1426508	CHEMBL:CHEMBL1426508	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.3977853881492006	Amitifadine	ncit:C169780	AMITIFADINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00575742	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	TCMDC-123605	chembl:CHEMBL547285	CHEMBL:CHEMBL547285	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004386606	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.364636606	GAMBOGIC AMIDE	chembl:CHEMBL444109	GAMBOGIC AMIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.030004384	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	6-CHLOROMELATONIN	iuphar.ligand:1346	6-CL-MLT	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010332088	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.029301156	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	OXYBENZONE	rxcui:32673	OXYBENZONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	SJ000113372	chembl:CHEMBL589912	CHEMBL:CHEMBL589912	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 1	hgnc:11036	SLC5A1	TTD	2020.06.01	NULL	4.200613698855561	LIK-066	ncit:C150375	LICOGLIFLOZIN	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.035382528	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	STILONIUM IODIDE	ncit:C73168	STILONIUM IODIDE	FALSE	FALSE	FALSE
RCE1	hgnc:13721	RCE1	DTC	9/2/20	NULL	1.071585127259071	ACRIDIN-1-YLAMINE	chembl:CHEMBL146525	CHEMBL:CHEMBL146525	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PHENYLARSINE OXIDE	iuphar.ligand:9201	PHENYLARSINE OXIDE	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	1.790034246671403	PRACTOLOL	rxcui:8620	PRACTOLOL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	FENOLDOPAM BROMIDE	chembl:CHEMBL1256646	FENOLDOPAM BROMIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.1223955040459079	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.4817217544559128	PHENCYCLIDINE HYDROCHLORIDE	ncit:C75101	PHENCYCLIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005653281	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	1.166837138570988	Oglemilast	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.017295017	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.012719882	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
EPHX2	hgnc:3402	EPHX2	DTC	9/2/20	NULL	3.000438356	ALOIN	ncit:C76760	ALOIN	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	1.141471113819445	MONOCILLIN I	chembl:CHEMBL215853	MONOCILLIN I	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.040515178	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	1.029562181092048	Cadi-05	ncit:C77884	TLR AGONIST CADI-05	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.066662299	ADENOSINE TRIPHOSPHATE	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004972317	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.100976291	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.041672755	NSC-720622	chembl:CHEMBL1287980	CHEMBL:CHEMBL1287980	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	3.000438356	LY-377604	drugbank:DB12858	LY-377604	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.9376369863516875	EMTRICITABINE	rxcui:276237	EMTRICITABINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	FPL-64176	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	KAINIC ACID	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	SJ000119988	chembl:CHEMBL589694	CHEMBL:CHEMBL589694	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.027752469	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.010346339	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.4773424657790409	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	2-(2'-METHOXYPHENYL)-1H-INDOLE	chembl:CHEMBL1449007	2-(2'-METHOXYPHENYL)-1H-INDOLE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.027177884	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	3.889457128569962	TRU-015	drugbank:DB05580	TRU-015	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.138178082	2-PHENYLACETYLAMINOBENZOTHIAZOLE	chembl:CHEMBL1405979	CHEMBL:CHEMBL1405979	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.022315202	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002737341	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00393537	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	6-O-BENZYLGUANINE	drugbank:DB11919	6-O-BENZYLGUANINE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.7395446652914718	CEFQUINOME	ncit:C79564	CEFQUINOME	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.1041818873724097	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	CORONOPILIN	chembl:CHEMBL248564	CORONOPILIN	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.05565201	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
P2RY2	hgnc:8541	P2RY2	DTC	9/2/20	NULL	3.500511415712966	ISO-IANTHERAN A	chembl:CHEMBL240681	ISO-IANTHERAN A	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	DNDI1417268	chembl:CHEMBL1517542	CHEMBL:CHEMBL1517542	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	DNDI1417268	chembl:CHEMBL1517542	CHEMBL:CHEMBL1517542	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	GNF-PF-1654	chembl:CHEMBL602776	CHEMBL:CHEMBL602776	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	(+)-TAXIFOLIN	chembl:CHEMBL66	(+)-TAXIFOLIN	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	DTC	9/2/20	NULL	0.595325071	RIVAROXABAN	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	GNF-PF-4814	chembl:CHEMBL585443	CHEMBL:CHEMBL585443	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.03292017	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	1.093909817410302	4-AMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL60824	4-AMINO-[1,2]NAPHTHOQUINONE	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.038467158	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	8.751278539282417	DIETHYL-2-PENTADECYLIDENEMALONATE	chembl:CHEMBL404916	CHEMBL:CHEMBL404916	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.1581556362520918	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00988845	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	0.9053046764774912	20(S)-GINSENOSIDE RG3	iuphar.ligand:7658	GINSENOSIDE RG3	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006381584	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.08780547	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.084214389	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.045579576	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
SUMO2	hgnc:11125	SUMO2	DTC	9/2/20	NULL	3.750547945406749	BITHIONOLOXIDE	ncit:C78040	BITHIONOLOXIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	METHYSTICIN	chembl:CHEMBL579224	METHYSTICIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	RO-106-9920	chembl:CHEMBL271023	CHEMBL:CHEMBL271023	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	MRS-1220	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	1.000146118775133	MACROCARPAL B	chembl:CHEMBL396848	MACROCARPAL B	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	RAZOXANE	rxcui:9154	RAZOXANE	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.077217164	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014993624	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HEPATOCYTE NUCLEAR FACTOR 1-ALPHA	hgnc:11621	HNF1A	TTD	2020.06.01	NULL	26.25383561784724	Norleucine	ncit:C87587	NORLEUCINE	FALSE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	4.039051633514961	KURARINONE	chembl:CHEMBL243796	KURARINONE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.138178082	TOSYL-L-LYSINE CHLOROMETHYL KETONE	chembl:CHEMBL466465	CHEMBL:CHEMBL466465	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.032173818	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	GNF-PF-1192	chembl:CHEMBL584854	CHEMBL:CHEMBL584854	FALSE	FALSE	FALSE
DYRK4	hgnc:3095	DYRK4	DTC	9/2/20	NULL	0.3977853881492008	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	1.458546423213736	GHRP-2	rxcui:1492039	PRALMORELIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	AZOSEMIDE	rxcui:18651	AZOSEMIDE	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.3281729452230906	CURCUMIN PYRAZOLE	chembl:CHEMBL180239	CURCUMIN PYRAZOLE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NCI-17383	chembl:CHEMBL188641	CHEMBL:CHEMBL188641	FALSE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	1.141471113819445	Atrasentan	ncit:C61606	ATRASENTAN	FALSE	FALSE	FALSE
RPS6KA6	hgnc:10435	RPS6KA6	DTC	9/2/20	NULL	1.944728564284981	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	DTC	9/2/20	NULL	0.075496292	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.044198376	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
ESTROGEN-RELATED RECEPTOR-ALPHA	hgnc:3471	ESRRA	TTD	2020.06.01	NULL	8.751278539282415	Dexamethasone palmitate	chemidplus:14899-36-6	DEXAMETHASONE PALMITATE	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	1.944728564284981	TG-100435	chembl:CHEMBL230686	CHEMBL:CHEMBL230686	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.006216868	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1988926940746003	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.093763699	DNDI1417254	chembl:CHEMBL2094567	CHEMBL:CHEMBL2094567	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.010718039	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	Carfentanil	ncit:C80574	CARFENTANIL	FALSE	FALSE	FALSE
PNLIP	hgnc:9155	PNLIP	DTC	9/2/20	NULL	3.029288725136221	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.2500365296937833	GNF-PF-1295	chembl:CHEMBL579837	CHEMBL:CHEMBL579837	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.06375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-1692	chembl:CHEMBL582055	CHEMBL:CHEMBL582055	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	AM-630	iuphar.ligand:750	AM-630	FALSE	FALSE	FALSE
RASGRP1	hgnc:9878	RASGRP1	DTC	9/2/20	NULL	2.333674277141977	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.078958904	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	3-METHOXYFLAVONOL	chembl:CHEMBL272005	CHEMBL:CHEMBL272005	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CORTICOSTERONE	drugbank:DB04652	CORTICOSTERONE	FALSE	FALSE	FALSE
PHOSPHOGLUCONATE DEHYDROGENASE	hgnc:8891	PGD	TTD	2020.06.01	NULL	8.751278539282415	GHRP-2	rxcui:1492039	PRALMORELIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.020542907	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002269228	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	PIRARUBICIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.4688184931758437	N6-CYCLOPENTYLADENOSINE	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	2-MORPHOLINOETHYL 1-PHENYLCYCLOHEXANECARBOXYLATE	iuphar.ligand:6678	PRE-084	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.040082192	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.021951368	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	BIX-01294	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	ANTHRACENE-9-CARBOXYLIC ACID	iuphar.ligand:4113	9-ANTHROIC ACID	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.3889457128569962	Carfentanil	ncit:C80574	CARFENTANIL	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.8204323630577265	CETIRIZINE DIHYDROCHLORIDE	chembl:CHEMBL1607273	CETIRIZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	(S)-MAP4 HCL	chembl:CHEMBL1256510	CHEMBL:CHEMBL1256510	FALSE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	1.500219178	OBP-301	ncit:C119617	SURATADENOTUREV	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.078958904	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.006359941	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.023616644	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006233104	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.062509132	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.2592971419046641	22(S)-HYDROXYCHOLESTEROL	chembl:CHEMBL1243244	CHEMBL:CHEMBL1243244	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW780056X	chembl:CHEMBL1882194	GW780056X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TCMDC-123634	chembl:CHEMBL530499	CHEMBL:CHEMBL530499	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.3365876361262467	ISOBOLDINE	chembl:CHEMBL462880	ISOBOLDINE	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.9907107780319716	Rinfabate	rxcui:1426631	RINFABATE	FALSE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	DTC	9/2/20	NULL	5.250767123569449	LIPOIC ACID	rxcui:6417	THIOCTIC ACID	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-4218	chembl:CHEMBL585269	CHEMBL:CHEMBL585269	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.020713085	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.1105424657593568	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	0.546954909	SILODOSIN	rxcui:720825	SILODOSIN	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.006227191	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	PURVALANOLA	chembl:CHEMBL23327	PURVALANOLA	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ABSCISIC ACID	drugbank:DB16829	ABSCISIC ACID	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
SSTR3	hgnc:11332	SSTR3	DTC	9/2/20	NULL	3.500511415712966	ODT-8	chembl:CHEMBL452157	CHEMBL:CHEMBL452157	FALSE	FALSE	FALSE
CHLORIDE CHANNEL UNSPECIFIC	hgnc:2014	CLC	TTD	2020.06.01	NULL	13.12691780892362	131I-TM-601	ncit:C48263	IODINE I 131 TM-601	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.1704794520639431	TG-02	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.077444943	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	chembl:CHEMBL1226	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.032412143	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.017620024	N-DESMETHYLCLOZAPINE	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	2,6-DIMETHOXYQUINONE	chembl:CHEMBL448515	2,6-DIMETHOXYQUINONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004252322	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009320613	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003262967	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	DANTROLENE SODIUM	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.3889457128569962	Butorphanol	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	ETHAVERINE	rxcui:24464	ETHAVERINE	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	7.501095891	DIDODECANOYLPHLOROGLUCINOL	chembl:CHEMBL470757	DIDODECANOYLPHLOROGLUCINOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	RU-24969	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	SJ000029259	chembl:CHEMBL592558	CHEMBL:CHEMBL592558	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
NR5A2	hgnc:7984	NR5A2	DTC	9/2/20	NULL	13.12691780892362	TDR79154	chembl:CHEMBL597670	CHEMBL:CHEMBL597670	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	NSC-319994	chembl:CHEMBL1329443	CHEMBL:CHEMBL1329443	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.3977853881492008	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003703461	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.050246575	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.035502144	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001612346	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.1691068316769549	Methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	DNDI1417623	chembl:CHEMBL2002849	CHEMBL:CHEMBL2002849	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001678098	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	GNF-PF-265	chembl:CHEMBL602418	CHEMBL:CHEMBL602418	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	ROSE BENGAL	rxcui:9471	ROSE BENGAL	FALSE	FALSE	FALSE
FOLLICLE-STIMULATING HORMONE RECEPTOR	hgnc:3969	FSHR	TTD	2020.06.01	NULL	18.37768493249307	Urofollitropin	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
LGALS9	hgnc:6570	LGALS9	DTC	9/2/20	NULL	35.00511415712966	LACTOSE, ANHYDROUS	chembl:CHEMBL417016	LACTOSE, ANHYDROUS	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004674828	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013825085	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	0.095295229	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.2344092465879218	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.091159151	EFAROXAN	ncit:C72923	EFAROXAN	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	0.4167275494896388	Methylnaltrexone bromide	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002042305	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.055271233	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	CIS-RESVERATROL	chembl:CHEMBL87333	CIS-RESVERATROL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	1,3-DIBENZYLTHIOUREA	chembl:CHEMBL1388908	CHEMBL:CHEMBL1388908	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	2.500365296937833	T-226296	iuphar.ligand:1314	T-226296	FALSE	FALSE	FALSE
EP300	hgnc:3373	EP300	DTC	9/2/20	NULL	8.751278539282415	DIETHYL-2-PENTADECYLIDENEMALONATE	chembl:CHEMBL404916	CHEMBL:CHEMBL404916	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	CHOLINE CHLORIDE	rxcui:1425426	CHOLINE CHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	2,6-DIMETHOXYQUINONE	chembl:CHEMBL448515	2,6-DIMETHOXYQUINONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.005609794	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	TOLNAFTATE	rxcui:10637	TOLNAFTATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	GNF-PF-5029	chembl:CHEMBL1198140	CHEMBL:CHEMBL1198140	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.004428785	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
PTPN11	hgnc:9644	PTPN11	DTC	9/2/20	NULL	1.071585127259071	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.027929612	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	0.3671865121377238	Vasopressin	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
TXN	hgnc:12435	TXN	DTC	9/2/20	NULL	2.917092846427472	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.023943307	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005581766	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.027177884	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	DTC	9/2/20	NULL	0.1041818873724097	ISONIPECOTIC ACID	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.07631929	Pagoclone	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007232462	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.016764901	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.023080295	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006940869	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.1232574442152452	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 2	hgnc:2358	CRHR2	TTD	2020.06.01	NULL	1.875273972703375	NBI-34041	iuphar.ligand:10375	NBI-34041	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	FDA	10-Apr-24	NULL	0.053361455	Amifampridine Phosphate	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.038741518	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
NAT2	hgnc:7646	NAT2	FDA	10-Apr-24	NULL	0.052090944	Amifampridine	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
F5	hgnc:3542	F5	FDA	10-Apr-24	NULL	0.1685639526025505	Avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	0.5707355569097228	Alprostadil	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.026458892	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
F2	hgnc:3535	F2	FDA	10-Apr-24	NULL	0.3947945205691315	Avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	FDA	10-Apr-24	NULL	0.038270897	Carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.016602341	Dextromethorphan	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.006199253	Clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.000912844	Clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.7095631248066824	ABT-510	drugbank:DB05434	ABT-510	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.5676505	THYROTROPIN	rxcui:10579	THYROTROPIN	TRUE	FALSE	FALSE
FHIT	hgnc:3701	FHIT	NCI	14-Sep-17	NULL	0.8751278539282418	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
FKBP4	hgnc:3720	FKBP4	NCI	14-Sep-17	NULL	0.6141248097742046	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	2.100306849	BETA-INTERFERON	ncit:C495	RECOMBINANT INTERFERON BETA	FALSE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	1.750255707856483	ANTI-ANDROGEN	ncit:C242	ANTI-ANDROGEN	FALSE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.5000730593875666	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
GAL	hgnc:4114	GAL	NCI	14-Sep-17	NULL	0.7292732116068681	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.210030685	ZNCL2	rxcui:39937	ZINC CHLORIDE	TRUE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	NCI	14-Sep-17	NULL	2.625383561784724	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.087512785	BROMODEOXYURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.1750255707856483	NORETHISTERONE ACETATE	rxcui:31983	NORETHINDRONE ACETATE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.075010959	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	3.500511415712966	INHIBINS	ncit:C578	RECOMBINANT INHIBIN	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.2885036881082115	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	2.917092846427472	Capromab	ncit:C174682	CAPROMAB	TRUE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	0.2692701089009974	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
GALP	hgnc:24840	GALP	NCI	14-Sep-17	NULL	17.50255707856483	THYROID-STIMULATING HORMONE	rxcui:4952	THYROTROPIN ALFA	TRUE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	0.041426171	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.089298761	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	NCI	14-Sep-17	NULL	0.044310271	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1785975212098452	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	1.875273972703375	Trichlormethiazide	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
GYPA	hgnc:4702	GYPA	NCI	14-Sep-17	NULL	1.875273972703375	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	1.591141552596803	LY-518674	drugbank:DB12988	LY-518674	FALSE	FALSE	FALSE
GTF2B	hgnc:4648	GTF2B	NCI	14-Sep-17	NULL	3.281729452230906	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.8751278539282416	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.034727296	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1752592497853621	Dienestrol	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	2.763561643983921	DISTAMYCIN	ncit:C1517	STALLIMYCIN	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.041872146	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	1.640864726115453	UK-371800	chembl:CHEMBL460293	CHEMBL:CHEMBL460293	FALSE	FALSE	FALSE
HOXB1	hgnc:5111	HOXB1	NCI	14-Sep-17	NULL	1.750255707856483	BROMODEOXYURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.014857858	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.2692701089009974	Doxazosin	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
HSF1	hgnc:5224	HSF1	NCI	14-Sep-17	NULL	3.938075342677087	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1526385791735305	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPD1	hgnc:5261	HSPD1	NCI	14-Sep-17	NULL	11.66837138570988	CETRORELIX	rxcui:68147	CETRORELIX	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.1121958787087489	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	1.521961485092594	Turofexorate isopropyl	ncit:C81536	TUROFEXORATE ISOPROPYL	FALSE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.3365876361262467	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	3.182283105193605	RECOMBINANT PROTHYMOSIN ALPHA	ncit:C1203	RECOMBINANT PROTHYMOSIN ALPHA	FALSE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	3.182283105193605	PROTHYMOSIN ALPHA	ncit:C1203	RECOMBINANT PROTHYMOSIN ALPHA	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	1.363835616511545	AT7519	ncit:C64761	CDK INHIBITOR AT7519	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	NCI	14-Sep-17	NULL	0.070765056	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.4487835148349958	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	4.039051633514961	SANDOSTATIN	chembl:CHEMBL408687	SANDOSTATIN	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.4018444227221517	INTERFERON ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	1.166837138570989	SU5402	drugbank:DB08577	3-[(3-(2-CARBOXYETHYL)-4-METHYLPYRROL-2-YL)METHYLENE]-2-INDOLINONE	FALSE	FALSE	FALSE
C1 ESTERASE INHIBITOR	hgnc:1228	SERPING1	TTD	2020.06.01	NULL	26.25383561784724	Cinryze	rxcui:1599832	C1 ESTERASE INHIBITOR	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	1.875273972703375	RECOMBINANT INTERLEUKIN-1-BETA	ncit:C585	RECOMBINANT INTERLEUKIN-1-BETA	FALSE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	1.346350544504987	DROLOXIFENE	ncit:C969	DROLOXIFENE	FALSE	FALSE	FALSE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	0.1654653505326507	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.175610941	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.6731752722524935	MANNITOL	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
IL1A	hgnc:5991	IL1A	NCI	14-Sep-17	NULL	0.5834185692854945	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.6863747873946993	AUTOANTIGEN	ncit:C20972	AUTOANTIGEN	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	2.059124362184098	IL-2 GENE	ncit:C2549	INTERLEUKIN-2 GENE	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.2500365296937833	Methylnaltrexone bromide	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.3571950424196904	SELECTIVE ESTROGEN RECEPTOR MODULATORS	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.1530835896084387	INTERFERON ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
COMPLEMENT C1S COMPONENT	hgnc:1247	C1S	TTD	2020.06.01	NULL	2.625383561784724	Cinryze	rxcui:1599832	C1 ESTERASE INHIBITOR	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.1852122442176172	ACE INHIBITOR	ncit:C247	ACE INHIBITOR	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.6482428547616604	DEOXYSPERGUALIN	drugbank:DB12991	DEOXYSPERGUALIN	FALSE	FALSE	FALSE
LIPA	hgnc:6617	LIPA	NCI	14-Sep-17	NULL	0.5834185692854944	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	1.419126249613364	Tarafenacin	ncit:C87644	TARAFENACIN	FALSE	FALSE	FALSE
LOH19CR1	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	1.615620653405984	STEEL FACTOR	ncit:C1410	RECOMBINANT HUMAN STEM CELL FACTOR	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.2007335520076852	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	1.250182648468916	ANABOLIC STEROID	ncit:C2360	ANABOLIC STEROID	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.2500365296937833	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.2282942227638891	TGF-BETA 2	ncit:C1286	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA-2	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.2941606231691568	ACE INHIBITOR	ncit:C247	ACE INHIBITOR	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.2201579506737715	SERMS	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	2.282942227638891	MV-CEA	ncit:C64775	CARCINOEMBRYONIC ANTIGEN-EXPRESSING MEASLES VIRUS	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.021309932	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.3182283105193606	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	5.834185692854944	INCOMPLETE FREUNDS ADJUVANT	ncit:C1573	INCOMPLETE FREUND'S ADJUVANT	FALSE	FALSE	FALSE
MT-CO1	hgnc:7419	MT-CO1	NCI	14-Sep-17	NULL	0.9723642821424908	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
P2Y PURINOCEPTOR 12	hgnc:18124	P2RY12	TTD	2020.06.01	NULL	3.828684360936057	Prasugrel	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
MT1JP	hgnc:7402	MT1JP	NCI	14-Sep-17	NULL	1.329308132549227	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	8.751278539282415	BCM	chembl:CHEMBL460283	MANNOMUSTINE	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1666910197958555	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.034888818	PRED	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.1715936968486748	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.025948936	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.5048814541893701	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.5966780822238011	DFMO	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	1.640864726115453	ACTH	iuphar.ligand:1331	ACTH	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	2.019525817	BETA-INTERFERON	ncit:C495	RECOMBINANT INTERFERON BETA	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.030607794	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.6908904109959803	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.046965717	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.012844342	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.21578495	INTERFERON GAMMA	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.1215455352678113	RAS INHIBITOR	ncit:C1902	RAS INHIBITOR	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	1.250182648468916	RAZOXANE	rxcui:9154	RAZOXANE	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.079798892	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	ALPHA-ADRENERGIC AGONIST	ncit:C29709	ALPHA-ADRENERGIC AGONIST	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.047561296	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1215455352678113	CYPROHEPTADINE HYDROCHLORIDE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	0.3088686543276147	PTC299	drugbank:DB05173	PTC299	FALSE	FALSE	FALSE
PTGES3	hgnc:16049	PTGES3	NCI	14-Sep-17	NULL	1.060761035064535	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	NCI	14-Sep-17	NULL	0.2386712328895204	SULINDAC SULFIDE	ncit:C29854	SULINDAC SULFIDE	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	2.625383561784724	PF-4878691	ncit:C61104	TLR7 AGONIST 852A	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	NCI	14-Sep-17	NULL	0.05068308	CHEMOTHERAPEUTIC AGENT	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	NCI	14-Sep-17	NULL	0.6563458904461812	GINGER	rxcui:899420	GINGER ALLERGENIC EXTRACT	TRUE	FALSE	FALSE
MONOCYTE CHEMOTACTIC AND ACTIVATING FACTOR	hgnc:10618	CCL2	TTD	2020.06.01	NULL	4.375639269641208	Bindarit	ncit:C96701	BINDARIT	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.2983390411119005	berberine	rxcui:1437	BERBERINE	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.1750255707856483	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
MYT1L	hgnc:7623	MYT1L	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.2333674277141977	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
SCLEROSTIN	hgnc:13771	SOST	TTD	2020.06.01	NULL	6.563458904461812	LY2541546	chembl:CHEMBL1742993	BLOSOZUMAB	FALSE	FALSE	FALSE
PKD2	hgnc:9009	PKD2	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
PLA2G4A	hgnc:9035	PLA2G4A	PharmGKB	4/5/24	NULL	0.062065805	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PROTEASOME	hgnc:9338	PRB2	TTD	2020.06.01	NULL	7.501095891	Delanzomib	ncit:C74075	DELANZOMIB	FALSE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	PharmGKB	4/5/24	NULL	1.640864726115453	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.082472782	nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
LYMPHOTOXIN BETA RECEPTOR	hgnc:6718	LTBR	TTD	2020.06.01	NULL	52.50767123569449	HCBE-11	chembl:CHEMBL2109509	HCBE-11	FALSE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.1228249619548409	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.017620024	n-desmethylclozapine	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.001276813	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.018354192	diltiazem	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.3387591692625452	trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	1.193356164447602	E6005	chembl:CHEMBL3989967	LOTAMILAST	FALSE	FALSE	FALSE
F13A1	hgnc:3531	F13A1	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.004669216	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	1.400204566285186	asunaprevir	rxcui:1652103	ASUNAPREVIR	FALSE	FALSE	FALSE
PLCD3	hgnc:9061	PLCD3	PharmGKB	4/5/24	NULL	6.563458904461812	diltiazem	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	1.381780822	penicillin v	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
P-SELECTIN	hgnc:10721	SELP	TTD	2020.06.01	NULL	5.250767123569449	PSI-697	drugbank:DB12211	PSI-697	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.4605936073306534	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1151484018326633	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.017835486	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.1893305453210138	ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
CSPG4	hgnc:2466	CSPG4	PharmGKB	4/5/24	NULL	0.1764963739014941	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.3977853881492006	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1835932560688619	ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	1.009762908	oxazine 89	iuphar.ligand:6944	OXAZINE 89	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	PharmGKB	4/5/24	NULL	1.500219178	trandolapril	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	PharmGKB	4/5/24	NULL	0.1562728310586145	cemiplimab-rwlc	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
IMMUNOGLOBULIN E	hgnc:5522	IGHE	TTD	2020.06.01	NULL	17.50255707856483	MEDI4212	chembl:CHEMBL2109452	MEDI-4212	FALSE	FALSE	FALSE
GTPASE NRAS	hgnc:7989	NRAS	TTD	2020.06.01	NULL	0.6351734423672721	GI-4000	drugbank:DB05698	GI-4000	FALSE	FALSE	FALSE
KLKB1	hgnc:6371	KLKB1	PharmGKB	4/5/24	NULL	11.25164383622025	ecallantide	rxcui:658708	ECALLANTIDE	TRUE	FALSE	FALSE
NFATC1	hgnc:7775	NFATC1	PharmGKB	4/5/24	NULL	1.193356164447602	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.4167275494896388	Taberminogene vadenovec	drugbank:DB05011	TABERMINOGENE VADENOVEC	FALSE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	TALC	12-May-16	NULL	0.2500365296937833	ETIDRONATE	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
EPCAM	hgnc:11529	EPCAM	TALC	12-May-16	NULL	1.575230137070835	MT110	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.2273059360852575	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	1.591141552596802	MK-3697	iuphar.ligand:9307	MK-3697	FALSE	FALSE	FALSE
PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9	hgnc:20001	PCSK9	TTD	2020.06.01	NULL	8.078103267029922	Bococizumab	ncit:C166723	BOCOCIZUMAB	FALSE	FALSE	FALSE
ASPARAGINASE	hgnc:16448	ASRGL1	TTD	2020.06.01	NULL	26.25383561784724	Calaspargase pegol	rxcui:2121416	CALASPARGASE PEGOL	TRUE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.2692701089009974	Abexinostat	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	1.166837138570988	CG-200745	drugbank:DB12259	CG-200745	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.6134073742487676	RAD-1901	rxcui:2628469	ELACESTRANT	TRUE	FALSE	TRUE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	XmAb-20717	chembl:CHEMBL4594617	VUDALIMAB	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	MGD013	ncit:C143957	TEBOTELIMAB	FALSE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	0.8751278539282416	Fremanezumab	rxcui:2056691	FREMANEZUMAB	TRUE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	1.193356164447602	Tezacaftor and ivacaftor	drugsatfda.nda:210491	TEZACAFTOR AND IVACAFTOR	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.2841324201065719	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	3.500511415712966	Tagraxofusp	rxcui:2109054	TAGRAXOFUSP-ERZS	TRUE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	TALC	12-May-16	inhibitor	0.096432821	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Diphenylpyraline	rxcui:23386	DIPHENYLPYRALINE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	0.2542744369767287	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
GSR	hgnc:4623	GSR	TALC	12-May-16	NULL	2.386712328895204	NOV-002	drugbank:DB05393	NOV-002	FALSE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.2573905452730122	Flavoxate	rxcui:4440	FLAVOXATE	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.086007651	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.2651902587661338	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.7836965856073805	AZD 1152	hemonc:60	BARASERTIB	FALSE	FALSE	TRUE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	0.3512218811752141	Oxytocin	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	TALC	12-May-16	inhibitor	1.640864726115453	AZD4877	iuphar.ligand:7708	AZD4877	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1479089330582944	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.5903640284436551	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	2.187819634820604	Proguanil	rxcui:2382	PROGUANIL	TRUE	FALSE	FALSE
MMP14	hgnc:7160	MMP14	TALC	12-May-16	vaccine	1.071585127259071	PRINOMASTAT	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	1.500219178	SGX523	ncit:C74062	MET TYROSINE KINASE INHIBITOR SGX523	FALSE	FALSE	TRUE
MUC1	hgnc:7508	MUC1	TALC	12-May-16	vaccine	1.093909817410302	MVA-MUC1-IL2	ncit:C2241	MESMULOGENE ANCOVACIVEC	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.1215455352678113	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.1143957978991165	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.1118771404169627	Isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	TALC	12-May-16	inhibitor	0.05486695	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	1.944728564284981	Altropane	drugbank:DB04947	ALTROPANE	FALSE	FALSE	FALSE
SIRT4	hgnc:14932	SIRT4	TALC	12-May-16	inhibitor	1.591141552596803	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
TEK	hgnc:11724	TEK	TALC	12-May-16	inhibitor	0.9845188356692718	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	4.773424657790408	Miglitol	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	TALC	12-May-16	agonist	29.17092846427472	LEXATUMUMAB	ncit:C64621	LEXATUMUMAB	FALSE	TRUE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	TALC	12-May-16	agonist	17.50255707856483	LBY135	chembl:CHEMBL2109247	LBY-135	FALSE	TRUE	TRUE
BIRC2	hgnc:590	BIRC2	TALC	12-May-16	inhibitor	1.875273972703375	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
DLL4	hgnc:2910	DLL4	TALC	12-May-16	inhibitor	4.200613698855561	REGN421	ncit:C82367	ENOTICUMAB	FALSE	FALSE	TRUE
CYP19A1	hgnc:2594	CYP19A1	TALC	12-May-16	inhibitor	0.7693431682885642	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
UNIPROT:P01903	hgnc:4947	HLA-DRA	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	1D09C3	drugbank:DB05121	1D09C3	FALSE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.3302369260106572	4SC-202	drugbank:DB13101	4SC-202	FALSE	FALSE	FALSE
UNIPROT:P16671	hgnc:1663	CD36	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	ABT-510	drugbank:DB05434	ABT-510	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.1296485709523321	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.030176823	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.089501712	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
UNIPROT:P43119	hgnc:9602	PTGIR	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	BERAPROST	ncit:C76896	BERAPROST	FALSE	FALSE	FALSE
UNIPROT:P00491	hgnc:7892	PNP	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	ULODESINE	ncit:C152793	ULODESINE	FALSE	FALSE	FALSE
UNIPROT:Q96BI3	hgnc:29509	APH1A	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	BMS-299897	chembl:CHEMBL247471	CHEMBL:CHEMBL247471	FALSE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.1187956362798518	VORTIOXETINE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.1795134059339983	VORTIOXETINE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.024384367	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A	hgnc:7943	NPR1	TTD	2020.06.01	NULL	1.009762908	Cenderitide	ncit:C171663	CENDERITIDE	FALSE	FALSE	FALSE
UNIPROT:P28566	hgnc:5291	HTR1E	TdgClinicalTrial	Jan-14	NULL	0.138178082	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.01535312	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.007196775	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.007196775	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.019739726	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P15509	hgnc:2435	CSF2RA	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	ONCOVEX GM-CSF	rxcui:1721264	TALIMOGENE LAHERPAREPVEC	TRUE	FALSE	FALSE
UNIPROT:P42081	hgnc:1705	CD86	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	ABATACEPT	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.1552333222045661	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.054398002	PROPAFENONE	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	2.561349816375341	SGN-19A	ncit:C105150	DENINTUZUMAB MAFODOTIN	FALSE	FALSE	FALSE
UNIPROT:P23786	hgnc:2330	CPT2	TdgClinicalTrial	Jan-14	NULL	0.1426838892274307	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
UNIPROT:A5X5Y0	hgnc:24005	HTR3E	TdgClinicalTrial	Jan-14	NULL	1.400204566285186	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.048260727	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.061628722	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
UNIPROT:Q9UQB9	hgnc:11391	AURKC	TdgClinicalTrial	Jan-14	NULL	0.059330702	R763	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:P56696	hgnc:6298	KCNQ4	TdgClinicalTrial	Jan-14	NULL	1.500219178162699	RETIGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
UNIPROT:O43526	hgnc:6296	KCNQ2	TdgClinicalTrial	Jan-14	NULL	3.000438356325399	RETIGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
CANCER/TESTIS ANTIGEN 1	hgnc:2491	CTAG1B	TTD	2020.06.01	NULL	3.281729452230906	GSK-2241658A	ncit:C116847	ANTI-NY-ESO-1 IMMUNOTHERAPEUTIC GSK-2241658A	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	ROFLUMILAST	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
UNIPROT:P98160	hgnc:5273	HSPG2	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	0.138178082	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.01858569	RISPERDAL	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	2.917092846427472	Anti-CD22 CAR-T cells	ncit:C201173	ANTI-CD22 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
UNIPROT:P08709	hgnc:3544	F7	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	RECOMBINANT NEMATODE ANTICOAGULANT PROTEIN C2	chembl:CHEMBL4298082	RECOMBINANT NEMATODE ANTICOAGULANT PROTEIN C2	FALSE	FALSE	FALSE
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TdgClinicalTrial	Jan-14	NULL	0.3500511415712966	RIMCAZOLE	ncit:C152218	RIMCAZOLE	FALSE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TdgClinicalTrial	Jan-14	NULL	0.051277023	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q9NY46	hgnc:10590	SCN3A	TdgClinicalTrial	Jan-14	NULL	0.054695491	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q9UQD0	hgnc:10596	SCN8A	TdgClinicalTrial	Jan-14	NULL	0.055622533	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P05362	hgnc:5344	ICAM1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	SAR 1118	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	4SCAR19 cells	ncit:C148156	AUTOLOGOUS CD19CAR-CD28-CD137/CD27/CD3ZETA-ICASP9-EXPRESSING T-LYMPHOCYTES	FALSE	FALSE	FALSE
UNIPROT:P35499	hgnc:10591	SCN4A	TdgClinicalTrial	Jan-14	NULL	0.050488145	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P20701	hgnc:6148	ITGAL	TdgClinicalTrial	Jan-14	NULL	1.357957014716237	SAR 1118	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.020936073	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.008774678	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CALCITONIN RECEPTOR	hgnc:1440	CALCR	TTD	2020.06.01	NULL	6.563458904461812	Calcitonin Human	rxcui:235481	HUMAN CALCITONIN	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	0.07458476	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P32970	hgnc:11937	CD70	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	SGN-75	chembl:CHEMBL2108672	VORSETUZUMAB MAFODOTIN	FALSE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	3.750547945	Carboprost Tromethamine	rxcui:20259	CARBOPROST TROMETHAMINE	TRUE	FALSE	FALSE
UNIPROT:P78527	hgnc:9413	PRKDC	TdgClinicalTrial	Jan-14	NULL	0.7292732116068681	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.032173818	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:Q6V0L0	hgnc:20577	CYP26C1	TdgClinicalTrial	Jan-14	NULL	10.50153425	TALAROZOLE	ncit:C90792	TALAROZOLE	FALSE	FALSE	FALSE
UNIPROT:O43174	hgnc:2603	CYP26A1	TdgClinicalTrial	Jan-14	NULL	15.75230137070834	TALAROZOLE	ncit:C90792	TALAROZOLE	FALSE	FALSE	FALSE
UNIPROT:P13569	hgnc:1884	CFTR	TdgClinicalTrial	Jan-14	NULL	2.983390411119005	IVACAFTOR	rxcui:1243041	IVACAFTOR	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.2536602475154323	NRP104	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
UNIPROT:P31749	hgnc:391	AKT1	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	XL418	drugbank:DB05204	XL418	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.03729238	Dextromethorphan Polistirex	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
UNIPROT:P23443	hgnc:10436	RPS6KB1	TdgClinicalTrial	Jan-14	NULL	1.064344687210023	XL418	drugbank:DB05204	XL418	FALSE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.064824285	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:O00329	hgnc:8977	PIK3CD	TdgClinicalTrial	Jan-14	NULL	0.1852122442176172	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.2853677784548614	XL888	ncit:C79835	HSP90 INHIBITOR XL888	FALSE	FALSE	TRUE
UNIPROT:P50579	hgnc:16672	METAP2	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	XMT-1107	ncit:C88321	FUMAGILLIN-DERIVED POLYMER CONJUGATE XMT-1107	FALSE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	3.500511415712966	Ibandronate	rxcui:115264	IBANDRONATE	TRUE	FALSE	FALSE
UNIPROT:P98170	hgnc:592	XIAP	TdgClinicalTrial	Jan-14	NULL	0.8334550989792777	CUDC-427	ncit:C103825	SMAC MIMETIC GDC-0917	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.693795846312725	ALCAFTADINE	rxcui:1000082	ALCAFTADINE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	2.316514907	AMBENONIUM	rxcui:623	AMBENONIUM	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TdgClinicalTrial	Jan-14	NULL	0.7501095890813498	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2004109589148645	ALCLOMETASONE	rxcui:108088	ALCLOMETASONE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.4817217544559128	ANILERIDINE	rxcui:17933	ANILERIDINE	TRUE	FALSE	FALSE
UNIPROT:P05546	hgnc:4838	SERPIND1	TdgClinicalTrial	Jan-14	NULL	7.501095890813499	ARDEPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	BENZTHIAZIDE	rxcui:19008	BENZTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	ARDEPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1635752997996713	Sibutramine	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.3040984820600068	CEVIMELINE	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	1.250182648468916	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.078194596	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.068191781	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1875273972703375	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.066465407	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1346350544504987	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.064824285	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.1988926940746003	DESOXIMETASONE	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.040703621	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TEND	1-Aug-11	NULL	1.014640990061729	DESMOPRESSIN	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
T-BOX TRANSCRIPTION FACTOR T	hgnc:11515	TBXT	TTD	2020.06.01	NULL	26.25383561784724	GI-6301	drugbank:DB17533	GI-6301	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	5.250767123569449	Valbenazine Tosylate	rxcui:1923002	VALBENAZINE TOSYLATE	TRUE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TEND	1-Aug-11	NULL	0.5834185692854945	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.1041818873724097	Trilostane	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.1193356164447602	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	0.4449802647092754	IRBESARTAN	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TEND	1-Aug-11	NULL	0.025390557	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	3.889457128569962	BI-853520	chembl:CHEMBL3544961	BI-853520	FALSE	FALSE	FALSE
UNIPROT:P43088	hgnc:9600	PTGFR	TEND	1-Aug-11	NULL	15.00219178	LATANOPROST	rxcui:43611	LATANOPROST	TRUE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.041214813	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.1219218372345847	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	1.491695205559502	Carteolol	rxcui:2116	CARTEOLOL	TRUE	FALSE	FALSE
UNIPROT:P02671	hgnc:3661	FGA	TEND	1-Aug-11	NULL	0.4773424657790409	ALTEPLASE	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
SODIUM PUMP	hgnc:15879	CTNNBL1	TTD	2020.06.01	NULL	26.25383561784724	Beta-acetyldigoxin	chembl:CHEMBL2074725	ACETYLDIGOXIN	FALSE	FALSE	FALSE
UNIPROT:P16233	hgnc:9155	PNLIP	TEND	1-Aug-11	NULL	3.029288725136221	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.1154014752432845	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.099446347	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.097236428	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.060761035064535	Cetrorelix	rxcui:68147	CETRORELIX	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	0.729273212	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.2	hgnc:1395	CACNA1H	TTD	2020.06.01	NULL	0.4440395030502706	Flunarizine	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.2792961235941196	Glycopyrrolate	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.6563458904461812	NEPAFENAC	rxcui:298665	NEPAFENAC	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.056826484	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.2117244807890907	Mepyramine	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.2692701089009974	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	1.000146118775133	Mepindolol	rxcui:29518	MEPINDOLOL	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.081407242	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TEND	1-Aug-11	NULL	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.1141471113819445	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.2234368988752957	Pirenzepine	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.1262203635473425	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	0.3563869088395554	Oxytocin	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.096050618	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.5645986154375752	Pilsicainide	ncit:C72582	PILSICAINIDE	FALSE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TEND	1-Aug-11	NULL	0.9723642821424906	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.2019525816757481	Sarpogrelate	ncit:C73158	SARPOGRELATE	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	OXYPHENCYCLIMINE	rxcui:32698	OXYPHENCYCLIMINE	TRUE	FALSE	FALSE
SUCCINATE-SEMIALDEHYDE DEHYDROGENASE	hgnc:408	ALDH5A1	TTD	2020.06.01	NULL	3.750547945	Succinic acid	rxcui:37255	SUCCINIC ACID	TRUE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TEND	1-Aug-11	NULL	0.2237542808339254	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.056622219	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
UNIPROT:Q15858	hgnc:10597	SCN9A	TEND	1-Aug-11	NULL	0.1103102336884338	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TEND	1-Aug-11	NULL	0.1795134059339982	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TEND	1-Aug-11	NULL	7.955707762984016	PRANLUKAST	ncit:C96712	PRANLUKAST	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL	hgnc:1527	CAV1	TTD	2020.06.01	NULL	4.375639269641208	Tolperisone	rxcui:10639	TOLPERISONE	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.071585127259071	Human coagulation factor X	rxcui:1426166	COAGULATION FACTOR X, HUMAN	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.2154897588332195	Yohimbine	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
SODIUM/HYDROGEN EXCHANGER 3	hgnc:11073	SLC9A3	TTD	2020.06.01	NULL	13.12691780892362	AZD1722	iuphar.ligand:8449	TENAPANOR	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.9907107780319716	AEW-541	chembl:CHEMBL551064	AEW-541	FALSE	FALSE	FALSE
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	3.500511415712966	CVX-241	chembl:CHEMBL4650388	CVX-241	FALSE	FALSE	FALSE
PROTEIN CEREBLON	hgnc:30185	CRBN	TTD	2020.06.01	NULL	5.834185692854944	CC-122	ncit:C160786	AVADOMIDE	FALSE	FALSE	FALSE
B-CELL-ACTIVATING FACTOR	hgnc:11929	TNFSF13B	TTD	2020.06.01	NULL	32.81729452230906	Belimumab	rxcui:1092437	BELIMUMAB	TRUE	TRUE	TRUE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	1.750255707856483	WP-1066	drugbank:DB12679	WP-1066	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	1.544343271638073	IMO-2055	drugbank:DB06181	IMO-2055	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.2557191780959147	ITI-007	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.0504235	INK128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.7955707762984013	LIRIMILAST	ncit:C82304	LIRIMILAST	FALSE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	1.810609352954982	BPX-101	ncit:C82361	AUTOLOGOUS PROSTATE CANCER ANTIGEN-EXPRESSING DENDRITIC CELL VACCINE BPX-101	FALSE	FALSE	FALSE
CATIONIC TRYPSINOGEN	hgnc:9475	PRSS1	TTD	2020.06.01	NULL	8.751278539282415	Alpha-1 antitrypsin	ncit:C82258	ALPHA-1-PROTEINASE INHIBITOR HUMAN	FALSE	FALSE	FALSE
LYSOPHOSPHATIDATE-3 RECEPTOR	hgnc:14298	LPAR3	TTD	2020.06.01	NULL	17.50255707856483	SAR-100842	iuphar.ligand:11315	SAR100842	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.041508041	Naphazoline	rxcui:7247	NAPHAZOLINE	TRUE	FALSE	FALSE
AMINOTRANSFERASE	hgnc:4175	GATM	TTD	2020.06.01	NULL	3.750547945	F-351	chembl:CHEMBL4297288	HYDRONIDONE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.8655110643246346	Chlorothiazide	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	1.250182648468916	Amylin	ncit:C169781	AMLINTIDE	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.057260274	Prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Fluoroquinolones	ncit:C126712	FLUOROQUINOLONE ANTIBIOTIC	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.6543011991986852	Phentermine	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	1.458546423213736	Methsuximide	rxcui:47858	METHSUXIMIDE	TRUE	FALSE	FALSE
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	2.386712328895204	SLV 306	ncit:C73039	DAGLUTRIL	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.3922986931402463	Amsacrine	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.2692701089009974	Alfuzosin	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
DIACYLGLYCEROL O-ACYLTRANSFERASE 2	hgnc:16940	DGAT2	TTD	2020.06.01	NULL	3.750547945406749	Vitamin B3	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	0.2302968036653267	Anisindione	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
TUBULIN BETA-2 CHAIN	hgnc:12412	TUBB2A	TTD	2020.06.01	NULL	0.073540156	Vinblastine	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.104285345	NVP-LAQ824	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.3443125982668492	Norethindrone	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 1	hgnc:11330	SSTR1	TTD	2020.06.01	NULL	0.8751278539282418	ODT-8	chembl:CHEMBL452157	CHEMBL:CHEMBL452157	FALSE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	1.029562181092048	UE-2343	iuphar.ligand:12037	UE2343	FALSE	FALSE	FALSE
T-CELL SURFACE ANTIGEN CD2	hgnc:1639	CD2	TTD	2020.06.01	NULL	17.50255707856483	Siplizumab	ncit:C38685	SIPLIZUMAB	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.3889457128569962	Codeine	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	1.750255707856483	Tebipenem	chembl:CHEMBL576981	TEBIPENEM	FALSE	FALSE	FALSE
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	3.750547945	SNAP-7941	iuphar.ligand:1313	SNAP-7941	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.2004109589148645	Betamethasone	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	Anileridine	rxcui:17933	ANILERIDINE	TRUE	FALSE	FALSE
ENDOGLIN CD105	hgnc:3349	ENG	TTD	2020.06.01	NULL	26.25383561784724	TRC105	ncit:C74010	CAROTUXIMAB	FALSE	FALSE	FALSE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	0.5048814541893701	Cholic Acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	1.419126249613364	CP-122721	drugbank:DB05421	CP-122721	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1635752997996713	Spiroglumide	ncit:C73219	SPIROGLUMIDE	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.006694845	Methyldopa	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
TYROSINE 3-MONOOXYGENASE	hgnc:11782	TH	TTD	2020.06.01	NULL	1.500219178	Tetrahydrobiopterin	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
VASOPRESSIN V1B RECEPTOR	hgnc:896	AVPR1B	TTD	2020.06.01	NULL	0.4688184931758437	ATOSIBAN	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.1555782851427985	Tropisetron	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	21.00306849427779	Methoxy polyethylene glycol-epoetin beta	rxcui:729596	METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.2500365296937833	Remifentanil	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Cryptenamine Acetates	rxcui:235225	CRYPTENAMINE ACETATES	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.068191781	Citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
THYROID HORMONE RECEPTOR ALPHA	hgnc:11796	THRA	TTD	2020.06.01	NULL	7.501095891	Dextrothyroxine Sodium	rxcui:40070	DEXTROTHYROXINE SODIUM	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Estradiol Cypionate	rxcui:1000146	ESTRADIOL CYPIONATE	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.038382801	Midazolam	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.3017682254924971	Teniposide	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
GUANYLYL CYCLASE C	hgnc:4688	GUCY2C	TTD	2020.06.01	NULL	19.69037671338543	Plecanatide	rxcui:1873752	PLECANATIDE	TRUE	FALSE	FALSE
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	1.909369863116163	IMC-CS4	chembl:CHEMBL2109323	IMC-CS4	FALSE	FALSE	FALSE
TRANSFERASE UNSPECIFIC	hgnc:11740	TF	TTD	2020.06.01	NULL	13.12691780892362	Ademetionine	ncit:C100098	ADEMETIONINE	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.3977853881492007	GFT-505	ncit:C166574	ELAFIBRANOR	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	0.1973972602845657	GFT-505	ncit:C166574	ELAFIBRANOR	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.071439008	Verubulin	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	0.7501095890813501	BUTAPROST	ncit:C74369	BUTAPROST	FALSE	FALSE	FALSE
MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN	hgnc:7467	MTTP	TTD	2020.06.01	NULL	5.250767123569449	BMS-201038	rxcui:1364478	LOMITAPIDE MESYLATE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1221108633388244	Butabarbital	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.116943588	Dromostanolone	rxcui:23678	DROMOSTANOLONE	TRUE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.091796628	Duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.090530468	IUPHAR.LIGAND:7191	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	1.458546423213736	Enoxaparin	rxcui:221095	ENOXAPARIN SODIUM	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	Ketotifen	rxcui:11404	KETOTIFEN FUMARATE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.09963505	Lidocaine	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Lurasidone hydrochloride	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	0.384671584	Prinomastat	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	0.1842374429322614	Ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.2864054794674245	Tenoxicam	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	0.192335792	Sulindac	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
HYPERPOLARIZATION CYCLIC NUCLEOTIDE-GATED CHANNEL	hgnc:29665	MALAT1	TTD	2020.06.01	NULL	3.500511415712967	Cilobradine	ncit:C81347	CILOBRADINE	FALSE	FALSE	FALSE
AURORA KINASE C	hgnc:11391	AURKC	TTD	2020.06.01	NULL	1.750255707856483	GSK1070916A	ncit:C91081	AURORA B/C KINASE INHIBITOR GSK1070916A	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.1025540453822158	GSK690693	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	0.789589041	RVX-208	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.047518255	GDC0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
METASTASIS-SUPPRESSOR KISS-1	hgnc:6341	KISS1	TTD	2020.06.01	NULL	52.50767123569449	TAK-448	drugbank:DB11975	TAK-448	FALSE	FALSE	FALSE
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	21.00306849427779	LCQ908	ncit:C166592	PRADIGASTAT	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.5357925636295356	PRT4445	rxcui:2045114	ANDEXANET ALFA	TRUE	FALSE	FALSE
NCBIGENE:1519	hgnc:2542	CTSO	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8181	iuphar.ligand:8181	COMPOUND 1 [PMID: 20005102]	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.050294704	IUPHAR.LIGAND:45	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:388	drugbank:DB07954	3-ISOBUTYL-1-METHYL-7H-XANTHINE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:11	iuphar.ligand:11	CP 93129	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.075442056	IUPHAR.LIGAND:46	ncit:C76441	OCAPERIDONE	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:401	iuphar.ligand:401	MRS923	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:11153	ncit:C148039	IMARADENANT	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1136529680426287	IUPHAR.LIGAND:457	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.5413161983061289	IUPHAR.LIGAND:5736	iuphar.ligand:5736	[3H]HEMADO	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.112919723	IUPHAR.LIGAND:587	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1715936968486748	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:8863	ncit:C127116	DUBERMATINIB	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:11887	iuphar.ligand:11887	TINENGOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1403948428761885	IUPHAR.LIGAND:7332	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.045265234	IUPHAR.LIGAND:7427	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2792	hgnc:4411	GNGT1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:7710	iuphar.ligand:7710	AZD5582	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:6165	iuphar.ligand:6165	RHODEI-LITORIN	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:6939	iuphar.ligand:6939	AZ-4217	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:6940	iuphar.ligand:6940	TAK-070	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.059397818	IUPHAR.LIGAND:556	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:547	iuphar.ligand:547	SR59230A	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:550	ncit:C72615	BUPRANOLOL	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8548	iuphar.ligand:8548	COMPOUND 2 [PMID: 26061392]	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:9814	iuphar.ligand:9814	CCT241161	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.090530468	IUPHAR.LIGAND:94	ncit:C152139	RACLOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:2893	hgnc:4574	GRIA4	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12232	iuphar.ligand:12232	BAY-069	FALSE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.2885036881082115	IUPHAR.LIGAND:5501	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.089298761	IUPHAR.LIGAND:152	iuphar.ligand:152	&ALPHA;-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:2598	hgnc:1372	CA14	GuideToPharmacology	2024.1	inhibitor	0.7292732116068681	IUPHAR.LIGAND:7147	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.2885036881082115	IUPHAR.LIGAND:6792	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2598	hgnc:1372	CA14	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:6792	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:6810	rxcui:60207	DORZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:5295	iuphar.ligand:5295	Z-DQMD-FMK	FALSE	FALSE	FALSE
NCBIGENE:528	hgnc:856	ATP6V1C1	GuideToPharmacology	2024.1	activator	1.166837138570989	IUPHAR.LIGAND:2518	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	blocker	1.166837138570989	IUPHAR.LIGAND:10159	ncit:C81680	BENIDIPINE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.1054370908347279	IUPHAR.LIGAND:46	ncit:C76441	OCAPERIDONE	FALSE	FALSE	FALSE
NCBIGENE:1581	hgnc:2651	CYP7A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7892	iuphar.ligand:7892	EXAMPLE 166  [WO2014154727]	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:730	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
NCBIGENE:391	hgnc:672	RHOG	GuideToPharmacology	2024.1	activator	0.1483267549030918	IUPHAR.LIGAND:2377	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.065799087	IUPHAR.LIGAND:733	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10177	iuphar.ligand:10177	AM10257	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:733	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:9772	ncit:C174799	LENABASUM	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:8410	iuphar.ligand:8410	DESULFATED GASTRIN-71	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:7557	rxcui:8348	PIPOTHIAZINE	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.039361073	IUPHAR.LIGAND:940	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.057073556	IUPHAR.LIGAND:939	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.008428198	IUPHAR.LIGAND:958	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.065226921	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:1232	hgnc:1604	CCR3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:10707	ncit:C167156	QUEMLICLUSTAT	FALSE	FALSE	FALSE
NCBIGENE:2889	hgnc:4568	RAPGEF1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:9033	iuphar.ligand:9033	PSB-6426	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12987	iuphar.ligand:12987	COMPOUND 18J [PMID: 35446588]	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.041672755	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:4862	iuphar.ligand:4862	AG1478	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:11136	ncit:C133691	AUMOLERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:9912	iuphar.ligand:9912	ALLITINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	NULL	0.2500365296937833	IUPHAR.LIGAND:4948	iuphar.ligand:4948	HB-EGF	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.42006137	IUPHAR.LIGAND:1894	ncit:C79571	CLOPROSTENOL	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	NULL	0.2500365296937833	IUPHAR.LIGAND:4873	iuphar.ligand:4873	BETACELLULIN	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:12300	iuphar.ligand:12300	SMTP-7	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.7955707762984013	IUPHAR.LIGAND:1940	ncit:C76900	FLUPROSTENOL	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12520	iuphar.ligand:12520	TG8-260	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.1600843635234588	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.033854076	IUPHAR.LIGAND:1013	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	NULL	0.9053046764774912	IUPHAR.LIGAND:5030	iuphar.ligand:5030	NEUREGULIN-3	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.041672755	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	antibody	2.917092846427472	IUPHAR.LIGAND:8930	iuphar.ligand:8930	ISTIRATUMAB	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:132	iuphar.ligand:132	CYANOPINDOLOL	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:8899	iuphar.ligand:8899	(S)-LIQUIRITIGENIN	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.1302273592155121	IUPHAR.LIGAND:1015	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.093098708	IUPHAR.LIGAND:1013	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:2822	iuphar.ligand:2822	R,R-THC	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3519	iuphar.ligand:3519	PD164333	FALSE	FALSE	FALSE
NCBIGENE:623	hgnc:1029	BDKRB1	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:2829	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
NCBIGENE:2016	hgnc:3340	EMX1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:6026	iuphar.ligand:6026	PKR INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2014	hgnc:3335	EMP3	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8743	iuphar.ligand:8743	COMPOUND 34 [PMID: 20189382]	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.014699796	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:870	hgnc:10939	SLC1A1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:4626	iuphar.ligand:4626	NBI-59159	FALSE	FALSE	FALSE
NCBIGENE:870	hgnc:10939	SLC1A1	GuideToPharmacology	2024.1	NULL	0.3409589041278864	IUPHAR.LIGAND:4698	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	NULL	0.5303805175322677	IUPHAR.LIGAND:4698	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:4317	iuphar.ligand:4317	SYM2081	FALSE	FALSE	FALSE
NCBIGENE:868	hgnc:1542	CBLB	GuideToPharmacology	2024.1	NULL	1.050153425	IUPHAR.LIGAND:4534	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1718	hgnc:2859	DHCR24	GuideToPharmacology	2024.1	agonist	0.3860858179095184	IUPHAR.LIGAND:4921	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9603	iuphar.ligand:9603	BIA 10-2639	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4241	iuphar.ligand:4241	L838417	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:4083	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	blocker	0.145450613	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.6403374540938354	IUPHAR.LIGAND:10427	ncit:C167009	BASMISANIL	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.100589408	IUPHAR.LIGAND:4839	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
NCBIGENE:411	hgnc:714	ARSB	GuideToPharmacology	2024.1	blocker	0.6908904109959803	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.036847489	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:412	hgnc:11425	STS	GuideToPharmacology	2024.1	blocker	0.1842374429322614	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:416	hgnc:721	ARSF	GuideToPharmacology	2024.1	agonist	0.4565884455277782	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:4143	iuphar.ligand:4143	AZA-THIP	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6087	iuphar.ligand:6087	GALANIN(1-16) (RAT/MOUSE/PIG)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:3593	iuphar.ligand:3593	GALANIN	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:5870	iuphar.ligand:5870	GSK1614343	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:3538	iuphar.ligand:3538	YIL781	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:4070	drugbank:DB02966	FLUORO-WILLARDIINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:206	ncit:C83940	MESULERGINE	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:10005	iuphar.ligand:10005	COMPOUND 17 [PMID: 29741897]	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:9325	ncit:C171915	VELSECORAT	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	0.5527123287967842	IUPHAR.LIGAND:4317	iuphar.ligand:4317	SYM2081	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:4276	iuphar.ligand:4276	NVP-AAM077	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4243	iuphar.ligand:4243	LY233053	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.1411496538593938	IUPHAR.LIGAND:2403	ncit:C65450	DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	blocker	0.2651902587661338	IUPHAR.LIGAND:2291	iuphar.ligand:2291	PICROTOXININ	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:9198	iuphar.ligand:9198	COMPOUND 4G [PMID: 2680437]	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:5955	drugbank:DB08325	2-({6-[(3-CHLOROPHENYL)AMINO]-9-ISOPROPYL-9H-PURIN-2-YL}AMINO)ETHANOL	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.044498026	IUPHAR.LIGAND:8019	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:11407	iuphar.ligand:11407	COMPOUND 5 [PMID: 19338355]	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:6929	ncit:C97364	TIDEGLUSIB	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	modulator	2.282942227638891	IUPHAR.LIGAND:5795	iuphar.ligand:5795	COMPOUND 9N [PMID: 18752940]	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.055155117	IUPHAR.LIGAND:152	iuphar.ligand:152	&ALPHA;-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:4850	iuphar.ligand:4850	[125I]STA	FALSE	FALSE	FALSE
NCBIGENE:608	hgnc:11913	TNFRSF17	GuideToPharmacology	2024.1	agonist	0.3947945205691315	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.066297565	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:1887	ncbigene:1887	EBVM1	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:5070	iuphar.ligand:5070	LIGHT	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:7495	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.035098711	IUPHAR.LIGAND:150	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1275	iuphar.ligand:1275	[125I]CCL16 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:1251	iuphar.ligand:1251	IMMEPIP	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.013879903	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	0.064824285	IUPHAR.LIGAND:5552	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.019304291	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5743	iuphar.ligand:5743	COMPOUND 1 [PMID: 21939274]	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:2885	iuphar.ligand:2885	25-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:10543	iuphar.ligand:10543	CLUL1 (52-77)	FALSE	FALSE	FALSE
NCBIGENE:114	hgnc:239	ADCY8	GuideToPharmacology	2024.1	modulator	8.751278539282415	IUPHAR.LIGAND:10440	iuphar.ligand:10440	MS48107	FALSE	FALSE	FALSE
NCBIGENE:147	hgnc:278	ADRA1B	GuideToPharmacology	2024.1	agonist	0.2536602475154323	IUPHAR.LIGAND:3698	iuphar.ligand:3698	R-SPONDIN-2	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:235	iuphar.ligand:235	ML 10302	FALSE	FALSE	FALSE
NCBIGENE:150	hgnc:281	ADRA2A	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:7041	iuphar.ligand:7041	CGEN-856	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:3699	iuphar.ligand:3699	R-SPONDIN-3	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4383	iuphar.ligand:4383	R-SPONDIN-4	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.019233579	IUPHAR.LIGAND:1626	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.064111931	IUPHAR.LIGAND:1663	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.3621218705909966	IUPHAR.LIGAND:5689	iuphar.ligand:5689	JNJ-28312141	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.1458546423213736	IUPHAR.LIGAND:7427	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.064347636	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:5685	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6491	ncit:C77602	CANDOXATRILAT	FALSE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:6502	iuphar.ligand:6502	FASIDOTRILAT	FALSE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:9091	iuphar.ligand:9091	COMPOUND 1A [PMID: 25692029]	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:4009	iuphar.ligand:4009	&ALPHA;-CONOTOXIN-GIC	FALSE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:3964	iuphar.ligand:3964	&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:264	iuphar.ligand:264	SB 699551	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:5742	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:5769	iuphar.ligand:5769	SB 414240	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1473	iuphar.ligand:1473	NEUROMEDIN U-8	FALSE	FALSE	FALSE
NCBIGENE:304	hgnc:539	ANXA2P2	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:1501	iuphar.ligand:1501	NEUROPEPTIDE B-23	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1477	iuphar.ligand:1477	1DME	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1483	iuphar.ligand:1483	[125I]1DME	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:5306	iuphar.ligand:5306	KH28	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:4016	iuphar.ligand:4016	RFRP-3	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:1569	iuphar.ligand:1569	JMV431	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2886	ncit:C87423	ALMOREXANT	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:12604	iuphar.ligand:12604	CVN45502	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:4460	ncit:C169980	FILOREXANT	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:4461	iuphar.ligand:4461	SB-649868	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9465	iuphar.ligand:9465	[3H]-ALMOREXANT	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:1703	iuphar.ligand:1703	SB-334867	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:4461	iuphar.ligand:4461	SB-649868	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8181	iuphar.ligand:8181	COMPOUND 1 [PMID: 20005102]	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:1757	iuphar.ligand:1757	BZATP	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:4093	iuphar.ligand:4093	&ALPHA;&BETA;-MEATP	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	agonist	0.6563458904461813	IUPHAR.LIGAND:1757	iuphar.ligand:1757	BZATP	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:4093	iuphar.ligand:4093	&ALPHA;&BETA;-MEATP	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1755	iuphar.ligand:1755	ADP&BETA;S	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:1760	iuphar.ligand:1760	DATP	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10503	iuphar.ligand:10503	GSK1370319A	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1710	iuphar.ligand:1710	2MESADP	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.087952548	IUPHAR.LIGAND:1776	rxcui:1656052	CANGRELOR	TRUE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.051177067	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	0.5645986154375752	IUPHAR.LIGAND:1763	iuphar.ligand:1710	2MESADP	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1748	iuphar.ligand:1748	MRS2782	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1711	iuphar.ligand:1711	2MESATP	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:4043	iuphar.ligand:4043	MRS2768	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1833	drugbank:DB02261	PLATELET ACTIVATING FACTOR	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	NULL	0.8751278539282416	IUPHAR.LIGAND:4375	iuphar.ligand:4375	EUROPIUM-LABELLED INSL5	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:8432	iuphar.ligand:8432	JNJ-18038683	FALSE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	activator	0.1256164383629055	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:768	hgnc:1383	CA9	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:11745	ncit:C1405	VALSPODAR	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1999	iuphar.ligand:1999	[125I]RELAXIN-3 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11599	iuphar.ligand:11599	SD-91	FALSE	FALSE	FALSE
NCBIGENE:2201	hgnc:3604	FBN2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8827	iuphar.ligand:8827	COMPOUND 11J [PMID: 23021994]	FALSE	FALSE	FALSE
NCBIGENE:1173	hgnc:564	AP2M1	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4670	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10217	iuphar.ligand:10217	SLC4101431	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.064033745	IUPHAR.LIGAND:9693	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2023	iuphar.ligand:2023	[125I]LTT-SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:2007	iuphar.ligand:2007	CORTISTATIN-14	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:2011	iuphar.ligand:2011	DES-AA1,5-[TYR2,D-TRP8,IAMP9]SRIF	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:7763	iuphar.ligand:7763	ANALOG 32 [PMID:18543899]	FALSE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:8144	iuphar.ligand:8144	COMPOUND 13R [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:10114	iuphar.ligand:10114	MK-4256	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2047	iuphar.ligand:2047	L-363,301	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:2040	iuphar.ligand:2040	BIM 23068	FALSE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:10192	iuphar.ligand:10192	ADU-S100	FALSE	FALSE	FALSE
NCBIGENE:1784	ncbigene:1784	DNCM	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8144	iuphar.ligand:8144	COMPOUND 13R [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:3356	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1972	iuphar.ligand:1972	U46609	FALSE	FALSE	FALSE
NCBIGENE:2421	hgnc:3931	FRA8C	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:10732	ncit:C90704	OTAMIXABAN	FALSE	FALSE	FALSE
NCBIGENE:1660	hgnc:2750	DHX9	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:10421	iuphar.ligand:10421	AM237	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:4256	iuphar.ligand:4256	ML9	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.5147810905460244	IUPHAR.LIGAND:4206	iuphar.ligand:4206	GSMTX-4	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.6908904109959803	IUPHAR.LIGAND:2443	iuphar.ligand:2443	ACAA	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:12531	iuphar.ligand:12531	BTDM	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	0.026045472	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.729273212	IUPHAR.LIGAND:10298	iuphar.ligand:10298	NARINGENIN	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	0.4861821410712453	IUPHAR.LIGAND:2452	drugbank:DB03203	SPHINGOSINE	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:7890	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	0.8751278539282418	IUPHAR.LIGAND:4186	iuphar.ligand:4186	ETHYLISOPROPYLAMILORIDE	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.750109589	IUPHAR.LIGAND:4283	iuphar.ligand:4283	PHENYLACETYLRINVANIL	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.2500365296937833	IUPHAR.LIGAND:2488	ncit:C166774	OLVANIL	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	activator	0.066465407	IUPHAR.LIGAND:2299	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:1658	hgnc:188	ADAM10	GuideToPharmacology	2024.1	inhibitor	0.1312691780892362	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:9432	iuphar.ligand:9432	PF-06263276	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:11895	iuphar.ligand:11895	COMPOUND 13 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	NULL	1.810609352954982	IUPHAR.LIGAND:9440	iuphar.ligand:9440	[125I]N-BIOTIN-[AHX0, BPA3]U-II (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:2197	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.006496866	IUPHAR.LIGAND:2182	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.009745299	IUPHAR.LIGAND:2197	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.002248915	IUPHAR.LIGAND:2168	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:2646	hgnc:4196	GCKR	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:6795	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.1981421556063943	IUPHAR.LIGAND:515	ncit:C77294	CIRAZOLINE	FALSE	FALSE	FALSE
NCBIGENE:2282	hgnc:3714	FKBP1AP1	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7710	iuphar.ligand:7710	AZD5582	FALSE	FALSE	FALSE
NCBIGENE:1614	hgnc:13557	ACE2	GuideToPharmacology	2024.1	NULL	5.250767123569449	IUPHAR.LIGAND:5132	iuphar.ligand:5132	ABZ-SER-PRO-TYR(NO2)-OH	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1508	iuphar.ligand:1508	NPY-(2-36) (PIG)	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.008681824	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.066297565	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:690	hgnc:1126	BTF3P11	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
NCBIGENE:695	hgnc:1133	BTK	GuideToPharmacology	2024.1	inhibitor	0.1029562181092049	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
NCBIGENE:688	hgnc:6349	KLF5	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:604	iuphar.ligand:604	[3H](PYR1)[MET(0)11]-APELIN-13	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:11471	iuphar.ligand:11471	COMPOUND 5B [PMID: 25974655]	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.007717177	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.070860555	IUPHAR.LIGAND:2713	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
ABCC3	hgnc:54	ABCC3	CIViC	10-Apr-24	NULL	0.017363648	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.043636393	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.1256164383629055	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
PDGFB	hgnc:8800	PDGFB	CIViC	10-Apr-24	NULL	0.3571950424196904	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	CIViC	10-Apr-24	NULL	0.074927706	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	3.088686543276147	IUPHAR.LIGAND:11475	iuphar.ligand:11475	UGR 9-1	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.3241214273808302	FLT3 INHIBITOR FF-10101 SUCCINATE	ncit:C137988	FLT3 INHIBITOR FF-10101 SUCCINATE	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1621858570986702	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
TOP1	hgnc:11986	TOP1	CIViC	10-Apr-24	NULL	0.097236428	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:5604	ncit:C96195	ROLOFYLLINE	FALSE	FALSE	FALSE
STMN1	hgnc:6510	STMN1	CIViC	10-Apr-24	NULL	0.1620607136904151	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CIViC	10-Apr-24	NULL	0.5000730593875666	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.1438566335224507	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.1269527834518725	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.1604757678352521	VORASIDENIB	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.05068308	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:3290	ncit:C74246	APADENOSON	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	CIViC	10-Apr-24	NULL	0.3500511415712966	TRABECTEDIN	rxcui:1716278	TRABECTEDIN	TRUE	FALSE	TRUE
PBK	hgnc:18282	PBK	CIViC	10-Apr-24	NULL	0.1544343271638073	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:400	iuphar.ligand:400	MRS1132	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.08334551	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	ncit:C69145	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.3968833804663227	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CASP8	hgnc:1509	CASP8	CIViC	10-Apr-24	NULL	2.625383561784724	CONATUMUMAB	ncit:C71015	CONATUMUMAB	FALSE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.069454592	LOMUSTINE	rxcui:6466	LOMUSTINE	TRUE	FALSE	TRUE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:453	iuphar.ligand:449	MRS1754	FALSE	FALSE	FALSE
DDX43	hgnc:18677	DDX43	CIViC	10-Apr-24	NULL	0.3500511415712966	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	1.029562181092049	PATRITUMAB DERUXTECAN	ncit:C136987	PATRITUMAB DERUXTECAN	FALSE	FALSE	TRUE
MYC	hgnc:7553	MYC	CIViC	10-Apr-24	NULL	0.1250182648468916	PREXASERTIB	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.085239726	IUPHAR.LIGAND:5605	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	CIViC	10-Apr-24	NULL	0.1060761035064535	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.076098074	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.048061942	Vincristine Sulfate	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:5590	iuphar.ligand:5590	TCPA	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.040452751	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	1.193356164447602	Pyrvinium	rxcui:35163	PYRVINIUM	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1060761035064535	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	2.386712328895204	ICG-001	drugbank:DB18024	ICG-001	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.2651902587661338	Veliparib	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	modulator	0.5413161983061289	IUPHAR.LIGAND:9446	iuphar.ligand:9446	LUF6000	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.3596415838061266	Veliparib	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1591141552596803	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	13.12691780892362	GVAX	drugbank:DB17276	GVAX	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	1.374546367426557	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.082472782	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.028937818	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:11930	iuphar.ligand:11930	COMPOUND 1 [PMID: 28379944]	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:7949	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.026519026	IUPHAR.LIGAND:5932	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.015516451	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:5691	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:7937	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
NCBIGENE:2792	hgnc:4411	GNGT1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:7732	iuphar.ligand:7732	SM-337	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8507	iuphar.ligand:8507	COMPOUND 17C [PMID: 25497965]	FALSE	FALSE	FALSE
NCBIGENE:2846	hgnc:4478	LPAR4	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8320	iuphar.ligand:8320	ABT-737	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.2344092465879218	IUPHAR.LIGAND:532	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.2344092465879218	IUPHAR.LIGAND:532	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.1339481409073839	IUPHAR.LIGAND:554	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:12165	iuphar.ligand:12165	CHF-6366	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.3387591692625452	IUPHAR.LIGAND:7445	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:3467	iuphar.ligand:3467	L742791	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:554	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:8475	iuphar.ligand:8475	AZ628	FALSE	FALSE	FALSE
NCBIGENE:3092	hgnc:4913	HIP1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:10434	iuphar.ligand:10434	COMPOUND 5B  [PMID: 31287314]	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.054243462	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:1624	hgnc:2692	DBIP1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:5296	iuphar.ligand:5296	Z-IETD-FMK	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.067751834	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.2465148884304905	GAMBOGIC AMIDE	chembl:CHEMBL444109	GAMBOGIC AMIDE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	7,3'-DIMETHOXYFLAVONE	chembl:CHEMBL1326944	7,3'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.004067052	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.050879526	Flumazenil	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:714	iuphar.ligand:714	CALHEX 231	FALSE	FALSE	FALSE
P2Y PURINOCEPTOR 12	hgnc:18124	P2RY12	TTD	2020.06.01	NULL	3.281729452230906	INS-50589	rxcui:1313722	REGRELOR	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.030124883	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:2328	hgnc:3771	FMO3	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8563	iuphar.ligand:8563	ARI-3099	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:9004	iuphar.ligand:9004	ADL5859	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:12235	ncit:C166837	UPACICALCET	FALSE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9490	rxcui:1872441	TELOTRISTAT ETHYL	TRUE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.2143170254518143	IUPHAR.LIGAND:1432	iuphar.ligand:1432	SIB-1893	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:308	iuphar.ligand:308	P-F-HHSID	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2270	rxcui:236901	SOMATORELIN	FALSE	FALSE	FALSE
NCBIGENE:1581	hgnc:2651	CYP7A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7891	iuphar.ligand:7891	COMPOUND 8A [PMID: 22861813]	FALSE	FALSE	FALSE
NCBIGENE:2344	hgnc:2528	CTSC	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:8622	iuphar.ligand:8622	COMPOUND 3D [PMID: 3941405]	FALSE	FALSE	FALSE
ETV5	hgnc:3494	ETV5	CIViC	10-Apr-24	NULL	1.050153425	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.013890918	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.090530468	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	inhibitor	1.458546423213736	SEMULOPARIN SODIUM	ncit:C143000	SEMULOPARIN SODIUM	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.4070362111294147	IUPHAR.LIGAND:7721	iuphar.ligand:7721	ABT-639	FALSE	FALSE	FALSE
FSIP1	hgnc:21674	FSIP1	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.046798281	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	4.039051633514961	Evacetrapib	ncit:C166804	EVACETRAPIB	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:12753	drugbank:DB11903	GW842166	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	0.4688184931758437	L-Tryptophan	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12724	iuphar.ligand:12724	LEO 29102	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:1993	iuphar.ligand:1993	RELAXIN	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.2278978786271462	AKT INHIBITOR MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.052090944	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.729273212	ESOMEPRAZOLE STRONTIUM	rxcui:1435522	ESOMEPRAZOLE STRONTIUM	TRUE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:10221	iuphar.ligand:10221	CCK-39	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	2.059124362184098	AV-203	chembl:CHEMBL2109401	AV-203	FALSE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	agonist	1.235474617310459	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	blocker	0.1346350544504987	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	GNF-PF-1211	chembl:CHEMBL600968	CHEMBL:CHEMBL600968	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2075402025126264	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	PROPYLPARABEN	rxcui:34706	PROPYLPARABEN	TRUE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3566	iuphar.ligand:3566	GASTRIN-71	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	DTC	9/2/20	NULL	0.7721716358190367	BODILISANT	chembl:CHEMBL2323582	BODILISANT	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.1193356164447602	Belinostat	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:3476	iuphar.ligand:3476	[3H]DEVAZEPIDE	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.058212496	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	0.276356164	ARQ 087	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3562	iuphar.ligand:3562	GASTRIN-34	FALSE	FALSE	FALSE
UNIPROT:Q04609	hgnc:3788	FOLH1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	CAPROMAB	ncit:C174682	CAPROMAB	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.056622219	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	inhibitor	0.093763699	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2664	ncit:C75192	RAGAGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:203	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:868	iuphar.ligand:868	SR146131	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2365210416022274	ARQ 751	ncit:C128250	PAN-AKT INHIBITOR ARQ751	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	1,7-O-DIACETYLMETHYLGEOPYXIN A	chembl:CHEMBL1889303	CHEMBL:CHEMBL1889303	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:764	iuphar.ligand:764	[125I]CCL5 (HUMAN)	FALSE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	DTC	9/2/20	NULL	0.065634589	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.085378327	IUPHAR.LIGAND:7502	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:66	hgnc:139	ACTBP6	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:817	iuphar.ligand:817	CCL25	FALSE	FALSE	FALSE
NCBIGENE:988	hgnc:1743	CDC5L	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:10605	iuphar.ligand:10605	AZD3965	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	CIViC	10-Apr-24	NULL	0.4773424657790409	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.1458546423213736	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1591141552596803	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
NCBIGENE:2995	hgnc:4704	GYPC	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:9864	iuphar.ligand:9864	TREGALIZUMAB	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.068115956	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP2B	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.4102161815288632	LEVAMISOLE	rxcui:6371	LEVAMISOLE	TRUE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:8920	iuphar.ligand:8920	UBLITUXIMAB	FALSE	FALSE	FALSE
UNIPROT:Q02880	hgnc:11990	TOP2B	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	VORELOXIN	ncit:C95148	VOSAROXIN	FALSE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TEND	1-Aug-11	NULL	1.346350544504987	MOCLOBEMIDE	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
NCBIGENE:1877	hgnc:3121	E4F1	GuideToPharmacology	2024.1	antibody	0.9723642821424908	IUPHAR.LIGAND:6772	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	5.834185692854944	MOR-103	iuphar.ligand:11132	OTILIMAB	FALSE	FALSE	FALSE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.4605936073306535	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	DIPHENIDOL HYDROCHLORIDE	rxcui:47877	DIPHENIDOL HYDROCHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
CTSG	hgnc:2532	CTSG	NCI	14-Sep-17	NULL	0.8751278539282417	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
NCBIGENE:2745	hgnc:4330	GLRX	GuideToPharmacology	2024.1	NULL	5.250767124	IUPHAR.LIGAND:6892	rxcui:1112973	BELATACEPT	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	TCMDC-123480	chembl:CHEMBL588683	CHEMBL:CHEMBL588683	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	blocker	0.1930429089547592	IUPHAR.LIGAND:2397	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	0.4565884455277783	IUPHAR.LIGAND:8161	iuphar.ligand:8161	COMPOUND 17 [PMID: 23642479]	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.3113103037689397	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.068637479	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-123781	chembl:CHEMBL581194	CHEMBL:CHEMBL581194	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	EVANS BLUE	rxcui:4191	EVANS BLUE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	LOMERIZINE	ncit:C66029	LOMERIZINE	FALSE	FALSE	FALSE
NCBIGENE:2733	hgnc:4315	GLE1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8824	iuphar.ligand:8824	COMPOUND 50 [PMID: 24313754]	FALSE	FALSE	FALSE
DAGLA	hgnc:1165	DAGLA	DTC	9/2/20	NULL	0.8078103267029924	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
NCBIGENE:1507	hgnc:1737	CDC42BPA	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.4735986033023426	nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.081597003	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	2.763561643983921	KBP-5074	iuphar.ligand:12040	OCEDURENONE	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	agonist	0.4375639269641209	IUPHAR.LIGAND:1757	iuphar.ligand:1757	BZATP	FALSE	FALSE	FALSE
NCBIGENE:1993	hgnc:3313	ELAVL2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10167	iuphar.ligand:10167	TOMIVOSERTIB	FALSE	FALSE	FALSE
SMARCB1	hgnc:11103	SMARCB1	CIViC	10-Apr-24	NULL	0.7955707762984016	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2852	hgnc:4485	GPER1	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:8404	iuphar.ligand:8404	POLATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	ChEMBL	33	cleavage	0.09869863	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	0.3088686543276147	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:12735	iuphar.ligand:12735	GLPG1837	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:7817	ncit:C79841	TALMAPIMOD	FALSE	FALSE	FALSE
UNIPROT:Q969P6	hgnc:29787	TOP1MT	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	PEG-IRINOTECAN	ncit:C74069	ETIRINOTECAN PEGOL	FALSE	FALSE	TRUE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.077217164	IUPHAR.LIGAND:213	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.305277158	LAS-100977	ncit:C132738	ABEDITEROL	FALSE	FALSE	FALSE
NCBIGENE:706	hgnc:1158	TSPO	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:4275	iuphar.ligand:4275	NS5818	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.089501712	MESALAZINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1491695205559502	VENLAFAXINE	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.043074382	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:6950	iuphar.ligand:6950	COMPOUND 2 [PMID: 22911925]	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:1403	iuphar.ligand:1403	PTBE	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:8069	iuphar.ligand:8069	CP-673451	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.024479101	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
NCBIGENE:2340	hgnc:2097	CMA1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:6503	iuphar.ligand:6503	NK3201	FALSE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	modulator	0.5000730593875667	SUVECALTAMIDE	ncit:C174710	SUVECALTAMIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.020721259	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.4688184931758437	SAPONARIN	chembl:CHEMBL538921	SAPONARIN	FALSE	FALSE	FALSE
NCBIGENE:700	hgnc:1153	BVR1	GuideToPharmacology	2024.1	activator	1.346350544504987	IUPHAR.LIGAND:2439	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1011	hgnc:1752	CDH12P2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524936	IUPHAR.LIGAND:4823	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	ChEMBL	33	inhibitor	0.1544343271638073	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.03409589	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
NCBIGENE:700	hgnc:1153	BVR1	GuideToPharmacology	2024.1	blocker	1.346350544504987	IUPHAR.LIGAND:2439	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.063530153	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:701	hgnc:1149	BUB1B	GuideToPharmacology	2024.1	activator	1.346350544504987	IUPHAR.LIGAND:2439	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
TRPM6	hgnc:17995	TRPM6	PharmGKB	4/5/24	NULL	26.25383561784724	Proton pump inhibitors	ncit:C29723	PROTON PUMP INHIBITOR	FALSE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TEND	1-Aug-11	NULL	0.111481255	ERGOCALCIFEROL	rxcui:4018	ERGOCALCIFEROL	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.039598545	IUPHAR.LIGAND:2713	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2A	hgnc:4585	GRIN2A	TTD	2020.06.01	NULL	0.1268301237577161	Glycine	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	1.944728564284981	99mTc-MIP-1404	ncit:C116887	TECHNETIUM TC 99M TROFOLASTAT	FALSE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:4688	rxcui:26143	GLYCYRRHIZIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:5715	iuphar.ligand:5715	TG-100-115	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10375	iuphar.ligand:10375	NBI-34041	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.235474617310458	INCB086550	iuphar.ligand:11528	INCB086550	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	1.640864726115453	ANTITUMOR ANTIBIOTIC	ncit:C259	ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	N-METHYLHISTAMINE DIHYDROCHLORIDE	chembl:CHEMBL1487156	N-METHYLHISTAMINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	Tislelizumab	rxcui:2677426	TISLELIZUMAB	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.077273983	TOPICAL CORTICOSTEROIDS	ncit:C29505	TOPICAL CORTICOSTEROID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NSC-747268	chembl:CHEMBL595911	CHEMBL:CHEMBL595911	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.045579576	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	2.333674277141978	AZASERINE	ncit:C289	AZASERINE	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:920	iuphar.ligand:920	UROCORTIN 1	FALSE	FALSE	FALSE
INTERFERON GAMMA RECEPTOR	hgnc:5440	IFNGR2	TTD	2020.06.01	NULL	105.0153424713889	Interferon gamma-1b	rxcui:5882	INTERFERON GAMMA-1B	TRUE	TRUE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:8592	iuphar.ligand:8592	[3H]TIOTROPIUM	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:688	iuphar.ligand:688	AMYLIN	FALSE	FALSE	FALSE
GLRB	hgnc:4329	GLRB	ChEMBL	33	positive modulator	0.1693795846312726	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.00897567	GLEEVEC	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.1154014752432846	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:689	iuphar.ligand:689	AC187	FALSE	FALSE	FALSE
CBR3	hgnc:1549	CBR3	PharmGKB	4/5/24	NULL	0.2430910705356226	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.014699796	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1282238613814273	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:3135	hgnc:4964	HLA-G	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:11122	iuphar.ligand:11122	LITIFILIMAB	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	ERYTHROMYCIN GLUCEPTATE	rxcui:24346	ERYTHROMYCIN GLUCEPTATE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	PharmGKB	4/5/24	NULL	0.040328473	propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NCBIGENE:1840	hgnc:3060	DTX1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8137	iuphar.ligand:8137	COMPOUND 8E [PMID: 24432909]	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	1.419126249613364	PBF-509	iuphar.ligand:10193	PBF-509	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.4167275494896388	Tivozanib	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.03251249	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:486	hgnc:4026	FXYD2	GuideToPharmacology	2024.1	blocker	1.458546423213736	IUPHAR.LIGAND:4206	iuphar.ligand:4206	GSMTX-4	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.089298761	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:10660	iuphar.ligand:10660	KBP-066	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.3387591692625452	CLOFAZIMINE	rxcui:2592	CLOFAZIMINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	0.8751278539282416	IUPHAR.LIGAND:2315	iuphar.ligand:2315	LEI-DAB7	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:7919	iuphar.ligand:7919	GNE-9605	FALSE	FALSE	FALSE
NCBIGENE:3081	hgnc:4892	HGD	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:10353	iuphar.ligand:10353	TEPODITAMAB	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.2044691247495891	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	VB-201	drugbank:DB15259	VB-201	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:7971	iuphar.ligand:7971	XL019	FALSE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TEND	1-Aug-11	NULL	0.078136416	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:718	hgnc:1318	C3	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
MAPKAPK2	hgnc:6887	MAPKAPK2	DTC	9/2/20	NULL	0.1325951293830669	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	inhibitor	0.021309932	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	LOXOPROFEN	rxcui:28908	LOXOPROFEN	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.4795221117415022	KU-55933	iuphar.ligand:5928	KU-55933	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.015268296	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.012794267	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:73	hgnc:146	ACTG1P1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:855	iuphar.ligand:855	CXCL16	FALSE	FALSE	FALSE
UNIPROT:Q9Y233	hgnc:21160	LINC00473	TEND	1-Aug-11	NULL	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.045818212	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	ncit:C69145	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	FALSE	FALSE	TRUE
MME	hgnc:7154	MME	ChEMBL	33	inhibitor	2.386712328895204	DAGLUTRIL	ncit:C73039	DAGLUTRIL	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.015993808	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.023524942	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
NCBIGENE:1965	hgnc:3265	EIF2S1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11841	iuphar.ligand:11841	SY-5609	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.1442518440541057	Flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
POLD2	hgnc:9176	POLD2	ChEMBL	33	inhibitor	0.108040476	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.28382525	ST1535	iuphar.ligand:5613	ST-1535	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:10002	iuphar.ligand:10002	TRIPLE MODULATOR 10 [PMID: 29878767]	FALSE	FALSE	FALSE
UQCRB	hgnc:12582	UQCRB	DTC	9/2/20	NULL	105.0153424713889	TERPESTACIN	chembl:CHEMBL1669042	TERPESTACIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	CHLORPHENIRAMINE MALEATE	rxcui:142429	CHLORPHENIRAMINE MALEATE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.050978322	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1750255707856483	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
NCBIGENE:1353	hgnc:2261	COX11	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11378	iuphar.ligand:11378	FUREGRELATE SODIUM	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1855	iuphar.ligand:1855	SDZ 64-412	FALSE	FALSE	FALSE
INTERLEUKIN-1 ALPHA	hgnc:5991	IL1A	TTD	2020.06.01	NULL	5.250767123569449	MABp1	wikidata:Q30314044	MABP1	FALSE	FALSE	FALSE
CHLORIDE CHANNEL UNSPECIFIC	hgnc:2014	CLC	TTD	2020.06.01	NULL	13.12691780892362	Moxidectin	rxcui:1047072	MOXIDECTIN	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.3125456621172291	TETOMILAST	ncit:C90922	TETOMILAST	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	0.4861821410712453	GLOFITAMAB	rxcui:2639782	GLOFITAMAB	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	PTEROSTILBENE	ncit:C153353	PTEROSTILBENE	FALSE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8551	iuphar.ligand:8551	1G244	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.577007376	ANGIOTENSIN CONVERTING ENZYME INHIBITOR	ncit:C247	ACE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:122	iuphar.ligand:122	DIPROPYL-5-CT	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	ChEMBL	33	inhibitor	0.3000438356325399	CTS-1027	drugbank:DB08490	CTS-1027	FALSE	FALSE	FALSE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2983390411119005	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.047734247	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:5697	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	0.077789143	IUPHAR.LIGAND:5687	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:10179	iuphar.ligand:10179	ARRY-502	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:1881	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.043902735	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	ANISOCOUMARIN H	chembl:CHEMBL408980	ANISOCOUMARIN H	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:12503	iuphar.ligand:12503	COMPOUND 6641	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	Pyrvinium	rxcui:35163	PYRVINIUM	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:484	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.081030357	Enasidenib	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	PLICAMYCIN	rxcui:6995	PLICAMYCIN	TRUE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:8996	iuphar.ligand:8996	QAV680	FALSE	FALSE	FALSE
NCBIGENE:3245	hgnc:115	ACLY	GuideToPharmacology	2024.1	inhibitor	39.38075342677087	IUPHAR.LIGAND:8321	rxcui:2282403	BEMPEDOIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1581	hgnc:2651	CYP7A1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7871	rxcui:1102261	TELAPREVIR	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1621	iuphar.ligand:1621	DYNORPHIN A-(1-8)	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5641	iuphar.ligand:5641	Y-KE88	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	1.658136986390352	B-701	ncit:C116863	VOFATAMAB	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	NCI	14-Sep-17	NULL	0.2763561643983921	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.060772768	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.076098074	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	NCI	14-Sep-17	NULL	0.1944728564284981	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	1.750255707856483	TIROFIBAN HYDROCHLORIDE	rxcui:253202	TIROFIBAN HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.017502557	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
FGF22	hgnc:3679	FGF22	DTC	9/2/20	NULL	3.750547945	MORACIN M	chembl:CHEMBL512578	MORACIN M	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.1875273972703375	IUPHAR.LIGAND:484	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	ISOPROPAMIDE IODIDE	rxcui:6051	ISOPROPAMIDE IODIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.010199625	ketoconazole	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:1827	iuphar.ligand:1827	TIP39-(7-39) (HUMAN/BOVINE)	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	2.080014029626545	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
UNIPROT:P24941	hgnc:1771	CDK2	TdgClinicalTrial	Jan-14	NULL	0.6819178082557726	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:8811	iuphar.ligand:8811	COMPOUND 53 [PMID: 19631533]	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	ChEMBL	33	modulator	0.1166837138570988	MOFAROTENE	ncit:C63667	MOFAROTENE	FALSE	FALSE	FALSE
NCBIGENE:2833	hgnc:4540	CXCR3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12785	iuphar.ligand:12785	DDO-3055	FALSE	FALSE	FALSE
UNIPROT:P23921	hgnc:10451	RRM1	TdgClinicalTrial	Jan-14	NULL	0.2725311655831894	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1223955040459079	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:2151	hgnc:3539	F2RL2	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8839	iuphar.ligand:8839	TORIN 2	FALSE	FALSE	FALSE
NCBIGENE:2169	hgnc:3556	FABP2	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:5666	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
NCBIGENE:2010	hgnc:3331	EMD	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:8161	iuphar.ligand:8161	COMPOUND 17 [PMID: 23642479]	FALSE	FALSE	FALSE
MOTHERS AGAINST DECAPENTAPLEGIC HOMOLOG 3	hgnc:6769	SMAD3	TTD	2020.06.01	NULL	0.032755877	FLUORESCEIN	rxcui:25138	FLUORESCEIN	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:2207	iuphar.ligand:2207	[125I]OH-LVA	FALSE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:6507	iuphar.ligand:6507	KC-12615	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.046881849	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.059397818	IUPHAR.LIGAND:1247	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7000	iuphar.ligand:7000	CURCUMIN	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:7925	iuphar.ligand:7925	HAS-NMU	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.096521454	METHIXENE HYDROCHLORIDE	rxcui:258230	METHIXENE HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2778183663264259	LAPATINIB DITOSYLATE	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.091159151	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1429428436543407	interferon alfa-2a, recombinant	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.4070362111294147	OXPRENOLOL	rxcui:7801	OXPRENOLOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	MRS-1220	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	NULL	0.5000730593875666	IUPHAR.LIGAND:4916	iuphar.ligand:4916	EGF	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.1216662358986632	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	NCI	14-Sep-17	NULL	0.3689063552859098	MEDROXYPROGESTERONE	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.025613498	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
PRIM1	hgnc:9369	PRIM1	ChEMBL	33	inhibitor	0.3947945205691315	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
BIRC7	hgnc:13702	BIRC7	TALC	12-May-16	inhibitor	3.750547945406749	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.051277023	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	inhibitor	0.081281225	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
RARB	hgnc:9865	RARB	NCI	14-Sep-17	NULL	0.1992701	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.039331589	IUPHAR.LIGAND:954	ncit:C152121	QUINELORANE	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.2083637747448194	4SC-202	drugbank:DB13101	4SC-202	FALSE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	VIA-2291	chembl:CHEMBL59356	ATRELEUTON	FALSE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TEND	1-Aug-11	NULL	0.8751278539282417	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1204304386139782	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:1881	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	2.500365296937833	IMC-3C5	chembl:CHEMBL2109602	IMC-3C5	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:1921	iuphar.ligand:1921	ONO-8713	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.045167889	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.069134524	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.029573456	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:12303	iuphar.ligand:12303	T532	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001180611	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	TCMDC-124522	chembl:CHEMBL526776	CHEMBL:CHEMBL526776	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.024309107	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.023620185	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.096167896	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:5816	ncit:C152512	TAPRENEPAG	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:5429	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	ANTHRALIN	rxcui:873	ANTHRALIN	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.033207482	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	OXENDOLONE	ncit:C174717	OXENDOLONE	FALSE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.5385402178019949	ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.3241214273808302	IUPHAR.LIGAND:1892	iuphar.ligand:1892	BUTAPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.4375639269641208	GNF-PF-4068	chembl:CHEMBL584668	CHEMBL:CHEMBL584668	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	0.8334550989792776	ABIETIC ACID	chembl:CHEMBL71893	ABIETIC ACID	FALSE	FALSE	FALSE
GPI	hgnc:4458	GPI	NCI	14-Sep-17	NULL	1.875273972703374	HEREGULIN	ncit:C1426	RECOMBINANT HEREGULIN	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.2155487324946408	CYCLOSPORIN	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
PTPN22	hgnc:9652	PTPN22	PharmGKB	4/5/24	NULL	1.166837138570989	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:10103	ncit:C73055	RUPATADINE	FALSE	FALSE	FALSE
NCBIGENE:1880	hgnc:3128	GPR183	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:9334	iuphar.ligand:9334	TIGATUZUMAB	FALSE	FALSE	FALSE
ZBTB4	hgnc:23847	ZBTB4	PharmGKB	4/5/24	NULL	10.50153425	varenicline	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.080042182	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:3164	drugbank:DB06548	MINODRONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:12804	iuphar.ligand:12804	J27644	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:6986	iuphar.ligand:6986	SYN-BRP-LPA	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.090530468	CYCLOSERINE	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	activator	0.072927321	IUPHAR.LIGAND:5483	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
KCNV2	hgnc:19698	KCNV2	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.1600843635234588	IUPHAR.LIGAND:1935	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	positive modulator	0.8751278539282416	OLINCIGUAT	ncit:C153148	OLINCIGUAT	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.325124899	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	0.1666910197958555	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.4526523382387456	DTS-201	drugbank:DB06071	DTS-201	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:12017	iuphar.ligand:12017	COMPOUND 47 [PMID: 35640059]	FALSE	FALSE	FALSE
LAMA3	hgnc:6483	LAMA3	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	LEO-15520	chembl:CHEMBL3545074	LEO-15520	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:12783	iuphar.ligand:12783	BAY1316957	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.049723174	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.086361301	IUPHAR.LIGAND:5667	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:7646	ncit:C80868	FALNIDAMOL	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	1.779921058837101	TAS-119	chembl:CHEMBL3545326	TAS-119	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:10204	iuphar.ligand:10204	NORENDOXIFEN	FALSE	FALSE	FALSE
SLC6A1	hgnc:11042	SLC6A1	ChEMBL	33	inhibitor	14.00204566285186	TIAGABINE HYDROCHLORIDE	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2311077079035849	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004458114	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.058602312	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:8898	iuphar.ligand:8898	FERB 033	FALSE	FALSE	FALSE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8385	iuphar.ligand:8385	LTK-14	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.2108741816694558	HQP1351	ncit:C165549	OLVEREMBATINIB	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:1002	iuphar.ligand:1002	[125I]PD164333	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	DTC	9/2/20	NULL	0.04339477	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	0.3281729452230906	IUPHAR.LIGAND:7384	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:1996	iuphar.ligand:1996	[125I]INSL3 (HUMAN)	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	LAPATINIB DITOSYLATE	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
IMPDH2	hgnc:6053	IMPDH2	PharmGKB	4/5/24	NULL	2.625383561784724	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3479	iuphar.ligand:3479	[3H]S0139	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-732881	chembl:CHEMBL261129	CHEMBL:CHEMBL261129	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3837	iuphar.ligand:3837	[ALA1,3,11,15]ET-1	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	PharmGKB	4/5/24	NULL	0.3409589041278864	motesanib	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
CHRFAM7A	hgnc:15781	CHRFAM7A	PharmGKB	4/5/24	NULL	10.50153425	varenicline	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.4526523382387456	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9651	iuphar.ligand:9651	K-8794	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10888	rxcui:2625882	ADAGRASIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ALFAXALONE	rxcui:1544577	ALFAXALONE	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.4605936073306534	IUPHAR.LIGAND:4366	iuphar.ligand:4366	[3H]CGS8216	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.055563673	IUPHAR.LIGAND:12616	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.040893825	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.5114383561918295	crisaborole	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	NCI	14-Sep-17	NULL	0.093763699	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
SLAM FAMILY MEMBER 7 SLAMF7	hgnc:21394	SLAMF7	TTD	2020.06.01	NULL	26.25383561784724	Elotuzumab	rxcui:1726104	ELOTUZUMAB	TRUE	FALSE	FALSE
NCBIGENE:2652	hgnc:4206	OPN1MW	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7014	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
POLD2	hgnc:9176	POLD2	ChEMBL	33	inhibitor	0.2573905452730122	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	FEPRAZONE	rxcui:8673	FEPRAZONE	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.166837138570989	CYTISINICLINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8247	iuphar.ligand:8247	LDC1267	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:8434	iuphar.ligand:8434	LP-12	FALSE	FALSE	FALSE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	CNF1010	chembl:CHEMBL109480	TANESPIMYCIN	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.364636606	BENZPHETAMINE	rxcui:1422	BENZPHETAMINE	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:243	rxcui:2107310	PRUCALOPRIDE	TRUE	FALSE	FALSE
NCBIGENE:394	hgnc:675	ARHGAP5	GuideToPharmacology	2024.1	activator	3.500511415712967	IUPHAR.LIGAND:2347	iuphar.ligand:2347	CYCLIC GMP	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:7352	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
NCBIGENE:410	hgnc:713	ARSA	GuideToPharmacology	2024.1	blocker	0.1151484018326633	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.2536602475154323	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	DTC	9/2/20	NULL	2.045753424767318	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	QUINOXALINE1	iuphar.ligand:5947	CDK1/5 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2651	hgnc:4204	GCNT2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7015	iuphar.ligand:7015	UNC0638	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.008109293	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.1630673019742065	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CLMN	hgnc:19972	CLMN	PharmGKB	4/5/24	NULL	0.6364566210387212	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	CORALYNE	chembl:CHEMBL363506	CORALYNE	FALSE	FALSE	FALSE
NCBIGENE:868	hgnc:1542	CBLB	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:4609	iuphar.ligand:4609	UCPH-101	FALSE	FALSE	FALSE
HBA2	hgnc:4824	HBA2	ChEMBL	33	positive modulator	4.375639269641208	VOXELOTOR	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1320	iuphar.ligand:1320	&ALPHA;-MSH	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.006105543	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.091796628	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.252440727	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
LPL	hgnc:6677	LPL	PharmGKB	4/5/24	NULL	0.1389091831632129	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3171	iuphar.ligand:3171	NE97220	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	TALC	12-May-16	inhibitor	0.3621218705909965	RETASPIMYCIN	ncit:C80378	RETASPIMYCIN	FALSE	FALSE	TRUE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	DESMOPRESSIN	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.2408608772279564	TD-1211	chembl:CHEMBL3137313	AXELOPRAN	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:12150	iuphar.ligand:12150	LJ-4517	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.053361455	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.095468493	Prilocaine	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
NCBIGENE:664	hgnc:1084	BNIP3	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:11027	iuphar.ligand:11027	OLEUROPEIN	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.2059124362184098	IUPHAR.LIGAND:2646	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8606	iuphar.ligand:8606	JZL195	FALSE	FALSE	FALSE
NCBIGENE:1736	hgnc:2890	DKC1	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:9665	iuphar.ligand:9665	MAB92	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.1151484018326633	IUPHAR.LIGAND:1649	iuphar.ligand:1649	GR 89696	FALSE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.098513454	IUPHAR.LIGAND:5661	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1981421556063943	SJ000114741	chembl:CHEMBL591370	CHEMBL:CHEMBL591370	FALSE	FALSE	FALSE
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	0.1190650141398968	LY3303560	iuphar.ligand:10471	ZAGOTENEMAB	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	CID 1540951	chembl:CHEMBL259421	CHEMBL:CHEMBL259421	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1396480617970598	2-PHENYLACETYLAMINOBENZOTHIAZOLE	chembl:CHEMBL1405979	CHEMBL:CHEMBL1405979	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	TALC	12-May-16	inhibitor	0.3314878234576672	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
PSORS1C3	hgnc:17203	PSORS1C3	PharmGKB	4/5/24	NULL	0.8334550989792776	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.1988926940746003	IUPHAR.LIGAND:4368	iuphar.ligand:4368	[18F]FLUOROETHYLFLUMAZENIL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	TDR78109	chembl:CHEMBL1304363	CHEMBL:CHEMBL1304363	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:12579	iuphar.ligand:12579	NDD-713	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	0.4688184931758437	IUPHAR.LIGAND:10090	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.2488515224440497	IUPHAR.LIGAND:9577	iuphar.ligand:9577	AZ13102909	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.3697723326457359	PROPOXYPHENE	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	INDOCYANINE GREEN SODIUM	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
CR2	hgnc:2336	CR2	NCI	14-Sep-17	NULL	1.875273972703374	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.002830755	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.1909369863116163	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.4605936073306534	IUPHAR.LIGAND:4368	iuphar.ligand:4368	[18F]FLUOROETHYLFLUMAZENIL	FALSE	FALSE	FALSE
CDH23	hgnc:13733	CDH23	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.2678962818147679	FRUQUINTINIB	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1693795846312726	GDC0879	iuphar.ligand:5681	GDC-0879	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.008511537	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
CD86	hgnc:1705	CD86	NCI	14-Sep-17	NULL	0.5834185692854945	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
MGAM	hgnc:7043	MGAM	DTC	9/2/20	NULL	9.546849315580817	RESVERATROL 4'-METHYL ETHER	chembl:CHEMBL291501	RESVERATROL 4'-METHYL ETHER	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	CGI	2/1/22	NULL	0.070574827	MEK inhibitor	ncit:C69145	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	FALSE	FALSE	TRUE
NCBIGENE:615	hgnc:7973	NR2E1	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.116943588	LGD-2941	chembl:CHEMBL467888	LGD-2941	FALSE	FALSE	FALSE
UNIPROT:P01024	hgnc:1318	C3	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	POT-4	iuphar.ligand:9219	AL-78898A	FALSE	FALSE	FALSE
PSMA3	hgnc:9532	PSMA3	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
IGHE	hgnc:5522	IGHE	ChEMBL	33	inhibitor	17.50255707856483	QUILIZUMAB	ncit:C152116	QUILIZUMAB	FALSE	FALSE	FALSE
LTBR	hgnc:6718	LTBR	ChEMBL	33	agonist	52.50767123569449	HCBE-11	chembl:CHEMBL2109509	HCBE-11	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.062808219	IUPHAR.LIGAND:4277	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
MMP8	hgnc:7175	MMP8	ChEMBL	33	inhibitor	1.071585127259071	CTS-1027	drugbank:DB08490	CTS-1027	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.087537101	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.057574201	IUPHAR.LIGAND:4192	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:733	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:8846	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.5048814541893701	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006756874	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.2302968036653267	IUPHAR.LIGAND:4368	iuphar.ligand:4368	[18F]FLUOROETHYLFLUMAZENIL	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.019059046	IUPHAR.LIGAND:224	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.080471527	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW795486X	chembl:CHEMBL396107	GW795486X	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	DTC	9/2/20	NULL	0.1521961485092594	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.6403374540938354	PUCOTENLIMAB	ncit:C160717	PUCOTENLIMAB	FALSE	FALSE	FALSE
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.058212496	IUPHAR.LIGAND:4277	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	LICOFELONE	ncit:C63957	LICOFELONE	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:491	iuphar.ligand:491	A-123189	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DESOGESTREL	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CRKL	hgnc:2363	CRKL	CIViC	10-Apr-24	NULL	0.051478109	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	NCI	14-Sep-17	NULL	0.2035181055647073	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.1422972120208523	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	1.419126249613364	DAPITANT	ncit:C97963	DAPITANT	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
ALOX5AP	hgnc:436	ALOX5AP	ChEMBL	33	inhibitor	7.501095891	FIBOFLAPON SODIUM	ncit:C166995	FIBOFLAPON SODIUM	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	2.143170254518142	LETAXABAN	ncit:C96541	LETAXABAN	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	0.3947945205691315	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6116	iuphar.ligand:6116	GAL-B2-MPEG4	FALSE	FALSE	FALSE
NCBIGENE:114	hgnc:239	ADCY8	GuideToPharmacology	2024.1	modulator	8.751278539282415	IUPHAR.LIGAND:9155	iuphar.ligand:9155	OGERIN	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.3017682254924971	IUPHAR.LIGAND:4368	iuphar.ligand:4368	[18F]FLUOROETHYLFLUMAZENIL	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:7689	iuphar.ligand:7689	&GAMMA;-KTX1.7	FALSE	FALSE	FALSE
NCBIGENE:2667	hgnc:4228	GDI2P1	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:12938	iuphar.ligand:12938	PF-9363	FALSE	FALSE	FALSE
NCBIGENE:1311	hgnc:2227	COMP	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7299	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:5056	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	agonist	0.2011788169949981	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:1492	hgnc:9414	PRKG1	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:5261	iuphar.ligand:5261	RP-8-CPT-CGMPS	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.3017682254924971	IUPHAR.LIGAND:4365	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:2837	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	antibody	0.2011788169949981	IUPHAR.LIGAND:8253	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.078136416	TCMDC-124336	chembl:CHEMBL527271	CHEMBL:CHEMBL527271	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	1.060761035064535	IL-18	iuphar.ligand:4983	IL-18	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	2.763561643983921	GNF-PF-3060	chembl:CHEMBL581449	CHEMBL:CHEMBL581449	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	MRS-1845	chembl:CHEMBL1256776	CHEMBL:CHEMBL1256776	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.073540156	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.3633748874442526	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW801372X	chembl:CHEMBL359999	GW801372X	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.08780547	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	ERGOCALCIFEROL	rxcui:4018	ERGOCALCIFEROL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	2',BETA-DIHYDROXYCHALCONE	chembl:CHEMBL1451434	2',BETA-DIHYDROXYCHALCONE	FALSE	FALSE	FALSE
PRKCB	hgnc:9395	PRKCB	ChEMBL	33	inhibitor	0.1640864726115453	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	modulator	0.133607306	ABBV-3373	iuphar.ligand:12917	ABBV-3373	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.1630673019742065	NEZULCITINIB	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.33338204	AN-2728	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
NCBIGENE:411	hgnc:714	ARSB	GuideToPharmacology	2024.1	blocker	0.5707355569097228	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.027093742	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:Q9UKG9	hgnc:2366	CROT	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
UNIPROT:O95264	hgnc:5298	HTR3B	TdgClinicalTrial	Jan-14	NULL	1.235474617310459	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	blocker	0.05853698	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:912	iuphar.ligand:912	CORTICOTROPHIN-RELEASING HORMONE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.025111273	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.2419708351875322	BITHIONOLOXIDE	ncit:C78040	BITHIONOLOXIDE	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	DTC	9/2/20	NULL	2.763561643983921	CHROMOCARB	ncit:C78116	CHROMOCARB	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.050488145	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL20	hgnc:6002	IL20	ChEMBL	33	inhibitor	52.50767123569449	FLETIKUMAB	ncit:C171836	FLETIKUMAB	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	LISOCABTAGENE MARALEUCEL	rxcui:2479136	LISOCABTAGENE MARALEUCEL	TRUE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2681242786503549	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
UNIPROT:P31751	hgnc:392	AKT2	TdgClinicalTrial	Jan-14	NULL	0.7778914257139926	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6448	iuphar.ligand:6448	COMPOUND 8 [PMID: 15482908]	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.070956312	IUPHAR.LIGAND:357	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.039420174	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	TRANSTORINE	iuphar.ligand:2918	KYNURENIC ACID	FALSE	FALSE	FALSE
UNIPROT:P24752	hgnc:93	ACAT1	TEND	1-Aug-11	NULL	0.2083637747448194	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:4099	iuphar.ligand:4099	TRANS-3-ACPBPA	FALSE	FALSE	FALSE
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	0.280789686	Hydroquinone	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.062645859	Estradiol Acetate	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	PharmGKB	4/5/24	NULL	0.1767935058440892	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	2.917092846427472	PBF-1129	ncit:C148435	ADENOSINE A2B RECEPTOR ANTAGONIST PBF-1129	FALSE	FALSE	FALSE
VASOPRESSIN V1B RECEPTOR	hgnc:896	AVPR1B	TTD	2020.06.01	NULL	0.9376369863516875	SSR149415	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	negative modulator	0.027693919	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.038894571	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:4328	iuphar.ligand:4328	TPMPA	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	binder	0.2470949234620917	BINTRAFUSP ALFA	ncit:C124229	BINTRAFUSP ALFA	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.2112984757975633	PENTAZOCINE	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	0.189216833	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	blocker	0.175610941	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:526	hgnc:854	ATP6V1B2	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:2503	rxcui:1362698	CHLOROFORM	TRUE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.027433475	IUPHAR.LIGAND:5269	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:6164	iuphar.ligand:6164	5-OXO-ODE	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:2181	hgnc:3570	ACSL3	GuideToPharmacology	2024.1	inhibitor	0.1215455352678113	IUPHAR.LIGAND:9381	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1041818873724097	NIFUROXAZIDE	rxcui:31782	NIFUROXAZIDE	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	0.5048814541893701	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.01609924	DAPSONE	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	PharmGKB	4/5/24	NULL	0.1567393171214761	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6099	iuphar.ligand:6099	M242	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	DTC	9/2/20	NULL	1.544343271638073	DESOXYCORDIFOLINE	chembl:CHEMBL453150	DESOXYCORDIFOLINE	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.085239726	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.057700738	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.060772768	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.014603719	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	0.2778183663264259	Vitamin A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
NCBIGENE:240	hgnc:435	ALOX5	GuideToPharmacology	2024.1	agonist	0.5147810905460244	IUPHAR.LIGAND:7705	ncit:C166751	LESOGABERAN	FALSE	FALSE	FALSE
MIR1912	hgnc:35396	MIR1912	PharmGKB	4/5/24	NULL	0.2706580991530644	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1037701012563132	ASENAPINE MALEATE	rxcui:860647	ASENAPINE MALEATE	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	modulator	0.1215455352678113	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
NCBIGENE:987	hgnc:1742	LRBA	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4670	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6113	iuphar.ligand:6113	GAL-B2-C12	FALSE	FALSE	FALSE
TSPYL2	hgnc:24358	TSPYL2	NCI	14-Sep-17	NULL	2.187819634820604	BROMODEOXYURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.750255707856483	Cilansetron	ncit:C76106	CILANSETRON	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	KOS-1803	ncit:C97332	ISO-FLUDELONE	FALSE	FALSE	FALSE
TUT7	hgnc:25817	TUT7	PharmGKB	4/5/24	NULL	1.381780822	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8972	iuphar.ligand:8972	HUMAN GIP(5-30)NH2	FALSE	FALSE	FALSE
UNIPROT:P10912	hgnc:4263	GHR	TEND	1-Aug-11	NULL	10.50153424713889	PEGVISOMANT	rxcui:278739	PEGVISOMANT	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ETHISTERONE	rxcui:4129	ETHISTERONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TEBUFENOZIDE	chembl:CHEMBL226968	TEBUFENOZIDE	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:5867	rxcui:1805438	IBUTAMOREN	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.093098708	ESTRADIOL VALERATE	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:6777	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.053038052	AMITRIPTYLINE HYDROCHLORIDE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	modulator	0.9907107780319716	IUPHAR.LIGAND:11927	iuphar.ligand:11927	LSN3318839	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	1.500219178	INSULIN ASPART	rxcui:352385	INSULIN ASPART PROTAMINE, HUMAN	TRUE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.4688184931758437	IUPHAR.LIGAND:4165	iuphar.ligand:4165	CX516	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.088935758	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3009	iuphar.ligand:3009	COMPOUND 1 [PATEL ET AL., 1991]	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DARGLITAZONE	ncit:C75187	DARGLITAZONE	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:4248	iuphar.ligand:4248	LY392098	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.172722603	METHYLCURCUMIN	chembl:CHEMBL494826	METHYLCURCUMIN	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	immunotherapy	2.561349816375341	AMP-224	drugbank:DB15767	AMP-224	FALSE	TRUE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	antibody	2.561349816375341	AMP-224	drugbank:DB15767	AMP-224	FALSE	TRUE	TRUE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.4688184931758437	IUPHAR.LIGAND:4248	iuphar.ligand:4248	LY392098	FALSE	FALSE	FALSE
FAP	hgnc:3590	FAP	ChEMBL	33	binder	4.039051633514961	F19 131I	chembl:CHEMBL2109643	F19 131I	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.042174836	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:4210	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:10122	iuphar.ligand:10122	H-151	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	DTC	9/2/20	NULL	3.938075342677087	MARAVIROC	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
NCBIGENE:1890	hgnc:3148	TYMP	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:5072	iuphar.ligand:5072	TL6	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.053145416	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2711	hgnc:14933	SIRT5	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8823	iuphar.ligand:8823	COMPOUND 2 [MAURER ET AL., 2012]	FALSE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:9025	iuphar.ligand:9025	852A	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:4268	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	PharmGKB	4/5/24	NULL	2.500365296937833	cotinine	ncit:C70941	COTININE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.070010228	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.041639708	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4170	iuphar.ligand:4170	D-CCPENE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.8975670296699914	Y-27632	drugbank:DB08756	Y-27632	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.062645859	ESTRADIOL VALERATE	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.2059124362184098	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.2822993077187876	IUPHAR.LIGAND:4171	rxcui:1742747	SERINE, D-	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	BETA-TOXICAROL	chembl:CHEMBL1556035	BETA-TOXICAROL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.002567612	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4332	iuphar.ligand:4332	UBP141	FALSE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	CIViC	10-Apr-24	NULL	1.640864726115453	PASIREOTIDE	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.1166837138570989	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1521961485092594	IUPHAR.LIGAND:4239	iuphar.ligand:4239	L689560	FALSE	FALSE	FALSE
DUTP PYROPHOSPHATASE	hgnc:3078	DUT	TTD	2020.06.01	NULL	52.50767123569449	TAS-114	ncit:C116885	DUTPASE/DPD INHIBITOR TAS-114	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.067317527	IUPHAR.LIGAND:3309	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	DTC	9/2/20	NULL	1.250182648468916	RO-0505124	iuphar.ligand:8203	RO-0505124	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	5-METHYLFURMETHIDE	iuphar.ligand:300	METHYLFURMETHIDE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.1976759387696734	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	DL-TRYPTOPHAN	chembl:CHEMBL484901	DL-TRYPTOPHAN	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.1268301237577161	IUPHAR.LIGAND:727	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
ITGA4	hgnc:6140	ITGA4	ChEMBL	33	inhibitor	5.834185692854944	NATALIZUMAB	rxcui:354770	NATALIZUMAB	TRUE	TRUE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	1.923357921	CISAPRIDE	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4168	iuphar.ligand:4168	D-AP5	FALSE	FALSE	FALSE
KCNS3	hgnc:6302	KCNS3	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.084553416	IUPHAR.LIGAND:4268	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	0.6908904109959803	PREXASERTIB	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	EVT-101	drugbank:DB05956	EVT-101	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.1268301237577161	IUPHAR.LIGAND:4084	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
NCBIGENE:2017	hgnc:3338	CTTN	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6740	iuphar.ligand:6740	GSK2606414	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2311	iuphar.ligand:2311	APAMIN	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.035902681	TESTOSTERONE UNDECANOATE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4170	iuphar.ligand:4170	D-CCPENE	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.2625383561784725	TENOXICAM	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002188184	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	DTC	9/2/20	NULL	7.001022831425932	3-((4-NITROPHENYL)AMINO)BENZOIC ACID	chembl:CHEMBL1682200	CHEMBL:CHEMBL1682200	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:4239	iuphar.ligand:4239	L689560	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.03729238	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	ChEMBL	33	inhibitor	0.9723642821424907	TREMELIMUMAB	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
HTR1A	hgnc:5286	HTR1A	DTC	9/2/20	NULL	0.1419126249613365	5-MEO-DMT	iuphar.ligand:145	5-MEO-DMT	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4208	iuphar.ligand:4208	GV196771A	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.5000730593875667	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.081533651	IUPHAR.LIGAND:7270	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006077277	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	blocker	0.1121958787087489	IUPHAR.LIGAND:2403	ncit:C65450	DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4332	iuphar.ligand:4332	UBP141	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6295	drugbank:DB13716	DIBUTYLPHTHALATE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.009220191	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.1060761035064535	IUPHAR.LIGAND:260	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	0.08119743	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.1905904582057876	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	CIViC	10-Apr-24	NULL	0.088665436	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
F8	hgnc:3546	F8	ChEMBL	33	positive modulator	6.177373086552294	EFMOROCTOCOG ALFA	rxcui:1543095	EFMOROCTOCOG ALFA	TRUE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	blocker	0.3977853881492007	IUPHAR.LIGAND:1862	iuphar.ligand:1862	GINKGOLIDE B	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.375054795	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1848861663228679	RAF-265	drugbank:DB05984	RAF-265	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:10521	iuphar.ligand:10521	MRI-1867	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1321	iuphar.ligand:1321	HS014	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:12237	iuphar.ligand:12237	CH7057288	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:6741	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
CD44	hgnc:1681	CD44	NCI	14-Sep-17	NULL	0.5527123287967842	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.073954467	AS-605240	drugbank:DB04769	5-QUINOXALIN-6-YLMETHYLENE-THIAZOLIDINE-2,4-DIONE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.005097832	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	blocker	1.009762908	IUPHAR.LIGAND:1862	iuphar.ligand:1862	GINKGOLIDE B	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.01338969	propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NEUROPEPTIDE Y RECEPTOR TYPE 2	hgnc:7957	NPY2R	TTD	2020.06.01	NULL	3.281729452230906	NEUROPEPTIDE-Y	chembl:CHEMBL267633	NEUROPEPTIDE-Y	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	EDROPHONIUM CHLORIDE	rxcui:3754	EDROPHONIUM CHLORIDE	TRUE	FALSE	FALSE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	0.1666910197958555	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2187819634820604	1-NAPHTHYLISOTHIOCYANATE	chembl:CHEMBL1381098	1-NAPHTHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.9053046764774912	(S)-ONDANSETRON	chembl:CHEMBL399705	(S)-ONDANSETRON	FALSE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	NCI	14-Sep-17	NULL	0.4039051633514962	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	blocker	0.1201548540862574	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
KCNH8	hgnc:18864	KCNH8	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.1816874437221263	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2029	hgnc:3360	ENSA	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:5924	drugbank:DB07364	6-PHENYL[5H]PYRROLO[2,3-B]PYRAZINE	FALSE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	2.917092846427472	CALCIUM OXYBATE	rxcui:2387307	CALCIUM OXYBATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.010923169	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.068458502	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
HP	hgnc:5141	HP	NCI	14-Sep-17	NULL	2.500365296937833	PYRIDOXINE	rxcui:42954	VITAMIN B6	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.068637479	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.088396753	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	ETICLOPRIDE	ncit:C65572	ETICLOPRIDE	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.100976291	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:8470	iuphar.ligand:8470	GSK256073	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DoCM	10-Apr-24	NULL	2.080014029626545	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	DNDI1417623	chembl:CHEMBL2002849	CHEMBL:CHEMBL2002849	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.003632995	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	METYRAPONE	rxcui:6923	METYRAPONE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.063110182	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
NCBIGENE:1444	hgnc:2442	CSHL1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8859	iuphar.ligand:8859	&BETA;-CYANO-L-ALANINE	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.064268875	IUPHAR.LIGAND:6699	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.1215455352678113	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:1969	iuphar.ligand:1969	CAY10441	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.3043922970185188	Idasanutlin	ncit:C99131	IDASANUTLIN	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.192335792	CHEMOTHERAPEUTIC AGENT	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	NSC-724440	chembl:CHEMBL515617	CHEMBL:CHEMBL515617	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.4257378748840094	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	2,6-DIMETHOXYQUINONE	chembl:CHEMBL448515	2,6-DIMETHOXYQUINONE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	FORMONONETIN	drugbank:DB15335	FORMONONETIN	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.251232877	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	0.2083637747448194	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	DEXMEDETOMIDINE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:3622	rxcui:2001986	PALMIDROL	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	PharmGKB	4/5/24	NULL	0.108711535	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.8334550989792776	METHSUXIMIDE	rxcui:47858	METHSUXIMIDE	TRUE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	blocker	0.2019525816757481	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.01484106	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.2625383561784725	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:1782	iuphar.ligand:1782	UDP-GALACTOSE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.6168664383892681	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.42006137	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.4605936073306534	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.112919723	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
NCBIGENE:105	hgnc:227	ADARB2	GuideToPharmacology	2024.1	agonist	0.7955707762984016	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	PharmGKB	4/5/24	NULL	0.6886251965336985	avapritinib	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	0.1692703779358301	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:Q14627	hgnc:5975	IL13RA2	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	CINTREDEKIN BESUDOTOX	ncit:C2599	CINTREDEKIN BESUDOTOX	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9338	iuphar.ligand:9338	AM6538	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.1367387271762877	TIZATERKIB	ncit:C176765	TIZATERKIB	FALSE	FALSE	TRUE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.069454592	ICI 182780	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NCBIGENE:108	hgnc:233	ADCY2	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:9804	iuphar.ligand:9804	DERIVATIVE 17 [NAKAHATA ET AL., 2018]	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.011171845	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2892984641085096	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	WIN-62577	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.192335792	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.025298806	flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5125748858722557	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:11211	iuphar.ligand:11211	ZQ-16	FALSE	FALSE	FALSE
UNIPROT:P27707	hgnc:2704	DCK	TdgClinicalTrial	Jan-14	NULL	0.06714536	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.108040476	SIBUTRAMINE	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:45	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:6973	rxcui:36118	SALMON CALCITONIN	TRUE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.018860514	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003125457	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:9995	iuphar.ligand:9995	GNE-4997	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.4907258993990139	GW7604	chembl:CHEMBL1091137	CHEMBL:CHEMBL1091137	FALSE	FALSE	FALSE
TRH	hgnc:12298	TRH	NCI	14-Sep-17	NULL	0.6177373086552295	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.060008767	TREQUINSIN HYDROCHLORIDE	chembl:CHEMBL1256910	TREQUINSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.1159109740302306	QPI-1002	chembl:CHEMBL4297574	TEPRASIRAN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.004219178	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NCBIGENE:147	hgnc:278	ADRA1B	GuideToPharmacology	2024.1	agonist	0.2536602475154323	IUPHAR.LIGAND:3697	iuphar.ligand:3697	R-SPONDIN-1	FALSE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	4.773424657790408	AC-264613	iuphar.ligand:9460	AC264613	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.021697385	n-desmethylclozapine	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.6863747873946994	IL-1RA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.7395446652914718	CT-322	ncit:C62791	PEGDINETANIB	FALSE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.3509871071904712	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	0.1223955040459079	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.03574382	budesonide	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.058212496	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:5111	iuphar.ligand:5111	2-AMINO-4-METHYLPYRIDINE	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.2456499239096818	ONDANSETRON HYDROCHLORIDE	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	ChEMBL	33	inhibitor	1.151484018326633	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
UNIPROT:P04114	hgnc:603	APOB	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	MIPOMERSEN	rxcui:1367839	MIPOMERSEN	TRUE	FALSE	FALSE
NCBIGENE:1402	hgnc:736	NAAA	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9178	iuphar.ligand:9178	ARN726	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:8434	iuphar.ligand:8434	LP-12	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	activator	0.033658764	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1521961485092594	IUPHAR.LIGAND:4080	iuphar.ligand:4080	[3H]CGS19755	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1667	iuphar.ligand:1667	TIFLUADOM	FALSE	FALSE	FALSE
NCBIGENE:2455	hgnc:3852	FRA13C	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:10450	iuphar.ligand:10450	COMPOUND 7 [PMID: 31381331]	FALSE	FALSE	FALSE
LGR5	hgnc:4504	LGR5	CIViC	10-Apr-24	NULL	1.323722804261206	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
COL5A1	hgnc:2209	COL5A1	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	1.458546423213736	LEMBOREXANT	rxcui:2272403	LEMBOREXANT	TRUE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:7873	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.016856395	IUPHAR.LIGAND:965	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	FLUAZINAM	chembl:CHEMBL1878267	FLUAZINAM	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW780159X	chembl:CHEMBL365663	GW780159X	FALSE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	1.810609352954982	ABBV-428	ncit:C132681	ANTI-CD40/ANTI-MESOTHELIN BISPECIFIC ANTIBODY ABBV-428	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.079256862	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	PREDNISOLONE ACETATE	rxcui:34372	PREDNISOLONE ACETATE	TRUE	FALSE	FALSE
SENP2	hgnc:23116	SENP2	DTC	9/2/20	NULL	21.00306849	N-ETHYLMALEIMIDE	drugbank:DB02967	N-ETHYLMALEIMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.002645889	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005867434	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.066297565	Dyclonine	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8984	iuphar.ligand:8984	JNJ-39758979	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1339481409073839	TETRAHYDROZOLINE HYDROCHLORIDE	rxcui:57983	TETRAHYDROZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP11B1	hgnc:2591	CYP11B1	ChEMBL	33	inhibitor	0.9723642821424908	MITOTANE	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	NSC-636948	chembl:CHEMBL1998001	CHEMBL:CHEMBL1998001	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1583941817064691	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:1415	iuphar.ligand:1415	MPPG	FALSE	FALSE	FALSE
NCBIGENE:2396	hgnc:3907	FRA5C	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8612	iuphar.ligand:8612	COMPOUND 37 [PMID: 24418773]	FALSE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2441	iuphar.ligand:2441	SKF96365	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.5173169579871378	Refametinib	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.2094720926955897	Biperiden	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.072165573	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.009205412	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.043611023	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.3081436105381133	RAMUCIRUMAB	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.023004456	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2234368988752957	BENIDIPINE	ncit:C81680	BENIDIPINE	FALSE	FALSE	FALSE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	4.039051633514961	RO-4929097	chembl:CHEMBL4297422	RG-4733	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	ITASETRON	ncit:C65990	ITASETRON	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	NCI	14-Sep-17	NULL	0.2763561643983921	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	0.5048814541893701	Rilapladib	ncit:C76401	RILAPLADIB	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	CancerCommons	25-Jul-13	inhibitor	0.2263261691193728	STA-9090	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	CancerCommons	25-Jul-13	inhibitor	1.500219178	INC280	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	CancerCommons	25-Jul-13	inhibitor	1.225178995499538	ABT-888	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
CRBN	hgnc:30185	CRBN	CGI	2/1/22	NULL	2.917092846427472	Pomalidomide	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.03043923	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PRKCH	hgnc:9403	PRKCH	CGI	2/1/22	NULL	0.063645662	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CGI	2/1/22	NULL	0.118072806	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
VHL	hgnc:12687	VHL	CGI	2/1/22	NULL	0.1984416902331613	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.1411496538593938	TRIPROLIDINE HYDROCHLORIDE	rxcui:71534	TRIPROLIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2419708351875322	CETIRIZINE HYDROCHLORIDE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	DIPHENHYDRAMINE CITRATE	rxcui:82004	DIPHENHYDRAMINE CITRATE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.068436196	ADALIMUMAB	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
IGHE	hgnc:5522	IGHE	ChEMBL	33	inhibitor	2.187819634820604	OMALIZUMAB	rxcui:302379	OMALIZUMAB	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.8899605294185507	AZILSARTAN KAMEDOXOMIL	rxcui:1294597	AZILSARTAN KAMEDOXOMIL	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.546954909	DAPIPRAZOLE HYDROCHLORIDE	rxcui:235757	DAPIPRAZOLE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2792961235941196	GLYCOPYRROLATE	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
ALDH5A1	hgnc:408	ALDH5A1	ChEMBL	33	inhibitor	3.750547945	DIVALPROEX SODIUM	rxcui:266856	DIVALPROEX SODIUM	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.099446347	NEFAZODONE HYDROCHLORIDE	rxcui:236082	NEFAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.1491695205559502	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	2.187819634820604	FAMOTIDINE	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
GHR	hgnc:4263	GHR	ChEMBL	33	inhibitor	10.50153424713889	PEGVISOMANT	rxcui:278739	PEGVISOMANT	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	1.154014752432846	RIZATRIPTAN BENZOATE	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.075732218	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.064347636	NEFAZODONE HYDROCHLORIDE	rxcui:236082	NEFAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	0.4318065068724876	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	OXYCODONE TEREPHTHALATE	rxcui:159821	OXYCODONE TEREPHTHALATE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1691068316769549	METHYLPHENIDATE HYDROCHLORIDE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.1603287671318916	RIMEXOLONE	rxcui:55681	RIMEXOLONE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	FLUPREDNISOLONE	rxcui:4497	FLUPREDNISOLONE	TRUE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	agonist	0.3563869088395554	OXYTOCIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:2459	hgnc:3856	FRA15A	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:10450	iuphar.ligand:10450	COMPOUND 7 [PMID: 31381331]	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.062645859	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.2083637747448194	ROFLUMILAST	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.1785975212098452	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.1810609352954983	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.1013661606866689	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.2180551131050435	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.3125456621172291	ESOMEPRAZOLE SODIUM	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.3125456621172291	SYNTHETIC CONJUGATED ESTROGENS, B	rxcui:618365	SYNTHETIC CONJUGATED ESTROGENS, B	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.364636606	OMEPRAZOLE MAGNESIUM	rxcui:236486	OMEPRAZOLE MAGNESIUM	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.2083637747448194	DIETHYLSTILBESTROL DIPHOSPHATE	chembl:CHEMBL1200598	DIETHYLSTILBESTROL DIPHOSPHATE	TRUE	FALSE	FALSE
CA9	hgnc:1383	CA9	ChEMBL	33	inhibitor	0.2500365296937833	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
CA3	hgnc:1374	CA3	ChEMBL	33	inhibitor	0.8751278539282417	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.077789143	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.4375639269641209	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.2430910705356227	TAMSULOSIN HYDROCHLORIDE	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:11904	iuphar.ligand:11904	ZOMIRADOMIDE	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.2853677784548614	MIDODRINE HYDROCHLORIDE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.2536602475154323	TAMSULOSIN HYDROCHLORIDE	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.098451884	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	DICLOFENAC EPOLAMINE	rxcui:40968	DICLOFENAC EPOLAMINE	TRUE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.7001022831425934	SODIUM NITROPRUSSIDE	rxcui:9895	SODIUM NITROPRUSSIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.078136416	TETRAHYDROZOLINE HYDROCHLORIDE	rxcui:57983	TETRAHYDROZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.9053046764774912	TOLBUTAMIDE SODIUM, STERILE	chembl:CHEMBL1200874	TOLBUTAMIDE SODIUM, STERILE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.2715914029432474	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NCBIGENE:1700	hgnc:5974	IL13RA1	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:11770	iuphar.ligand:11770	EBLASAKIMAB	FALSE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	1.750255707856483	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
THRA	hgnc:11796	THRA	ChEMBL	33	agonist	1.875273972703375	DEXTROTHYROXINE	rxcui:3292	DEXTROTHYROXINE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.1848861663228679	BUPRENORPHINE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.1093909817410302	TELAPREVIR	rxcui:1102261	TELAPREVIR	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.3697723326457359	LEVALLORPHAN TARTRATE	rxcui:235419	LEVALLORPHAN TARTRATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.067839369	NEBIVOLOL HYDROCHLORIDE	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
GSC1	hgnc:4612	GSC	ChEMBL	33	inhibitor	10.50153424713889	ANIDULAFUNGIN	rxcui:341018	ANIDULAFUNGIN	TRUE	FALSE	FALSE
DIO1	hgnc:2883	DIO1	ChEMBL	33	inhibitor	5.250767124	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
COL4A1	hgnc:2202	COL4A1	ChEMBL	33	cleavage	0.3454452054979901	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
COL5A2	hgnc:2210	COL5A2	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	negative modulator	2.187819634820604	TICAGRELOR	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	agonist	0.3409589041278864	SUCCINYLCHOLINE CHLORIDE	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	negative modulator	0.050879526	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.091476779	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.055155117	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.052648066	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.056500364	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.096050618	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.024422173	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.023867123	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.025613498	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.024422173	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:1696	ncbigene:1696	DFNA19	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:10659	ncit:C131019	BEMPEGALDESLEUKIN	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.023336743	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.050879526	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.050879526	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.093763699	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.092988792	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.081365193	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.039598545	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.088396753	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.020656047	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.018819954	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	DIRITHROMYCIN	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1968	ncit:C76403	TAPROSTENE	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	inhibitor	0.6000876712650799	MUROMONAB-CD3	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	inhibitor	0.8334550989792776	MUROMONAB-CD3	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
POLA1	hgnc:9173	POLA1	ChEMBL	33	inhibitor	0.081030357	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
POLD1	hgnc:9175	POLD1	ChEMBL	33	inhibitor	0.054020238	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:5215	iuphar.ligand:5215	LUTEOLIN	FALSE	FALSE	FALSE
POLA2	hgnc:30073	POLA2	ChEMBL	33	inhibitor	0.092606122	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
POLD1	hgnc:9175	POLD1	ChEMBL	33	inhibitor	0.1286952726365061	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
NCBIGENE:674	ncbigene:674	BRAFPS1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:12460	rxcui:1310546	ACESULFAME	TRUE	FALSE	FALSE
POLE	hgnc:9177	POLE	ChEMBL	33	inhibitor	0.2763561643983921	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.039068208	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.055622533	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.1256164383629055	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.052090944	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.04464938	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:682	hgnc:1116	BSG	GuideToPharmacology	2024.1	agonist	0.3281729452230906	IUPHAR.LIGAND:6650	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.064624826	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.2586584789935689	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	SIMEPREVIR SODIUM	rxcui:1484518	SIMEPREVIR SODIUM	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.092606122	AFATINIB DIMALEATE	rxcui:1430441	AFATINIB DIMALEATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.062808219	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
MTNR1A	hgnc:7463	MTNR1A	ChEMBL	33	agonist	5.625821918110125	TASIMELTEON	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.1151484018326633	AFATINIB DIMALEATE	rxcui:1430441	AFATINIB DIMALEATE	TRUE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	0.4296082192011368	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
ITGA4	hgnc:6140	ITGA4	ChEMBL	33	inhibitor	5.834185692854944	VEDOLIZUMAB	rxcui:1538097	VEDOLIZUMAB	TRUE	FALSE	FALSE
PSMA7	hgnc:9536	PSMA7	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.1419126249613365	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
PSMC1	hgnc:9547	PSMC1	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMD13	hgnc:9558	PSMD13	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMB4	hgnc:9541	PSMB4	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMD2	hgnc:9559	PSMD2	ChEMBL	33	inhibitor	0.5385402178019948	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMD6	hgnc:9564	PSMD6	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMA8	hgnc:22985	PSMA8	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMD11	hgnc:9556	PSMD11	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMB10	hgnc:9538	PSMB10	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
RARB	hgnc:9865	RARB	ChEMBL	33	modulator	0.5147810905460244	MOFAROTENE	ncit:C63667	MOFAROTENE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.029235897	GSK2881078	iuphar.ligand:11151	GSK2881078	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1848861663228679	BMS-794833	chembl:CHEMBL3545119	BMS-794833	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	BMS-794833	chembl:CHEMBL3545119	BMS-794833	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.116943588	LGD-2941	chembl:CHEMBL467888	LGD-2941	FALSE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	ChEMBL	33	agonist	2.019525817	HYODEOXYCHOLIC_ACID	chembl:CHEMBL272621	HYODEOXYCHOLIC_ACID	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.5707355569097228	AC-430	drugbank:DB12535	AC-430	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.2397610558707511	AZD-7451	chembl:CHEMBL3545179	AZD-7451	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.5546584989686039	AZD-8055	drugbank:DB12774	AZD-8055	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	SC-80036	chembl:CHEMBL3544930	SC-80036	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.071780822	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.046303061	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.075768645	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.1562728310586145	IDOXIFENE	ncit:C1406	IDOXIFENE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	cleavage	0.6134073742487676	ELACESTRANT	rxcui:2628469	ELACESTRANT	TRUE	FALSE	TRUE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	1.381780822	LY2623091	chembl:CHEMBL3545275	LY2623091	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.222962511	ELOCALCITOL	drugbank:DB06194	ELOCALCITOL	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.4475085616678508	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2678962818147679	FRUQUINTINIB	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.2243917574174978	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PRKCI	hgnc:9404	PRKCI	ChEMBL	33	inhibitor	0.2625383561784725	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.1458546423213736	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	ChEMBL	33	inhibitor	0.1312691780892362	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.038159645	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.041672755	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
CHRM5	hgnc:1954	CHRM5	ChEMBL	33	inhibitor	0.2059124362184098	DAROTROPIUM BROMIDE	ncit:C76000	DAROTROPIUM BROMIDE	FALSE	FALSE	FALSE
MLNR	hgnc:4495	MLNR	ChEMBL	33	agonist	10.50153424713889	CAMICINAL	ncit:C166668	CAMICINAL	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	inhibitor	2.917092846427472	LY545694	chembl:CHEMBL3545161	LY545694	FALSE	FALSE	FALSE
CCR1	hgnc:1602	CCR1	ChEMBL	33	inhibitor	5.834185692854944	AZD4818	chembl:CHEMBL2178570	AZD4818	FALSE	FALSE	FALSE
CHRM4	hgnc:1953	CHRM4	ChEMBL	33	inhibitor	0.2778183663264258	AFACIFENACIN	ncit:C90741	AFACIFENACIN	FALSE	FALSE	FALSE
CHRM5	hgnc:1954	CHRM5	ChEMBL	33	inhibitor	0.1470803115845784	AFACIFENACIN	ncit:C90741	AFACIFENACIN	FALSE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	ChEMBL	33	inhibitor	3.580068493342807	NETAZEPIDE	ncit:C87692	NETAZEPIDE	FALSE	FALSE	FALSE
KCNB2	hgnc:6232	KCNB2	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.1682938180631233	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	ChEMBL	33	inhibitor	0.6250913242344582	ASM-024	chembl:CHEMBL3707249	ASM-024	FALSE	FALSE	FALSE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	blocker	0.075010959	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	modulator	0.1630673019742065	ASM-024	chembl:CHEMBL3707249	ASM-024	FALSE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	ChEMBL	33	blocker	0.047734247	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.1315981735230438	ASM-024	chembl:CHEMBL3707249	ASM-024	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.2263261691193728	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
ABCC9	hgnc:60	ABCC9	ChEMBL	33	potentiator	1.193356164447602	NAMINIDIL	ncit:C77076	NAMINIDIL	FALSE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	potentiator	0.6563458904461812	NAMINIDIL	ncit:C77076	NAMINIDIL	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	ChEMBL	33	inhibitor	0.2625383561784725	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.182318303	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.1798207919030633	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.130291988	MOMELOTINIB	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.1902451856365742	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
IL5	hgnc:6016	IL5	ChEMBL	33	inhibitor	17.50255707856483	RESLIZUMAB	rxcui:1746889	RESLIZUMAB	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	4.039051633514961	IXEKIZUMAB	rxcui:1745099	IXEKIZUMAB	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	1.334940794127826	AZILSARTAN	rxcui:1091642	AZILSARTAN MEDOXOMIL	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	negative modulator	0.2778183663264258	ESKETAMINE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	ChEMBL	33	agonist	0.7955707762984014	LARAZOTIDE ACETATE	ncit:C81670	LARAZOTIDE ACETATE	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	3.500511415712966	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
CASP8	hgnc:1509	CASP8	ChEMBL	33	inhibitor	3.500511415712966	NIVOCASAN	ncit:C98213	NIVOCASAN	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6300	iuphar.ligand:6300	CITRONELLAL	FALSE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	ChEMBL	33	inhibitor	1.640864726115453	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
PSEN1	hgnc:9508	PSEN1	ChEMBL	33	inhibitor	1.514644363	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	ChEMBL	33	positive modulator	3.750547945	FASIGLIFAM	ncit:C132780	FASIGLIFAM	FALSE	FALSE	FALSE
XPO1	hgnc:12825	XPO1	ChEMBL	33	inhibitor	5.250767123569449	SELINEXOR	rxcui:2178390	SELINEXOR	TRUE	FALSE	TRUE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9112	iuphar.ligand:9112	GIV3727	FALSE	FALSE	FALSE
ITGB5	hgnc:6160	ITGB5	ChEMBL	33	inhibitor	7.876150685354174	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.07631929	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:5994	iuphar.ligand:5994	JAK3 INHIBITOR IV	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	2.917092846427472	IBUTAMOREN MESYLATE	rxcui:1805437	IBUTAMOREN MESYLATE	TRUE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	7.001022831425932	ERENUMAB	rxcui:2045613	ERENUMAB	TRUE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	ChEMBL	33	inhibitor	0.6482428547616604	EPTINEZUMAB	rxcui:2282660	EPTINEZUMAB	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.3302369260106572	TEPROTUMUMAB	rxcui:2274802	TEPROTUMUMAB-TRBW	TRUE	FALSE	TRUE
CD4	hgnc:1678	CD4	ChEMBL	33	agonist	3.281729452230906	TREGALIZUMAB	ncit:C152722	TREGALIZUMAB	FALSE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	other/unknown	2.100306849	TUCOTUZUMAB CELMOLEUKIN	ncit:C2630	TUCOTUZUMAB CELMOLEUKIN	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	ChEMBL	33	inhibitor	1.591141552596803	CINPANEMAB	ncit:C169852	CINPANEMAB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.072927321	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	DIHYDROSTREPTOMYCIN SULFATE	rxcui:1549556	DIHYDROSTREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
IFNA8	hgnc:5429	IFNA8	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
IFNA2	hgnc:5423	IFNA2	ChEMBL	33	inhibitor	0.8078103267029924	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.007349898	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CD38	hgnc:1667	CD38	ChEMBL	33	inhibitor	5.834185692854944	HUMAX-IL15	chembl:CHEMBL2109468	HUMAX-IL15	FALSE	FALSE	FALSE
IFNA6	hgnc:5427	IFNA6	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	ChEMBL	33	inhibitor	0.067317527	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	ChEMBL	33	inhibitor	0.7001022831425933	FENFLURAMINE HYDROCHLORIDE	rxcui:82018	FENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TNNC1	hgnc:11943	TNNC1	ChEMBL	33	positive modulator	4.500657534	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.085796848	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	agonist	0.062065805	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.3889457128569963	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.031929262	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
SSTR4	hgnc:11333	SSTR4	ChEMBL	33	binder	1.750255707856483	LUTETIUM DOTATATE LU-177	chembl:CHEMBL3989924	LUTETIUM DOTATATE LU-177	TRUE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.062808219	IUPHAR.LIGAND:10316	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	binder	1.029562181092049	ANTI-TAC 90 Y-HAT	chembl:CHEMBL2109366	ANTI-TAC 90 Y-HAT	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	1.029562181092049	LUMRETUZUMAB	ncit:C104058	LUMRETUZUMAB	FALSE	FALSE	FALSE
FN1	hgnc:3778	FN1	ChEMBL	33	binder	4.039051633514961	MU-BC-1	chembl:CHEMBL2109529	MU-BC-1	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:9392	iuphar.ligand:9392	HG-10-102-01	FALSE	FALSE	FALSE
MSLN	hgnc:7371	MSLN	ChEMBL	33	binder	0.364636606	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
MSTN	hgnc:4223	MSTN	ChEMBL	33	inhibitor	2.187819634820604	PF-03446879	chembl:CHEMBL2109522	PF-03446879	FALSE	FALSE	FALSE
IL3RA	hgnc:6012	IL3RA	ChEMBL	33	binder	3.500511415712966	TAGRAXOFUSP	rxcui:2109054	TAGRAXOFUSP-ERZS	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.05814803	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.2397610558707511	LAROTRECTINIB SULFATE	rxcui:2104548	LAROTRECTINIB SULFATE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.2108741816694558	PEXIDARTINIB HYDROCHLORIDE	rxcui:2183103	PEXIDARTINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.108040476	PEXIDARTINIB HYDROCHLORIDE	rxcui:2183103	PEXIDARTINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.3804903712731485	PF-06651600	chembl:CHEMBL4085457	PF-06651600	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	inhibitor	0.029766254	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	inhibitor	0.031784305	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.024041974	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
HBA1	hgnc:4823	HBA1	ChEMBL	33	positive modulator	4.375639269641208	VOXELOTOR	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.020607406	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	1.016277507787635	UPADACITINIB	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.2853677784548614	FEDRATINIB HYDROCHLORIDE	rxcui:2197594	FEDRATINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1193356164447602	ESFLURBIPROFEN	ncit:C80544	ESFLURBIPROFEN	FALSE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	GEMIGLIPTIN	ncit:C118446	GEMIGLIPTIN	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.078136416	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.2453629496995069	LASOFOXIFENE	ncit:C80679	LASOFOXIFENE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	0.2051080907644316	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:9005	iuphar.ligand:9005	AR-M1000390	FALSE	FALSE	FALSE
SLC5A1	hgnc:11036	SLC5A1	ChEMBL	33	inhibitor	4.200613698855561	LICOGLIFLOZIN	ncit:C150375	LICOGLIFLOZIN	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.1491695205559502	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
ERG1	hgnc:6251	KCNH2	ChEMBL	33	inhibitor	0.074797252	LIRANAFTATE	ncit:C66019	LIRANAFTATE	FALSE	FALSE	FALSE
PTGER2	hgnc:9594	PTGER2	ChEMBL	33	agonist	3.281729452230906	OMIDENEPAG	rxcui:2612691	OMIDENEPAG	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	SITAFLOXACIN	ncit:C76922	SITAFLOXACIN	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.2263261691193728	PAZUFLOXACIN	ncit:C66331	PAZUFLOXACIN	FALSE	FALSE	FALSE
EGLN2	hgnc:14660	EGLN2	ChEMBL	33	inhibitor	4.200613698855561	VADADUSTAT	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	3.281729452230906	LAFUTIDINE	ncit:C79117	LAFUTIDINE	FALSE	FALSE	FALSE
NCBIGENE:2372	hgnc:3880	FRA1M	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8484	iuphar.ligand:8484	PEPTIDE KLK2B(C1)	FALSE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	ChEMBL	33	inhibitor	2.019525817	MARALIXIBAT	rxcui:2571074	MARALIXIBAT	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.2500365296937833	BENIDIPINE	ncit:C81680	BENIDIPINE	FALSE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	ChEMBL	33	inhibitor	0.4773424657790409	PELABRESIB	ncit:C188265	PELABRESIB	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.210030685	SAROGLITAZAR	ncit:C152303	SAROGLITAZAR	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
FGF1	hgnc:3665	FGF1	ChEMBL	33	agonist	2.917092846427472	FAZPILODEMAB	ncit:C188644	FAZPILODEMAB	FALSE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	1.250182648468916	VELDOREOTIDE	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.1750255707856483	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.8334550989792776	VELDOREOTIDE	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
SSTR4	hgnc:11333	SSTR4	ChEMBL	33	agonist	2.500365296937833	VELDOREOTIDE	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.064824285	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.1731022128649269	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.5834185692854945	ATACIGUAT	ncit:C79587	ATACIGUAT	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	ChEMBL	33	inhibitor	0.5135224570728067	IDH305	chembl:CHEMBL4167360	IDH305	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1682938180631233	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
GSC1	hgnc:4612	GSC	ChEMBL	33	inhibitor	10.50153424713889	IBREXAFUNGERP CITRATE	rxcui:2560215	IBREXAFUNGERP CITRATE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	modulator	1.721562991334245	VILAPRISAN	ncit:C148505	VILAPRISAN	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	ELRANATAMAB	rxcui:2644880	ELRANATAMAB	TRUE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	0.3889457128569963	ZILUCOPLAN	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
TPH1	hgnc:12008	TPH1	ChEMBL	33	inhibitor	13.12691780892362	RODATRISTAT ETHYL	ncit:C171781	RODATRISTAT ETHYL	FALSE	FALSE	FALSE
GCK	hgnc:4195	GCK	ChEMBL	33	activator	7.001022831425932	PF-04937319	drugbank:DB15009	PF-04937319	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.640864726115453	YM-543	chembl:CHEMBL2397450	YM-543	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	GLOFITAMAB	rxcui:2639782	GLOFITAMAB	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.050879526	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.42006137	LERIGLITAZONE	ncit:C170108	LERIGLITAZONE	FALSE	FALSE	FALSE
TNFRSF17	hgnc:11913	TNFRSF17	ChEMBL	33	binder	0.6908904109959803	ELRANATAMAB	rxcui:2644880	ELRANATAMAB	TRUE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.8751278539282416	RUNCACIGUAT	ncit:C166842	RUNCACIGUAT	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	0.7095631248066824	ELINZANETANT	ncit:C174774	ELINZANETANT	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.038104261	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.096167896	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1037701012563132	TRAZPIROBEN	ncit:C171664	TRAZPIROBEN	FALSE	FALSE	FALSE
MMP13	hgnc:7159	MMP13	ChEMBL	33	inhibitor	0.9376369863516874	CTS-1027	drugbank:DB08490	CTS-1027	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	ChEMBL	33	inhibitor	0.1121958787087489	ENCEQUIDAR	ncit:C111994	ENCEQUIDAR	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1000146118775133	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.053253216	IUPHAR.LIGAND:5688	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.08937476	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3314878234576672	XL518	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4475085616678508	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.375054795	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.5000730593875667	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1377250393067396	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.31919557	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	COSMIC	4-Sep-20	NULL	2.080014029626545	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
NCBIGENE:2372	hgnc:3880	FRA1M	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8672	iuphar.ligand:8672	HK2P01 DERIVATIVE KLK2 INHIBITOR	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	COSMIC	4-Sep-20	NULL	0.6667640791834221	PF-04217903	drugbank:DB12848	PF-04217903	FALSE	FALSE	TRUE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	0.6250913242344582	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	NSC-106547	chembl:CHEMBL223575	CHEMBL:CHEMBL223575	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.033615667	PROPAFENONE	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
NCBIGENE:973	hgnc:1698	CD79A	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4589	iuphar.ligand:4589	DIOA	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.053854022	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.034727296	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-4102	chembl:CHEMBL596836	CHEMBL:CHEMBL596836	FALSE	FALSE	FALSE
VCP	hgnc:12666	VCP	DTC	9/2/20	NULL	0.4268916360625569	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ERGOCALCIFEROL	rxcui:4018	ERGOCALCIFEROL	TRUE	FALSE	FALSE
ANXA2	hgnc:537	ANXA2	DTC	9/2/20	NULL	1.500219178	N-ETHYLMALEIMIDE	drugbank:DB02967	N-ETHYLMALEIMIDE	FALSE	FALSE	FALSE
NCBIGENE:2757	hgnc:23177	KEAP1	GuideToPharmacology	2024.1	NULL	2.100306849	IUPHAR.LIGAND:10487	iuphar.ligand:10487	RA839	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	DTC	9/2/20	NULL	0.7143900848393808	PHILANTHOTOXIN 343	chembl:CHEMBL16117	PHILANTHOTOXIN 343	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.012364929	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	GNF-PF-4012	chembl:CHEMBL584269	CHEMBL:CHEMBL584269	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.008704853	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	1,3-DIPROPYL-8-CYCLOPENTYLXANTHINE [DPCPX]	iuphar.ligand:386	DPCPX	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	NSC-50690	chembl:CHEMBL1388703	CHEMBL:CHEMBL1388703	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.02339914	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	0.3070624048871023	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	GNF-PF-2906	chembl:CHEMBL579957	CHEMBL:CHEMBL579957	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.018699313	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.1442518440541058	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	DNDI1416917	chembl:CHEMBL1335833	CHEMBL:CHEMBL1335833	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.03574382	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.004419838	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.2524407270946851	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	CYSTAMINE DIHYDROCHLORIDE	ncit:C97356	CYSTAMINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.3500511415712966	TCMDC-123516	chembl:CHEMBL547304	CHEMBL:CHEMBL547304	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1193356164447602	DNDI1383301	chembl:CHEMBL1509103	CHEMBL:CHEMBL1509103	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	1.491695205559502	CARTEOLOL	rxcui:2116	CARTEOLOL	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	BIX-01294	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.063722902	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	DTC	9/2/20	NULL	0.1315981735230438	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.7501095890813501	DNDI1416917	chembl:CHEMBL1335833	CHEMBL:CHEMBL1335833	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.02075402	IUPHAR.LIGAND:5703	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	CID 1225609	chembl:CHEMBL444376	CHEMBL:CHEMBL444376	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	SPIPERONE	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	SIB-1893	iuphar.ligand:1432	SIB-1893	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.005151852	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	SJ000193360	chembl:CHEMBL607253	CHEMBL:CHEMBL607253	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.212581665	GNF-PF-4510	chembl:CHEMBL586024	CHEMBL:CHEMBL586024	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	GERONTOXANTHONE I	chembl:CHEMBL478791	GERONTOXANTHONE I	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.053038052	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-108	chembl:CHEMBL578929	CHEMBL:CHEMBL578929	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.006943622	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.067317527	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013887244	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	1-AMINOBENZOTRIAZOLE	chembl:CHEMBL101168	CHEMBL:CHEMBL101168	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.036162308	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2273059360852575	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.2625383561784725	SJ000029259	chembl:CHEMBL592558	CHEMBL:CHEMBL592558	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2651902587661338	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1704794520639431	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002542252	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.021501913	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2220197515251353	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2580229544751573	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	NSC-699479	chembl:CHEMBL1701915	CHEMBL:CHEMBL1701915	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	DEXTROMETHORPHAN HYDROBROMIDE MONOHYDRATE	chembl:CHEMBL1256818	DEXTROMETHORPHAN HYDROBROMIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	GW405833	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.053854022	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.1389091831632129	METHYLCURCUMIN	chembl:CHEMBL494826	METHYLCURCUMIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.077789143	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.0023813	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.041508041	IUPHAR.LIGAND:5712	iuphar.ligand:5712	SU-14813	FALSE	FALSE	FALSE
MMP14	hgnc:7160	MMP14	DTC	9/2/20	NULL	0.300043836	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.007631929	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	BUTANE-2,3-DIONE MONOOXIME	chembl:CHEMBL335741	CHEMBL:CHEMBL335741	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.072324616	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	3.000438356	AMBROXOL	rxcui:625	AMBROXOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.018301733	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.028413242	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.011124507	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.2546668357992238	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	E1501	chembl:CHEMBL1233714	E1501	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	MECLOFENAMATE SODIUM	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	1.093909817410302	EMTRICITABINE	rxcui:276237	EMTRICITABINE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	HERBIMYCIN	ncit:C1124	HERBIMYCIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.035358701	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	LOFEPRAMINE	rxcui:6465	LOFEPRAMINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.026858144	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	DIMETHYL SUCCINATE	rxcui:2393581	DIMETHYL SUCCINATE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1232574442152452	ZOLANTIDINE	chembl:CHEMBL419296	ZOLANTIDINE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	NOMIFENSINE MALEATE	rxcui:262302	NOMIFENSINE MALEATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.079557078	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.096167896	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.072524408	(+)-TAXIFOLIN	chembl:CHEMBL66	(+)-TAXIFOLIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002213645	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
AMOT	hgnc:17810	AMOT	DTC	9/2/20	NULL	11.66837138570989	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	GAMOLENIC ACID	rxcui:25605	GAMMA-LINOLENIC ACID	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.075010959	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	ACRYLAMIDE	rxcui:1368125	ACRYLAMIDE	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2580229544751573	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	0.5303805175322677	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	2-MERCAPTONICOTINIC ACID	chembl:CHEMBL1521174	2-MERCAPTONICOTINIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	NSC-747267	chembl:CHEMBL610767	CHEMBL:CHEMBL610767	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1773907812016706	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	PIRARUBICIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DIMETHYLPHENYLPIPERAZINIUM IODIDE	chembl:CHEMBL47814	DIMETHYLPHENYLPIPERAZINIUM IODIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009309871	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	1.640864726115453	NSC-119911	chembl:CHEMBL502775	CHEMBL:CHEMBL502775	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	SJ000001516	chembl:CHEMBL592316	CHEMBL:CHEMBL592316	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.014658758	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.023482858	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.033401826	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.3621218705909966	ALOSETRON HYDROCHLORIDE	rxcui:85247	ALOSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.085239726	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	DTC	9/2/20	NULL	1.400204566285186	ISOSILYBIN B	chembl:CHEMBL3542340	ISOSILYBIN B	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	chembl:CHEMBL1226	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	VUF-5574	iuphar.ligand:3280	VUF5574	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	TOREMIFENE CITRATE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	1.750255707856483	NSC-176327	chembl:CHEMBL363332	CHEMBL:CHEMBL363332	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	SJ000114741	chembl:CHEMBL591370	CHEMBL:CHEMBL591370	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.5250767123569451	ALOSETRON HYDROCHLORIDE	rxcui:85247	ALOSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004889893	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:10222	iuphar.ligand:10222	TAK-448	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	GNF-PF-3237	chembl:CHEMBL602206	CHEMBL:CHEMBL602206	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.375054795	MORACIN M	chembl:CHEMBL512578	MORACIN M	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.048708415	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	ONONETIN	chembl:CHEMBL241858	ONONETIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	BENFLUOREX HYDROCHLORIDE	rxcui:235953	BENFLUOREX HYDROCHLORIDE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	1.500219178	NSC-50650	chembl:CHEMBL1561747	CHEMBL:CHEMBL1561747	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.012504804	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	HYDROXYPROGESTERONE	ncit:C87242	HYDROXYPROGESTERONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ESTRADIOL PHOSPHATE	chembl:CHEMBL1642763	ESTRADIOL PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:6043	drugbank:DB08009	SU-11652	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.056581542	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	OXYBENZONE	rxcui:32673	OXYBENZONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00292359	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.043109746	FLUORESCEIN	rxcui:25138	FLUORESCEIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001359809	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.3125456621172291	GAMOLENIC ACID	rxcui:25605	GAMMA-LINOLENIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV006169	chembl:CHEMBL597248	CHEMBL:CHEMBL597248	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006434764	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:11868	iuphar.ligand:11868	BEZUCLASTINIB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.01351201	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.010819631	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.3977853881492007	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1363835616511545	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.022439176	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE	chembl:CHEMBL1513686	12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.020383413	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	TREQUINSIN HYDROCHLORIDE	chembl:CHEMBL1256910	TREQUINSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	6-CHLOROMELATONIN	iuphar.ligand:1346	6-CL-MLT	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:12357	ncit:C180833	ELENESTINIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	SJ000047241	chembl:CHEMBL601933	CHEMBL:CHEMBL601933	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	2,2,3,3,4,4,5,5,6,6,7,7,8,8,9,9,9-HEPTADECAFLUORO-NONANOIC ACID	chembl:CHEMBL426404	CHEMBL:CHEMBL426404	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE	chembl:CHEMBL1513686	12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE	FALSE	FALSE	FALSE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.1164249916534246	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.028004091	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.1355619739303644	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	4-(HEXYLOXY)PHENOL	chembl:CHEMBL225563	CHEMBL:CHEMBL225563	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.007349898	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	TCMDC-124063	chembl:CHEMBL534535	CHEMBL:CHEMBL534535	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:5712	iuphar.ligand:5712	SU-14813	FALSE	FALSE	FALSE
GZMB	hgnc:4709	GZMB	DTC	9/2/20	NULL	0.5122699632750682	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.010539476	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	GNF-PF-2356	chembl:CHEMBL601547	CHEMBL:CHEMBL601547	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	TCMDC-124307	chembl:CHEMBL546865	CHEMBL:CHEMBL546865	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	ETHYL NITRITE [SPIRIT]	chembl:CHEMBL1551365	ETHYL NITRITE [SPIRIT]	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	2.625383561784724	IUPHAR.LIGAND:2319	iuphar.ligand:2319	TAMAPIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	DEXMEDETOMIDINE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.009571212	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.032312413	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
GABRR1	hgnc:4090	GABRR1	DTC	9/2/20	NULL	0.3125456621172291	ISONIPECOTIC ACID	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	CYSTEINE METHYL-ESTER HCL	chembl:CHEMBL1426508	CHEMBL:CHEMBL1426508	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007003824	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.2548916079402645	2,2,3,3,4,4,5,5,6,6,7,7,8,8,9,9,9-HEPTADECAFLUORO-NONANOIC ACID	chembl:CHEMBL426404	CHEMBL:CHEMBL426404	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.098451884	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2317	iuphar.ligand:2317	NS309	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.049349315	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.1084869240406911	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
NEU3	hgnc:7760	NEU3	DTC	9/2/20	NULL	52.50767123569449	OSELTAMIVIR	rxcui:259275	OSELTAMIVIR PHOSPHATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	SJ000281118	chembl:CHEMBL592561	CHEMBL:CHEMBL592561	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.085239726	AMINACRINE HYDROCHLORIDE	rxcui:81949	AMINACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.00767656	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	activator	1.875273972703375	IUPHAR.LIGAND:2395	ncit:C152558	TENIDAP	FALSE	FALSE	FALSE
HIF1AN	hgnc:17113	HIF1AN	DTC	9/2/20	NULL	17.50255707856483	L-4-THIOPROLINE	chembl:CHEMBL1800368	CHEMBL:CHEMBL1800368	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.020117882	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.046590658	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PBK	hgnc:18282	PBK	DTC	9/2/20	NULL	0.1591141552596803	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007374673	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	CID 3238892	chembl:CHEMBL261118	CHEMBL:CHEMBL261118	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002712173	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.014222013	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
NCBIGENE:433	hgnc:743	ASGR2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.03591496	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	1.221108633388244	SJ000291864	chembl:CHEMBL592566	CHEMBL:CHEMBL592566	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.019107595	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	ALOSETRON HYDROCHLORIDE	rxcui:85247	ALOSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	TREQUINSIN HYDROCHLORIDE	chembl:CHEMBL1256910	TREQUINSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:442	hgnc:755	ASNSP2	GuideToPharmacology	2024.1	inhibitor	0.4526523382387457	IUPHAR.LIGAND:2414	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
UTS2R	hgnc:4468	UTS2R	DTC	9/2/20	NULL	5.431828058864948	URANTIDE	iuphar.ligand:2167	URANTIDE	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	1.129197231	CEFMETAZOLE	rxcui:2182	CEFMETAZOLE	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.3547815624033412	2-PHENYLACETYLAMINOBENZOTHIAZOLE	chembl:CHEMBL1405979	CHEMBL:CHEMBL1405979	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	GNF-PF-2356	chembl:CHEMBL601547	CHEMBL:CHEMBL601547	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2507	iuphar.ligand:2507	CLOFILIUM	FALSE	FALSE	FALSE
MSTN	hgnc:4223	MSTN	DTC	9/2/20	NULL	0.4861821410712454	SB-431542	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	FURAMIDINE	chembl:CHEMBL24057	FURAMIDINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	LEUCINE	rxcui:6308	LEUCINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003668018	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	ACRIDIN-1-YLAMINE	chembl:CHEMBL146525	CHEMBL:CHEMBL146525	FALSE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.079557078	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	TRIAZOPHOS	ncit:C163712	TRIAZOPHOS	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
NCBIGENE:1243	ncbigene:1243	CMM	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:5114	iuphar.ligand:5114	3-CHLOROTYROSINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	2.500365296937833	ETHYL 2,4,6-TRIHYDROXYBENZOATE	chembl:CHEMBL2204435	CHEMBL:CHEMBL2204435	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	NECROSTATIN	iuphar.ligand:9750	NECROSTATIN-1	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.036212187	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.020296742	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.034830959	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.07182992	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.03251249	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.019361236	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SEROTONIN HYDROCHLORIDE	rxcui:1356129	SEROTONIN HYDROCHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	GALANTAMINE HYDROBROMIDE	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.007489327	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.01036063	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.1060761035064535	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12524	iuphar.ligand:12524	COMPOUND 66 [PMID: 36126387]	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	ETHYLISOTHIOUREA	chembl:CHEMBL321691	ETHYLISOTHIOUREA	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.08334551	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.01160647	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	FPL-64176	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	PHENAMIL METHANESULFONATE	chembl:CHEMBL1256775	PHENAMIL METHANESULFONATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	XANTHONE	chembl:CHEMBL186784	XANTHONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.222962511	TRICIFEROL	chembl:CHEMBL1164992	TRICIFEROL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	4-AMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL60824	4-AMINO-[1,2]NAPHTHOQUINONE	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.596678082	BENZANTHRONE	chembl:CHEMBL1607517	BENZANTHRONE	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.3182283105193606	6-AZAURIDINE	ncit:C291	6-AZAURIDINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1810609352954982	PROCATEROL HYDROCHLORIDE	rxcui:58918	PROCATEROL HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:5126	iuphar.ligand:5126	6-FLUOROTRYPTOPHAN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	HALOBETASOL PROPIONATE	rxcui:41208	HALOBETASOL	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.026045472	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	LEUCINE	rxcui:6308	LEUCINE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.012056871	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.004930298	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.033919684	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	SJ000111875	chembl:CHEMBL590949	CHEMBL:CHEMBL590949	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.1646008502686348	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GERONTOXANTHONE I	chembl:CHEMBL478791	GERONTOXANTHONE I	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	DTC	9/2/20	NULL	0.1469979597863787	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
NCBIGENE:1242	hgnc:20692	TPH2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5240	ncit:C81112	FENCLONINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00517674	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.049256727	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	ISOQUINOLINE-3-CARBOXYLIC ACID	chembl:CHEMBL1728638	CHEMBL:CHEMBL1728638	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.002976625	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002088278	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001535581	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	TYRPHOSTIN 1	iuphar.ligand:5917	AG 9	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.7395446652914718	CANTHIN-6-ONE	chembl:CHEMBL156897	CANTHIN-6-ONE	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.4861821410712453	CID 4970947	chembl:CHEMBL1451921	CHEMBL:CHEMBL1451921	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.3302369260106572	GNF-PF-2906	chembl:CHEMBL579957	CHEMBL:CHEMBL579957	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	TCMDC-124063	chembl:CHEMBL534535	CHEMBL:CHEMBL534535	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	1.458546423213736	TCMDC-123591	chembl:CHEMBL588234	CHEMBL:CHEMBL588234	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	NSC-116702	chembl:CHEMBL1477383	CHEMBL:CHEMBL1477383	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	ETIDRONIC ACID	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.01274458	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
NCBIGENE:2853	hgnc:4486	GPR31	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10486	iuphar.ligand:10486	COMPOUND 21B [PMID: 31430136]	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005424346	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	WIN-62577	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.03251249	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	0.1151484018326633	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	DICYCLOMINE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TRIPHENYLBISMUTHINE	chembl:CHEMBL203014	TRIPHENYLBISMUTHINE	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:9360	iuphar.ligand:9360	KU-0063794	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.3211478363039418	Z160	iuphar.ligand:7765	NP118809	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.015498132	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	PIRENPERONE	ncit:C66417	PIRENPERONE	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	DTC	9/2/20	NULL	0.090843722	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	LOTEPREDNOL ETABONATE	rxcui:237027	LOTEPREDNOL	TRUE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.577007376	2,6-DIMETHOXYQUINONE	chembl:CHEMBL448515	2,6-DIMETHOXYQUINONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.015791781	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:9837	iuphar.ligand:9837	CZ415	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.192335792	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NSC-74429	chembl:CHEMBL1269022	CHEMBL:CHEMBL1269022	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003632492	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.044198376	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.01763778	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.008458066	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	[14C]-TACRINE MONOHYDRATE MONOHYDROCHLORIDE	chembl:CHEMBL1337960	CHEMBL:CHEMBL1337960	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TCMDC-125810	chembl:CHEMBL528119	CHEMBL:CHEMBL528119	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	RS-16566	chembl:CHEMBL145725	CHEMBL:CHEMBL145725	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	DEXKETOPROFEN	rxcui:237162	DEXKETOPROFEN	TRUE	FALSE	FALSE
NCBIGENE:3181	hgnc:5033	HNRNPA2B1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11529	iuphar.ligand:11529	STM2457	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.059397818	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.097236428	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.022108493	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.021590325	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	2.100306849	NAPHTHALENE-1,2-DIOL	drugbank:DB07610	1,2-DIHYDROXYNAPHTHALENE	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.2059124362184097	IUPHAR.LIGAND:11869	ncit:C162676	ELZOVANTINIB	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004540811	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	TCMDC-125180	chembl:CHEMBL586163	CHEMBL:CHEMBL586163	FALSE	FALSE	FALSE
PPM1D	hgnc:9277	PPM1D	DTC	9/2/20	NULL	0.7001022831425933	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003646366	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:3372	iuphar.ligand:3372	CBIPES	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.1581556362520918	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GNF-PF-108	chembl:CHEMBL578929	CHEMBL:CHEMBL578929	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	BISANHYDRORUTILANTINONE	chembl:CHEMBL1436035	BISANHYDRORUTILANTINONE	FALSE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	2.500365296937833	GSK9772	iuphar.ligand:8693	GSK9772	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	(-)-GRACILIOETHER C	chembl:CHEMBL2178583	CHEMBL:CHEMBL2178583	FALSE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	DTC	9/2/20	NULL	6.300920548	(+)-[3H]-PENTAZOCINE	iuphar.ligand:6683	[3H]PENTAZOCINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004427291	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.3125456621172291	LESCOL	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.760980743	SILYBIN B	chembl:CHEMBL592675	SILYBIN B	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002229625	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	DIHYDROERGOCRISTINE	rxcui:3416	DIHYDROERGOCRISTINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.071341945	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.4134462302023188	HYPERFORIN	drugbank:DB01892	HYPERFORIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.052824619	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	3-FLUOROEVODIAMINE	chembl:CHEMBL2171781	CHEMBL:CHEMBL2171781	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	EFAROXAN	ncit:C72923	EFAROXAN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	PROCHLORAZ	chembl:CHEMBL522782	PROCHLORAZ	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	UH-301	iuphar.ligand:61	(S)-UH 301	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.069824031	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	OLOMOUCINE	drugbank:DB02116	OLOMOUCINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003632995	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.014634245	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.009318132	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003279475	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.038159645	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	SJ000029259	chembl:CHEMBL592558	CHEMBL:CHEMBL592558	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	NSC-117079	chembl:CHEMBL471225	CHEMBL:CHEMBL471225	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.1458546423213736	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	MOSAPRAMINE	ncit:C66203	MOSAPRAMINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	GNF-PF-4864	chembl:CHEMBL583558	CHEMBL:CHEMBL583558	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665929	chembl:CHEMBL584841	CHEMBL:CHEMBL584841	FALSE	FALSE	FALSE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.280789686	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	(R)-PINOCEMBRIN	chembl:CHEMBL399249	(R)-PINOCEMBRIN	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.7778914257139926	DIHYDROTANSHINONE I	chembl:CHEMBL227075	DIHYDROTANSHINONE I	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001169436	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	DIBENZ[A,H]ANTHRACENE	chembl:CHEMBL1346946	DIBENZ[A,H]ANTHRACENE	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.8899605294185507	2-PYRIDYLCARBOXALDEHYDE P-BROMOBENZOYLHYDRAZONE	chembl:CHEMBL400912	CHEMBL:CHEMBL400912	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.008832241	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00506733	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.036212187	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007841647	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	RO-106-9920	chembl:CHEMBL271023	CHEMBL:CHEMBL271023	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004557958	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.015599427	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.3621218705909966	TCMDC-124381	chembl:CHEMBL579919	CHEMBL:CHEMBL579919	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.008651783	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.2651902587661338	IOXYNIL	chembl:CHEMBL509523	IOXYNIL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.057073556	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.1548898856510162	GNF-PF-4579	chembl:CHEMBL584626	CHEMBL:CHEMBL584626	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	FLUORESCEIN	rxcui:25138	FLUORESCEIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	MANUMYCIN A	chembl:CHEMBL285848	MANUMYCIN A	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	EXISULIND	ncit:C1239	EXISULIND	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.030038714	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.047432404	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
FGF22	hgnc:3679	FGF22	DTC	9/2/20	NULL	0.1875273972703375	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	BUTANE-2,3-DIONE MONOOXIME	chembl:CHEMBL335741	CHEMBL:CHEMBL335741	FALSE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	DTC	9/2/20	NULL	0.066297565	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	1.093909817410302	GONIOTHALAMIN	chembl:CHEMBL464443	GONIOTHALAMIN	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	0.080042182	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1848861663228679	N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL199592	CHEMBL:CHEMBL199592	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001580319	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	0.3281729452230906	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.022201975	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	PROPANTHELINE BROMIDE	rxcui:8762	PROPANTHELINE BROMIDE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	N6-BENZYLADENOSINE	chembl:CHEMBL388757	N6-BENZYLADENOSINE	FALSE	FALSE	FALSE
GLI1	hgnc:4317	GLI1	DTC	9/2/20	NULL	1.166837138570989	BETULINIC ACID	ncit:C38126	BETULINIC ACID	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	SJ000117447	chembl:CHEMBL592611	CHEMBL:CHEMBL592611	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	DTC	9/2/20	NULL	0.4296082192011368	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1415301111474245	GNF-PF-107	chembl:CHEMBL578675	CHEMBL:CHEMBL578675	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	CID 1540545	chembl:CHEMBL259784	CHEMBL:CHEMBL259784	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1902451856365742	MECHLORETHAMINE HYDROCHLORIDE	rxcui:155036	MECHLORETHAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.086361301	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	NSC-724440	chembl:CHEMBL515617	CHEMBL:CHEMBL515617	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	GNF-PF-4481	chembl:CHEMBL597251	CHEMBL:CHEMBL597251	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	ISOETHARINE MESYLATE	rxcui:6024	ISOETHARINE MESYLATE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.093098708	PHENAMIL METHANESULFONATE	chembl:CHEMBL1256775	PHENAMIL METHANESULFONATE	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.1902451856365742	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	PENFLURIDOL	rxcui:7974	PENFLURIDOL	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	4.039051633514961	PD-194035	chembl:CHEMBL415893	CHEMBL:CHEMBL415893	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	BENOMYL	chembl:CHEMBL327919	BENOMYL	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.035358701	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.047432404	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	THIOLACTOMYCIN	drugbank:DB04302	4-HYDROXY-3,5-DIMETHYL-5-(2-METHYL-BUTA-1,3-DIENYL)-5H-THIOPHEN-2-ONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.000772808	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.546954909	PIRENPERONE	ncit:C66417	PIRENPERONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001656812	FLUFENAMIC ACID	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009320613	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.066676408	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	TCMDC-123748	chembl:CHEMBL530609	CHEMBL:CHEMBL530609	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.099071078	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2917092846427472	DIPHENYLUREA	chembl:CHEMBL354676	DIPHENYLUREA	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007063179	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	DTC	9/2/20	NULL	1.591141552596802	L-655708	chembl:CHEMBL52030	CHEMBL:CHEMBL52030	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	2.282942227638891	NEOCHAMAEJASMIN A	chembl:CHEMBL452374	NEOCHAMAEJASMIN A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	IOXYNIL	chembl:CHEMBL509523	IOXYNIL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	2-AMINOBIPHENYL	chembl:CHEMBL296021	CHEMBL:CHEMBL296021	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	SJ000111875	chembl:CHEMBL590949	CHEMBL:CHEMBL590949	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.019724895	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	SCOULERINE	chembl:CHEMBL1235966	SCOULERINE	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	DTC	9/2/20	NULL	2.500365296937833	NSC-613604	chembl:CHEMBL572637	CHEMBL:CHEMBL572637	FALSE	FALSE	FALSE
SPSB2	hgnc:29522	SPSB2	DTC	9/2/20	NULL	52.50767123569449	PHENYLTHIAZOL-2-AMINE	chembl:CHEMBL175296	CHEMBL:CHEMBL175296	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	SJ000202381	chembl:CHEMBL591598	CHEMBL:CHEMBL591598	FALSE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	DTC	9/2/20	NULL	0.055271233	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	CITALOPRAM HYDROBROMIDE	rxcui:221078	CITALOPRAM HYDROBROMIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	GNF-PF-3125	chembl:CHEMBL534288	CHEMBL:CHEMBL534288	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-124316	chembl:CHEMBL534214	CHEMBL:CHEMBL534214	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.011355465	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	NSC-128437	chembl:CHEMBL1370698	CHEMBL:CHEMBL1370698	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003439517	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.012067955	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	DIPROPYLDOPAMINE HYDROBROMIDE	chembl:CHEMBL1255747	DIPROPYLDOPAMINE HYDROBROMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	TEBUFENOZIDE	chembl:CHEMBL226968	TEBUFENOZIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	NCG-C00094408-01	chembl:CHEMBL1256885	CHEMBL:CHEMBL1256885	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	NSC-37173	chembl:CHEMBL221733	CHEMBL:CHEMBL221733	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.018225502	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	DICYCLOMINE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	CID 1540951	chembl:CHEMBL259421	CHEMBL:CHEMBL259421	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	FENOLDOPAM BROMIDE	chembl:CHEMBL1256646	FENOLDOPAM BROMIDE	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.2958178661165888	AKT INHIBITOR VIII	iuphar.ligand:5921	AKT INHIBITOR VIII	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.1193356164447602	SALMETEROL	rxcui:36117	SALMETEROL	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1238388472539964	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	NIRIDAZOLE	ncit:C90757	NIRIDAZOLE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DNDI1417254	chembl:CHEMBL2094567	CHEMBL:CHEMBL2094567	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.00453826	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
PRKAG1	hgnc:9385	PRKAG1	DTC	9/2/20	NULL	1.795134059339982	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MILBEMYCIN A4	chembl:CHEMBL2272397	MILBEMYCIN A4	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FENOVERINE	rxcui:24855	FENOVERINE	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.1491695205559502	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002088278	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	OLOMOUCINE	drugbank:DB02116	OLOMOUCINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	GNF-PF-107	chembl:CHEMBL578675	CHEMBL:CHEMBL578675	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	GNF-PF-4945	chembl:CHEMBL585628	CHEMBL:CHEMBL585628	FALSE	FALSE	FALSE
PRKAG1	hgnc:9385	PRKAG1	DTC	9/2/20	NULL	5.000730593875666	SAPONARIN	chembl:CHEMBL538921	SAPONARIN	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.112919723	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.013505059	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	DTC	9/2/20	NULL	1.363835616511545	SAPONARIN	chembl:CHEMBL538921	SAPONARIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	GNF-PF-2844	chembl:CHEMBL576353	CHEMBL:CHEMBL576353	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.2763561643983921	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	TCMDC-123927	chembl:CHEMBL531268	CHEMBL:CHEMBL531268	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1286952726365061	RS-16566	chembl:CHEMBL145725	CHEMBL:CHEMBL145725	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002719055	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.070010228	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.068191781	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	6-AMINONICOTINAMIDE	ncit:C38127	6-AMINONICOTINAMIDE	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	DTC	9/2/20	NULL	1.544343271638073	TURBINATINE	chembl:CHEMBL452240	TURBINATINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	ANISOCOUMARIN H	chembl:CHEMBL408980	ANISOCOUMARIN H	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ESTRADIOL PROPIONATE	chembl:CHEMBL2356687	ESTRADIOL PROPIONATE	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.189216833	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	N-BENZOYLANTHRANILIC ACID	chembl:CHEMBL198666	CHEMBL:CHEMBL198666	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	CEFOTAXIME	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1750255707856483	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	chembl:CHEMBL1226	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.023759127	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	CID 2093195	chembl:CHEMBL411085	CHEMBL:CHEMBL411085	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	WIN-62577	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	MOCLOBEMIDE	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	(2-NITROVINYL)BENZENE	chembl:CHEMBL230156	(2-NITROVINYL)BENZENE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	SJ000149318	chembl:CHEMBL600662	CHEMBL:CHEMBL600662	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.041872146	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	GERANIOL	rxcui:1368875	GERANIOL	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.036212187	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-300014A	chembl:CHEMBL475599	GSK-300014A	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	2-PHENYLPHENOL	rxcui:236677	2-PHENYLPHENOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.034888818	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.026519026	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.007114861	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	SJ000117447	chembl:CHEMBL592611	CHEMBL:CHEMBL592611	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.071439008	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001144706	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	REL-HUEAFURANOID A	chembl:CHEMBL2207339	CHEMBL:CHEMBL2207339	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	GNF-PF-3799	chembl:CHEMBL597244	CHEMBL:CHEMBL597244	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.1981421556063943	DNDI1417368	chembl:CHEMBL2094652	CHEMBL:CHEMBL2094652	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	N-DESMETHYLCLOZAPINE	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006987979	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	7-O-ACETYLAFROMOSIN	chembl:CHEMBL446567	CHEMBL:CHEMBL446567	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	NALIDIXATE SODIUM	ncit:C80641	NALIDIXATE SODIUM	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005669763	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.11707396	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.006614723	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001180611	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	ETHYLNOREPINEPHRINE HYDROCHLORIDE	rxcui:289080	ETHYLNOREPINEPHRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	NSC-50690	chembl:CHEMBL1388703	CHEMBL:CHEMBL1388703	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	DTC	9/2/20	NULL	0.015002192	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	OCTADEC-17-YNOIC ACID	iuphar.ligand:8851	17-OCTADECYNOIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
PRMT1	hgnc:5187	PRMT1	DTC	9/2/20	NULL	2.625383561784725	FURAMIDINE	chembl:CHEMBL24057	FURAMIDINE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.041182487	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.030598876	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
ADRBK1	hgnc:289	GRK2	DTC	9/2/20	NULL	0.6731752722524936	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.016992774	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	CORALYNE	chembl:CHEMBL363506	CORALYNE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	SJ000121255	chembl:CHEMBL590422	CHEMBL:CHEMBL590422	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	ONONETIN	chembl:CHEMBL241858	ONONETIN	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.1458546423213736	SB-431542	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CID 1225609	chembl:CHEMBL444376	CHEMBL:CHEMBL444376	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.021742307	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	METHOXSALEN	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.021301287	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	0.6213925590023018	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.006460892	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.001341192	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	P-CYANOCHALCONE	chembl:CHEMBL445153	CHEMBL:CHEMBL445153	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.003806283	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2187819634820604	DIMETHYL YELLOW	chembl:CHEMBL263116	DIMETHYL YELLOW	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.007649719	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007699637	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1290114772375786	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.090064616	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ERGOCALCIFEROL	rxcui:4018	ERGOCALCIFEROL	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.02832129	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1056492378987816	TETROQUINONE	chembl:CHEMBL1329029	TETROQUINONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005208578	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.03729238	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.02339914	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2075402025126264	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.1346350544504987	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-720622	chembl:CHEMBL1287980	CHEMBL:CHEMBL1287980	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.041150213	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	SJ000260156	chembl:CHEMBL590695	CHEMBL:CHEMBL590695	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	GNF-PF-4786	chembl:CHEMBL602363	CHEMBL:CHEMBL602363	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	PENFLURIDOL	rxcui:7974	PENFLURIDOL	FALSE	FALSE	FALSE
FOXO3	hgnc:3821	FOXO3	DTC	9/2/20	NULL	52.50767123569449	SYRINGARESINOL	chembl:CHEMBL361362	SYRINGARESINOL	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GNF-PF-2356	chembl:CHEMBL601547	CHEMBL:CHEMBL601547	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	PALMITOYL-DL-CARNITINE CHLORIDE	chembl:CHEMBL1256761	CHEMBL:CHEMBL1256761	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.015516451	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003313623	SPIPERONE	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.017811286	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.027855529	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.5097832158805291	AZORUBINE	chembl:CHEMBL1552837	AZORUBINE	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.1187956362798518	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.056826484	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
ARRB1	hgnc:711	ARRB1	DTC	9/2/20	NULL	0.036590712	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	GNF-PF-4786	chembl:CHEMBL602363	CHEMBL:CHEMBL602363	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.020575106	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007003824	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	SPIPERONE	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.034318739	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.058602312	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.1479089330582944	DNDI1417254	chembl:CHEMBL2094567	CHEMBL:CHEMBL2094567	FALSE	FALSE	FALSE
GLA	hgnc:4296	GLA	DTC	9/2/20	NULL	0.1154014752432846	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.020836377	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.087512785	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.006614723	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004937716	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.04907259	PROPYLPARABEN	rxcui:34706	PROPYLPARABEN	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.030832455	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003401858	ESCITALOPRAM OXALATE	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.033338204	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	NORTRIPTYLINE HYDROCHLORIDE	rxcui:203130	NORTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DOCUSATE SODIUM	rxcui:71722	DOCUSATE SODIUM	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004754838	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.02726255	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.005688805	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	AMCINAFIDE	ncit:C80807	AMCINAFIDE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	SIB-1893	iuphar.ligand:1432	SIB-1893	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	DNDI1417599	chembl:CHEMBL2094833	CHEMBL:CHEMBL2094833	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	7,3'-DIMETHOXYFLAVONE	chembl:CHEMBL1326944	7,3'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.021832712	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.016077058	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	DTC	9/2/20	NULL	0.2083637747448194	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MALTOTRIOSE	chembl:CHEMBL1234363	MALTOTRIOSE	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.1620607136904151	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.6604738520213144	ISORHAMNETIN	drugbank:DB16767	ISORHAMNETIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	NSC-724440	chembl:CHEMBL515617	CHEMBL:CHEMBL515617	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
PROS1	hgnc:9456	PROS1	FDA	10-Apr-24	NULL	2.143170254518142	Avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.047734247	Dapsone	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.059030547	Deutetrabenazine	rxcui:1876905	DEUTETRABENAZINE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	FDA	10-Apr-24	NULL	0.8204323630577265	Nusinersen	rxcui:1863556	NUSINERSEN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.035418328	Pitolisant	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.092606122	Ramucirumab	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.018081154	Prasugrel	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	9.451380822	Simeprevir	rxcui:1482790	SIMEPREVIR	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.3918482928036902	DANUSERTIB	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.04525223	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.023759127	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.095500063	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	0.1832728489902076	XL281	drugbank:DB05190	XL281	FALSE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	MyCancerGenome	20-Jun-17	inhibitor	0.2243917574174978	LGX818	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	MyCancerGenome	20-Jun-17	inhibitor	1.346350544504987	XL281	drugbank:DB05190	XL281	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	0.074975256	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.1852122442176172	MM-151	iuphar.ligand:9125	MM-151	FALSE	TRUE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.09699693	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	antibody	0.8255923150266431	GANITUMAB	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.8607814956671229	EPIPODOPHYLLOTOXINS	ncit:C1331	EPIPODOPHYLLOTOXIN COMPOUND	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.090608578	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB4	hgnc:45	ABCB4	NCI	14-Sep-17	NULL	0.2592971419046642	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.2869271652223742	DROLOXIFENE	ncit:C969	DROLOXIFENE	FALSE	FALSE	FALSE
ABCB4	hgnc:45	ABCB4	NCI	14-Sep-17	NULL	0.6177373086552295	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.032817295	GLEEVEC	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ADM	hgnc:259	ADM	NCI	14-Sep-17	NULL	0.3547815624033412	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	1.521961485092594	PROTHYMOSIN ALPHA	ncit:C1203	RECOMBINANT PROTHYMOSIN ALPHA	FALSE	FALSE	FALSE
ADH4	hgnc:252	ADH4	NCI	14-Sep-17	NULL	0.1107756777124356	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.1544343271638073	INTERFERON GAMMA	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.4150804050252529	PROGESTOGENS	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	NCI	14-Sep-17	NULL	0.058471794	NAFOXIDINE	ncit:C677	NAFOXIDINE	FALSE	FALSE	FALSE
B2M	hgnc:914	B2M	NCI	14-Sep-17	NULL	4.375639269641208	THYROGLOBULIN	rxcui:10565	THYROGLOBULIN	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.038894571	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.7001022831425933	INHIBINS	ncit:C578	RECOMBINANT INHIBIN	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.051859428	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1067229090156392	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	2.333674277141977	TOPICAL CORTICOSTEROIDS	ncit:C29505	TOPICAL CORTICOSTEROID	FALSE	FALSE	FALSE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	0.9546849315580819	DIFFERENTIATING AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	1.166837138570989	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
CD44	hgnc:1681	CD44	NCI	14-Sep-17	NULL	0.3684748858645228	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
CD55	hgnc:2665	CD55	NCI	14-Sep-17	NULL	0.5676504998453459	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
CD44	hgnc:1681	CD44	NCI	14-Sep-17	NULL	0.5527123287967842	INTERFERON GAMMA	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
CDA	hgnc:1712	CDA	NCI	14-Sep-17	NULL	0.1613138901250215	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	1.693795846312725	FTI	ncit:C2020	FARNESYL TRANSFERASE INHIBITOR	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	NCI	14-Sep-17	NULL	0.2763561643983921	GEMTUZUMAB OZOGAMICIN	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	NCI	14-Sep-17	NULL	0.145450613	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
COIL	hgnc:2184	COIL	NCI	14-Sep-17	NULL	2.059124362184098	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.070010228	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.029170928	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.4667348554283955	TETANUS TOXOID	chembl:CHEMBL2108875	TETANUS TOXOID	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.050007306	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	IL-12 GENE	ncit:C2222	INTERLEUKIN-12 GENE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.041182487	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.044310271	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CST3	hgnc:2475	CST3	NCI	14-Sep-17	NULL	0.921187215	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.2692701089009974	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.7001022831425934	CTLA4-IG	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	0.3125456621172291	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.012364929	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.03151721	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	5.834185692854944	OXYGEN THERAPY	wikidata:Q1988216	OXYGEN THERAPY	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	NCI	14-Sep-17	NULL	0.007033376	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.5431828058864948	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.077047207	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.1178623372293928	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.058277105	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.035040154	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
FLG	hgnc:3748	FLG	NCI	14-Sep-17	NULL	52.50767123569449	PROPIONIBACTERIUM ACNES	rxcui:1310910	PROPIONIBACTERIUM ACNES	FALSE	FALSE	FALSE
FPGS	hgnc:3824	FPGS	NCI	14-Sep-17	NULL	0.080225625	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.5834185692854944	FREUNDS ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	NCI	14-Sep-17	NULL	0.069454592	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.053172325	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.4039051633514962	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
GAL	hgnc:4114	GAL	NCI	14-Sep-17	NULL	0.3977853881492008	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
GAS6	hgnc:4168	GAS6	NCI	14-Sep-17	NULL	1.060761035064535	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.2500365296937833	IL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.5357925636295358	HEREGULIN	ncit:C1426	RECOMBINANT HEREGULIN	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.089298761	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6428	iuphar.ligand:6428	GRN-529	FALSE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	NCI	14-Sep-17	NULL	0.074797252	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
H2AFX	hgnc:4739	H2AX	NCI	14-Sep-17	NULL	0.384671584	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	NCI	14-Sep-17	NULL	0.042602573	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.09869863	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.1242785118004603	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.4039051633514962	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.3241214273808303	ROFECOXIB	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	1.615620653405984	IL-10	iuphar.ligand:4975	IL-10	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	NCI	14-Sep-17	NULL	1.923357921	CISAPRIDE	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6427	iuphar.ligand:6427	COMPOUND 16A [PMID: 14697765]	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	NCI	14-Sep-17	NULL	0.072175493	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.5834185692854945	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	NCI	14-Sep-17	NULL	0.1320947704042629	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.09869863	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.1315981735230438	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.5834185692854945	ROFECOXIB	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.5250767123569451	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6430	iuphar.ligand:6430	COMPOUND 29B [PMID: 20809633]	FALSE	FALSE	FALSE
IL3RA	hgnc:6012	IL3RA	NCI	14-Sep-17	NULL	0.3088686543276147	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	1.29648571	BIOSTIM	ncit:C1018	KLEBSIELLA PNEUMONIAE GLYCOPROTEIN	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	2.143170254518142	IMIPENEM CILASTATIN SODIUM	ncit:C2338	IMIPENEM-CILASTATIN SODIUM	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.081030357	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.049864835	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.037042449	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
LIPE	hgnc:6621	LIPE	NCI	14-Sep-17	NULL	0.9053046764774914	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1973972602845657	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1339481409073839	RU 486	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.063916824	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6395	iuphar.ligand:6395	LSN2814617	FALSE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	NCI	14-Sep-17	NULL	0.3454452054979901	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.2344092465879218	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
MICA	hgnc:7090	MICA	NCI	14-Sep-17	NULL	5.250767124	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.079197091	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6400	iuphar.ligand:6400	VU0360172	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	NCI	14-Sep-17	NULL	0.6250913242344582	HEXAMETHYLENE BISACETAMIDE	ncit:C1125	HEXAMETHYLENE BISACETAMIDE	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	NCI	14-Sep-17	NULL	0.3125456621172291	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	0.086007651	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	LOBAPLATIN	ncit:C1434	LOBAPLATIN	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.040546464	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.1562728310586145	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1433	ncit:C80667	FENOBAM ANHYDROUS	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	NCI	14-Sep-17	NULL	0.027693919	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	NCI	14-Sep-17	NULL	0.040515178	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.007406922	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.013990853	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.3241214273808303	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1056492378987816	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.037925367	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	NCI	14-Sep-17	NULL	0.01045553	ARABINOFURANOSYLCYTOSINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.2692701089009974	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.017760078	ARABINOFURANOSYLCYTOSINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.075714018	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	0.2083637747448194	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.037857009	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.02213179	TAM	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.02213179	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.1620607136904151	I3C	ncit:C1135	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.048618214	IL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.024759276	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.016574391	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.089756703	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.06757744	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.4167275494896388	EOTAXIN	ncit:C1531	RECOMBINANT EOTAXIN	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	1.093909817410302	DEOXYCOFORMYCIN	rxcui:8011	PENTOSTATIN	TRUE	FALSE	TRUE
PPY	hgnc:9327	PPY	NCI	14-Sep-17	NULL	5.000730593875666	CISAPRIDE	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	FLUOXYMESTERONE	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.2430910705356226	MANNITOL	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	NCI	14-Sep-17	NULL	0.4167275494896389	INTERLEUKIN-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	NCI	14-Sep-17	NULL	0.053038052	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:1373	iuphar.ligand:1373	(+)-MCPG	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.2692701089009974	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.6731752722524935	CLOMIPHENE CITRATE	rxcui:142431	CLOMIPHENE CITRATE	TRUE	FALSE	FALSE
PTHR1	hgnc:9608	PTH1R	NCI	14-Sep-17	NULL	0.1595977849109255	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.8975670296699914	ENDOTHELIN RECEPTOR ANTAGONIST	ncit:C28313	ENDOTHELIN RECEPTOR ANTAGONIST	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.3365876361262467	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
PTPN13	hgnc:9646	PTPN13	NCI	14-Sep-17	NULL	7.001022831425933	ANTIESTROGENS	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9836	ncit:C152510	TANZISERTIB	FALSE	FALSE	FALSE
PYGM	hgnc:9726	PYGM	NCI	14-Sep-17	NULL	1.875273972703374	RU 486	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
PTP4A1	hgnc:9634	PTP4A1	NCI	14-Sep-17	NULL	17.50255707856483	HALOFUGINONE	ncit:C1120	HALOFUGINONE	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	NCI	14-Sep-17	NULL	0.040005845	GLEEVEC	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
SAA1	hgnc:10513	SAA1	NCI	14-Sep-17	NULL	5.834185692854945	IL-1RA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:8179	iuphar.ligand:8179	PF-03715455	FALSE	FALSE	FALSE
SLC25A5	hgnc:10991	SLC25A5	NCI	14-Sep-17	NULL	0.1207072901969988	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
SLC16A1	hgnc:10922	SLC16A1	NCI	14-Sep-17	NULL	2.500365296937833	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.3500511415712966	FREUND&APOS;S ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
TBXA2R	hgnc:11608	TBXA2R	NCI	14-Sep-17	NULL	0.2206204673768676	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:8074	iuphar.ligand:8074	NG-25	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.037870661	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.2071308530007672	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
TJP1	hgnc:11827	TJP1	NCI	14-Sep-17	NULL	0.3323270331373069	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.080656945	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.1881995384791917	PYRIDOXINE	rxcui:42954	VITAMIN B6	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.2258394461750301	FLUOCINOLONE ACETONIDE	rxcui:4461	FLUOCINOLONE ACETONIDE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.3763990769583834	TETRANDRINE	ncit:C28952	TETRANDRINE	FALSE	FALSE	FALSE
NCBIGENE:2080	hgnc:6857	MAP3K5	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8133	iuphar.ligand:8133	COMPOUND 10 [PMID: 23147077]	FALSE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	NCI	14-Sep-17	NULL	4.375639269641208	AUTOANTIGEN	ncit:C20972	AUTOANTIGEN	FALSE	FALSE	FALSE
TNFRSF11B	hgnc:11909	TNFRSF11B	NCI	14-Sep-17	NULL	0.384671584	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.011176601	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TNFSF10	hgnc:11925	TNFSF10	NCI	14-Sep-17	NULL	2.500365296937833	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.038636991	YONDELIS	rxcui:1716278	TRABECTEDIN	TRUE	FALSE	TRUE
TRH	hgnc:12298	TRH	NCI	14-Sep-17	NULL	0.5000730593875666	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	5.527123287967842	ANTIEMETIC	ncit:C267	ANTIEMETIC AGENT	FALSE	FALSE	FALSE
TYMP	hgnc:3148	TYMP	NCI	14-Sep-17	NULL	1.312691780892362	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.1141471113819445	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.034374908	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.093098708	MITOMYCIN C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
NCBIGENE:2084	hgnc:6861	MAP3K9	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
UGT1A9	hgnc:12541	UGT1A9	NCI	14-Sep-17	NULL	0.175610941	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.145450613	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
VIM	hgnc:12692	VIM	NCI	14-Sep-17	NULL	21.00306849427779	GANGLIOSIDE GM2	ncit:C516	GANGLIOSIDE GM2	FALSE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.06823609	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CDA	hgnc:1712	CDA	PharmGKB	4/5/24	NULL	0.375054795	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.019739726	alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.036770078	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CHRNE	hgnc:1966	CHRNE	PharmGKB	4/5/24	NULL	0.3070624048871023	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.3182283105193606	isosorbide dinitrate	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.2143170254518142	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:2086	hgnc:3454	ERV3-1	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:8074	iuphar.ligand:8074	NG-25	FALSE	FALSE	FALSE
C9ORF72	hgnc:28337	C9orf72	PharmGKB	4/5/24	NULL	5.250767124	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.069638821	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.028467157	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.042242696	ampicillin	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.023233483	flutamide	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.020203029	doxycycline	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
PTGER2	hgnc:9594	PTGER2	PharmGKB	4/5/24	NULL	0.046549354	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1548898856510162	sulfamethazine	rxcui:10178	SULFAMETHAZINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.007596596	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.003038638	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	0.4375639269641208	atomoxetine	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HCN1	hgnc:4845	HCN1	PharmGKB	4/5/24	NULL	7.501095890813499	o-desmethyltramadol	chembl:CHEMBL4650315	DESMETRAMADOL	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	PharmGKB	4/5/24	NULL	0.3025133322221082	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NCF4	hgnc:7662	NCF4	PharmGKB	4/5/24	NULL	0.4667348554283955	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CXCL13	hgnc:10639	CXCL13	PharmGKB	4/5/24	NULL	1.166837138570988	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:2084	hgnc:6861	MAP3K9	GuideToPharmacology	2024.1	inhibitor	0.9376369863516874	IUPHAR.LIGAND:8137	iuphar.ligand:8137	COMPOUND 8E [PMID: 24432909]	FALSE	FALSE	FALSE
MIR1264	hgnc:35246	MIR1264	PharmGKB	4/5/24	NULL	0.2706580991530644	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
RUNDC3B	hgnc:30286	RUNDC3B	PharmGKB	4/5/24	NULL	1.400204566285186	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CRY1	hgnc:2384	CRY1	PharmGKB	4/5/24	NULL	1.250182648468916	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:6505	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
SCNN1G	hgnc:10602	SCNN1G	PharmGKB	4/5/24	NULL	0.6482428547616605	bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
MTTP	hgnc:7467	MTTP	PharmGKB	4/5/24	NULL	0.6482428547616604	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	PharmGKB	4/5/24	NULL	0.1241316104862754	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
SRP19	hgnc:11300	SRP19	PharmGKB	4/5/24	NULL	1.312691780892362	sertraline	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	0.2344092465879218	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:1639	hgnc:2711	DCTN1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.015627283	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	PharmGKB	4/5/24	NULL	0.010505737	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.084598826	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CORO7	hgnc:26161	CORO7	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.018560506	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	1.111273465305703	mobocertinib	rxcui:2570736	MOBOCERTINIB	TRUE	FALSE	TRUE
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	0.4412409347537353	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
PLCG1	hgnc:9065	PLCG1	PharmGKB	4/5/24	NULL	0.5147810905460245	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
SLC22A7	hgnc:10971	SLC22A7	PharmGKB	4/5/24	NULL	0.5147810905460245	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9014	iuphar.ligand:9014	PF-152	FALSE	FALSE	FALSE
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	0.041377203	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	PharmGKB	4/5/24	NULL	0.024709492	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	0.076374795	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.04339477	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
PRDM16	hgnc:14000	PRDM16	PharmGKB	4/5/24	NULL	0.9546849315580819	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
APOA5	hgnc:17288	APOA5	PharmGKB	4/5/24	NULL	0.5728109589348491	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
SLC6A12	hgnc:11045	SLC6A12	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	10.74020548002842	tezacaftor	rxcui:1999382	TEZACAFTOR	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.1342907192728759	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.7059854956059763	avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	51.82575342743873	succinylcholine	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	0.1260688385010672	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:8606	iuphar.ligand:8606	JZL195	FALSE	FALSE	FALSE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	21.82136986418472	methoxyflurane	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.088248187	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	0.092118721	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.1442518440541057	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NR1I3	hgnc:7969	NR1I3	PharmGKB	4/5/24	NULL	0.2296253844126581	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	7.501095891	isepamicin	ncit:C83838	ISEPAMICIN	FALSE	FALSE	FALSE
HMMR	hgnc:5012	HMMR	PharmGKB	4/5/24	NULL	0.2206204673768676	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.28382525	betaine	rxcui:1512	BETAINE	TRUE	FALSE	FALSE
PSORS1C3	hgnc:17203	PSORS1C3	PharmGKB	4/5/24	NULL	1.166837138570988	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
HFE	hgnc:4886	HFE	PharmGKB	4/5/24	NULL	0.7721716358190368	epoetin alfa	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
CNNM2	hgnc:103	CNNM2	PharmGKB	4/5/24	NULL	2.333674277141977	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
NCBIGENE:2881	hgnc:23248	MOGAT2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12738	iuphar.ligand:12738	BMS-963272	FALSE	FALSE	FALSE
GREM2	hgnc:17655	GREM2	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
STX4	hgnc:11439	STX4	PharmGKB	4/5/24	NULL	7.001022831425934	acenocoumarol	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9482	iuphar.ligand:9482	KML29	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	PharmGKB	4/5/24	NULL	0.007607602	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011746683	telithromycin	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.002629854	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.005593658	sertindole	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.005339401	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003632995	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.018687904	ketoconazole	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.009788902	mephenytoin	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.005339401	methoxyflurane	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
CALU	hgnc:1458	CALU	PharmGKB	4/5/24	NULL	31.50460274141669	acenocoumarol	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	0.061197752	carvedilol	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	1.193356164447602	canakinumab	rxcui:853491	CANAKINUMAB	TRUE	TRUE	TRUE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1462	iuphar.ligand:1462	MOTILIN-(1-13) (HUMAN)	FALSE	FALSE	FALSE
AOC1	hgnc:80	AOC1	PharmGKB	4/5/24	NULL	0.024605282	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	1.228249619548409	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2461297089173179	thiotepa	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.760980743	elagolix	rxcui:2049846	ELAGOLIX	TRUE	FALSE	FALSE
EPM2AIP1	hgnc:19735	EPM2AIP1	PharmGKB	4/5/24	NULL	3.500511415712966	dacarbazine	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.064824285	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	0.1666910197958555	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.05073205	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	PharmGKB	4/5/24	NULL	0.096264064	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UGT2A1	hgnc:12542	UGT2A1	PharmGKB	4/5/24	NULL	1.400204566285186	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
C20ORF194	hgnc:17721	DNAAF9	PharmGKB	4/5/24	NULL	1.381780822	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.031115657	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:7266	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
BCL2L11	hgnc:994	BCL2L11	PharmGKB	4/5/24	NULL	0.525076712	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.3786610906420276	irbesartan	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.038894571	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.054695491	trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
COLEC10	hgnc:2220	COLEC10	PharmGKB	4/5/24	NULL	0.8824818695074705	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:4035	ncit:C166668	CAMICINAL	FALSE	FALSE	FALSE
NPC1L1	hgnc:7898	NPC1L1	PharmGKB	4/5/24	NULL	1.944728564284981	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	PharmGKB	4/5/24	NULL	1.500219178	ethosuximide	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	PharmGKB	4/5/24	NULL	0.011517366	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
TRAC	hgnc:12029	TRAC	PharmGKB	4/5/24	NULL	0.2706580991530644	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:7266	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	PharmGKB	4/5/24	NULL	0.2778183663264259	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.05913026	caffeine	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	1.166837138570988	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.3409589041278864	ampicillin	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.099305288	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PTPN11	hgnc:9644	PTPN11	PharmGKB	4/5/24	NULL	0.1875273972703375	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
BMP5	hgnc:1072	BMP5	PharmGKB	4/5/24	NULL	3.000438356	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
TMEM167A	hgnc:28330	TMEM167A	PharmGKB	4/5/24	NULL	0.8824818695074705	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	14.00204566285186	simeprevir	rxcui:1482790	SIMEPREVIR	FALSE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	9.451380822	simeprevir	rxcui:1482790	SIMEPREVIR	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	PharmGKB	4/5/24	NULL	0.01877621	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	PharmGKB	4/5/24	NULL	0.02262774	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:4036	iuphar.ligand:4036	MA-2029	FALSE	FALSE	FALSE
DLG5	hgnc:2904	DLG5	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
OSGEP	hgnc:18028	OSGEP	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CHN2	hgnc:1944	CHN2	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1460	iuphar.ligand:1460	MOTILIN-(1-11) (HUMAN)	FALSE	FALSE	FALSE
OASL	hgnc:8090	OASL	PharmGKB	4/5/24	NULL	1.381780822	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.09869863	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	PharmGKB	4/5/24	NULL	0.4118248724368196	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.1535312024435511	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1500219178162699	glipizide	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	1.050153425	moviprep	rxcui:267366	SODIUM ASCORBATE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.760980743	dulaglutide	rxcui:1551291	DULAGLUTIDE	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.040328473	Methyldopa	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
HNRNPH2	hgnc:5042	HNRNPH2	PharmGKB	4/5/24	NULL	17.50255707856483	migalastat	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
GLCCI1	hgnc:18713	GLCCI1	PharmGKB	4/5/24	NULL	1.615620653405984	budesonide	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
PROS1	hgnc:9456	PROS1	PharmGKB	4/5/24	NULL	2.143170254518142	avatrombopag	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	PharmGKB	4/5/24	NULL	0.2287915957982331	talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.053038052	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
SLIT1	hgnc:11085	SLIT1	PharmGKB	4/5/24	NULL	0.8899605294185507	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.011219588	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BLMH	hgnc:1059	BLMH	PharmGKB	4/5/24	NULL	0.2224901323546377	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
SLC22A4	hgnc:10968	SLC22A4	PharmGKB	4/5/24	NULL	2.625383561784725	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.3947945205691315	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.1553481397505754	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.031254566	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
TLR2	hgnc:11848	TLR2	PharmGKB	4/5/24	NULL	0.1630673019742065	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	8.078103267029922	buprenorphine / naloxone	wikidata:Q25048068	BUPRENORPHINE/NALOXONE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.2363572458670459	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:6937	iuphar.ligand:6937	IPEROXO	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	TALC	12-May-16	inhibitor	0.2044691247495891	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.079376676	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	TALC	12-May-16	inhibitor	0.1402073998282897	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.1480479452134243	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.3409589041278864	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.151537291	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.2251615404618117	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
IL2	hgnc:6001	IL2	TALC	12-May-16	vaccine	0.4102161815288632	MVA-MUC1-IL2	ncit:C2241	MESMULOGENE ANCOVACIVEC	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.023004456	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	1.250182648468916	AZD8330	iuphar.ligand:8474	AZD8330	FALSE	FALSE	TRUE
MMP3	hgnc:7173	MMP3	TALC	12-May-16	vaccine	0.5357925636295356	PRINOMASTAT	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	1.500219178	INCB28060	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:291	iuphar.ligand:291	NNC 11-1314	FALSE	FALSE	FALSE
MMP13	hgnc:7159	MMP13	TALC	12-May-16	vaccine	0.9376369863516874	PRINOMASTAT	ncit:C1811	PRINOMASTAT	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.2386712328895204	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
PRKCA	hgnc:9393	PRKCA	TALC	12-May-16	antisense oligonucleotide	1.093909817410302	AFFINITAC	rxcui:2634355	APRINOCARSEN	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	TALC	12-May-16	inhibitor	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ROS1	hgnc:10261	ROS1	TALC	12-May-16	inhibitor	1.346350544504987	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:7354	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	TALC	12-May-16	inhibitor	0.1691068316769549	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
BIRC3	hgnc:591	BIRC3	TALC	12-May-16	inhibitor	1.071585127259071	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
XIAP	hgnc:592	XIAP	TALC	12-May-16	inhibitor	0.3571950424196904	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
UNIPROT:P13762	hgnc:4952	HLA-DRB4	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	1D09C3	drugbank:DB05121	1D09C3	FALSE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	TALC	12-May-16	inhibitor	0.729273212	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
UNIPROT:Q08722	hgnc:1682	CD47	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	ABT-510	drugbank:DB05434	ABT-510	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.276356164	IUPHAR.LIGAND:338	iuphar.ligand:338	KT 5823	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.069454592	AC480	ncit:C48380	PAN-HER KINASE INHIBITOR AC480	FALSE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	ACOTIAMIDE	ncit:C65214	ACOTIAMIDE	FALSE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	0.1215455352678113	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	0.1620607136904151	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.050246575	IUPHAR.LIGAND:356	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	0.085796848	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	ZALEPLON	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
UNIPROT:Q9NZ42	hgnc:30100	PSENEN	TdgClinicalTrial	Jan-14	NULL	0.729273212	BMS-299897	chembl:CHEMBL247471	CHEMBL:CHEMBL247471	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.083016081	CARIPRAZINE	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	CHIDAMIDE	hemonc:99	CHIDAMIDE	FALSE	FALSE	FALSE
UNIPROT:Q8TDS4	hgnc:24827	HCAR2	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	CILANSETRON	ncit:C76106	CILANSETRON	FALSE	FALSE	FALSE
UNIPROT:P07947	hgnc:12841	YES1	TdgClinicalTrial	Jan-14	NULL	0.013113804	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.056142926	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.070543222	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.033458584	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	ECOPIPAM	ncit:C74188	ECOPIPAM	FALSE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	9.845188356692718	ELINOGREL	ncit:C96896	ELINOGREL	FALSE	FALSE	FALSE
UNIPROT:Q16739	hgnc:12524	UGCG	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	ELIGLUSTAT	rxcui:1547220	ELIGLUSTAT	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.03251249	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
UNIPROT:O00206	hgnc:11850	TLR4	TdgClinicalTrial	Jan-14	NULL	4.565884455277782	ERITORAN	ncit:C80053	ERITORAN	FALSE	FALSE	FALSE
UNIPROT:A5X5Y0	hgnc:24005	HTR3E	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	GLYCOPYRROLATE	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:314	iuphar.ligand:314	MUSCARINIC TOXIN 7	FALSE	FALSE	FALSE
UNIPROT:Q9Y5N1	hgnc:5184	HRH3	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	GSK-1004723	drugbank:DB12806	GSK-1004723	FALSE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	FAMOTIDINE	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	IBANDRONATE	rxcui:115264	IBANDRONATE	TRUE	FALSE	FALSE
NCBIGENE:1216	hgnc:25588	SLC47A1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:1231	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
UNIPROT:P07949	hgnc:9967	RET	TdgClinicalTrial	Jan-14	NULL	0.034572952	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.096264064	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	1.029066006546944	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	TASIDOTIN	ncit:C77067	TASIDOTIN	FALSE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	INS-50589	rxcui:1313722	REGRELOR	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1642918374083057	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P06213	hgnc:6091	INSR	TdgClinicalTrial	Jan-14	NULL	1.500219178	INSULIN GLULISINE	rxcui:400008	INSULIN GLULISINE, HUMAN	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.077789143	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P04062	hgnc:4177	GBA1	TdgClinicalTrial	Jan-14	NULL	4.500657534488099	ISOFAGOMINE	ncit:C83520	AFEGOSTAT	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.42006137	JB991	drugbank:DB05081	JB991	FALSE	FALSE	FALSE
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	KC706	drugbank:DB05157	KC706	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.272767123	KETOPROFEN	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.9546849315580818	LIRAGLUTIDE	rxcui:475968	LIRAGLUTIDE	TRUE	FALSE	FALSE
UNIPROT:P01589	hgnc:6008	IL2RA	TdgClinicalTrial	Jan-14	NULL	0.3431873936973496	INTERLEUKIN-2	ncit:C587	RECOMBINANT INTERLEUKIN-2	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	GLYCOPYRRONIUM	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	BETAHISTINE	rxcui:1511	BETAHISTINE	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.020320306	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:Q9NR61	hgnc:2910	DLL4	TdgClinicalTrial	Jan-14	NULL	31.50460274141669	DEMCIZUMAB	ncit:C80041	DEMCIZUMAB	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.099446347	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	PTC299	drugbank:DB05173	PTC299	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.060215219	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.6134073742487676	RAD1901	rxcui:2628469	ELACESTRANT	TRUE	FALSE	TRUE
UNIPROT:Q96GD4	hgnc:11390	AURKB	TdgClinicalTrial	Jan-14	NULL	0.033207482	R763	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:O14965	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.04525223	R763	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.4268916360625568	RG2833	iuphar.ligand:7501	RGFP109	FALSE	FALSE	FALSE
UNIPROT:Q08499	hgnc:8783	PDE4D	TdgClinicalTrial	Jan-14	NULL	0.025513932	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1355	iuphar.ligand:1355	S26284	FALSE	FALSE	FALSE
UNIPROT:O43525	hgnc:6297	KCNQ3	TdgClinicalTrial	Jan-14	NULL	2.678962818147678	RETIGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
UNIPROT:P05113	hgnc:6016	IL5	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	RESLIZUMAB	rxcui:1746889	RESLIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P22455	hgnc:3691	FGFR4	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
UNIPROT:Q9UI33	hgnc:10583	SCN11A	TdgClinicalTrial	Jan-14	NULL	0.05293112	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:O00305	hgnc:1404	CACNB4	TdgClinicalTrial	Jan-14	NULL	0.252440727	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.042073455	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.061628722	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.022949157	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	0.760980743	SPI-1620	ncit:C74027	SOVATELTIDE	FALSE	FALSE	FALSE
UNIPROT:Q9NR63	hgnc:20581	CYP26B1	TdgClinicalTrial	Jan-14	NULL	10.50153425	TALAROZOLE	ncit:C90792	TALAROZOLE	FALSE	FALSE	FALSE
UNIPROT:P11049	hgnc:1666	CD37	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	TRU-016	ncit:C74006	OTLERTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:1617	ncit:C166495	DIPRENORPHINE	FALSE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.1810609352954982	XL888	ncit:C79835	HSP90 INHIBITOR XL888	FALSE	FALSE	TRUE
UNIPROT:O96017	hgnc:16627	CHEK2	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	XL844	drugbank:DB05149	XL844	FALSE	FALSE	FALSE
UNIPROT:O14757	hgnc:1925	CHEK1	TdgClinicalTrial	Jan-14	NULL	1.381780822	XL844	drugbank:DB05149	XL844	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.1312691780892362	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
UNIPROT:P30530	hgnc:905	AXL	TdgClinicalTrial	Jan-14	NULL	0.1093909817410302	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.1434635826111871	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.063262255	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.2075402025126264	ACETOPHENAZINE	rxcui:16735	ACETOPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	9.845188356692718	BETAZOLE	drugbank:DB00272	BETAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	BIPERIDEN	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2094720926955897	BIPERIDEN	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.4565884455277783	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.1154014752432846	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	ETHOPROPAZINE	rxcui:4134	PROFENAMINE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	OXPRENOLOL	rxcui:7801	OXPRENOLOL	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.546954909	PHENYLPROPANOLAMINE	rxcui:8175	PHENYLPROPANOLAMINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.031555091	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	PHENDIMETRAZINE	rxcui:33272	PHENDIMETRAZINE	TRUE	FALSE	FALSE
UNIPROT:P00439	hgnc:8582	PAH	TdgClinicalTrial	Jan-14	NULL	3.500511415712967	SAPROPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.5427149481725528	RITODRINE	rxcui:9392	RITODRINE	TRUE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TEND	1-Aug-11	NULL	0.7001022831425934	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.5427149481725528	ALPRENOLOL	rxcui:597	ALPRENOLOL	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.7955707762984013	ALPRENOLOL	rxcui:597	ALPRENOLOL	FALSE	FALSE	FALSE
UNIPROT:Q9UGM1	hgnc:14079	CHRNA9	TEND	1-Aug-11	NULL	1.141471113819445	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	modulator	0.5770073762164231	IUPHAR.LIGAND:9159	iuphar.ligand:9159	BMS-986123	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.2075402025126264	ACETOPHENAZINE	rxcui:16735	ACETOPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:Q02127	hgnc:2867	DHODH	TEND	1-Aug-11	NULL	1.151484018326633	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
UNIPROT:P24530	hgnc:3180	EDNRB	TEND	1-Aug-11	NULL	2.250328767244049	AMBRISENTAN	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.2419708351875322	CETIRIZINE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TEND	1-Aug-11	NULL	3.750547945	CARBOPROST TROMETHAMINE	rxcui:20259	CARBOPROST TROMETHAMINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.047886613	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TEND	1-Aug-11	NULL	0.1491695205559502	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.076263865	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:7209	rxcui:6370	LEVALLORPHAN	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.064033745	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.061055432	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.061055432	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1215455352678113	DRONEDARONE	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.1325951293830669	DRONEDARONE	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	DIPHENYLPYRALINE	rxcui:23386	DIPHENYLPYRALINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1221108633388244	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TEND	1-Aug-11	NULL	5.834185692854944	GONADORELIN	rxcui:6384	GONADORELIN	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.1280674908187671	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.1166837138570989	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.4773424657790409	LUMIRACOXIB	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TEND	1-Aug-11	NULL	0.1976759387696734	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.1470803115845784	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.2778183663264258	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.1154014752432846	IUPHAR.LIGAND:1642	iuphar.ligand:1642	NOR-BINALTORPHIMINE	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.1861974157294131	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.1902451856365742	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:O43451	hgnc:7043	MGAM	TEND	1-Aug-11	NULL	4.773424657790408	MIGLITOL	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	1.334940794127826	MOEXIPRIL	rxcui:30131	MOEXIPRIL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.05814803	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.059532507	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.060984519	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.1457197166578015	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.051885051	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.093763699	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TEND	1-Aug-11	NULL	0.081030357	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.2112984757975633	PENTAZOCINE	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TEND	1-Aug-11	NULL	0.189216833	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1469979597863787	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.042073455	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TEND	1-Aug-11	NULL	0.3025133322221082	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.070956312	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.2365210416022274	IUPHAR.LIGAND:7435	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.04362008	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.5427149481725528	RITODRINE	rxcui:9392	RITODRINE	TRUE	FALSE	FALSE
UNIPROT:Q8TCC7	hgnc:10972	SLC22A8	TEND	1-Aug-11	NULL	2.045753424767318	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
UNIPROT:P00797	hgnc:9958	REN	TEND	1-Aug-11	NULL	15.75230137070834	REMIKIREN	ncit:C73099	REMIKIREN	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.096050618	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.083257407	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TEND	1-Aug-11	NULL	2.059124362184097	TAMIBAROTENE	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.081365193	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1223955040459079	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1835932560688619	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.091796628	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.093763699	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.092988792	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TEND	1-Aug-11	NULL	2.386712328895204	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TEND	1-Aug-11	NULL	0.9053046764774912	THIAMYLAL	rxcui:10464	THIAMYLAL	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	1.093909817410302	TOLBUTAMIDE	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.1646008502686348	IUPHAR.LIGAND:10316	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
UNIPROT:Q8NET8	hgnc:18084	TRPV3	TEND	1-Aug-11	NULL	8.751278539282415	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.1419126249613365	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.040893825	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.060215219	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TEND	1-Aug-11	NULL	0.7292732116068681	TREPROSTINIL	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.028229931	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1591141552596803	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.054243462	TRIMIPRAMINE	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.2044691247495891	VENLAFAXINE	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 4	hgnc:1605	CCR4	TTD	2020.06.01	NULL	6.177373086552294	AZD-1678	iuphar.ligand:9679	AZD1678	FALSE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	10.50153424713889	TAK-272	chembl:CHEMBL3969876	IMARIKIREN HYDROCHLORIDE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.021554873	Genistein	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.4167275494896388	OX-914	chembl:CHEMBL4297287	HT-0712	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.061628722	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	MCLA-128	ncit:C152948	ZENOCUTUZUMAB	FALSE	FALSE	FALSE
LYSOPHOSPHATIDIC ACID RECEPTOR 1	hgnc:3166	LPAR1	TTD	2020.06.01	NULL	26.25383561784724	BMS-986020	drugbank:DB14948	BMS-986020	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.250182648468916	Savolitinib	ncit:C104732	SAVOLITINIB	FALSE	FALSE	TRUE
B7 HOMOLOG 3	hgnc:19137	CD276	TTD	2020.06.01	NULL	31.50460274141669	Enoblituzumab	ncit:C97510	ENOBLITUZUMAB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.8334550989792777	Depatuxizumab	ncit:C95206	DEPATUXIZUMAB	FALSE	TRUE	TRUE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	CBT-501	ncit:C148159	GEPTANOLIMAB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1389091831632129	Sym015	ncit:C127906	ANTI-MET MONOCLONAL ANTIBODY MIXTURE SYM015	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.9723642821424906	REGN1979	ncit:C119615	ODRONEXTAMAB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	SYN004	ncit:C121550	ANTI-EGFR MONOCLONAL ANTIBODY SYN004	FALSE	FALSE	FALSE
NOCICEPTIN RECEPTOR	hgnc:8155	OPRL1	TTD	2020.06.01	NULL	6.563458904461812	BTRX-246040	drugbank:DB16048	BTRX-246040	FALSE	FALSE	FALSE
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	0.1190650141398968	BIIB092	chembl:CHEMBL3990042	GOSURANEMAB	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.080781033	Perifosine	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:7700	iuphar.ligand:7700	AZD1332	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	1.141471113819445	Aminoguanidine	rxcui:1311670	PIMAGEDINE	FALSE	FALSE	FALSE
MELANOMA-ASSOCIATED ANTIGEN 3	hgnc:6801	MAGEA3	TTD	2020.06.01	NULL	35.00511415712966	Astuprotimut-R	ncit:C78478	ASTUPROTIMUT-R	FALSE	FALSE	TRUE
MELANOMA ANTIGEN GP75	hgnc:12450	TYRP1	TTD	2020.06.01	NULL	105.0153424713889	Flanvotumab	ncit:C91384	FLANVOTUMAB	FALSE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	0.5147810905460245	NKP-1339	ncit:C97948	RUTHENIUM-BASED TRANSFERRIN TARGETING AGENT NKP-1339	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	2.282942227638891	NI-0101	ncit:C182630	PARIDIPRUBART	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.250182648468916	Volitinib	ncit:C104732	SAVOLITINIB	FALSE	FALSE	TRUE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.2365210416022274	Eltoprazine	ncit:C73286	ELTOPRAZINE	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:8137	iuphar.ligand:8137	COMPOUND 8E [PMID: 24432909]	FALSE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.087537101	Progesterone	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	6.177373086552294	BGC-20-1531	chembl:CHEMBL3260771	BGC-20-1531	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.068436196	ABP 501	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
EXPORTIN-1	hgnc:12825	XPO1	TTD	2020.06.01	NULL	5.250767123569449	KPT-330	rxcui:2178390	SELINEXOR	TRUE	FALSE	TRUE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	0.750109589	PRT-062607	iuphar.ligand:8070	P505-15	FALSE	FALSE	FALSE
LACTOTRANSFERRIN	hgnc:6720	LTF	TTD	2020.06.01	NULL	6.563458904461812	Parecoxib	rxcui:279950	PARECOXIB	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	0.2051080907644316	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Mephentermine	rxcui:6756	MEPHENTERMINE	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.5966780822238011	Ciprofibrate	rxcui:21149	CIPROFIBRATE	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.9723642821424906	Fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	2.282942227638891	TBC-3711	drugbank:DB05407	TBC-3711	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.056097939	Aniracetam	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	0.4605936073306534	Pyridoxal Phosphate	rxcui:1599827	PYRIDOXAL PHOSPHATE ANHYDROUS	FALSE	FALSE	FALSE
NICOTINIC ACID RECEPTOR	hgnc:24827	HCAR2	TTD	2020.06.01	NULL	2.500365296937833	Vitamin B3	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	0.172722603	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
PROLACTIN RECEPTOR	hgnc:9446	PRLR	TTD	2020.06.01	NULL	2.187819634820604	Endostatin	drugbank:DB06423	ENDOSTATIN	FALSE	FALSE	TRUE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.1256164383629055	Tetracaine	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:7700	iuphar.ligand:7700	AZD1332	FALSE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR3.4	hgnc:6266	KCNJ5	TTD	2020.06.01	NULL	0.3889457128569963	phorbol 12-myristate 13-acetate	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 5	hgnc:11334	SSTR5	TTD	2020.06.01	NULL	0.8751278539282418	ODT-8	chembl:CHEMBL452157	CHEMBL:CHEMBL452157	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.013340364	Gossypol	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1B	hgnc:278	ADRA1B	TTD	2020.06.01	NULL	0.5707355569097228	Phendimetrazine	rxcui:33272	PHENDIMETRAZINE	TRUE	FALSE	FALSE
TISSUE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9051	PLAT	TTD	2020.06.01	NULL	3.182283105193605	Aminocaproic Acid	rxcui:99	6-AMINOCAPROIC ACID	TRUE	FALSE	FALSE
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	1.640864726115453	NM-702	drugbank:DB05505	NM-702	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	NULL	1.875273972703375	IUPHAR.LIGAND:5033	iuphar.ligand:5033	NEUROTROPHIN-3	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE ENDOTHELIAL	hgnc:7876	NOS3	TTD	2020.06.01	NULL	1.250182648468916	Tilarginine acetate	ncit:C90899	TILARGININE ACETATE	FALSE	FALSE	FALSE
CERAMIDE GLUCOSYLTRANSFERASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	7.001022831425932	Miglustat	rxcui:402316	MIGLUSTAT	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.021053597	Interferon Alfa-2a, Recombinant	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.05814803	Nitrazepam	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	Sumanirole	ncit:C76651	SUMANIROLE	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	2.386712328895204	SARALASIN	rxcui:9556	SARALASIN	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	CCT-018159	drugbank:DB07594	CCT-018159	FALSE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.5834185692854945	SLV320	ncit:C96199	DERENOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:3981	iuphar.ligand:3981	[3H]&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	Tapentadol hydrochloride	rxcui:857492	TAPENTADOL HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.063110182	Colchicine	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR BETA-2	hgnc:4082	GABRB2	TTD	2020.06.01	NULL	0.1526385791735305	ZK-93423	drugbank:DB17063	ZK-93423	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA-2/DELTA-1	hgnc:1399	CACNA2D1	TTD	2020.06.01	NULL	0.6250913242344582	Lercanidipine	rxcui:135056	LERCANIDIPINE	TRUE	FALSE	FALSE
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	0.045579576	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	2.187819634820604	Pralatrexate	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.026045472	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.079376676	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
MITOCHONDRIAL COMPLEX I	hgnc:17194	NDUFA13	TTD	2020.06.01	NULL	13.12691780892362	Flurpiridaz F 18	ncit:C171889	FLURPIRIDAZ F-18	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	1.334940794127826	TAK-491	rxcui:1091642	AZILSARTAN MEDOXOMIL	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.2128689374420047	Vilazodone	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	0.2845944240417046	CHR-3996	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.305277158	LAS 100977	ncit:C132738	ABEDITEROL	FALSE	FALSE	FALSE
ILEAL SODIUM/BILE ACID COTRANSPORTER	hgnc:10906	SLC10A2	TTD	2020.06.01	NULL	4.039051633514961	A-3309	ncit:C171820	ELOBIXIBAT	FALSE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	2.187819634820604	Inotuzumab ozogamicin	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:3977	iuphar.ligand:3976	[125I]EPIBATIDINE	FALSE	FALSE	FALSE
CLAUDIN-18	hgnc:2039	CLDN18	TTD	2020.06.01	NULL	105.0153424713889	Claudiximab	ncit:C85475	ZOLBETUXIMAB	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	1.193356164447602	Antroquinonol	drugbank:DB12326	ANTROQUINONOL	FALSE	FALSE	FALSE
N-ACETYLGALACTOSAMINE 6 SULFATASE	hgnc:4122	GALNS	TTD	2020.06.01	NULL	105.0153424713889	BMN-110	rxcui:1489914	ELOSULFASE ALFA	TRUE	FALSE	FALSE
ALPHA-GALACTOSIDASE A	hgnc:4296	GLA	TTD	2020.06.01	NULL	4.039051633514961	PRX-102	chembl:CHEMBL4297801	PEGUNIGALSIDASE ALFA	FALSE	FALSE	FALSE
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	0.128537751	RXDX 101	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:463	hgnc:777	ZFHX3	GuideToPharmacology	2024.1	blocker	0.729273212	IUPHAR.LIGAND:3990	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	0.1919140030544389	RXDX 101	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
MHC CLASS I NK CELL RECEPTOR 2DL3	hgnc:6331	KIR2DL3	TTD	2020.06.01	NULL	4.375639269641208	IPH-2102	chembl:CHEMBL2109500	LIRILUMAB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.079376676	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
INTERLEUKIN 6 RECEPTOR	hgnc:6019	IL6R	TTD	2020.06.01	NULL	4.039051633514961	ALX-0061	iuphar.ligand:8363	VOBARILIZUMAB	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.081281225	Fludiazepam	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	PF-06801591	ncit:C124058	SASANLIMAB	FALSE	FALSE	FALSE
V-SET IMMUNOREGULATORY RECEPTOR	hgnc:30085	VSIR	TTD	2020.06.01	NULL	13.12691780892362	CA-170	drugbank:DB15772	CA-170	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.7160136986685613	Levobunolol	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	Methadyl Acetate	rxcui:6814	METHADYL ACETATE	TRUE	FALSE	FALSE
P-SELECTIN	hgnc:10721	SELP	TTD	2020.06.01	NULL	2.625383561784724	CY-1503	drugbank:DB17605	CY-1503	FALSE	FALSE	FALSE
E-SELECTIN	hgnc:10718	SELE	TTD	2020.06.01	NULL	2.386712328895204	CY-1503	drugbank:DB17605	CY-1503	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:3976	iuphar.ligand:3976	[125I]EPIBATIDINE	FALSE	FALSE	FALSE
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	0.092118721	Flufenamic Acid	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR BETA	hgnc:6009	IL2RB	TTD	2020.06.01	NULL	4.039051633514961	Leukocyte interleukin	drugbank:DB17315	LEUKOCYTE INTERLEUKIN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1B	hgnc:278	ADRA1B	TTD	2020.06.01	NULL	0.1268301237577161	MEDETOMIDINE	rxcui:52016	MEDETOMIDINE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	1.790034246671403	Arbutamine	rxcui:61609	ARBUTAMINE	TRUE	FALSE	FALSE
SOLUBLE GUANYLATE CYCLASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	0.5250767123569451	Nitric Oxide	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP3	hgnc:9595	PTGER3	TTD	2020.06.01	NULL	0.364636606	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.3580068493342807	Meloxicam	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
ILEAL SODIUM/BILE ACID COTRANSPORTER	hgnc:10906	SLC10A2	TTD	2020.06.01	NULL	4.039051633514961	S-8921	chembl:CHEMBL18380	CHEMBL:CHEMBL18380	FALSE	FALSE	FALSE
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	5.834185692854944	Antegren	rxcui:354770	NATALIZUMAB	TRUE	TRUE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.193356164447602	TAK-385	rxcui:2472778	RELUGOLIX	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	TAK-285	chembl:CHEMBL1614725	TAK-285	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.5834185692854944	NMS-1286937	chembl:CHEMBL1094408	NMS-1286937	FALSE	FALSE	TRUE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:5459	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	2.100306849	LY-2624587	chembl:CHEMBL4594572	LY-2624587	FALSE	FALSE	FALSE
MULTIDRUG RESISTANCE PROTEIN 1	hgnc:40	ABCB1	TTD	2020.06.01	NULL	0.1682938180631233	Biricodar	ncit:C71621	BIRICODAR	FALSE	FALSE	FALSE
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	5.250767123569449	CAR-GPC3 T Cells	ncit:C121638	ANTI-GPC3-CAR AUTOLOGOUS T LYMPHOCYTES	FALSE	FALSE	FALSE
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	5.250767123569449	CAR-GPC3 T cells	ncit:C121638	ANTI-GPC3-CAR AUTOLOGOUS T LYMPHOCYTES	FALSE	FALSE	FALSE
IRON	hgnc:4650	GTF2E1	TTD	2020.06.01	NULL	3.500511415712966	Etidronate Disodium	rxcui:9872	ETIDRONATE DISODIUM	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.7721716358190367	Echothiophate Iodide	rxcui:3740	ECHOTHIOPHATE IODIDE	TRUE	FALSE	FALSE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	0.5097832158805291	Dextrothyroxine Sodium	rxcui:40070	DEXTROTHYROXINE SODIUM	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.065799087	Flurazepam	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.1017590527823536	Isoetharine	rxcui:6023	ISOETHARINE	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.2160809515872201	Nateglinide	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.2386712328895204	Oxtriphylline	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.4861821410712453	Pinacidil	rxcui:33717	PINACIDIL	TRUE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	0.3500511415712966	Talimogene Laherparepvec	rxcui:1721264	TALIMOGENE LAHERPAREPVEC	TRUE	FALSE	FALSE
PARATHYROID HORMONE	hgnc:9606	PTH	TTD	2020.06.01	NULL	0.3365876361262467	Teriparatide	rxcui:32915	TERIPARATIDE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	0.2430910705356227	Tamsulosin	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	0.4318065068724876	Spironolactone	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.8204323630577265	Ecopipam	ncit:C74188	ECOPIPAM	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	0.7001022831425933	MEDI-565	chembl:CHEMBL2109372	MEDI-565	FALSE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	2.663432598912039	obeticholic acid	rxcui:1798288	OBETICHOLIC ACID	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Bevantolol	ncit:C79556	BEVANTOLOL	FALSE	FALSE	FALSE
ORNITHINE DECARBOXYLASE	hgnc:8109	ODC1	TTD	2020.06.01	NULL	2.864054794674245	Eflornithine	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	1.779921058837101	Delapril	ncit:C75022	DELAPRIL	FALSE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.6674703970639131	Deserpidine	rxcui:62174	DESERPIDINE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.596678082	Dexibuprofen	ncit:C166907	DEXIBUPROFEN	TRUE	FALSE	FALSE
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	0.1905904582057876	Dextroamphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.49187514	Levonorgestrel	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.056581542	Podofilox	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.7573221812840553	Pimavanserin	rxcui:1791685	PIMAVANSERIN	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.3182283105193605	Rofecoxib	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	0.6250913242344582	DSP-2230	chembl:CHEMBL5095026	DSP-2230	FALSE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.3918482928036902	GSK1070916A	ncit:C91081	AURORA B/C KINASE INHIBITOR GSK1070916A	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.4922594178346359	GSK2141795	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.067839369	Ganaxolone	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.9376369863516875	ERB-041	ncit:C76959	PRINABEREL	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.7095631248066824	Ensaculin hydrochloride	chembl:CHEMBL1940735	ENSACULIN HYDROCHLORIDE	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.070765056	Sodium butyrate	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	1.721562991334245	Vilaprisan	ncit:C148505	VILAPRISAN	FALSE	FALSE	FALSE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	0.2763561643983921	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	2.917092846427472	ISRAPAFANT	ncit:C65987	ISRAPAFANT	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	1.071585127259071	Sirukumab	ncit:C152371	SIRUKUMAB	FALSE	FALSE	FALSE
MONOCYTE CHEMOTACTIC AND ACTIVATING FACTOR	hgnc:10618	CCL2	TTD	2020.06.01	NULL	2.917092846427472	RS-504393	iuphar.ligand:781	RS-504393	FALSE	FALSE	FALSE
NCBIGENE:1878	ncbigene:1878	E11S	GuideToPharmacology	2024.1	NULL	13.12691780892362	IUPHAR.LIGAND:5081	iuphar.ligand:5081	4-1BB LIGAND	FALSE	FALSE	FALSE
NCBIGENE:1519	hgnc:2542	CTSO	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8009	iuphar.ligand:8009	PHT-427	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.5834185692854944	HBI-8000	ncit:C97263	TUCIDINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.1131630845596864	IUPHAR.LIGAND:8434	iuphar.ligand:8434	LP-12	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.019680536	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.048663273	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.3163112725041837	IUPHAR.LIGAND:110	iuphar.ligand:110	CP-122288	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.070291394	IUPHAR.LIGAND:45	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.062509132	IUPHAR.LIGAND:121	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:110	iuphar.ligand:110	CP-122288	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.089298761	IUPHAR.LIGAND:15	iuphar.ligand:15	L-694,247	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.032899543	IUPHAR.LIGAND:34	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:143	iuphar.ligand:143	SB 277011-A	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1241316104862754	IUPHAR.LIGAND:45	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:174	iuphar.ligand:174	AC-90179	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.005698065	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.019739726	IUPHAR.LIGAND:203	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.036847489	IUPHAR.LIGAND:213	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:249	iuphar.ligand:249	ML 10375	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:226	rxcui:139778	TEGASEROD	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.8899605294185507	IUPHAR.LIGAND:3240	iuphar.ligand:3240	WAY-181187	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.042379073	IUPHAR.LIGAND:87	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	modulator	0.5527123287967842	IUPHAR.LIGAND:10908	iuphar.ligand:10908	BAY1125976	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:8181	iuphar.ligand:8181	COMPOUND 1 [PMID: 20005102]	FALSE	FALSE	FALSE
NCBIGENE:1283	ncbigene:1283	CTD	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:5233	iuphar.ligand:5233	NKY80	FALSE	FALSE	FALSE
NCBIGENE:1382	hgnc:2339	CRABP2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:10262	iuphar.ligand:10262	KV-37	FALSE	FALSE	FALSE
NCBIGENE:174	hgnc:317	AFP	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:3638	rxcui:89959	PHOSPHATIDYLSERINE	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.010213513	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.1651184630053286	IUPHAR.LIGAND:483	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.061919424	IUPHAR.LIGAND:485	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.082559232	IUPHAR.LIGAND:277	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:7381	iuphar.ligand:7381	RS-100329	FALSE	FALSE	FALSE
NCBIGENE:1614	hgnc:13557	ACE2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:7866	iuphar.ligand:7866	MLN-4760	FALSE	FALSE	FALSE
NCBIGENE:688	hgnc:6349	KLF5	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:1773	iuphar.ligand:1773	PCMBS	FALSE	FALSE	FALSE
NCBIGENE:694	hgnc:1130	BTG1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10188	iuphar.ligand:10188	AUPHEN	FALSE	FALSE	FALSE
NCBIGENE:688	hgnc:6349	KLF5	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:4126	iuphar.ligand:4126	AG+	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:601	iuphar.ligand:601	[125I](PYR1)APELIN-13	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	1.029562181092048	IUPHAR.LIGAND:10307	ncit:C65409	DIMINAZENE	FALSE	FALSE	FALSE
NCBIGENE:685	hgnc:1121	BTC	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:10307	ncit:C65409	DIMINAZENE	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:383	iuphar.ligand:383	AS99	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:385	iuphar.ligand:385	8-CYCLOPENTYLTHEOPHYLLINE	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.100589408	IUPHAR.LIGAND:457	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:5616	iuphar.ligand:5616	ATL802	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:8420	iuphar.ligand:8420	UK-432,097	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:397	iuphar.ligand:397	MRS1084	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:455	iuphar.ligand:455	[3H]ZM 241385	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:12150	iuphar.ligand:12150	LJ-4517	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:444	iuphar.ligand:444	DAX	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:386	iuphar.ligand:386	DPCPX	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:446	iuphar.ligand:446	I-ABOPX	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:383	iuphar.ligand:383	AS99	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.025256215	IUPHAR.LIGAND:413	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:3286	iuphar.ligand:3286	PSB1115	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:443	iuphar.ligand:443	BW-A1433	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:6895	iuphar.ligand:6895	L-163,101	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	0.4234489615781814	IUPHAR.LIGAND:2504	rxcui:1999003	ANGIOTENSIN II	TRUE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:11944	iuphar.ligand:11944	TRV026	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:9375	iuphar.ligand:9375	VTX-11E	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8863	ncit:C127116	DUBERMATINIB	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.2206204673768676	IUPHAR.LIGAND:11887	iuphar.ligand:11887	TINENGOTINIB	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:621	iuphar.ligand:621	PD 168368	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:6192	iuphar.ligand:6192	PHENYLACETYL-ALA,DTRP-PHENTHYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9982	iuphar.ligand:9982	COMPOUND 15 [PMID: 25699151]	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.2344092465879218	IUPHAR.LIGAND:9326	ncit:C132738	ABEDITEROL	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:531	iuphar.ligand:531	[3H](-)CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:531	iuphar.ligand:531	[3H](-)CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:12065	iuphar.ligand:12065	BI-167107	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:570	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:565	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
NCBIGENE:2893	hgnc:4574	GRIA4	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:9085	iuphar.ligand:9085	COMPOUND 42 [PMID: 26938474]	FALSE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:6814	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1596	hgnc:210	ADAM3B	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8675	iuphar.ligand:8675	COMPOUND 3 [PMID: 14640538]	FALSE	FALSE	FALSE
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:5294	iuphar.ligand:5294	Z-DEVD-FMK	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:3947	iuphar.ligand:3947	AC265347	FALSE	FALSE	FALSE
NCBIGENE:1622	hgnc:2690	DBI	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:5300	iuphar.ligand:5300	Z-VEID-FMK	FALSE	FALSE	FALSE
NCBIGENE:2347	hgnc:2531	CTSF	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6535	iuphar.ligand:6535	COMPOUND (R)-26 [PMID: 22686657]	FALSE	FALSE	FALSE
NCBIGENE:388	hgnc:668	RHOB	GuideToPharmacology	2024.1	activator	0.098884503	IUPHAR.LIGAND:2377	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:2351	ncbigene:2351	FOLR2L	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10746	iuphar.ligand:10746	VBY-825	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:8705	iuphar.ligand:8705	TM38837	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:9233	ncit:C87598	SURINABANT	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:3316	iuphar.ligand:3316	AM1241	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	inhibitor	7.876150685354174	IUPHAR.LIGAND:889	ncit:C96871	DEXLOXIGLUMIDE	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:864	rxcui:9800	SINCALIDE	TRUE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10164	iuphar.ligand:10164	CCX354	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	0.4039051633514962	IUPHAR.LIGAND:770	iuphar.ligand:770	CCL13	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	3.580068493342807	IUPHAR.LIGAND:887	ncit:C87692	NETAZEPIDE	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:3500	iuphar.ligand:3500	E913	FALSE	FALSE	FALSE
NCBIGENE:66	hgnc:139	ACTBP6	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9252	iuphar.ligand:9252	COMPOUND 24 [PMID: 26987013 ]	FALSE	FALSE	FALSE
NCBIGENE:63	hgnc:136	ACTBP3	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:808	iuphar.ligand:808	CCL20	FALSE	FALSE	FALSE
NCBIGENE:3010	hgnc:4720	H1-6	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:9949	iuphar.ligand:9949	NARATUXIMAB EMTANSINE	FALSE	FALSE	FALSE
NCBIGENE:2863	hgnc:4496	GPR39	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:8460	iuphar.ligand:8460	LULIZUMAB PEGOL	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:7580	rxcui:1876366	OCRELIZUMAB	TRUE	FALSE	FALSE
NCBIGENE:2766	hgnc:4376	GMPR	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12111	iuphar.ligand:12111	MK-0159	FALSE	FALSE	FALSE
NCBIGENE:3104	hgnc:4930	ZBTB48	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:10588	iuphar.ligand:10588	PEPTIDE 5A	FALSE	FALSE	FALSE
NCBIGENE:1874	hgnc:3118	E2F4	GuideToPharmacology	2024.1	antibody	6.563458904461812	IUPHAR.LIGAND:9802	iuphar.ligand:9802	CFZ533	FALSE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	0.2536602475154323	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11936	iuphar.ligand:11936	COMPOUND 14F [PMID: 35063894]	FALSE	FALSE	FALSE
NCBIGENE:2982	hgnc:4685	GUCY1A1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9780	iuphar.ligand:9780	COMPOUND 7F [PMID: 29283260]	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6470	rxcui:60819	BIVALIRUDIN	TRUE	FALSE	FALSE
NCBIGENE:394	hgnc:675	ARHGAP5	GuideToPharmacology	2024.1	blocker	8.751278539282415	IUPHAR.LIGAND:2349	iuphar.ligand:2349	L-(CIS)-DILTIAZEM	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7727	iuphar.ligand:7727	AZ12971554	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.052142673	IUPHAR.LIGAND:5658	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.070765056	IUPHAR.LIGAND:5695	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
NCBIGENE:2360	hgnc:3868	FRA1A	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:11366	iuphar.ligand:11366	OSOCIMAB	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:11192	iuphar.ligand:11192	IACS-9439	FALSE	FALSE	FALSE
NCBIGENE:607	hgnc:1008	BCL9	GuideToPharmacology	2024.1	inhibitor	0.3547815624033412	IUPHAR.LIGAND:2330	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:6661	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:7401	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.029698909	IUPHAR.LIGAND:5239	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:7298	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
NCBIGENE:1424	hgnc:2414	CRYGGP	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8771	iuphar.ligand:8771	COMPOUND 57 [PMID: 16610804]	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:8531	iuphar.ligand:8531	CXCL12&DELTA;	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12207	iuphar.ligand:12207	ACT-660602	FALSE	FALSE	FALSE
NCBIGENE:73	hgnc:146	ACTG1P1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:3662	iuphar.ligand:3662	[125I]CXCL16 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:5861	ncit:C77981	IRALUKAST	FALSE	FALSE	FALSE
NCBIGENE:1341	hgnc:2642	CYP4A11	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12767	iuphar.ligand:12767	TP0472993	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8550	iuphar.ligand:8550	COMPOUND 24DD [PMID: 20684603]	FALSE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:8550	iuphar.ligand:8550	COMPOUND 24DD [PMID: 20684603]	FALSE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:10658	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:1902	iuphar.ligand:1902	15(R)-15-METHYL-PGD2	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.043430663	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.067317527	IUPHAR.LIGAND:939	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.049864835	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.067317527	IUPHAR.LIGAND:933	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.024141458	IUPHAR.LIGAND:940	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.2333674277141977	IUPHAR.LIGAND:954	ncit:C152121	QUINELORANE	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:944	iuphar.ligand:944	SKF-83566	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.022583945	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.023598953	IUPHAR.LIGAND:953	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.1666910197958555	IUPHAR.LIGAND:935	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.060077427	IUPHAR.LIGAND:3300	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.015466177	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:932	iuphar.ligand:932	(+)-ADTN	FALSE	FALSE	FALSE
NCBIGENE:2835	hgnc:4466	GPR12	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12282	ncit:C127114	VALEMETOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12412	iuphar.ligand:12412	COMPOUND 52 [PMID: 36749735]	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:9897	iuphar.ligand:9897	MPPA	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:7252	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:1949	iuphar.ligand:1949	AH23848	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:9912	iuphar.ligand:9912	ALLITINIB	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	NULL	0.4526523382387456	IUPHAR.LIGAND:4948	iuphar.ligand:4948	HB-EGF	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:9922	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.021554873	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:4052	iuphar.ligand:4052	WAY200070	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:4052	iuphar.ligand:4052	WAY200070	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:6700	ncit:C76959	PRINABEREL	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:992	iuphar.ligand:992	[125I]ET-2 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:1010	iuphar.ligand:1010	BQ788	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:3487	ncit:C61606	ATRASENTAN	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:10070	ncit:C174728	APROCITENTAN	TRUE	FALSE	FALSE
NCBIGENE:868	hgnc:1542	CBLB	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:4631	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4347	iuphar.ligand:4347	ZK93426	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4241	iuphar.ligand:4241	L838417	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	agonist	0.1201548540862574	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:4083	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4347	iuphar.ligand:4347	ZK93426	FALSE	FALSE	FALSE
NCBIGENE:413	hgnc:716	ARSC2	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:417	hgnc:723	ART1	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:414	hgnc:717	ARSD	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:418	hgnc:724	ART2P	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6116	iuphar.ligand:6116	GAL-B2-MPEG4	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6104	iuphar.ligand:6104	M1153	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6094	iuphar.ligand:6094	GALANIN(10-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6108	iuphar.ligand:6108	GAL-R2-DPEG24	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3195	iuphar.ligand:3195	COMPOUND 16 [PMID: 18800762]	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:6125	iuphar.ligand:6125	SNAP 398299	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:1095	iuphar.ligand:1095	[125I]TYR-ALA-HEXARELIN	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.090064616	IUPHAR.LIGAND:1136	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4081	iuphar.ligand:4081	[3H]CNQX	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	blocker	1.250182648468916	IUPHAR.LIGAND:4000	iuphar.ligand:4000	NS1738	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5751	ncit:C97962	EZLOPITANT	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:2114	iuphar.ligand:2114	FK-888	FALSE	FALSE	FALSE
NCBIGENE:2860	hgnc:4493	GPR36	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:8453	iuphar.ligand:8453	TAREXTUMAB	FALSE	FALSE	FALSE
NCBIGENE:304	hgnc:539	ANXA2P2	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1502	iuphar.ligand:1502	NEUROPEPTIDE B-29	FALSE	FALSE	FALSE
NCBIGENE:250	hgnc:439	ALPP	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:7049	rxcui:1364468	TEDUGLUTIDE	TRUE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	0.5527123287967842	IUPHAR.LIGAND:4181	drugbank:DB02852	DOMOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	blocker	0.3804903712731485	IUPHAR.LIGAND:2403	ncit:C65450	DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	blocker	0.05853698	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.1693795846312726	IUPHAR.LIGAND:4089	iuphar.ligand:4089	[3H]DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4243	iuphar.ligand:4243	LY233053	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:5978	iuphar.ligand:5978	GSK-3BETA INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:2029	hgnc:3360	ENSA	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:8019	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1166	iuphar.ligand:1166	[125I][DES-GLY10,D-ALA6]GNRH N-ETHYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5791	iuphar.ligand:5791	COMPOUND 2G [PMID: 19309152]	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:4945	iuphar.ligand:4945	GUANYLIN	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.076765601	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:8984	iuphar.ligand:8984	JNJ-39758979	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:1277	iuphar.ligand:1277	JNJ-10191584	FALSE	FALSE	FALSE
NCBIGENE:86	hgnc:24124	ACTL6A	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:1497	iuphar.ligand:1497	[125I]NPW-23 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4354	iuphar.ligand:4354	7&BETA;, 27-DIHYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:85	ncbigene:85	ACTL5	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:12666	iuphar.ligand:12666	EXAMPLE 31 [WO2018183145]	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:5541	iuphar.ligand:5541	R-SPONDIN-3	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:3698	iuphar.ligand:3698	R-SPONDIN-2	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:10171	iuphar.ligand:10171	GLPG1205	FALSE	FALSE	FALSE
NCBIGENE:148	hgnc:277	ADRA1A	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:3698	iuphar.ligand:3698	R-SPONDIN-2	FALSE	FALSE	FALSE
NCBIGENE:304	hgnc:539	ANXA2P2	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1497	iuphar.ligand:1497	[125I]NPW-23 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2625	hgnc:4172	GATA3	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:6831	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1480	iuphar.ligand:1480	PANCREATIC POLYPEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1455	hgnc:2455	CSNK1G2	GuideToPharmacology	2024.1	activator	1.875273972703375	IUPHAR.LIGAND:9249	ncit:C152258	ROSIPTOR	FALSE	FALSE	FALSE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9386	iuphar.ligand:9386	BMS-536924	FALSE	FALSE	TRUE
NCBIGENE:1802	hgnc:3004	DPH2	GuideToPharmacology	2024.1	inhibitor	7.501095890813499	IUPHAR.LIGAND:7423	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8083	iuphar.ligand:8083	ND-2158	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1491	iuphar.ligand:1491	NEUROPEPTIDE S	FALSE	FALSE	FALSE
NCBIGENE:1708	hgnc:6019	IL6R	GuideToPharmacology	2024.1	agonist	0.212581665	IUPHAR.LIGAND:4998	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
NCBIGENE:165	hgnc:303	AEBP1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:9166	iuphar.ligand:9166	[CY5-LYS19]NPS	FALSE	FALSE	FALSE
NCBIGENE:680	hgnc:1113	BRS3	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:10901	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
NCBIGENE:662	hgnc:1082	BNIP1	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:12426	iuphar.ligand:12426	PROCYANIDIN C2	FALSE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12469	iuphar.ligand:12469	BENGALENSOL	FALSE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:12458	iuphar.ligand:12458	ABSINTHIN	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:8403	ncit:C76681	RETOSIBAN	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:9712	iuphar.ligand:9712	COMPOUND 5E [PMID: 28580438]	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:7839	iuphar.ligand:7839	ILGINATINIB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:7913	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:9432	iuphar.ligand:9432	PF-06263276	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:9697	ncit:C152385	SOLCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:7839	iuphar.ligand:7839	ILGINATINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:7971	iuphar.ligand:7971	XL019	FALSE	FALSE	FALSE
NCBIGENE:2376	hgnc:3888	FRA2D	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8655	iuphar.ligand:8655	COMPOUND 5 {PMID: 24900446]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1651	ncit:C80585	NALFURAFINE	FALSE	FALSE	FALSE
NCBIGENE:2132	hgnc:3513	EXT2	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8219	iuphar.ligand:8219	COMPOUND 74 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1648	iuphar.ligand:1648	E2078	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:7362	iuphar.ligand:7362	JDTIC	FALSE	FALSE	FALSE
NCBIGENE:3236	hgnc:5133	HOXD10	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:13033	iuphar.ligand:13033	LY3522348	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:9194	ncit:C170144	ATICAPRANT	FALSE	FALSE	FALSE
NCBIGENE:972	hgnc:1697	CD74	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4665	iuphar.ligand:4665	VU0240551	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9304	iuphar.ligand:9304	TCS 1102	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:9383	iuphar.ligand:9383	OSI-930	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11851	iuphar.ligand:11851	MRTX1133	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.061919424	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2316	iuphar.ligand:2316	LEIUROTOXIN I	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	0.1458546423213736	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2315	iuphar.ligand:2315	LEI-DAB7	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	0.2885036881082116	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:11648	rxcui:2591497	DARIDOREXANT	TRUE	FALSE	FALSE
NCBIGENE:429	hgnc:738	ASCL1	GuideToPharmacology	2024.1	blocker	6.563458904461812	IUPHAR.LIGAND:10382	drugbank:DB11968	MK-7145	FALSE	FALSE	FALSE
NCBIGENE:433	hgnc:743	ASGR2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	0.2983390411119005	IUPHAR.LIGAND:2603	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.1025540453822158	IUPHAR.LIGAND:2603	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:7679	iuphar.ligand:7679	AZD3778	FALSE	FALSE	FALSE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	inhibitor	0.3860858179095184	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:540	hgnc:870	ATP7B	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:10050	iuphar.ligand:10050	VM24	FALSE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.2734774543525755	IUPHAR.LIGAND:2298	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:547	hgnc:888	KIF1A	GuideToPharmacology	2024.1	blocker	0.4861821410712454	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712454	IUPHAR.LIGAND:7465	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.4375639269641209	IUPHAR.LIGAND:2560	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:2562	iuphar.ligand:2562	S9947	FALSE	FALSE	FALSE
NCBIGENE:2138	hgnc:3519	EYA1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8941	iuphar.ligand:8941	COMPOUND 4 [PMID: 24432870]	FALSE	FALSE	FALSE
NCBIGENE:94	hgnc:175	ACVRL1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:2905	iuphar.ligand:2905	AM966	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:5450	iuphar.ligand:5450	VPC32179	FALSE	FALSE	FALSE
NCBIGENE:1240	hgnc:2121	CMKLR1	GuideToPharmacology	2024.1	activator	5.250767124	IUPHAR.LIGAND:5276	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12523	iuphar.ligand:12523	COMPOUND 65 [PMID: 36126387]	FALSE	FALSE	FALSE
NCBIGENE:94	hgnc:175	ACVRL1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:2911	iuphar.ligand:2911	FARNESYL MONOPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7035	iuphar.ligand:7035	H3-COA-20	FALSE	FALSE	FALSE
NCBIGENE:2136	hgnc:16059	PAK4	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8941	iuphar.ligand:8941	COMPOUND 4 [PMID: 24432870]	FALSE	FALSE	FALSE
NCBIGENE:2685	ncbigene:2685	GGTL2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:12807	iuphar.ligand:12807	ZAVONDEMSTAT	FALSE	FALSE	FALSE
NCBIGENE:2094	ncbigene:2094	ERVT4	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12167	iuphar.ligand:12167	GAMCEMETINIB	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1303	iuphar.ligand:1303	7-FLUOROCHROMONE-2-CARBOXAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:8247	iuphar.ligand:8247	LDC1267	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.038608582	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:5709	iuphar.ligand:5709	SGX-523	FALSE	FALSE	FALSE
NCBIGENE:2135	hgnc:3516	EXTL2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8941	iuphar.ligand:8941	COMPOUND 4 [PMID: 24432870]	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3214	iuphar.ligand:3214	DOLICHOL PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:1405	ncit:C83847	ISOSPAGLUMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1434	ncit:C80667	FENOBAM ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6420	iuphar.ligand:6420	COMPOUND 41 [PMID: 23434029]	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6426	iuphar.ligand:6426	COMPOUND 11A [PMID: 14697765]	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	0.8751278539282416	IUPHAR.LIGAND:1416	iuphar.ligand:1416	PHCCC	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1399	iuphar.ligand:1399	[3H]LY341495	FALSE	FALSE	FALSE
NCBIGENE:2137	hgnc:3518	EXTL3	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8941	iuphar.ligand:8941	COMPOUND 4 [PMID: 24432870]	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:3336	iuphar.ligand:3336	MTEP	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:1415	iuphar.ligand:1415	MPPG	FALSE	FALSE	FALSE
NCBIGENE:2100	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:12936	iuphar.ligand:12936	PCC0105003	FALSE	FALSE	FALSE
NCBIGENE:2097	hgnc:3464	ESB3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12936	iuphar.ligand:12936	PCC0105003	FALSE	FALSE	FALSE
NCBIGENE:2099	hgnc:3467	ESR1	GuideToPharmacology	2024.1	inhibitor	0.1226814748497534	IUPHAR.LIGAND:12937	iuphar.ligand:12937	PCC0208017	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	0.729273212	IUPHAR.LIGAND:2373	rxcui:6069	IVERMECTIN	TRUE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:9973	iuphar.ligand:9973	COMPOUND 27 [PMID: 29775310]	FALSE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:8014	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	0.046840028	IUPHAR.LIGAND:2377	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8842	iuphar.ligand:8842	COMPOUND 35 [PMID: 23916259]	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:7817	ncit:C79841	TALMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4147	iuphar.ligand:4147	BRILLIANT BLUE G	FALSE	FALSE	FALSE
NCBIGENE:2080	hgnc:6857	MAP3K5	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10602	iuphar.ligand:10602	COMPOUND 26 [PMID: 31710475]	FALSE	FALSE	FALSE
NCBIGENE:2073	hgnc:3437	ERCC5	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9355	iuphar.ligand:9355	GNE-3511	FALSE	FALSE	FALSE
NCBIGENE:1634	hgnc:2705	DCN	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	1.093909817410302	IUPHAR.LIGAND:5953	iuphar.ligand:5953	CHELERYTHRINE	FALSE	FALSE	FALSE
NCBIGENE:2087	ncbigene:2087	ERVK2	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:2086	hgnc:3454	ERV3-1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625569	IUPHAR.LIGAND:9693	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:7823	iuphar.ligand:7823	AZD6605	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:7722	iuphar.ligand:7722	AZ11657312 (SALT FREE)	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5288	iuphar.ligand:5288	WAY170523	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6468	ncit:C1705	TANOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1638	hgnc:2709	DCT	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:12057	iuphar.ligand:12057	TP0556351	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:7823	iuphar.ligand:7823	AZD6605	FALSE	FALSE	FALSE
NCBIGENE:1630	hgnc:2701	DCC	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8846	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:1784	iuphar.ligand:1784	UDP-GLUCURONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:11816	iuphar.ligand:11816	ABD-1970	FALSE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:8846	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11742	ncit:C169812	BIFEMELANE	FALSE	FALSE	FALSE
NCBIGENE:988	hgnc:1743	CDC5L	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8813	iuphar.ligand:8813	COMPOUND 30 [PMID: 16455256]	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:1772	iuphar.ligand:1772	CLOPIDOGREL (ACTIVE METABOLITE)	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:3278	iuphar.ligand:3278	[11C]XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:8593	iuphar.ligand:8593	[3H]ACETYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:321	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:319	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.045898314	IUPHAR.LIGAND:359	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.078958904	IUPHAR.LIGAND:9658	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.276356164	IUPHAR.LIGAND:8592	iuphar.ligand:8592	[3H]TIOTROPIUM	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1364	iuphar.ligand:1364	5-METHOXY-LUZINDOLE	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:10666	iuphar.ligand:10666	UCSF7447	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1359	iuphar.ligand:1359	K185	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:1664	iuphar.ligand:1664	NALOXONE BENZOYLHYDRAZONE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	modulator	0.5770073762164231	IUPHAR.LIGAND:9157	iuphar.ligand:9157	BMS-986122	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:9471	iuphar.ligand:9471	MRS4183	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:3534	rxcui:56795	SUFENTANIL	TRUE	FALSE	FALSE
NCBIGENE:3141	hgnc:4976	HLCS	GuideToPharmacology	2024.1	activator	26.25383561784724	IUPHAR.LIGAND:11142	iuphar.ligand:11142	NATURAL CYTOTOXICITY TRIGGERING RECEPTOR 3 LIGAND 1	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.1319288222002374	IUPHAR.LIGAND:1756	iuphar.ligand:1756	AR-C67085	FALSE	FALSE	FALSE
NCBIGENE:1749	hgnc:2918	DLX5	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:5036	iuphar.ligand:5036	OSTEOCRIN	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:7537	iuphar.ligand:7537	NORZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	modulator	1.810609352954982	IUPHAR.LIGAND:12223	ncit:C72600	PONAZURIL	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:12087	iuphar.ligand:12087	ANIZATRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:4636	iuphar.ligand:4636	[3H]NISOXETINE	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:5685	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:12237	iuphar.ligand:12237	CH7057288	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:12377	iuphar.ligand:12377	EMZELTRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:1725	iuphar.ligand:1725	PPADS	FALSE	FALSE	FALSE
NCBIGENE:470	ncbigene:470	ATHS	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3964	iuphar.ligand:3964	&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	modulator	1.250182648468916	IUPHAR.LIGAND:3992	iuphar.ligand:3992	LY2087101	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1743	iuphar.ligand:1743	ITP	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:2116	iuphar.ligand:2116	MEN 10376	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1679	iuphar.ligand:1679	AC-RYYRIK-NH2	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:9009	iuphar.ligand:9009	NM4-C16	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:5814	iuphar.ligand:5814	PI1	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:5815	iuphar.ligand:5815	QA1	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1859	ncit:C77989	APAFANT	FALSE	FALSE	FALSE
NCBIGENE:2823	hgnc:4460	GPM6A	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8024	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:3390	iuphar.ligand:3390	5S-HETE	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:2483	iuphar.ligand:2483	5S-HPETE	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:12604	iuphar.ligand:12604	CVN45502	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.1319288222002374	IUPHAR.LIGAND:1773	iuphar.ligand:1773	PCMBS	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:1736	ncit:C65436	DIQUAFOSOL	FALSE	FALSE	FALSE
NCBIGENE:2590	hgnc:4124	GALNT2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11433	ncit:C77404	CETILISTAT	FALSE	FALSE	FALSE
NCBIGENE:347	hgnc:612	APOD	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:10971	iuphar.ligand:10971	SCH-79797	FALSE	FALSE	FALSE
NCBIGENE:347	hgnc:612	APOD	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:4047	rxcui:1537034	VORAPAXAR	TRUE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:4702	iuphar.ligand:4702	4-AMBA	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	modulator	0.9053046764774912	IUPHAR.LIGAND:9560	iuphar.ligand:9560	AZ3451	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	1.544343271638073	IUPHAR.LIGAND:12597	iuphar.ligand:12597	[3H]MIROGABALIN	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9878	iuphar.ligand:9878	6-HYDROXY-5,7-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:12518	iuphar.ligand:12518	NERANDOMILAST	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.3182283105193606	IUPHAR.LIGAND:12287	iuphar.ligand:12287	CHIGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12518	iuphar.ligand:12518	NERANDOMILAST	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:5922	iuphar.ligand:5922	AKT INHIBITOR X	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:9367	iuphar.ligand:9367	LGB321	FALSE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.041377203	IUPHAR.LIGAND:4807	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:10618	ncit:C175203	SERALUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:11510	iuphar.ligand:11510	M4205	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.065634589	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:2751	hgnc:4340	GLUD1P5	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11388	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.043756393	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:12143	iuphar.ligand:12143	WNY0824	FALSE	FALSE	FALSE
NCBIGENE:1434	hgnc:2431	CSE1L	GuideToPharmacology	2024.1	activator	8.751278539282415	IUPHAR.LIGAND:5305	iuphar.ligand:5305	ADP-RIBOSYLATION FACTOR 1	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.1312691780892362	IUPHAR.LIGAND:10658	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:10073	iuphar.ligand:10073	COMPOUND 6 [PMID: 30125504]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:10618	ncit:C175203	SERALUTINIB	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	0.4412409347537352	IUPHAR.LIGAND:5666	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12904	iuphar.ligand:12904	COMPOUND (S)-29 [PMID: 37606563]	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:12905	iuphar.ligand:12905	DUAL VEGFR/PARP INHIBITOR 14B	FALSE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:12345	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
NCBIGENE:2170	hgnc:3557	FABP3	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:5666	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:9928	iuphar.ligand:9928	PUQUITINIB	FALSE	FALSE	FALSE
NCBIGENE:2171	hgnc:3560	FABP5	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12083	iuphar.ligand:12083	OCIFISERTIB	FALSE	FALSE	FALSE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11749	iuphar.ligand:11749	ONAMETOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:11627	ncit:C96718	PICLAMILAST	FALSE	FALSE	FALSE
NCBIGENE:1252	hgnc:5187	PRMT1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7037	iuphar.ligand:7037	C21	FALSE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:8739	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:12059	iuphar.ligand:12059	COMPOUND 23 [PMID: 35816678]	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	activator	0.3281729452230906	IUPHAR.LIGAND:7443	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
NCBIGENE:1432	hgnc:6876	MAPK14	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:6696	ncit:C72985	DARAPLADIB	FALSE	FALSE	FALSE
NCBIGENE:1486	hgnc:2496	CTBS	GuideToPharmacology	2024.1	inhibitor	0.1229687850953032	IUPHAR.LIGAND:7946	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
NCBIGENE:1484	ncbigene:1484	CTAA2	GuideToPharmacology	2024.1	activator	0.546954909	IUPHAR.LIGAND:7443	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
NCBIGENE:1488	hgnc:2495	CTBP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11186	ncit:C124796	DAROVASERTIB	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8034	iuphar.ligand:8034	CCG-203920	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:5887	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:11845	iuphar.ligand:11845	COMPOUND 1 [PMID: 34917254]	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:6431	iuphar.ligand:6431	TRIAZINE COMPOUND PC7	FALSE	FALSE	FALSE
NCBIGENE:611	hgnc:1012	OPN1SW	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:2816	iuphar.ligand:2816	UVI3003	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.060077427	IUPHAR.LIGAND:5658	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.2282942227638891	IUPHAR.LIGAND:9921	iuphar.ligand:9921	TAFETINIB	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8205	iuphar.ligand:8205	COMPOUND 22 [PMID: 20462760]	FALSE	FALSE	FALSE
NCBIGENE:2393	hgnc:3905	FRA5A	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:6498	iuphar.ligand:6498	WX-UK1	FALSE	FALSE	FALSE
NCBIGENE:2630	hgnc:4178	GBA1LP	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:4802	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:4374	iuphar.ligand:4374	EUROPIUM-LABELLED RELAXIN-3-B/INSL5 A CHIMERA	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.1312691780892362	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	0.5707355569097228	IUPHAR.LIGAND:1990	iuphar.ligand:1990	RELAXIN-3	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.1666910197958555	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.039390601	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:2708	hgnc:10886	SIRT2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9251	iuphar.ligand:9251	COMPOUND 86 [PMID: 26982234]	FALSE	FALSE	FALSE
NCBIGENE:922	hgnc:1690	CD5L	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:4820	rxcui:4331	FENOPROFEN	TRUE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.1312691780892362	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:6678	iuphar.ligand:6678	PRE-084	FALSE	FALSE	FALSE
NCBIGENE:2707	hgnc:4285	GJB3	GuideToPharmacology	2024.1	activator	8.751278539282415	IUPHAR.LIGAND:9514	iuphar.ligand:9514	SIRT1 ACTIVATOR 3	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:6680	iuphar.ligand:6680	BD-1047	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	agonist	6.300920548	IUPHAR.LIGAND:6683	iuphar.ligand:6683	[3H]PENTAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:8199	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
NCBIGENE:1721	hgnc:9446	PRLR	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:4894	iuphar.ligand:4894	CHORIONIC SOMATOMAMMOTROPIN HORMONE-LIKE 1	FALSE	FALSE	FALSE
NCBIGENE:2520	hgnc:4164	GAST	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10054	iuphar.ligand:10054	SPHINGOMYELIN SYNTHASE 2 INHIBITOR 15W	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10217	iuphar.ligand:10217	SLC4101431	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2013	iuphar.ligand:2013	KE 108	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:5263	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2019	iuphar.ligand:2019	SRIF-14	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2003	iuphar.ligand:2003	BIM 23050	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:5643	iuphar.ligand:5643	GA-NODAGA-LM3	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2019	iuphar.ligand:2019	SRIF-14	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2007	iuphar.ligand:2007	CORTISTATIN-14	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:2062	iuphar.ligand:2062	[125I]TYR3 SMS 201-995	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.2524407270946851	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:3247	ncbigene:3247	HPFH2	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:12907	iuphar.ligand:12907	BEXMARILIMAB	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:5693	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
NCBIGENE:3243	hgnc:11717	TEAD4	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12814	iuphar.ligand:12814	GNE-7883	FALSE	FALSE	FALSE
NCBIGENE:2257	hgnc:3668	FGF12	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:1486	hgnc:2496	CTBS	GuideToPharmacology	2024.1	inhibitor	0.5770073762164232	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:392	hgnc:673	ARHGAP1	GuideToPharmacology	2024.1	blocker	0.3889457128569962	IUPHAR.LIGAND:2406	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1949	iuphar.ligand:1949	AH23848	FALSE	FALSE	FALSE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	activator	6.563458904461812	IUPHAR.LIGAND:11848	iuphar.ligand:11848	TPC2-A1-N	FALSE	FALSE	FALSE
NCBIGENE:3015	hgnc:4741	H2AZ1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12803	iuphar.ligand:12803	COMPOUND 11 [PMID: 37449845]	FALSE	FALSE	FALSE
NCBIGENE:1484	ncbigene:1484	CTAA2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:5693	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.6482428547616604	IUPHAR.LIGAND:8194	iuphar.ligand:8194	COMPOUND 15B [PMID: 16539403]	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	2.282942227638891	IUPHAR.LIGAND:4293	iuphar.ligand:4293	PYR3	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.5707355569097228	IUPHAR.LIGAND:2443	iuphar.ligand:2443	ACAA	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:12529	iuphar.ligand:12529	GSK2332255B	FALSE	FALSE	FALSE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10374	iuphar.ligand:10374	I-C11	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.1041818873724097	IUPHAR.LIGAND:2593	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	inhibitor	0.05068308	IUPHAR.LIGAND:2330	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	1.500219178	IUPHAR.LIGAND:4091	iuphar.ligand:4091	[3H]RESINIFERATOXIN	FALSE	FALSE	FALSE
NCBIGENE:3084	hgnc:7997	NRG1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:10374	iuphar.ligand:10374	I-C11	FALSE	FALSE	FALSE
NCBIGENE:504	hgnc:828	ATP5F1AP2	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:2441	iuphar.ligand:2441	SKF96365	FALSE	FALSE	FALSE
NCBIGENE:511	hgnc:3145	TRPV5	GuideToPharmacology	2024.1	blocker	0.9376369863516875	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:10147	iuphar.ligand:10147	JAK INHIBITOR 20A	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:7839	iuphar.ligand:7839	ILGINATINIB	FALSE	FALSE	FALSE
NCBIGENE:1013	hgnc:1754	CDH15	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:4762	iuphar.ligand:4762	[123I]IODOBENZOVESAMICOL	FALSE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:10388	iuphar.ligand:10388	SZM594	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:3531	iuphar.ligand:3531	SB-611812	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2280	iuphar.ligand:2280	HELODERMIN	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.092606122	IUPHAR.LIGAND:2182	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2214	iuphar.ligand:2214	D(CH2)5[D-ILE2,ILE4,ALA-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:3813	iuphar.ligand:3813	[3H]D(CH2)5[TYR(ME)2]AVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2195	iuphar.ligand:2195	OH-LVA	FALSE	FALSE	FALSE
NCBIGENE:611	hgnc:1012	OPN1SW	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2807	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:1520	iuphar.ligand:1520	[125I]PYY (PIG)	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1544	iuphar.ligand:1544	[D-TRP32]NPY	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	CIViC	10-Apr-24	NULL	0.011925431	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.01214331	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	0.5125748858722557	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.546954909	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	1.250182648468916	SAVOLITINIB	ncit:C104732	SAVOLITINIB	FALSE	FALSE	TRUE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8910	iuphar.ligand:8910	SAR407899	FALSE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.3125456621172291	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.075768645	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.005483257	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
RICTOR	hgnc:28611	RICTOR	CIViC	10-Apr-24	NULL	1.071585127259071	VISTUSERTIB	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	1.250182648468916	JQEZ5	iuphar.ligand:9332	JQEZ5	FALSE	FALSE	TRUE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:4172	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	CIViC	10-Apr-24	NULL	0.4055851016423223	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.1374546367426557	U0126	iuphar.ligand:5282	U0126	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	CIViC	10-Apr-24	NULL	0.1193356164447602	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.056622219	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	0.036770078	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:11915	iuphar.ligand:11915	INSL5 ANALOGUE 13	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	CIViC	10-Apr-24	NULL	0.008103036	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SMAD4	hgnc:6770	SMAD4	CIViC	10-Apr-24	NULL	0.088248187	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
TFF3	hgnc:11757	TFF3	CIViC	10-Apr-24	NULL	0.4039051633514962	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
EGF	hgnc:3229	EGF	CIViC	10-Apr-24	NULL	0.4861821410712454	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4303	iuphar.ligand:4303	RYANODINE	FALSE	FALSE	FALSE
PDCD1LG2	hgnc:18731	PDCD1LG2	CIViC	10-Apr-24	NULL	0.750109589	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
AURKA	hgnc:11393	AURKA	CIViC	10-Apr-24	NULL	0.00747866	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PTPRF	hgnc:9670	PTPRF	CIViC	10-Apr-24	NULL	17.50255707856483	ERLOTINIB HYDROCHLORIDE	rxcui:477320	ERLOTINIB HYDROCHLORIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.017386646	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	CIViC	10-Apr-24	NULL	0.059219178	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:4303	iuphar.ligand:4303	RYANODINE	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:7436	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.1988926940746004	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.1691976516724849	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.118072806	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1637453364938497	ENZALUTAMIDE	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	CIViC	10-Apr-24	NULL	0.008240375	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:2707	hgnc:4285	GJB3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8101	iuphar.ligand:8101	SPLITOMICIN	FALSE	FALSE	FALSE
PTP4A3	hgnc:9636	PTP4A3	CIViC	10-Apr-24	NULL	0.7292732116068681	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
KDM5C	hgnc:11114	KDM5C	CIViC	10-Apr-24	NULL	0.1785975212098452	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.045421861	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NCBIGENE:1170	hgnc:13448	SLC38A2	GuideToPharmacology	2024.1	NULL	10.50153425	IUPHAR.LIGAND:4542	rxcui:426	ALANINE	TRUE	FALSE	FALSE
ETV4	hgnc:3493	ETV4	CIViC	10-Apr-24	NULL	0.525076712	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.010001461	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.0545251	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.028598949	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.5527123287967841	TYROSINE KINASE INHIBITOR SU5402	ncit:C1725	TYROSINE KINASE INHIBITOR SU5402	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	CIViC	10-Apr-24	NULL	0.044878351	BAFETINIB	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	CIViC	10-Apr-24	NULL	1.193356164447602	LOMUSTINE	rxcui:6466	LOMUSTINE	TRUE	FALSE	TRUE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:11905	ncit:C171901	ENAVOGLIFLOZIN	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.006714536	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1988926940746003	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.7192831676122533	Elimusertib	ncit:C146807	ELIMUSERTIB	FALSE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.090922374	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.1106589488634236	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	0.4375639269641208	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.2187819634820604	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.5527123287967842	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:8201	rxcui:2105845	GLASDEGIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.2647445608522412	Cemiplimab	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.2059124362184097	Vactosertib	ncit:C116357	VACTOSERTIB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.235474617310458	CS1003	ncit:C156726	NOFAZINLIMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	MT-6402	ncit:C181982	ENGINEERED TOXIN BODY TARGETING PD-L1 MT-6402	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.1223955040459079	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.044198376	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	2.092697042002317	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	5.527123287967842	MRK-003	drugbank:DB17015	MRK-003	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.2453629496995069	Zotatifin	ncit:C165746	ZOTATIFIN	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.02726255	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6783936852156912	Infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.006659185	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.016005996	Tamatinib	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2546668357992238	Tandutinib	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.064824285	Altiratinib	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.029465584	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.8444216134395313	Tipifarnib	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.4375639269641209	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.2917092846427472	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	2.187819634820604	Vorasidenib	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.1902451856365742	Lestaurtinib	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.1902451856365742	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.031707531	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	YM-254890	iuphar.ligand:9335	YM-254890	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.045369532	Gedatolisib	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.07699072	BI-847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1725162436059257	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2991890098899972	Taselisib	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	1.810609352954982	Fostamatinib	rxcui:2044896	FOSTAMATINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.2592971419046642	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.4254093734373397	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.018540844	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.1093909817410302	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	1.093909817410302	SAF-189s	ncit:C175475	FORITINIB SUCCINATE	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.2263261691193728	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.015454797	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.053815809	Adavosertib	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.014049815	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.007727398	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1931849567170511	RG7112	drugbank:DB14793	RO-5045337	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.021733308	Navitoclax	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.2318219480604613	CHIR-124	drugbank:DB06852	CHIR-124	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.009272878	Topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	modulator	1.050153425	SOLITOMAB	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006987979	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.027752469	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.048618214	NEOSTIGMINE BROMIDE	rxcui:82055	NEOSTIGMINE BROMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.047432404	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.075333818	CA4P	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TSC1	hgnc:12362	TSC1	PharmGKB	4/5/24	NULL	0.1861974157294131	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P29275	hgnc:264	ADORA2B	TdgClinicalTrial	Jan-14	NULL	0.3241214273808303	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.0545251	MEGESTROL	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.075333818	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.1521961485092594	Zoledronic acid	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	0.1403948428761885	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007378818	CYPROHEPTADINE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.1250182648468916	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	TREQUINSIN HYDROCHLORIDE	chembl:CHEMBL1256910	TREQUINSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.009723643	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	1.875273972703375	GNF-PF-574	chembl:CHEMBL582737	CHEMBL:CHEMBL582737	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	PHENANTHRIDIN-6(5H)-ONE	chembl:CHEMBL45245	CHEMBL:CHEMBL45245	FALSE	FALSE	FALSE
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	0.9546849315580819	DIFFERENTIATION AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.072927321	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.057574201	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
UNIPROT:P41595	hgnc:5294	HTR2B	TEND	1-Aug-11	NULL	0.3125456621172291	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.075010959	IUPHAR.LIGAND:933	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:1011	hgnc:1752	CDH12P2	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	(S)-NITRENDIPINE	chembl:CHEMBL251230	(S)-NITRENDIPINE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	SJ000001516	chembl:CHEMBL592316	CHEMBL:CHEMBL592316	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.2983390411119005	SJ000116228	chembl:CHEMBL577887	CHEMBL:CHEMBL577887	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	NCI	14-Sep-17	NULL	0.084553416	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	TALC	12-May-16	antibody	0.9723642821424907	TREMELIMUMAB	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	0.2941606231691568	Exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.061919424	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.007174649	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.052090944	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1442518440541057	VIT C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	4.773424657790408	LB80380	chembl:CHEMBL1652128	LB80380	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	DINALINE	ncit:C79870	DINALINE	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.1795134059339982	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	1.029562181092049	THYMOSIN FRACTION 5	ncit:C2700	HUMAN THYMOSIN-FRACTION 5	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.038104261	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.2083637747448194	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.09963505	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	10.50153424713889	Novaferon	chembl:CHEMBL4650410	NOVAFERON	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2B	hgnc:282	ADRA2B	TTD	2020.06.01	NULL	0.1562728310586145	MEDETOMIDINE	rxcui:52016	MEDETOMIDINE	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:7707	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	0.3409589041278863	TENOFOVIR	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.03151721	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	GSK163929	chembl:CHEMBL1784521	CHEMBL:CHEMBL1784521	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.055441823	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.081281225	Alprazolam	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:6179	iuphar.ligand:6179	(D-ALA11]BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.072324616	IUPHAR.LIGAND:359	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	NSC-145669	chembl:CHEMBL191611	CHEMBL:CHEMBL191611	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.007905401	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:12039	ncit:C171675	APARARENONE	FALSE	FALSE	FALSE
APC	hgnc:583	APC	NCI	14-Sep-17	NULL	0.072324616	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	OncoKB	23-Jul-20	NULL	5.469549087051511	Enasidenib	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.2163777660811586	ITI-007	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
NCBIGENE:235	hgnc:4045	FZD7	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:10324	iuphar.ligand:10324	FZ7-21	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	AM-630	iuphar.ligand:750	AM-630	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	TETROQUINONE	chembl:CHEMBL1329029	TETROQUINONE	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.025663573	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001770916	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NCBIGENE:2599	hgnc:1375	CA4	GuideToPharmacology	2024.1	inhibitor	0.4861821410712454	IUPHAR.LIGAND:7147	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	4.500657534488099	AFEGOSTAT	ncit:C83520	AFEGOSTAT	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	TCMDC-125180	chembl:CHEMBL586163	CHEMBL:CHEMBL586163	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014160645	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1193356164447602	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NCBIGENE:1530	hgnc:10435	RPS6KA6	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8038	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
DCN	hgnc:2705	DCN	NCI	14-Sep-17	NULL	1.500219178	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.043665423	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:178	iuphar.ligand:178	LY063518	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	TRICLOSAN	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	1.381780822	CYANIDIN	chembl:CHEMBL404515	CYANIDIN	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.086219493	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.048708415	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.016992774	CANDESARTAN CILEXETIL	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TRIPROLIDINE HYDROCHLORIDE	rxcui:71534	TRIPROLIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	TOSYL-L-LYSINE CHLOROMETHYL KETONE	chembl:CHEMBL466465	CHEMBL:CHEMBL466465	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.09963505	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
LIPA	hgnc:6617	LIPA	NCI	14-Sep-17	NULL	0.5303805175322677	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	0.3387591692625452	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	CIViC	10-Apr-24	NULL	5.469549087051511	ENASIDENIB	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.062509132	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.032362201	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9993	iuphar.ligand:9993	RILZABRUTINIB	FALSE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DL1	hgnc:6329	KIR2DL1	TTD	2020.06.01	NULL	5.834185692854944	IPH-2102	chembl:CHEMBL2109500	LIRILUMAB	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.04321619	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	BIX-01294	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2229	iuphar.ligand:2229	SKF-105494	FALSE	FALSE	FALSE
ERCC2	hgnc:3434	ERCC2	CIViC	10-Apr-24	NULL	0.044198376	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	CIViC	10-Apr-24	NULL	0.4102161815288632	EPZ004777	iuphar.ligand:7377	EPZ004777	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	OncoKB	23-Jul-20	NULL	0.2778183663264259	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
CYP2A7	hgnc:2611	CYP2A7	PharmGKB	4/5/24	NULL	0.5834185692854944	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	0.546954909	AVB-S6-500	ncit:C156017	BATIRAXCEPT	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA-2/DELTA-1	hgnc:1399	CACNA2D1	TTD	2020.06.01	NULL	0.2500365296937833	Nitrendipine	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11144	iuphar.ligand:11144	COMPOUND 49 [PMID: 30889352]	FALSE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	binder	2.386712328895204	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	DILTIAZEM	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.093098708	EXISULIND	ncit:C1239	EXISULIND	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	RU-24969	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
QUINONE REDUCTASE 1	hgnc:2874	NQO1	TTD	2020.06.01	NULL	2.019525817	ARQ 761	ncit:C99146	BETA-LAPACHONE PRODRUG ARQ 761	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.8950171233357017	Hexylcaine	rxcui:26879	HEXYLCAINE	TRUE	FALSE	FALSE
BILE-SALT-ACTIVATED LIPASE	hgnc:1848	CEL	TTD	2020.06.01	NULL	7.501095891	Bucelipase alfa	ncit:C166667	BUCELIPASE ALFA	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:8260	ncit:C79485	AVOSENTAN	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	0.3025133322221082	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.031254566	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	agonist	0.8751278539282416	NONABINE	ncit:C72950	NONABINE	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	0.8514757497680189	BINODENOSON	ncit:C174671	BINODENOSON	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	CHLORPHENIRAMINE MALEATE	rxcui:142429	CHLORPHENIRAMINE MALEATE	TRUE	FALSE	FALSE
SIRT5	hgnc:14933	SIRT5	DTC	9/2/20	NULL	0.5181678082469852	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
UNIPROT:P28907	hgnc:1667	CD38	TdgClinicalTrial	Jan-14	NULL	23.33674277141977	SAR650984	rxcui:2282018	ISATUXIMAB	TRUE	FALSE	FALSE
UNIPROT:P13569	hgnc:1884	CFTR	TdgClinicalTrial	Jan-14	NULL	8.353493151133215	VX-809	rxcui:1655922	LUMACAFTOR	TRUE	FALSE	FALSE
PROTEIN DELTA HOMOLOG 1	hgnc:2907	DLK1	TTD	2020.06.01	NULL	26.25383561784724	GDC0134	iuphar.ligand:11506	GDC-0134	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.5000730593875666	(-)-OLEOCANTHAL	iuphar.ligand:6308	OLEOCANTHAL	FALSE	FALSE	FALSE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.056097939	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	2.838252499226729	Figopitant	ncit:C81498	FIGOPITANT	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	ChEMBL	33	inhibitor	2.100306849	OTILIMAB	ncit:C170271	OTILIMAB	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:12597	iuphar.ligand:12597	[3H]MIROGABALIN	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:12345	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.010923169	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	TD-1211	chembl:CHEMBL3137313	AXELOPRAN	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.069089041	Halazepam	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.2470949234620917	PRAMIPEXOLE	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.4953553890159858	PARTHENOLIDE	rxcui:32941	PARTHENOLIDE	FALSE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.2134458180312784	4SC-202	drugbank:DB13101	4SC-202	FALSE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.3680444245492605	ARQ 087	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	1.750255707856483	articaine / epinephrine	wikidata:Q48566634	ARTICAINE / EPINEPHRINE	FALSE	FALSE	FALSE
NCBIGENE:531	hgnc:1393	CACNA1F	GuideToPharmacology	2024.1	inhibitor	0.04464938	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:11869	ncit:C162676	ELZOVANTINIB	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:9760	iuphar.ligand:9760	NNC1702	FALSE	FALSE	FALSE
NCBIGENE:1836	hgnc:10994	SLC26A2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:7953	iuphar.ligand:7953	BMS-777607	FALSE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.010518364	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.053038052	ketoconazole	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
HEPATOCYTE GROWTH FACTOR	hgnc:4893	HGF	TTD	2020.06.01	NULL	0.4861821410712453	ABI-011	ncit:C116890	NANOPARTICLE ALBUMIN-BOUND THIOCOLCHICINE DIMER NAB-5404	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-4	hgnc:3682	FGF4	TTD	2020.06.01	NULL	10.50153424713889	Ad5FGF-4	ncit:C184852	ALFERMINOGENE TADENOVEC	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.07631929	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:10107	iuphar.ligand:10107	TUG-1375	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.1691068316769549	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	modulator	1.944728564284981	CENERIMOD	ncit:C169837	CENERIMOD	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.2365210416022274	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.014299475	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:9496	iuphar.ligand:9496	A-971432	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.051885051	SARIZOTAN HYDROCHLORIDE	ncit:C76654	SARIZOTAN HYDROCHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003840807	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.089756703	telithromycin	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.2647445608522412	cemiplimab-rwlc	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
NCBIGENE:2093	ncbigene:2093	ERVT3	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8064	iuphar.ligand:8064	BIX02188	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4017	iuphar.ligand:4017	AC262620	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1691068316769549	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6091	iuphar.ligand:6091	GALANIN(3-29) (PIG)	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.546954909	MK-2201	chembl:CHEMBL3545000	MK-2201	FALSE	FALSE	FALSE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.058341857	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008103036	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1591141552596803	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.050488145	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.2725311655831894	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.091159151	IUPHAR.LIGAND:2829	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.033821366	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	0.2763561643983921	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
APH1B	hgnc:24080	APH1B	ChEMBL	33	inhibitor	1.009762908	AVAGACESTAT	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
REN	hgnc:9958	REN	ChEMBL	33	inhibitor	10.50153424713889	IMARIKIREN HYDROCHLORIDE	chembl:CHEMBL3969876	IMARIKIREN HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.006977764	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.028290771	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.022889133	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.069180068	AMINEPTINE	rxcui:17698	AMINEPTIN	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	1.591141552596803	BUSERELIN	rxcui:1825	BUSERELIN	TRUE	FALSE	FALSE
UNIPROT:P47901	hgnc:896	AVPR1B	TdgClinicalTrial	Jan-14	NULL	1.666910197958555	DESMOPRESSIN	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.069180068	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2218633995874415	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.029399592	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.060772768	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.081281225	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002623285	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	1.312691780892362	SJ000047241	chembl:CHEMBL601933	CHEMBL:CHEMBL601933	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.011124507	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.1704794520639431	OLOMOUCINE	drugbank:DB02116	OLOMOUCINE	FALSE	FALSE	FALSE
BMP2	hgnc:1069	BMP2	DTC	9/2/20	NULL	4.375639269641208	BUTAMBEN	rxcui:19861	BUTAMBEN	TRUE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.729273212	SJ000040837	chembl:CHEMBL590672	CHEMBL:CHEMBL590672	FALSE	FALSE	FALSE
TNFSF10	hgnc:11925	TNFSF10	NCI	14-Sep-17	NULL	1.750255707856483	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
NPPA-AS1	hgnc:37635	NPPA-AS1	PharmGKB	4/5/24	NULL	1.944728564284981	bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.023171964	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.008448539	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1682938180631233	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613069	IUPHAR.LIGAND:8431	iuphar.ligand:8431	DR-4004	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.052142673	IUPHAR.LIGAND:5658	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6185	iuphar.ligand:6185	[D-PRO4,D-TRP7,9,10]SUBSTANCE P (4-11)	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.067059606	IUPHAR.LIGAND:7199	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
NCBIGENE:1795	hgnc:2989	DOCK3	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:7797	ncit:C116891	GALUNISERTIB	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	NEOMYCIN SULFATE	rxcui:7300	NEOMYCIN SULFATE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.005135727	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.068191781	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	4-NONYLPHENOL	rxcui:1788868	4-NONYLPHENOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	6-3'-DIMETHYLFLAVONE	chembl:CHEMBL137498	CHEMBL:CHEMBL137498	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2004	iuphar.ligand:2004	BIM 23052	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:1377	iuphar.ligand:1377	DCG-IV	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.7095631248066824	IMARADENANT	ncit:C148039	IMARADENANT	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.019607047	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.2332563532602643	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.040390516	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.4070362111294147	HMPL-453	chembl:CHEMBL4650297	HMPL-453	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:2026	iuphar.ligand:2026	BIM 23454	FALSE	FALSE	FALSE
PGP	hgnc:8909	PGP	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1620607136904151	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PSMC3	hgnc:9549	PSMC3	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2024	iuphar.ligand:2024	[125I]TYR10-CST14	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	OXITRIPTAN	rxcui:94	5-HYDROXYTRYPTOPHAN	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1029562181092048	TCMDC-123730	chembl:CHEMBL530280	CHEMBL:CHEMBL530280	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SQ-789	chembl:CHEMBL211042	CHEMBL:CHEMBL211042	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.9460841664089098	PHOTOSENSITIZER	ncit:C1420	PHOTOSENSITIZING AGENT	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1186614039224734	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2082	iuphar.ligand:2082	L-803,087	FALSE	FALSE	FALSE
UNIPROT:P42338	hgnc:8976	PIK3CB	TdgClinicalTrial	Jan-14	NULL	0.046303061	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:8160	iuphar.ligand:8160	COMPOUND 9B [PMID: 18986805]	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:7707	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	AZD2936	ncit:C188211	RILVEGOSTOMIG	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:9630	ncit:C25951	MALEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2418	hgnc:3929	FRA8A	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8624	iuphar.ligand:8624	INHIBITOR 1 [COLOMBO ET AL., 2012]	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	CancerCommons	25-Jul-13	antibody	0.8255923150266431	AMG 479	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.013442824	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	1.071585127259071	SIRUKUMAB	ncit:C152371	SIRUKUMAB	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.026789628	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.01893533	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2024	iuphar.ligand:2024	[125I]TYR10-CST14	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.095122593	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:6561	iuphar.ligand:6561	PSB-0788	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:4081	iuphar.ligand:4081	[3H]CNQX	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1776	rxcui:1656052	CANGRELOR	TRUE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:9207	iuphar.ligand:9207	2'3'-CGAMP	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9131	iuphar.ligand:9131	PLIXORAFENIB	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	KAINIC ACID	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.078136416	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:275	iuphar.ligand:275	RO 63-0563	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:4096	iuphar.ligand:4096	CIS-3-ACPBPA	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.048663273	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	1.944728564284981	DIDEOXYADENOSINE	ncit:C429	DIDEOXYADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	1.117184494376478	IUPHAR.LIGAND:10116	iuphar.ligand:10116	S5A1	FALSE	FALSE	FALSE
UNIPROT:P05155	hgnc:1228	SERPING1	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	C1-INH	rxcui:1599832	C1 ESTERASE INHIBITOR	TRUE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:11977	iuphar.ligand:11977	COMPOUND 27 [WO2019226977A1]	FALSE	FALSE	FALSE
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1	hgnc:2357	CRHR1	TTD	2020.06.01	NULL	2.917092846427472	ONO-2333Ms	iuphar.ligand:10376	ONO-2333MS	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006210251	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10078	iuphar.ligand:10078	RORC2 INVERSE AGONIST 66 [PMID: 30130103]	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.072125922	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	SPIRAMIDE	ncit:C66559	SPIRAMIDE	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	PharmGKB	4/5/24	NULL	1.400204566285186	ulinastatin	ncit:C102851	ULINASTATIN	FALSE	FALSE	FALSE
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	0.6250913242344582	Amediplase	ncit:C169777	AMEDIPLASE	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1981	iuphar.ligand:1981	[125I]PTA-OH	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	0.6177373086552295	BUTAPROST	ncit:C74369	BUTAPROST	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.070860555	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.8078103267029924	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
NCBIGENE:1795	hgnc:2989	DOCK3	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:9713	iuphar.ligand:9713	H. POLYGYRUS TGF-&BETA; MIMIC	FALSE	FALSE	FALSE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.497231735	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	PharmGKB	4/5/24	NULL	0.030221982	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.1648075054478797	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004716823	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.016377939	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.040235763	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.066297565	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.071341945	IUPHAR.LIGAND:2326	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	1.193356164447602	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	1.675776741564718	Cycrimine	rxcui:22037	CYCRIMINE	TRUE	FALSE	FALSE
NCBIGENE:3182	hgnc:5034	HNRNPAB	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:11530	iuphar.ligand:11530	TEMELIMAB	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.364636606	IUPHAR.LIGAND:2340	iuphar.ligand:2340	NA+	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.4795221117415022	AZD1390	iuphar.ligand:11277	AZD1390	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	GNF-PF-1654	chembl:CHEMBL602776	CHEMBL:CHEMBL602776	FALSE	FALSE	FALSE
SIRT5	hgnc:14933	SIRT5	TALC	12-May-16	inhibitor	0.1988926940746004	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.078545507	Refametinib	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.010468037	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.008327942	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	0.2430910705356226	IUPHAR.LIGAND:2453	iuphar.ligand:2453	DIHYDROSPHINGOSINE	FALSE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.2187819634820604	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	ABT-702	iuphar.ligand:5131	ABT702	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	GNF-PF-1737	chembl:CHEMBL531710	CHEMBL:CHEMBL531710	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	0.4375639269641208	desvenlafaxine	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.042863405	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:9783	iuphar.ligand:9783	MK6-83	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.019318496	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.07458476	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	6.563458904461812	ONO-1301	iuphar.ligand:1964	ONO-1301	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	NIFUROXAZIDE	rxcui:31782	NIFUROXAZIDE	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.049349315	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:317	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.3241214273808302	FLT3 TYROSINE KINASE INHIBITOR TTT-3002	ncit:C123362	FLT3 TYROSINE KINASE INHIBITOR TTT-3002	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.025298806	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003053304	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	1.500219178	IUPHAR.LIGAND:2494	iuphar.ligand:2494	DIPHENYLBORONIC ANHYDRIDE	FALSE	FALSE	FALSE
DCK	hgnc:2704	DCK	NCI	14-Sep-17	NULL	1.141471113819445	FMDC	ncit:C1539	TEZACITABINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.008600765	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.2282942227638891	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.040021091	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11147	iuphar.ligand:11147	COMPOUND 60 [PMID: 30889352]	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.5585922471882393	IUPHAR.LIGAND:9401	iuphar.ligand:9401	NMS-P715	FALSE	FALSE	FALSE
NCBIGENE:3239	hgnc:5136	HOXD13	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12799	iuphar.ligand:12799	GPX4 INHIBITOR C18	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.1105424657593568	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:1577	iuphar.ligand:1577	LARGE NEUROTENSIN	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR-I	hgnc:5464	IGF1	TTD	2020.06.01	NULL	13.12691780892362	BI-836845	chembl:CHEMBL4297850	XENTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:8148	iuphar.ligand:8148	COMPOUND 31 [PMID: 24915291]	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
ADCY2	hgnc:233	ADCY2	PharmGKB	4/5/24	NULL	0.6250913242344582	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2187819634820604	N,N'-DIPHENYL-GUANIDINE	chembl:CHEMBL77675	CHEMBL:CHEMBL77675	FALSE	FALSE	FALSE
CATIONIC TRYPSINOGEN	hgnc:9475	PRSS1	TTD	2020.06.01	NULL	2.917092846427472	Ulinastatin	ncit:C102851	ULINASTATIN	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.2206204673768676	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-4612	chembl:CHEMBL601550	CHEMBL:CHEMBL601550	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.070574827	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
SIRT3	hgnc:14931	SIRT3	DTC	9/2/20	NULL	0.6908904109959803	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.002213645	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.6250913242344582	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.063645662	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
NCBIGENE:2246	hgnc:3665	FGF1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8193	iuphar.ligand:8193	COMPOUND 30 [PMID: 17280833]	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	DTC	9/2/20	NULL	1.141471113819445	PNU-120596	iuphar.ligand:3991	PNU-120596	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.060772768	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
TIRAP	hgnc:17192	TIRAP	PharmGKB	4/5/24	NULL	5.250767124	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.251232877	DURVALUMAB	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
MAP3K11	hgnc:6850	MAP3K11	DTC	9/2/20	NULL	17.50255707856483	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.049817525	IUPHAR.LIGAND:5688	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.038382801	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	DTC	9/2/20	NULL	0.3409589041278864	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
NCBIGENE:1133	hgnc:1954	CHRM5	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:4821	rxcui:14851	VIGABATRIN	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.05593857	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.6908904109959803	DSP-2230	chembl:CHEMBL5095026	DSP-2230	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3127	iuphar.ligand:3127	COMPOUND 13 [PMID: 19456099]	FALSE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:11791	iuphar.ligand:11791	BIIB091	FALSE	FALSE	FALSE
COL1A1	hgnc:2197	COL1A1	PharmGKB	4/5/24	NULL	1.363835616511545	pamidronate	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	PharmGKB	4/5/24	NULL	0.2143170254518142	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
UNIPROT:Q8N9I0	hgnc:11510	SYT2	TEND	1-Aug-11	NULL	35.00511415712966	BOTULINUM TOXIN TYPE B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.087222045	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	CIViC	10-Apr-24	NULL	0.6908904109959803	PREXASERTIB	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1013	hgnc:1754	CDH15	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4768	iuphar.ligand:4768	AMINOBENZOVESAMICOL	FALSE	FALSE	FALSE
MTNR1B	hgnc:7464	MTNR1B	ChEMBL	33	agonist	7.876150685354174	TASIMELTEON	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	3.750547945	BRIAKINUMAB	ncit:C95321	BRIAKINUMAB	FALSE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.3182283105193606	ISOSORBIDE DINITRATE	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.021003068	trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.3684748858645228	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:455	iuphar.ligand:455	[3H]ZM 241385	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7033	iuphar.ligand:7033	MOLIBRESIB	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.075010959	IUPHAR.LIGAND:985	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.4605936073306534	Sotorasib	rxcui:2550714	SOTORASIB	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.133607306	HYDROCORTISONE SODIUM SUCCINATE	rxcui:235483	HYDROCORTISONE SODIUM SUCCINATE	TRUE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	NCI	14-Sep-17	NULL	0.2430910705356226	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1000146118775133	GAMBOGIC AMIDE	chembl:CHEMBL444109	GAMBOGIC AMIDE	FALSE	FALSE	FALSE
UNIPROT:P51788	hgnc:2020	CLCN2	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	LUBIPROSTONE	rxcui:623033	LUBIPROSTONE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.023867123	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.008621949	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.5427149481725528	ALPRENOLOL	rxcui:597	ALPRENOLOL	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	PharmGKB	4/5/24	NULL	5.469549087051511	enasidenib	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4088	iuphar.ligand:4088	[3H]MDL105519	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.1682938180631234	IUPHAR.LIGAND:2510	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NCBIGENE:2102	hgnc:16870	MELK	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:9366	iuphar.ligand:9366	MELK-TI	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:5457	iuphar.ligand:5457	EPPTB	FALSE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.8975670296699914	Piboserod	ncit:C74393	PIBOSEROD	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:10886	iuphar.ligand:10886	SR101099	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.090530468	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	0.201178817	Pyridoxal Phosphate	rxcui:1599827	PYRIDOXAL PHOSPHATE ANHYDROUS	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.6775183385250904	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
ABCA3	hgnc:33	ABCA3	PharmGKB	4/5/24	NULL	0.014435099	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	1.312691780892362	TOLBUTAMIDE SODIUM, STERILE	chembl:CHEMBL1200874	TOLBUTAMIDE SODIUM, STERILE	TRUE	FALSE	FALSE
PRKCI	hgnc:9404	PRKCI	ChEMBL	33	inhibitor	0.3088686543276147	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	5.431828058864948	IUPHAR.LIGAND:2167	iuphar.ligand:2167	URANTIDE	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.4167275494896388	TABERMINOGENE VADENOVEC	drugbank:DB05011	TABERMINOGENE VADENOVEC	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:752	iuphar.ligand:752	BP-CCL3	FALSE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:4764	iuphar.ligand:4764	[125I]IODOVINYL-TBZ	FALSE	FALSE	FALSE
NCBIGENE:2373	hgnc:6364	KLK3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8486	iuphar.ligand:8486	COMPOUND 20 [PMID: 23692593]	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.1229687850953032	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
HCAR2	hgnc:24827	HCAR2	DTC	9/2/20	NULL	2.500365296937833	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.023080295	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.2243917574174978	CYCLOBENZAPRINE HYDROCHLORIDE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.067317527	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2277	iuphar.ligand:2277	[125I]VIP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:1625	ncbigene:1625	DBIL3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:5298	iuphar.ligand:5298	Z-LEHD-FMK	FALSE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.1842374429322614	methylene blue	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.00502947	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.5556367326528519	ICOTINIB	ncit:C138996	ICOTINIB	FALSE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	1.419126249613364	ESTRADIOL DIPROPIONATE	ncit:C29770	ESTRADIOL DIPROPIONATE	FALSE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	NCI	14-Sep-17	NULL	0.1172046232939609	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:2226	rxcui:358257	TOLVAPTAN	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.04724037	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
FGF4	hgnc:3682	FGF4	CGI	2/1/22	NULL	0.1039755866053356	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12985	iuphar.ligand:12985	CH7233163	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2204	iuphar.ligand:2204	YM 218	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.082429625	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1500219178162699	ACRIDIN-1-YLAMINE	chembl:CHEMBL146525	CHEMBL:CHEMBL146525	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.074797252	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	(S)-MAP4 HCL	chembl:CHEMBL1256510	CHEMBL:CHEMBL1256510	FALSE	FALSE	FALSE
AMP-ACTIVATED PROTEIN KINASE	hgnc:9377	PRKAA2	TTD	2020.06.01	NULL	4.773424657790408	Imeglimin	ncit:C132841	IMEGLIMIN	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1930429089547591	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	ALPRENOLOL	rxcui:597	ALPRENOLOL	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:9772	ncit:C174799	LENABASUM	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5533	ncit:C152801	UNDECANOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:7372	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.03591496	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2211	iuphar.ligand:2211	[PHAA1,D-TYR2,VAL4,ARG6,ARG-NH29]AVP	FALSE	FALSE	FALSE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.097236428	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
UNIPROT:P20648	hgnc:819	ATP4A	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	PANTOPRAZOLE	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	DTC	9/2/20	NULL	4.039051633514961	CYPATE	chembl:CHEMBL2071606	CYPATE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.035098711	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.4412409347537352	RIVASTIGMINE	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.050912416	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.019418517	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
NCBIGENE:1921	hgnc:19679	AAK1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11893	iuphar.ligand:11893	COMPOUND 6 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:542	iuphar.ligand:542	H87/07	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:1228	rxcui:10849	TRIPROLIDINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:288	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	0.091796628	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	SJ000281118	chembl:CHEMBL592561	CHEMBL:CHEMBL592561	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.3231241306811969	PROPERICIAZINE	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	MICONAZOLE NITRATE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.02339914	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
SODIUM-DEPENDENT MULTIVITAMIN TRANSPORTER	hgnc:11041	SLC5A6	TTD	2020.06.01	NULL	1.944728564284981	Gabapentin enacarbil	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CancerCommons	25-Jul-13	inhibitor	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.5427149481725528	Ritodrine	rxcui:9392	RITODRINE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.2386712328895204	Aminosalicylic Acid	rxcui:7833	AMINOSALICYLIC ACID	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DINITROPHENYLENE	chembl:CHEMBL114070	DINITROPHENYLENE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
ZFP36L2	hgnc:1108	ZFP36L2	NCI	14-Sep-17	NULL	0.258658479	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2205	iuphar.ligand:2205	YM 471	FALSE	FALSE	FALSE
NCBIGENE:2068	hgnc:3434	ERCC2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:12104	iuphar.ligand:12104	COMPOUND 1K [PMID: 35912476]	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.406619897	Etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.3580068493342807	MELOXICAM	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.546954909	SILODOSIN	rxcui:720825	SILODOSIN	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.021554873	IUPHAR.LIGAND:87	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.011940798	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:667	rxcui:1148138	ICATIBANT	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	EXALAMIDE	ncit:C65607	EXALAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2831	hgnc:4522	NPBWR1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12000	iuphar.ligand:12000	MS40	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	0.8751278539282416	Deutetrabenazine	rxcui:1876905	DEUTETRABENAZINE	TRUE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	1.166837138570988	FEXOFENADINE HYDROCHLORIDE	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	PD-173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.077789143	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	0.8078103267029924	IUPHAR.LIGAND:1504	iuphar.ligand:1504	NEUROPEPTIDE Y	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	GR-4661	chembl:CHEMBL344127	CHEMBL:CHEMBL344127	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.019142425	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	DTC	9/2/20	NULL	3.150460274	KU-0058948	drugbank:DB08058	4-[3-(1,4-DIAZEPAN-1-YLCARBONYL)-4-FLUOROBENZYL]PHTHALAZIN-1(2H)-ONE	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	3.750547945	CELL SURFACE ANTIGENS	ncit:C269	CELL SURFACE ANTIGEN	FALSE	FALSE	FALSE
REEP5	hgnc:30077	REEP5	PharmGKB	4/5/24	NULL	1.050153425	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:3802	iuphar.ligand:3802	[125I]PYY-(3-36) (HUMAN)	FALSE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	FLUVASTATIN	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.067317527	IUPHAR.LIGAND:985	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.036847489	IUPHAR.LIGAND:34	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:3867	iuphar.ligand:3867	D(CH2)5[TYR(ME)2,ARG8]VP	FALSE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.3621218705909965	RETASPIMYCIN	ncit:C80378	RETASPIMYCIN	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	N-ACETYLCOLCHINOL	chembl:CHEMBL486504	N-ACETYLCOLCHINOL	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1750255707856483	DIBENZ[A,H]ANTHRACENE	chembl:CHEMBL1346946	DIBENZ[A,H]ANTHRACENE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002165622	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.035430277	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	5.250767123569449	Aliskiren	rxcui:325646	ALISKIREN	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.9845188356692718	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	CIViC	10-Apr-24	NULL	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:10658	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:7056	iuphar.ligand:7056	COMPOUND 7D [PMID: 19111466]	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.037721028	IUPHAR.LIGAND:2603	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.025588534	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
CCNE1	hgnc:1589	CCNE1	CIViC	10-Apr-24	NULL	0.1071585127259071	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
TLR4	hgnc:11850	TLR4	NCI	14-Sep-17	NULL	0.057796006	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.2983390411119005	CLOBETASOL	rxcui:2590	CLOBETASOL	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.039598545	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	1.235474617310458	KN035	ncit:C129714	ENVAFOLIMAB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005107253	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
TYROSINE 3-MONOOXYGENASE	hgnc:11782	TH	TTD	2020.06.01	NULL	0.8334550989792776	ProSavin	wikidata:Q7246687	PROSAVIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	CIViC	10-Apr-24	NULL	0.2243917574174978	COBIMETINIB	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.2590839041234926	TUCATINIB	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.068757317	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.4102161815288632	ranitidine	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00809055	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
CRKL	hgnc:2363	CRKL	CIViC	10-Apr-24	NULL	0.045461187	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	4.200613699	KRH-3955	chembl:CHEMBL2062277	CHEMBL:CHEMBL2062277	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005903055	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
GALACTOSYLTRANSFERASE	hgnc:4135	GALT	TTD	2020.06.01	NULL	52.50767123569449	Algenpantucel-L	ncit:C61082	ALGENPANTUCEL-L	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.075768645	BRIGATINIB	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	11.66837138570988	IUPHAR.LIGAND:8387	iuphar.ligand:8387	EPZ005687	FALSE	FALSE	TRUE
NCBIGENE:2094	ncbigene:2094	ERVT4	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8763	iuphar.ligand:8763	COMPOUND 8 [PMID: 17480064]	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.3977853881492008	BRIGATINIB	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
IKZF1	hgnc:13176	IKZF1	CIViC	10-Apr-24	NULL	0.3088686543276147	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.3977853881492006	NEBIVOLOL	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.6886251965336985	AVAPRITINIB	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	CIViC	10-Apr-24	NULL	0.018106094	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	CIViC	10-Apr-24	NULL	0.074690855	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
ALPHA-1-ANTITRYPSIN	hgnc:8941	SERPINA1	TTD	2020.06.01	NULL	8.751278539282415	Glassia	rxcui:535	ALPHA 1-ANTITRYPSIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	3-((2-PHENETHYLPHENOXY)METHYL)PYRIDINE	chembl:CHEMBL217425	CHEMBL:CHEMBL217425	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.077789143	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.016116535	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	CID 3238892	chembl:CHEMBL261118	CHEMBL:CHEMBL261118	FALSE	FALSE	FALSE
FZD1	hgnc:4038	FZD1	DTC	9/2/20	NULL	26.25383561784724	GNF-PF-3411	chembl:CHEMBL593726	CHEMBL:CHEMBL593726	FALSE	FALSE	FALSE
NCOR2	hgnc:7673	NCOR2	DTC	9/2/20	NULL	1.591141552596803	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	SJ000124275	chembl:CHEMBL602150	CHEMBL:CHEMBL602150	FALSE	FALSE	FALSE
SLFN11	hgnc:26633	SLFN11	CIViC	10-Apr-24	NULL	1.250182648468916	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	CHLOROACETOXYQUINOLINE	chembl:CHEMBL1450499	CHLOROACETOXYQUINOLINE	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.1682938180631233	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.03729238	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.029833904	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:10287	iuphar.ligand:10287	TONANTZITLOLONE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	6-CHLORONICOTINIC ACID	chembl:CHEMBL1723657	6-CHLORONICOTINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.018867291	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:8069	iuphar.ligand:8069	CP-673451	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.062509132	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1325951293830669	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	1.166837138570988	GNF-PF-4371	chembl:CHEMBL585651	CHEMBL:CHEMBL585651	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1635752997996713	SIBUTRAMINE	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
UNIPROT:P48443	hgnc:10479	RXRG	TdgClinicalTrial	Jan-14	NULL	0.1049104320393496	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6101	iuphar.ligand:6101	M1145	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	0.192335792	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.035574303	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.071780822	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	CID 1225609	chembl:CHEMBL444376	CHEMBL:CHEMBL444376	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	FLUORODIFEN	chembl:CHEMBL1892429	FLUORODIFEN	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.065226921	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
UNIPROT:Q02750	hgnc:6840	MAP2K1	TdgClinicalTrial	Jan-14	NULL	0.5125748858722557	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
UNIPROT:O00757	hgnc:3607	FBP2	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	MB07803	chembl:CHEMBL4297400	MB-07803	FALSE	FALSE	FALSE
ZEB1	hgnc:11642	ZEB1	CIViC	10-Apr-24	NULL	0.1166837138570988	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	5.469549087051511	Enasidenib	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
GSTA1	hgnc:4626	GSTA1	PharmGKB	4/5/24	NULL	0.3500511415712967	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.029515273	nebivolol	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.1411496538593938	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	DTC	9/2/20	NULL	0.072175493	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001225383	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.021301287	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	3',5-DIHYDROXYFLAVONE	chembl:CHEMBL502242	CHEMBL:CHEMBL502242	FALSE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	0.729273212	APINOCALTAMIDE	ncit:C190345	APINOCALTAMIDE	FALSE	FALSE	FALSE
UNIPROT:Q7L0J3	hgnc:20566	SV2A	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	BRIVARACETAM	rxcui:1739745	BRIVARACETAM	TRUE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	CIViC	10-Apr-24	NULL	0.3977853881492007	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:5927	iuphar.ligand:5927	AMINOPURVALANOL A	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	Revumenib	ncit:C165776	REVUMENIB	FALSE	FALSE	FALSE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.1193356164447602	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
GNAS	hgnc:4392	GNAS	CIViC	10-Apr-24	NULL	0.012606884	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
UNIPROT:Q9Y5N1	hgnc:5184	HRH3	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	BETAHISTINE	rxcui:1511	BETAHISTINE	TRUE	FALSE	FALSE
UNIPROT:P47901	hgnc:896	AVPR1B	TEND	1-Aug-11	NULL	1.666910197958555	DESMOPRESSIN	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.033458584	DOXEPIN HYDROCHLORIDE	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.039688338	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CTLA4	hgnc:2505	CTLA4	ChEMBL	33	inhibitor	1.750255707856483	ZALIFRELIMAB	ncit:C126113	ZALIFRELIMAB	FALSE	FALSE	FALSE
UNIPROT:Q16739	hgnc:12524	UGCG	TdgClinicalTrial	Jan-14	NULL	7.001022831425932	MIGLUSTAT	rxcui:402316	MIGLUSTAT	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:6502	iuphar.ligand:6502	FASIDOTRILAT	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.4440395030502706	IUPHAR.LIGAND:12488	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.091159151	B-RAF/VEGFR-2 INHIBITOR RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:770	iuphar.ligand:770	CCL13	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:3499	iuphar.ligand:3499	DMP696	FALSE	FALSE	FALSE
NCBIGENE:3230	hgnc:5131	HOXD@	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12656	iuphar.ligand:12656	RP-6685	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-125254	chembl:CHEMBL547313	CHEMBL:CHEMBL547313	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.006375385	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.033658764	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	RAC-NUTLIN-3	chembl:CHEMBL211045	CHEMBL:CHEMBL211045	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	TCMDC-125575	chembl:CHEMBL587620	CHEMBL:CHEMBL587620	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.095122593	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.1341192113299987	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
LUM	hgnc:6724	LUM	NCI	14-Sep-17	NULL	8.751278539282415	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.6908904109959803	ISOPROPAMIDE IODIDE	rxcui:6051	ISOPROPAMIDE IODIDE	TRUE	FALSE	FALSE
STK11	hgnc:11389	STK11	CGI	2/1/22	NULL	0.4138535663897103	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	HYDROCORTISONE ACETATE	rxcui:27197	HYDROCORTISONE ACETATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.058471794	TESTOSTERONE CYPIONATE	rxcui:835827	TESTOSTERONE CYPIONATE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.083257407	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.047734247	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
KCNA3	hgnc:6221	KCNA3	ChEMBL	33	blocker	0.150021918	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.014425184	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.026253836	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	CI-218872	chembl:CHEMBL13662	CI-218872	FALSE	FALSE	FALSE
CRBN	hgnc:30185	CRBN	CIViC	10-Apr-24	NULL	2.917092846427472	POMALIDOMIDE	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	3.088686543276147	NSC-640584	chembl:CHEMBL476968	CHEMBL:CHEMBL476968	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:10938	iuphar.ligand:10938	SAR247799	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.062509132	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	PHENAMIL METHANESULFONATE	chembl:CHEMBL1256775	PHENAMIL METHANESULFONATE	FALSE	FALSE	FALSE
DYSTROPHIN NONSENSE MUTANT	hgnc:2928	DMD	TTD	2020.06.01	NULL	0.091476779	Ataluren	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	FDA	10-Apr-24	NULL	0.1919140030544389	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
SLC25A5	hgnc:10991	SLC25A5	NCI	14-Sep-17	NULL	0.1750255707856483	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	MECHLORETHAMINE HYDROCHLORIDE	rxcui:155036	MECHLORETHAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CREB1	hgnc:2345	CREB1	NCI	14-Sep-17	NULL	0.1208461938681116	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:3023	ncbigene:3023	H4F3	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:12601	ncit:C1146	LONIDAMINE	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	0.08607815	IUPHAR.LIGAND:7946	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5627	iuphar.ligand:5627	NODAGA-[TYR3]-OCTREOTIDE	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.3977853881492006	IUPHAR.LIGAND:2418	iuphar.ligand:2418	ACROLEIN	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:2172	iuphar.ligand:2172	LVP	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.7955707762984013	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.011762471	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.071341945	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN TREGOPIL	ncit:C166701	INSULIN TREGOPIL	FALSE	FALSE	FALSE
NCBIGENE:1638	hgnc:2709	DCT	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8846	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	SULFADIAZINE, SILVER	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.3088686543276147	ZNCL2	rxcui:39937	ZINC CHLORIDE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	(Z)-PIPLARTINE	chembl:CHEMBL1456697	(Z)-PIPLARTINE	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.2414145803939977	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
DSE	hgnc:21144	DSE	PharmGKB	4/5/24	NULL	4.375639269641208	abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	4.039051633514961	Ixekizumab	rxcui:1745099	IXEKIZUMAB	TRUE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.08914715	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.02726255	METHOXSALEN	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	CancerCommons	25-Jul-13	inhibitor	0.1810609352954982	XL888	ncit:C79835	HSP90 INHIBITOR XL888	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	CancerCommons	25-Jul-13	inhibitor	0.6250913242344582	RECENTIN	hemonc:94	CEDIRANIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.042793538	VENETOCLAX	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	CIViC	10-Apr-24	NULL	0.4296082192011368	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PDCD1	hgnc:8760	PDCD1	CancerCommons	25-Jul-13	antibody	2.561349816375341	CT-011	drugbank:DB05916	CT-011	FALSE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.546954909	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
RAD54L	hgnc:9826	RAD54L	CIViC	10-Apr-24	NULL	0.023867123	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
BCOR	hgnc:20893	BCOR	CGI	2/1/22	NULL	2.187819634820604	Enzastaurin	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	CGI	2/1/22	NULL	0.068191781	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.072165573	Exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
FGF3	hgnc:3681	FGF3	CGI	2/1/22	NULL	0.8751278539282417	Lucitanib	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.020029629	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
FGF3	hgnc:3681	FGF3	CGI	2/1/22	NULL	0.1299694832566695	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
FGF4	hgnc:3682	FGF4	CGI	2/1/22	NULL	0.7001022831425934	Lucitanib	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
EZH2	hgnc:3527	EZH2	CGI	2/1/22	NULL	11.66837138570988	EPZ-005687	iuphar.ligand:8387	EPZ005687	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CGI	2/1/22	NULL	0.006669123	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CGI	2/1/22	NULL	1.346350544504987	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CGI	2/1/22	NULL	1.029066006546944	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CGI	2/1/22	NULL	0.1088116604009326	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	CGI	2/1/22	NULL	0.3017682254924971	MEK inhibitor	ncit:C69145	MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.010573434	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	CGI	2/1/22	NULL	0.037505479	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	CIViC	10-Apr-24	NULL	0.03140411	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.1215455352678113	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
MTOR	hgnc:3942	MTOR	CGI	2/1/22	NULL	0.2007335520076852	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
PLG	hgnc:9071	PLG	ChEMBL	33	inhibitor	1.250182648468916	TRANEXAMIC ACID	rxcui:10691	TRANEXAMIC ACID	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	inhibitor	1.666910197958555	AMINOCAPROIC ACID	rxcui:99	6-AMINOCAPROIC ACID	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1861974157294131	OXYPHENCYCLIMINE HYDROCHLORIDE	rxcui:91164	OXYPHENCYCLIMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	CIViC	10-Apr-24	NULL	0.009529523	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.3977853881492006	NEBIVOLOL HYDROCHLORIDE	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	0.5834185692854945	INDAPAMIDE	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
PLAT	hgnc:9051	PLAT	ChEMBL	33	inhibitor	3.182283105193605	AMINOCAPROIC ACID	rxcui:99	6-AMINOCAPROIC ACID	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.1976759387696734	PIOGLITAZONE HYDROCHLORIDE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	0.2681242786503549	PEMETREXED DISODIUM	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	3.281729452230906	RANITIDINE BISMUTH CITRATE	rxcui:55471	RANITIDINE BISMUTH CITRATE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	ChEMBL	33	inhibitor	0.2941606231691568	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.013645445	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP EXTENDED BEEF	chembl:CHEMBL1201640	INSULIN ZINC SUSP EXTENDED BEEF	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP PROMPT BEEF	chembl:CHEMBL1201642	INSULIN ZINC SUSP PROMPT BEEF	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.04362008	AMITRIPTYLINE HYDROCHLORIDE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PGA5	hgnc:8887	PGA5	ChEMBL	33	inhibitor	17.50255707856483	SUCRALFATE	rxcui:10156	SUCRALFATE	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.050764748	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.4303907478335614	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.49187514	LEVONORGESTREL	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.053798843	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.1166837138570989	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
CA6	hgnc:1380	CA6	ChEMBL	33	inhibitor	0.5000730593875666	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	CODEINE PHOSPHATE	rxcui:2672	CODEINE PHOSPHATE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.064824285	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.028413242	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	CIViC	10-Apr-24	NULL	0.1396480617970598	FGFR INHIBITOR AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
ACTL6A	hgnc:24124	ACTL6A	CIViC	10-Apr-24	NULL	0.090530468	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.012154554	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.058212496	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
GNAQ	hgnc:4390	GNAQ	CIViC	10-Apr-24	NULL	1.312691780892362	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.032899543	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.03070624	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.028199609	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.089501712	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	CIViC	10-Apr-24	NULL	0.03292017	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.108711535	TETRAHYDROZOLINE HYDROCHLORIDE	rxcui:57983	TETRAHYDROZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.3750547945406749	TOLAZAMIDE	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.09699693	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.069824031	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.1315981735230438	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.012993732	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.4546118721705151	Tazemetostat	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.9590442234830044	Ceralasertib	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.025238006	Valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
LAMA5	hgnc:6485	LAMA5	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.030221982	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.4795221117415022	PJ34	iuphar.ligand:11348	PJ34	FALSE	FALSE	FALSE
LAMA4	hgnc:6484	LAMA4	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.030545475	Lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
LAMB3	hgnc:6490	LAMB3	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
COL4A3	hgnc:2204	COL4A3	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.063440602	Temsirolimus	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
COL6A6	hgnc:27023	COL6A6	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.074128477	Pemetrexed Disodium	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
COL6A1	hgnc:2211	COL6A1	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.3182283105193605	ROFECOXIB	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
ITK	hgnc:6171	ITK	ChEMBL	33	inhibitor	0.053253216	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.2059124362184097	Trabectedin	rxcui:1716278	TRABECTEDIN	TRUE	FALSE	TRUE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	1.944728564284981	YTTRIUM Y 90 IBRITUMOMAB TIUXETAN	chembl:CHEMBL2108667	YTTRIUM Y 90 IBRITUMOMAB TIUXETAN	TRUE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	0.3977853881492007	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	agonist	0.2273059360852575	SUCCINYLCHOLINE CHLORIDE	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	agonist	0.2386712328895204	SUCCINYLCHOLINE CHLORIDE	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.096167896	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	2.019525817	GSK461364	ncit:C70948	POLO-LIKE KINASE 1 INHIBITOR GSK461364	FALSE	FALSE	TRUE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.07631929	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.056826484	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.097236428	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.085239726	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.03591496	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.1835932560688619	Sapanisertib	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.085796848	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.03043923	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.326134604	TAE226	iuphar.ligand:9382	NVP-TAE 226	FALSE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	modulator	0.2160809515872201	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	modulator	0.1215455352678113	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	modulator	0.2160809515872201	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.9211872146613068	Ceralasertib	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	modulator	0.1495945049449985	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	modulator	0.2160809515872201	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1635752997996713	ICP-192	ncit:C178318	GUNAGRATINIB	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.030147945	Cediranib	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.054695491	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.036847489	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.050007306	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.043502627	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1124502911321247	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.088248187	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.016695603	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.072919531	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.010923169	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.1377250393067396	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1000146118775133	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	2.917092846427472	SUVOREXANT	rxcui:1547099	SUVOREXANT	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.1547594520630995	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.08937476	NINTEDANIB ESYLATE	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2386712328895204	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
PSMA2	hgnc:9531	PSMA2	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	ARQ 531	ncit:C138066	NEMTABRUTINIB	FALSE	FALSE	FALSE
PSMB8	hgnc:9545	PSMB8	ChEMBL	33	inhibitor	0.1223955040459079	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.054581779	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.054581779	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.108040476	Rebastinib	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.061197752	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.055563673	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.108040476	GMI-1359	drugbank:DB18092	GMI-1359	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1795134059339982	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
PRKACA	hgnc:9380	PRKACA	ChEMBL	33	inhibitor	0.1544343271638073	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.076765601	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PRKCA	hgnc:9393	PRKCA	ChEMBL	33	inhibitor	0.1286952726365061	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.3889457128569963	LY-2780301	chembl:CHEMBL3545134	LY-2780301	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.2302968036653267	RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.037884323	PAXALISIB	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1666910197958555	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.4167275494896388	SAR-260301	chembl:CHEMBL3545008	SAR-260301	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.596678082	RO-4987655	drugbank:DB12933	RO-4987655	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1666910197958555	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
FZD8	hgnc:4046	FZD8	ChEMBL	33	inhibitor	3.750547945406749	VANTICTUMAB	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.1256164383629055	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.026259671	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.03140411	Sapanisertib	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.054695491	Azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.025942525	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2853677784548614	C220	rxcui:203203	ALFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	TAK-632	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	FCN-159	ncit:C172382	MEK 1/2 INHIBITOR FCN-159	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	ChEMBL	33	agonist	3.750547945	LY2881835	chembl:CHEMBL3545086	LY2881835	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1693795846312726	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2035181055647073	LAS190792	chembl:CHEMBL3545272	LAS190792	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.007867496	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.048394167	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
CSNK2A1	hgnc:2457	CSNK2A1	ChEMBL	33	inhibitor	1.875273972703375	SILMITASERTIB	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1764963739014941	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1209854175937661	E6201	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
PRKD1	hgnc:9407	PRKD1	ChEMBL	33	inhibitor	0.2625383561784725	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	Ipatasertib	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.039068208	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.1605739181519709	ODELEPRAN	chembl:CHEMBL2103878	ODELEPRAN	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.1315981735230438	AFACIFENACIN	ncit:C90741	AFACIFENACIN	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.5834185692854945	DERENOFYLLINE	ncit:C96199	DERENOFYLLINE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.086818239	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	1.369765336583334	SPARSENTAN	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.054020238	M2698	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	1.009762908	PRATOSARTAN	ncit:C72935	PRATOSARTAN	FALSE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	1.500219178	RAFABEGRON	ncit:C96753	RAFABEGRON	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	inhibitor	1.029562181092048	TRELANSERIN	ncit:C90946	TRELANSERIN	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.1166837138570989	AZD7325	iuphar.ligand:7712	AZD7325	FALSE	FALSE	FALSE
RAMP1	hgnc:9843	RAMP1	ChEMBL	33	agonist	3.281729452230906	DAVALINTIDE	ncit:C83650	DAVALINTIDE	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.6731752722524935	EVT-101	drugbank:DB05956	EVT-101	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.2586584789935689	GW468816	chembl:CHEMBL1207366	GW468816	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.5357925636295356	EVT-101	drugbank:DB05956	EVT-101	FALSE	FALSE	FALSE
P2RX7	hgnc:8537	P2RX7	ChEMBL	33	inhibitor	17.50255707856483	CE-224535	drugbank:DB12113	CE-224535	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.458546423213736	POZANICLINE	ncit:C81045	POZANICLINE	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	ChEMBL	33	inhibitor	3.281729452230906	BEMCENTINIB	ncit:C121854	BEMCENTINIB	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.3365876361262467	RADIPRODIL	ncit:C152143	RADIPRODIL	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.084146909	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.011933562	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNS1	hgnc:6300	KCNS1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNH4	hgnc:6253	KCNH4	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCND1	hgnc:6237	KCND1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNB1	hgnc:6231	KCNB1	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.2393966773663883	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.1544343271638073	SARIZOTAN HYDROCHLORIDE	ncit:C76654	SARIZOTAN HYDROCHLORIDE	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inverse agonist	0.7573221812840553	PIMAVANSERIN TARTRATE	rxcui:1791685	PIMAVANSERIN	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.029833904	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.043756393	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.090530468	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.034544521	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	LOXO-783	ncit:C187335	MUTANT-SELECTIVE PI3K-ALPHA H1047R INHIBITOR LOXO-783	FALSE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	activator	0.6563458904461812	FLINDOKALNER	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	other/unknown	2.917092846427472	BECTUMOMAB	drugbank:DB04962	BECTUMOMAB	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	3.962843112127886	FIGITUMUMAB	ncit:C52187	FIGITUMUMAB	FALSE	TRUE	TRUE
BCL2	hgnc:990	BCL2	ChEMBL	33	inhibitor	0.1219690388750162	VENETOCLAX	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.011049594	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.9723642821424906	ALBINTERFERON ALFA-2B	ncit:C87296	ALBINTERFERON ALFA-2B	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.729273212	TQ-B3139	ncit:C148513	ALK/C-MET INHIBITOR TQ-B3139	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	negative modulator	0.042174836	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
MYL7	hgnc:21719	MYL7	ChEMBL	33	activator	2.187819634820604	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.087512785	Pemetrexed Disodium	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
RHD	hgnc:10009	RHD	ChEMBL	33	inhibitor	26.25383561784724	ROLEDUMAB	ncit:C152241	ROLEDUMAB	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.4138535663897103	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
TPBG	hgnc:12004	TPBG	ChEMBL	33	other/unknown	10.50153424713889	ANATUMOMAB MAFENATOX	ncit:C190321	ANATUMOMAB MAFENATOX	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	modulator	0.3889457128569963	AMISELIMOD HYDROCHLORIDE	ncit:C142922	AMISELIMOD HYDROCHLORIDE	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	PIRPROFEN	ncit:C170327	PIRPROFEN	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	PIRPROFEN	ncit:C170327	PIRPROFEN	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.063110182	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.070574827	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	inhibitor	0.090843722	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	blocker	0.1262203635473425	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CCR4	hgnc:1605	CCR4	ChEMBL	33	modulator	12.35474617310458	MOGAMULIZUMAB	rxcui:2054068	MOGAMULIZUMAB	TRUE	TRUE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.029698909	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.9546849315580818	AMG-820	chembl:CHEMBL2109322	AMG-820	FALSE	FALSE	FALSE
MCAM	hgnc:6934	MCAM	ChEMBL	33	inhibitor	52.50767123569449	ABX-MA1	chembl:CHEMBL2109519	ABX-MA1	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.056097939	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1591141552596802	ACECLOFENAC	rxcui:16689	ACECLOFENAC	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.069180068	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	2.917092846427472	PITAVASTATIN SODIUM	rxcui:1944734	PITAVASTATIN SODIUM	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	1.944728564284981	OCARATUZUMAB	ncit:C2524	OCARATUZUMAB	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	2.187819634820604	AS-1403	chembl:CHEMBL2109360	AS-1403	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	modulator	0.760980743	MEDI-565	chembl:CHEMBL2109372	MEDI-565	FALSE	FALSE	FALSE
CR1	hgnc:2334	CR1	ChEMBL	33	inhibitor	13.12691780892362	MIROCOCEPT	ncit:C170185	MIROCOCEPT	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.03378872	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2465148884304905	LOFEXIDINE HYDROCHLORIDE	rxcui:235853	LOFEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.03049226	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.032055965	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.068369364	AVIPTADIL	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.364636606	SELITRECTINIB	ncit:C138160	SELITRECTINIB	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2442217266776488	BENIDIPINE	ncit:C81680	BENIDIPINE	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2442217266776488	NILVADIPINE	rxcui:53692	NILVADIPINE	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1981421556063943	BENIDIPINE	ncit:C81680	BENIDIPINE	FALSE	FALSE	FALSE
MGAM	hgnc:7043	MGAM	ChEMBL	33	inhibitor	2.386712328895204	CELGOSIVIR	ncit:C79567	CELGOSIVIR	FALSE	FALSE	FALSE
TNKS2	hgnc:15677	TNKS2	ChEMBL	33	inhibitor	13.12691780892362	2X-121	drugbank:DB16063	2X-121	FALSE	FALSE	FALSE
SI	hgnc:10856	SI	ChEMBL	33	inhibitor	1.640864726115453	CELGOSIVIR	ncit:C79567	CELGOSIVIR	FALSE	FALSE	FALSE
IDO1	hgnc:6059	IDO1	ChEMBL	33	inhibitor	7.501095891	LINRODOSTAT	ncit:C141135	LINRODOSTAT	FALSE	FALSE	FALSE
TNFRSF17	hgnc:11913	TNFRSF17	ChEMBL	33	binder	2.763561643983921	IDECABTAGENE VICLEUCEL	rxcui:2536430	IDECABTAGENE VICLEUCEL	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	TETOMILAST	ncit:C90922	TETOMILAST	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2917092846427472	CILOMILAST	ncit:C95232	CILOMILAST	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	ChEMBL	33	inhibitor	0.5707355569097228	ELRAGLUSIB	ncit:C156792	ELRAGLUSIB	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2983390411119005	CILOMILAST	ncit:C95232	CILOMILAST	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.9053046764774912	NEMONOXACIN	ncit:C174838	NEMONOXACIN	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.082300425	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PTPN11	hgnc:9644	PTPN11	ChEMBL	33	inhibitor	5.000730593875666	BATOPROTAFIB	ncit:C139559	BATOPROTAFIB	FALSE	FALSE	FALSE
TSPO	hgnc:1158	TSPO	ChEMBL	33	inhibitor	2.763561643983921	ONO-2952	drugbank:DB14802	ONO-2952	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.095295229	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	AMG 900	ncit:C82349	AURORA KINASE INHIBITOR AMG 900	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.2430910705356226	TESOFENSINE	ncit:C66589	TESOFENSINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	BLZ945	chembl:CHEMBL4227505	BLZ945	FALSE	FALSE	FALSE
TIGIT	hgnc:26838	TIGIT	ChEMBL	33	inhibitor	6.563458904461812	VIBOSTOLIMAB	ncit:C140041	VIBOSTOLIMAB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	TEBUFENPYRAD	chembl:CHEMBL1897070	TEBUFENPYRAD	FALSE	FALSE	FALSE
MTTP	hgnc:7467	MTTP	ChEMBL	33	inhibitor	13.12691780892362	SLX-4090	drugbank:DB05678	SLX-4090	FALSE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.7001022831425934	ATACIGUAT	ncit:C79587	ATACIGUAT	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	VU001171	iuphar.ligand:6228	VU0001171	FALSE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	ZINLIRVIMAB	ncit:C188593	ZINLIRVIMAB	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.4861821410712453	SERDEXMETHYLPHENIDATE CHLORIDE	rxcui:2562177	SERDEXMETHYLPHENIDATE CHLORIDE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.037213091	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.024309107	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NPR1	hgnc:7943	NPR1	ChEMBL	33	agonist	1.346350544504987	CARPERITIDE	ncit:C169829	CARPERITIDE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.3017682254924971	SJ000120515	chembl:CHEMBL592314	CHEMBL:CHEMBL592314	FALSE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	1.009762908	RUNCACIGUAT	ncit:C166842	RUNCACIGUAT	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	agonist	0.1861974157294131	TALSACLIDINE	ncit:C96885	TALSACLIDINE	FALSE	FALSE	FALSE
IL1RL2	hgnc:5999	IL1RL2	ChEMBL	33	inhibitor	8.751278539282415	SPESOLIMAB	rxcui:2610417	SPESOLIMAB	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	binder	0.3454452054979901	TRASTUZUMAB DUOCARMAZINE	ncit:C118674	TRASTUZUMAB DUOCARMAZINE	FALSE	FALSE	FALSE
EREG	hgnc:3443	EREG	ChEMBL	33	inhibitor	4.375639269641208	FEPIXNEBART	ncit:C188574	FEPIXNEBART	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	ChEMBL	33	inhibitor	0.1682938180631233	BIRICODAR	ncit:C71621	BIRICODAR	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.3621218705909966	GLICLAZIDE	rxcui:4816	GLICLAZIDE	TRUE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	agonist	2.187819634820604	GILORALIMAB	ncit:C139553	GILORALIMAB	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.038608582	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
HTR6	hgnc:5301	HTR6	ChEMBL	33	inhibitor	3.500511415712966	MASUPIRDINE	ncit:C175121	MASUPIRDINE	FALSE	FALSE	FALSE
F11	hgnc:3529	F11	ChEMBL	33	inhibitor	0.6908904109959803	MILVEXIAN	ncit:C175138	MILVEXIAN	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.092443083	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
TRHR	hgnc:12299	TRHR	ChEMBL	33	agonist	8.751278539282415	ROVATIRELIN	ncit:C152262	ROVATIRELIN	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	EMB-01	drugbank:DB16091	EMB-01	FALSE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	2.625383561784724	CIBINETIDE	ncit:C171683	CIBINETIDE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	DNDI1416988	chembl:CHEMBL1389794	CHEMBL:CHEMBL1389794	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	positive modulator	1.193356164447602	NAVOCAFTOR	ncit:C174930	NAVOCAFTOR	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	FDA	10-Apr-24	NULL	2.512328767	Abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	blocker	0.2019525816757481	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.4303907478335614	NOMEGESTROL ACETATE	rxcui:53744	NOMEGESTROL ACETATE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	EMB-01	drugbank:DB16091	EMB-01	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.4167275494896388	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	ChEMBL	33	inhibitor	0.192335792	CTS-1027	drugbank:DB08490	CTS-1027	FALSE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.729273212	ABEPRAZAN	ncit:C171876	FEXUPRAZAN	FALSE	FALSE	FALSE
MAGEA3	hgnc:6801	MAGEA3	ChEMBL	33	vaccine	35.00511415712966	ASTUPROTIMUT-R	ncit:C78478	ASTUPROTIMUT-R	FALSE	FALSE	TRUE
S1PR4	hgnc:3170	S1PR4	ChEMBL	33	binder	1.166837138570989	FINGOLIMOD LAURYL SULFATE	rxcui:2610292	FINGOLIMOD LAURYL SULFATE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.04685396	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1117184494376478	E7449	ncit:C102746	PARP/TANKYRASE INHIBITOR 2X-121	FALSE	FALSE	TRUE
ATR	hgnc:882	ATR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3500511415712967	E7449	ncit:C102746	PARP/TANKYRASE INHIBITOR 2X-121	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.056622219	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.0545251	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.056622219	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CCND1	hgnc:1582	CCND1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.032899543	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1099061668983662	NVP-BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.4773424657790409	TEMOLOZOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2243917574174978	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1795134059339982	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2311077079035849	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.062065805	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
TLE3	hgnc:11839	TLE3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2430910705356226	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1547594520630995	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	COSMIC	4-Sep-20	NULL	1.250182648468916	Savolitinib	ncit:C104732	SAVOLITINIB	FALSE	FALSE	TRUE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	RIMSULFURON	chembl:CHEMBL1867091	RIMSULFURON	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	RO-046790	iuphar.ligand:274	RO 04-6790	FALSE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.3409589041278863	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW279320X	chembl:CHEMBL1909397	GW279320X	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.006073762	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.2187819634820604	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	OXATOMIDE	rxcui:54236	OXATOMIDE	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.06466462	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	SJ000117447	chembl:CHEMBL592611	CHEMBL:CHEMBL592611	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.1450488155682168	PROTOCATECHUIC ACID	chembl:CHEMBL37537	PROTOCATECHUIC ACID	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.2323348284765243	20(S)-GINSENOSIDE RG3	iuphar.ligand:7658	GINSENOSIDE RG3	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.019483366	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	GNF-PF-516	chembl:CHEMBL602970	CHEMBL:CHEMBL602970	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.038173516	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.1470803115845784	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.036062961	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1060761035064535	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	GERONTOXANTHONE I	chembl:CHEMBL478791	GERONTOXANTHONE I	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CARBENDAZIM	ncit:C1154	CARBENDAZIM	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	1.500219178	N-NONYLDEOXYNOJIRIMYCIN	chembl:CHEMBL408500	CHEMBL:CHEMBL408500	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-1737	chembl:CHEMBL531710	CHEMBL:CHEMBL531710	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	NEOCUPROINE	chembl:CHEMBL375781	NEOCUPROINE	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.039960176	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007937668	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	ISOBONDUCELLIN	chembl:CHEMBL1253830	ISOBONDUCELLIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004176557	REPAGLINIDE	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	BUTAMBEN	rxcui:19861	BUTAMBEN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	NSC-133896	chembl:CHEMBL512908	CHEMBL:CHEMBL512908	FALSE	FALSE	FALSE
ADH1A	hgnc:249	ADH1A	PharmGKB	4/5/24	NULL	0.081030357	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.040703621	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.022220766	IUPHAR.LIGAND:320	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
SLC22A5	hgnc:10969	SLC22A5	DTC	9/2/20	NULL	35.00511415712966	CARNITINE	rxcui:2106	CARNITINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00988845	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1396480617970598	6-HYDROXYFLAVONE	chembl:CHEMBL138649	6-HYDROXYFLAVONE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	GNF-PF-4612	chembl:CHEMBL601550	CHEMBL:CHEMBL601550	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00808059	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
DHRS9	hgnc:16888	DHRS9	DTC	9/2/20	NULL	15.00219178	(+)-ZONAROL	chembl:CHEMBL461471	CHEMBL:CHEMBL461471	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005208578	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
SMARCA2	hgnc:11098	SMARCA2	DTC	9/2/20	NULL	1.875273972703374	AMINACRINE HYDROCHLORIDE	rxcui:81949	AMINACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:1891	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	LAVENDUSTIN A	ncit:C1142	LAVENDUSTIN A	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	0.9546849315580819	AKT INHIBITOR VIII	iuphar.ligand:5921	AKT INHIBITOR VIII	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	CYSTAMINE DIHYDROCHLORIDE	ncit:C97356	CYSTAMINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-5478	chembl:CHEMBL586982	CHEMBL:CHEMBL586982	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001426141	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003849818	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NSC-83217	chembl:CHEMBL120806	CHEMBL:CHEMBL120806	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00224853	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.010795163	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.118072806	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	METHYSTICIN	chembl:CHEMBL579224	METHYSTICIN	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.075010959	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	TCMDC-123605	chembl:CHEMBL547285	CHEMBL:CHEMBL547285	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.082043236	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
PSMC3	hgnc:9549	PSMC3	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	TROVAFLOXACIN MESYLATE	rxcui:221177	TROVAFLOXACIN MESYLATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	LEVOMETHADYL ACETATE HYDROCHLORIDE	rxcui:82043	LEVOMETHADYL ACETATE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A7	hgnc:2640	CYP3A7	NCI	14-Sep-17	NULL	0.4688184931758437	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.2206204673768676	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.3113103037689397	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.046673486	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.060492709	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.046673486	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.2590839041234926	ARRY-380	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	BREFELDIN A	drugbank:DB07348	BREFELDIN A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	CGP-13501	iuphar.ligand:7848	CGP13501	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	BROQUINALDOL	ncit:C73256	BROQUINALDOL	FALSE	FALSE	FALSE
PROTEIN C-ETS-2	hgnc:3489	ETS2	TTD	2020.06.01	NULL	5.250767123569449	TK216	drugbank:DB17414	TK216	FALSE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.054187483	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001284874	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.078136416	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
ERAP2	hgnc:29499	ERAP2	DTC	9/2/20	NULL	1.250182648468916	ESCULETIN	iuphar.ligand:5180	ESCULETIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	DECYLUBIQUINONE	chembl:CHEMBL217894	DECYLUBIQUINONE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.024861587	DICYCLOMINE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	8,2'-DIMETHOXYFLAVONE	chembl:CHEMBL1516007	8,2'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.034888818	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00149902	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
P2Y PURINOCEPTOR 12	hgnc:18124	P2RY12	TTD	2020.06.01	NULL	2.187819634820604	Brilinta	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.043502627	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006780433	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.033919684	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	0.364636606	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.006221288	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:837	iuphar.ligand:837	CXCL9	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.010966514	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	TYRPHOSTIN 1	iuphar.ligand:5917	AG 9	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	RS-23597-190	iuphar.ligand:254	RS 39604	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	TCMDC-123730	chembl:CHEMBL530280	CHEMBL:CHEMBL530280	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.05010274	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1215455352678113	GNF-PF-1295	chembl:CHEMBL579837	CHEMBL:CHEMBL579837	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1500219178162699	AMINACRINE HYDROCHLORIDE	rxcui:81949	AMINACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	BISANHYDRORUTILANTINONE	chembl:CHEMBL1436035	BISANHYDRORUTILANTINONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002269228	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.015930725	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1060761035064535	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.5469549087051511	MIGLITOL	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	OMEPRAZOLE MAGNESIUM	rxcui:236486	OMEPRAZOLE MAGNESIUM	TRUE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.7501095890813498	BREFELDIN A	drugbank:DB07348	BREFELDIN A	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	SJ000007704	chembl:CHEMBL589469	CHEMBL:CHEMBL589469	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.024709492	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	NSC-50690	chembl:CHEMBL1388703	CHEMBL:CHEMBL1388703	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NSC-74429	chembl:CHEMBL1269022	CHEMBL:CHEMBL1269022	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.075010959	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.036162308	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.026830696	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW827396X	chembl:CHEMBL427159	GW827396X	FALSE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.5834185692854944	PURVALANOLA	chembl:CHEMBL23327	PURVALANOLA	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.009571212	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.054243462	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.029074015	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.037003292	IUPHAR.LIGAND:4277	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.044198376	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6238	iuphar.ligand:6238	ADX88178	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	GNF-PF-2906	chembl:CHEMBL579957	CHEMBL:CHEMBL579957	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.011176601	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.546954909	TCMDC-124307	chembl:CHEMBL546865	CHEMBL:CHEMBL546865	FALSE	FALSE	FALSE
RCE1	hgnc:13721	RCE1	DTC	9/2/20	NULL	1.250182648468916	LEVOFLOXACIN	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.6422956726078837	DAMGO	iuphar.ligand:1647	DAMGO	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.021869084	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.364636606	GNF-PF-4612	chembl:CHEMBL601550	CHEMBL:CHEMBL601550	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.057700738	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.092443083	CEFOXITIN SODIUM	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	BENZANTHRONE	chembl:CHEMBL1607517	BENZANTHRONE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008027468	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.038608582	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2734774543525755	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.05814803	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.056826484	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009487052	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	ACETOSIDE	chembl:CHEMBL444478	ACETOSIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00383828	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	NSC-724440	chembl:CHEMBL515617	CHEMBL:CHEMBL515617	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.076098074	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	PREDNISOLONE ACETATE	rxcui:34372	PREDNISOLONE ACETATE	TRUE	FALSE	FALSE
GCLM	hgnc:4312	GCLM	NCI	14-Sep-17	NULL	0.7343730242754476	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.187193124	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.067403943	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	SULCONAZOLE NITRATE	rxcui:56798	SULCONAZOLE NITRATE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.6250913242344582	CHLORPYRAMIN HYDROCHLORIDE	chembl:CHEMBL550011	CHLORPYRAMIN HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BIFENOX	chembl:CHEMBL449928	BIFENOX	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	RS-16566	chembl:CHEMBL145725	CHEMBL:CHEMBL145725	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.082950507	GNF-PF-1241	chembl:CHEMBL528724	CHEMBL:CHEMBL528724	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.027781837	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	6-OXIMOTRYPTANTHRIN	chembl:CHEMBL308106	CHEMBL:CHEMBL308106	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	MANSONONE F	chembl:CHEMBL197655	MANSONONE F	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.022286787	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	AM-630	iuphar.ligand:750	AM-630	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1193356164447602	TCMDC-125575	chembl:CHEMBL587620	CHEMBL:CHEMBL587620	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.008178765	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.2375912725597036	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	TCMDC-123992	chembl:CHEMBL530149	CHEMBL:CHEMBL530149	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1115286134997759	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PREDNICARBATE	rxcui:34369	PREDNICARBATE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.7001022831425933	METRIBUZIN	chembl:CHEMBL1902519	METRIBUZIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005483257	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.070860555	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
LECITHIN-CHOLESTEROL ACYLTRANSFERASE	hgnc:6522	LCAT	TTD	2020.06.01	NULL	21.00306849427779	MEDI6012	drugbank:DB14833	MEDI6012	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	RIBOFLAVIN	rxcui:9346	RIBOFLAVIN	TRUE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	DTC	9/2/20	NULL	0.16256245	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIC	chembl:CHEMBL1095014	AESCULIOSIDE IIC	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.096167896	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	GANGLEOIDIN ACETATE	chembl:CHEMBL1590432	GANGLEOIDIN ACETATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.003744663	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	PAXILLINE	iuphar.ligand:2309	PAXILLINE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.016485925	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DIMETHYL YELLOW	chembl:CHEMBL263116	DIMETHYL YELLOW	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DINALINE	ncit:C79870	DINALINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	TCMDC-137192	chembl:CHEMBL268584	CHEMBL:CHEMBL268584	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.023004456	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.1154014752432846	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DESMEDIPHAM	chembl:CHEMBL16024	DESMEDIPHAM	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.002575799	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.01879301	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.03591496	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.039778539	NSC-377852	chembl:CHEMBL1466186	CHEMBL:CHEMBL1466186	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DOCUSATE SODIUM	rxcui:71722	DOCUSATE SODIUM	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	NSC-7387	chembl:CHEMBL119878	CHEMBL:CHEMBL119878	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.1022212937748757	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	DESMEDIPHAM	chembl:CHEMBL16024	DESMEDIPHAM	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NSC-123526	chembl:CHEMBL271165	CHEMBL:CHEMBL271165	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	ISONIAZID	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004540811	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.1229687850953032	TENOFOVIR	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	CHELERYTHRINE CHLORIDE	chembl:CHEMBL258893	CHELERYTHRINE CHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.002430911	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DYDROGESTERONE	rxcui:3706	DYDROGESTERONE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.008746905	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	DNDI1416917	chembl:CHEMBL1335833	CHEMBL:CHEMBL1335833	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	GNF-PF-1211	chembl:CHEMBL600968	CHEMBL:CHEMBL600968	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	HYDROCORTISONE VALERATE	rxcui:27199	HYDROCORTISONE VALERATE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.009767052	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.042619863	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1426838892274307	ATOMOXETINE HYDROCHLORIDE	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.021240967	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	SYROSINGOPINE	ncit:C152485	SYROSINGOPINE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	FLUORESCEIN	rxcui:25138	FLUORESCEIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	RO-194603	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	8-{[(4-BROMOPHENYL)METHYL]SULFANYL}CAFFEINE	chembl:CHEMBL1927670	CHEMBL:CHEMBL1927670	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	CANDESARTAN CILEXETIL	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	CAFFEIC ACID	rxcui:1311397	CAFFEIC ACID	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004861821	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1136529680426287	BREFELDIN A	drugbank:DB07348	BREFELDIN A	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	DTC	9/2/20	NULL	0.1367387271762877	VORICONAZOLE	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.021554873	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
PRKG2	hgnc:9416	PRKG2	DTC	9/2/20	NULL	0.3977853881492008	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.066676408	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	0.1562728310586145	Ranolazine	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.072927321	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.010195664	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	ADEFOVIR DIPIVOXIL	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.020399251	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.078722146	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.022099188	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	GLABRIDIN	rxcui:1603522	GLABRIDIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	NSC-133896	chembl:CHEMBL512908	CHEMBL:CHEMBL512908	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013825085	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	REL-CARINATIN B	chembl:CHEMBL2332126	CHEMBL:CHEMBL2332126	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	SHINJULACTONE B	chembl:CHEMBL1723340	SHINJULACTONE B	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.021608095	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.3443125982668492	MK-571	iuphar.ligand:10346	MK-571	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010588359	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003217973	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	BISSALICYL FUMARATE	chembl:CHEMBL1374986	BISSALICYL FUMARATE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012112496	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.025390557	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1136529680426287	IMETIT	iuphar.ligand:1250	IMETIT	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	DIFENPIRAMIDE	drugbank:DB13371	DIFENPIRAMIDE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.364636606	3-(4'-HYDROXYPHENYL)COUMARIN	chembl:CHEMBL71271	CHEMBL:CHEMBL71271	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.021240967	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
MKNK1	hgnc:7110	MKNK1	DTC	9/2/20	NULL	17.50255707856483	CGP-57380	iuphar.ligand:6010	MNK1 INHIBITOR	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.066297565	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.057700738	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	2.625383561784724	RITODRINE HYDROCHLORIDE	rxcui:105470	RITODRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	GNF-PF-4945	chembl:CHEMBL585628	CHEMBL:CHEMBL585628	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124995	chembl:CHEMBL529348	CHEMBL:CHEMBL529348	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.1640864726115453	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	NSC-116702	chembl:CHEMBL1477383	CHEMBL:CHEMBL1477383	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006999156	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.082429625	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	DTC	9/2/20	NULL	1.666910197958555	RALTITREXED	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	[14C]-TACRINE MONOHYDRATE MONOHYDROCHLORIDE	chembl:CHEMBL1337960	CHEMBL:CHEMBL1337960	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	DIETHANOLAMINE	rxcui:1362911	DIETHANOLAMINE	TRUE	FALSE	FALSE
CHRM4	hgnc:1953	CHRM4	DTC	9/2/20	NULL	1.944728564284981	VU10010	iuphar.ligand:7633	VU0010010	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	GNF-PF-2755	chembl:CHEMBL600738	CHEMBL:CHEMBL600738	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-2844	chembl:CHEMBL576353	CHEMBL:CHEMBL576353	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	CID 1540951	chembl:CHEMBL259421	CHEMBL:CHEMBL259421	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.6250913242344582	SJ000247817	chembl:CHEMBL590408	CHEMBL:CHEMBL590408	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.023620185	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.018206543	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1752592497853621	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.075442056	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.3977853881492007	AMINOQUINURIDE	rxcui:17747	AMINOQUINURIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DEFLAZACORT	rxcui:22396	DEFLAZACORT	TRUE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:6037	iuphar.ligand:6037	SB 218078	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.035670972	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	1.521961485092594	ALVESPIMYCIN	ncit:C38142	ALVESPIMYCIN	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-2356	chembl:CHEMBL601547	CHEMBL:CHEMBL601547	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.010742159	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	RS-16566	chembl:CHEMBL145725	CHEMBL:CHEMBL145725	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NONYL 4-HYDROXYBENZOATE	chembl:CHEMBL2271362	NONYL 4-HYDROXYBENZOATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005835482	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.2983390411119005	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.009018837	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.002956513	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DNDI1267127	chembl:CHEMBL135115	CHEMBL:CHEMBL135115	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.031032903	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	ALTANSERIN	ncit:C77258	ALTANSERIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	NORETHINDRONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.4907258993990139	GLYCITEIN	chembl:CHEMBL513024	GLYCITEIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016959842	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007699637	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	DTC	9/2/20	NULL	1.458546423213736	CURCUMIN PYRAZOLE	chembl:CHEMBL180239	CURCUMIN PYRAZOLE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.097870776	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.078722146	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1193356164447602	GNF-PF-3343	chembl:CHEMBL599943	CHEMBL:CHEMBL599943	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.050294704	TCMDC-123730	chembl:CHEMBL530280	CHEMBL:CHEMBL530280	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.082300425	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
VPS35	hgnc:13487	VPS35	DTC	9/2/20	NULL	15.00219178162699	MELAGATRAN	ncit:C66077	MELAGATRAN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.044124093	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.020117882	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.047518255	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	0.750109589	R-348	drugbank:DB06321	R-348	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	DTC	9/2/20	NULL	1.458546423213736	CHROMOCARB	ncit:C78116	CHROMOCARB	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.018081154	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	ACROLEIN	iuphar.ligand:2418	ACROLEIN	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2282942227638891	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005402024	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007873395	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011049594	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.3182283105193606	DNDI1417254	chembl:CHEMBL2094567	CHEMBL:CHEMBL2094567	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	OCTADEC-17-YNOIC ACID	iuphar.ligand:8851	17-OCTADECYNOIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001025821	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	DIHYDRALAZINE	rxcui:3409	DIHYDRALAZINE	FALSE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.047518255	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	DNDI1317721	chembl:CHEMBL1385558	CHEMBL:CHEMBL1385558	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.011110383	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010588359	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.092118721	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	CLOCAPRAMINE	ncit:C78010	CLOCAPRAMINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV011522	chembl:CHEMBL587892	CHEMBL:CHEMBL587892	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.057073556	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	CIS-RESVERATROL	chembl:CHEMBL87333	CIS-RESVERATROL	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	PIRARUBICIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	MESO-HEXESTROL	drugbank:DB07931	HEXESTROL	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1041818873724097	TCMDC-124336	chembl:CHEMBL527271	CHEMBL:CHEMBL527271	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.091796628	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BUNAMIDINE HYDROCHLORIDE	ncit:C75211	BUNAMIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	NIFUROXAZIDE	rxcui:31782	NIFUROXAZIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BENZOXIQUINE	rxcui:314521	BENZOXIQUINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	SPIPERONE	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
RASGRP3	hgnc:14545	RASGRP3	DTC	9/2/20	NULL	5.250767124	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	ROPINIROLE HYDROCHLORIDE	rxcui:236553	ROPINIROLE HYDROCHLORIDE	TRUE	FALSE	FALSE
RGS12	hgnc:9994	RGS12	DTC	9/2/20	NULL	1.640864726115453	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.2638576444004749	VITEXIN	drugbank:DB16836	VITEXIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002610374	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005107253	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	GRINIMIBINE	chembl:CHEMBL1477760	GRINIMIBINE	FALSE	FALSE	FALSE
GPR12	hgnc:4466	GPR12	DTC	9/2/20	NULL	15.00219178	CYCLOCITRINOL	chembl:CHEMBL523073	CYCLOCITRINOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001976425	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	1.312691780892362	BETULINIC ACID	ncit:C38126	BETULINIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.014330696	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	GNF-PF-3343	chembl:CHEMBL599943	CHEMBL:CHEMBL599943	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.03140411	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002529881	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.002541391	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004847011	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	DTC	9/2/20	NULL	0.1290114772375786	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	TRYPAN BLUE	rxcui:10878	TRYPAN BLUE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MINOPAFANT HYDROCHLORIDE	chembl:CHEMBL2104419	MINOPAFANT	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.212152207	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	BROMPERIDOL	rxcui:19777	BROMPERIDOL	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	CHLORPYRIFOS-METHYL	ncit:C163642	CHLORPYRIFOS-METHYL	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	PHENIDONE	chembl:CHEMBL7660	PHENIDONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	DICHLORODIPHENYLDICHLOROETHYLENE	chembl:CHEMBL363207	DICHLORODIPHENYLDICHLOROETHYLENE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003345716	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	3.500511415712966	8ALPHA-HYDROXYHIRSUTINOLIDE	chembl:CHEMBL2062863	CHEMBL:CHEMBL2062863	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124635	chembl:CHEMBL525519	CHEMBL:CHEMBL525519	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.014849455	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1AN	hgnc:17113	HIF1AN	DTC	9/2/20	NULL	1.346350544504987	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	TRIPROLIDINE HYDROCHLORIDE	rxcui:71534	TRIPROLIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IVA	chembl:CHEMBL1094677	AESCULIOSIDE IVA	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	NSC-50690	chembl:CHEMBL1388703	CHEMBL:CHEMBL1388703	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.012504804	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.017751072	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	2.100306849	SPERMINE TETRAHYDROCHLORIDE	chembl:CHEMBL1256357	SPERMINE TETRAHYDROCHLORIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	PHENELZINE	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	NSC-638080	chembl:CHEMBL136344	CHEMBL:CHEMBL136344	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	STILONIUM IODIDE	ncit:C73168	STILONIUM IODIDE	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.08334551	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	GNF-PF-1134	chembl:CHEMBL600694	CHEMBL:CHEMBL600694	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-872	chembl:CHEMBL600342	CHEMBL:CHEMBL600342	FALSE	FALSE	FALSE
PMM2	hgnc:9115	PMM2	DTC	9/2/20	NULL	1.500219178	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.003411804	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.033002936	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	7,3'-DIMETHOXYFLAVONE	chembl:CHEMBL1326944	7,3'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.016429184	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.032837818	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	2.187819634820604	L-3,4-DIHYDROXYPHENYLALANINE METHYL ESTER HCL	chembl:CHEMBL1255756	CHEMBL:CHEMBL1255756	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.050294704	ISOBOLDINE	chembl:CHEMBL462880	ISOBOLDINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.040515178	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.055622533	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007378818	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	MOXISYLYTE	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	DTC	9/2/20	NULL	0.3431873936973497	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.05853698	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.1121958787087489	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	DNDI1383301	chembl:CHEMBL1509103	CHEMBL:CHEMBL1509103	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007727398	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.015892152	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
CTSL	hgnc:2537	CTSL	DTC	9/2/20	NULL	26.25383561784724	GALLINAMIDE A	chembl:CHEMBL541700	GALLINAMIDE A	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	GNF-PF-265	chembl:CHEMBL602418	CHEMBL:CHEMBL602418	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
CDC42	hgnc:1736	CDC42	DTC	9/2/20	NULL	17.50255707856483	SECRAMINE B	chembl:CHEMBL1222039	SECRAMINE B	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW833373X	chembl:CHEMBL189459	GW833373X	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.5000730593875666	DNDI1417319	chembl:CHEMBL1392244	CHEMBL:CHEMBL1392244	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002933717	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	RO-046790	iuphar.ligand:274	RO 04-6790	FALSE	FALSE	FALSE
NPY1R	hgnc:7956	NPY1R	DTC	9/2/20	NULL	0.128067491	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	LASSBIO-1182	chembl:CHEMBL1173140	CHEMBL:CHEMBL1173140	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	XANTHOANGELOL F	chembl:CHEMBL1722838	XANTHOANGELOL F	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.027563082	CANDESARTAN CILEXETIL	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.039778539	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	NIHYDRAZONE	ncit:C175162	NIHYDRAZONE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.023080295	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	1.591141552596803	DAPHNORETIN	chembl:CHEMBL508494	DAPHNORETIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	TCMDC-123808	chembl:CHEMBL546493	CHEMBL:CHEMBL546493	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	METHYSTICIN	chembl:CHEMBL579224	METHYSTICIN	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.3977853881492007	SJ000024553	chembl:CHEMBL589238	CHEMBL:CHEMBL589238	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV006087	chembl:CHEMBL317364	CHEMBL:CHEMBL317364	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.42006137	DNDI1417368	chembl:CHEMBL2094652	CHEMBL:CHEMBL2094652	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	GR-113808	iuphar.ligand:247	GR 113808	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	DTC	9/2/20	NULL	0.043430663	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.026748686	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DNDI1383301	chembl:CHEMBL1509103	CHEMBL:CHEMBL1509103	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	MRS-1220	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.041214813	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.577007376	ACRIDIN-1-YLAMINE	chembl:CHEMBL146525	CHEMBL:CHEMBL146525	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.1988926940746004	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV008212	chembl:CHEMBL529984	CHEMBL:CHEMBL529984	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NSC-49789	chembl:CHEMBL469309	CHEMBL:CHEMBL469309	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.009205412	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	TCMDC-123927	chembl:CHEMBL531268	CHEMBL:CHEMBL531268	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.2386712328895204	CURCUMIN PYRAZOLE	chembl:CHEMBL180239	CURCUMIN PYRAZOLE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.033919684	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	ACETAMIDE	rxcui:2475952	ACETAMIDE	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.108374966	INDIRUBIN-3'-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.014537008	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
ABHD6	hgnc:21398	ABHD6	DTC	9/2/20	NULL	8.078103267029924	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW621431X	chembl:CHEMBL191705	GW621431X	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.2294915700860773	METOPROLOL	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	DTC	9/2/20	NULL	3.088686543276147	TIPLASININ	ncit:C77020	TIPLASININ	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2051080907644316	PIRENOXINE	rxcui:228080	PIRENOXINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	8-CYCLOPENTYLTHEOPHYLLINE	iuphar.ligand:385	8-CYCLOPENTYLTHEOPHYLLINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	(-)-ESEROLINE	chembl:CHEMBL310934	CHEMBL:CHEMBL310934	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.053038052	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.020195258	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005903055	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	LUPEOL	drugbank:DB12622	LUPEOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NSC-747260	chembl:CHEMBL595912	CHEMBL:CHEMBL595912	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.025942525	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
RARB	hgnc:9865	RARB	DTC	9/2/20	NULL	0.3633748874442526	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001392186	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	NIFUROXAZIDE	rxcui:31782	NIFUROXAZIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.01609924	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.043466615	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1232574442152452	GNF-PF-2755	chembl:CHEMBL600738	CHEMBL:CHEMBL600738	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.8468979231563628	CEFUROXIME	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.1396480617970598	CYSTAMINE HYDROCHLORIDE	chembl:CHEMBL1256388	CYSTAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	GNF-PF-1134	chembl:CHEMBL600694	CHEMBL:CHEMBL600694	FALSE	FALSE	FALSE
RCE1	hgnc:13721	RCE1	DTC	9/2/20	NULL	7.501095891	HTS-9915	chembl:CHEMBL512935	CHEMBL:CHEMBL512935	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.005164012	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	NSC-133896	chembl:CHEMBL512908	CHEMBL:CHEMBL512908	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005712634	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	DICYCLOMINE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	GAVESTINEL SODIUM	chembl:CHEMBL419045	GAVESTINEL SODIUM	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.002976625	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.038722471	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NIMETAZEPAM	ncit:C76536	NIMETAZEPAM	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.082950507	DNDI1417388	chembl:CHEMBL1528359	CHEMBL:CHEMBL1528359	FALSE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	1.060761035064535	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	CHELERYTHRINE CHLORIDE	chembl:CHEMBL258893	CHELERYTHRINE CHLORIDE	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.041872146	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(+)-9-DEMETHYLELEUTHERIN	chembl:CHEMBL594695	CHEMBL:CHEMBL594695	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	TOLNAFTATE	rxcui:10637	TOLNAFTATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	U-0124	chembl:CHEMBL97858	CHEMBL:CHEMBL97858	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.004546119	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.042516333	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	CID 670282	chembl:CHEMBL260213	CHEMBL:CHEMBL260213	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.088996053	DEQUALINIUM CHLORIDE	rxcui:3120	DEQUALINIUM CHLORIDE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.040112812	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	RILMENIDINE	rxcui:55679	RILMENIDINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	DNDI1417701	chembl:CHEMBL1326164	CHEMBL:CHEMBL1326164	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003132729	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.079557078	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1286952726365061	RS-67506	iuphar.ligand:3230	RS67506	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	1.050153425	DNDI1417502	chembl:CHEMBL1344912	CHEMBL:CHEMBL1344912	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,7-BIS[3-(DIETHYLAMINO)PROPIONAMIDO]ANTHRAQUINONE	chembl:CHEMBL91163	CHEMBL:CHEMBL91163	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.2122951667211368	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.063722902	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.001831769	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005593658	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	GNF-PF-107	chembl:CHEMBL578675	CHEMBL:CHEMBL578675	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	NSC-720622	chembl:CHEMBL1287980	CHEMBL:CHEMBL1287980	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005903055	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	TIOXOLONE	rxcui:2059173	TIOXOLONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	RO-106-9920	chembl:CHEMBL271023	CHEMBL:CHEMBL271023	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	GNF-PF-4864	chembl:CHEMBL583558	CHEMBL:CHEMBL583558	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.014732792	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	RESCINNAMINE	rxcui:9259	RESCINNAMINE	TRUE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.1988926940746003	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00347273	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.02654584	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	TCMDC-123992	chembl:CHEMBL530149	CHEMBL:CHEMBL530149	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.013411921	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	1.400204566285186	PHYTANIC ACID	iuphar.ligand:2813	PHYTANIC ACID	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.02654584	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	NSC-748118	chembl:CHEMBL2063681	CHEMBL:CHEMBL2063681	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	METHYL 2-(4-FLUOROBENZAMIDO)BENZOATE	chembl:CHEMBL250428	CHEMBL:CHEMBL250428	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	DTC	9/2/20	NULL	0.16256245	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	CLOFAZIMINE	rxcui:2592	CLOFAZIMINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.015184405	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.07596596	Flurbiprofen	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.020029629	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.026253836	Oxymetazoline	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.2590839041234926	ARRY380	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.6168664383892681	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.021751314	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.052824619	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.1099061668983662	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.041214813	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.1190650141398968	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.024513385	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.375054795	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.075768645	AP26113	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.043866058	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1808115400678185	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4296082192011368	AZD 2281	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1988926940746004	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1767935058440892	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.037666909	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2160809515872201	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.063440602	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.030202859	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.074797252	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.096167896	DOMPERIDONE	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.009756163	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.074797252	FEXOFENADINE HYDROCHLORIDE	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.08780547	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.3365876361262467	BROMODEOXYURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.1779921058837101	INTERFERON GAMMA	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	NCI	14-Sep-17	NULL	0.8751278539282416	METHYLCELLULOSE	rxcui:6873	METHYLCELLULOSE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.3879877184903534	ACE INHIBITOR	ncit:C247	ACE INHIBITOR	FALSE	FALSE	FALSE
APP	hgnc:620	APP	NCI	14-Sep-17	NULL	0.052116795	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1422972120208523	EGFR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1067229090156392	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.050222545	TETRAHYDROCANNABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.042689164	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FENHEXAMID	chembl:CHEMBL1688541	FENHEXAMID	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.043665423	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.032252869	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.086007651	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
BHLHB2	hgnc:1046	BHLHE40	NCI	14-Sep-17	NULL	2.625383561784725	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.042968634	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.060156088	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	0.082043236	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
CA3	hgnc:1374	CA3	NCI	14-Sep-17	NULL	1.640864726115453	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
CEACAM1	hgnc:1814	CEACAM1	NCI	14-Sep-17	NULL	0.8468979231563629	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.03136659	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	NCI	14-Sep-17	NULL	0.029715717	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
PSMA4	hgnc:9533	PSMA4	ChEMBL	33	inhibitor	0.1785975212098452	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	0.3153613888029699	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.3241214273808302	FREUNDS ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
CR1	hgnc:2334	CR1	NCI	14-Sep-17	NULL	8.751278539282415	TETANUS TOXOID	chembl:CHEMBL2108875	TETANUS TOXOID	FALSE	FALSE	FALSE
CRHR2	hgnc:2358	CRHR2	NCI	14-Sep-17	NULL	3.750547945	BRONCHODILATOR	ncit:C319	BRONCHODILATOR	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.089756703	RECOMBINANT INTERFERON	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.6250913242344582	BIOFLAVONOID	ncit:C306	BIOFLAVONOID	FALSE	FALSE	FALSE
PROTEIN KINASE N3	hgnc:17999	PKN3	TTD	2020.06.01	NULL	17.50255707856483	Atu-027	drugbank:DB12171	ATU-027	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.009838424	INTERLEUKIN-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.018641225	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.009838424	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.042073455	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.029515273	ACTH	iuphar.ligand:1331	ACTH	FALSE	FALSE	FALSE
CYP2B	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.1262203635473425	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.004195244	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.3684748858645228	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1878628666751145	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.072324616	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	0.4773424657790409	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.050488145	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.3302369260106572	TEGAFUR	rxcui:10995	URACIL	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	NCI	14-Sep-17	NULL	0.005254182	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
EIF4EBP1	hgnc:3288	EIF4EBP1	NCI	14-Sep-17	NULL	0.044198376	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
EPO	hgnc:3415	EPO	NCI	14-Sep-17	NULL	0.5770073762164232	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.138178082	INFIGRATINIB PHOSPHATE	ncit:C175088	INFIGRATINIB PHOSPHATE	TRUE	FALSE	FALSE
ELA2	hgnc:3309	ELANE	NCI	14-Sep-17	NULL	0.1223004764806549	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.167488584	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.3454452054979901	ANTHRAQUINONE	chembl:CHEMBL55659	ANTHRAQUINONE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.6908904109959803	VACCINE ADJUVANT	ncit:C2554	VACCINE ADJUVANT	FALSE	FALSE	FALSE
POLR3A	hgnc:30074	POLR3A	ChEMBL	33	inhibitor	17.50255707856483	TAS-106	drugbank:DB06656	TAS-106	FALSE	FALSE	FALSE
EZR	hgnc:12691	EZR	NCI	14-Sep-17	NULL	13.12691780892362	RO 31-8220	ncit:C1310	RO 31-8220	FALSE	FALSE	FALSE
ESRRG	hgnc:3474	ESRRG	NCI	14-Sep-17	NULL	0.5303805175322677	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.040097496	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.036013492	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.6035364509849942	SILICON PHTHALOCYANINE 4	ncit:C2651	SILICON PHTHALOCYANINE 4	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.7955707762984014	PENICILLIN	wikidata:Q12190	PENICILLIN	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	0.577007376	IUPHAR.LIGAND:9285	iuphar.ligand:9285	PRN694	FALSE	FALSE	FALSE
GALR1	hgnc:4132	GALR1	NCI	14-Sep-17	NULL	1.346350544504987	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.4167275494896388	DEMECOLCINE	ncit:C419	DEMECOLCINE	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1470803115845784	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	NCI	14-Sep-17	NULL	1.591141552596803	BUSERELIN	rxcui:1825	BUSERELIN	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.040766825	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.2917092846427472	DROLOXIFENE	ncit:C969	DROLOXIFENE	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.8751278539282416	DX-8951F	ncit:C1679	EXATECAN MESYLATE	FALSE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	0.1022544717345559	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	1.570742301922485	INTERLEUKIN-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.2287915957982331	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.016916131	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.182318303	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.082043236	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.079557078	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1143957978991165	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
IL5	hgnc:6016	IL5	NCI	14-Sep-17	NULL	0.9723642821424906	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
IL5	hgnc:6016	IL5	NCI	14-Sep-17	NULL	5.834185692854944	INTERLEUKIN-3	rxcui:1311225	INTERLEUKIN-3	FALSE	FALSE	FALSE
ITGA2B	hgnc:6138	ITGA2B	NCI	14-Sep-17	NULL	0.729273212	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
IRS1	hgnc:6125	IRS1	NCI	14-Sep-17	NULL	0.1661635165686534	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.3977853881492007	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
KCNA1	hgnc:6218	KCNA1	NCI	14-Sep-17	NULL	0.6819178082557728	DFMO	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.8751278539282418	INTRALIPID	rxcui:1309980	SOYBEAN SEED OIL	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	1.141471113819445	ANTI-CD20 ANTIBODY	ncit:C2543	TOSITUMOMAB	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.4118248724368196	ICRF-187	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	3.500511415712966	TUMOR VACCINES	ncit:C1663	ANTINEOPLASTIC VACCINE	FALSE	FALSE	FALSE
MT1E	hgnc:7397	MT1E	NCI	14-Sep-17	NULL	7.001022831425933	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.8036888454443035	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
MT1IP	hgnc:7401	MT1IP	NCI	14-Sep-17	NULL	3.621218705909965	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.016748858	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.1988926940746004	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.6563458904461813	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.008310806	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.002209082	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.041972559	PROTHYMOSIN ALPHA	ncit:C1203	RECOMBINANT PROTHYMOSIN ALPHA	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.1051204629343233	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	1.790034246671403	ANTIHYPERTENSIVE AGENT	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.091556532	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	2.187819634820604	ICR62	ncit:C2720	MONOCLONAL ANTIBODY ICR62	FALSE	FALSE	FALSE
PAEP	hgnc:8573	PAEP	NCI	14-Sep-17	NULL	5.000730593875666	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.2692701089009974	I3C	ncit:C1135	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.100976291	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1154014752432845	HEREGULIN	ncit:C1426	RECOMBINANT HEREGULIN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.201952582	RAS INHIBITOR	ncit:C1902	RAS INHIBITOR	FALSE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	0.3365876361262468	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	0.212581665	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	NCI	14-Sep-17	NULL	0.175610941	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.089298761	RU 486	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
PML	hgnc:9113	PML	NCI	14-Sep-17	NULL	1.591141552596803	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
SLC4A8	hgnc:11034	SLC4A8	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
PLAUR	hgnc:9053	PLAUR	NCI	14-Sep-17	NULL	13.12691780892362	RECOMBINANT INTERFERON GAMMA	ncit:C583	RECOMBINANT INTERFERON GAMMA	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.729273212	BENZNIDAZOLE	rxcui:18994	BENZNIDAZOLE	TRUE	FALSE	FALSE
RARG	hgnc:9866	RARG	NCI	14-Sep-17	NULL	0.2989051493493045	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
NCBIGENE:2907	hgnc:4589	GRINA	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9829	drugbank:DB02424	GELDANAMYCIN	FALSE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	1.750255707856483	3-HYDROXYTAMOXIFEN	ncit:C969	DROLOXIFENE	FALSE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	0.5527123287967842	BUSULPHAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.3462044257298538	ACE INHIBITOR	ncit:C247	ACE INHIBITOR	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.3231241306811969	INTRALIPID	rxcui:1309980	SOYBEAN SEED OIL	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1615620653405984	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.095036509	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	NCI	14-Sep-17	NULL	0.1691068316769549	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
SOAT1	hgnc:11177	SOAT1	NCI	14-Sep-17	NULL	0.2447910080918158	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:7459	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	NCI	14-Sep-17	NULL	0.07643038	HALOFUGINONE	ncit:C1120	HALOFUGINONE	FALSE	FALSE	FALSE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	0.4375639269641208	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
SULT2A1	hgnc:11458	SULT2A1	NCI	14-Sep-17	NULL	10.50153424713889	OXANDROLONE	rxcui:7779	OXANDROLONE	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	1.050153425	KLH	ncit:C1139	KEYHOLE LIMPET HEMOCYANIN	FALSE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.1489579325835305	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.2447910080918158	ALPHA-DIFLUOROMETHYLORNITHINE	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.028953775	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.11707396	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	OncoKB	23-Jul-20	NULL	1.346350544504987	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.596678082	CETYLPYRIDINIUM CHLORIDE HYDRATE	chembl:CHEMBL2003538	CETYLPYRIDINIUM CHLORIDE	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	OncoKB	23-Jul-20	NULL	1.367387271762877	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	OncoKB	23-Jul-20	NULL	2.080014029626545	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	OncoKB	23-Jul-20	NULL	1.500219178	Capmatinib	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.789589041	BESTATIN	ncit:C1015	UBENIMEX	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	OncoKB	23-Jul-20	NULL	0.2991890098899972	Taselisib	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	OncoKB	23-Jul-20	NULL	0.6783936852156912	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	PharmGKB	4/5/24	NULL	0.8975670296699914	ulinastatin	ncit:C102851	ULINASTATIN	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.1544343271638073	ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	TAS-115	chembl:CHEMBL3545144	TAS-115	FALSE	FALSE	FALSE
LEPR	hgnc:6554	LEPR	PharmGKB	4/5/24	NULL	0.3182283105193606	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	7.609807425462971	simvastatin acid	ncit:C96309	TENIVASTATIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.2713574740862764	pindolol	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.096521454	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:1617	ncit:C166495	DIPRENORPHINE	FALSE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.1842374429322614	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	PharmGKB	4/5/24	NULL	1.029066006546944	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
LGR5	hgnc:4504	LGR5	PharmGKB	4/5/24	NULL	1.323722804261206	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.034727296	flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.020257589	erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.048618214	ospemifene	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.040515178	rimegepant	rxcui:2282307	RIMEGEPANT	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.040515178	brivaracetam	rxcui:1739745	BRIVARACETAM	TRUE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2042	iuphar.ligand:2042	BOC-ATE	FALSE	FALSE	FALSE
FAM177A1	hgnc:19829	FAM177A1	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
RGL4	hgnc:31911	RGL4	PharmGKB	4/5/24	NULL	2.187819634820604	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.1325951293830669	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
OR52E2	hgnc:14769	OR52E2	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	PharmGKB	4/5/24	NULL	0.1241316104862754	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.28382525	sertraline	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HMBS	hgnc:4982	HMBS	PharmGKB	4/5/24	NULL	5.834185692854944	givosiran	rxcui:2265712	GIVOSIRAN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00626658	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
CYP2C18	hgnc:2620	CYP2C18	PharmGKB	4/5/24	NULL	0.8751278539282418	sertraline	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
P3H3	hgnc:19318	P3H3	PharmGKB	4/5/24	NULL	5.250767124	sertraline	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	0.2344092465879218	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
MT-ND1	hgnc:7455	MT-ND1	PharmGKB	4/5/24	NULL	6.620532460152785	gentamicin	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.016086909	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.1025540453822158	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.034251579	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
ZNF565	hgnc:26726	ZNF565	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.6250913242344582	levomethadone	rxcui:236913	LEVOMETHADONE	FALSE	FALSE	FALSE
ZNF211	hgnc:13003	ZNF211	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.076765601	WAY-100135	iuphar.ligand:79	WAY-100135	FALSE	FALSE	FALSE
IL18	hgnc:5986	IL18	PharmGKB	4/5/24	NULL	0.1905904582057876	interferon alfa-2a, recombinant	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
KLF4	hgnc:6348	KLF4	PharmGKB	4/5/24	NULL	2.500365296937833	hydroxyurea	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.044878351	tetrabenazine	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.1682938180631233	Biricodar	ncit:C71621	BIRICODAR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.014024485	diltiazem	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.016829382	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
ADD1	hgnc:243	ADD1	PharmGKB	4/5/24	NULL	1.640864726115453	spironolactone	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.015768069	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TP53AIP1	hgnc:29984	TP53AIP1	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	2-(PHENOXYMETHYL)BENZOTHIAZOLE	chembl:CHEMBL233302	2-(PHENOXYMETHYL)BENZOTHIAZOLE	FALSE	FALSE	FALSE
ELAVL2	hgnc:3313	ELAVL2	PharmGKB	4/5/24	NULL	0.1546617709446082	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	PharmGKB	4/5/24	NULL	0.019592415	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CACNA2D2	hgnc:1400	CACNA2D2	PharmGKB	4/5/24	NULL	0.1119566550867686	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:5385	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	PharmGKB	4/5/24	NULL	0.1567393171214761	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
ATP2A2	hgnc:812	ATP2A2	PharmGKB	4/5/24	NULL	0.068147529	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11159	iuphar.ligand:11159	COMPOUND 3 [PMID: 32636746]	FALSE	FALSE	FALSE
PTGER4	hgnc:9596	PTGER4	PharmGKB	4/5/24	NULL	0.092199598	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CCKBR	hgnc:1571	CCKBR	PharmGKB	4/5/24	NULL	0.024605282	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CA12	hgnc:1371	CA12	PharmGKB	4/5/24	NULL	0.1119566550867686	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:2744	drugbank:DB02545	FEXARAMINE	FALSE	FALSE	FALSE
PRKAB2	hgnc:9379	PRKAB2	PharmGKB	4/5/24	NULL	0.2165264793224515	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
SPTA1	hgnc:11272	SPTA1	PharmGKB	4/5/24	NULL	17.50255707856483	benazepril	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
SLCO1A2	hgnc:10956	SLCO1A2	PharmGKB	4/5/24	NULL	0.1750255707856483	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.2125816649218401	ticlopidine	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1318	iuphar.ligand:1318	[3H]SNAP-7941	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	PharmGKB	4/5/24	NULL	0.261046661	lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
RGS5	hgnc:10001	RGS5	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.059030547	deutetrabenazine	rxcui:1876905	DEUTETRABENAZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.035418328	pitolisant	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
ECHS1	hgnc:3151	ECHS1	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12644	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.3106962795011509	carvedilol	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UGT2B10	hgnc:12544	UGT2B10	PharmGKB	4/5/24	NULL	3.500511415712967	n-desmethylclozapine	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.070956312	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	1.750255707856483	interferon alfa-n1	rxcui:202912	INTERFERON ALFA-N1	FALSE	TRUE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.08334551	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.1250182648468916	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
PLCG1	hgnc:9065	PLCG1	PharmGKB	4/5/24	NULL	0.1241316104862754	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
WNT5B	hgnc:16265	WNT5B	PharmGKB	4/5/24	NULL	0.8824818695074705	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.2333674277141977	dacarbazine	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
NFATC2	hgnc:7776	NFATC2	PharmGKB	4/5/24	NULL	0.5645986154375753	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
RALBP1	hgnc:9841	RALBP1	PharmGKB	4/5/24	NULL	0.1260688385010672	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HLA-DPB1	hgnc:4940	HLA-DPB1	PharmGKB	4/5/24	NULL	0.2706580991530644	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
HLA-DPB1	hgnc:4940	HLA-DPB1	PharmGKB	4/5/24	NULL	0.5585922471882393	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.2083637747448194	AZELNIDIPINE	ncit:C73023	AZELNIDIPINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	PharmGKB	4/5/24	NULL	0.1988926940746003	risdiplam	rxcui:2390935	RISDIPLAM	TRUE	FALSE	FALSE
CYP2F1	hgnc:2632	CYP2F1	PharmGKB	4/5/24	NULL	0.7001022831425933	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.3561566847382379	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
CFHR4	hgnc:16979	CFHR4	PharmGKB	4/5/24	NULL	2.500365296937833	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.1031078472964055	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.1084869240406911	brivaracetam	rxcui:1739745	BRIVARACETAM	TRUE	FALSE	FALSE
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	0.3125456621172291	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.00182331	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.002712173	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.054243462	tolbutamide	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.019724895	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	PharmGKB	4/5/24	NULL	0.037925367	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.1268301237577161	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.2243917574174978	dabigatran	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
CHIA	hgnc:17432	CHIA	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.2592971419046642	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.040112812	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.2763561643983921	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	PharmGKB	4/5/24	NULL	0.106290832	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.2651902587661338	lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
HLA-DPB2	hgnc:4941	HLA-DPB2	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.088935758	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
IVL	hgnc:6187	IVL	PharmGKB	4/5/24	NULL	0.5645986154375753	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
SRD5A2	hgnc:11285	SRD5A2	PharmGKB	4/5/24	NULL	4.375639269641208	abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
SEPTIN3	hgnc:10750	SEPTIN3	PharmGKB	4/5/24	NULL	1.312691780892362	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
SULT2B1	hgnc:11459	SULT2B1	PharmGKB	4/5/24	NULL	0.546954909	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.138178082	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.4605936073306534	OXYPHENCYCLIMINE	rxcui:32698	OXYPHENCYCLIMINE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.1029562181092049	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.017859752	alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
CYP4F11	hgnc:13265	CYP4F11	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.099446347	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.099446347	buprenorphine	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.099258358	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
ARRB2	hgnc:712	ARRB2	PharmGKB	4/5/24	NULL	0.3017682254924971	buprenorphine	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.108711535	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
ABI1	hgnc:11320	ABI1	PharmGKB	4/5/24	NULL	0.8204323630577265	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.1093909817410302	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
CEP68	hgnc:29076	CEP68	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.026599631	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PTGER3	hgnc:9595	PTGER3	PharmGKB	4/5/24	NULL	0.1241316104862754	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.1909369863116163	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:833	iuphar.ligand:833	SB 225002	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	PharmGKB	4/5/24	NULL	0.6783936852156912	infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.1342907192728759	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
RHBDF2	hgnc:20788	RHBDF2	PharmGKB	4/5/24	NULL	0.760980743	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.2071308530007672	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.1037701012563132	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	TALC	12-May-16	inhibitor	0.2775246894064191	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.2300445618212245	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.1754935535952356	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
UNIPROT:P02675	hgnc:3662	FGB	TdgClinicalTrial	Jan-14	NULL	2.333674277141977	ALFIMEPRASE	ncit:C79877	ALFIMEPRASE	FALSE	FALSE	FALSE
UNIPROT:O75899	hgnc:4507	GABBR2	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
UNIPROT:P04275	hgnc:12726	VWF	TdgClinicalTrial	Jan-14	NULL	8.290684931951763	ALX-0681	rxcui:2110604	CAPLACIZUMAB-YHDP	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.5114383561918295	AN-2728	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.053038052	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.04362008	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	ANTI-CD3 MONOCLONAL ANTIBODY	ncit:C112883	ANTI-CD3 MONOCLONAL ANTIBODY	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.055563673	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.175415383	APC-100	chembl:CHEMBL37676	APC-100	FALSE	FALSE	FALSE
UNIPROT:Q9UBU3	hgnc:18129	GHRL	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	ARD-07	rxcui:1999420	MACIMORELIN	TRUE	FALSE	FALSE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.1182605208011137	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
UNIPROT:Q02750	hgnc:6840	MAP2K1	TdgClinicalTrial	Jan-14	NULL	0.375054795	ARRY-162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
UNIPROT:P36507	hgnc:6842	MAP2K2	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	ARRY-162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
UNIPROT:Q08289	hgnc:1402	CACNB2	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	1.129197231	ART621	chembl:CHEMBL2108739	PLACULUMAB	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1223955040459079	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.081597003	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P61812	hgnc:11768	TGFB2	TdgClinicalTrial	Jan-14	NULL	15.00219178	BELAGENPUMATUCEL-L	ncit:C73438	BELAGENPUMATUCEL-L	FALSE	FALSE	TRUE
UNIPROT:P08235	hgnc:7979	NR3C2	TdgClinicalTrial	Jan-14	NULL	0.046840028	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	agonist	0.3621218705909966	IUPHAR.LIGAND:4156	iuphar.ligand:4156	CGS8216	FALSE	FALSE	FALSE
UNIPROT:P68366	hgnc:12407	TUBA4A	TdgClinicalTrial	Jan-14	NULL	0.058212496	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
UNIPROT:P30874	hgnc:11331	SSTR2	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P11177	hgnc:8808	PDHB	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	1.500219178	INSULIN GLULISINE	rxcui:400008	INSULIN GLULISINE, HUMAN	TRUE	FALSE	FALSE
UNIPROT:Q15118	hgnc:8809	PDK1	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
UNIPROT:Q15120	hgnc:8811	PDK3	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.42006137	CS-7017	ncit:C64764	EFATUTAZONE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	EW-A-401	drugbank:DB05525	EW-A-401	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.042845917	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.106290832	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.4930297768609811	FIPAMEZOLE	ncit:C65684	FIPAMEZOLE	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2004109589148645	FLUOCINONIDE	rxcui:4462	FLUOCINONIDE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	DEXMETHYLPHENIDATE	rxcui:352372	DEXMETHYLPHENIDATE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.3271505995993426	DEXMETHYLPHENIDATE	rxcui:352372	DEXMETHYLPHENIDATE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1077080435603989	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.2812910959055062	KETOPROFEN	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	LASOFOXIFENE	ncit:C80679	LASOFOXIFENE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.064824285	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	M0002	drugbank:DB05091	M0002	FALSE	FALSE	FALSE
UNIPROT:P15391	hgnc:1633	CD19	TdgClinicalTrial	Jan-14	NULL	3.842024724563012	MDX-1342	chembl:CHEMBL2109337	MDX-1342	FALSE	FALSE	FALSE
UNIPROT:P02778	hgnc:10637	CXCL10	TdgClinicalTrial	Jan-14	NULL	6.177373086552294	MDX-1100	iuphar.ligand:9047	ELDELUMAB	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.2294915700860773	METOPROLOL	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1245241215075758	PRAMIPEXOLE	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
UNIPROT:P31749	hgnc:391	AKT1	TdgClinicalTrial	Jan-14	NULL	0.3697723326457359	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
UNIPROT:P31751	hgnc:392	AKT2	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
UNIPROT:Q9Y243	hgnc:393	AKT3	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
UNIPROT:O43613	hgnc:4848	HCRTR1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	SUVOREXANT	rxcui:1547099	SUVOREXANT	TRUE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	MOCLOBEMIDE	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
UNIPROT:P28908	hgnc:11923	TNFRSF8	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	MOR208	rxcui:2387211	TAFASITAMAB	TRUE	FALSE	FALSE
UNIPROT:A8K7I4	hgnc:2015	CLCA1	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	TALNIFLUMATE	rxcui:236770	TALNIFLUMATE	FALSE	FALSE	FALSE
UNIPROT:P12268	hgnc:6053	IMPDH2	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.1810609352954982	MPC-3100	ncit:C84836	HSP90 INHIBITOR LAM-003A	FALSE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.061055432	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	1.225178995499538	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.062509132	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.1235474617310458	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.08178765	NORELGESTROMIN	rxcui:326374	NORELGESTROMIN	TRUE	FALSE	FALSE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.1037701012563132	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.151537291	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344583	RECOMBINANT INTERFERON ALFA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	2.423430980108977	PONEZUMAB	ncit:C97941	PONEZUMAB	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.009745299	PRASTERONE	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	1.369765336583334	PS433540	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.1562728310586145	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P40238	hgnc:7217	MPL	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	SB-559448	drugbank:DB05930	SB-559448	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.2083637747448194	TABERMINOGENE VADENOVEC	drugbank:DB05011	TABERMINOGENE VADENOVEC	FALSE	FALSE	FALSE
UNIPROT:O60895	hgnc:9844	RAMP2	TdgClinicalTrial	Jan-14	NULL	7.501095890813499	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	0.3236220106976548	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
UNIPROT:P11597	hgnc:1869	CETP	TdgClinicalTrial	Jan-14	NULL	8.078103267029922	TORCETRAPIB	ncit:C91058	TORCETRAPIB	FALSE	FALSE	FALSE
UNIPROT:P08887	hgnc:6019	IL6R	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	TOCILIZUMAB	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	V24343	drugbank:DB05201	V24343	FALSE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	1.009762908	VEGLIN	drugbank:DB05890	VEGLIN	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1640864726115453	VB-201	drugbank:DB15259	VB-201	FALSE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	VELUSETRAG	ncit:C84238	VELUSETRAG	FALSE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.2128689374420047	VILAZODONE	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P25103	hgnc:11526	TACR1	TdgClinicalTrial	Jan-14	NULL	2.128689374420047	VESTIPITANT	ncit:C95194	VESTIPITANT	FALSE	FALSE	FALSE
UNIPROT:P30559	hgnc:8529	OXTR	TdgClinicalTrial	Jan-14	NULL	4.118248724368195	CARBETOCIN	ncit:C96858	CARBETOCIN	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.096167896	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.091476779	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.087222045	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	0.099446347	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	1.666910197958555	DECAMETHONIUM	ncit:C77363	DECAMETHONIUM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	DESOGESTREL	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.088945801	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.076098074	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.07963752	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.075261832	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.081533651	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.11707396	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TdgClinicalTrial	Jan-14	NULL	18.37768493249307	FOLLITROPIN BETA	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.09969811	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.089501712	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.086551106	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.2019525816757481	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P10827	hgnc:11796	THRA	TdgClinicalTrial	Jan-14	NULL	0.9092237443410304	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.085147575	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.7160136986685613	LEVOBUNOLOL	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.07160137	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.080781033	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.076840494	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.079758488	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q02127	hgnc:2867	DHODH	TdgClinicalTrial	Jan-14	NULL	1.151484018326633	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.3580068493342807	MELOXICAM	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.1842374429322614	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.2651902587661338	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.1861974157294131	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.1682938180631233	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	MILRINONE	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.049629179	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1383601350084176	MOLINDONE	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.1457197166578015	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:Q9UGM1	hgnc:14079	CHRNA9	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1620607136904151	PACRITINIB CITRATE	rxcui:2595242	PACRITINIB CITRATE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1640864726115453	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1325951293830669	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.4303907478335614	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.08178765	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.1290114772375786	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.070574827	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.049723174	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TdgClinicalTrial	Jan-14	NULL	0.4023576339899961	TIAGABINE	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ZOXAMIDE	chembl:CHEMBL1893025	ZOXAMIDE	FALSE	FALSE	FALSE
UNIPROT:P30531	hgnc:11042	SLC6A1	TdgClinicalTrial	Jan-14	NULL	14.00204566285186	TIAGABINE	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.1750255707856483	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008857569	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
UNIPROT:P08183	hgnc:40	ABCB1	TEND	1-Aug-11	NULL	0.012945678	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.1731022128649269	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.054243462	TRIMIPRAMINE	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	0.7955707762984016	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.0037759	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
UNIPROT:P23415	hgnc:4326	GLRA1	TEND	1-Aug-11	NULL	0.1591141552596803	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1204304386139782	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TEND	1-Aug-11	NULL	0.2180551131050435	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TEND	1-Aug-11	NULL	0.1785975212098452	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:O15399	hgnc:4588	GRIN2D	TEND	1-Aug-11	NULL	0.7778914257139926	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	1.675776741564718	CYCRIMINE	rxcui:22037	CYCRIMINE	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.021370644	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
UNIPROT:P38484	hgnc:5440	IFNGR2	TEND	1-Aug-11	NULL	105.0153424713889	INTERFERON GAMMA-1B	rxcui:5882	INTERFERON GAMMA-1B	TRUE	TRUE	FALSE
UNIPROT:P13612	hgnc:6140	ITGA4	TEND	1-Aug-11	NULL	5.834185692854944	NATALIZUMAB	rxcui:354770	NATALIZUMAB	TRUE	TRUE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1115286134997759	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.2775246894064191	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	ETHOPROPAZINE	rxcui:4134	PROFENAMINE	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TEND	1-Aug-11	NULL	0.2941606231691568	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.047886613	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.073540156	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.1555782851427985	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.067883221	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.068637479	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.054953083	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.056826484	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.192335792	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.3697723326457359	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
UNIPROT:P23945	hgnc:3969	FSHR	TEND	1-Aug-11	NULL	18.37768493249307	FOLLITROPIN BETA	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.305277158	FOSPROPOFOL	rxcui:828682	FOSPROPOFOL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.059532507	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.2234368988752957	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1265245090016735	TIVOZANIB HYDROCHLORIDE	rxcui:2534245	TIVOZANIB HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TEND	1-Aug-11	NULL	3.500511415712966	IBANDRONATE	rxcui:115264	IBANDRONATE	TRUE	FALSE	FALSE
UNIPROT:P63316	hgnc:11943	TNNC1	TEND	1-Aug-11	NULL	4.500657534	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.1754935535952356	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-466314A	chembl:CHEMBL218720	GSK-466314A	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TEND	1-Aug-11	NULL	0.1228249619548409	AMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TEND	1-Aug-11	NULL	0.9546849315580818	LIRAGLUTIDE RECOMBINANT	rxcui:475968	LIRAGLUTIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1562728310586145	METARAMINOL	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	PH-011685	chembl:CHEMBL126804	CHEMBL:CHEMBL126804	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.1013661606866689	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.079798892	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.1315981735230438	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.1071585127259071	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.108711535	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.2651902587661338	METHYLPHENOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013964806	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P12268	hgnc:6053	IMPDH2	TEND	1-Aug-11	NULL	2.625383561784724	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TEND	1-Aug-11	NULL	1.406455479527531	MISOPROSTOL	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
TDO2	hgnc:11708	TDO2	NCI	14-Sep-17	NULL	0.3962843112127886	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.049629179	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.06757744	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.014699796	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.027093742	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.05814803	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TEND	1-Aug-11	NULL	0.7242437411819932	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.1693795846312726	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TEND	1-Aug-11	NULL	0.7721716358190367	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.4605936073306534	OXYPHENCYCLIMINE	rxcui:32698	OXYPHENCYCLIMINE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.097236428	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.053038052	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.375054795	gemtuzumab ozogamicin	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.093763699	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.1093909817410302	ABI-011	ncit:C116890	NANOPARTICLE ALBUMIN-BOUND THIOCOLCHICINE DIMER NAB-5404	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	1.779921058837101	TAS-119	chembl:CHEMBL3545326	TAS-119	FALSE	FALSE	FALSE
STIMULATOR OF INTERFERON GENES PROTEIN	hgnc:27962	STING1	TTD	2020.06.01	NULL	52.50767123569449	ADU-S100	drugbank:DB14722	ADU-S100	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.2386712328895204	DCC-3014	ncit:C175876	VIMSELTINIB	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.2187819634820604	PATRITUMAB DERUXTECAN	ncit:C136987	PATRITUMAB DERUXTECAN	FALSE	FALSE	TRUE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	2.625383561784724	MEDI9197	ncit:C124653	TELRATOLIMOD	FALSE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.2778183663264258	ME-401	ncit:C123925	ZANDELISIB	FALSE	FALSE	FALSE
AMP-ACTIVATED PROTEIN KINASE	hgnc:9377	PRKAA2	TTD	2020.06.01	NULL	4.773424657790408	IM156	ncit:C153372	LIXUMISTAT ACETATE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	GNF-PF-5294	chembl:CHEMBL579725	CHEMBL:CHEMBL579725	FALSE	FALSE	FALSE
OXALOSUCCINATE DECARBOXYLASE	hgnc:5382	IDH1	TTD	2020.06.01	NULL	0.5135224570728067	IDH305	chembl:CHEMBL4167360	IDH305	FALSE	FALSE	FALSE
HEPATITIS A VIRUS CELLULAR RECEPTOR 2	hgnc:18437	HAVCR2	TTD	2020.06.01	NULL	8.751278539282415	LY3321367	ncit:C137820	ANTI-TIM3 MONOCLONAL ANTIBODY LY3321367	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.022477599	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 BETA	hgnc:5258	HSP90AB1	TTD	2020.06.01	NULL	1.141471113819445	PU-H71	chembl:CHEMBL200102	PU-H71	FALSE	FALSE	FALSE
EPHRIN TYPE-B RECEPTOR 2	hgnc:3393	EPHB2	TTD	2020.06.01	NULL	0.1151484018326633	MK-8353	iuphar.ligand:9974	MK-8353	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	1.640864726115453	BAL-101553	ncit:C97664	LISAVANBULIN	FALSE	FALSE	FALSE
PROTEIN KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	0.1367387271762877	MGCD516	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	Vecabrutinib	ncit:C136416	VECABRUTINIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003313623	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
CYTOKINE ML-1	hgnc:16404	IL17F	TTD	2020.06.01	NULL	7.501095891	Bimekizumab	rxcui:2668041	BIMEKIZUMAB	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	L-755507	iuphar.ligand:3931	L 755507	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION GENE 3 PROTEIN	hgnc:6476	LAG3	TTD	2020.06.01	NULL	6.563458904461812	GSK2831781	wikidata:Q19904145	GSK2831781	FALSE	FALSE	FALSE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	2.019525817	Bimekizumab	rxcui:2668041	BIMEKIZUMAB	TRUE	FALSE	FALSE
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	0.3804903712731485	PF-06651600	chembl:CHEMBL4085457	PF-06651600	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	1.109316997937207	Difelikefalin	rxcui:2569089	DIFELIKEFALIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
GLUCAGON	hgnc:4191	GCG	TTD	2020.06.01	NULL	2.019525817	MEDI0382	chembl:CHEMBL4297630	COTADUTIDE	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	0.8078103267029924	(+)-JQ1	iuphar.ligand:7511	(+)-JQ1	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
CYTOCHROME P450 3A	ncbigene:1574	CYP3A	TTD	2020.06.01	NULL	0.4039051633514962	Cobicistat	rxcui:1306284	COBICISTAT	TRUE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1A	hgnc:7463	MTNR1A	TTD	2020.06.01	NULL	5.625821918110125	Tasimelteon	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	CLANFENUR	ncit:C78082	CLANFENUR	FALSE	FALSE	FALSE
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	2.692701089009974	Lesinurad	rxcui:1731031	LESINURAD	TRUE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1B	hgnc:7464	MTNR1B	TTD	2020.06.01	NULL	7.876150685354174	Tasimelteon	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
GLUCOSE-DEPENDENT INSULINOTROPIC RECEPTOR	hgnc:19060	GPR119	TTD	2020.06.01	NULL	1.750255707856483	LEZ763	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.7395446652914718	Pegdinetanib	ncit:C62791	PEGDINETANIB	FALSE	FALSE	TRUE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	0.750109589	AGT-182	drugbank:DB17630	AGT-182	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	0.750109589	DM-199	chembl:CHEMBL4297936	RECOMBINANT HUMAN KALLIKREIN-1	FALSE	FALSE	FALSE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	2.282942227638891	POL-6014	iuphar.ligand:11275	LONODELESTAT	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.4412409347537352	Rivastigmine	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	8.078103267029922	Ranirestat	ncit:C96307	RANIRESTAT	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	0.2051080907644316	Mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.05293112	IUPHAR.LIGAND:6953	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE BETA	hgnc:5960	IKBKB	TTD	2020.06.01	NULL	7.501095891	SAR-113945	chembl:CHEMBL3544945	SAR-113945	FALSE	FALSE	FALSE
INTERLEUKIN-22	hgnc:14900	IL22	TTD	2020.06.01	NULL	78.76150685354175	Fezakinumab	ncit:C87764	FEZAKINUMAB	FALSE	FALSE	FALSE
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	6.058577450272442	RDEA3170	ncit:C152863	VERINURAD	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.002737341	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
METHYLMALONYL-COA MUTASE	hgnc:7526	MMUT	TTD	2020.06.01	NULL	26.25383561784724	Hydroxocobalamin	rxcui:5514	HYDROXOCOBALAMIN	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	2.669881588255652	Saprisartan	ncit:C152297	SAPRISARTAN	FALSE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR ALPHA	hgnc:6008	IL2RA	TTD	2020.06.01	NULL	2.059124362184098	LMB-2	chembl:CHEMBL2109367	LMB-2	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:5586	rxcui:2472778	RELUGOLIX	TRUE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.8975670296699914	HTF 919	rxcui:139778	TEGASEROD	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.4167275494896388	DENBUFYLLINE	ncit:C76316	DENBUFYLLINE	FALSE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	0.2344092465879218	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
SOMATOTROPIN	hgnc:4261	GH1	TTD	2020.06.01	NULL	4.375639269641208	Albutropin	chembl:CHEMBL4298125	ALBUSOMATROPIN	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	1.346350544504987	Moclobemide	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:2089	iuphar.ligand:2089	NEUROKININ A	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.034590034	Ocaperidone	ncit:C76441	OCAPERIDONE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.2393966773663883	Propantheline	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
GLUTATHIONE-DEPENDENT PGD SYNTHASE	hgnc:17890	HPGDS	TTD	2020.06.01	NULL	13.12691780892362	Praziquantel	rxcui:8628	PRAZIQUANTEL	TRUE	FALSE	FALSE
ALPHA-1-ANTITRYPSIN	hgnc:8941	SERPINA1	TTD	2020.06.01	NULL	13.12691780892362	Igmesine	ncit:C170052	IGMESINE	FALSE	FALSE	FALSE
S-ADENOSYLMETHIONINE DECARBOXYLASE PROENZYME	hgnc:457	AMD1	TTD	2020.06.01	NULL	0.6035364509849942	Tromethamine	rxcui:10865	TROMETHAMINE	TRUE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.9723642821424906	DEXMETHYLPHENIDATE HYDROCHLORIDE	rxcui:352372	DEXMETHYLPHENIDATE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.021751314	MIBEFRADIL	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
CALCINEURIN	hgnc:9314	PPP3CA	TTD	2020.06.01	NULL	0.1508841127462485	Cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CONNECTIVE TISSUE GROWTH FACTOR	hgnc:2500	CCN2	TTD	2020.06.01	NULL	0.3365876361262467	Ocaperidone	ncit:C76441	OCAPERIDONE	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.010569177	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CARCINOEMBRYONIC ANTIGEN CGM1	hgnc:1815	CEACAM3	TTD	2020.06.01	NULL	17.50255707856483	Arcitumomab	ncit:C1494	ARCITUMOMAB	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-4	hgnc:3682	FGF4	TTD	2020.06.01	NULL	10.50153424713889	Alferminogene tadenovec	ncit:C184852	ALFERMINOGENE TADENOVEC	FALSE	FALSE	FALSE
PSMD4	hgnc:9561	PSMD4	MyCancerGenome	20-Jun-17	other/unknown	0.3488881809680698	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.1232574442152452	Zotarolimus	ncit:C82294	ZOTAROLIMUS	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	4.565884455277782	ERITORAN	ncit:C80053	ERITORAN	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	BIIB-021	ncit:C62517	HSP90 INHIBITOR BIIB021	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.1071585127259071	Mebendazole	rxcui:6672	MEBENDAZOLE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.3977853881492006	Nebivolol	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.3236220106976548	Telmisartan	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.1286952726365061	Malathion	rxcui:6606	MALATHION	TRUE	FALSE	FALSE
PANCREATIC ELASTASE 1	hgnc:3308	CELA1	TTD	2020.06.01	NULL	1.944728564284981	Sivelestat	ncit:C66539	SIVELESTAT	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.062139256	Carvedilol	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.3918482928036902	PHA-739358	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	1.193356164447602	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	12.11715490054488	MDX-1411	chembl:CHEMBL2109492	MDX-1411	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.9546849315580818	Taspoglutide	ncit:C152518	TASPOGLUTIDE	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.5114383561918295	AN2728	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	0.2983390411119005	SSR149415	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.020446912	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.6213925590023018	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
NICOTINIC ACID RECEPTOR	hgnc:24827	HCAR2	TTD	2020.06.01	NULL	8.751278539282415	MK-0354	drugbank:DB05939	MK-0354	FALSE	FALSE	FALSE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	1.640864726115453	CH-4051	iuphar.ligand:9844	CH-4051	FALSE	FALSE	FALSE
ILEAL SODIUM/BILE ACID COTRANSPORTER	hgnc:10906	SLC10A2	TTD	2020.06.01	NULL	2.019525817	264W94	iuphar.ligand:6529	264W94	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.3860858179095183	Ladostigil	ncit:C77584	LADOSTIGIL	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	7.876150685354174	AZD-8848	drugbank:DB14868	AZD-8848	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 1	hgnc:11036	SLC5A1	TTD	2020.06.01	NULL	6.300920548283339	LX-4211	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
UNIPROT:Q96LZ3	hgnc:9318	PPP3R2	TEND	1-Aug-11	NULL	1.207072901969988	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
STEROID 17-ALPHA-MONOOXYGENASE	hgnc:2593	CYP17A1	TTD	2020.06.01	NULL	7.501095891	CFG920	ncit:C102855	CYP17/CYP11B2 INHIBITOR LAE001	FALSE	FALSE	FALSE
ILEAL SODIUM/BILE ACID COTRANSPORTER	hgnc:10906	SLC10A2	TTD	2020.06.01	NULL	4.039051633514961	GSK2330672	chembl:CHEMBL2387408	LINERIXIBAT	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	2.625383561784724	GS-9620	chembl:CHEMBL2424780	VESATOLIMOD	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	SAR-3419	hemonc:114	COLTUXIMAB RAVTANSINE	FALSE	FALSE	FALSE
LEUKOCYTE ANTIGEN CD37	hgnc:1666	CD37	TTD	2020.06.01	NULL	35.00511415712966	IMGN529	ncit:C100101	NARATUXIMAB EMTANSINE	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	0.2386712328895204	Thiopental	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
HISTAMINE H2 RECEPTOR	hgnc:5183	HRH2	TTD	2020.06.01	NULL	9.845188356692718	Betazole	drugbank:DB00272	BETAZOLE	TRUE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.6177373086552294	MSB2311	ncit:C155931	BETIFISOLIMAB	FALSE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	7.001022831425932	Erenumab	rxcui:2045613	ERENUMAB	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.1715936968486748	Mepenzolate	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.012561644	Flufenamic Acid	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	0.091159151	MEDETOMIDINE	rxcui:52016	MEDETOMIDINE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.1232574442152452	MEDETOMIDINE	rxcui:52016	MEDETOMIDINE	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	0.2917092846427472	Apremilast	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:2006	iuphar.ligand:2006	CH 275	FALSE	FALSE	FALSE
GTP CYCLOHYDROLASE-I	hgnc:4193	GCH1	TTD	2020.06.01	NULL	8.751278539282415	ProSavin	wikidata:Q7246687	PROSAVIN	FALSE	FALSE	FALSE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	5.250767123569449	PF-06291874	drugbank:DB15065	PF-06291874	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	3.281729452230906	DE-117	chembl:CHEMBL4297666	OMIDENEPAG ISOPROPYL	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	1.826353782111112	X-396	drugbank:DB13104	X-396	FALSE	FALSE	TRUE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	3.281729452230906	ATLCAR.CD30 cells	ncit:C155294	AUTOLOGOUS CD30CAR-CD28-CD3ZETA-EXPRESSING T-LYMPHOCYTES	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	2.561349816375341	YESCARTA	rxcui:1987398	AXICABTAGENE CILOLEUCEL	TRUE	FALSE	FALSE
NKG2 D ACTIVATING NK RECEPTOR	hgnc:18788	KLRK1	TTD	2020.06.01	NULL	13.12691780892362	CYAD-101	ncit:C121536	AUTOLOGOUS NKG2D CAR-CD3ZETA-DAP10-EXPRESSING T-LYMPHOCYTES CYAD-01	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	1.029066006546944	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
SURFACE GLYCOPROTEIN LFA-3	hgnc:1688	CD58	TTD	2020.06.01	NULL	8.751278539282415	Alefacept	rxcui:299635	ALEFACEPT	TRUE	TRUE	FALSE
SOMATOSTATIN RECEPTOR TYPE 4	hgnc:11333	SSTR4	TTD	2020.06.01	NULL	3.500511415712967	177Lu-DOTATATE	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	5.834185692854944	MOR-202	chembl:CHEMBL4594579	FELZARTAMAB	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.1930429089547591	SR46349B	ncit:C95215	EPLIVANSERIN FUMARATE	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.1591141552596802	LY2944876	chembl:CHEMBL3990012	PEGAPAMODUTIDE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	MTC-DOX	ncit:C2644	DOXORUBICIN-MAGNETIC TARGETED CARRIER COMPLEX	FALSE	FALSE	FALSE
APOPTOSIS INHIBITOR SURVIVIN	hgnc:593	BIRC5	TTD	2020.06.01	NULL	0.596678082	EZN-3042	ncit:C92578	SURVIVIN MRNA ANTAGONIST EZN-3042	FALSE	FALSE	FALSE
ENDOTHELIN-CONVERTING ENZYME	hgnc:3146	ECE1	TTD	2020.06.01	NULL	5.250767123569449	SLV-334	drugbank:DB15356	SLV-334	FALSE	FALSE	FALSE
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	7.501095891	SAR164877	iuphar.ligand:8965	FASINUMAB	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.400821918	ETIPREDNOL DICLOACETATE	ncit:C80816	ETIPREDNOL DICLOACETATE	FALSE	FALSE	FALSE
TAX TRANSCRIPTIONALLY-ACTIVATED GLYCOPROTEIN 1	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	0.5834185692854944	AMG 386	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.015534814	CUDC-907	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.290901226	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	0.4412409347537352	Alitretinoin	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	1.666910197958555	Aminocaproic Acid	rxcui:99	6-AMINOCAPROIC ACID	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.8468979231563628	Acrivastine	rxcui:19959	ACRIVASTINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	Acetophenazine	rxcui:16735	ACETOPHENAZINE	TRUE	FALSE	FALSE
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE BETA	hgnc:5960	IKBKB	TTD	2020.06.01	NULL	0.192335792	Arsenic trioxide	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	1.193356164447602	Ampiroxicam	ncit:C73073	AMPIROXICAM	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	ZINC 02849675	chembl:CHEMBL605959	CHEMBL:CHEMBL605959	FALSE	FALSE	FALSE
SYNAPTIC VESICLE GLYCOPROTEIN 2A	hgnc:20566	SV2A	TTD	2020.06.01	NULL	10.50153424713889	Brivaracetam	rxcui:1739745	BRIVARACETAM	TRUE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	1.790034246671403	Conivaptan	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
DKK1	hgnc:2891	DKK1	NCI	14-Sep-17	NULL	0.6141248097742047	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 2	hgnc:6930	MC2R	TTD	2020.06.01	NULL	13.12691780892362	Cosyntropin	rxcui:2890	COSYNTROPIN	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.007156559	Dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.2294915700860773	Metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	13.12691780892362	Live attenuated influenza vaccine	ncit:C96402	LIVE ATTENUATED INFLUENZA VACCINE	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C9	hgnc:60	ABCC9	TTD	2020.06.01	NULL	0.9546849315580819	Nicorandil	rxcui:31748	NICORANDIL	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.305277158	Nicergoline	rxcui:7398	NICERGOLINE	FALSE	FALSE	FALSE
INTERFERON ALPHA/BETA RECEPTOR 2	hgnc:5433	IFNAR2	TTD	2020.06.01	NULL	0.2187819634820604	Sifalimumab	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.1773907812016706	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.8078103267029922	Trimazosin	ncit:C75059	TRIMAZOSIN	FALSE	FALSE	FALSE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	5.250767123569449	REMD-477	ncit:C167005	VOLAGIDEMAB	FALSE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 1 ALPHA	hgnc:4910	HIF1A	TTD	2020.06.01	NULL	1.086365611772989	PX-478	drugbank:DB06082	PX-478	FALSE	FALSE	TRUE
OX40L RECEPTOR	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	7.001022831425932	PF-04518600	ncit:C121927	IVUXOLIMAB	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.1159109740302306	SAR-405838	drugbank:DB12541	SAR-405838	FALSE	FALSE	FALSE
AURORA KINASE C	hgnc:11391	AURKC	TTD	2020.06.01	NULL	0.2500365296937833	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.4150804050252529	Aplindore fumarate	ncit:C76649	APLINDORE FUMARATE	FALSE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	1.810609352954982	Lucatumumab	ncit:C48405	LUCATUMUMAB	FALSE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	2.917092846427472	SELODENOSON	ncit:C75135	SELODENOSON	FALSE	FALSE	FALSE
CAM-KINASE II	hgnc:1461	CAMK2B	TTD	2020.06.01	NULL	5.250767123569449	Rimacalib	ncit:C87325	RIMACALIB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	2.059124362184098	PRN1008	ncit:C174769	RILZABRUTINIB	FALSE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.2612321952024601	VX-680	ncit:C61319	TOZASERTIB LACTATE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.2108741816694558	IUPHAR.LIGAND:123	iuphar.ligand:123	LYSERGOL	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.020407179	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.020407179	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1035654265003836	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.079197091	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.053199262	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.026045472	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.032055965	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:7670	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.018942161	IUPHAR.LIGAND:85	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.013442824	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.018118589	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.024513385	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:165	iuphar.ligand:165	MK-212	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.020470827	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.047561296	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:3246	iuphar.ligand:275	RO 63-0563	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.040051618	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.037775303	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.041972559	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:2919	hgnc:4602	CXCL1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9480	iuphar.ligand:9480	WWL123	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.1539814405738841	IUPHAR.LIGAND:7741	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:8461	iuphar.ligand:8461	AH 11110	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:4450	iuphar.ligand:4450	(+)-ADRENALINE	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.013202834	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.098513454	IUPHAR.LIGAND:7302	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.032016873	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:4450	iuphar.ligand:4450	(+)-ADRENALINE	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.023609564	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.037775303	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.009443826	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.03849536	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:7241	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:520	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.025244073	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:524	iuphar.ligand:524	ARC-239	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:9061	iuphar.ligand:9061	PF-03882845	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:386	iuphar.ligand:386	DPCPX	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:476	iuphar.ligand:476	VUF8507	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:6898	ncit:C152517	TASOSARTAN	FALSE	FALSE	FALSE
NCBIGENE:969	hgnc:1694	CD69	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:4742	rxcui:33770	PIRETANIDE	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:6165	iuphar.ligand:6165	RHODEI-LITORIN	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:6163	iuphar.ligand:6163	NEUROMEDIN B (1-30) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2938	hgnc:4626	GSTA1	GuideToPharmacology	2024.1	antibody	5.250767123569449	IUPHAR.LIGAND:12586	iuphar.ligand:12586	OBRINDATAMAB	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:632	iuphar.ligand:632	[D-PHE6,&BETA;-ALA11,PHE13,NLE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9131	iuphar.ligand:9131	PLIXORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7513	iuphar.ligand:7513	CPI-203	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:12143	iuphar.ligand:12143	WNY0824	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:10564	iuphar.ligand:10564	ARV-771	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7509	iuphar.ligand:7509	MS436	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:11730	iuphar.ligand:11730	TAK-020	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:646	iuphar.ligand:646	[DES-ARG9]BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:939	hgnc:11922	CD27	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11227	iuphar.ligand:11227	INHIBITOR E4	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:671	iuphar.ligand:671	[TYR8]BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:12326	iuphar.ligand:12326	ACT-1014-6470	FALSE	FALSE	FALSE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:9385	iuphar.ligand:9385	P59 [PMID: 27108698]	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5760	iuphar.ligand:5760	WWGKKYRASKLGLAR	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:10595	iuphar.ligand:10595	JR14A	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.1172046232939609	IUPHAR.LIGAND:203	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1558	hgnc:2622	CYP2C8	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:9366	iuphar.ligand:9366	MELK-TI	FALSE	FALSE	FALSE
NCBIGENE:1593	hgnc:2605	CYP27A1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:8675	iuphar.ligand:8675	COMPOUND 3 [PMID: 14640538]	FALSE	FALSE	FALSE
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:6527	iuphar.ligand:6527	AC-DEVD-CHO	FALSE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	inhibitor	0.043611023	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	blocker	1.166837138570989	IUPHAR.LIGAND:2525	iuphar.ligand:2525	PB2+	FALSE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	0.4773424657790409	IUPHAR.LIGAND:12488	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
NCBIGENE:389	hgnc:669	RHOC	GuideToPharmacology	2024.1	activator	0.1483267549030918	IUPHAR.LIGAND:2377	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:2349	hgnc:2535	CTSH	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9550	iuphar.ligand:9550	COMPOUND 1E [PMID: 27285276]	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:740	rxcui:1976	CANNABINOL	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:3536	iuphar.ligand:3536	UCB35625	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:759	iuphar.ligand:759	CCL7	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:769	iuphar.ligand:769	CCL11	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:11598	iuphar.ligand:11598	BMS-741672	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:7679	iuphar.ligand:7679	AZD3778	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:9678	iuphar.ligand:9678	AZD2098	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:11724	iuphar.ligand:11724	MG-277	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	0.8975670296699916	IUPHAR.LIGAND:7331	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:9000	iuphar.ligand:9000	(R)-ARN2508	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.021951368	IUPHAR.LIGAND:5239	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:10240	iuphar.ligand:10240	SC-560	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:11391	iuphar.ligand:11391	SC-58125	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:921	iuphar.ligand:921	UROCORTIN 2	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:830	iuphar.ligand:830	CXCL7	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:769	iuphar.ligand:769	CCL11	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:808	iuphar.ligand:808	CCL20	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:8533	iuphar.ligand:8533	CXCL12&PHI;	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:9405	iuphar.ligand:9405	BS-181	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12881	iuphar.ligand:12881	TIBREMCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:11662	iuphar.ligand:11662	CP-10	FALSE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:8311	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
NCBIGENE:1883	hgnc:11910	TNFRSF25	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:5071	iuphar.ligand:5071	TL1A	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1161674142382621	IUPHAR.LIGAND:9004	iuphar.ligand:9004	ADL5859	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1161674142382621	IUPHAR.LIGAND:1611	iuphar.ligand:1611	SNC80	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1630	ncit:C170234	NORMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:2603	hgnc:2861	DHFR	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:8890	iuphar.ligand:8890	COMPOUND 9 [PMID: 15615544]	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	1.151484018326633	IUPHAR.LIGAND:6825	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
NCBIGENE:3211	hgnc:5111	HOXB1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12241	ncit:C179085	ERVOGASTAT	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11164	iuphar.ligand:11164	S416	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:9099	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.005618798	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.048394167	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.051731696	IUPHAR.LIGAND:940	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
NCBIGENE:2012	hgnc:3333	EMP1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8602	iuphar.ligand:8602	COMPOUND 10F [PMID: 24556381]	FALSE	FALSE	FALSE
NCBIGENE:2835	hgnc:4466	GPR12	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8240	iuphar.ligand:8240	GSK343	FALSE	FALSE	FALSE
NCBIGENE:1615	hgnc:2678	DARS1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:6507	iuphar.ligand:6507	KC-12615	FALSE	FALSE	FALSE
NCBIGENE:1823	hgnc:3035	DSC1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12282	ncit:C127114	VALEMETOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:10468	iuphar.ligand:10468	MOBOCERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9196	ncit:C101791	OLMUTINIB	FALSE	FALSE	TRUE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:2745	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:3059	rxcui:115264	IBANDRONATE	TRUE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1050	iuphar.ligand:1050	GW9508	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.076765601	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:11414	iuphar.ligand:11414	TASURGRATINIB	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.004972317	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:2609	hgnc:4145	GAPDHP67	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:6031	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.01823183	IUPHAR.LIGAND:7649	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
NCBIGENE:3177	hgnc:11004	SLC29A2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:11483	iuphar.ligand:11483	GPI-1046	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.039068208	IUPHAR.LIGAND:11887	iuphar.ligand:11887	TINENGOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:9712	iuphar.ligand:9712	COMPOUND 5E [PMID: 28580438]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.043180651	IUPHAR.LIGAND:5658	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:9366	iuphar.ligand:9366	MELK-TI	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.034184682	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.009092237	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:5832	iuphar.ligand:5832	AG-11/03	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1030	iuphar.ligand:1030	T-BOC-FLFLF	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:3424	iuphar.ligand:3424	AS604872	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:3386	iuphar.ligand:3386	AL12180	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.3889457128569962	IUPHAR.LIGAND:1048	iuphar.ligand:1048	WKYMVM	FALSE	FALSE	FALSE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:232	hgnc:4042	FZD4	GuideToPharmacology	2024.1	modulator	26.25383561784724	IUPHAR.LIGAND:10322	iuphar.ligand:10322	FZM1	FALSE	FALSE	FALSE
NCBIGENE:234	hgnc:4044	FZD6	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:3547	iuphar.ligand:3547	WNT-4	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4094	iuphar.ligand:4094	&ALPHA;3IA	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.051885051	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	inhibitor	0.045226246	IUPHAR.LIGAND:4083	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.2302968036653267	IUPHAR.LIGAND:4366	iuphar.ligand:4366	[3H]CGS8216	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6074	iuphar.ligand:6074	M1160	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3199	drugbank:DB08180	2-[METHYL-(5-GERANYL-4-METHYL-PENT-3-ENYL)-AMINO]-ETHYL-DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2977	hgnc:4684	GUCY1A2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:12843	iuphar.ligand:12843	LY3463251	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	modulator	0.5147810905460244	IUPHAR.LIGAND:9135	iuphar.ligand:9135	MK-0893	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	agonist	0.1403948428761885	IUPHAR.LIGAND:1136	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.014198938	IUPHAR.LIGAND:3447	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:452	hgnc:4581	GRIK3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:4085	iuphar.ligand:4085	[3H]KAINATE	FALSE	FALSE	FALSE
NCBIGENE:454	hgnc:772	ASS1P9	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:4085	iuphar.ligand:4085	[3H]KAINATE	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.6563458904461813	IUPHAR.LIGAND:4216	iuphar.ligand:4216	HOMOQUINOLINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:454	hgnc:772	ASS1P9	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:4317	iuphar.ligand:4317	SYM2081	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.1693795846312726	IUPHAR.LIGAND:4216	iuphar.ligand:4216	HOMOQUINOLINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	blocker	0.1346350544504987	IUPHAR.LIGAND:4089	iuphar.ligand:4089	[3H]DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:4276	iuphar.ligand:4276	NVP-AAM077	FALSE	FALSE	FALSE
NCBIGENE:936	hgnc:1647	CD24P2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4622	iuphar.ligand:4622	ALX 1393	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:9341	iuphar.ligand:9341	FERTIRELIN	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4602	iuphar.ligand:4602	[3H](R)-NPTS	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1172	iuphar.ligand:1172	[TRP8]GNRH	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:12784	iuphar.ligand:12784	BAY1214784	FALSE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:610	rxcui:3194	DEOXYCHOLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2234368988752957	PIRENZEPINE	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4896	iuphar.ligand:4896	C-TYPE NATRIURETIC PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:6480	iuphar.ligand:6480	G36	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4856	iuphar.ligand:4856	A-71915	FALSE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:722	rxcui:2567	CITRULLINE	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.2344092465879218	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
NCBIGENE:1441	hgnc:2439	CSF3R	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8873	iuphar.ligand:8873	COMPOUND 1 [PMID: 16821802]	FALSE	FALSE	FALSE
ORGANIC ANION TRANSPORTER M1	hgnc:23612	SLCO4C1	TTD	2020.06.01	NULL	1.029562181092049	Digoxin	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NCBIGENE:311	hgnc:535	ANXA11	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:1588	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:1597	iuphar.ligand:1597	IBC 293	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.3113103037689397	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.062733179	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.1881995384791917	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.2430910705356227	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.1835932560688619	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:9891	iuphar.ligand:9891	MARBOSTAT-100	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.1495945049449985	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.028078969	IUPHAR.LIGAND:5932	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1201	iuphar.ligand:1201	UR-PG153	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:8924	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:1217	iuphar.ligand:1217	A-349821	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1245	iuphar.ligand:1245	VUF 5207	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9103	iuphar.ligand:9103	GSK334429	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:1217	iuphar.ligand:1217	A-349821	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3010	iuphar.ligand:3010	COMPOUND 33 [PMID: 17574412]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3001	iuphar.ligand:3001	COMPOUND 42 [PMID: 17574411]	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:5526	iuphar.ligand:5526	ABNORMAL CANNABIDIOL	FALSE	FALSE	FALSE
NCBIGENE:114	hgnc:239	ADCY8	GuideToPharmacology	2024.1	modulator	0.3500511415712966	IUPHAR.LIGAND:5884	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	positive modulator	0.2778183663264258	NEBOGLAMINE	ncit:C66222	NEBOGLAMINE	FALSE	FALSE	FALSE
NCBIGENE:2039	hgnc:3382	DMTN	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9646	iuphar.ligand:9646	COMPOUND 47 [PMID: 28737909]	FALSE	FALSE	FALSE
NCBIGENE:2039	hgnc:3382	DMTN	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10134	iuphar.ligand:10134	IKK-BETA INHIBITOR R-28	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5635	iuphar.ligand:5635	AM3	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:5851	iuphar.ligand:5851	BAY-73-1449	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:1664	iuphar.ligand:1664	NALOXONE BENZOYLHYDRAZONE	FALSE	FALSE	FALSE
NCBIGENE:2757	hgnc:23177	KEAP1	GuideToPharmacology	2024.1	NULL	0.7001022831425933	IUPHAR.LIGAND:2717	ncit:C48382	BARDOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.003773458	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.017295017	IUPHAR.LIGAND:9039	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.018867291	IUPHAR.LIGAND:5660	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.016605842	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1285	iuphar.ligand:1285	KISSPEPTIN-14	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11715	iuphar.ligand:11715	OPNURASIB	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2311	iuphar.ligand:2311	APAMIN	FALSE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.1458546423213736	TERGURIDE	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	blocker	1.250182648468916	IUPHAR.LIGAND:2325	iuphar.ligand:2325	P05	FALSE	FALSE	FALSE
NCBIGENE:544	hgnc:881	ALDH7A1P4	GuideToPharmacology	2024.1	blocker	0.5834185692854945	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:544	hgnc:881	ALDH7A1P4	GuideToPharmacology	2024.1	blocker	0.2333674277141977	IUPHAR.LIGAND:2406	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:2596	iuphar.ligand:2596	XE991	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	activator	0.3125456621172291	IUPHAR.LIGAND:2593	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:12662	iuphar.ligand:12662	EXAMPLE 320 [WO2018198077A2]	FALSE	FALSE	FALSE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.31919557	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.300043836	IUPHAR.LIGAND:5689	iuphar.ligand:5689	JNJ-28312141	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9814	iuphar.ligand:9814	CCT241161	FALSE	FALSE	FALSE
NCBIGENE:1570	hgnc:6656	LNPEP	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8621	iuphar.ligand:8621	INHIBITOR 19 [PMID: 21476495]	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:2742	iuphar.ligand:2742	22R-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8690	iuphar.ligand:8690	GSK2033	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:10095	iuphar.ligand:10095	RO3306	FALSE	FALSE	FALSE
NCBIGENE:2591	hgnc:4125	GALNT3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10664	iuphar.ligand:10664	COMPOUND 12 [PMID: 31990537]	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:2905	iuphar.ligand:2905	AM966	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:12522	iuphar.ligand:12522	UCM-14216	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:9498	iuphar.ligand:9498	BMS-986020	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:2911	iuphar.ligand:2911	FARNESYL MONOPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10230	iuphar.ligand:10230	AS2717638	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1226814748497534	EC145	ncit:C62525	VINTAFOLIDE	FALSE	FALSE	TRUE
NCBIGENE:2666	hgnc:17582	KAT6B	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:12938	iuphar.ligand:12938	PF-9363	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7023	iuphar.ligand:7023	OG-L002	FALSE	FALSE	FALSE
NCBIGENE:2664	hgnc:4226	GDI1	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:12938	iuphar.ligand:12938	PF-9363	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1301	iuphar.ligand:1301	MCH (SALMON)	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.406619897	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NCBIGENE:2102	hgnc:16870	MELK	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11457	iuphar.ligand:11457	CC-401	FALSE	FALSE	FALSE
NCBIGENE:2094	ncbigene:2094	ERVT4	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:6009	iuphar.ligand:6009	MK2A INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:283	hgnc:483	ANG	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:6967	ncit:C169866	CORTICOTROPIN-ZINC HYDROXIDE	TRUE	FALSE	FALSE
NCBIGENE:283	hgnc:483	ANG	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:3767	iuphar.ligand:3767	[125I]ACTH-(1-24)	FALSE	FALSE	FALSE
NCBIGENE:281	hgnc:479	AMYP1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1301	iuphar.ligand:1301	MCH (SALMON)	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:10408	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
NCBIGENE:283	hgnc:483	ANG	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:6965	rxcui:2890	COSYNTROPIN	TRUE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	0.3750547945406749	IUPHAR.LIGAND:10408	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	0.8751278539282418	IUPHAR.LIGAND:9272	iuphar.ligand:9272	SETMELANOTIDE	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1341	iuphar.ligand:1341	PG-901	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	0.3500511415712967	IUPHAR.LIGAND:9272	iuphar.ligand:9272	SETMELANOTIDE	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:1339	iuphar.ligand:1339	MBP10	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:1320	iuphar.ligand:1320	&ALPHA;-MSH	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6221	iuphar.ligand:6221	MNI-137	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	0.5527123287967842	IUPHAR.LIGAND:1365	iuphar.ligand:1365	(1S,3R)-ACPD	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10563	iuphar.ligand:10563	MS432	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.072125922	IUPHAR.LIGAND:9658	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11406	ncit:C179135	ZALOGLANSTAT	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.072125922	IUPHAR.LIGAND:297	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.100976291	IUPHAR.LIGAND:342	iuphar.ligand:342	BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.027635616	IUPHAR.LIGAND:357	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:8593	iuphar.ligand:8593	[3H]ACETYLCHOLINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW805758X	chembl:CHEMBL359963	GW805758X	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:317	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:366	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:308	iuphar.ligand:308	P-F-HHSID	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:288	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.025244073	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:318	iuphar.ligand:318	[3H]QNB	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:321	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.035098711	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:339	iuphar.ligand:339	WIN 51,708	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:342	iuphar.ligand:342	BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:306	ncit:C152278	SABCOMELINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:321	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.1591141552596803	IUPHAR.LIGAND:342	iuphar.ligand:342	BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.048935388	IUPHAR.LIGAND:224	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:3274	iuphar.ligand:3274	VU0255035	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:5388	iuphar.ligand:5388	[3H]DIHYDROALPRENOLOL	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1349	iuphar.ligand:1349	GR 196429	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:1362	iuphar.ligand:1362	S26131	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.2885036881082115	IUPHAR.LIGAND:1607	iuphar.ligand:1607	DADLE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.2885036881082115	IUPHAR.LIGAND:11694	iuphar.ligand:11694	SRI22141	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:5192	iuphar.ligand:5192	G&OUML; 6983	FALSE	FALSE	FALSE
NCBIGENE:750	hgnc:1197	GAS8-AS1	GuideToPharmacology	2024.1	blocker	0.2917092846427472	IUPHAR.LIGAND:2406	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NCBIGENE:1553	hgnc:2608	CYP2A13	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:6740	iuphar.ligand:6740	GSK2606414	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:2574	iuphar.ligand:2574	JINGZHAOTOXIN-III	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8413	ncit:C174857	ELECLAZINE	FALSE	FALSE	FALSE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:2615	iuphar.ligand:2615	BC-III	FALSE	FALSE	FALSE
NCBIGENE:2245	hgnc:3663	FGD1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8057	iuphar.ligand:8057	XMD8-92	FALSE	FALSE	FALSE
NCBIGENE:1888	hgnc:3143	EBVS1	GuideToPharmacology	2024.1	NULL	13.12691780892362	IUPHAR.LIGAND:5034	iuphar.ligand:5034	NEUROTROPHIN-4	FALSE	FALSE	FALSE
NCBIGENE:467	hgnc:785	ATF3	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:4010	iuphar.ligand:4010	&ALPHA;-CONOTOXIN MII [H9A, L15A]	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:3964	iuphar.ligand:3964	&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CHLORMADINONE	rxcui:78904	CHLORMADINONE	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5758	ncit:C71635	CASOPITANT	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:7623	rxcui:1731071	FOSAPREPITANT	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1448487482363986	EMETINE	rxcui:3820	EMETINE	FALSE	FALSE	FALSE
NCBIGENE:2122	hgnc:3498	MECOM	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8205	iuphar.ligand:8205	COMPOUND 22 [PMID: 20462760]	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:2127	iuphar.ligand:2127	SENKTIDE	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:2128	iuphar.ligand:2128	GR138676	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.027121731	FLUPHENAZINE HYDROCHLORIDE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:2106	iuphar.ligand:2106	SCH 206272	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1472	iuphar.ligand:1472	NEUROMEDIN U-8	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:1681	iuphar.ligand:1681	NOCICEPTIN/ORPHANIN FQ	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:10381	iuphar.ligand:10381	NY0116	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1490	iuphar.ligand:1490	NEUROPEPTIDE S	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	NCI	14-Sep-17	NULL	0.2051080907644316	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:1579	iuphar.ligand:1579	NEUROTENSIN	FALSE	FALSE	FALSE
NCBIGENE:1763	hgnc:2939	DNA2	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:5024	iuphar.ligand:5024	MURAMYL DIPEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	NULL	0.084553416	IUPHAR.LIGAND:2953	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	NULL	1.050153425	IUPHAR.LIGAND:4687	iuphar.ligand:4687	[3H]ESTRADIOL-17&BETA;-GLUCURONIDE	FALSE	FALSE	FALSE
NCBIGENE:1227	hgnc:23612	SLCO4C1	GuideToPharmacology	2024.1	NULL	1.029562181092049	IUPHAR.LIGAND:4725	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:11453	iuphar.ligand:11453	MRS4625	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	modulator	1.693795846312725	IUPHAR.LIGAND:1729	iuphar.ligand:1729	2,2'-PYRIDYLISATOGEN TOSYLATE	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1753	iuphar.ligand:1753	MRS2578	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10270	iuphar.ligand:10270	P4PAL-10	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10269	iuphar.ligand:10269	BMS-986120	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:3740	iuphar.ligand:3740	SLIGKV-NH2	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	0.7573221812840553	dicumarol	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
NCBIGENE:2139	hgnc:3520	EYA2	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:5704	iuphar.ligand:5704	PP-242	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:6742	iuphar.ligand:6742	MRL20	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:8700	iuphar.ligand:8700	TIROTUNDIN	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2717	ncit:C48382	BARDOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	modulator	0.1966579447029756	IUPHAR.LIGAND:8968	iuphar.ligand:8968	PIK-108	FALSE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:8839	iuphar.ligand:8839	TORIN 2	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:8827	iuphar.ligand:8827	COMPOUND 11J [PMID: 23021994]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.036873365	IUPHAR.LIGAND:9916	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.2949869170544634	IUPHAR.LIGAND:8978	iuphar.ligand:8978	QUINOSTATIN	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.098328972	IUPHAR.LIGAND:9728	ncit:C107686	DEZAPELISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:9563	ncit:C125471	EGANELISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	modulator	0.1389091831632129	IUPHAR.LIGAND:8968	iuphar.ligand:8968	PIK-108	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:8915	iuphar.ligand:8915	AZD8835	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:12062	iuphar.ligand:12062	COMPOUND 27 [PMID: 35834807]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:8915	iuphar.ligand:8915	AZD8835	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:9800	iuphar.ligand:9800	SELETALISIB	FALSE	FALSE	FALSE
NCBIGENE:1299	hgnc:2219	COL9A3	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:2347	iuphar.ligand:2347	CYCLIC GMP	FALSE	FALSE	FALSE
NCBIGENE:1312	hgnc:2228	COMT	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8811	iuphar.ligand:8811	COMPOUND 53 [PMID: 19631533]	FALSE	FALSE	FALSE
NCBIGENE:2387	hgnc:3899	FRA3D	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8658	iuphar.ligand:8658	PEPTIDE 18 [PMID: 24350995]	FALSE	FALSE	FALSE
NCBIGENE:1162	hgnc:18762	SLC36A2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4671	rxcui:94	5-HYDROXYTRYPTOPHAN	TRUE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:4449	iuphar.ligand:4449	PTH-(1-34) (RAT)	FALSE	FALSE	FALSE
NCBIGENE:1213	hgnc:2092	CLTC	GuideToPharmacology	2024.1	NULL	0.3125456621172291	IUPHAR.LIGAND:4562	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:3624	iuphar.ligand:3624	TIP39	FALSE	FALSE	FALSE
NCBIGENE:598	hgnc:992	BCL2L1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:2718	rxcui:2438	CHOLESTEROL	TRUE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:11308	ncit:C177073	ECLITASERTIB	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12059	iuphar.ligand:12059	COMPOUND 23 [PMID: 35816678]	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8209	iuphar.ligand:8209	COMPOUND 35 [PMID: 20684608]	FALSE	FALSE	FALSE
NCBIGENE:1528	hgnc:2570	CYB5A	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:8038	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
NCBIGENE:2631	hgnc:4179	NIPSNAP2	GuideToPharmacology	2024.1	inhibitor	0.3860858179095184	IUPHAR.LIGAND:4802	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
NCBIGENE:1860	hgnc:9675	PTPRM	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8856	iuphar.ligand:8856	COMPOUND 8A [PMID: 23713581]	FALSE	FALSE	FALSE
ATP-CITRATE SYNTHASE	hgnc:115	ACLY	TTD	2020.06.01	NULL	39.38075342677087	ETC-1002	rxcui:2282403	BEMPEDOIC ACID	TRUE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.201952582	IUPHAR.LIGAND:1990	iuphar.ligand:1990	RELAXIN-3	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:1990	iuphar.ligand:1990	RELAXIN-3	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:2924	iuphar.ligand:2924	FINGOLIMOD-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	blocker	0.596678082	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:2924	iuphar.ligand:2924	FINGOLIMOD-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:11496	iuphar.ligand:11496	S1P D20:1	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:2937	iuphar.ligand:2937	AFD(R)	FALSE	FALSE	FALSE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	agonist	0.7292732116068681	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:2937	iuphar.ligand:2937	AFD(R)	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.3431873936973497	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:9569	iuphar.ligand:9569	ASP4058	FALSE	FALSE	FALSE
NCBIGENE:252	hgnc:10608	SCTR	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:3755	iuphar.ligand:3755	[(CH2NH)4,5]SECRETIN	FALSE	FALSE	FALSE
NCBIGENE:2213	hgnc:3618	FCGR2B	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:11893	iuphar.ligand:11893	COMPOUND 6 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:2225	hgnc:11408	STK4	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11812	iuphar.ligand:11812	XMU-MP-1	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1017590527823536	IUPHAR.LIGAND:7321	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.061055432	IUPHAR.LIGAND:357	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:9099	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
NCBIGENE:2522	ncbigene:2522	FUSE	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9851	iuphar.ligand:9851	LX2931	FALSE	FALSE	FALSE
NCBIGENE:1115	hgnc:11002	SLC28A2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8485	iuphar.ligand:8485	COMPOUND 48 [PMID: 25815140]	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10218	iuphar.ligand:10218	COMPOUND 27D [PMID: 28231433]	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3085	iuphar.ligand:3085	COMPOUND 3A [PMID: 12238936]	FALSE	FALSE	FALSE
NCBIGENE:3048	hgnc:4832	HBG2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12696	iuphar.ligand:12696	SLB1122168	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2036	iuphar.ligand:2036	BIM 23056	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.1151484018326633	IUPHAR.LIGAND:2007	iuphar.ligand:2007	CORTISTATIN-14	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2013	iuphar.ligand:2013	KE 108	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2079	iuphar.ligand:2079	H-C[CYS-PHE-LAGL(N&BETA;ME,BENZOYL)-DTRP-LYS-THR-PHE-CYS]-OH	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2019	iuphar.ligand:2019	SRIF-14	FALSE	FALSE	FALSE
NCBIGENE:2633	hgnc:4182	GBP1	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:6818	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10672	iuphar.ligand:10672	COMPOUND 5 [TOMASSI ET AL., 2020]	FALSE	FALSE	FALSE
NCBIGENE:2716	hgnc:4295	GK4P	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12664	iuphar.ligand:12664	EXAMPLE 203 [WO2017058503A1]	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:10294	iuphar.ligand:10294	COMPOUND 130 [PMID: 29157600]	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.3454452054979901	minocycline	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
NCBIGENE:2239	hgnc:4452	GPC4	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8118	iuphar.ligand:8118	COMPOUND 30 [PMID: 22902653]	FALSE	FALSE	FALSE
NCBIGENE:2258	hgnc:3670	FGF13	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:1759	hgnc:2972	DNM1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7198	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
SRP19	hgnc:11300	SRP19	PharmGKB	4/5/24	NULL	0.750109589	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:1754	hgnc:11850	TLR4	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:9137	iuphar.ligand:9137	NEOCEPTIN-3	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.1593072549626653	IUPHAR.LIGAND:2635	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.3241214273808302	IUPHAR.LIGAND:7797	ncit:C116891	GALUNISERTIB	FALSE	FALSE	FALSE
NCBIGENE:2423	hgnc:3933	FRA8E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8582	iuphar.ligand:8582	PEPTIDE 4 [PMID: 18294843]	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:2499	rxcui:10553	THYMOL	TRUE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	0.729273212	IUPHAR.LIGAND:2441	iuphar.ligand:2441	SKF96365	FALSE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.1491695205559502	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.3281729452230906	IUPHAR.LIGAND:2525	iuphar.ligand:2525	PB2+	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:10292	iuphar.ligand:10292	AM12	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.07458476	IUPHAR.LIGAND:1056	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.027811267	IUPHAR.LIGAND:2377	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	1.544343271638073	IUPHAR.LIGAND:12528	iuphar.ligand:12528	AM-0883	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.028290771	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:6387	iuphar.ligand:6387	SF-51	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:11846	iuphar.ligand:11846	ML1-SA1	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.3947945205691315	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:10698	iuphar.ligand:10698	KPR-5714	FALSE	FALSE	FALSE
NCBIGENE:498	hgnc:823	ATP5F1A	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.1241316104862754	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:2271	hgnc:3700	FH	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11339	iuphar.ligand:11339	SBI-0206965	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2220	iuphar.ligand:2220	D(CH2)5[TYR(ME)2,THR4,TYR(3125I)-NH29]OVT	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:1520	iuphar.ligand:1520	[125I]PYY (PIG)	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.2453629496995069	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
UNIPROT:P43088	hgnc:9600	PTGFR	TEND	1-Aug-11	NULL	15.00219178	TRAVOPROST	rxcui:283809	TRAVOPROST	TRUE	FALSE	FALSE
MDM4	hgnc:6974	MDM4	CIViC	10-Apr-24	NULL	0.2500365296937833	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MDM2	hgnc:6973	MDM2	CIViC	10-Apr-24	NULL	0.150021918	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
AKT3	hgnc:393	AKT3	CIViC	10-Apr-24	NULL	0.045579576	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
AREG	hgnc:651	AREG	CIViC	10-Apr-24	NULL	0.2917092846427472	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
ERCC1	hgnc:3433	ERCC1	CIViC	10-Apr-24	NULL	0.040515178	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.2592971419046642	ALECTINIB	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	9.845188356692718	ARRY-520	ncit:C68937	FILANESIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.6783936852156912	INFIGRATINIB	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.1124502911321247	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.026885648	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	CIViC	10-Apr-24	NULL	0.076765601	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.054695491	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	0.1389091831632129	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.077217164	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
RAD50	hgnc:9816	RAD50	CIViC	10-Apr-24	NULL	26.25383561784724	CHECKPOINT KINASE INHIBITOR AZD7762	ncit:C66961	CHECKPOINT KINASE INHIBITOR AZD7762	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.3547815624033412	IPATASERTIB	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.2332563532602643	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	CIViC	10-Apr-24	NULL	1.325951293830669	DURVALUMAB	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.7192831676122533	ELIMUSERTIB	ncit:C146807	ELIMUSERTIB	FALSE	FALSE	TRUE
ATXN1L	hgnc:33279	ATXN1L	CIViC	10-Apr-24	NULL	0.3500511415712966	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
PTPN12	hgnc:9645	PTPN12	CIViC	10-Apr-24	NULL	0.3571950424196904	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	CIViC	10-Apr-24	NULL	0.2386712328895204	GW-2580	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.4145342465975881	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.6134073742487676	ELACESTRANT	rxcui:2628469	ELACESTRANT	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.015627283	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.003574869	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	CIViC	10-Apr-24	NULL	2.187819634820604	VORASIDENIB	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.048394167	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
STAG2	hgnc:11355	STAG2	CIViC	10-Apr-24	NULL	1.458546423213736	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
VPS37A	hgnc:24928	VPS37A	CIViC	10-Apr-24	NULL	1.458546423213736	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.00459626	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.024256701	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DoCM	10-Apr-24	NULL	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	DoCM	10-Apr-24	NULL	0.1660584163051692	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.057073556	Navitoclax	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.043406727	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.024256701	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	YM-254890	iuphar.ligand:9335	YM-254890	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.068727318	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.01683118	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.082472782	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.5250767123569451	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.4735986033023426	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.1902451856365742	Dinaciclib	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.066591847	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.3316273972780705	SU5402	drugbank:DB08577	3-[(3-(2-CARBOXYETHYL)-4-METHYLPYRROL-2-YL)METHYLENE]-2-INDOLINONE	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.063415062	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	1.897867635025102	PLX9486	ncit:C121647	BEZUCLASTINIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.253049018	Toripalimab-tpzi	rxcui:2669407	TORIPALIMAB-TPZI	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.072299719	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.070291394	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.010939098	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.2500365296937833	GDC0879	iuphar.ligand:5681	GDC-0879	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.3125456621172291	AZD0364	ncit:C176765	TIZATERKIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.069454592	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.1389091831632129	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.9845188356692718	SAR405838	ncit:C106120	P53-HDM2 INTERACTION INHIBITOR MI-773	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.150021918	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.079557078	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1209854175937661	Refametinib	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1058622403945453	Obatoclax	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.048394167	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.095500063	Gedatolisib	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2278978786271462	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.016574391	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	Nab-paclitaxel	ncit:C2688	NAB-PACLITAXEL	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.7095631248066824	UMI-77	iuphar.ligand:8105	UMI-77	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2365210416022274	PKI-179	drugbank:DB13109	PKI-179	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1637453364938497	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.028382525	Topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.008548953	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CancerCommons	25-Jul-13	inhibitor	0.5000730593875667	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1389091831632129	Gedatolisib	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CancerCommons	25-Jul-13	inhibitor	0.1250182648468916	RO4987655	ncit:C82696	MEK INHIBITOR RO4987655	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	HARMAN	chembl:CHEMBL12014	HARMAN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.133607306	HYDROCORTISONE VALERATE	rxcui:27199	HYDROCORTISONE VALERATE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.005571697	FLUFENAMIC ACID	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009974862	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.2546668357992238	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.020936073	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.2169738480813822	6beta-hydroxytestosterone	chembl:CHEMBL2074878	6BETA-HYDROXYTESTOSTERONE	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.089501712	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	0.192335792	Psoralen	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	1.184383561707394	KD3010	drugbank:DB05188	KD3010	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.1615620653405984	Prazosin	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4094	iuphar.ligand:4094	&ALPHA;3IA	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:1576	iuphar.ligand:1576	LARGE NEUROMEDIN N	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:8865	iuphar.ligand:8865	PWT2-N/OFQ	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.079798892	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:10601	iuphar.ligand:10601	AZD7648	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:6023	drugbank:DB04769	5-QUINOXALIN-6-YLMETHYLENE-THIAZOLIDINE-2,4-DIONE	FALSE	FALSE	FALSE
NCBIGENE:1171	hgnc:14679	SLC38A4	GuideToPharmacology	2024.1	NULL	2.187819634820604	IUPHAR.LIGAND:4635	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.096167896	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2059	iuphar.ligand:2059	[111IN,90Y]DOTA-TOC	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.022632617	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1422972120208522	ACTH	iuphar.ligand:1331	ACTH	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.069454592	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	NCI	14-Sep-17	NULL	0.2625383561784725	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
IL12A	hgnc:5969	IL12A	ChEMBL	33	inhibitor	3.500511415712966	BRIAKINUMAB	ncit:C95321	BRIAKINUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	1.336059069138614	trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.051277023	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.1801292323694494	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	ORTHOTOLIDINE	chembl:CHEMBL85109	ORTHOTOLIDINE	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.3088686543276147	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	0.1682938180631233	4SC-202	drugbank:DB13101	4SC-202	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.2540693769469088	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.036847489	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PRKCZ	hgnc:9412	PRKCZ	ChEMBL	33	inhibitor	0.2573905452730122	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	CHINOMETHIONAT	chembl:CHEMBL1595865	CHINOMETHIONAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.006026014	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00239313	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.032817295	Chloroquine	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.014299475	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
UNIPROT:Q06432	hgnc:1405	CACNG1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461813	NITRENDIPINE	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.167488584	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.080225625	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	4.118248724368196	MM-121	chembl:CHEMBL2109402	MM-121	FALSE	TRUE	TRUE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:7977	drugbank:DB07404	BPH-608	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	NULL	1.544343271638073	IUPHAR.LIGAND:3413	iuphar.ligand:3413	[3H]LTB4	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:1634	iuphar.ligand:1634	BNTX	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	TCMDC-123748	chembl:CHEMBL530609	CHEMBL:CHEMBL530609	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.020721259	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004579424	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.1182605208011137	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.2639729920045843	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:2024	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2886	ncit:C87423	ALMOREXANT	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	VENLAFAXINE HYDROCHLORIDE	rxcui:235988	VENLAFAXINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	0.2692701089009974	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	ChEMBL	33	inhibitor	3.500511415712966	QUAVONLIMAB	ncit:C150679	QUAVONLIMAB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004051518	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.005716987	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.1810609352954982	IPI-504	ncit:C48401	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	TRUE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	0.3281729452230906	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6345	iuphar.ligand:6345	COMPOUND 23C [PMID: 17929793]	FALSE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	ChEMBL	33	inhibitor	2.917092846427472	EMICERFONT	ncit:C174801	EMICERFONT	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.069332312	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
TPO	hgnc:12015	TPO	ChEMBL	33	inhibitor	8.751278539282415	CARBIMAZOLE	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.014464923	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	CAS 902561-11-9	chembl:CHEMBL494081	CHEMBL:CHEMBL494081	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001439355	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UNIPROT:P09884	hgnc:9173	POLA1	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	NELARABINE	rxcui:274771	NELARABINE	TRUE	FALSE	TRUE
UNIPROT:P08887	hgnc:6019	IL6R	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	SIRUKUMAB	ncit:C152371	SIRUKUMAB	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:12534	iuphar.ligand:12534	DS88790512	FALSE	FALSE	FALSE
NCBIGENE:1888	hgnc:3143	EBVS1	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:5033	iuphar.ligand:5033	NEUROTROPHIN-3	FALSE	FALSE	FALSE
IL18	hgnc:5986	IL18	ChEMBL	33	inhibitor	8.290684931951763	GSK-1070806	chembl:CHEMBL2109606	GSK-1070806	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	1.458546423213736	ARDEPARIN SODIUM	rxcui:87865	ARDEPARIN SODIUM	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	2-METHOXY-1,4-NAPHTHOQUINONE	chembl:CHEMBL106562	2-METHOXY-1,4-NAPHTHOQUINONE	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.040005845	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1512704997187101	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.090821275	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
UGT1A5	hgnc:12537	UGT1A5	NCI	14-Sep-17	NULL	0.3684748858645228	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.007529925	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.061412481	loratadine	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	1.419126249613364	CIFORADENANT	ncit:C125659	CIFORADENANT	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	PEG-SN38	ncit:C70651	FIRTECAN PEGOL	FALSE	FALSE	FALSE
NCBIGENE:80	hgnc:153	ACTG1P8	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:844	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.1810609352954982	CNF1010	chembl:CHEMBL109480	TANESPIMYCIN	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.2692701089009974	NIC5-15	chembl:CHEMBL493737	METHYLINOSITOL	FALSE	FALSE	FALSE
UNIPROT:Q09428	hgnc:59	ABCC8	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	DIAZOXIDE CHOLINE	chembl:CHEMBL4297276	DIAZOXIDE CHOLINE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Hyoscyamine	rxcui:153970	HYOSCYAMINE	TRUE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	3.938075342677087	NBI-98854	rxcui:1918219	VALBENAZINE	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA-2/DELTA-1	hgnc:1399	CACNA2D1	TTD	2020.06.01	NULL	0.192335792	Imagabalin	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:5260	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.105015342	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.051177067	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	SODIUM NITRITE	rxcui:9894	SODIUM NITRITE	TRUE	FALSE	FALSE
CRABP2	hgnc:2339	CRABP2	NCI	14-Sep-17	NULL	0.6775183385250904	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.1785975212098452	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	COAGULATION FACTOR VIIA	rxcui:2386863	COAGULATION FACTOR VIIA (RECOMBINANT)-JNCW	TRUE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.1256164383629055	IUPHAR.LIGAND:7382	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:7502	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.05676505	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:463	hgnc:777	ZFHX3	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:3979	iuphar.ligand:3979	[3H]CYTISINE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.040515178	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008995661	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.004836742	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006489639	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	VINDESINE SULFATE	rxcui:11205	VINDESINE SULFATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	HYDROCORTISONE VALERATE	rxcui:27199	HYDROCORTISONE VALERATE	TRUE	FALSE	FALSE
UNIPROT:P05093	hgnc:2593	CYP17A1	TdgClinicalTrial	Jan-14	NULL	3.125456621172291	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.347732922	thioureidobutyronitrile	ncit:C102881	THIOUREIDOBUTYRONITRILE	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3882	iuphar.ligand:3882	GR94800	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.003929186	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	FDA	10-Apr-24	NULL	0.084598826	Carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
ARAF	hgnc:646	ARAF	MyCancerGenome	20-Jun-17	inhibitor	0.6364566210387211	XL281	drugbank:DB05190	XL281	FALSE	FALSE	TRUE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.057073556	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
STRYCHNINE-BINDING GLYCINE RECEPTOR	hgnc:4326	GLRA1	TTD	2020.06.01	NULL	0.7955707762984014	D-Serine	ncit:C61739	D-SERINE	FALSE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	ChEMBL	33	blocker	0.1312691780892362	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.2210849315187136	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.06466462	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1962903597596056	CHLOROTRIANISENE	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.064111931	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	CIViC	10-Apr-24	NULL	0.027519744	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BCAR1	hgnc:971	BCAR1	PharmGKB	4/5/24	NULL	1.567393171214761	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
BOMBESIN RECEPTOR	hgnc:1058	BLM	TTD	2020.06.01	NULL	0.5097832158805291	BAY-86-7548	chembl:CHEMBL4297341	RM-2 GA-68	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.1172046232939609	AVIPTADIL	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.2778183663264259	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.6105543166941221	ORCIPRENALINE	rxcui:7688	METAPROTERENOL	TRUE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.100589408	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CNR1	hgnc:2159	CNR1	ChEMBL	33	agonist	0.6177373086552295	DRONABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	blocker	0.1442518440541058	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.00453826	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
PIP4K2A	hgnc:8997	PIP4K2A	DTC	9/2/20	NULL	1.166837138570989	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.020399251	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.212152207	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.03849536	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.8899605294185507	MLN8054	drugbank:DB13061	MLN8054	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.045579576	IUPHAR.LIGAND:7397	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.093763699	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1391	hgnc:6719	LTC4S	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10479	iuphar.ligand:10479	AZD9898	FALSE	FALSE	FALSE
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	0.2187819634820604	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.08178765	POLYESTRADIOL PHOSPHATE	rxcui:34120	POLYESTRADIOL PHOSPHATE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.065389379	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	SPECTINOMYCIN HYDROCHLORIDE	rxcui:267342	SPECTINOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	BISPHENOL A	rxcui:1433347	BISPHENOL A	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004427291	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
FGB	hgnc:3662	FGB	ChEMBL	33	inhibitor	0.8751278539282416	FIBRINOLYSIN, HUMAN	rxcui:4388	PLASMIN	TRUE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	PharmGKB	4/5/24	NULL	0.463302981	pitolisant	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8166	iuphar.ligand:8166	COMPOUND 72 [WO2013026806]	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1215455352678113	SJ000111875	chembl:CHEMBL590949	CHEMBL:CHEMBL590949	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	modulator	1.944728564284981	OZANIMOD HYDROCHLORIDE	rxcui:2288235	OZANIMOD HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	DTC	9/2/20	NULL	3.281729452230906	LORNEIC ACID A	chembl:CHEMBL1079947	LORNEIC ACID A	FALSE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.1363835616511545	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
MIR4278	hgnc:38243	MIR4278	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
SOST	hgnc:13771	SOST	ChEMBL	33	inhibitor	6.563458904461812	SETRUSUMAB	ncit:C152352	SETRUSUMAB	FALSE	FALSE	FALSE
AMACR	hgnc:451	AMACR	PharmGKB	4/5/24	NULL	1.346350544504987	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:Q01668	hgnc:1391	CACNA1D	TdgClinicalTrial	Jan-14	NULL	0.1221108633388244	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:6160	iuphar.ligand:6160	12-EPI LTB4	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.546954909	I-CBP112	iuphar.ligand:8236	I-CBP112	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.058645947	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	BEZAFIBRATE	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2599	ncit:C82306	LINOPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:4093	iuphar.ligand:4093	&ALPHA;&BETA;-MEATP	FALSE	FALSE	FALSE
TIGIT	hgnc:26838	TIGIT	ChEMBL	33	inhibitor	6.563458904461812	ETIGILIMAB	ncit:C142821	ETIGILIMAB	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:2003	iuphar.ligand:2003	BIM 23050	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	MEPREDNISONE	rxcui:29523	MEPREDNISONE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	FDA	10-Apr-24	NULL	1.029066006546944	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	0.077789143	Ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1164249916534246	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.1232574442152452	PIMECROLIMUS	rxcui:321952	PIMECROLIMUS	TRUE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.3182283105193605	Semaglutide	rxcui:1991302	SEMAGLUTIDE	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.053361455	IUPHAR.LIGAND:4192	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:7679	iuphar.ligand:7679	AZD3778	FALSE	FALSE	FALSE
SLC16A1	hgnc:10922	SLC16A1	NCI	14-Sep-17	NULL	1.207072901969988	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	0.2386712328895204	EVANS BLUE	rxcui:4191	EVANS BLUE	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.069089041	Quazepam	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.082559232	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
NEUROPEPTIDE Y RECEPTOR TYPE 1	hgnc:7956	NPY1R	TTD	2020.06.01	NULL	2.625383561784724	NEUROPEPTIDE-Y	chembl:CHEMBL267633	NEUROPEPTIDE-Y	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.086361301	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
KCNMA1	hgnc:6284	KCNMA1	ChEMBL	33	potentiator	0.729273212	FLINDOKALNER	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.189216833	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.028413242	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.078840347	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.1187956362798518	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.8607814956671229	NOMEGESTROL	rxcui:31930	NOMEGESTROL	TRUE	FALSE	FALSE
CCHCR1	hgnc:13930	CCHCR1	PharmGKB	4/5/24	NULL	4.773424657790409	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:3902	rxcui:28656	NAFARELIN	TRUE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	2.051080907644316	IUPHAR.LIGAND:7299	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:9151	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
NCBIGENE:3096	hgnc:4920	HIVEP1	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:12069	iuphar.ligand:12069	SOS1 PROTAC 9D	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1808115400678185	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.049864835	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1067229090156392	IUPHAR.LIGAND:277	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:10441	iuphar.ligand:10441	COMPOUND 5D [PMID: 31335136]	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.036062961	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.012738397	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.091796628	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.065092154	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.060492709	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BCL2L10	hgnc:993	BCL2L10	ChEMBL	33	inhibitor	8.751278539282415	OBATOCLAX MESYLATE	ncit:C62771	OBATOCLAX MESYLATE	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.4070362111294147	APINOCALTAMIDE	ncit:C190345	APINOCALTAMIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TCMDC-124685	chembl:CHEMBL587579	CHEMBL:CHEMBL587579	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	CYCLOSERINE	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.028977744	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	NULL	2.763561643983921	IUPHAR.LIGAND:4073	iuphar.ligand:4073	[125I]PSALMOTOXIN 1	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.064111931	IBUTILIDE FUMARATE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.1097721349875146	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.064268875	IUPHAR.LIGAND:6322	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	DESERPIDINE	rxcui:62174	DESERPIDINE	TRUE	FALSE	FALSE
IRON	hgnc:4650	GTF2E1	TTD	2020.06.01	NULL	10.50153424713889	SPD602	chembl:CHEMBL487465	DEFERITAZOLE	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:9613	iuphar.ligand:9613	AM841	FALSE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8082	iuphar.ligand:8082	ND-2110	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3063	iuphar.ligand:3063	COMPOUND 6 [PMID: 7629799]	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	HQP1351	ncit:C165549	OLVEREMBATINIB	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.03729238	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.004585823	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.071341945	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.5114383561918295	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.2218633995874415	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
UGT2B17	hgnc:12547	UGT2B17	PharmGKB	4/5/24	NULL	0.6731752722524935	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.021878196	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RAC2	hgnc:9802	RAC2	PharmGKB	4/5/24	NULL	1.640864726115453	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004101201	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
AKT3	hgnc:393	AKT3	CIViC	10-Apr-24	NULL	0.3076621361466474	AKT INHIBITOR MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
SLC1A1	hgnc:10939	SLC1A1	PharmGKB	4/5/24	NULL	0.1546617709446082	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	inhibitor	0.1579178082276526	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.1141471113819445	6-AZAURIDINE	ncit:C291	6-AZAURIDINE	FALSE	FALSE	FALSE
ATM SERINE/THREONINE KINASE	hgnc:795	ATM	TTD	2020.06.01	NULL	0.2397610558707511	AZD0156	iuphar.ligand:9942	AZD0156	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.022583945	IUPHAR.LIGAND:59	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.3860858179095183	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.3241214273808302	SUN-K0706	ncit:C174748	VODOBATINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:5971	iuphar.ligand:5971	FLT-3 INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9000	iuphar.ligand:9000	(R)-ARN2508	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:11410	ncit:C175770	DEURUXOLITINIB	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	2.500365296937833	Mivacurium	rxcui:30077	MIVACURIUM	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.047415271	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.1539814405738841	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.096167896	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.8751278539282416	Exatecan	ncit:C66720	EXATECAN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	NSC-37031	chembl:CHEMBL222993	CHEMBL:CHEMBL222993	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.049302978	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.1001290450718812	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P50391	hgnc:9329	NPY4R	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	TM30339	drugbank:DB05085	TM30339	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	3.214755381777214	COAGULATION FACTOR IX	wikidata:Q20801778	COAGULATION FACTOR IX	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.068727318	Obatoclax	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	0.351221881	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	QUISQUALATE	drugbank:DB02999	QUISQUALIC ACID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	TCMDC-125575	chembl:CHEMBL587620	CHEMBL:CHEMBL587620	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.018423744	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.019949723	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008279355	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.596678082	JATRORRHIZINE	chembl:CHEMBL251055	JATRORRHIZINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-125733	chembl:CHEMBL530788	CHEMBL:CHEMBL530788	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
BCL2L2	hgnc:995	BCL2L2	ChEMBL	33	inhibitor	1.093909817410302	OBATOCLAX MESYLATE	ncit:C62771	OBATOCLAX MESYLATE	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.032252869	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.072826174	FLUORESCEIN	rxcui:25138	FLUORESCEIN	TRUE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.2263261691193728	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1293292394967844	STILONIUM IODIDE	ncit:C73168	STILONIUM IODIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004616194	FLUFENAMIC ACID	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.3547815624033412	OPC-14523	drugbank:DB05422	OPC-14523	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.086551106	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.096758608	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.030527716	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:10190	ncit:C125659	CIFORADENANT	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:7713	iuphar.ligand:7713	AZD7762	FALSE	FALSE	TRUE
CA7	hgnc:1381	CA7	ChEMBL	33	inhibitor	1.166837138570988	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.08334551	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	ChEMBL	33	positive modulator	2.763561643983921	VONICOG ALFA	rxcui:1812589	VONICOG ALFA	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	PharmGKB	4/5/24	NULL	0.037318885	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.1458546423213736	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TOB1	hgnc:11979	TOB1	NCI	14-Sep-17	NULL	13.12691780892362	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.00740849	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.067317527	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:11597	iuphar.ligand:11597	BMS-753426	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2822	iuphar.ligand:2822	R,R-THC	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.1521961485092594	IUPHAR.LIGAND:4216	iuphar.ligand:4216	HOMOQUINOLINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:6479	iuphar.ligand:6479	CXCL17	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2237	iuphar.ligand:2237	D(CH2)5[D-ILE2,VAL4,TYR-NH29]AVP	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.9883796938483671	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.055681518	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.026927011	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
RGS12	hgnc:9994	RGS12	DTC	9/2/20	NULL	1.009762908	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
NCBIGENE:1638	hgnc:2709	DCT	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8578	iuphar.ligand:8578	COMPOUND 29E [PMID: 23631440]	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:9383	iuphar.ligand:9383	OSI-930	FALSE	FALSE	FALSE
VEGFC	hgnc:12682	VEGFC	CIViC	10-Apr-24	NULL	0.1190650141398968	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	0.1063985232739503	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.1875273972703375	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.2408608772279564	OXYCODEGOL	ncit:C170277	OXYCODEGOL	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.187193124	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.561579372	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	0.145450613	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.014849455	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.073437302	BCP9000383	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
UNIPROT:P42336	hgnc:8975	PIK3CA	TdgClinicalTrial	Jan-14	NULL	0.1350505947420126	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:424	iuphar.ligand:424	[3H]CGS 21680	FALSE	FALSE	FALSE
NCBIGENE:1989	hgnc:1974	CHUK	GuideToPharmacology	2024.1	inhibitor	0.091476779	IUPHAR.LIGAND:9693	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:925	iuphar.ligand:925	ASTRESSIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	PharmGKB	4/5/24	NULL	0.2778183663264259	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.087512785	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.525076712	Nalidixic Acid	rxcui:7240	NALIDIXIC ACID	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	CID 1540951	chembl:CHEMBL259421	CHEMBL:CHEMBL259421	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.085796848	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
PSMD3	hgnc:9560	PSMD3	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.038894571	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004287741	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.016086909	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.364636606	AR42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.039778539	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.591141552596803	NAFARELIN	rxcui:28656	NAFARELIN	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:11757	drugbank:DB15435	BMS-986158	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.561579372	MEDI4736	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.2103110997424346	MILNACIPRAN	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.096167896	IUPHAR.LIGAND:5501	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:2347	hgnc:2531	CTSF	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:10746	iuphar.ligand:10746	VBY-825	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003541833	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.6977763619361395	ACY-1215	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.098884503	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8024	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:45	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4241	iuphar.ligand:4241	L838417	FALSE	FALSE	FALSE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12209	iuphar.ligand:12209	VIPOGLANSTAT	FALSE	FALSE	FALSE
NCBIGENE:2632	hgnc:4180	GBE1	GuideToPharmacology	2024.1	activator	1.500219178162699	IUPHAR.LIGAND:6846	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	ACROLEIN	iuphar.ligand:2418	ACROLEIN	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	CIViC	10-Apr-24	NULL	0.045461187	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.01763778	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.9723642821424906	ASP-4058	drugbank:DB11819	ASP-4058	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	BETA-TOXICAROL	chembl:CHEMBL1556035	BETA-TOXICAROL	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.055155117	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	PIRENPERONE	ncit:C66417	PIRENPERONE	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.027781837	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.1151484018326633	Trifluridine	rxcui:10803	TRIFLURIDINE	TRUE	FALSE	FALSE
NCBIGENE:2105	hgnc:7111	MKNK2	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:9366	iuphar.ligand:9366	MELK-TI	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	4.145342465975881	OC-000459	iuphar.ligand:9277	TIMAPIPRANT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.1770916399180253	ETIOCHOLANOLONE	ncit:C29023	ETIOCHOLANOLONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005284588	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.040515178	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00445925	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.088695391	GLYCOPYRROLATE	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.036718651	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
APLN	hgnc:16665	APLN	NCI	14-Sep-17	NULL	1.875273972703374	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	PharmGKB	4/5/24	NULL	0.082732675	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:4264	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:9432	iuphar.ligand:9432	PF-06263276	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.056097939	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	6-O-BENZYLGUANINE	drugbank:DB11919	6-O-BENZYLGUANINE	FALSE	FALSE	FALSE
UNIPROT:P31639	hgnc:11037	SLC5A2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	IPRAGLIFLOZIN	ncit:C166685	IPRAGLIFLOZIN	FALSE	FALSE	FALSE
SIGLEC8	hgnc:10877	SIGLEC8	ChEMBL	33	inhibitor	52.50767123569449	LIRENTELIMAB	ncit:C129591	LIRENTELIMAB	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	ChEMBL	33	inhibitor	0.062808219	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:7707	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.028929846	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.02179646	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124226	chembl:CHEMBL586344	CHEMBL:CHEMBL586344	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:317	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.4605936073306534	SOLIFENACIN SUCCINATE	rxcui:476588	SOLIFENACIN SUCCINATE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.16256245	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P48454	hgnc:9316	PPP3CC	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	VOCLOSPORIN	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:7852	iuphar.ligand:7852	EXAMPLE 2 [WO2013004676]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:12867	iuphar.ligand:12867	CINSEBRUTINIB	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.046673486	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	DEXKETOPROFEN	rxcui:237162	DEXKETOPROFEN	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	AMINACRINE HYDROCHLORIDE	rxcui:81949	AMINACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
COL2A1	hgnc:2200	COL2A1	ChEMBL	33	cleavage	0.4605936073306535	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	2.917092846427472	INOTUZUMAB	chembl:CHEMBL4297558	INOTUZUMAB	TRUE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:1132	iuphar.ligand:1132	GLUCAGON-LIKE PEPTIDE 1-(7-36) AMIDE	FALSE	FALSE	FALSE
NCBIGENE:147	hgnc:278	ADRA1B	GuideToPharmacology	2024.1	agonist	0.2536602475154323	IUPHAR.LIGAND:3699	iuphar.ligand:3699	R-SPONDIN-3	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	TRANSTORINE	iuphar.ligand:2918	KYNURENIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	GNF-PF-4579	chembl:CHEMBL584626	CHEMBL:CHEMBL584626	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.2476776945079929	2-PHENYLACETYLAMINOBENZOTHIAZOLE	chembl:CHEMBL1405979	CHEMBL:CHEMBL1405979	FALSE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.1084869240406911	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PRMT1	hgnc:5187	PRMT1	DTC	9/2/20	NULL	13.12691780892362	NSC-47762	chembl:CHEMBL1092740	CHEMBL:CHEMBL1092740	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.091796628	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.066297565	INTERLEUKIN-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.0136917	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.023813003	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	PharmGKB	4/5/24	NULL	0.068637479	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.027010119	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.080781033	Ascorbic Acid	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
UNIPROT:Q02880	hgnc:11990	TOP2B	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	RTA 744	drugbank:DB05920	RTA 744	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:496	ncit:C75061	UPIDOSIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	P-HYDROXYPHENETHYL ANISATE	chembl:CHEMBL1078244	CHEMBL:CHEMBL1078244	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.045109683	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.4039051633514962	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
GCKR	hgnc:4196	GCKR	PharmGKB	4/5/24	NULL	0.5770073762164232	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TEND	1-Aug-11	NULL	1.826353782111113	AMBRISENTAN	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.032982206	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.026572708	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.029833904	IUPHAR.LIGAND:479	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.6563458904461813	IUPHAR.LIGAND:4113	iuphar.ligand:4113	9-ANTHROIC ACID	FALSE	FALSE	FALSE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	1.312691780892362	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003174779	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	Fenoterol	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	5.250767123569449	T863	iuphar.ligand:7828	T863	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	PharmGKB	4/5/24	NULL	3.000438356	velaglucerase alfa	rxcui:901805	VELAGLUCERASE ALFA	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	EVENAMIDE	ncit:C174804	EVENAMIDE	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6101	iuphar.ligand:6101	M1145	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.2263261691193728	DIPHYLLIN	chembl:CHEMBL221190	DIPHYLLIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.023274677	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
ACTR2	hgnc:169	ACTR2	NCI	14-Sep-17	NULL	6.563458904461812	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011352028	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	NSC-319994	chembl:CHEMBL1329443	CHEMBL:CHEMBL1329443	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW680191X	chembl:CHEMBL517907	GW680191X	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1876	iuphar.ligand:1876	&DELTA;12-PGJ2	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:4171	rxcui:1742747	SERINE, D-	FALSE	FALSE	FALSE
NCBIGENE:434	hgnc:745	ASIP	GuideToPharmacology	2024.1	blocker	5.250767123569449	IUPHAR.LIGAND:7704	iuphar.ligand:7704	AZD2927	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:25	iuphar.ligand:25	S-14671	FALSE	FALSE	FALSE
ITIH3	hgnc:6168	ITIH3	PharmGKB	4/5/24	NULL	1.082632396612257	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2734774543525755	TCMDC-123591	chembl:CHEMBL588234	CHEMBL:CHEMBL588234	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.009437037	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.2638576444004749	METHANESULFONIC ACID METHYL ESTER	chembl:CHEMBL313493	METHANESULFONIC ACID METHYL ESTER	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.059837802	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.4145342465975881	MARGETUXIMAB	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TEGASEROD MALEATE	rxcui:339270	TEGASEROD MALEATE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1483267549030917	METHOCTRAMINE HYDROCHLORIDE	chembl:CHEMBL500996	METHOCTRAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	blocker	0.6563458904461812	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	SJ000173328	chembl:CHEMBL591613	CHEMBL:CHEMBL591613	FALSE	FALSE	FALSE
NCBIGENE:1871	hgnc:3115	E2F3	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:5073	iuphar.ligand:5073	TUMOUR NECROSIS FACTOR MEMBRANE FORM	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	0.1902451856365742	PF-04965842	rxcui:2591476	ABROCITINIB	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007012242	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1852122442176172	ERLOTINIB HYDROCHLORIDE	rxcui:477320	ERLOTINIB HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:2336	hgnc:1476	CAPN1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10883	iuphar.ligand:10883	GC-376	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3658	iuphar.ligand:3658	[125I]CXCL7 (HUMAN)	FALSE	FALSE	FALSE
TP53AIP1	hgnc:29984	TP53AIP1	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:11728	iuphar.ligand:11728	BMS-986318	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1630	ncit:C170234	NORMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:9800	iuphar.ligand:9800	SELETALISIB	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.1973972602845657	IUPHAR.LIGAND:2446	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:2197	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	1.544343271638073	TCMDC-123961	chembl:CHEMBL587759	CHEMBL:CHEMBL587759	FALSE	FALSE	FALSE
CALCINEURIN	hgnc:9314	PPP3CA	TTD	2020.06.01	NULL	0.4688184931758437	Tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.2083637747448194	BIOFLAVONOID	ncit:C306	BIOFLAVONOID	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.4449802647092754	SARALASIN	rxcui:9556	SARALASIN	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	PharmGKB	4/5/24	NULL	0.045898314	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
F7	hgnc:3544	F7	ChEMBL	33	positive modulator	0.6250913242344582	EPTACOG ALFA PEGOL (ACTIVATED)	ncit:C166689	EPTACOG ALFA PEGOL (ACTIVATED)	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1852122442176172	ERLOTINIB HYDROCHLORIDE	rxcui:477320	ERLOTINIB HYDROCHLORIDE	TRUE	FALSE	TRUE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.05814803	ALLOPREGNANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2044	iuphar.ligand:2044	EC 5-21	FALSE	FALSE	FALSE
UGT2B4	hgnc:12553	UGT2B4	PharmGKB	4/5/24	NULL	2.692701089009974	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	1.750255707856483	ALPHA-ADRENERGIC AGONIST	ncit:C29709	ALPHA-ADRENERGIC AGONIST	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	negative modulator	0.2586584789935689	ESKETAMINE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
NCBIGENE:731	hgnc:1352	C8A	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	0.8078103267029922	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.5527123287967841	CPL304110	ncit:C173964	FGFR INHIBITOR CPL304110	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.1168135066422569	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	TCMDC-124381	chembl:CHEMBL579919	CHEMBL:CHEMBL579919	FALSE	FALSE	FALSE
NPIPB8	hgnc:37490	NPIPB8	PharmGKB	4/5/24	NULL	8.751278539282415	tapentadol	rxcui:787390	TAPENTADOL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005349192	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:12313	iuphar.ligand:12313	COMPOUND 29 [PMID: 36356320]	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.2461297089173179	KETOROLAC TROMETHAMINE	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
KCNJ8	hgnc:6269	KCNJ8	ChEMBL	33	potentiator	1.640864726115453	NAMINIDIL	ncit:C77076	NAMINIDIL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001193302	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	ChEMBL	33	agonist	0.9053046764774912	ULOTARONT	ncit:C179130	ULOTARONT	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:374	iuphar.ligand:374	CCPA	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:8175	iuphar.ligand:8175	COMPOUND 8H [PMID: 22765894]	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.305277158	CUPRESSUFLAVONE	chembl:CHEMBL1208973	CUPRESSUFLAVONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.014658758	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	AG1295	iuphar.ligand:5914	AG 1295	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.023080295	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	ZK-164015	chembl:CHEMBL184074	CHEMBL:CHEMBL184074	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	PharmGKB	4/5/24	NULL	0.2822993077187876	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	ENDRIN	chembl:CHEMBL44072	ENDRIN	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.03292017	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.040328473	ENMD 2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	OncoKB	23-Jul-20	NULL	0.3677319929494733	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ALDH1A2	hgnc:15472	ALDH1A2	NCI	14-Sep-17	NULL	0.6775183385250904	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.028290771	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8417	iuphar.ligand:8417	GLPG0974	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	inhibitor	0.1630673019742065	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11756	ncit:C175855	SIVOPIXANT	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	agonist	2.625383561784724	GLUCAGON HYDROCHLORIDE	rxcui:253170	GLUCAGON HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	12-HYDROXY-OCTADECANOIC ACID	chembl:CHEMBL292352	CHEMBL:CHEMBL292352	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.015241704	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
GLRA2	hgnc:4327	GLRA2	DTC	9/2/20	NULL	0.9376369863516874	HU-210	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	GNF-PF-3084	chembl:CHEMBL601135	CHEMBL:CHEMBL601135	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:1894	ncit:C79571	CLOPROSTENOL	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.4102161815288632	IUPHAR.LIGAND:2508	iuphar.ligand:2508	LYSOPHOSPHATIDYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.4646696569530486	IUPHAR.LIGAND:3873	iuphar.ligand:3873	DSTBULET	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004292999	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	SJ000089108	chembl:CHEMBL605708	CHEMBL:CHEMBL605708	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.049723174	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.6563458904461813	IL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
NCBIGENE:698	ncbigene:698	BTS1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4113	iuphar.ligand:4113	9-ANTHROIC ACID	FALSE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	ChEMBL	33	inhibitor	0.7955707762984013	RG-4733	drugbank:DB11870	RG-4733	FALSE	FALSE	FALSE
NCBIGENE:2943	hgnc:1682	CD47	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:11592	iuphar.ligand:11592	EVORPACEPT	FALSE	FALSE	FALSE
NCBIGENE:2136	hgnc:16059	PAK4	GuideToPharmacology	2024.1	inhibitor	0.1367387271762877	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.098884503	bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.4375639269641208	PRODIGIOSIN	chembl:CHEMBL275787	PRODIGIOSIN	FALSE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	ChEMBL	33	inhibitor	3.125456621172291	ABIRATERONE ACETATE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.021138354	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CHRNA5	hgnc:1959	CHRNA5	ChEMBL	33	agonist	2.187819634820604	POZANICLINE	ncit:C81045	POZANICLINE	FALSE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.068637479	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	3.088686543276147	BMS-770767	chembl:CHEMBL4802167	BMS-770767	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.1597596487901455	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:712	iuphar.ligand:712	COMPOUND (S)-3H [PMID: 15686947]	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.011668371	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.03357268	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1321	iuphar.ligand:1321	HS014	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	FEPRAZONE	rxcui:8673	FEPRAZONE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.059397818	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P41231	hgnc:8541	P2RY2	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	DIQUAFOSOL	ncit:C65436	DIQUAFOSOL	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	CID 670282	chembl:CHEMBL260213	CHEMBL:CHEMBL260213	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.080471527	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:3290	ncit:C74246	APADENOSON	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	1.363835616511545	KB07	chembl:CHEMBL373822	CHEMBL:CHEMBL373822	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.093931433	IUPHAR.LIGAND:7189	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CancerCommons	25-Jul-13	inhibitor	0.1750255707856483	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
IL7R	hgnc:6024	IL7R	CGI	2/1/22	NULL	3.088686543276147	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.055504938	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
CCL2	hgnc:10618	CCL2	ChEMBL	33	inhibitor	17.50255707856483	CARLUMAB	ncit:C71010	CARLUMAB	FALSE	FALSE	FALSE
NPR2	hgnc:7944	NPR2	ChEMBL	33	binder	2.917092846427472	VOSORITIDE	rxcui:2586354	VOSORITIDE	TRUE	FALSE	FALSE
UNIPROT:P22748	hgnc:1375	CA4	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:3297	iuphar.ligand:3297	[3H]NGD941	FALSE	FALSE	FALSE
PROTEASE	hgnc:39004	ERVK-10	ChEMBL	33	inhibitor	52.50767123569449	BMS-955176	drugbank:DB15193	BMS-955176	FALSE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	1.458546423213736	Alendronate	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
PTGER1	hgnc:9593	PTGER1	DTC	9/2/20	NULL	0.9376369863516875	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.091796628	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.011710007	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.085378327	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
DOPAMINE BETA HYDROXYLASE	hgnc:2689	DBH	TTD	2020.06.01	NULL	3.500511415712966	Etamicastat	ncit:C90846	ETAMICASTAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004540811	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	CGI	2/1/22	NULL	0.088333021	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	ChEMBL	33	inhibitor	0.192335792	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV000753	chembl:CHEMBL532141	CHEMBL:CHEMBL532141	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:8705	iuphar.ligand:8705	TM38837	FALSE	FALSE	FALSE
NCBIGENE:585	hgnc:969	BBS4	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12630	iuphar.ligand:12630	SUZETRIGINE	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:10441	iuphar.ligand:10441	COMPOUND 5D [PMID: 31335136]	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	CX-6258	iuphar.ligand:9368	CX-6258	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010678802	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.063110182	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.053253216	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-125066	chembl:CHEMBL533577	CHEMBL:CHEMBL533577	FALSE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	DTC	9/2/20	NULL	0.059940264	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	0.9723642821424906	KF-17837	chembl:CHEMBL27508	CHEMBL:CHEMBL27508	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.004352426	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10126	iuphar.ligand:10126	TRYPTANTHRIN 5I	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:5715	iuphar.ligand:5715	TG-100-115	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.028413242	IUPHAR.LIGAND:7875	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NCBIGENE:2916	hgnc:4598	GRM6	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9419	iuphar.ligand:9419	NEXINHIB20	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	KANZONOL X	chembl:CHEMBL606241	KANZONOL X	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.033658764	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8517	iuphar.ligand:8517	IS1	FALSE	FALSE	FALSE
ADAM17	hgnc:195	ADAM17	PharmGKB	4/5/24	NULL	0.5645986154375753	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
POLE	hgnc:9177	POLE	ChEMBL	33	inhibitor	0.1544343271638073	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	CHLOROPYRAMINE	rxcui:20861	CHLOROPYRAMINE	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1193356164447602	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	CIViC	10-Apr-24	NULL	0.9376369863516875	MCL-1 INHIBITOR MIK665	ncit:C133174	MCL-1 INHIBITOR MIK665	FALSE	FALSE	TRUE
P2RY11	hgnc:8540	P2RY11	DTC	9/2/20	NULL	17.50255707856483	ISO-IANTHERAN A	chembl:CHEMBL240681	ISO-IANTHERAN A	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.035358701	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1458546423213736	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	LASSBIO-123	chembl:CHEMBL573111	CHEMBL:CHEMBL573111	FALSE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	AMV564	ncit:C135632	VIXTIMOTAMAB	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.007941269	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.090843722	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.1004931506903244	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.760980743	RXDX-105	ncit:C107245	AGERAFENIB	FALSE	FALSE	TRUE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TdgClinicalTrial	Jan-14	NULL	0.1025540453822158	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.2692701089009974	TAMSULOSIN HYDROCHLORIDE	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	modulator	0.099446347	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.1190650141398968	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
TBC1D1	hgnc:11578	TBC1D1	PharmGKB	4/5/24	NULL	0.5413161983061289	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.020269319	clodronate	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2051080907644316	AMINOQUINURIDE	rxcui:17747	AMINOQUINURIDE	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.8751278539282416	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.09869863	SELADELPAR	ncit:C167015	SELADELPAR	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.093596562	MILCICLIB	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.03409589	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.2885036881082115	GW468816	chembl:CHEMBL1207366	GW468816	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.055247971	Sapanisertib	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
UNIPROT:P07202	hgnc:12015	TPO	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	CARBIMAZOLE	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:5661	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:1990	iuphar.ligand:1990	RELAXIN-3	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	COSMIC	4-Sep-20	NULL	0.4055851016423223	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:11537	iuphar.ligand:11537	NTP42	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.2103110997424346	MILNACIPRAN	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.006233104	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.1117184494376478	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	0.3860858179095183	Netarsudil	rxcui:1992864	NETARSUDIL	TRUE	FALSE	FALSE
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	0.108711535	Doramapimod	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	1.131630845596864	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.05073205	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:965	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1451	iuphar.ligand:1451	[L-BPA5,ILE13]MOTILIN (HUMAN)	FALSE	FALSE	FALSE
CXCR2	hgnc:6027	CXCR2	ChEMBL	33	inhibitor	4.375639269641208	NAVARIXIN	ncit:C156730	NAVARIXIN	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	inhibitor	2.625383561784724	ADOMEGLIVANT	ncit:C166989	ADOMEGLIVANT	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.044611445	TRIMIPRAMINE	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:7381	iuphar.ligand:7381	RS-100329	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:10011	ncit:C153478	DOLCANATIDE	FALSE	FALSE	FALSE
LCK TYROSINE PROTEIN KINASE	hgnc:6524	LCK	TTD	2020.06.01	NULL	0.3431873936973496	VX-680	ncit:C61319	TOZASERTIB LACTATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	MESO-HEXESTROL	drugbank:DB07931	HEXESTROL	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.076263865	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:Q03431	hgnc:9608	PTH1R	TEND	1-Aug-11	NULL	2.812910959055062	TERIPARATIDE	rxcui:32915	TERIPARATIDE	TRUE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9058	iuphar.ligand:9058	PF-03654746	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.1848861663228679	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.090634645	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
CCNK	hgnc:1596	CCNK	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006909813	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	TCMDC-123605	chembl:CHEMBL547285	CHEMBL:CHEMBL547285	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.09869863	AFACIFENACIN	ncit:C90741	AFACIFENACIN	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:2600	iuphar.ligand:2600	(S)-N-[1-(3-MORPHOLIN-4-YL-PHENYL)-ETHYL]-3-PHENYL-ACRYLAMIDE	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.2302968036653267	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.035418328	Mirabegron	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.002213645	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1346350544504987	MANNITOL	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1137761023525341	HYDROMORPHONE	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	AMINOQUINURIDE	rxcui:17747	AMINOQUINURIDE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.014528963	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	CGI	2/1/22	NULL	0.017409705	Ilorasertib	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.049349315	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CGI	2/1/22	NULL	0.1900426678745596	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PDGFB	hgnc:8800	PDGFB	CGI	2/1/22	NULL	0.3500511415712966	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CGI	2/1/22	NULL	1.009762908	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	PHENIRAMINE MALEATE	rxcui:266959	PHENIRAMINE MALEATE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	HYDROXYZINE HYDROCHLORIDE	rxcui:154987	HYDROXYZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RYR1	hgnc:10483	RYR1	ChEMBL	33	inhibitor	2.083637747448194	DANTROLENE SODIUM	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ChEMBL	33	inhibitor	2.917092846427472	PIMECROLIMUS	rxcui:321952	PIMECROLIMUS	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1893305453210138	LURASIDONE HYDROCHLORIDE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.020320306	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.2430910705356226	PHENDIMETRAZINE TARTRATE	rxcui:33272	PHENDIMETRAZINE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.4861821410712453	DIETHYLPROPION HYDROCHLORIDE	rxcui:81998	DIETHYLPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.2408608772279564	LEVALLORPHAN TARTRATE	rxcui:235419	LEVALLORPHAN TARTRATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1204304386139782	BUPRENORPHINE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	TAPENTADOL HYDROCHLORIDE	rxcui:857492	TAPENTADOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	PREDNISOLONE SODIUM PHOSPHATE	rxcui:55062	PREDNISOLONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	FLUOROMETHOLONE ACETATE	rxcui:221101	FLUOROMETHOLONE ACETATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	TRIAMCINOLONE DIACETATE	rxcui:10762	TRIAMCINOLONE DIACETATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.801643836	METHYLPREDNISOLONE ACETATE	rxcui:155323	METHYLPREDNISOLONE ACETATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.1226814748497534	CLOMIPHENE CITRATE	rxcui:142431	CLOMIPHENE CITRATE	TRUE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	ChEMBL	33	inhibitor	0.525076712	PEMETREXED DISODIUM	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	ChEMBL	33	agonist	0.068369364	FENOLDOPAM MESYLATE	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1226814748497534	SYNTHETIC CONJUGATED ESTROGENS, B	rxcui:618365	SYNTHETIC CONJUGATED ESTROGENS, B	TRUE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.1136529680426287	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.1442518440541058	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.4688184931758437	OMEPRAZOLE MAGNESIUM	rxcui:236486	OMEPRAZOLE MAGNESIUM	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.1041818873724097	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
CA12	hgnc:1371	CA12	ChEMBL	33	inhibitor	0.7501095890813501	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
CA5B	hgnc:1378	CA5B	ChEMBL	33	inhibitor	1.750255707856483	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.031254566	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
ITGB7	hgnc:6162	ITGB7	ChEMBL	33	inhibitor	2.187819634820604	NATALIZUMAB	rxcui:354770	NATALIZUMAB	TRUE	TRUE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.032016873	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.036977233	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.2817943000126717	CLONIDINE HYDROCHLORIDE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.2386712328895204	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1442518440541058	CLONIDINE HYDROCHLORIDE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.201952582	MIDODRINE HYDROCHLORIDE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	FENOPROFEN CALCIUM	rxcui:267171	FENOPROFEN CALCIUM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2983390411119005	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.01354163	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	FENOPROFEN CALCIUM	rxcui:267171	FENOPROFEN CALCIUM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	DICLOFENAC POTASSIUM	rxcui:81997	DICLOFENAC POTASSIUM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1074020548002842	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1790034246671403	KETOROLAC TROMETHAMINE	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.8078103267029924	SODIUM NITROPRUSSIDE	rxcui:9895	SODIUM NITROPRUSSIDE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.1873044158229292	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.058799184	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	0.2548916079402645	DEXTROTHYROXINE	rxcui:3292	DEXTROTHYROXINE	TRUE	FALSE	FALSE
ITGB1	hgnc:6153	ITGB1	ChEMBL	33	inhibitor	1.093909817410302	NATALIZUMAB	rxcui:354770	NATALIZUMAB	TRUE	TRUE	FALSE
BCHE	hgnc:983	BCHE	ChEMBL	33	inhibitor	0.5625821918110125	RIVASTIGMINE	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
CD80	hgnc:1700	CD80	ChEMBL	33	inhibitor	5.250767123569449	ABATACEPT	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
COL3A1	hgnc:2201	COL3A1	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
COL28A1	hgnc:22442	COL28A1	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	ChEMBL	33	positive modulator	0.1539814405738841	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.3409589041278864	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	negative modulator	0.099446347	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.05814803	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	negative modulator	0.02804897	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.089298761	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.087222045	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.082429625	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.031254566	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.033232703	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.032016873	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.093763699	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.023080295	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.026927011	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.028382525	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.055387839	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.030527716	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.032412143	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.033658764	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.03409589	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.091796628	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.035098711	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.039097298	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.087318744	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.023943307	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.021997349	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.021715331	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.6035364509849942	TROVAFLOXACIN MESYLATE	rxcui:221177	TROVAFLOXACIN MESYLATE	TRUE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	inhibitor	0.4688184931758437	MUROMONAB-CD3	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	1.125164383622024	USTEKINUMAB	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
POLA1	hgnc:9173	POLA1	ChEMBL	33	inhibitor	1.036335616	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
POLD4	hgnc:14106	POLD4	ChEMBL	33	inhibitor	0.4605936073306535	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
PRIM2	hgnc:9370	PRIM2	ChEMBL	33	inhibitor	0.108040476	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
POLA2	hgnc:30073	POLA2	ChEMBL	33	inhibitor	0.2206204673768676	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLD3	hgnc:20932	POLD3	ChEMBL	33	inhibitor	0.108040476	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
POLE3	hgnc:13546	POLE3	ChEMBL	33	inhibitor	0.108040476	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.052090944	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.051277023	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.063568609	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.062509132	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.049723174	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.058602312	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.098451884	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
RAMP2	hgnc:9844	RAMP2	ChEMBL	33	agonist	6.563458904461812	PRAMLINTIDE ACETATE	rxcui:356773	PRAMLINTIDE ACETATE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.077789143	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	CAPREOMYCIN SULFATE	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	ESLICARBAZEPINE ACETATE	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
ITGB7	hgnc:6162	ITGB7	ChEMBL	33	inhibitor	8.751278539282415	VEDOLIZUMAB	rxcui:1538097	VEDOLIZUMAB	TRUE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	ChEMBL	33	inhibitor	0.3365876361262467	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMB1	hgnc:9537	PSMB1	ChEMBL	33	inhibitor	0.384671584	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMC5	hgnc:9552	PSMC5	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMD12	hgnc:9557	PSMD12	ChEMBL	33	inhibitor	0.2692701089009974	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMB7	hgnc:9544	PSMB7	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
RARG	hgnc:9866	RARG	ChEMBL	33	modulator	0.5147810905460244	MOFAROTENE	ncit:C63667	MOFAROTENE	FALSE	FALSE	FALSE
RXRB	hgnc:10478	RXRB	ChEMBL	33	modulator	0.9723642821424906	MOFAROTENE	ncit:C63667	MOFAROTENE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.175415383	GLPG0492	chembl:CHEMBL3545417	GLPG0492	FALSE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	ChEMBL	33	agonist	1.250182648468916	HYODEOXYCHOLIC_ACID	chembl:CHEMBL272621	HYODEOXYCHOLIC_ACID	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.018006746	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.4930297768609811	MIRANSERTIB	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.2966535098061835	AMG-900	drugbank:DB17197	AMG-900	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	1.000146118775133	TELISOTUZUMAB	ncit:C106262	TELISOTUZUMAB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.2612321952024601	AMG-900	drugbank:DB17197	AMG-900	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	AZD-4769	chembl:CHEMBL422872	AZD-4769	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.2083637747448194	CEP-7055	chembl:CHEMBL346631	CEP-7055	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.4398548375764984	TOVORAFENIB	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	ChEMBL	33	inhibitor	8.078103267029922	NMS-1116354	chembl:CHEMBL3545321	NMS-1116354	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.3977853881492007	NSC-123414	chembl:CHEMBL16751	CHEMBL:CHEMBL16751	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.2047082699247349	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	SB-85635	chembl:CHEMBL3545384	SB-85635	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	3.424413341458336	WHI-P131	chembl:CHEMBL405130	WHI-P131	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.5834185692854944	TAK-960	chembl:CHEMBL2392545	TAK-960	FALSE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	2.763561643983921	XL550	chembl:CHEMBL3545393	XL550	FALSE	FALSE	FALSE
IL12A	hgnc:5969	IL12A	ChEMBL	33	inhibitor	1.750255707856483	EBDAROKIMAB	ncit:C179082	EBDAROKIMAB	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	ZYH7	chembl:CHEMBL3545093	ZYH7	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.3906820776465364	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.1902451856365742	AZD-1480	drugbank:DB12588	AZD-1480	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.060956201	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.016807833	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.067317527	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1470803115845784	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
EPHB4	hgnc:3395	EPHB4	ChEMBL	33	inhibitor	0.8204323630577265	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	ChEMBL	33	inhibitor	0.1093909817410302	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:1500	iuphar.ligand:1500	DES-BR-NEUROPEPTIDE B-29	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.082043236	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
FGR	hgnc:3697	FGR	ChEMBL	33	inhibitor	0.1562728310586145	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.075768645	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	ChEMBL	33	inhibitor	0.015777545	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.8334550989792777	INCB-40093	chembl:CHEMBL3545054	INCB-40093	FALSE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	ChEMBL	33	inhibitor	2.917092846427472	VERUCERFONT	ncit:C152869	VERUCERFONT	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1117184494376478	DAROTROPIUM BROMIDE	ncit:C76000	DAROTROPIUM BROMIDE	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	2.282942227638891	AZD2423	iuphar.ligand:7825	AZD2423	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	2.128689374420047	TRADIPITANT	ncit:C152707	TRADIPITANT	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.079798892	AFACIFENACIN	ncit:C90741	AFACIFENACIN	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	modulator	2.917092846427472	DIPRAGLURANT	ncit:C171677	DIPRAGLURANT	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.2430910705356226	INDANTADOL	ncit:C83796	INDANTADOL	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.6674703970639131	angiotensin II	rxcui:1999003	ANGIOTENSIN II	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	blocker	0.105015342	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	blocker	0.105015342	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	blocker	0.058341857	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	MAPRACORAT	ncit:C166458	MAPRACORAT	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.2453629496995069	ACOLBIFENE	ncit:C64183	ACOLBIFENE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.111481255	PEFCALCITOL	ncit:C170289	PEFCALCITOL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.0403388	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	ChEMBL	33	inhibitor	1.367387271762877	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.054020238	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	negative modulator	0.096167896	ESKETAMINE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	0.6141248097742047	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TEND	1-Aug-11	NULL	2.692701089009974	ERYTHRITYL TETRANITRATE	rxcui:4040	ERYTHRITYL TETRANITRATE	TRUE	FALSE	FALSE
LY96	hgnc:17156	LY96	ChEMBL	33	inhibitor	26.25383561784724	ERITORAN TETRASODIUM	ncit:C91759	ERITORAN TETRASODIUM	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	1.432027397337122	ETORICOXIB	rxcui:307296	ETORICOXIB	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	BENZYDAMINE	rxcui:1425	BENZYDAMINE	TRUE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	2.019525817	LIPEGFILGRASTIM	rxcui:1440046	LIPEGFILGRASTIM	TRUE	FALSE	FALSE
APH1B	hgnc:24080	APH1B	ChEMBL	33	inhibitor	1.514644363	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	ChEMBL	33	inhibitor	2.386712328895204	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.1875273972703374	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.5048814541893701	EPLIVANSERIN	ncit:C65517	EPLIVANSERIN	FALSE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	ChEMBL	33	inhibitor	1.193356164447602	AVAGACESTAT	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
RPE65	hgnc:10294	RPE65	ChEMBL	33	inhibitor	15.00219178	EMIXUSTAT	ncit:C171669	EMIXUSTAT	FALSE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	3.938075342677087	VALBENAZINE	rxcui:1918219	VALBENAZINE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1801292323694494	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
PDGFB	hgnc:8800	PDGFB	ChEMBL	33	inhibitor	8.751278539282415	PEGPLERANIB SODIUM	ncit:C170304	PEGPLERANIB SODIUM	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	ChEMBL	33	inhibitor	1.346350544504987	NIVOCASAN	ncit:C98213	NIVOCASAN	FALSE	FALSE	FALSE
BCL2L1	hgnc:992	BCL2L1	ChEMBL	33	inhibitor	0.6250913242344582	OBATOCLAX MESYLATE	ncit:C62771	OBATOCLAX MESYLATE	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.1875273972703374	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.3409589041278863	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	3.281729452230906	GUSELKUMAB	rxcui:1928588	GUSELKUMAB	TRUE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	1.250182648468916	TILDRAKIZUMAB	rxcui:2053436	TILDRAKIZUMAB	TRUE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	2.187819634820604	TILDRAKIZUMAB	rxcui:2053436	TILDRAKIZUMAB	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	ChEMBL	33	inhibitor	0.2966535098061835	FRESOLIMUMAB	ncit:C63546	FRESOLIMUMAB	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:11497	iuphar.ligand:11497	[3H]4-DAMP	FALSE	FALSE	FALSE
ICAM1	hgnc:5344	ICAM1	ChEMBL	33	inhibitor	8.751278539282415	ENLIMOMAB PEGOL	chembl:CHEMBL2108401	ENLIMOMAB PEGOL	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.040515178	GSK690693	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
UMPS	hgnc:12563	UMPS	ChEMBL	33	inhibitor	3.281729452230906	AZARIBINE	ncit:C1008	AZARIBINE	TRUE	FALSE	FALSE
S1PR3	hgnc:3167	S1PR3	ChEMBL	33	modulator	2.625383561784725	AMISELIMOD HYDROCHLORIDE	ncit:C142922	AMISELIMOD HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.050912416	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	inhibitor	0.091159151	AMINEPTINE	rxcui:17698	AMINEPTIN	TRUE	FALSE	FALSE
IFNA5	hgnc:5426	IFNA5	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.032899543	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
IFNA7	hgnc:5428	IFNA7	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	inhibitor	0.059397818	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HTR6	hgnc:5301	HTR6	ChEMBL	33	inhibitor	0.1346350544504987	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
UNIPROT:P08684	hgnc:2637	CYP3A4	TdgClinicalTrial	Jan-14	NULL	0.007341677	TESMILIFENE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
CPT2	hgnc:2330	CPT2	ChEMBL	33	inhibitor	0.1037701012563132	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	ZATUXIMAB	chembl:CHEMBL2109395	ZATUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	1.381780822	IUPHAR.LIGAND:2450	iuphar.ligand:2450	NAADP	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	ChEMBL	33	inhibitor	2.187819634820604	NARNATUMAB	ncit:C91382	NARNATUMAB	FALSE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	binder	0.8751278539282418	LUTETIUM DOTATATE LU-177	chembl:CHEMBL3989924	LUTETIUM DOTATATE LU-177	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	BICTEGRAVIR	rxcui:1999660	BICTEGRAVIR	TRUE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	binder	1.944728564284981	HUJ591 111IN	chembl:CHEMBL2109677	HUJ591 111IN	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.05814803	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.059532507	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	3.281729452230906	RISANKIZUMAB	rxcui:2166040	RISANKIZUMAB	TRUE	FALSE	FALSE
EEF2	hgnc:3214	EEF2	ChEMBL	33	inhibitor	0.9723642821424906	TAGRAXOFUSP	rxcui:2109054	TAGRAXOFUSP-ERZS	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	BICTEGRAVIR SODIUM	rxcui:1999661	BICTEGRAVIR SODIUM	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.3365876361262467	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
BMX	hgnc:1079	BMX	ChEMBL	33	inhibitor	1.750255707856483	PF-06651600	chembl:CHEMBL4085457	PF-06651600	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.017566969	palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
TEC	hgnc:11719	TEC	ChEMBL	33	inhibitor	0.6731752722524935	PF-06651600	chembl:CHEMBL4085457	PF-06651600	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.02232469	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.02534154	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.014537008	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	inhibitor	0.02232469	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.021309932	CENOBAMATE	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1593072549626653	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
PPIA	hgnc:9253	PPIA	ChEMBL	33	inhibitor	7.501095891	ALISPORIVIR	ncit:C169774	ALISPORIVIR	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1620607136904151	FEDRATINIB HYDROCHLORIDE	rxcui:2197594	FEDRATINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.1141471113819445	UPADACITINIB	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.2453629496995069	ESTRIOL	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.3125456621172291	ESTRIOL	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	5.250767123569449	EPOETIN DELTA	ncit:C166731	EPOETIN DELTA	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	CYCLOBENZAPRINE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	ESFLURBIPROFEN	ncit:C80544	ESFLURBIPROFEN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.2263261691193728	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.1491695205559502	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	GNF-PF-4467	chembl:CHEMBL598883	CHEMBL:CHEMBL598883	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.4167275494896388	LASOFOXIFENE	ncit:C80679	LASOFOXIFENE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.1346350544504987	NAFTOPIDIL	ncit:C72927	NAFTOPIDIL	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.2224901323546377	IMIDAPRIL	rxcui:60245	IMIDAPRIL	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	LOXOPROFEN	rxcui:28908	LOXOPROFEN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.4907258993990139	IOBENGUANE I 131	rxcui:2053281	IOBENGUANE I-131	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	RG-7841	chembl:CHEMBL4297935	RG-7841	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.036162308	phenprocoumon	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
TRAF3IP2	hgnc:1343	TRAF3IP2	ChEMBL	33	inhibitor	3.750547945406749	IGURATIMOD	ncit:C65886	IGURATIMOD	FALSE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	1.312691780892362	MITIGLINIDE CALCIUM DIHYDRATE	chembl:CHEMBL4298005	MITIGLINIDE CALCIUM DIHYDRATE	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.9053046764774912	MITIGLINIDE CALCIUM DIHYDRATE	chembl:CHEMBL4298005	MITIGLINIDE CALCIUM DIHYDRATE	FALSE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	ChEMBL	33	inhibitor	4.039051633514961	VOLIXIBAT	ncit:C152907	VOLIXIBAT	FALSE	FALSE	FALSE
INTERLEUKIN-4	hgnc:6014	IL4	TTD	2020.06.01	NULL	21.00306849427779	Pascolizumab	ncit:C88618	PASCOLIZUMAB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	AZINTUXIZUMAB VEDOTIN	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
TGFB3	hgnc:11769	TGFB3	ChEMBL	33	binder	2.625383561784725	BINTRAFUSP ALFA	ncit:C124229	BINTRAFUSP ALFA	FALSE	FALSE	FALSE
TGFB2	hgnc:11768	TGFB2	ChEMBL	33	binder	1.500219178	BINTRAFUSP ALFA	ncit:C124229	BINTRAFUSP ALFA	FALSE	FALSE	FALSE
FGF1	hgnc:3665	FGF1	ChEMBL	33	agonist	1.944728564284981	PEGBELFERMIN	ncit:C174833	PEGBELFERMIN	FALSE	FALSE	FALSE
KLB	hgnc:15527	KLB	ChEMBL	33	agonist	4.375639269641208	PEGBELFERMIN	ncit:C174833	PEGBELFERMIN	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.068191781	TENOFOVIR	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.075333818	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
DKK1	hgnc:2891	DKK1	ChEMBL	33	inhibitor	5.834185692854944	DKN-01	chembl:CHEMBL4297562	DKN-01	FALSE	FALSE	FALSE
BRDT	hgnc:1105	BRDT	ChEMBL	33	inhibitor	0.7501095890813501	PELABRESIB	ncit:C188265	PELABRESIB	FALSE	FALSE	FALSE
GRB14	hgnc:4565	GRB14	NCI	14-Sep-17	NULL	0.6604738520213144	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	ChEMBL	33	inhibitor	5.527123287967842	OLECLUMAB	ncit:C123914	OLECLUMAB	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.210030685	MK-0767	drugbank:DB12055	MK-0767	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	BILR 355	chembl:CHEMBL1630842	BILR 355	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	ChEMBL	33	inhibitor	0.1190650141398968	GOSURANEMAB	ncit:C175078	GOSURANEMAB	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	TNP-2092	drugbank:DB16312	TNP-2092	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	ACETOSIDE	chembl:CHEMBL444478	ACETOSIDE	FALSE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.8334550989792776	APINOCALTAMIDE	ncit:C190345	APINOCALTAMIDE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	1.458546423213736	RELAMORELIN	ncit:C152174	RELAMORELIN	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.023535487	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.1810609352954982	SNX 5422	ncit:C141504	SNX 5422	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	0.1835932560688619	LENOGRASTIM	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
AGTR2	hgnc:338	AGTR2	ChEMBL	33	inhibitor	4.773424657790408	OLODANRIGAN	ncit:C174823	OLODANRIGAN	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.1790034246671403	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.062509132	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	2.461297089173179	ZICONOTIDE	rxcui:68503	ZICONOTIDE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.2518353536484148	VODOBATINIB	ncit:C174748	VODOBATINIB	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	ZOLIFLODACIN	ncit:C152962	ZOLIFLODACIN	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.4039051633514961	BELUMOSUDIL	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	ERYTHROMYCIN ACISTRATE	ncit:C166893	ERYTHROMYCIN ACISTRATE	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.1392776425349986	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	GLOFITAMAB	rxcui:2639782	GLOFITAMAB	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.096167896	LEVOSULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
FCGRT	hgnc:3621	FCGRT	ChEMBL	33	inhibitor	5.834185692854944	NIPOCALIMAB	ncit:C170891	NIPOCALIMAB	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.5147810905460245	PIRTOBRUTINIB	rxcui:2629338	PIRTOBRUTINIB	TRUE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	2.386712328895204	ORN-0829 HYDRATE	chembl:CHEMBL4650522	ORN-0829 HYDRATE	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN, PROTAMINE ZINC	chembl:CHEMBL2109046	INSULIN, PROTAMINE ZINC	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	0.6177373086552294	INCB-086550	chembl:CHEMBL4802209	INCB-086550	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	ChEMBL	33	positive modulator	2.763561643983921	TRENONACOG ALFA	ncit:C152727	TRENONACOG ALFA	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	binder	0.1881995384791917	ABBV-3373	iuphar.ligand:12917	ABBV-3373	FALSE	FALSE	FALSE
NOX1	hgnc:7889	NOX1	ChEMBL	33	inhibitor	8.751278539282415	SETANAXIB	ncit:C166721	SETANAXIB	FALSE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	blocker	0.1262203635473425	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	blocker	0.2243917574174979	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.8607814956671229	TRIMEGESTONE	ncit:C152746	TRIMEGESTONE	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.048083948	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	blocker	0.1553481397505754	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.036770078	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
IL5	hgnc:6016	IL5	ChEMBL	33	inhibitor	5.834185692854944	DEPEMOKIMAB	ncit:C175768	DEPEMOKIMAB	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	2.019525817	REGRAMOSTIM	ncit:C170366	REGRAMOSTIM	FALSE	FALSE	FALSE
APLNR	hgnc:339	APLNR	ChEMBL	33	agonist	26.25383561784724	APELIN	chembl:CHEMBL4650373	APELIN	FALSE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.9376369863516875	ABEPRAZAN	ncit:C171876	FEXUPRAZAN	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.525076712	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3906820776465364	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
HMGCR	hgnc:5006	HMGCR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.121958787087489	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.049026771	GDC-0942	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PDCD1	hgnc:8760	PDCD1	ClearityFoundationClinicalTrial	15-Jun-13	blocker	0.2561349816375342	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
TLR8	hgnc:15632	TLR8	ClearityFoundationClinicalTrial	15-Jun-13	immunotherapy	13.12691780892362	SURECN254984	ncit:C80521	MOTOLIMOD	FALSE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.046940525	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	COSMIC	4-Sep-20	NULL	2.341819737097098	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.3864200913449379	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	E-4031	iuphar.ligand:2605	E4031	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.040515178	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CHLORMADINONE ACETATE	rxcui:2369	CHLORMADINONE ACETATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009922085	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.1450488155682168	N-BENZOYLANTHRANILIC ACID	chembl:CHEMBL198666	CHEMBL:CHEMBL198666	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	DTC	9/2/20	NULL	0.5073204950308646	PHILANTHOTOXIN 343	chembl:CHEMBL16117	PHILANTHOTOXIN 343	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.020446912	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	MAYTANSINE	ncit:C626	MAYTANSINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE	chembl:CHEMBL1569494	CHEMBL:CHEMBL1569494	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	2,6-DIMETHOXYQUINONE	chembl:CHEMBL448515	2,6-DIMETHOXYQUINONE	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	DTC	9/2/20	NULL	1.193356164447602	6-O-BENZYLGUANINE	drugbank:DB11919	6-O-BENZYLGUANINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	P-HYDROXYPHENETHYL ANISATE	chembl:CHEMBL1078244	CHEMBL:CHEMBL1078244	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	1,7-O-DIACETYLMETHYLGEOPYXIN A	chembl:CHEMBL1889303	CHEMBL:CHEMBL1889303	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.072424374	NSC-117079	chembl:CHEMBL471225	CHEMBL:CHEMBL471225	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	1.500219178	TDR78826	chembl:CHEMBL1500913	CHEMBL:CHEMBL1500913	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	DNDI1417701	chembl:CHEMBL1326164	CHEMBL:CHEMBL1326164	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	AMDINOCILLIN	rxcui:626	AMDINOCILLIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	HARPAGOSIDE	rxcui:2048124	HARPAGOSIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	NSC-747261	chembl:CHEMBL593366	CHEMBL:CHEMBL593366	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.037693949	ROSE BENGAL	rxcui:9471	ROSE BENGAL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	RO-84304	iuphar.ligand:4300	RO 8-4304	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	CID 670282	chembl:CHEMBL260213	CHEMBL:CHEMBL260213	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	TRYPAN BLUE	rxcui:10878	TRYPAN BLUE	TRUE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.1067229090156392	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
ENPP2	hgnc:3357	ENPP2	DTC	9/2/20	NULL	17.50255707856483	NSC-12188	chembl:CHEMBL1089321	CHEMBL:CHEMBL1089321	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.055563673	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.085239726	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004128935	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	ISOETHARINE	rxcui:6023	ISOETHARINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	BREFELDIN A	drugbank:DB07348	BREFELDIN A	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	2.019525817	NSC-640584	chembl:CHEMBL476968	CHEMBL:CHEMBL476968	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	RUTAECARPINE	chembl:CHEMBL85139	RUTAECARPINE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.006707674	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.082171629	PIRARUBICIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	FURAMIDINE	chembl:CHEMBL24057	FURAMIDINE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	LUFENURON	rxcui:83586	LUFENURON	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.001873601	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1363835616511545	N-ETHYLMALEIMIDE	drugbank:DB02967	N-ETHYLMALEIMIDE	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.3409589041278863	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	DNDI1417319	chembl:CHEMBL1392244	CHEMBL:CHEMBL1392244	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.7001022831425933	IMIDOCARB DIPROPIONATE	rxcui:1740238	IMIDOCARB DIPROPIONATE	TRUE	FALSE	FALSE
GRM1	hgnc:4593	GRM1	DTC	9/2/20	NULL	4.375639269641208	PHILANTHOTOXIN 343	chembl:CHEMBL16117	PHILANTHOTOXIN 343	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.011065895	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
TNNT2	hgnc:11949	TNNT2	DTC	9/2/20	NULL	0.525076712	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01535312	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2447910080918158	SUBEROHYDROXAMIC ACID	chembl:CHEMBL320497	SUBEROHYDROXAMIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ANECORTAVE ACETATE	ncit:C171908	ANECORTAVE ACETATE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.061628722	PROSTAGLANDIN B1	chembl:CHEMBL1561148	PROSTAGLANDIN B1	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NSC-83217	chembl:CHEMBL120806	CHEMBL:CHEMBL120806	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-117023	chembl:CHEMBL2059274	CHEMBL:CHEMBL2059274	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.1535312024435511	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.010175905	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.017485072	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.04907259	4-NONYLPHENOL	rxcui:1788868	4-NONYLPHENOL	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.061055432	THIOLACTOMYCIN	drugbank:DB04302	4-HYDROXY-3,5-DIMETHYL-5-(2-METHYL-BUTA-1,3-DIENYL)-5H-THIOPHEN-2-ONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.006614723	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006987979	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.084963869	TCMDC-123730	chembl:CHEMBL530280	CHEMBL:CHEMBL530280	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	OXYPHENONIUM BROMIDE	rxcui:42833	OXYPHENONIUM BROMIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PYRIDOSTIGMINE BROMIDE	rxcui:9001	PYRIDOSTIGMINE BROMIDE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.005834186	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003185179	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	FENTHION	drugbank:DB11412	FENTHION	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.021832712	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	NSC-22225	chembl:CHEMBL462314	CHEMBL:CHEMBL462314	FALSE	FALSE	FALSE
EPAS1	hgnc:3374	EPAS1	DTC	9/2/20	NULL	8.751278539282415	HALICLONADIAMINE	chembl:CHEMBL2177349	HALICLONADIAMINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-98	chembl:CHEMBL244023	CHEMBL:CHEMBL244023	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.1779921058837101	GNF-PF-3832	chembl:CHEMBL261693	CHEMBL:CHEMBL261693	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	METOLAZONE	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.2035181055647073	1-DEOXYRUBRALACTONE	chembl:CHEMBL260980	CHEMBL:CHEMBL260980	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	NIHYDRAZONE	ncit:C175162	NIHYDRAZONE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.7395446652914718	GARENOXACIN	ncit:C65800	GARENOXACIN	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1100789753368857	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.157680694	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	TYRPHOSTIN 1	iuphar.ligand:5917	AG 9	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.058341857	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.007544206	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BROQUINALDOL	ncit:C73256	BROQUINALDOL	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.00937637	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	4-(2-AMINOETHYL)BENZENESULFONYL FLUORIDE	drugbank:DB07347	4-(2-AMINOETHYL)BENZENESULFONYL FLUORIDE	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.059667808	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	FURATHIOCARB	chembl:CHEMBL1551453	FURATHIOCARB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	RESORCINOL MONOACETATE	rxcui:2106739	RESORCINOL MONOACETATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIFLUCORTOLONE 21-VALERATE	chembl:CHEMBL2358130	DIFLUCORTOLONE 21-VALERATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	PT-102	chembl:CHEMBL317356	CHEMBL:CHEMBL317356	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004762601	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.3088686543276147	TIOXOLONE	rxcui:2059173	TIOXOLONE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008887554	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	ZOLANTIDINE	chembl:CHEMBL419296	ZOLANTIDINE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.3725599732909588	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.037884323	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.069089041	CID 867101	chembl:CHEMBL406557	CHEMBL:CHEMBL406557	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011810092	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.031822831	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.9546849315580819	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003528741	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	3.750547945	TRIS(4-ISOPROPYLPHENYL) PHOSPHATE	chembl:CHEMBL458602	CHEMBL:CHEMBL458602	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	CID 2093195	chembl:CHEMBL411085	CHEMBL:CHEMBL411085	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.3977853881492007	TCMDC-125603	chembl:CHEMBL528734	CHEMBL:CHEMBL528734	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	20(S)-GINSENOSIDE RG3	iuphar.ligand:7658	GINSENOSIDE RG3	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	SJ000116228	chembl:CHEMBL577887	CHEMBL:CHEMBL577887	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003313623	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-125435	chembl:CHEMBL525888	CHEMBL:CHEMBL525888	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.01327292	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.034727296	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	QUINOXALINE1	iuphar.ligand:5947	CDK1/5 INHIBITOR	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.02617531	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.034184682	SB-242084	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	GNF-PF-1192	chembl:CHEMBL584854	CHEMBL:CHEMBL584854	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.039527003	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007596596	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.021357605	DAPSONE	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	DTC	9/2/20	NULL	1.521961485092594	TAK-779	iuphar.ligand:783	TAK-779	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	DTC	9/2/20	NULL	1.640864726115453	TDR79154	chembl:CHEMBL597670	CHEMBL:CHEMBL597670	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.03729238	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.017982079	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
MIF	hgnc:7097	MIF	DTC	9/2/20	NULL	17.50255707856483	TCMDC-124484	chembl:CHEMBL524449	CHEMBL:CHEMBL524449	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009433646	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.1071585127259071	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006324701	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.058602312	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.010148371	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	0.3106962795011509	NIFLUMIC ACID	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.4487835148349957	N-METHYL-N-NITROSOUREA	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	1.591141552596802	QUERCITRIN	chembl:CHEMBL82242	QUERCITRIN	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.2651902587661338	IMIDOCARB DIPROPIONATE	rxcui:1740238	IMIDOCARB DIPROPIONATE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	RHAMNETIN	drugbank:DB16772	RHAMNETIN	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.010777437	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.010777437	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	SULCONAZOLE NITRATE	rxcui:56798	SULCONAZOLE NITRATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007596596	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.098605955	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
EEF2	hgnc:3214	EEF2	DTC	9/2/20	NULL	0.061412481	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	GNF-PF-1134	chembl:CHEMBL600694	CHEMBL:CHEMBL600694	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1491695205559502	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.2476776945079929	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.023943307	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.063110182	ABT-702	iuphar.ligand:5131	ABT702	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.03070624	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.007866318	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	METHYL 3-(2,5-DIHYDROXYPHENYL)ACRYLATE	chembl:CHEMBL17329	CHEMBL:CHEMBL17329	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.1491695205559502	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2083637747448194	GNF-PF-5029	chembl:CHEMBL1198140	CHEMBL:CHEMBL1198140	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.1630673019742065	ZERANOL	rxcui:1368476	ZERANOL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.005753635	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.020688602	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NSC-74429	chembl:CHEMBL1269022	CHEMBL:CHEMBL1269022	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	CHLORPYRIFOS-METHYL	ncit:C163642	CHLORPYRIFOS-METHYL	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.020351811	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	TCMDC-125319	chembl:CHEMBL527586	CHEMBL:CHEMBL527586	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	MESO-HEXESTROL	drugbank:DB07931	HEXESTROL	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1312691780892362	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	ChEMBL	33	agonist	2.461297089173179	CORTICOTROPIN	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.2201579506737715	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
TLR2	hgnc:11848	TLR2	DTC	9/2/20	NULL	7.501095891	RESVERATROL HEXANOIC ACID	chembl:CHEMBL504510	RESVERATROL HEXANOIC ACID	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
HNF4A	hgnc:5024	HNF4A	DTC	9/2/20	NULL	0.2524407270946851	TOREMIFENE CITRATE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	AG-1288	chembl:CHEMBL166486	CHEMBL:CHEMBL166486	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.058931169	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	NORETHINDRONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.002668073	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
NCBIGENE:511	hgnc:3145	TRPV5	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6418	iuphar.ligand:6418	TETRAHYDROCANNABIVARIN	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	1.250182648468916	2,3,5-TRIS(4-HYDROXYPHENYL)THIOPHENE	chembl:CHEMBL2332580	CHEMBL:CHEMBL2332580	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.013673873	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.03292017	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.018962684	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	GNF-PF-1211	chembl:CHEMBL600968	CHEMBL:CHEMBL600968	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	12-CHLOROEVODIAMINE	chembl:CHEMBL2171803	CHEMBL:CHEMBL2171803	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	AZASERINE	ncit:C289	AZASERINE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.596678082	PALMATINE CHLORIDE	chembl:CHEMBL274189	PALMATINE CHLORIDE	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	DTC	9/2/20	NULL	0.025256215	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.1118771404169627	ISOPROTERENOL HYDROCHLORIDE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.017444409	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.039068208	CGP-7930	iuphar.ligand:1079	CGP7930	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002610374	VERAPAMIL HYDROCHLORIDE	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	RU-24969	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	DTC	9/2/20	NULL	4.773424657790408	L-4-THIOPROLINE	chembl:CHEMBL1800368	CHEMBL:CHEMBL1800368	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.040235763	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.1419126249613365	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
ADCY1	hgnc:232	ADCY1	DTC	9/2/20	NULL	8.751278539282415	NSC-270718	chembl:CHEMBL401844	CHEMBL:CHEMBL401844	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	CHLORPHRIFOS OXON	chembl:CHEMBL444970	CHLORPHRIFOS OXON	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.099446347	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.2263261691193728	GNF-PF-4612	chembl:CHEMBL601550	CHEMBL:CHEMBL601550	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	GNF-PF-2414	chembl:CHEMBL601353	CHEMBL:CHEMBL601353	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	NSC-638080	chembl:CHEMBL136344	CHEMBL:CHEMBL136344	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	N-ETHYLMALEIMIDE	drugbank:DB02967	N-ETHYLMALEIMIDE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2713574740862764	TERTATOLOL	rxcui:37840	TERTATOLOL	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.060353645	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.3500511415712966	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	chembl:CHEMBL1226	AMINODIMETHOXYQUINAZOLINYLPIPERAZINE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.015268296	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010569177	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	GNF-PF-4814	chembl:CHEMBL585443	CHEMBL:CHEMBL585443	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.025942525	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	OXATOMIDE	rxcui:54236	OXATOMIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PYRIDALYL	chembl:CHEMBL2136658	PYRIDALYL	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.7501095890813501	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
GPBAR1	hgnc:19680	GPBAR1	DTC	9/2/20	NULL	1.346350544504987	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.091159151	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	1.640864726115453	3,4,5,6-TETRACHLORO-[1,2]BENZOQUINONE	chembl:CHEMBL364729	CHEMBL:CHEMBL364729	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	NSC-638080	chembl:CHEMBL136344	CHEMBL:CHEMBL136344	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.011741429	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.052824619	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.021706354	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2393966773663883	PROPANTHELINE	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	DNDI1417457	chembl:CHEMBL1530911	CHEMBL:CHEMBL1530911	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.060562481	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.1704794520639431	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.010271454	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.029057925	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.087512785	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	2-PYRIDYLKETONE THIOPHENECARBOXYL HYDRAZONE	chembl:CHEMBL255068	CHEMBL:CHEMBL255068	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1988926940746003	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ENDRIN	chembl:CHEMBL44072	ENDRIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIFLOXACIN HYDROCHLORIDE	ncit:C72740	DIFLOXACIN HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.026626608	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.1785975212098452	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.02287916	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GNF-PF-2260	chembl:CHEMBL601351	CHEMBL:CHEMBL601351	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.054020238	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	NSC-81747	chembl:CHEMBL1371696	CHEMBL:CHEMBL1371696	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	CYCLOTHIAZIDE	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.005905046	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:959	hgnc:11935	CD40LG	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:7104	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1250182648468916	TCMDC-123808	chembl:CHEMBL546493	CHEMBL:CHEMBL546493	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000040837	chembl:CHEMBL590672	CHEMBL:CHEMBL590672	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.546954909	TOSYL-L-LYSINE CHLOROMETHYL KETONE	chembl:CHEMBL466465	CHEMBL:CHEMBL466465	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	LAVENDUSTIN A	ncit:C1142	LAVENDUSTIN A	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.07458476	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.042863405	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.1172046232939609	ROSMARINIC ACID	rxcui:2531311	ROSMARINIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00747866	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1367387271762877	AMPEROZIDE	ncit:C74191	AMPEROZIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	DIPHENIDOL	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	METRONIDAZOLE	rxcui:6922	METRONIDAZOLE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	(R)-PINOCEMBRIN	chembl:CHEMBL399249	(R)-PINOCEMBRIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	SJ000001516	chembl:CHEMBL592316	CHEMBL:CHEMBL592316	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.3070624048871023	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.07458476	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-125779	chembl:CHEMBL531451	CHEMBL:CHEMBL531451	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	TUBERCIDIN	ncit:C911	TUBERCIDIN	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	DTC	9/2/20	NULL	0.3182283105193606	L-GLUTAMATE	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.080781033	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.1312691780892362	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.01630673	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DNDI1317721	chembl:CHEMBL1385558	CHEMBL:CHEMBL1385558	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.011890324	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.001759051	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	ARTEMISININ	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.051226996	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00684585	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	EDARAVONE	rxcui:1921877	EDARAVONE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.063110182	PURVALANOL B	iuphar.ligand:7806	PURVALANOL B	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.011668371	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1056492378987816	DAPHNORIN	chembl:CHEMBL1209491	DAPHNORIN	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	3.281729452230906	TCMDC-124245	chembl:CHEMBL587615	CHEMBL:CHEMBL587615	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.026319635	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008136519	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.004155732	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.082171629	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
SOD1	hgnc:11179	SOD1	DTC	9/2/20	NULL	0.5834185692854945	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	DTC	9/2/20	NULL	0.3671865121377238	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	DNDI1416917	chembl:CHEMBL1335833	CHEMBL:CHEMBL1335833	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	TCMDC-123808	chembl:CHEMBL546493	CHEMBL:CHEMBL546493	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.068907705	GAMOLENIC ACID	rxcui:25605	GAMMA-LINOLENIC ACID	FALSE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	2.692701089009974	LESINURAD	rxcui:1731031	LESINURAD	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	OLEOYLETHANOLAMIDE	iuphar.ligand:2661	N-OLEOYLETHANOLAMIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.022099188	DAPSONE	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	TCMDC-123730	chembl:CHEMBL530280	CHEMBL:CHEMBL530280	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1293292394967844	GNF-PF-5029	chembl:CHEMBL1198140	CHEMBL:CHEMBL1198140	FALSE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.009673484	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	2.917092846427472	NSC-39249	chembl:CHEMBL482792	CHEMBL:CHEMBL482792	FALSE	FALSE	FALSE
CDK5R1	hgnc:1775	CDK5R1	DTC	9/2/20	NULL	0.2885036881082116	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
ADAM17	hgnc:195	ADAM17	DTC	9/2/20	NULL	1.166837138570988	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	5.250767123569449	DIPICOLINIC ACID	drugbank:DB04267	DIPICOLINIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.009553798	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.083744292	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.041312094	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.061197752	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.305277158	GNF-PF-2100	chembl:CHEMBL576175	CHEMBL:CHEMBL576175	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV396704	chembl:CHEMBL2028056	CHEMBL:CHEMBL2028056	FALSE	FALSE	FALSE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.095500063	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	THIOLACTOMYCIN	drugbank:DB04302	4-HYDROXY-3,5-DIMETHYL-5-(2-METHYL-BUTA-1,3-DIENYL)-5H-THIOPHEN-2-ONE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	FURAMIDINE	chembl:CHEMBL24057	FURAMIDINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.3621218705909965	3-NITROPROPIONIC ACID	chembl:CHEMBL451226	CHEMBL:CHEMBL451226	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	ANTIMYCIN A	chembl:CHEMBL211501	ANTIMYCIN A	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.3017682254924971	GNF-PF-1477	chembl:CHEMBL582675	CHEMBL:CHEMBL582675	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	DTC	9/2/20	NULL	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	PIROCTONE	rxcui:2058907	PIROCTONE	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.2983390411119005	OLOMOUCINE	drugbank:DB02116	OLOMOUCINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	BENFLUOREX HYDROCHLORIDE	rxcui:235953	BENFLUOREX HYDROCHLORIDE	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	2.282942227638891	COUMERMYCIN A1	ncit:C81447	COUMERMYCIN	FALSE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	activator	0.7292732116068681	IUPHAR.LIGAND:4150	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.1562728310586145	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.1600843635234588	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.1682938180631233	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	DIMETHYLPINOCEMBRIN	chembl:CHEMBL107131	DIMETHYLPINOCEMBRIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	TCMDC-123605	chembl:CHEMBL547285	CHEMBL:CHEMBL547285	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.1097339001790898	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.3088686543276147	DNDI1417368	chembl:CHEMBL2094652	CHEMBL:CHEMBL2094652	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.021258166	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-108	chembl:CHEMBL578929	CHEMBL:CHEMBL578929	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.047734247	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE	chembl:CHEMBL1569494	CHEMBL:CHEMBL1569494	FALSE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.2243917574174978	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	NSC-7387	chembl:CHEMBL119878	CHEMBL:CHEMBL119878	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002669701	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.3697723326457359	GNF-PF-2442	chembl:CHEMBL578420	CHEMBL:CHEMBL578420	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.023336743	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.046673486	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	LESCOL	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.018031481	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW300657X	chembl:CHEMBL272165	GW300657X	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.061412481	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.157680694	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.091796628	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1100789753368857	10-METHOXYLRUTAECARPINE	chembl:CHEMBL85826	CHEMBL:CHEMBL85826	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	SJ000168197	chembl:CHEMBL590670	CHEMBL:CHEMBL590670	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.009860596	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.041672755	NSC-699479	chembl:CHEMBL1701915	CHEMBL:CHEMBL1701915	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	CAMPHOR	rxcui:1297880	CAMPHOR OIL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NSC-49789	chembl:CHEMBL469309	CHEMBL:CHEMBL469309	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	LOMEFLOXACIN	rxcui:28872	LOMEFLOXACIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	SJ000167432	chembl:CHEMBL589909	CHEMBL:CHEMBL589909	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TCMDC-125232	chembl:CHEMBL531079	CHEMBL:CHEMBL531079	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	SB-431542	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
TMPRSS15	hgnc:9490	TMPRSS15	DTC	9/2/20	NULL	0.6177373086552295	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001174668	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.012501826	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	GNF-PF-793	chembl:CHEMBL604311	CHEMBL:CHEMBL604311	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.021805511	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.078136416	DNDI1417599	chembl:CHEMBL2094833	CHEMBL:CHEMBL2094833	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1019566431761058	FENOLDOPAM BROMIDE	chembl:CHEMBL1256646	FENOLDOPAM BROMIDE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.013638356	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	DEQUALINIUM CHLORIDE	rxcui:3120	DEQUALINIUM CHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	IODOQUINOL	rxcui:3435	IODOQUINOL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	FUROXAN	chembl:CHEMBL336467	FUROXAN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	(S)-NITRENDIPINE	chembl:CHEMBL251230	(S)-NITRENDIPINE	FALSE	FALSE	FALSE
APOA1	hgnc:600	APOA1	DTC	9/2/20	NULL	4.565884455277782	BMS-309403	iuphar.ligand:6735	BMS309403	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.020195258	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	DNDI1417621	chembl:CHEMBL1431017	CHEMBL:CHEMBL1431017	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003469746	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.049442252	AG-527	chembl:CHEMBL258767	CHEMBL:CHEMBL258767	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	DNDI1417368	chembl:CHEMBL2094652	CHEMBL:CHEMBL2094652	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.031536139	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	LEUCINE	rxcui:6308	LEUCINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	SJ000113107	chembl:CHEMBL589245	CHEMBL:CHEMBL589245	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	2,6-DIMETHOXYQUINONE	chembl:CHEMBL448515	2,6-DIMETHOXYQUINONE	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.1403948428761885	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.3017682254924971	TCMDC-125764	chembl:CHEMBL586670	CHEMBL:CHEMBL586670	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	PURVALANOLA	chembl:CHEMBL23327	PURVALANOLA	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007873395	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002956679	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.090530468	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	NSC-720622	chembl:CHEMBL1287980	CHEMBL:CHEMBL1287980	FALSE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.08334551	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	SB-431542	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	2.282942227638891	MANZAMINE A	chembl:CHEMBL403233	MANZAMINE A	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-123852	chembl:CHEMBL547656	CHEMBL:CHEMBL547656	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	MICONAZOLE NITRATE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-124328	chembl:CHEMBL532143	CHEMBL:CHEMBL532143	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000769366	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1312691780892362	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.026830696	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004889893	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004384042	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.050488145	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.2125816649218401	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.081533651	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.089298761	GNF-PF-5029	chembl:CHEMBL1198140	CHEMBL:CHEMBL1198140	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.019461702	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.015930725	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	CEAROIN	chembl:CHEMBL1613209	CEAROIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	BARDOXOLONE METHYL	ncit:C98250	BARDOXOLONE METHYL	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.056097939	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.050488145	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.1628144844517658	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	DTC	9/2/20	NULL	0.012154554	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.6908904109959803	NAKIJIQUINONE I	chembl:CHEMBL499609	NAKIJIQUINONE I	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.086361301	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.090064616	AURIN	chembl:CHEMBL210868	AURIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.035890411	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.020117882	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	1.591141552596803	LICARIN A	chembl:CHEMBL463526	LICARIN A	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001531729	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.031612084	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.045265234	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.023420014	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.009031247	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124617	chembl:CHEMBL582767	CHEMBL:CHEMBL582767	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	GW405833	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.039960176	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.008217163	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.3281729452230906	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	0.3671865121377238	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.030527716	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	DNDI1417701	chembl:CHEMBL1326164	CHEMBL:CHEMBL1326164	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.08178765	ALACHLOR	chembl:CHEMBL1414154	ALACHLOR	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	NSC-699479	chembl:CHEMBL1701915	CHEMBL:CHEMBL1701915	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-7387	chembl:CHEMBL119878	CHEMBL:CHEMBL119878	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	HELIOMYCIN	ncit:C75147	HELIOMYCIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.011810092	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	0.091796628	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004829624	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	COLCHICEINE	rxcui:2174385	COLCHICEINE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.029170928	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	1.640864726115453	XR-9577	chembl:CHEMBL428402	CHEMBL:CHEMBL428402	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	OXYPHENBUTAZONE	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.2019525816757481	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	QUISQUALATE	drugbank:DB02999	QUISQUALIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	CEPHARANTHINE	ncit:C83611	CEPHARANTHINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.019447286	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
PARP3	hgnc:273	PARP3	DTC	9/2/20	NULL	8.751278539282415	KU-0058948	drugbank:DB08058	4-[3-(1,4-DIAZEPAN-1-YLCARBONYL)-4-FLUOROBENZYL]PHTHALAZIN-1(2H)-ONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	DNDI1417268	chembl:CHEMBL1517542	CHEMBL:CHEMBL1517542	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.029465584	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.034590034	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.039068208	2-CHLORO-ADENOSINETRIPHOSPHATE	iuphar.ligand:1716	2-CHLOROADENOSINE-5-TRIPHOSPHATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-124552	chembl:CHEMBL547245	CHEMBL:CHEMBL547245	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	SJ000244621	chembl:CHEMBL600175	CHEMBL:CHEMBL600175	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.001620607	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002330153	FLUFENAMIC ACID	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	APAZONE	rxcui:1029	APAZONE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016959842	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
PRKAB2	hgnc:9379	PRKAB2	DTC	9/2/20	NULL	1.077080435603989	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.084146909	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	SPIPERONE	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	3.000438356	TCMDC-124242	chembl:CHEMBL529177	CHEMBL:CHEMBL529177	FALSE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	DTC	9/2/20	NULL	3.182283105193606	3-(DIMETHYLAMINO)BUTYL 3-PHENYLPROPYLCARBAMATE	chembl:CHEMBL448084	CHEMBL:CHEMBL448084	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.010195664	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012977675	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	DTC	9/2/20	NULL	0.3500511415712966	SILIBININ	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.00679975	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.020399251	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006193403	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
PRKAG3	hgnc:9387	PRKAG3	DTC	9/2/20	NULL	5.000730593875666	SAPONARIN	chembl:CHEMBL538921	SAPONARIN	FALSE	FALSE	FALSE
PRKAB2	hgnc:9379	PRKAB2	DTC	9/2/20	NULL	3.000438356325399	SAPONARIN	chembl:CHEMBL538921	SAPONARIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.009368006	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	SJ000001516	chembl:CHEMBL592316	CHEMBL:CHEMBL592316	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	TCMDC-125298	chembl:CHEMBL581152	CHEMBL:CHEMBL581152	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.1201548540862574	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	7,8-DIHYDROXYFLAVONE	chembl:CHEMBL75267	7,8-DIHYDROXYFLAVONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	OCTOCRYLENE	rxcui:77674	OCTOCRYLENE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-223133	chembl:CHEMBL1888586	CHEMBL:CHEMBL1888586	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.007537708	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.01535312	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	SB-431542	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	DTC	9/2/20	NULL	0.045579576	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-4156	chembl:CHEMBL585279	CHEMBL:CHEMBL585279	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	L-161982	iuphar.ligand:1952	L-161,982 (EP4A)	FALSE	FALSE	FALSE
ADCY5	hgnc:236	ADCY5	DTC	9/2/20	NULL	26.25383561784724	NSC-270718	chembl:CHEMBL401844	CHEMBL:CHEMBL401844	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	CGP-7930	iuphar.ligand:1079	CGP7930	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.00679975	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	ADENINE	rxcui:290	ADENINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	CID 670282	chembl:CHEMBL260213	CHEMBL:CHEMBL260213	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.035358701	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	CHLOROXURON	chembl:CHEMBL1568699	CHLOROXURON	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001988927	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ALAPROCLATE	ncit:C72685	ALAPROCLATE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.019447286	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	WAY-629	chembl:CHEMBL258465	CHEMBL:CHEMBL258465	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1988926940746003	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.025827679	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	QUISQUALATE	drugbank:DB02999	QUISQUALIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.026372512	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.2397610558707511	GAMBOGIC AMIDE	chembl:CHEMBL444109	GAMBOGIC AMIDE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.760980743	TALMAPIMOD	ncit:C79841	TALMAPIMOD	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.08178765	CAMPHOR	rxcui:1297880	CAMPHOR OIL	TRUE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.019889269	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.087952548	SULOCHRIN	chembl:CHEMBL61133	SULOCHRIN	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	GNF-PF-1211	chembl:CHEMBL600968	CHEMBL:CHEMBL600968	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	NCG-C00094421-01	chembl:CHEMBL553503	CHEMBL:CHEMBL553503	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.4167275494896389	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.099446347	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	RESCINNAMINE	rxcui:9259	RESCINNAMINE	TRUE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.047518255	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	CEPHARANTHINE	ncit:C83611	CEPHARANTHINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.020737627	TCMDC-139459	chembl:CHEMBL86464	CHEMBL:CHEMBL86464	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-663	chembl:CHEMBL596847	CHEMBL:CHEMBL596847	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	QUINOXALINE1	iuphar.ligand:5947	CDK1/5 INHIBITOR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	LOTEPREDNOL ETABONATE	rxcui:237027	LOTEPREDNOL	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.5834185692854944	GNF-PF-52	chembl:CHEMBL601142	CHEMBL:CHEMBL601142	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	SJ000124275	chembl:CHEMBL602150	CHEMBL:CHEMBL602150	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SJ000029259	chembl:CHEMBL592558	CHEMBL:CHEMBL592558	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.041672755	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.018501646	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	DIMETHYLPINOCEMBRIN	chembl:CHEMBL107131	DIMETHYLPINOCEMBRIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ESCULIN	rxcui:1314351	ESCULIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NSC-117079	chembl:CHEMBL471225	CHEMBL:CHEMBL471225	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.009115915	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.1145205479513511	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	AM-630	iuphar.ligand:750	AM-630	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.021554873	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	ENOXAMAST	ncit:C72586	ENOXAMAST	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.069824031	TRANSTORINE	iuphar.ligand:2918	KYNURENIC ACID	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1902451856365742	DICHLORODIPHENYLDICHLOROETHYLENE	chembl:CHEMBL363207	DICHLORODIPHENYLDICHLOROETHYLENE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	DNDI1417599	chembl:CHEMBL2094833	CHEMBL:CHEMBL2094833	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	TANSHINONE IIA	chembl:CHEMBL187266	TANSHINONE IIA	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.1268301237577161	MESO-HEXESTROL	drugbank:DB07931	HEXESTROL	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	TERBUTALINE SULFATE	rxcui:10369	TERBUTALINE SULFATE	TRUE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.1193356164447602	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	TOREMIFENE CITRATE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	MEFLOQUINE HYDROCHLORIDE	rxcui:82130	MEFLOQUINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	MESO-HEXESTROL	drugbank:DB07931	HEXESTROL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.2651902587661338	N-ACETYLCOLCHINOL	chembl:CHEMBL486504	N-ACETYLCOLCHINOL	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.044763573	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.016377939	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007479725	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-278538	chembl:CHEMBL275200	CHEMBL:CHEMBL275200	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	ALLOXAN	rxcui:2466730	ALLOXAN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004501686	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	ZERANOL	rxcui:1368476	ZERANOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	TCMDC-125066	chembl:CHEMBL533577	CHEMBL:CHEMBL533577	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	COLCHICEINE	rxcui:2174385	COLCHICEINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	(S)-NITRENDIPINE	chembl:CHEMBL251230	(S)-NITRENDIPINE	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.095295229	ONDANSETRON HYDROCHLORIDE	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2616661357260523	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	SJ000114741	chembl:CHEMBL591370	CHEMBL:CHEMBL591370	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	THEONELLASTEROL F	chembl:CHEMBL1782581	THEONELLASTEROL F	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.2917092846427472	PTEROSTILBENE	ncit:C153353	PTEROSTILBENE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	CID 1225609	chembl:CHEMBL444376	CHEMBL:CHEMBL444376	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.008334551	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	DTC	9/2/20	NULL	0.4167275494896389	NECA	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	NSC-60339	chembl:CHEMBL1448793	CHEMBL:CHEMBL1448793	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	DTC	9/2/20	NULL	2.917092846427472	NAPHTHALENE-1,2-DIOL	drugbank:DB07610	1,2-DIHYDROXYNAPHTHALENE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	COLCHICEINE	rxcui:2174385	COLCHICEINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	GNF-PF-1872	chembl:CHEMBL600103	CHEMBL:CHEMBL600103	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.013695272	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1861974157294131	DITOLYLGUANIDINE	iuphar.ligand:6684	1,3-DITOLYLGUANIDINE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	CCT241161	iuphar.ligand:9814	CCT241161	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	BENZOQUINONE	iuphar.ligand:6307	BENZOQUINONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	GNF-PF-1654	chembl:CHEMBL602776	CHEMBL:CHEMBL602776	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.012282496	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	DEQUALINIUM CHLORIDE	rxcui:3120	DEQUALINIUM CHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010569177	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.053038052	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.05454398	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.4118248724368196	DEXRAZOXANE	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	DILTIAZEM	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	2.700394520692859	Boceprevir	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	SJ000173328	chembl:CHEMBL591613	CHEMBL:CHEMBL591613	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	0.108711535	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.00591236	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.020741723	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.004216468	Iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.004660306	Ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.020257589	Prasugrel	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.022789788	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	FDA	10-Apr-24	NULL	0.097236428	Prasugrel	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
POLG	hgnc:9179	POLG	FDA	10-Apr-24	NULL	0.3070624048871023	Valproic Acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1245241215075758	Pramipexole	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.009327235	Vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.3337351985319565	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.034341185	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.2938862196027677	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.284980577	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	MyCancerGenome	20-Jun-17	inhibitor	1.521961485092594	ASP3026	ncit:C116727	ALK INHIBITOR ASP3026	FALSE	FALSE	TRUE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.019361236	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	MyCancerGenome	20-Jun-17	inhibitor	0.012534655	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	1.334940794127826	PF-03814735	drugbank:DB13059	PF-03814735	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.2083637747448194	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.1715936968486748	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.1607377690888607	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.079197091	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.2822993077187876	REMTOLUMAB	ncit:C152189	REMTOLUMAB	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.3704244884352345	CAL-101	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	MyCancerGenome	20-Jun-17	inhibitor	1.367387271762877	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
PRKCG	hgnc:9402	PRKCG	MyCancerGenome	20-Jun-17	inhibitor	0.1902451856365742	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:7633	iuphar.ligand:7633	VU0010010	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	MyCancerGenome	20-Jun-17	inhibitor	0.5303805175322677	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	1.282909942931453	LGX818	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.067231333	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.3697723326457359	APATINIB	hemonc:40	APATINIB	FALSE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenome	20-Jun-17	antibody	4.118248724368196	MM-121	chembl:CHEMBL2109402	MM-121	FALSE	TRUE	TRUE
VEGFA	hgnc:12680	VEGFA	MyCancerGenome	20-Jun-17	antibody	0.2019525816757481	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	modulator	1.500219178	IUPHAR.LIGAND:12545	iuphar.ligand:12545	MRS-1477	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.017059022	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	2.341819737097098	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1166837138570988	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3677319929494733	LAPATINIB DITOSYLATE	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	CLN-049	ncit:C185677	ANTI-FLT3/CD3 BISPECIFIC ANTIBODY CLN-049	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	2.407466349146467	AP26113	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.028498058	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1512704997187101	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	CRYSTAL VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.007873395	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.022439176	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02804897	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.182318303	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.546954909	SILYMARIN	rxcui:9794	SILYMARIN	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1912847768149162	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
SYNUCLEIN ALPHA	hgnc:11138	SNCA	TTD	2020.06.01	NULL	1.591141552596803	BIIB054	chembl:CHEMBL3833330	CINPANEMAB	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	0.030246354	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	0.4167275494896388	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	NCI	14-Sep-17	NULL	0.06714536	NDGA	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	MyCancerGenome	20-Jun-17	inhibitor	0.4055851016423223	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
APLN	hgnc:16665	APLN	NCI	14-Sep-17	NULL	13.12691780892362	CYCLOOXYGENASE INHIBITOR	ncit:C1323	CYCLOOXYGENASE INHIBITOR	FALSE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.11707396	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
ATIC	hgnc:794	ATIC	NCI	14-Sep-17	NULL	0.1875273972703374	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.2000292237550266	MEDROXYPROGESTERONE	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.3500511415712966	ADM	ncit:C186783	ACELLULAR DERMAL MATRIX	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.012501826	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.7001022831425933	NFX	ncit:C677	NAFOXIDINE	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	0.2625383561784725	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
NCBIGENE:1271	hgnc:2170	CNTFR	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:5217	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.1250182648468916	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
CCL22	hgnc:10621	CCL22	NCI	14-Sep-17	NULL	4.375639269641208	EOTAXIN	ncit:C1531	RECOMBINANT EOTAXIN	FALSE	FALSE	FALSE
CCNA2	hgnc:1578	CCNA2	NCI	14-Sep-17	NULL	0.3454452054979901	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.5173169579871378	ANTI CD3	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.3860858179095183	PROPANIDID	rxcui:8758	PROPANIDID	TRUE	FALSE	FALSE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	0.4861821410712454	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	5.250767123569449	CTLA4-IG	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002258977	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
CDH1	hgnc:1748	CDH1	NCI	14-Sep-17	NULL	6.563458904461812	PROTEOLYTIC ENZYMES	ncit:C38728	PANCREATIC PROTEOLYTIC ENZYMES	FALSE	FALSE	FALSE
CDC42	hgnc:1736	CDC42	NCI	14-Sep-17	NULL	4.375639269641208	GNRH	chembl:CHEMBL1200511	GONADORELIN ACETATE	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	0.4070362111294147	EOTAXIN	ncit:C1531	RECOMBINANT EOTAXIN	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	1.129197231	DTPA	rxcui:3690	PENTETIC ACID	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.085009721	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.1363835616511545	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.072026984	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	1.166837138570989	NORETHINDRONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	11.66837138570988	GOSSYPOL ACETIC ACID	ncit:C1118	GOSSYPOL ACETIC ACID	FALSE	FALSE	FALSE
CHAT	hgnc:1912	CHAT	NCI	14-Sep-17	NULL	0.2991890098899971	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
CETP	hgnc:1869	CETP	NCI	14-Sep-17	NULL	0.1242785118004603	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1132444383228493	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
CHAT	hgnc:1912	CHAT	NCI	14-Sep-17	NULL	0.6141248097742047	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2B	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.182318303	BHT	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.018071819	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.006909813	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.4487835148349958	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.010685322	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
EDNRB	hgnc:3180	EDNRB	NCI	14-Sep-17	NULL	0.069454592	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.9723642821424906	NORETHISTERONE ACETATE	rxcui:31983	NORETHINDRONE ACETATE	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.078722146	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.3677319929494733	GW2016	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.026572708	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.012561644	SUBEROYLANILIDE HYDROXAMIC ACID	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.1508841127462485	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.2651902587661338	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	METHAPYRILENE	rxcui:6822	METHAPYRILENE	FALSE	FALSE	FALSE
FOXO1	hgnc:3819	FOXO1	NCI	14-Sep-17	NULL	1.750255707856483	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
UNIPROT:Q04609	hgnc:3788	FOLH1	TEND	1-Aug-11	NULL	2.917092846427472	CAPROMAB	ncit:C174682	CAPROMAB	TRUE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	NCI	14-Sep-17	NULL	0.3889457128569963	ANTIESTROGENS	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	NCI	14-Sep-17	NULL	0.1023541349623674	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	NCI	14-Sep-17	NULL	0.1682938180631234	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.043756393	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.095468493	PROGESTOGENS	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1389091831632129	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1041818873724097	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	1.250182648468916	PCB	rxcui:66925	PROCARBAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.062509132	RU 486	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	IODOPHENPROPIT	iuphar.ligand:1266	IODOPHENPROPIT	FALSE	FALSE	FALSE
HIST3H2A	hgnc:20507	H2AC25	NCI	14-Sep-17	NULL	7.876150685354174	GNRH	chembl:CHEMBL1200511	GONADORELIN ACETATE	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.6141248097742047	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.7955707762984013	ALPRENOLOL	rxcui:597	ALPRENOLOL	FALSE	FALSE	FALSE
HP	hgnc:5141	HP	NCI	14-Sep-17	NULL	0.31919557	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1436598392221464	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1744440904840348	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.05309168	NDGA	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.093931433	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	NCI	14-Sep-17	NULL	0.3365876361262467	INTERFERONS	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	NCI	14-Sep-17	NULL	13.12691780892362	GRANULOCYTE MACROPHAGE COLONY-STIMULATING FACTOR	ncit:C1288	RECOMBINANT GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.2083637747448194	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.1022544717345559	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	PALMITIC ACID	rxcui:1370621	PALMITATE	TRUE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.1417211099478934	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.1389091831632129	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	4.039051633514961	BUSERELIN	rxcui:1825	BUSERELIN	TRUE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	7.501095891	IMMUNOLOGICAL ADJUVANT	ncit:C210	IMMUNOADJUVANT	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.2083637747448194	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.070860555	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.2059124362184098	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.039598545	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
IL5	hgnc:6016	IL5	NCI	14-Sep-17	NULL	0.8334550989792776	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.2386712328895204	GW632580X	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
IL6R	hgnc:6019	IL6R	NCI	14-Sep-17	NULL	0.067883221	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	1.29648571	ALUMINUM HYDROXIDE	rxcui:612	ALUMINUM HYDROXIDE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.038131933	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.5527123287967842	IMMUNOMODULATORS	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
IL7	hgnc:6023	IL7	NCI	14-Sep-17	NULL	0.3070624048871023	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.3241214273808302	BIOFLAVONOID	ncit:C306	BIOFLAVONOID	FALSE	FALSE	FALSE
IL7	hgnc:6023	IL7	NCI	14-Sep-17	NULL	1.944728564284981	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.012004497	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	1.381780822	CLOMIPHENE CITRATE	rxcui:142431	CLOMIPHENE CITRATE	TRUE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.8607814956671229	PDGF-BB	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
LTF	hgnc:6720	LTF	NCI	14-Sep-17	NULL	8.751278539282415	BACITRACIN	rxcui:1291	BACITRACIN	TRUE	FALSE	FALSE
LPO	hgnc:6678	LPO	NCI	14-Sep-17	NULL	0.6364566210387212	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.042741287	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P53350	hgnc:9077	PLK1	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	TKM-PLK1	ncit:C116889	LIPID ENCAPSULATED ANTI-PLK1 SIRNA TKM-PLK1	FALSE	FALSE	FALSE
MBP	hgnc:6925	MBP	NCI	14-Sep-17	NULL	3.750547945	BIOFLAVONOID	ncit:C306	BIOFLAVONOID	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.032899543	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	3.182283105193606	G207	hemonc:34886	G207	FALSE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.5250767123569451	LUPRON	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.056581542	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	1.750255707856483	TENECTEPLASE	rxcui:259280	TENECTEPLASE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	0.035927247	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.045461187	6-TG	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	0.6563458904461813	C-1311	chembl:CHEMBL338604	C-1311	FALSE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.061737415	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.075010959	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
NEUROD1	hgnc:7762	NEUROD1	NCI	14-Sep-17	NULL	0.9460841664089098	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.062958838	NEUROPROTECTIVE AGENT	ncit:C1509	NEUROPROTECTIVE AGENT	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.087005255	ANTIBIOTICS	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.054781086	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.047712559	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.052824619	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.054781086	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1643432589536604	IL-1RA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	agonist	0.021422958	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.3547815624033412	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.1892168332817819	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.2282942227638891	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.1988926940746004	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.3684748858645228	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.096167896	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.1223955040459079	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.049864835	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.08780547	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
OSM	hgnc:8506	OSM	NCI	14-Sep-17	NULL	10.50153425	IL-10	iuphar.ligand:4975	IL-10	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.1198805279353755	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.048618214	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.040515178	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	MELOXICAM	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.026885648	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.2778183663264258	I3C	ncit:C1135	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.2423430980108976	ACTIVIN	ncit:C2689	IH636 GRAPE SEED PROANTHOCYANIDIN EXTRACT	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.073437302	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.100976291	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
PRKAR2B	hgnc:9392	PRKAR2B	NCI	14-Sep-17	NULL	3.889457128569963	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.4861821410712453	BACITRACIN	rxcui:1291	BACITRACIN	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.076765601	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1325951293830669	DFMO	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.015036561	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.024861587	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
PSMD4	hgnc:9561	PSMD4	NCI	14-Sep-17	NULL	0.7501095890813501	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.012573676	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
PSMD7	hgnc:9565	PSMD7	NCI	14-Sep-17	NULL	0.8751278539282418	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	NCI	14-Sep-17	NULL	1.500219178	IL-10	iuphar.ligand:4975	IL-10	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.045898314	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
PTHLH	hgnc:9607	PTHLH	NCI	14-Sep-17	NULL	0.5147810905460245	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
PTHLH	hgnc:9607	PTHLH	NCI	14-Sep-17	NULL	1.591141552596803	DIFFERENTIATION AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	2.917092846427472	GM-CSF/IL-3 FUSION PROTEIN	ncit:C1477	MILODISTIM	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.1666910197958555	ANTIESTROGENS	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.019776901	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RAB5A	hgnc:9783	RAB5A	NCI	14-Sep-17	NULL	10.50153425	HGF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.4953553890159858	SIGNAL TRANSDUCTION INHIBITORS	ncit:C2189	SIGNAL TRANSDUCTION INHIBITOR	FALSE	FALSE	FALSE
RPE65	hgnc:10294	RPE65	NCI	14-Sep-17	NULL	0.7259125055625967	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.5147810905460244	NORETHISTERONE ACETATE	rxcui:31983	NORETHINDRONE ACETATE	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.1187956362798518	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	1.029562181092048	CETRORELIX	rxcui:68147	CETRORELIX	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.3088686543276147	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.1250182648468916	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	NCI	14-Sep-17	NULL	0.1546617709446082	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
TFAP2A	hgnc:11742	TFAP2A	NCI	14-Sep-17	NULL	1.166837138570988	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
TGFBR3	hgnc:11774	TGFBR3	NCI	14-Sep-17	NULL	2.625383561784725	TGF-BETA 2	ncit:C1286	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA-2	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.088996053	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1047012387551236	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	1.250182648468916	ACTH	iuphar.ligand:1331	ACTH	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.2991890098899971	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.9376369863516875	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.075442056	BROMODEOXYURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.015454797	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.028977744	PUROMYCIN	ncit:C787	PUROMYCIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.006439499	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.023182195	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.025757994	SELECTIVE ESTROGEN RECEPTOR MODULATORS	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.082624188	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
TPK1	hgnc:17358	TPK1	NCI	14-Sep-17	NULL	52.50767123569449	ANTIMETABOLITE	ncit:C272	ANTIMETABOLITE	FALSE	FALSE	FALSE
TRH	hgnc:12298	TRH	NCI	14-Sep-17	NULL	0.9131768910555564	ERYTHRO	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.2031244535229961	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.027584802	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.2234368988752957	INTERFERON GAMMA	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
UGCG	hgnc:12524	UGCG	NCI	14-Sep-17	NULL	0.5527123287967842	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	NCI	14-Sep-17	NULL	0.1342907192728759	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.2482632209725508	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.080781033	TAM	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
UCP2	hgnc:12518	UCP2	NCI	14-Sep-17	NULL	3.500511415712967	INTRALIPID	rxcui:1309980	SOYBEAN SEED OIL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.005145289	TAM	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.006026014	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.005145289	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	0.3454452054979901	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.167488584	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.1579178082276526	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	PharmGKB	4/5/24	NULL	0.1767935058440892	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
STXBP2	hgnc:11445	STXBP2	PharmGKB	4/5/24	NULL	13.12691780892362	emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	PharmGKB	4/5/24	NULL	15.75230137070834	fluindione	rxcui:50097	FLUINDIONE	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	0.1400204566285186	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	PharmGKB	4/5/24	NULL	0.3231241306811969	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.1235474617310458	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.01151484	nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
SRP19	hgnc:11300	SRP19	PharmGKB	4/5/24	NULL	1.050153425	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.1367387271762877	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
CYB5R1	hgnc:13397	CYB5R1	PharmGKB	4/5/24	NULL	0.9546849315580819	isosorbide dinitrate	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.2344092465879218	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.026240715	dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.018860514	dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1032599237673441	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.029041854	spironolactone	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	PharmGKB	4/5/24	NULL	1.458546423213736	cotinine	ncit:C70941	COTININE	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	PharmGKB	4/5/24	NULL	0.2083637747448194	emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.525076712	sulfadiazine	rxcui:10171	SULFADIAZINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.010848692	norethindrone	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.010678802	propafenone	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
MDGA2	hgnc:19835	MDGA2	PharmGKB	4/5/24	NULL	2.692701089009974	fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
ARVCF	hgnc:728	ARVCF	PharmGKB	4/5/24	NULL	0.1630673019742065	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.8204323630577265	diflomotecan	ncit:C90824	DIFLOMOTECAN	FALSE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.1342907192728759	vinblastine	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003454907	vinblastine	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
HCN1	hgnc:4845	HCN1	PharmGKB	4/5/24	NULL	2.187819634820604	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.1172046232939609	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
MECP2	hgnc:6990	MECP2	PharmGKB	4/5/24	NULL	4.375639269641208	trofinetide	rxcui:2632852	TROFINETIDE	TRUE	FALSE	FALSE
SLC26A8	hgnc:14468	SLC26A8	PharmGKB	4/5/24	NULL	1.875273972703374	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.021301287	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
NT5C1A	hgnc:17819	NT5C1A	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
MYO1H	hgnc:13879	MYO1H	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
HLA-DRA	hgnc:4947	HLA-DRA	PharmGKB	4/5/24	NULL	1.666910197958555	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
CEL	hgnc:1848	CEL	NCI	14-Sep-17	NULL	0.300043836	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
SCN2A	hgnc:10588	SCN2A	PharmGKB	4/5/24	NULL	0.1389091831632129	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.2051080907644316	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
GATA4	hgnc:4173	GATA4	PharmGKB	4/5/24	NULL	3.500511415712967	acenocoumarol	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
FXR2	hgnc:4024	FXR2	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
FARP2	hgnc:16460	FARP2	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
ETFDH	hgnc:3483	ETFDH	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
OPCML	hgnc:8143	OPCML	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.1620607136904151	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ZNF134	hgnc:12918	ZNF134	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
PIGM	hgnc:18858	PIGM	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	1.944728564284981	FENCAMFAMINE	ncit:C87695	FENCAMFAMIN	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	PharmGKB	4/5/24	NULL	0.041639708	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
IL13	hgnc:5973	IL13	PharmGKB	4/5/24	NULL	0.4375639269641209	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.9546849315580819	timolol	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.2375912725597036	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
PLA2G4A	hgnc:9035	PLA2G4A	PharmGKB	4/5/24	NULL	0.2573905452730122	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.018184475	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.051604591	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
MYLIP	hgnc:21155	MYLIP	PharmGKB	4/5/24	NULL	1.909369863116163	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.027538988	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.095468493	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	0.1272913242077442	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CYSLTR1	hgnc:17451	CYSLTR1	PharmGKB	4/5/24	NULL	1.325951293830669	zafirlukast	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	PharmGKB	4/5/24	NULL	0.039778539	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
STAT4	hgnc:11365	STAT4	PharmGKB	4/5/24	NULL	0.8751278539282418	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
DTNBP1	hgnc:17328	DTNBP1	PharmGKB	4/5/24	NULL	0.2165264793224515	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.158394182	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.077387872	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	15.48613345200206	enflurane	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.019776901	progesterone	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.018081154	moclobemide	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
AQP4	hgnc:637	AQP4	PharmGKB	4/5/24	NULL	0.6908904109959803	inebilizumab	rxcui:2373950	INEBILIZUMAB-CDON	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	PharmGKB	4/5/24	NULL	0.039688338	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004794564	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	PharmGKB	4/5/24	NULL	0.1205533268166455	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	0.1346350544504987	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.022136455	chlorpheniramine	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	IMC-3C5	chembl:CHEMBL2109602	IMC-3C5	FALSE	FALSE	FALSE
PSORS1C2	hgnc:17199	PSORS1C2	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	agonist	0.7955707762984013	DESMOPRESSIN ACETATE	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
TRIB2	hgnc:30809	TRIB2	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
CFLAR	hgnc:1876	CFLAR	PharmGKB	4/5/24	NULL	0.4375639269641208	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.2059124362184098	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	BRL-52537	chembl:CHEMBL1256835	CHEMBL:CHEMBL1256835	FALSE	FALSE	FALSE
NOTCH4	hgnc:7884	NOTCH4	PharmGKB	4/5/24	NULL	0.5834185692854944	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
TSHZ2	hgnc:13010	TSHZ2	PharmGKB	4/5/24	NULL	3.500511415712966	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.2500365296937833	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.037081689	SB-224289	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	PharmGKB	4/5/24	NULL	0.039390601	propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.033148782	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	PharmGKB	4/5/24	NULL	0.09963505	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
ZNF816	hgnc:26995	ZNF816	PharmGKB	4/5/24	NULL	1.312691780892362	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.014668586	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.019577804	chlorzoxazone	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003670838	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.001468335	gabapentin	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003670838	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.1555782851427985	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
TACR3	hgnc:11528	TACR3	DTC	9/2/20	NULL	5.834185692854944	RO-4603325	chembl:CHEMBL2203705	CHEMBL:CHEMBL2203705	FALSE	FALSE	FALSE
NAT1	hgnc:7645	NAT1	PharmGKB	4/5/24	NULL	0.1325951293830669	mesalazine	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00903591	zolpidem	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.058832125	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	PharmGKB	4/5/24	NULL	0.1243602739792764	trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CCL25	hgnc:10624	CCL25	NCI	14-Sep-17	NULL	4.375639269641208	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	PharmGKB	4/5/24	NULL	0.1567393171214761	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.5385402178019949	TRANSFORMING GROWTH FACTOR-BETA 2	ncit:C1286	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA-2	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	PharmGKB	4/5/24	NULL	0.05056107	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CACNB2	hgnc:1402	CACNB2	PharmGKB	4/5/24	NULL	0.097962073	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.071225816	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.021697385	belzutifan	rxcui:2567226	BELZUTIFAN	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2051080907644316	mephenytoin	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.2966535098061835	benazepril	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	PharmGKB	4/5/24	NULL	0.8325740682192574	futibatinib	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
UNIPROT:P55157	hgnc:7467	MTTP	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	SLX-4090	drugbank:DB05678	SLX-4090	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.088396753	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
CPOX	hgnc:2321	CPOX	PharmGKB	4/5/24	NULL	35.00511415712966	givosiran	rxcui:2265712	GIVOSIRAN	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	PharmGKB	4/5/24	NULL	0.1511209794852536	tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ALPL	hgnc:438	ALPL	PharmGKB	4/5/24	NULL	0.063916824	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.023612219	dacarbazine	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.009486481	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.1458546423213736	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.05073205	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.089756703	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
OAS1	hgnc:8086	OAS1	PharmGKB	4/5/24	NULL	0.921187215	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
ARID5B	hgnc:17362	ARID5B	PharmGKB	4/5/24	NULL	0.4667348554283955	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
GNMT	hgnc:4415	GNMT	PharmGKB	4/5/24	NULL	0.7778914257139925	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
IMPDH1	hgnc:6052	IMPDH1	PharmGKB	4/5/24	NULL	0.31115657	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.095122593	diltiazem	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	PharmGKB	4/5/24	NULL	0.2365210416022275	caffeine	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	PharmGKB	4/5/24	NULL	1.125164383622024	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
TRAT1	hgnc:30698	TRAT1	PharmGKB	4/5/24	NULL	1.082632396612257	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.098421127	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
EPM2A	hgnc:3413	EPM2A	PharmGKB	4/5/24	NULL	0.1546617709446082	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.090219366	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.012302641	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.3182283105193606	lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	2.902758237845518	caffeine	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.080327901	caffeine	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
DCK	hgnc:2704	DCK	PharmGKB	4/5/24	NULL	0.095122593	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
MEGF11	hgnc:29635	MEGF11	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CBR1	hgnc:1548	CBR1	PharmGKB	4/5/24	NULL	0.1470803115845784	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP4X1	hgnc:20244	CYP4X1	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.040112812	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
EXO1	hgnc:3511	EXO1	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.069332312	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
TCL1A	hgnc:11648	TCL1A	PharmGKB	4/5/24	NULL	3.088686543276147	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.03140411	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.006106608	thioridazine	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.2625383561784725	acetaminophen / codeine	wikidata:Q48566735	ACETAMINOPHEN / CODEINE	FALSE	FALSE	FALSE
TXNRD1	hgnc:12437	TXNRD1	PharmGKB	4/5/24	NULL	0.6731752722524936	vitamin c	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	PharmGKB	4/5/24	NULL	0.5250767123569451	varenicline	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
FTO	hgnc:24678	FTO	PharmGKB	4/5/24	NULL	0.4526523382387457	interferon alfa-2a, recombinant	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	0.2172731223545979	interferon alfa-2a, recombinant	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.044763573	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.045579576	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	PharmGKB	4/5/24	NULL	0.7501095890813501	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.032134438	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	NCI	14-Sep-17	NULL	0.3889457128569963	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
LMNA	hgnc:6636	LMNA	PharmGKB	4/5/24	NULL	1.944728564284981	lonafarnib	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	0.3977853881492006	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
MAGEA3	hgnc:6801	MAGEA3	TALC	12-May-16	vaccine	2.187819634820604	EP-2101	ncit:C26645	MULTI-NEO-EPITOPE VACCINE OSE 2101	FALSE	FALSE	TRUE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.1630673019742065	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.075550606	blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	OncoKB	23-Jul-20	NULL	0.128537751	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CD19	hgnc:1633	CD19	PharmGKB	4/5/24	NULL	0.5122699632750684	blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.052824619	SU-014813	chembl:CHEMBL1721885	SU-014813	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	0.8899605294185507	MLN 8237	hemonc:19	ALISERTIB	FALSE	FALSE	TRUE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:2026	iuphar.ligand:2026	BIM 23454	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	TALC	12-May-16	inhibitor	0.088396753	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	1.334940794127826	PF-03814735	drugbank:DB13059	PF-03814735	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.028766073	Leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
UNIPROT:P01375	hgnc:11892	TNF	TEND	1-Aug-11	NULL	0.068436196	ADALIMUMAB	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	1.790034246671403	ANTIHYPERTENSIVE DRUGS	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:5946	drugbank:DB07664	K-00546	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:7909	ncit:C116857	GANDOTINIB	FALSE	FALSE	TRUE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.082429625	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.2500365296937833	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	0.1682938180631233	R-flurbiprofen	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.0403388	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	3.962843112127886	DALOTUZUMAB	rxcui:1432293	DALOTUZUMAB	FALSE	TRUE	TRUE
ABL1	hgnc:76	ABL1	TALC	12-May-16	inhibitor	0.6241137025199848	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	HEXYLRESORCINOL	rxcui:5321	HEXYLRESORCINOL	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	Noberastine	ncit:C74582	NOBERASTINE	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.3906820776465364	AS-703026	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	1.000146118775133	AMG 208	ncit:C82677	C-MET INHIBITOR AMG 208	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MST1R	hgnc:7381	MST1R	TALC	12-May-16	inhibitor	0.6563458904461812	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5207	iuphar.ligand:5207	JZL184	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	TALC	12-May-16	antibody	0.2561349816375342	MDX-1106	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.035800685	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.1750255707856483	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	TALC	12-May-16	inhibitor	0.1618941559168381	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
SRC	hgnc:11283	SRC	TALC	12-May-16	inhibitor	0.4167275494896389	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2239	iuphar.ligand:2239	COMPOUND 37 [PMID: 16250654]	FALSE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	TALC	12-May-16	inhibitor	0.1325951293830669	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
CENPE	hgnc:1856	CENPE	TALC	12-May-16	inhibitor	17.50255707856483	GSK-923295	drugbank:DB06097	GSK-923295	FALSE	FALSE	TRUE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:3907	iuphar.ligand:3907	R3(B&DELTA;23-27)R/I5 CHIMERIC PEPTIDE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	TALC	12-May-16	inhibitor	2.341819737097098	GSK2118436	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
WEE1	hgnc:12761	WEE1	TALC	12-May-16	inhibitor	0.7212592202705288	MK-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.2243917574174978	4SC-202	drugbank:DB13101	4SC-202	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.086361301	AC480	ncit:C48380	PAN-HER KINASE INHIBITOR AC480	FALSE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.1325951293830669	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:Q01726	hgnc:6929	MC1R	TdgClinicalTrial	Jan-14	NULL	4.500657534488099	AFAMELANOTIDE	rxcui:2262250	AFAMELANOTIDE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.1268301237577161	AGN-214868	chembl:CHEMBL3137348	SENREBOTASE	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.1232574442152452	AGN-214868	chembl:CHEMBL3137348	SENREBOTASE	FALSE	FALSE	FALSE
UNIPROT:P48058	hgnc:4574	GRIA4	TdgClinicalTrial	Jan-14	NULL	0.596678082	BGG-492	chembl:CHEMBL3545042	SELURAMPANEL	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:3907	iuphar.ligand:3907	R3(B&DELTA;23-27)R/I5 CHIMERIC PEPTIDE	FALSE	FALSE	FALSE
UNIPROT:P49810	hgnc:9509	PSEN2	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	BMS-299897	chembl:CHEMBL247471	CHEMBL:CHEMBL247471	FALSE	FALSE	FALSE
ALCOHOL DEHYDROGENASE 1A	hgnc:249	ADH1A	TTD	2020.06.01	NULL	3.281729452230906	Fomepizole	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
UNIPROT:P49768	hgnc:9508	PSEN1	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	BMS-299897	chembl:CHEMBL247471	CHEMBL:CHEMBL247471	FALSE	FALSE	FALSE
UNIPROT:Q03431	hgnc:9608	PTH1R	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	PARATHYROID HORMONE	rxcui:1427222	PARATHYROID HORMONE	TRUE	FALSE	FALSE
UNIPROT:O00311	hgnc:1745	CDC7	TdgClinicalTrial	Jan-14	NULL	12.11715490054488	BMS-863233	drugbank:DB12357	BMS-863233	FALSE	FALSE	FALSE
UNIPROT:O00329	hgnc:8977	PIK3CD	TdgClinicalTrial	Jan-14	NULL	0.3704244884352345	CAL-101	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.3201687270469177	CHIDAMIDE	hemonc:99	CHIDAMIDE	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.030868707	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
UNIPROT:P49019	hgnc:16824	HCAR3	TdgClinicalTrial	Jan-14	NULL	1.875273972703374	NIACIN	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	CH-1504	chembl:CHEMBL4802141	CH-1504	FALSE	FALSE	FALSE
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	1.125164383622024	CNTO 1275	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	ESTROGEN	chembl:CHEMBL592868	ESTROGEN	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.1219218372345847	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
UNIPROT:P42684	hgnc:77	ABL2	TdgClinicalTrial	Jan-14	NULL	0.039341412	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	DARUSENTAN	ncit:C75991	DARUSENTAN	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	TALC	12-May-16	inhibitor	0.064268875	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P25942	hgnc:11919	CD40	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	DACETUZUMAB	ncit:C62179	DACETUZUMAB	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	0.6141248097742047	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	3.962843112127886	DALOTUZUMAB	rxcui:1432293	DALOTUZUMAB	FALSE	TRUE	TRUE
UNIPROT:P01019	hgnc:333	AGT	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	CYT006-ANGQB	drugbank:DB05739	CYT006-ANGQB	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.596678082	DAPOXETINE	ncit:C75168	DAPOXETINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
UNIPROT:P12931	hgnc:11283	SRC	TdgClinicalTrial	Jan-14	NULL	0.1136529680426287	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	DC-RTS-IL-12	ncit:C101789	ADENOVIRAL TRANSDUCED HIL-12-EXPRESSING AUTOLOGOUS DENDRITIC CELLS INXN-3001 PLUS ACTIVATOR LIGAND INXN-1001	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.067059606	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TdgClinicalTrial	Jan-14	NULL	0.4102161815288632	DILTIAZEM	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.069638821	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.063160791	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.061725319	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.060353645	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	0.5966780822238011	SILDENAFIL	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
UNIPROT:Q15761	hgnc:7958	NPY5R	TdgClinicalTrial	Jan-14	NULL	1.500219178	PEPTIDE YY	iuphar.ligand:1514	PEPTIDE YY	FALSE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.2941606231691568	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
UNIPROT:Q13698	hgnc:1397	CACNA1S	TdgClinicalTrial	Jan-14	NULL	0.1165542091802319	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.046343929	PRIMAQUINE PHOSPHATE	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
UNIPROT:P15559	hgnc:2874	NQO1	TdgClinicalTrial	Jan-14	NULL	2.019525817	EPI-743	chembl:CHEMBL1812161	VATIQUINONE	FALSE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	1.019566431761058	EPROTIROME	ncit:C81533	EPROTIROME	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.033701971	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.066297565	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.071148606	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	2.128689374420047	GEPIRONE	rxcui:2672253	GEPIRONE	TRUE	FALSE	FALSE
UNIPROT:Q70Z44	hgnc:24004	HTR3D	TdgClinicalTrial	Jan-14	NULL	0.3409589041278864	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
UNIPROT:P14151	hgnc:10720	SELL	TdgClinicalTrial	Jan-14	NULL	23.33674277141977	GMI-1070	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
UNIPROT:O95264	hgnc:5298	HTR3B	TdgClinicalTrial	Jan-14	NULL	0.280789686	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.5966780822238011	GW501516	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	3.424413341458336	GTS-21	drugbank:DB05708	GTS-21	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.048958202	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.2287915957982331	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.760980743	RETASPIMYCIN	ncit:C80378	RETASPIMYCIN	FALSE	FALSE	TRUE
UNIPROT:Q14568	hgnc:5256	HSP90AA2P	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	IPI-504	ncit:C48401	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.070010228	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.050007306	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.081830137	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.085147575	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	LOBELINE	rxcui:6464	LOBELINE	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.2386712328895204	LICOFELONE	ncit:C63957	LICOFELONE	FALSE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.1346350544504987	VORTIOXETINE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.1091635576625665	VORTIOXETINE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	0.034544521	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.020320306	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.011143394	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.02302968	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.009730851	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.018672714	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.051177067	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.020025809	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P33681	hgnc:1700	CD80	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	ABATACEPT	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
UNIPROT:Q8WXI7	hgnc:15582	MUC16	TdgClinicalTrial	Jan-14	NULL	22.50328767	OREGOVAMAB	ncit:C1784	OREGOVOMAB	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1491695205559502	OPC-14523	drugbank:DB05422	OPC-14523	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.025003653	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P50052	hgnc:338	AGTR2	TdgClinicalTrial	Jan-14	NULL	0.9546849315580819	PS433540	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
UNIPROT:P43155	hgnc:2342	CRAT	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
UNIPROT:P50416	hgnc:2328	CPT1A	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	PROPIONYL-L-CARNITINE	drugbank:DB15980	LEVOCARNITINE PROPIONATE	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.049723174	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.020351811	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
UNIPROT:Q8WXA8	hgnc:24003	HTR3C	TdgClinicalTrial	Jan-14	NULL	1.500219178	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.067231333	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.023813003	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
UNIPROT:Q8NER1	hgnc:12716	TRPV1	TdgClinicalTrial	Jan-14	NULL	0.7684049449126024	RESINIFERATOXIN	ncit:C1214	RESINIFERATOXIN	FALSE	FALSE	FALSE
UNIPROT:P43235	hgnc:2536	CTSK	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	RELACATIB	ncit:C66512	RELACATIB	FALSE	FALSE	FALSE
UNIPROT:P51787	hgnc:6294	KCNQ1	TdgClinicalTrial	Jan-14	NULL	0.6819178082557726	RETIGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.7395446652914718	RIDAFOROLIMUS	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.061340737	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	agonist	0.1469979597863787	PILOCARPINE HYDROCHLORIDE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P17326	hgnc:3541	F3	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	RECOMBINANT NEMATODE ANTICOAGULANT PROTEIN C2	chembl:CHEMBL4298082	RECOMBINANT NEMATODE ANTICOAGULANT PROTEIN C2	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.2263261691193728	RTA 744	drugbank:DB05920	RTA 744	FALSE	FALSE	FALSE
UNIPROT:P23280	hgnc:1380	CA6	TdgClinicalTrial	Jan-14	NULL	7.501095891	SAR566658	ncit:C95764	ANTI-CA6-DM4 IMMUNOCONJUGATE SAR566658	FALSE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	TETRAHYDROCANNABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
UNIPROT:P42336	hgnc:8975	PIK3CA	TdgClinicalTrial	Jan-14	NULL	0.027010119	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.02339914	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.1215455352678113	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.012695278	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.016126435	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:378	iuphar.ligand:378	PENECA	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.017352172	IUPHAR.LIGAND:5682	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	CILOSTAMIDE	ncit:C76315	CILOSTAMIDE	FALSE	FALSE	FALSE
UNIPROT:P50750	hgnc:1780	CDK9	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	FDA	10-Apr-24	NULL	0.1230648544586589	Efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
UNIPROT:Q9Y243	hgnc:393	AKT3	TdgClinicalTrial	Jan-14	NULL	0.6563458904461813	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
UNIPROT:P31749	hgnc:391	AKT1	TdgClinicalTrial	Jan-14	NULL	0.443726799	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
UNIPROT:P13631	hgnc:9866	RARG	TdgClinicalTrial	Jan-14	NULL	0.1357664414626878	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.2917092846427472	CC-1088	ncit:C2210	SELECTIVE CYTOKINE INHIBITORY DRUG CC-1088	FALSE	FALSE	FALSE
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.2778183663264258	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
SLCO1A2	hgnc:10956	SLCO1A2	PharmGKB	4/5/24	NULL	1.250182648468916	nadolol	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
PARP1	hgnc:270	PARP1	TALC	12-May-16	inhibitor	0.4296082192011368	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.272767123	Ketoprofen	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
UNIPROT:P00797	hgnc:9958	REN	TdgClinicalTrial	Jan-14	NULL	15.75230137070834	VTP-27999	drugbank:DB12416	VTP-27999	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 4	hgnc:1605	CCR4	TTD	2020.06.01	NULL	12.35474617310458	Mogamulizumab	rxcui:2054068	MOGAMULIZUMAB	TRUE	TRUE	TRUE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.080164384	POTASSIUM DICHROMATE	rxcui:8595	POTASSIUM DICHROMATE	FALSE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	NRP104	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	REMACEMIDE HYDROCHLORIDE	ncit:C152184	REMACEMIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q9NR97	hgnc:15632	TLR8	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	VTX-2337	ncit:C80521	MOTOLIMOD	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.2983390411119005	Dipivefrin	rxcui:23410	DIPIVEFRIN	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.058212496	IUPHAR.LIGAND:4360	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:1236	iuphar.ligand:1236	(R)-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
UNIPROT:P48736	hgnc:8978	PIK3CG	TdgClinicalTrial	Jan-14	NULL	0.089756703	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
NCBIGENE:1881	ncbigene:1881	EBM	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:5066	iuphar.ligand:5066	RANK LIGAND	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1109316997937207	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:P31751	hgnc:392	AKT2	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	XL418	drugbank:DB05204	XL418	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	activator	4.773424657790408	IUPHAR.LIGAND:12552	iuphar.ligand:12552	KS0365	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.026779381	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:3474	iuphar.ligand:1485	BIBP3226	FALSE	FALSE	FALSE
UNIPROT:O43570	hgnc:1371	CA12	TdgClinicalTrial	Jan-14	NULL	0.8036888454443035	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.4605936073306534	BENZOCAINE	rxcui:1399	BENZOCAINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	1.790034246671403	BENZONATATE	rxcui:18993	BENZONATATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.4189441853911795	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.1280674908187671	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.087222045	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.089298761	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.1535312024435511	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	ESTRIOL	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	FENOTEROL	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
UNIPROT:P32239	hgnc:1571	CCKBR	TdgClinicalTrial	Jan-14	NULL	3.580068493342807	PENTAGASTRIN	rxcui:7993	PENTAGASTRIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1352294697019358	KRT-232	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	NORSTICTIC ACID	chembl:CHEMBL228281	NORSTICTIC ACID	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.6105543166941221	PHENYLPROPANOLAMINE	rxcui:8175	PHENYLPROPANOLAMINE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.1615620653405984	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.072927321	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	0.138178082	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
UNIPROT:P22748	hgnc:1375	CA4	TEND	1-Aug-11	NULL	1.250182648468916	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P32239	hgnc:1571	CCKBR	TEND	1-Aug-11	NULL	3.580068493342807	PENTAGASTRIN	rxcui:7993	PENTAGASTRIN	TRUE	FALSE	FALSE
UNIPROT:Q9GZZ6	hgnc:13800	CHRNA10	TEND	1-Aug-11	NULL	0.4565884455277782	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1396480617970598	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	GEDUNIN	chembl:CHEMBL465226	GEDUNIN	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TEND	1-Aug-11	NULL	0.5357925636295356	ANTIHEMOPHILIC FACTOR	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.4861821410712453	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.1219218372345847	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.077827576	CABERGOLINE	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.068637479	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.075333818	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.064033745	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.2019525816757481	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.062509132	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.070956312	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.207267123	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.158793361	DIPHENHYDRAMINE	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TEND	1-Aug-11	NULL	1.193356164447602	GONADORELIN	rxcui:6384	GONADORELIN	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.6012328767445935	HYDROCORTAMATE	ncit:C65862	HYDROCORTAMATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.1250182648468916	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.2983390411119005	ISOETHARINE	rxcui:6023	ISOETHARINE	TRUE	FALSE	FALSE
UNIPROT:Q14432	hgnc:8778	PDE3A	TEND	1-Aug-11	NULL	0.251232877	AMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.2713574740862764	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TEND	1-Aug-11	NULL	0.7955707762984014	BEZAFIBRATE	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.1067229090156392	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.1041818873724097	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.097236428	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.5073204950308646	METHOXAMINE	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.054953083	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18031	hgnc:9642	PTPN1	TEND	1-Aug-11	NULL	1.400204566285186	TILUDRONATE	rxcui:11476	TILUDRONIC ACID	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.8950171233357017	PENBUTOLOL	rxcui:7973	PENBUTOLOL	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.1117184494376478	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.096967075	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.100976291	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TEND	1-Aug-11	NULL	0.1215455352678113	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.2019525816757481	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1875273972703375	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.2237542808339254	RANOLAZINE	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.062262061	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	0.5147810905460245	THC	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.4145342465975881	ROPIVACAINE	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.027347745	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
UNIPROT:P07101	hgnc:11782	TH	TEND	1-Aug-11	NULL	0.9616789603607051	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.2282942227638891	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.090634645	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.087318744	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.089501712	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P07202	hgnc:12015	TPO	TEND	1-Aug-11	NULL	8.751278539282415	CARBIMAZOLE	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.007496384	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
C1S	hgnc:1247	C1S	NCI	14-Sep-17	NULL	2.625383561784724	MBL	ncit:C1151	MANNOSE-BINDING LECTIN	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.2035181055647073	THIAMYLAL	rxcui:10464	THIAMYLAL	TRUE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TEND	1-Aug-11	NULL	3.043922970185188	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.056826484	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.036463661	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.083744292	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.061197752	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.054243462	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.053038052	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.044611445	TRIMIPRAMINE	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	TRIPELENNAMINE	rxcui:10847	TRIPELENNAMINE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.060423097	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TEND	1-Aug-11	NULL	3.281729452230906	VARDENAFIL	rxcui:306674	VARDENAFIL	TRUE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TEND	1-Aug-11	NULL	1.633571993999384	ZOLEDRONATE	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	1.265245090016735	AMG-191	chembl:CHEMBL2109325	AMG-191	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	0.8334550989792776	Trilaciclib	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.3571950424196904	Trilaciclib	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	GDC-0853	ncit:C116844	FENEBRUTINIB	FALSE	FALSE	FALSE
PPCDC	hgnc:28107	PPCDC	PharmGKB	4/5/24	NULL	0.5834185692854944	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NKG2 D ACTIVATING NK RECEPTOR	hgnc:18788	KLRK1	TTD	2020.06.01	NULL	13.12691780892362	NN8555	chembl:CHEMBL4594564	TESNATILIMAB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	CIViC	10-Apr-24	NULL	0.034830959	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	0.2333674277141977	Mavrilimumab	ncit:C95788	MAVRILIMUMAB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	1.009762908	BI-836880	drugbank:DB17484	BI-836880	FALSE	FALSE	FALSE
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	2.625383561784724	IMCgp100	rxcui:2590743	TEBENTAFUSP	TRUE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	1.875273972703375	PF-06840003	iuphar.ligand:9565	PF-06840003	FALSE	FALSE	FALSE
LEUKOCYTE COMMON ANTIGEN	hgnc:9666	PTPRC	TTD	2020.06.01	NULL	2.917092846427472	Iomab-B	ncit:C2527	IODINE I 131 APAMISTAMAB	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.4167275494896388	Ronomilast	ncit:C97274	RONOMILAST	FALSE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.4167275494896388	AMG 319	ncit:C95891	PI3K-DELTA INHIBITOR AMG 319	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	0.1442518440541057	PLX-3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	1.544343271638073	GNKG-168	chembl:CHEMBL4297962	GNKG-168	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.7395446652914718	BFH-772	chembl:CHEMBL4080062	BFH-772	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.1250182648468916	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	0.1093909817410302	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	3.443125982668491	MEDI-575	ncit:C82684	TOVETUMAB	FALSE	TRUE	TRUE
LEUKEMIA INHIBITORY FACTOR RECEPTOR	hgnc:6597	LIFR	TTD	2020.06.01	NULL	105.0153424713889	Emfilermin	ncit:C1384	EMFILERMIN	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.4145342465975881	MGAH22	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
ALDOSTERONE SYNTHASE	hgnc:2592	CYP11B2	TTD	2020.06.01	NULL	5.834185692854944	LCI699	rxcui:2286252	OSILODROSTAT	TRUE	FALSE	FALSE
OVARIAN CARCINOMA ANTIGEN CA125	hgnc:15582	MUC16	TTD	2020.06.01	NULL	22.50328767	Oregovomab	ncit:C1784	OREGOVOMAB	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR	hgnc:2438	CSF3	TTD	2020.06.01	NULL	17.50255707856483	Neugranin	ncit:C81936	RECOMBINANT HUMAN ALBUMIN-HUMAN GRANULOCYTE COLONY-STIMULATING FACTOR	FALSE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	15.75230137070834	VTP-27999	drugbank:DB12416	VTP-27999	FALSE	FALSE	FALSE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	1.193356164447602	Bismuth	rxcui:1599	BISMUTH	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.201952582	Midodrine	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA2.3	hgnc:6292	KCNN3	TTD	2020.06.01	NULL	3.281729452230906	dequalinium	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE BETA	hgnc:5960	IKBKB	TTD	2020.06.01	NULL	0.6250913242344582	Parthenolide	rxcui:32941	PARTHENOLIDE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 3	hgnc:10912	SLC12A3	TTD	2020.06.01	NULL	11.66837138570988	Polythiazide	rxcui:8565	POLYTHIAZIDE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.023060023	Aniracetam	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	1.117184494376478	A-85380	iuphar.ligand:5460	A-85380	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.5515511684421691	Tacrine	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 4	hgnc:11333	SSTR4	TTD	2020.06.01	NULL	1.750255707856483	ODT-8	chembl:CHEMBL452157	CHEMBL:CHEMBL452157	FALSE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 2	hgnc:11331	SSTR2	TTD	2020.06.01	NULL	0.5834185692854945	ODT-8	chembl:CHEMBL452157	CHEMBL:CHEMBL452157	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.1363835616511545	Phenylbutazone	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.3125456621172291	METHYLDOPATE HYDROCHLORIDE	rxcui:91241	METHYLDOPATE HYDROCHLORIDE	TRUE	FALSE	FALSE
AROMATIC-L-AMINO-ACID DECARBOXYLASE	hgnc:2719	DDC	TTD	2020.06.01	NULL	1.750255707856483	Vitamin B6	rxcui:42954	VITAMIN B6	TRUE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	0.4167275494896388	AMG 386	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.008647508	Methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.5000730593875666	CAPMATINIB HYDROCHLORIDE	rxcui:2362259	CAPMATINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-RAF	hgnc:9829	RAF1	TTD	2020.06.01	NULL	0.3365876361262467	Semapimod	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
INTERLEUKIN-10	hgnc:5962	IL10	TTD	2020.06.01	NULL	2.625383561784724	Ilodecakin	rxcui:2604685	ILODECAKIN	FALSE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	4.039051633514961	QR-333	drugbank:DB05533	QR-333	FALSE	FALSE	FALSE
LIVER CARBOXYLESTERASE	hgnc:1863	CES1	TTD	2020.06.01	NULL	0.760980743	K-604	iuphar.ligand:10150	K-604	FALSE	FALSE	FALSE
TYROSINE 3-MONOOXYGENASE	hgnc:11782	TH	TTD	2020.06.01	NULL	0.9616789603607051	Metyrosine	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.8514757497680189	SCH 420814	ncit:C76394	PRELADENANT	FALSE	FALSE	FALSE
RPL34	hgnc:10340	RPL34	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
VITAMIN K-DEPENDENT PROTEIN C	hgnc:9451	PROC	TTD	2020.06.01	NULL	15.75230137070834	Sodium Tetradecyl Sulfate	rxcui:9913	SODIUM TETRADECYL SULFATE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	1.790034246671403	Benzonatate	rxcui:18993	BENZONATATE	TRUE	FALSE	FALSE
LACTOTRANSFERRIN	hgnc:6720	LTF	TTD	2020.06.01	NULL	13.12691780892362	Talactoferrin	rxcui:1425932	TALACTOFERRIN ALFA	FALSE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.2	hgnc:6256	KCNJ10	TTD	2020.06.01	NULL	2.500365296937833	Mitiglinide	ncit:C81699	MITIGLINIDE	TRUE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.3241214273808302	Spiroglumide	ncit:C73219	SPIROGLUMIDE	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	0.06697407	Ibudilast	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 22 MEMBER 8	hgnc:10972	SLC22A8	TTD	2020.06.01	NULL	0.5357925636295356	FLUORESCEIN	rxcui:25138	FLUORESCEIN	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.070956312	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
UNIPROT:Q02641	hgnc:1401	CACNB1	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
NCBIGENE:128	hgnc:253	ADH5	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12944	iuphar.ligand:12944	NOX-6-18	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.6908904109959803	CP-724714	drugbank:DB12302	CP-724714	FALSE	FALSE	FALSE
IRON	hgnc:4650	GTF2E1	TTD	2020.06.01	NULL	1.312691780892362	Exjade	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:11190	ncit:C175876	VIMSELTINIB	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.088945801	Pardoprunox	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
INTERLEUKIN-15	hgnc:5977	IL15	TTD	2020.06.01	NULL	3.750547945	AMG-714	iuphar.ligand:13046	ORDESEKIMAB	FALSE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	0.9546849315580819	Pamidronate	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	Triprolidine	rxcui:10849	TRIPROLIDINE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.026071336	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 3	hgnc:1604	CCR3	TTD	2020.06.01	NULL	2.917092846427472	YM-355179	iuphar.ligand:793	YM-355179	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.3431873936973496	Methantheline	rxcui:6821	METHANTHELINE	TRUE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	5.000730593875666	Streptokinase	rxcui:10106	STREPTOKINASE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	GLIQUIDONE	rxcui:25793	GLIQUIDONE	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.089756703	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Bromodiphenhydramine	rxcui:19759	BROMODIPHENHYDRAMINE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE MER	hgnc:7027	MERTK	TTD	2020.06.01	NULL	0.4375639269641208	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	METHIXENE HYDROCHLORIDE	rxcui:258230	METHIXENE HYDROCHLORIDE	TRUE	FALSE	FALSE
MACROPHAGE-STIMULATING PROTEIN RECEPTOR	hgnc:7381	MST1R	TTD	2020.06.01	NULL	0.091159151	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
CASP14	hgnc:1502	CASP14	ChEMBL	33	inhibitor	4.039051633514962	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.025439763	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.9907107780319716	OSI-906	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	0.029918901	M100907	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.031254566	MGCD516	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
INTEGRIN ALPHA-2	hgnc:6137	ITGA2	TTD	2020.06.01	NULL	26.25383561784724	E7820	chembl:CHEMBL4297376	E-7820	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	7.876150685354174	PRO-140	ncit:C137824	LERONLIMAB	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.1315981735230438	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
THYROID HORMONE RECEPTOR ALPHA	hgnc:11796	THRA	TTD	2020.06.01	NULL	1.250182648468916	tiratricol	rxcui:13982	TIRATRICOL	FALSE	FALSE	FALSE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	0.169927739	tiratricol	rxcui:13982	TIRATRICOL	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.8078103267029922	ELND005	ncit:C122987	SCYLLITOL	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
PROTO-ONCOGENE MAS	hgnc:6899	MAS1	TTD	2020.06.01	NULL	8.751278539282415	Angiotensin-(1-7)	iuphar.ligand:582	ANGIOTENSIN-(1-7)	FALSE	FALSE	FALSE
DIHYDROOROTATE DEHYDROGENASE	hgnc:2867	DHODH	TTD	2020.06.01	NULL	5.527123287967842	Teriflunomide	rxcui:1310520	TERIFLUNOMIDE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.5000730593875666	MK-8033	chembl:CHEMBL2323775	MK-8033	FALSE	FALSE	FALSE
CFD	hgnc:2771	CFD	ChEMBL	33	inhibitor	17.50255707856483	DANICOPAN	ncit:C148181	DANICOPAN	FALSE	FALSE	FALSE
T-CELL DIFFERENTIATION ANTIGEN CD6	hgnc:1691	CD6	TTD	2020.06.01	NULL	52.50767123569449	Itolizumab	ncit:C95787	ITOLIZUMAB	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.3697723326457359	GDC-0349	drugbank:DB13072	GDC-0349	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	GTx-758	drugbank:DB14969	GTX-758	FALSE	FALSE	FALSE
FREE FATTY ACID RECEPTOR 2	hgnc:4501	FFAR2	TTD	2020.06.01	NULL	13.12691780892362	GLPG0974	iuphar.ligand:8417	GLPG0974	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.042174836	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 5	hgnc:14299	S1PR5	TTD	2020.06.01	NULL	6.563458904461812	ASP-4058	drugbank:DB11819	ASP-4058	FALSE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.284980577	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.2678962818147678	BAL-101553	ncit:C97664	LISAVANBULIN	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.2561349816375342	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	4.773424657790408	LCZ696	ncit:C162629	SACUBITRIL/VALSARTAN	FALSE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	4.375639269641208	PLEGRIDY	rxcui:1546168	PEGINTERFERON BETA-1A	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.079236928	PF-05212384	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.736088849	ARN-810	ncit:C106235	BRILANESTRANT	FALSE	FALSE	TRUE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.2263261691193728	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	3.424413341458336	CCX-140	ncit:C175798	ILACIRNON	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.8537832721251137	Spartalizumab	ncit:C121625	SPARTALIZUMAB	FALSE	FALSE	FALSE
PHENYLALANINE HYDROXYLASE	hgnc:8582	PAH	TTD	2020.06.01	NULL	8.751278539282415	Pegvaliase	rxcui:2046360	PEGVALIASE	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV7.3	hgnc:6297	KCNQ3	TTD	2020.06.01	NULL	3.750547945	XEN1101	ncit:C188540	AZETUKALNER	FALSE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	1.458546423213736	O-desulfated heparin	ncit:C99130	DOCIPARSTAT SODIUM	FALSE	FALSE	FALSE
PROLYL ENDOPEPTIDASE	hgnc:9358	PREP	TTD	2020.06.01	NULL	17.50255707856483	ONO-1603	chembl:CHEMBL1087333	CHEMBL:CHEMBL1087333	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	0.1930429089547591	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
UNIPROT:P19838	hgnc:7794	NFKB1	TdgClinicalTrial	Jan-14	NULL	0.138178082	THYMOSIN BETA-4	drugbank:DB12003	THYMOSIN BETA-4	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.08334551	Apremilast	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	3.424413341458336	TC-6987	drugbank:DB14854	TC-6987	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.400821918	Deflazacort	rxcui:22396	DEFLAZACORT	TRUE	FALSE	FALSE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	0.6731752722524935	Brodalumab	rxcui:1872251	BRODALUMAB	TRUE	FALSE	FALSE
IRON	hgnc:4650	GTF2E1	TTD	2020.06.01	NULL	0.6177373086552295	Deferoxamine Mesylate	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
TRIPEPTIDYL-PEPTIDASE I	hgnc:2073	TPP1	TTD	2020.06.01	NULL	157.5230137070835	Cerliponase Alfa	rxcui:1922436	CERLIPONASE ALFA	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.1219218372345847	Bupivacaine	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.06286838	Epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.1436598392221464	Etomidate	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	CIViC	10-Apr-24	NULL	0.9479406894984094	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.6012328767445935	Hydrocortamate	ncit:C65862	HYDROCORTAMATE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.061055432	Metharbital	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	2.100306849	Niraparib Tosylate	rxcui:2637447	NIRAPARIB TOSYLATE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.6105543166941221	Mebutamate	ncit:C66062	MEBUTAMATE	TRUE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	1.633571993999384	Zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	2.100306849	ABT-767	ncit:C96795	PARP-1/2 INHIBITOR ABT-767	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	Pelitinib	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
PROSTAGLANDIN E2 RECEPTOR EP3	hgnc:9595	PTGER3	TTD	2020.06.01	NULL	1.166837138570989	BUTAPROST	ncit:C74369	BUTAPROST	FALSE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.2051080907644316	Daclizumab	rxcui:190353	DACLIZUMAB	TRUE	TRUE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1556551518844698	Carphenazine	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.1539814405738841	Cinnarizine	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.075496292	Duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.445925021	Dihydrotachysterol	rxcui:3429	DIHYDROTACHYSTEROL	TRUE	FALSE	FALSE
INTERFERON ALPHA/BETA RECEPTOR 2	hgnc:5433	IFNAR2	TTD	2020.06.01	NULL	2.461297089173179	Interferon alfa-n1	rxcui:202912	INTERFERON ALFA-N1	FALSE	TRUE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.1893305453210138	Lurasidone hydrochloride	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.1848861663228679	Rilmenidine	rxcui:55679	RILMENIDINE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.6105543166941221	Stiripentol	rxcui:2054968	STIRIPENTOL	TRUE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.089756703	CUDC-907	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.6250913242344582	BPN14770	iuphar.ligand:10451	BPN14770	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.201952582	TG100-115	drugbank:DB05552	TG100-115	FALSE	FALSE	FALSE
GANGLIOSIDE GM2 ACTIVATOR	hgnc:4367	GM2A	TTD	2020.06.01	NULL	3.281729452230906	BIW-8962	chembl:CHEMBL2109426	BIW-8962	FALSE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	0.5147810905460244	Eltoprazine	ncit:C73286	ELTOPRAZINE	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	2.100306849	INO-1001	ncit:C61315	INO-1001	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	4.039051633514961	Lanabecestat	ncit:C170091	LANABECESTAT	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.071585127259071	Semuloparin	rxcui:2368733	SEMULOPARIN	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.7395446652914718	Ridaforolimus	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.071585127259071	SSR-126517E	drugbank:DB05362	SSR-126517E	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.1131630845596864	IUPHAR.LIGAND:8435	iuphar.ligand:8435	LP-44	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.026626608	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.016764901	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.090374649	IUPHAR.LIGAND:15	iuphar.ligand:15	L-694,247	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.039068208	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.6863747873946993	CC-292	ncit:C97037	SPEBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:126	iuphar.ligand:126	(+)-WAY 100135	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.065716735	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:123	iuphar.ligand:123	LYSERGOL	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:207	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:8430	iuphar.ligand:8430	[11C]GSK215083	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:192	iuphar.ligand:192	SB 228357	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.019844169	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.03251249	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.02271093	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.011277421	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3244	iuphar.ligand:3244	[11C]SB207145	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:782	hgnc:1401	CACNB1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8802	iuphar.ligand:8802	ESTRADIOL DISULFATE	FALSE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	MyCancerGenome	20-Jun-17	inhibitor	0.033232703	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.2518353536484148	IUPHAR.LIGAND:11191	ncit:C174748	VODOBATINIB	FALSE	FALSE	FALSE
NCBIGENE:1263	hgnc:2154	PLK3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12243	iuphar.ligand:12243	CP-640186	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:1279	hgnc:2199	COL1AR	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:944	iuphar.ligand:944	SKF-83566	FALSE	FALSE	FALSE
NCBIGENE:3070	hgnc:4861	HELLS	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10250	iuphar.ligand:10250	DO264	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:6663	iuphar.ligand:6663	&RHO;-DA1A	FALSE	FALSE	FALSE
NCBIGENE:1921	hgnc:19679	AAK1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10403	iuphar.ligand:10403	COMPOUND 21B [PMID: 31136173]	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:11837	iuphar.ligand:11837	COMPOUND 14A [PMID: 34795866]	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:6453	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.9211872146613068	IUPHAR.LIGAND:10307	ncit:C65409	DIMINAZENE	FALSE	FALSE	FALSE
NCBIGENE:685	hgnc:1121	BTC	GuideToPharmacology	2024.1	blocker	0.5966780822238011	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:4292	iuphar.ligand:4292	PSALMOTOXIN 1	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:10308	iuphar.ligand:10308	MAMBALGIN-1	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.5527123287967842	IUPHAR.LIGAND:4186	iuphar.ligand:4186	ETHYLISOPROPYLAMILORIDE	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	modulator	0.6035364509849942	IUPHAR.LIGAND:8895	iuphar.ligand:8895	VPC171	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:10351	iuphar.ligand:10351	LUF7602	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:5616	iuphar.ligand:5616	ATL802	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:393	iuphar.ligand:393	MRS1042	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:392	iuphar.ligand:392	MRS1041	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.018699313	IUPHAR.LIGAND:413	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:411	iuphar.ligand:411	MORIN	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.2273059360852575	IUPHAR.LIGAND:423	iuphar.ligand:423	N(6)-CYCLOHEXYLADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:5368	iuphar.ligand:5368	ANGIOTENSIN IV	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10354	iuphar.ligand:10354	ELIMUSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8477	iuphar.ligand:8477	AZ20	FALSE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.013505059	IUPHAR.LIGAND:9381	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:5930	iuphar.ligand:5930	AURORA KINASE INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:8190	iuphar.ligand:8190	COMPOUND 1 [PMID: 21742770]	FALSE	FALSE	FALSE
NCBIGENE:2901	hgnc:4583	GRIK5	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9561	ncit:C170396	ZIRITAXESTAT	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:7953	iuphar.ligand:7953	BMS-777607	FALSE	FALSE	TRUE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:621	iuphar.ligand:621	PD 168368	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7852	iuphar.ligand:7852	EXAMPLE 2 [WO2013004676]	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9831	iuphar.ligand:9831	PF-06684511	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:538	rxcui:39801	XAMOTEROL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.07767407	IUPHAR.LIGAND:558	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9809	iuphar.ligand:9809	BUTOXAMINE	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:10564	iuphar.ligand:10564	ARV-771	FALSE	FALSE	FALSE
NCBIGENE:2598	hgnc:1372	CA14	GuideToPharmacology	2024.1	inhibitor	0.8751278539282417	IUPHAR.LIGAND:6814	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2598	hgnc:1372	CA14	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:6810	rxcui:60207	DORZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:3093	hgnc:4914	UBE2K	GuideToPharmacology	2024.1	activator	0.921187215	IUPHAR.LIGAND:4804	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:2598	hgnc:1372	CA14	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:6797	rxcui:194881	BRINZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:5143	iuphar.ligand:5143	AZ10417808	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	1.009762908	IUPHAR.LIGAND:8375	rxcui:1876119	ETELCALCETIDE	TRUE	FALSE	FALSE
NCBIGENE:533	hgnc:861	ATP6V0B	GuideToPharmacology	2024.1	blocker	3.500511415712967	IUPHAR.LIGAND:2525	iuphar.ligand:2525	PB2+	FALSE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	0.4773424657790409	IUPHAR.LIGAND:12488	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
NCBIGENE:2472	hgnc:3882	FRA20B	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:6647	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.3029288725136221	IUPHAR.LIGAND:730	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:3497	iuphar.ligand:3497	CP-481,715	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.3182283105193606	IUPHAR.LIGAND:770	iuphar.ligand:770	CCL13	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:759	iuphar.ligand:759	CCL7	FALSE	FALSE	FALSE
NCBIGENE:2943	hgnc:1682	CD47	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:12036	iuphar.ligand:12036	ONTORPACEPT	FALSE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8191	iuphar.ligand:8191	COMPOUND 18 [PMID: 20873740]	FALSE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:9784	iuphar.ligand:9784	TETHERED CHEMERIN 9	FALSE	FALSE	FALSE
NCBIGENE:3187	hgnc:5041	HNRNPH1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11617	iuphar.ligand:11617	GLPG4716	FALSE	FALSE	FALSE
NCBIGENE:2982	hgnc:4685	GUCY1A1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11617	iuphar.ligand:11617	GLPG4716	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005308631	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
NCBIGENE:396	hgnc:678	ARHGDIA	GuideToPharmacology	2024.1	activator	3.500511415712967	IUPHAR.LIGAND:2347	iuphar.ligand:2347	CYCLIC GMP	FALSE	FALSE	FALSE
NCBIGENE:2363	hgnc:3871	FRA1D	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8493	iuphar.ligand:8493	COMPOUND 11 [PMID: 16413183]	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7688	iuphar.ligand:7688	AR-H067637	FALSE	FALSE	FALSE
NCBIGENE:2360	hgnc:3868	FRA1A	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6549	iuphar.ligand:6549	ALPHA-KETOTHIAZOLE ANALOGUE 36	FALSE	FALSE	FALSE
NCBIGENE:1989	hgnc:1974	CHUK	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9646	iuphar.ligand:9646	COMPOUND 47 [PMID: 28737909]	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	PD-123319	iuphar.ligand:597	PD123319	FALSE	FALSE	FALSE
NCBIGENE:2842	hgnc:4473	GPR19	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11282	iuphar.ligand:11282	COMPOUND 2 [PMID: 28621538]	FALSE	FALSE	FALSE
NCBIGENE:2339	hgnc:3782	FNTA	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8653	iuphar.ligand:8653	COMPOUND 51 [PMID: 19743866]	FALSE	FALSE	FALSE
NCBIGENE:2335	hgnc:3778	FN1	GuideToPharmacology	2024.1	antibody	4.039051633514961	IUPHAR.LIGAND:9807	iuphar.ligand:9807	SUTIMLIMAB	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.069824031	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10378	ncit:C152869	VERUCERFONT	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:3489	iuphar.ligand:3489	ANTALARMIN	FALSE	FALSE	FALSE
NCBIGENE:2734	hgnc:4316	GLG1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:7506	iuphar.ligand:7506	ISCHEMIN	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:3891	iuphar.ligand:3891	K41498	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:3919	iuphar.ligand:3919	X4-HIV-1 GP120	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:8160	iuphar.ligand:8160	COMPOUND 9B [PMID: 18986805]	FALSE	FALSE	FALSE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	0.1400204566285186	IUPHAR.LIGAND:5890	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	6-METHOXY-HARMALAN	chembl:CHEMBL338115	CHEMBL:CHEMBL338115	FALSE	FALSE	FALSE
NCBIGENE:1344	hgnc:2645	CYP4F2	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12767	iuphar.ligand:12767	TP0472993	FALSE	FALSE	FALSE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:2406	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	4'-EPICHAETOVIRIDIN A	chembl:CHEMBL1306556	CHEMBL:CHEMBL1306556	FALSE	FALSE	FALSE
NCBIGENE:1348	hgnc:2290	COX7A2P2	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11373	iuphar.ligand:11373	HET0016	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:1894	ncit:C79571	CLOPROSTENOL	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	0.3000438356325399	IUPHAR.LIGAND:1910	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:935	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:932	iuphar.ligand:932	(+)-ADTN	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.043756393	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.072927321	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1400204566285186	IUPHAR.LIGAND:953	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.001216441	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2010	hgnc:3331	EMD	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8166	iuphar.ligand:8166	COMPOUND 72 [WO2013026806]	FALSE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	NCI	14-Sep-17	NULL	0.1816874437221263	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7035	iuphar.ligand:7035	H3-COA-20	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	antibody	0.2500365296937833	IUPHAR.LIGAND:8090	rxcui:1723738	NECITUMUMAB	TRUE	TRUE	TRUE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:3322	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:8245	iuphar.ligand:8245	ZM-306416	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.029970132	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.1290114772375786	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	1.029066006546944	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P19793	hgnc:10477	RXRA	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	R-ETODOLAC	chembl:CHEMBL1716091	SDX-101	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	activator	0.108711535	IUPHAR.LIGAND:2326	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:12380	iuphar.ligand:12380	MIFANERTINIB	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:3510	ncit:C79124	LANEPITANT	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1942	iuphar.ligand:1942	ONO-AE3-208	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3057	iuphar.ligand:3057	ZARAGOZIC ACID A	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:8686	iuphar.ligand:8686	MARGETUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:8715	iuphar.ligand:8715	ELGEMTUMAB	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:9912	iuphar.ligand:9912	ALLITINIB	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.07458476	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	NULL	5.834185692854944	IUPHAR.LIGAND:9241	iuphar.ligand:9241	TX1-85-1	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.3211478363039418	MET-ENKEPHALIN	rxcui:1349278	METENKEFALIN	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.031254566	IUPHAR.LIGAND:7071	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	ALVERINE CITRATE	rxcui:71767	ALVERINE CITRATE	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.079557078	IUPHAR.LIGAND:7071	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:3487	ncit:C61606	ATRASENTAN	FALSE	FALSE	FALSE
NCBIGENE:622	hgnc:1027	BDH1	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2829	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:999	iuphar.ligand:999	PD-156707	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:1004	iuphar.ligand:1004	ENDOTHELIN-3	FALSE	FALSE	FALSE
NCBIGENE:870	hgnc:10939	SLC1A1	GuideToPharmacology	2024.1	NULL	0.375054795	IUPHAR.LIGAND:4534	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:4531	iuphar.ligand:4531	WAY-213613	FALSE	FALSE	FALSE
NCBIGENE:872	hgnc:10945	SLC1A7	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4631	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:4631	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
NCBIGENE:872	hgnc:10945	SLC1A7	GuideToPharmacology	2024.1	NULL	1.750255707856483	IUPHAR.LIGAND:4534	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
NCBIGENE:872	hgnc:10945	SLC1A7	GuideToPharmacology	2024.1	NULL	1.591141552596803	IUPHAR.LIGAND:4698	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:3435	rxcui:1798288	OBETICHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:871	hgnc:1546	SERPINH1	GuideToPharmacology	2024.1	NULL	0.7955707762984016	IUPHAR.LIGAND:4698	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10124	iuphar.ligand:10124	DUAL SEH/FAAH INHIBITOR 11	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3168	iuphar.ligand:3168	NE58018	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.049723174	IUPHAR.LIGAND:4192	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	blocker	0.072725306	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:9908	iuphar.ligand:9908	ONO-8590580	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	inhibitor	0.2011788169949981	IUPHAR.LIGAND:4083	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	blocker	0.095295229	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:4096	iuphar.ligand:4096	CIS-3-ACPBPA	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	inhibitor	0.175610941	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:4143	iuphar.ligand:4143	AZA-THIP	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:4096	iuphar.ligand:4096	CIS-3-ACPBPA	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	blocker	0.1973972602845657	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:419	hgnc:725	ART3	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:4320	iuphar.ligand:4320	TBPS	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	inhibitor	0.05853698	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:4143	iuphar.ligand:4143	AZA-THIP	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6091	iuphar.ligand:6091	GALANIN(3-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3191	drugbank:DB07873	LAURYL ALCOHOL DIPHOSPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:5866	iuphar.ligand:5866	SM-130,686	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:9724	rxcui:1991302	SEMAGLUTIDE	TRUE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:4070	drugbank:DB02966	FLUORO-WILLARDIINE	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	NULL	0.3125456621172291	IUPHAR.LIGAND:4081	iuphar.ligand:4081	[3H]CNQX	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:4085	iuphar.ligand:4085	[3H]KAINATE	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:9654	ncit:C166458	MAPRACORAT	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.1268301237577161	IUPHAR.LIGAND:4171	rxcui:1742747	SERINE, D-	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	blocker	0.1521961485092594	IUPHAR.LIGAND:4089	iuphar.ligand:4089	[3H]DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4088	iuphar.ligand:4088	[3H]MDL105519	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:4080	iuphar.ligand:4080	[3H]CGS19755	FALSE	FALSE	FALSE
NCBIGENE:2891	hgnc:4572	GRIA2	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:9053	ncit:C114381	TELAGLENASTAT	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	blocker	0.3387591692625452	IUPHAR.LIGAND:4089	iuphar.ligand:4089	[3H]DIZOCILPINE	FALSE	FALSE	FALSE
NCBIGENE:2029	hgnc:3360	ENSA	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:8014	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	blocker	0.6731752722524935	IUPHAR.LIGAND:2291	iuphar.ligand:2291	PICROTOXININ	FALSE	FALSE	FALSE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	blocker	0.8751278539282416	IUPHAR.LIGAND:2291	iuphar.ligand:2291	PICROTOXININ	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.1315981735230438	IUPHAR.LIGAND:733	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
NCBIGENE:311	hgnc:535	ANXA11	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4711	rxcui:1546380	4-HYDROXYBUTYRIC ACID	TRUE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	0.2885036881082115	IUPHAR.LIGAND:1588	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:12804	iuphar.ligand:12804	J27644	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.1881995384791917	IUPHAR.LIGAND:8391	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:9891	iuphar.ligand:9891	MARBOSTAT-100	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.106290832	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.091796628	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:8391	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.1035654265003836	IUPHAR.LIGAND:1247	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:8924	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1270	iuphar.ligand:1270	N,N-DIMETHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:112	hgnc:237	ADCY6	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:2921	iuphar.ligand:2921	DIHYDROSPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:10542	iuphar.ligand:10542	SPAG11B (61-103)	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:7423	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.251232877	IUPHAR.LIGAND:7741	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:7397	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:5990	iuphar.ligand:5990	IRAK-1/4 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2044	hgnc:3389	EPHA5	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:11785	iuphar.ligand:11785	IRAK3 PROTAC 23	FALSE	FALSE	FALSE
NCBIGENE:1727	hgnc:2873	CYB5R3	GuideToPharmacology	2024.1	agonist	0.7001022831425934	IUPHAR.LIGAND:4975	iuphar.ligand:4975	IL-10	FALSE	FALSE	FALSE
NCBIGENE:671	hgnc:1095	BPI	GuideToPharmacology	2024.1	agonist	0.9723642821424908	IUPHAR.LIGAND:12457	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
NCBIGENE:676	hgnc:1105	BRDT	GuideToPharmacology	2024.1	agonist	0.2885036881082116	IUPHAR.LIGAND:2510	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:2291	iuphar.ligand:2291	PICROTOXININ	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:12377	iuphar.ligand:12377	EMZELTRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:9991	rxcui:2591476	ABROCITINIB	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:9803	iuphar.ligand:9803	SAR-20347	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.086361301	IUPHAR.LIGAND:7913	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
NCBIGENE:2757	hgnc:23177	KEAP1	GuideToPharmacology	2024.1	NULL	2.100306849	IUPHAR.LIGAND:10488	iuphar.ligand:10488	COMPOUND 10 [PMID: 31411465]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:10452	iuphar.ligand:10452	NMRA-140	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:7563	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.041508041	IUPHAR.LIGAND:9383	iuphar.ligand:9383	OSI-930	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:8069	iuphar.ligand:8069	CP-673451	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.024163678	IUPHAR.LIGAND:5661	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1286	iuphar.ligand:1286	KISSPEPTIN-15	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.070765056	IUPHAR.LIGAND:5695	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:12988	iuphar.ligand:12988	ERAS-5024	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2314	iuphar.ligand:2314	EBIO	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	blocker	0.1389091831632129	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	2.500365296937833	IUPHAR.LIGAND:2331	iuphar.ligand:2331	SENICAPOC	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	2.500365296937833	IUPHAR.LIGAND:9318	iuphar.ligand:9318	NS6180	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	0.8334550989792776	IUPHAR.LIGAND:2324	iuphar.ligand:2324	DC-EBIO	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2320	iuphar.ligand:2320	UCL1684	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2314	iuphar.ligand:2314	EBIO	FALSE	FALSE	FALSE
NCBIGENE:546	hgnc:886	ATRX	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:7759	iuphar.ligand:7759	RY796	FALSE	FALSE	FALSE
NCBIGENE:2890	hgnc:4571	GRIA1	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:9027	iuphar.ligand:9027	L6H21	FALSE	FALSE	FALSE
NCBIGENE:2983	hgnc:4687	GUCY1B1	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:9782	iuphar.ligand:9782	PECAZINE	FALSE	FALSE	FALSE
NCBIGENE:2983	hgnc:4687	GUCY1B1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:11883	iuphar.ligand:11883	SAFIMALTIB	FALSE	FALSE	FALSE
NCBIGENE:1816	hgnc:3026	DRD5	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:7953	iuphar.ligand:7953	BMS-777607	FALSE	FALSE	TRUE
NCBIGENE:2096	hgnc:3463	ESAT	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8177	iuphar.ligand:8177	COMPOUND 16 [PMID: 17480064]	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1321	iuphar.ligand:1321	HS014	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:1335	iuphar.ligand:1335	AGOUTI-RELATED PROTEIN	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1335	iuphar.ligand:1335	AGOUTI-RELATED PROTEIN	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:7948	iuphar.ligand:7948	TIVANTINIB	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6252	iuphar.ligand:6252	GSK1331258	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6331	iuphar.ligand:6331	[3H]JNJ-40068782	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1421	iuphar.ligand:1421	BOMA	FALSE	FALSE	FALSE
NCBIGENE:2100	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:11896	iuphar.ligand:11896	COMPOUND 14 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1407	iuphar.ligand:1407	(S)-3,4-DCPG	FALSE	FALSE	FALSE
NCBIGENE:2098	hgnc:3465	ESD	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12936	iuphar.ligand:12936	PCC0105003	FALSE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	1.050153425	Grazoprevir	rxcui:1734630	GRAZOPREVIR	TRUE	FALSE	FALSE
NCBIGENE:3024	hgnc:4715	H1-1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:6647	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:2874	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
NCBIGENE:3023	ncbigene:3023	H4F3	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:6647	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:10703	drugbank:DB15624	HALICIN	FALSE	FALSE	FALSE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9700	iuphar.ligand:9700	COMPOUND 25 [PMID: 28038940]	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:7812	iuphar.ligand:7812	RXP470.1	FALSE	FALSE	FALSE
UNIPROT:P06213	hgnc:6091	INSR	TdgClinicalTrial	Jan-14	NULL	1.500219178	INSULIN ASPART	rxcui:352385	INSULIN ASPART PROTAMINE, HUMAN	TRUE	FALSE	FALSE
NCBIGENE:1628	hgnc:2697	DBP	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:5145	ncit:C1529	BATIMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:6568	iuphar.ligand:6568	COMPOUND 20 [PMID: 22153340]	FALSE	FALSE	FALSE
NCBIGENE:1628	hgnc:2697	DBP	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6466	iuphar.ligand:6466	CIPEMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1630	hgnc:2701	DCC	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6528	iuphar.ligand:6528	UK-356618	FALSE	FALSE	FALSE
NCBIGENE:1630	hgnc:2701	DCC	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:5145	ncit:C1529	BATIMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1647	hgnc:4095	GADD45A	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:8846	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.019261802	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:6639	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:8578	iuphar.ligand:8578	COMPOUND 29E [PMID: 23631440]	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	NIGULDIPINE	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
NCBIGENE:2881	hgnc:23248	MOGAT2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12971	iuphar.ligand:12971	BMS-986172	FALSE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	antibody	2.282942227638891	IUPHAR.LIGAND:9510	iuphar.ligand:9510	ANDECALIXIMAB	FALSE	FALSE	FALSE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:7428	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	0.1521961485092594	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	1.346350544504987	DNDI1417434	chembl:CHEMBL394883	CHEMBL:CHEMBL394883	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.029698909	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.050488145	IUPHAR.LIGAND:288	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:3259	iuphar.ligand:3259	VU0090157	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:351	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:299	ncit:C76041	FURTRETHONIUM IODIDE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:296	drugbank:DB04365	ARECOLINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:368	iuphar.ligand:3264	AFDX384	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:7777	iuphar.ligand:7777	UCM 793	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.2365210416022274	IUPHAR.LIGAND:1343	drugbank:DB08190	N-[2-(2-IODO-5-METHOXY-1H-INDOL-3-YL)ETHYL]ACETAMIDE	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.7778914257139926	DEXRAZOXANE	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
NCBIGENE:1216	hgnc:25588	SLC47A1	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:4800	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:7777	iuphar.ligand:7777	UCM 793	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:7774	iuphar.ligand:7774	EFPPEA	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.040235763	IUPHAR.LIGAND:224	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
NCBIGENE:1749	hgnc:2918	DLX5	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4870	iuphar.ligand:4870	AP811	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:10314	iuphar.ligand:10314	SELITRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:12377	iuphar.ligand:12377	EMZELTRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:10360	iuphar.ligand:10360	UTATRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.036413087	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10314	iuphar.ligand:10314	SELITRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:12237	iuphar.ligand:12237	CH7057288	FALSE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3999	iuphar.ligand:3999	&ALPHA;-CONOTOXIN MI	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:3979	iuphar.ligand:3979	[3H]CYTISINE	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:6926	ncit:C166844	ENCENICLINE	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:2106	iuphar.ligand:2106	SCH 206272	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.014172111	FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1695	iuphar.ligand:1695	[NPHE1]N/OFQ-(1-13)-NH2	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:3917	iuphar.ligand:3917	UFP-112	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:4016	iuphar.ligand:4016	RFRP-3	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.029970132	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:1499	iuphar.ligand:1499	DES-BR-NEUROPEPTIDE B-23	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1484	iuphar.ligand:1484	[125I]Y-RFRP-3	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:1571	iuphar.ligand:1571	JMV457	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1477	iuphar.ligand:1477	1DME	FALSE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	TRELANSERIN	ncit:C90946	TRELANSERIN	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:2201	iuphar.ligand:2201	SSR126768A	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:12439	iuphar.ligand:12439	RTOXA-43	FALSE	FALSE	FALSE
NCBIGENE:2138	hgnc:3519	EYA1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	0.546954909	IUPHAR.LIGAND:7676	iuphar.ligand:7676	PD-118057	FALSE	FALSE	FALSE
NCBIGENE:479	hgnc:13816	ATP12A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9545	iuphar.ligand:9545	NF770	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11230	iuphar.ligand:11230	NF279	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	2.187819634820604	IUPHAR.LIGAND:9022	iuphar.ligand:9022	GW791343	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4118	iuphar.ligand:4118	A438079	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	1.029562181092048	IUPHAR.LIGAND:1714	iuphar.ligand:1714	ATP&GAMMA;S	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:1762	iuphar.ligand:1762	NF340	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004786261	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:1766	iuphar.ligand:1766	BX 048	FALSE	FALSE	FALSE
NCBIGENE:347	hgnc:612	APOD	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:3525	iuphar.ligand:3525	RWJ-56110	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.069180068	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
NCBIGENE:986	hgnc:18068	SLC15A3	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4670	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.039068208	IUPHAR.LIGAND:9916	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.016161179	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:9728	ncit:C107686	DEZAPELISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:6023	drugbank:DB04769	5-QUINOXALIN-6-YLMETHYLENE-THIAZOLIDINE-2,4-DIONE	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:5715	iuphar.ligand:5715	TG-100-115	FALSE	FALSE	FALSE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9878	iuphar.ligand:9878	6-HYDROXY-5,7-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:5260	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.019093699	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005412046	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.4487835148349958	IUPHAR.LIGAND:2510	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:5971	iuphar.ligand:5971	FLT-3 INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:5684	iuphar.ligand:5684	GSK-461364A	FALSE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11526	iuphar.ligand:11526	SARUPARIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	CARBETAPENTANE CITRATE	rxcui:283547	CARBETAPENTANE CITRATE	TRUE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10117	iuphar.ligand:10117	AUNP-12	FALSE	FALSE	FALSE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11844	iuphar.ligand:11844	PF-06939999	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	activator	0.2051080907644316	IUPHAR.LIGAND:7443	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:11186	ncit:C124796	DAROVASERTIB	FALSE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 5	hgnc:11334	SSTR5	TTD	2020.06.01	NULL	1.640864726115453	Pasireotide	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
NCBIGENE:1476	hgnc:2482	CSTB	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:1486	hgnc:2496	CTBS	GuideToPharmacology	2024.1	activator	0.4688184931758437	IUPHAR.LIGAND:7443	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:8839	iuphar.ligand:8839	TORIN 2	FALSE	FALSE	FALSE
PRKCB	hgnc:9395	PRKCB	PharmGKB	4/5/24	NULL	0.182318303	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
NCBIGENE:1489	hgnc:2499	CTF1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9681	iuphar.ligand:9681	COMPOUND 13C [PMID: 20684591]	FALSE	FALSE	FALSE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8850	iuphar.ligand:8850	COMPOUND 7B [HAFTCHENARY ET AL., 2013]	FALSE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	0.054020238	IUPHAR.LIGAND:9381	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:13032	iuphar.ligand:13032	YHJ1039	FALSE	FALSE	FALSE
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.1620607136904151	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:11564	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:5890	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12244	iuphar.ligand:12244	SIR1-365	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1367387271762877	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.7001022831425934	IUPHAR.LIGAND:4055	iuphar.ligand:4055	AC55649	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2652	iuphar.ligand:2652	CD666	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.027840759	IUPHAR.LIGAND:5661	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:8079	iuphar.ligand:8079	HX 531	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
NCBIGENE:597	hgnc:991	BCL2A1	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:4349	iuphar.ligand:4349	HEME	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:10709	iuphar.ligand:10709	WF-47-JS03	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.032817295	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8911	ncit:C152866	VEROSUDIL	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.045658845	IUPHAR.LIGAND:5890	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:11462	iuphar.ligand:11462	TAMRLX	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:1999	iuphar.ligand:1999	[125I]RELAXIN-3 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:11909	iuphar.ligand:11909	[G(B24)S]R3/I5	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:8337	iuphar.ligand:8337	RELAXIN-3 B CHAIN DIMER	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	activator	0.138178082	IUPHAR.LIGAND:1728	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:2937	iuphar.ligand:2937	AFD(R)	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.055563673	GNF-PF-5061	chembl:CHEMBL601385	CHEMBL:CHEMBL601385	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:9569	iuphar.ligand:9569	ASP4058	FALSE	FALSE	FALSE
NCBIGENE:2707	hgnc:4285	GJB3	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:9515	iuphar.ligand:9515	SRT2104	FALSE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:6975	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
NCBIGENE:922	hgnc:1690	CD5L	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:4795	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11147	iuphar.ligand:11147	COMPOUND 60 [PMID: 30889352]	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	GNF-PF-1083	chembl:CHEMBL530361	CHEMBL:CHEMBL530361	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:8146	iuphar.ligand:8146	COMPOUND 23 [PMID: 17600705]	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11970	iuphar.ligand:11970	COMPOUND 28 [PMID: 35439002]	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:7889	ncit:C105402	ENTOSPLETINIB	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.025588534	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:2207	hgnc:3611	FCER1G	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8212	iuphar.ligand:8212	COMPOUND 66 [PMID: 21802293]	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	GW642444	rxcui:1424884	VILANTEROL	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2023	iuphar.ligand:2023	[125I]LTT-SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:2071	iuphar.ligand:2071	BN-81,674	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2036	iuphar.ligand:2036	BIM 23056	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2013	iuphar.ligand:2013	KE 108	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2059	iuphar.ligand:2059	[111IN,90Y]DOTA-TOC	FALSE	FALSE	FALSE
MICROTUBULE AFFINITY REGULATING KINASE 3	hgnc:6897	MARK3	TTD	2020.06.01	NULL	1.250182648468916	CBP-501	drugbank:DB17277	CBP-501	FALSE	FALSE	FALSE
NCBIGENE:3202	hgnc:5106	HOXA5	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12063	iuphar.ligand:12063	PEPTIDE 22D	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:6951	rxcui:3292	DEXTROTHYROXINE	TRUE	FALSE	FALSE
NCBIGENE:1752	hgnc:11848	TLR2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:5044	iuphar.ligand:5044	PEPTIDOGLYCAN	FALSE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	inhibitor	0.3241214273808303	IUPHAR.LIGAND:7198	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	blocker	0.1458546423213736	IUPHAR.LIGAND:2406	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1939	iuphar.ligand:1939	STA2	FALSE	FALSE	FALSE
PSMD4	hgnc:9561	PSMD4	CIViC	10-Apr-24	NULL	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:6050	drugbank:DB03921	4-(3-PYRIDIN-2-YL-1H-PYRAZOL-4-YL)QUINOLINE	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:6049	iuphar.ligand:6049	TGF-BETA RI INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1984	ncit:C65463	DOMITROBAN	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.044198376	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.3860858179095183	IUPHAR.LIGAND:2443	iuphar.ligand:2443	ACAA	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.074690855	IUPHAR.LIGAND:2330	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:12532	iuphar.ligand:12532	AM-1473	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.364636606	IUPHAR.LIGAND:2503	rxcui:1362698	CHLOROFORM	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.4475085616678508	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:11847	iuphar.ligand:11847	ML3-SA1	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.750109589	IUPHAR.LIGAND:3390	iuphar.ligand:3390	5S-HETE	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:6401	iuphar.ligand:6401	SN-1	FALSE	FALSE	FALSE
NCBIGENE:511	hgnc:3145	TRPV5	GuideToPharmacology	2024.1	blocker	0.4688184931758437	IUPHAR.LIGAND:2449	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:11238	iuphar.ligand:11238	NSC151066	FALSE	FALSE	FALSE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	0.091796628	Oxyphenbutazone	rxcui:7816	OXYPHENBUTAZONE	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12557	iuphar.ligand:12557	GSK2798745	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:10304	iuphar.ligand:10304	RN-9893	FALSE	FALSE	FALSE
NCBIGENE:2424	ncbigene:2424	FRA8F	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	inhibitor	0.037398626	IUPHAR.LIGAND:5239	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8146	iuphar.ligand:8146	COMPOUND 23 [PMID: 17600705]	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:11893	iuphar.ligand:11893	COMPOUND 6 [PMID: 34333981]	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1058622403945453	IUPHAR.LIGAND:7913	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:2203	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2195	iuphar.ligand:2195	OH-LVA	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.019490598	IUPHAR.LIGAND:2172	iuphar.ligand:2172	LVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.014617949	IUPHAR.LIGAND:2221	iuphar.ligand:2221	D(CH2)5[TYR(ME)2,THR4,TYR-NH29]OVT	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.014617949	IUPHAR.LIGAND:2223	iuphar.ligand:2223	D(CH2)5[TYR(ME)2]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:2223	iuphar.ligand:2223	D(CH2)5[TYR(ME)2]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2214	iuphar.ligand:2214	D(CH2)5[D-ILE2,ILE4,ALA-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:2203	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:8529	iuphar.ligand:8529	RO5028442	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8855	iuphar.ligand:8855	SM-122	FALSE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:7837	ncit:C97037	SPEBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1549	iuphar.ligand:1549	NPY-(2-36)	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	CIViC	10-Apr-24	NULL	0.046940525	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	0.4906052389860809	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	1.336059069138614	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	CIViC	10-Apr-24	NULL	0.040390516	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.038382801	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.9845188356692719	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
MAPK1	hgnc:6871	MAPK1	CIViC	10-Apr-24	NULL	0.042863405	WZ4002	iuphar.ligand:9176	WZ4002	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.019739726	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	1.944728564284981	PRALSETINIB	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	0.5479061346333338	TAE684	ncit:C171615	ALK INHIBITOR TAE684	FALSE	FALSE	TRUE
CREBBP	hgnc:2348	CREBBP	CIViC	10-Apr-24	NULL	0.051885051	C646	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
GATA2	hgnc:4171	GATA2	CIViC	10-Apr-24	NULL	0.07631929	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.1372749574789398	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
EREG	hgnc:3443	EREG	CIViC	10-Apr-24	NULL	0.4375639269641209	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
SLFN11	hgnc:26633	SLFN11	CIViC	10-Apr-24	NULL	0.8751278539282418	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	CIViC	10-Apr-24	NULL	0.1666910197958555	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
TSC2	hgnc:12363	TSC2	CIViC	10-Apr-24	NULL	2.250328767	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
CSF1R	hgnc:2433	CSF1R	CIViC	10-Apr-24	NULL	0.028929846	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
RASA1	hgnc:9871	RASA1	CIViC	10-Apr-24	NULL	1.050153425	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.1339481409073839	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.1875273972703375	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.1187956362798518	ENZALUTAMIDE	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
RIT1	hgnc:10023	RIT1	CIViC	10-Apr-24	NULL	0.7955707762984016	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
FLCN	hgnc:27310	FLCN	CIViC	10-Apr-24	NULL	1.500219178	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
PIK3R2	hgnc:8980	PIK3R2	CIViC	10-Apr-24	NULL	0.037398626	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.4734548598913698	COBIMETINIB	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
KDM5C	hgnc:11114	KDM5C	CIViC	10-Apr-24	NULL	0.2500365296937833	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
CCND1	hgnc:1582	CCND1	CIViC	10-Apr-24	NULL	0.038467158	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
DKK1	hgnc:2891	DKK1	CIViC	10-Apr-24	NULL	0.049026771	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
DKK1	hgnc:2891	DKK1	CIViC	10-Apr-24	NULL	0.092606122	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
WEE1	hgnc:12761	WEE1	CIViC	10-Apr-24	NULL	0.7212592202705288	ADAVOSERTIB	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	0.1205533268166455	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ACTL6A	hgnc:24124	ACTL6A	CIViC	10-Apr-24	NULL	0.3977853881492008	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.4565884455277782	AZD3463	iuphar.ligand:7706	AZD3463	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.091317689	Topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	1.521961485092594	ASP3026	ncit:C116727	ALK INHIBITOR ASP3026	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.015477574	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.2282942227638891	SAF-189s	ncit:C175475	FORITINIB SUCCINATE	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	1.193356164447602	TetMYB	ncit:C153094	TETMYB DNA VACCINE	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.1835932560688619	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.047952211	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
ATR	hgnc:882	ATR	JAX-CKB	10-Apr-24	NULL	0.2692701089009974	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.1541321073454828	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	1.657092009619794	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	2.341819737097098	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.4123639102279672	AZ628	iuphar.ligand:8475	AZ628	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2199274187882492	GDC0879	iuphar.ligand:5681	GDC-0879	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.030545475	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.1458546423213736	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.926605963	Nab-paclitaxel	ncit:C2688	NAB-PACLITAXEL	FALSE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.008236497	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.2059124362184097	Cadonilimab	ncit:C153379	CADONILIMAB	FALSE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	3.500511415712966	RP-3500	ncit:C174206	CAMONSERTIB	FALSE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	0.5834185692854944	Veliparib	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	CPL304110	ncit:C173964	FGFR INHIBITOR CPL304110	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.5672124979164529	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.014732792	Mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.060772768	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.2302968036653267	Ganitumab	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.017117415	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.063415062	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.023295329	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1058622403945453	Rigosertib	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2540693769469088	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.047049885	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	AZD0364	ncit:C176765	TIZATERKIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2778183663264258	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.025588534	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.3684748858645228	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	Ganitumab	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.037398626	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.013890918	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.008103036	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.070956312	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.049275217	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	EP0031	ncit:C189067	RET INHIBITOR EP0031	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	1.29648571	Vepafestinib	ncit:C176968	VEPAFESTINIB	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	4.375639269641208	KPT-8602	ncit:C125193	ELTANEXOR	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.04636439	LB-100	drugbank:DB15412	LB-100	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.04636439	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1545479653736408	Idasanutlin	ncit:C99131	IDASANUTLIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.019318496	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.017832458	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.009659248	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.016558711	Ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	Serdemetan	ncit:C77904	SERDEMETAN	FALSE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	FURAPREVIR	ncit:C166437	FURAPREVIR	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	N-(BENZYLCARBAMOTHIOYL)BENZAMIDE	chembl:CHEMBL1478462	CHEMBL:CHEMBL1478462	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-4481	chembl:CHEMBL597251	CHEMBL:CHEMBL597251	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	1.790034246671403	clofibrate	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.056826484	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.3088686543276147	PHENSERINE	drugbank:DB04892	PHENSERINE	FALSE	FALSE	FALSE
UNIPROT:P00813	hgnc:186	ADA	TEND	1-Aug-11	NULL	0.032382159	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:914	hgnc:1639	CD2	GuideToPharmacology	2024.1	NULL	5.834185692854944	IUPHAR.LIGAND:4493	iuphar.ligand:4493	[3H]HEMICHOLINIUM-3	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:11879	iuphar.ligand:11879	NARAZACICLIB	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.1179947668217853	IUPHAR.LIGAND:970	iuphar.ligand:970	(+)-AJ76	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.046425881	IUPHAR.LIGAND:940	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
KCNG3	hgnc:18306	KCNG3	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.059532507	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.020164236	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
TNFRSF1B	hgnc:11917	TNFRSF1B	PharmGKB	4/5/24	NULL	1.016277507787635	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000007704	chembl:CHEMBL589469	CHEMBL:CHEMBL589469	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.2273059360852575	2-CHLORO-ADENOSINETRIPHOSPHATE	iuphar.ligand:1716	2-CHLOROADENOSINE-5-TRIPHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:Q02763	hgnc:11724	TEK	TdgClinicalTrial	Jan-14	NULL	0.3977853881492008	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.1470803115845784	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	0.020048748	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.078136416	IUPHAR.LIGAND:2514	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.2375912725597036	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:12298	iuphar.ligand:12298	MOSUNETUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:884	iuphar.ligand:884	T-0632	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:12377	iuphar.ligand:12377	EMZELTRECTINIB	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.010742159	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.7955707762984014	SJ000032155	chembl:CHEMBL590643	CHEMBL:CHEMBL590643	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.058341857	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.3889457128569962	LIRIMILAST	ncit:C82304	LIRIMILAST	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.037213091	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:2730	hgnc:4312	GCLM	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:8396	iuphar.ligand:8396	COMPOUND 34 [PMID: 25974391]	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:4283	iuphar.ligand:4283	PHENYLACETYLRINVANIL	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.1598407039138341	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011012515	MICONAZOLE NITRATE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
CAV1	hgnc:1527	CAV1	NCI	14-Sep-17	NULL	0.6731752722524935	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	LAVENDUSTIN A	ncit:C1142	LAVENDUSTIN A	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2282942227638891	ANTHRACENE-9-CARBOXYLIC ACID	iuphar.ligand:4113	9-ANTHROIC ACID	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	1.750255707856483	D-ALPHA-TOCOPHEROL ACETATE	ncit:C74962	D-ALPHA-TOCOPHEROL ACETATE	FALSE	FALSE	FALSE
HTR1E	hgnc:5291	HTR1E	ChEMBL	33	inhibitor	0.6177373086552295	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.3182283105193605	GLP-1	chembl:CHEMBL1240772	GLP-1	FALSE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	0.729273212	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.018301733	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.6035364509849942	TYRAMINE	rxcui:10958	TYRAMINE	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.2344092465879218	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
MECP2	hgnc:6990	MECP2	PharmGKB	4/5/24	NULL	0.2206204673768676	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.08914715	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	DNDI1417739	chembl:CHEMBL487356	CHEMBL:CHEMBL487356	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.3621218705909965	PUUPEHENONE	chembl:CHEMBL157844	PUUPEHENONE	FALSE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA2.1	hgnc:6290	KCNN1	TTD	2020.06.01	NULL	1.640864726115453	dequalinium	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.596678082	LANDIOLOL	ncit:C79125	LANDIOLOL	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	FDA	10-Apr-24	NULL	8.353493151133215	Lumacaftor	rxcui:1655922	LUMACAFTOR	TRUE	FALSE	FALSE
NCBIGENE:1606	hgnc:2849	DGKA	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:11982	ncit:C166793	VIPIVOTIDE TETRAXETAN	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	2.561349816375341	XEN-D0501	drugbank:DB18673	XEN-D0501	FALSE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	blocker	0.1262203635473425	PHLOROGLUCINOL	rxcui:8196	PHLOROGLUCINOL	TRUE	FALSE	FALSE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	0.3977853881492006	Sodium lauryl sulfate	rxcui:9871	SODIUM DODECYL SULFATE	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4327	iuphar.ligand:4327	TPA023	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TBXA2R	hgnc:11608	TBXA2R	ChEMBL	33	inhibitor	1.875273972703375	TERBOGREL	ncit:C96923	TERBOGREL	FALSE	FALSE	FALSE
RRM2	hgnc:10452	RRM2	ChEMBL	33	inhibitor	0.212581665	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.591141552596803	Nafarelin	rxcui:28656	NAFARELIN	TRUE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.077789143	IUPHAR.LIGAND:8014	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.463302981	IUPHAR.LIGAND:8924	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	DNDI1417260	chembl:CHEMBL2094573	CHEMBL:CHEMBL2094573	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.3409589041278863	2-CHLORO-ADENOSINETRIPHOSPHATE	iuphar.ligand:1716	2-CHLOROADENOSINE-5-TRIPHOSPHATE	FALSE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.2375912725597036	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.041021618	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11897	iuphar.ligand:11897	ORLUDODSTAT	FALSE	FALSE	FALSE
CFLAR	hgnc:1876	CFLAR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2625383561784725	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.4526523382387456	SJ000202381	chembl:CHEMBL591598	CHEMBL:CHEMBL591598	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	GENTIAN VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.0023813	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
IL6R	hgnc:6019	IL6R	NCI	14-Sep-17	NULL	0.4039051633514962	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10056	ncit:C166608	DAPANSUTRILE	FALSE	FALSE	FALSE
TNNC1	hgnc:11943	TNNC1	DTC	9/2/20	NULL	0.42006137	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:8435	iuphar.ligand:8435	LP-44	FALSE	FALSE	FALSE
PPAT	hgnc:9238	PPAT	ChEMBL	33	inhibitor	17.50255707856483	AZATHIOPRINE SODIUM	rxcui:267476	AZATHIOPRINE SODIUM	TRUE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:632	iuphar.ligand:632	[D-PHE6,&BETA;-ALA11,PHE13,NLE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
PRIM1	hgnc:9369	PRIM1	ChEMBL	33	inhibitor	0.092606122	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.1121958787087489	IUPHAR.LIGAND:4171	rxcui:1742747	SERINE, D-	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	1.591141552596803	DX-8951F	ncit:C1679	EXATECAN MESYLATE	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	1.141471113819445	A-1155463	chembl:CHEMBL3342332	A-1155463	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	1-AMINOCYCLOHEXANECARBOXYLIC ACID	chembl:CHEMBL559934	CHEMBL:CHEMBL559934	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	DNDI1417368	chembl:CHEMBL2094652	CHEMBL:CHEMBL2094652	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	NSC-753576	chembl:CHEMBL2088731	CHEMBL:CHEMBL2088731	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	NORTRIPTYLINE HYDROCHLORIDE	rxcui:203130	NORTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.030868707	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.006000877	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:2687	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
NCBIGENE:3102	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:10514	iuphar.ligand:10514	RO0094889	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.1392776425349986	diazepam	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	1.250182648468916	Chlorthalidone	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
ATIC	hgnc:794	ATIC	PharmGKB	4/5/24	NULL	0.2800409132570373	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.065389379	MILCICLIB	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
MAG	hgnc:6783	MAG	ChEMBL	33	inhibitor	17.50255707856483	REFANEZUMAB	ncit:C152172	REFANEZUMAB	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.3337351985319565	DANUSERTIB	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.017620024	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:9108	iuphar.ligand:9108	ARRY-382	FALSE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	blocker	0.2651902587661338	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.064111931	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.2365210416022274	TERTATOLOL	rxcui:37840	TERTATOLOL	FALSE	FALSE	FALSE
CD83	hgnc:1703	CD83	NCI	14-Sep-17	NULL	6.563458904461812	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.1615620653405984	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.1684738114514262	naproxen	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	0.2778183663264259	CHR-3996	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	JWCAR029	ncit:C155878	RELMACABTAGENE AUTOLEUCEL	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.070574827	RUFINAMIDE	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	1.093909817410302	Vabicaserin	ncit:C132725	VABICASERIN	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.027781837	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10672	iuphar.ligand:10672	COMPOUND 5 [TOMASSI ET AL., 2020]	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	MOLINDONE	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.3454452054979901	MUBRITINIB	ncit:C66212	MUBRITINIB	FALSE	FALSE	TRUE
NAT1	hgnc:7645	NAT1	PharmGKB	4/5/24	NULL	0.4861821410712453	cotinine	ncit:C70941	COTININE	FALSE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.2778183663264258	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.3860858179095183	Eptastigmine	ncit:C65525	EPTASTIGMINE	FALSE	FALSE	FALSE
NCBIGENE:871	hgnc:1546	SERPINH1	GuideToPharmacology	2024.1	NULL	0.8751278539282418	IUPHAR.LIGAND:4534	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.853211925965688	Sugemalimab	ncit:C154550	SUGEMALIMAB	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2045	iuphar.ligand:2045	[111IN]DOTA-NOC	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.2234368988752957	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.212152207	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1875273972703375	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
EDNRA	hgnc:3179	EDNRA	TALC	12-May-16	inhibitor	4.565884455277782	ZIBOTENTAN	ncit:C48430	ZIBOTENTAN	FALSE	FALSE	TRUE
UNIPROT:Q15858	hgnc:10597	SCN9A	TdgClinicalTrial	Jan-14	NULL	0.039068208	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.3182283105193606	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.3281729452230906	LY-2780301	chembl:CHEMBL3545134	LY-2780301	FALSE	FALSE	FALSE
NCBIGENE:2353	hgnc:3796	FOS	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:6535	iuphar.ligand:6535	COMPOUND (R)-26 [PMID: 22686657]	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:5817	iuphar.ligand:5817	PF-04418948	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1207072901969988	SALICYLHYDROXAMIC ACID	drugbank:DB03819	SALICYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.009357988	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:1161	hgnc:3439	ERCC8	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:4671	rxcui:94	5-HYDROXYTRYPTOPHAN	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	modulator	0.081030357	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014160645	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	LUFENURON	rxcui:83586	LUFENURON	TRUE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	0.301335273	CNTX-4975	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
INTERLEUKIN-21	hgnc:6005	IL21	TTD	2020.06.01	NULL	17.50255707856483	NN-8828	chembl:CHEMBL4297797	NNC0114-0006	FALSE	FALSE	FALSE
NCBIGENE:1389	hgnc:2350	CREBL2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8750	iuphar.ligand:8750	COMPOUND 21N [PMID: 17656086]	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	1.029562181092048	IUPHAR.LIGAND:4306	rxcui:9525	SALICYLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.090219366	IUPHAR.LIGAND:457	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	1.123158743009508	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
PLA2G6	hgnc:9039	PLA2G6	PharmGKB	4/5/24	NULL	0.4449802647092754	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.030886865	bupivacaine	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	0.082300425	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:4019	iuphar.ligand:4019	[3H]NPVF	FALSE	FALSE	FALSE
NCBIGENE:1573	hgnc:2634	CYP2J2	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8445	ncit:C90656	BELORANIB	FALSE	FALSE	FALSE
UNIPROT:P49190	hgnc:9609	PTH2R	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	PARATHYROID HORMONE	rxcui:1427222	PARATHYROID HORMONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007232462	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	0.301335273	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.061628722	(+)-TAXIFOLIN	chembl:CHEMBL66	(+)-TAXIFOLIN	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.2035181055647073	ESMIRTAZAPINE	ncit:C76963	ESMIRTAZAPINE	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.063300387	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:739	iuphar.ligand:739	ARACHIDONYLCYCLOPROPYLAMIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.5147810905460245	URIDINE-5'-MONOPHOSPHATE	drugbank:DB03685	URIDINE MONOPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:8846	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	PF-4708671	iuphar.ligand:8036	PF-4708671	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.055563673	IUPHAR.LIGAND:2953	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
CD38	hgnc:1667	CD38	ChEMBL	33	binder	5.834185692854944	MEZAGITAMAB	ncit:C148078	MEZAGITAMAB	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.047734247	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	NECROSTATIN	iuphar.ligand:9750	NECROSTATIN-1	FALSE	FALSE	FALSE
IGFBP3	hgnc:5472	IGFBP3	PharmGKB	4/5/24	NULL	0.4412409347537352	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	8.290684931951763	AM-211	chembl:CHEMBL2181753	AM-211	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:10233	iuphar.ligand:10233	AZ2	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.1535312024435511	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.2263261691193728	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	DIHYDROTANSHINONE I	chembl:CHEMBL227075	DIHYDROTANSHINONE I	FALSE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	3.500511415712966	THYROTROPIN	rxcui:10579	THYROTROPIN	TRUE	FALSE	FALSE
PRKACB	hgnc:9381	PRKACB	ChEMBL	33	inhibitor	1.544343271638073	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	1.019566431761058	RESMETIROM	ncit:C170368	RESMETIROM	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-124316	chembl:CHEMBL534214	CHEMBL:CHEMBL534214	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	TRIFLUPERIDOL	rxcui:10804	TRIFLUPERIDOL	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.8899605294185507	Losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006210251	ACID BLUE 129	chembl:CHEMBL133576	ACID BLUE 129	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.2386712328895204	TENOFOVIR DISOPROXIL FUMARATE	rxcui:322248	TENOFOVIR DISOPROXIL FUMARATE	TRUE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.076765601	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	3-METHOXY-MORPHANIN HCL	chembl:CHEMBL1257022	CHEMBL:CHEMBL1257022	FALSE	FALSE	FALSE
PLA2G4A	hgnc:9035	PLA2G4A	PharmGKB	4/5/24	NULL	0.2430910705356227	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	AURAPTENE	chembl:CHEMBL307341	AURAPTENE	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.2134458180312784	IUPHAR.LIGAND:1881	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	1.500219178	IUPHAR.LIGAND:12544	iuphar.ligand:12544	RHTX	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TIOCONAZOLE	rxcui:38298	TIOCONAZOLE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	BMS-509744	iuphar.ligand:9994	BMS-509744	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	THIOINOSINE	ncit:C877	THIOINOSINE	FALSE	FALSE	FALSE
TNNT2	hgnc:11949	TNNT2	ChEMBL	33	positive modulator	1.875273972703374	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
IL22RA1	hgnc:13700	IL22RA1	ChEMBL	33	agonist	26.25383561784724	EFLEPEDOCOKIN ALFA	ncit:C141419	EFLEPEDOCOKIN ALFA	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TRIMETHYL-TETRADECYL-AMMONIUM CHLORIDE	chembl:CHEMBL109747	TRIMETHYL-TETRADECYL-AMMONIUM CHLORIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.1232574442152452	ESMIRTAZAPINE MALEATE	ncit:C76940	ESMIRTAZAPINE MALEATE	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	CancerCommons	25-Jul-13	inhibitor	0.1801292323694494	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.7095631248066824	KLH	ncit:C1139	KEYHOLE LIMPET HEMOCYANIN	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.1025540453822158	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:11413	iuphar.ligand:11413	NEMTABRUTINIB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	HYDROXYZINE HYDROCHLORIDE	rxcui:154987	HYDROXYZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	ISOETHARINE	rxcui:6023	ISOETHARINE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.9376369863516875	R 75251	ncit:C1433	LIAROZOLE	FALSE	FALSE	FALSE
INTERLEUKIN-12 ALPHA	hgnc:5969	IL12A	TTD	2020.06.01	NULL	1.750255707856483	STA-5326	ncit:C90808	APILIMOD	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.1646008502686348	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6196	iuphar.ligand:6196	BAYCYSLT2	FALSE	FALSE	FALSE
NCBIGENE:2257	hgnc:3668	FGF12	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7397	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.05068308	Acalisib	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.025003653	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1767935058440892	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.034544521	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:121	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:11080	iuphar.ligand:11080	TATM2NX	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.1025540453822158	Mocetinostat	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.6105543166941221	orciprenaline	rxcui:7688	METAPROTERENOL	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.052090944	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.026045472	IUPHAR.LIGAND:548	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.045898314	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	TENONITROZOLE	rxcui:236186	TENONITROZOLE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00402481	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.007024438	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.4412409347537353	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.7778914257139925	Ronomilast	ncit:C97274	RONOMILAST	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	MIZOLASTINE	rxcui:61455	MIZOLASTINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	NSC-93817	chembl:CHEMBL1509789	CHEMBL:CHEMBL1509789	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW572401X	chembl:CHEMBL275473	GW572401X	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:491	iuphar.ligand:491	A-123189	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:8984	iuphar.ligand:8984	JNJ-39758979	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	L-3,4-DIHYDROXYPHENYLALANINE METHYL ESTER HCL	chembl:CHEMBL1255756	CHEMBL:CHEMBL1255756	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:2073	iuphar.ligand:2073	L-796,778	FALSE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	DTC	9/2/20	NULL	11.66837138570988	4-METHOXYPHENOXYBENZENE	chembl:CHEMBL398021	CHEMBL:CHEMBL398021	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.4286340509036286	RECOMBINANT HUMAN IL-4	rxcui:1426682	BINETRAKIN	FALSE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.044198376	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10732	ncit:C90704	OTAMIXABAN	FALSE	FALSE	FALSE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	1.193356164447602	Gadofosveset	rxcui:1364289	GADOFOSVESET TRISODIUM	TRUE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	activator	3.088686543276147	IUPHAR.LIGAND:4137	iuphar.ligand:4137	ARCAINE	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9755	iuphar.ligand:9755	PBT-3	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	CIS-RESVERATROL	chembl:CHEMBL87333	CIS-RESVERATROL	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW680975X	chembl:CHEMBL381948	GW680975X	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	1.166837138570988	3-BENZHYDRYL-PYRIDINE	chembl:CHEMBL149246	CHEMBL:CHEMBL149246	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001825687	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	1.381780822	Recombinant Factor IX	rxcui:1300488	NONACOG ALFA	TRUE	FALSE	FALSE
UNIPROT:Q8WW43	hgnc:24080	APH1B	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	BMS-299897	chembl:CHEMBL247471	CHEMBL:CHEMBL247471	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	EDARAVONE	rxcui:1921877	EDARAVONE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.4773424657790409	NEPAFENAC	rxcui:298665	NEPAFENAC	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.2	hgnc:1389	CACNA1B	TTD	2020.06.01	NULL	1.640864726115453	CNV-2197944	drugbank:DB15229	CNV-2197944	FALSE	FALSE	FALSE
DUSP3	hgnc:3069	DUSP3	DTC	9/2/20	NULL	0.4688184931758437	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.193356164447602	Gonadorelin	rxcui:6384	GONADORELIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.030386384	benzbromarone	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
EPHX2	hgnc:3402	EPHX2	PharmGKB	4/5/24	NULL	0.071439008	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.2778183663264258	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	modulator	0.4375639269641209	SUVECALTAMIDE	ncit:C174710	SUVECALTAMIDE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.076098074	Dinaciclib	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	GNF-PF-3832	chembl:CHEMBL261693	CHEMBL:CHEMBL261693	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
COL1A2	hgnc:2198	COL1A2	NCI	14-Sep-17	NULL	2.333674277141978	TGF-BETA 2	ncit:C1286	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA-2	FALSE	FALSE	FALSE
CD55	hgnc:2665	CD55	NCI	14-Sep-17	NULL	0.2658616265098455	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	0.5000730593875667	IUPHAR.LIGAND:770	iuphar.ligand:770	CCL13	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3121	iuphar.ligand:3121	BPH-830	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	BENZOFURAN	drugbank:DB04179	BENZOFURAN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	DEHYDROVARIABILIN	chembl:CHEMBL1520512	DEHYDROVARIABILIN	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.07182992	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	TENOXICAM	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	AMINACRINE HYDROCHLORIDE	rxcui:81949	AMINACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2045	iuphar.ligand:2045	[111IN]DOTA-NOC	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.092933931	metyrapone	rxcui:6923	METYRAPONE	TRUE	FALSE	FALSE
PHOSPHATIDYLINOSITOL-4-KINASE ALPHA	hgnc:8983	PI4KA	TTD	2020.06.01	NULL	1.500219178	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	ETHAVERINE	rxcui:24464	ETHAVERINE	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.182318303	SULFADIAZINE, SILVER	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
UNIPROT:Q9NYA1	hgnc:11240	SPHK1	TdgClinicalTrial	Jan-14	NULL	3.750547945406749	PHENOXODIOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6366	iuphar.ligand:6366	COMPOUND 24D [PMID: 23357634]	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.138178082	IUPHAR.LIGAND:339	iuphar.ligand:339	WIN 51,708	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	TEDIZOLID	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	XANTHOANGELOL F	chembl:CHEMBL1722838	XANTHOANGELOL F	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.9546849315580819	DIHYDROTANSHINONE I	chembl:CHEMBL227075	DIHYDROTANSHINONE I	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:3848	iuphar.ligand:3848	[PRO34]NPY	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.2678962818147678	TENOFOVIR	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	NSC-292213	chembl:CHEMBL222808	CHEMBL:CHEMBL222808	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	1.406455479527531	CD40L	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
NCBIGENE:2039	hgnc:3382	DMTN	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:5694	iuphar.ligand:5694	MLN-120B	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	1.591141552596803	FOTEMUSTINE	ncit:C1106	FOTEMUSTINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PUROMYCIN HYDROCHLORIDE	ncit:C75148	PUROMYCIN HYDROCHLORIDE	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.4688184931758437	PI3-KINASE INHIBITORS	ncit:C2152	PHOSPHATIDYLINOSITIDE 3-KINASE INHIBITOR	FALSE	FALSE	TRUE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.2282942227638891	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.1582152052299645	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.2573905452730122	PAROMOMYCIN SULFATE	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.064944553	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	1.584283183835609	AMONAFIDE	rxcui:1440270	AMONAFIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124696	chembl:CHEMBL546531	CHEMBL:CHEMBL546531	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.729273212	rifapentine	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	0.088333021	RXDX 101	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	TCMDC-125764	chembl:CHEMBL586670	CHEMBL:CHEMBL586670	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.033615667	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	2.100306849	SILYBIN B	chembl:CHEMBL592675	SILYBIN B	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004952619	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TEND	1-Aug-11	NULL	0.2275522047050683	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:10137	iuphar.ligand:10137	YH18968	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.035098711	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	0.6563458904461813	LICOGLIFLOZIN	ncit:C150375	LICOGLIFLOZIN	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.093763699	GRINIMIBINE	chembl:CHEMBL1477760	GRINIMIBINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	2-CHLORO-ADENOSINETRIPHOSPHATE	iuphar.ligand:1716	2-CHLOROADENOSINE-5-TRIPHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.049723174	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	ChEMBL	33	modulator	2.100306849	PENTAZOCINE LACTATE	rxcui:203196	PENTAZOCINE LACTATE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.062509132	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:870	hgnc:10939	SLC1A1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:4631	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.5250767123569451	GRINIMIBINE	chembl:CHEMBL1477760	GRINIMIBINE	FALSE	FALSE	FALSE
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	3.029288725136221	Triapine	ncit:C2242	TRIAPINE	FALSE	FALSE	TRUE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	modulator	2.500365296937833	IUPHAR.LIGAND:6217	iuphar.ligand:6217	ADX71743	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.038104261	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	blocker	0.2243917574174979	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	(+/-)-VANILLYLMANDELIC ACID	iuphar.ligand:6645	VANILLYLMANDELIC ACID	FALSE	FALSE	FALSE
MYL2	hgnc:7583	MYL2	ChEMBL	33	activator	2.187819634820604	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.01439355	SPIPERONE	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002731787	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:226	rxcui:139778	TEGASEROD	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.078958904	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	0.2763561643983921	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
LAMA2	hgnc:6482	LAMA2	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	1.050153425	Rivoceranib	ncit:C152237	RIVOCERANIB	FALSE	FALSE	FALSE
KCNG2	hgnc:6249	KCNG2	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
NME1	hgnc:7849	NME1	PharmGKB	4/5/24	NULL	0.4375639269641208	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
NCBIGENE:347	hgnc:612	APOD	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:3742	iuphar.ligand:3742	TFLLR-NH2	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	PROSTAGLANDIN B1	chembl:CHEMBL1561148	PROSTAGLANDIN B1	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	SJ000117447	chembl:CHEMBL592611	CHEMBL:CHEMBL592611	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.3977853881492007	PIRENOXINE	rxcui:228080	PIRENOXINE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	ChEMBL	33	inhibitor	0.064347636	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	0.084146909	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
PDE10A	hgnc:21160	LINC00473	ChEMBL	33	inhibitor	0.546954909	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.750109589	IUPHAR.LIGAND:12755	ncit:C170153	MAVATREP	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	0.252440727	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.092443083	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.4579157375205915	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
KIAA2026	hgnc:23378	BRD10	PharmGKB	4/5/24	NULL	1.093909817410302	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
NCBIGENE:1320	hgnc:2597	CYP1B1	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:12963	iuphar.ligand:12963	2,3',4,5'-TETRAMETHOXYSTILBENE	FALSE	FALSE	FALSE
GADD45G	hgnc:4097	GADD45G	NCI	14-Sep-17	NULL	6.177373086552294	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:6985	iuphar.ligand:6985	BRP-LPA	FALSE	FALSE	FALSE
METHIONINE AMINOPEPTIDASE 2	hgnc:16672	METAP2	TTD	2020.06.01	NULL	1.640864726115453	M8891	iuphar.ligand:12714	M8891	FALSE	FALSE	FALSE
CHRM4	hgnc:1953	CHRM4	DTC	9/2/20	NULL	0.3889457128569963	PIPERTRAMINE AMIDE	chembl:CHEMBL130835	PIPERTRAMINE AMIDE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.089046362	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	DESVENLAFAXINE FUMARATE	chembl:CHEMBL3989861	DESVENLAFAXINE FUMARATE	TRUE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	ChEMBL	33	agonist	2.500365296937833	BREMELANOTIDE ACETATE	rxcui:2176311	BREMELANOTIDE ACETATE	TRUE	FALSE	FALSE
EGLN3	hgnc:14661	EGLN3	ChEMBL	33	inhibitor	2.100306849	VADADUSTAT	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.092851762	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	METHYL DEOXYCHOLATE	chembl:CHEMBL1078051	METHYL DEOXYCHOLATE	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.058212496	IUPHAR.LIGAND:7496	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2023	iuphar.ligand:2023	[125I]LTT-SRIF-28	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.1320947704042629	Resminostat	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
ACTIVATION-INDUCIBLE TNFR FAMILY RECEPTOR	hgnc:11914	TNFRSF18	TTD	2020.06.01	NULL	26.25383561784724	TRX-518	drugbank:DB17534	TRX-518	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1458546423213736	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DS2	hgnc:6334	KIR2DS2	TTD	2020.06.01	NULL	10.50153425	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011188509	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.045304289	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.9546849315580819	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.1801292323694494	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.032055965	IUPHAR.LIGAND:2168	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.173866461	APG-115	ncit:C132991	ALRIZOMADLIN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	CID 670282	chembl:CHEMBL260213	CHEMBL:CHEMBL260213	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002663877	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1103102336884338	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
SRI	hgnc:11292	SRI	NCI	14-Sep-17	NULL	1.105424657593568	ADRIAMYCIN	wikidata:Q47520887	ADRIAMYCIN	FALSE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	0.351221881	Sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	1.078924751	RP-3500	ncit:C174206	CAMONSERTIB	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.9907107780319716	SK-7041	chembl:CHEMBL152133	CHEMBL:CHEMBL152133	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	SJ000113107	chembl:CHEMBL589245	CHEMBL:CHEMBL589245	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.021554873	IUPHAR.LIGAND:98	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:4069	drugbank:DB04152	2-AMINO-3-(3-HYDROXY-7,8-DIHYDRO-6H-CYCLOHEPTA[D]-4-ISOXAZOLYL)PROPIONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:7649	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	NULL	0.6250913242344582	IUPHAR.LIGAND:11974	iuphar.ligand:11974	COMPOUND 10 [O'MAHONY ET AL., 2022]	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.054981855	KO-947	iuphar.ligand:9976	KO-947	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	CID 4970947	chembl:CHEMBL1451921	CHEMBL:CHEMBL1451921	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.014206621	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.1136529680426287	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
MYH7	hgnc:7577	MYH7	ChEMBL	33	activator	2.187819634820604	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	agonist	1.500219178	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.08780547	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
TLR2	hgnc:11848	TLR2	PharmGKB	4/5/24	NULL	0.2419708351875322	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	N,N'-DIPHENYL-GUANIDINE	chembl:CHEMBL77675	CHEMBL:CHEMBL77675	FALSE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	NCI	14-Sep-17	NULL	3.029288725136221	BPDE	ncit:C196	BENZO(A)PYRENE-7,8-DIOL 9,10-EPOXIDE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.006100578	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
UNIPROT:Q9UP95	hgnc:10913	SLC12A4	TEND	1-Aug-11	NULL	5.834185692854945	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	ChEMBL	33	agonist	2.187819634820604	LABRADIMIL	ncit:C1606	LABRADIMIL	FALSE	FALSE	FALSE
UNIPROT:Q01118	hgnc:10594	SCN7A	TdgClinicalTrial	Jan-14	NULL	0.057574201	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:8915	iuphar.ligand:8915	AZD8835	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	BENFLUOREX HYDROCHLORIDE	rxcui:235953	BENFLUOREX HYDROCHLORIDE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.078958904	6-CHLOROMELATONIN	iuphar.ligand:1346	6-CL-MLT	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124632	chembl:CHEMBL533399	CHEMBL:CHEMBL533399	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.1458546423213736	THEOPHYLLINE SODIUM GLYCINATE	rxcui:155075	THEOPHYLLINE SODIUM GLYCINATE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TMPRSS15	hgnc:9490	TMPRSS15	DTC	9/2/20	NULL	1.050153425	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	CYSTEINE METHYL-ESTER HCL	chembl:CHEMBL1426508	CHEMBL:CHEMBL1426508	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	GW405833	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1415301111474245	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.078136416	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1000146118775133	INTERFERON ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	0.9723642821424908	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	4.039051633514961	ZEN-3694	ncit:C126805	BET BROMODOMAIN INHIBITOR ZEN-3694	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	1.693795846312725	ANTIMETABOLITE	ncit:C272	ANTIMETABOLITE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003279475	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:10577	iuphar.ligand:10577	ABBV-3221	FALSE	FALSE	FALSE
NCBIGENE:1330	hgnc:2270	COX5BP1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8756	iuphar.ligand:8756	COMPOUND 23 [PMID: 17125252]	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	1.875273972703375	SILMITASERTIB	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.038467158	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	GNF-PF-1872	chembl:CHEMBL600103	CHEMBL:CHEMBL600103	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	1.166837138570988	PAC-1	drugbank:DB13048	PAC-1	FALSE	FALSE	FALSE
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	22.50328767	Tanezumab	ncit:C71522	TANEZUMAB	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II ALPHA	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	PK1	ncit:C1366	DOXORUBICIN-HPMA CONJUGATE	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.100976291	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	0.1417211099478934	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2282942227638891	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.003204618	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	activator	0.212581665	IUPHAR.LIGAND:4804	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	PharmGKB	4/5/24	NULL	0.034830959	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006100578	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.1223955040459079	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1682938180631233	THIOTHIXENE HYDROCHLORIDE	rxcui:91135	THIOTHIXENE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.091317689	Taletrectinib	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.050007306	Fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.384671584	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.094864808	IONOMYCIN	ncit:C596	IONOMYCIN	FALSE	FALSE	FALSE
UNIPROT:P25103	hgnc:11526	TACR1	TdgClinicalTrial	Jan-14	NULL	1.419126249613364	AV608	drugbank:DB05072	AV608	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.3547815624033412	OXYPHENCYCLIMINE	rxcui:32698	OXYPHENCYCLIMINE	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.067317527	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
SIRT6	hgnc:14934	SIRT6	TALC	12-May-16	inhibitor	1.591141552596803	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.01524613	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	NSC-60340	chembl:CHEMBL1534034	CHEMBL:CHEMBL1534034	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005524797	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	PREDNISOLONE TEBUTATE	rxcui:34376	PREDNISOLONE TEBUTATE	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1361	iuphar.ligand:1361	S22153	FALSE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.192335792	phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.003139923	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.045898314	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	SJ000202381	chembl:CHEMBL591598	CHEMBL:CHEMBL591598	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	DTC	9/2/20	NULL	1.458546423213736	LUF-5962	iuphar.ligand:9813	LUF5962	FALSE	FALSE	FALSE
GSTO1	hgnc:13312	GSTO1	NCI	14-Sep-17	NULL	4.039051633514962	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FLUPREDNISOLONE	rxcui:4497	FLUPREDNISOLONE	TRUE	FALSE	FALSE
OXT	hgnc:8528	OXT	PharmGKB	4/5/24	NULL	0.5413161983061289	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TEND	1-Aug-11	NULL	0.6563458904461813	NITRENDIPINE	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.2917092846427472	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	HEXACONAZOLE	chembl:CHEMBL1898860	HEXACONAZOLE	FALSE	FALSE	FALSE
HEPATOCYTE GROWTH FACTOR	hgnc:4893	HGF	TTD	2020.06.01	NULL	1.944728564284981	TAK-701	ncit:C81939	ANTI-HGF MONOCLONAL ANTIBODY TAK-701	FALSE	FALSE	FALSE
NCBIGENE:562	hgnc:6297	KCNQ3	GuideToPharmacology	2024.1	activator	3.750547945	IUPHAR.LIGAND:12650	ncit:C188540	AZETUKALNER	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	NCI	14-Sep-17	NULL	0.01242344	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CALCR	hgnc:1440	CALCR	ChEMBL	33	agonist	1.640864726115453	DAVALINTIDE	ncit:C83650	DAVALINTIDE	FALSE	FALSE	FALSE
FN1	hgnc:3778	FN1	ChEMBL	33	binder	4.039051633514961	L19TNFA	chembl:CHEMBL2109589	L19TNFA	FALSE	FALSE	FALSE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	inhibitor	4.039051633514961	MIK-BETA-1	chembl:CHEMBL2109326	MIK-BETA-1	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	2.187819634820604	EPITUMOMAB CITUXETAN	ncit:C175781	EPITUMOMAB CITUXETAN	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.008317388	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.070860555	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	TECADENOSON	ncit:C77980	TECADENOSON	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.031621603	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	DNDI1417701	chembl:CHEMBL1326164	CHEMBL:CHEMBL1326164	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.089501712	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ORTHOTOLIDINE	chembl:CHEMBL85109	ORTHOTOLIDINE	FALSE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:8550	iuphar.ligand:8550	COMPOUND 24DD [PMID: 20684603]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2970	iuphar.ligand:2970	COMPOUND 4FF [PMID: 1656041]	FALSE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9667	iuphar.ligand:9667	ZIMLOVISERTIB	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.005204963	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2417	hgnc:3928	FRA7J	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6539	iuphar.ligand:6539	ST074946	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	1.000146118775133	GALLOCATECHIN GALLATE	chembl:CHEMBL264938	GALLOCATECHIN GALLATE	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.010434752	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	NSC-133896	chembl:CHEMBL512908	CHEMBL:CHEMBL512908	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.2651902587661338	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
IVL	hgnc:6187	IVL	NCI	14-Sep-17	NULL	5.834185692854944	TOPICAL CORTICOSTEROIDS	ncit:C29505	TOPICAL CORTICOSTEROID	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.062509132	sertraline	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00411841	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.040390516	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	ETHCHLORVYNOL	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
RARG	hgnc:9866	RARG	ChEMBL	33	inhibitor	1.029562181092048	IRX4310	chembl:CHEMBL3545173	IRX4310	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.4773424657790409	RILPIVIRINE	rxcui:1102270	RILPIVIRINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.00429616	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.105015342	Topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.073540156	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1635752997996713	FAXELADOL	ncit:C80579	FAXELADOL	FALSE	FALSE	FALSE
RHOA	hgnc:667	RHOA	PharmGKB	4/5/24	NULL	0.5556367326528519	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.039778539	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.1117184494376478	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GNF-PF-1241	chembl:CHEMBL528724	CHEMBL:CHEMBL528724	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:8978	iuphar.ligand:8978	QUINOSTATIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	2-MERCAPTONICOTINIC ACID	chembl:CHEMBL1521174	2-MERCAPTONICOTINIC ACID	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.1458546423213736	GNF-PF-3716	chembl:CHEMBL609606	CHEMBL:CHEMBL609606	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	PARBENDAZOLE	ncit:C96752	PARBENDAZOLE	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.1389091831632129	AL3818	ncit:C138997	ANLOTINIB	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	ATEVIRDINE MESYLATE	ncit:C73148	ATEVIRDINE MESYLATE	FALSE	FALSE	FALSE
UNIPROT:P49327	hgnc:3594	FASN	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	GT 389-255	drugbank:DB05894	GT 389-255	FALSE	FALSE	FALSE
CDH13	hgnc:1753	CDH13	PharmGKB	4/5/24	NULL	0.057291513	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	5.834185692854944	Molgramostim	rxcui:70161	MOLGRAMOSTIM	FALSE	FALSE	FALSE
UNIPROT:Q9UP95	hgnc:10913	SLC12A4	TdgClinicalTrial	Jan-14	NULL	5.834185692854945	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
STAG3	hgnc:11356	STAG3	CIViC	10-Apr-24	NULL	1.458546423213736	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	Polyglutamate camptothecin	ncit:C26664	POLYGLUTAMATE CAMPTOTHECIN	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:9882	iuphar.ligand:9882	TIQ-15	FALSE	FALSE	FALSE
KLKB1	hgnc:6371	KLKB1	ChEMBL	33	inhibitor	7.501095891	LANADELUMAB	rxcui:2055640	LANADELUMAB-FLYO	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	PIMURUTAMAB	ncit:C163981	PIMURUTAMAB	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.4449802647092754	LISINOPRIL	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:7571	iuphar.ligand:7571	PROTOXIN II	FALSE	FALSE	FALSE
UNIPROT:P39877	hgnc:9038	PLA2G5	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	VARESPLADIB	ncit:C152832	VARESPLADIB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	CHRYSEN-6-YLAMINE	chembl:CHEMBL313154	CHEMBL:CHEMBL313154	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.019318496	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.09869863	IUPHAR.LIGAND:2031	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.043692674	Aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1077080435603989	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ROBUSTONE	chembl:CHEMBL252722	ROBUSTONE	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1785975212098452	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.3431873936973497	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.2853677784548614	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:6797	rxcui:194881	BRINZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:5963	iuphar.ligand:5963	EGFR INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.025739055	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11742	ncit:C169812	BIFEMELANE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.2368767123414789	LY2874455	iuphar.ligand:8104	LY2874455	FALSE	FALSE	FALSE
ATF2	hgnc:784	ATF2	NCI	14-Sep-17	NULL	1.591141552596803	ALPHA-DIFLUOROMETHYLORNITHINE	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
ERK ACTIVATOR KINASE 2	hgnc:6842	MAP2K2	TTD	2020.06.01	NULL	0.1808115400678185	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:2377	hgnc:3889	FRA2E	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8488	iuphar.ligand:8488	COMPOUND 3 [PMID: 23849879]	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.069454592	Linsitinib	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.027752469	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.1105424657593568	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	TCMDC-125353	chembl:CHEMBL547924	CHEMBL:CHEMBL547924	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:419	iuphar.ligand:419	CV-1674	FALSE	FALSE	FALSE
CCL22	hgnc:10621	CCL22	NCI	14-Sep-17	NULL	5.834185692854944	RANTES	ncit:C1211	RECOMBINANT RANTES	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.157680694	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:O14786	hgnc:8004	NRP1	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
PTGER4	hgnc:9596	PTGER4	NCI	14-Sep-17	NULL	0.158394182	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:7461	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:6196	iuphar.ligand:6196	BAYCYSLT2	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:7651	iuphar.ligand:7651	UNC0006	FALSE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:10119	iuphar.ligand:10119	AM-6120	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.045421861	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:5260	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5649	iuphar.ligand:5649	TYR3-OCTREOTIDE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	NSC-7387	chembl:CHEMBL119878	CHEMBL:CHEMBL119878	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.3684748858645227	ISORHAMNETIN	drugbank:DB16767	ISORHAMNETIN	FALSE	FALSE	FALSE
METAP2	hgnc:16672	METAP2	ChEMBL	33	inhibitor	6.563458904461812	ACLIMOSTAT	ncit:C169760	ACLIMOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.091796628	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	1.458546423213736	E-7016	chembl:CHEMBL3527000	E-7016	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.4782119420372905	MEGESTROL	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
NCBIGENE:2917	hgnc:4599	GRM7	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:9421	iuphar.ligand:9421	ITOLIZUMAB	FALSE	FALSE	FALSE
GZMA	hgnc:4708	GZMA	NCI	14-Sep-17	NULL	7.501095891	CC CHEMOKINES	ncit:C1591	RECOMBINANT BETA CHEMOKINE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DoCM	10-Apr-24	NULL	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
POLR3G	hgnc:30075	POLR3G	PharmGKB	4/5/24	NULL	4.773424657790409	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.022869195	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.050879526	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.071148606	DIURETIC	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.026227608	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN CD47	hgnc:1682	CD47	TTD	2020.06.01	NULL	4.375639269641208	Hu5F9-G4	ncit:C117730	MAGROLIMAB	FALSE	FALSE	FALSE
CAST	hgnc:1515	CAST	NCI	14-Sep-17	NULL	2.143170254518142	ACE INHIBITOR	ncit:C247	ACE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	1.458546423213736	IUPHAR.LIGAND:10299	iuphar.ligand:10299	ISOSAKURANETIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	TYRPHOSTIN 1	iuphar.ligand:5917	AG 9	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	TECHTOCHRYSIN	chembl:CHEMBL164841	TECHTOCHRYSIN	FALSE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	0.280789686	Donitriptan	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.049770304	IUPHAR.LIGAND:11893	iuphar.ligand:11893	COMPOUND 6 [PMID: 34333981]	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.089501712	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009320613	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.010422325	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	inhibitor	0.1187956362798518	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	TIOXOLONE	rxcui:2059173	TIOXOLONE	FALSE	FALSE	FALSE
TPSD1	hgnc:14118	TPSD1	NCI	14-Sep-17	NULL	7.501095890813499	CETIRIZINE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.043866058	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:636	iuphar.ligand:636	D-LYS0-[DES-ARG10]KALLIDIN	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:2862	iuphar.ligand:2862	HYDROXYFLUTAMIDE	FALSE	FALSE	FALSE
UNIPROT:P06730	hgnc:3287	EIF4E	TdgClinicalTrial	Jan-14	NULL	1.810609352954982	LY2275796	drugbank:DB05165	LY2275796	FALSE	FALSE	FALSE
UNIPROT:P34972	hgnc:2160	CNR2	TdgClinicalTrial	Jan-14	NULL	0.1187956362798518	TETRAHYDROCANNABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	1.282909942931453	ENCORAFENIB	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:2007	iuphar.ligand:2007	CORTISTATIN-14	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	ALACHLOR	chembl:CHEMBL1414154	ALACHLOR	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.041672755	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:9787	drugbank:DB12903	DEBIO-1347	FALSE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	NCI	14-Sep-17	NULL	0.326134604	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.058602312	IUPHAR.LIGAND:5695	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.010704928	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	TCMDC-123598	chembl:CHEMBL547269	CHEMBL:CHEMBL547269	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR BETA-2	hgnc:1962	CHRNB2	TTD	2020.06.01	NULL	1.458546423213736	SUVN-911	iuphar.ligand:10700	SUVN-911	FALSE	FALSE	FALSE
TXNRD2	hgnc:18155	TXNRD2	PharmGKB	4/5/24	NULL	0.7721716358190368	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.2917092846427472	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1935172158563679	OXYBUTYNIN CHLORIDE	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:9814	iuphar.ligand:9814	CCT241161	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2333674277141978	DIFAMILAST	ncit:C169909	DIFAMILAST	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.2853677784548614	ALPHA-ADRENERGIC AGONIST	ncit:C29709	ALPHA-ADRENERGIC AGONIST	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CancerCommons	25-Jul-13	inhibitor	0.6019397937072561	PF-00299804	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	CancerCommons	25-Jul-13	inhibitor	1.521961485092594	ASP3026	ncit:C116727	ALK INHIBITOR ASP3026	FALSE	FALSE	TRUE
TOLL-LIKE RECEPTOR 2	hgnc:11848	TLR2	TTD	2020.06.01	NULL	2.500365296937833	Cadi-05	ncit:C77884	TLR AGONIST CADI-05	FALSE	FALSE	FALSE
CLU	hgnc:2095	CLU	CancerCommons	25-Jul-13	inhibitor	8.751278539282415	OGX-011	ncit:C1055	CUSTIRSEN SODIUM	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.6241137025199848	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	CGI	2/1/22	NULL	0.042259695	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	1.657092009619794	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CGI	2/1/22	NULL	0.1396480617970598	Veliparib	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.05454398	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	MEPIVACAINE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FLCN	hgnc:27310	FLCN	CGI	2/1/22	NULL	1.500219178	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.020320306	Exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.02103111	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
SH2B3	hgnc:29605	SH2B3	CGI	2/1/22	NULL	4.633029814914221	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	PHENAZINE-2,3-DIAMINE	chembl:CHEMBL274921	CHEMBL:CHEMBL274921	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	CGI	2/1/22	NULL	0.028413242	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	CGI	2/1/22	NULL	1.678633990910949	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CGI	2/1/22	NULL	0.049275217	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1115286134997759	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	CGI	2/1/22	NULL	0.4906052389860809	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.041508041	Cediranib	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CGI	2/1/22	NULL	0.2639729920045843	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	PROCYCLIDINE	rxcui:8718	PROCYCLIDINE	TRUE	FALSE	FALSE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.3913615247380956	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
TSC2	hgnc:12363	TSC2	CGI	2/1/22	NULL	2.250328767	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
TOP2A	hgnc:11989	TOP2A	CGI	2/1/22	NULL	0.1508841127462485	Anthracyclines	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.2365210416022274	TOLTERODINE TARTRATE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:819	iuphar.ligand:819	CXCL1	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	CGI	2/1/22	NULL	0.3472729579080323	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.064505739	TROPICAMIDE	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	SOLIFENACIN SUCCINATE	rxcui:476588	SOLIFENACIN SUCCINATE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.7095631248066824	TIOTROPIUM BROMIDE	rxcui:393575	TIOTROPIUM BROMIDE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.8899605294185507	SPIRAPRIL HYDROCHLORIDE	ncit:C66561	SPIRAPRIL HYDROCHLORIDE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.4123639102279672	Belvarafenib	ncit:C121646	BELVARAFENIB	FALSE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	PROPIOMAZINE HYDROCHLORIDE	rxcui:6232	PROPIOMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3677319929494733	LAPATINIB DITOSYLATE	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	PROCYCLIDINE HYDROCHLORIDE	rxcui:142443	PROCYCLIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1396480617970598	METHIXENE HYDROCHLORIDE	rxcui:258230	METHIXENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:324	iuphar.ligand:324	HIMBACINE	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	0.1902451856365742	HYDROCHLOROTHIAZIDE	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1988926940746003	CLOMIPRAMINE HYDROCHLORIDE	rxcui:81984	CLOMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	3.281729452230906	CIMETIDINE HYDROCHLORIDE	rxcui:91251	CIMETIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.351221881	SUMATRIPTAN SUCCINATE	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP PURIFIED BEEF/PORK	chembl:CHEMBL1201634	INSULIN ZINC SUSP PURIFIED BEEF/PORK	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.4907258993990139	PSEUDOEPHEDRINE POLISTIREX	rxcui:407885	PSEUDOEPHEDRINE POLISTIREX	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.08178765	NEFAZODONE HYDROCHLORIDE	rxcui:236082	NEFAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	ChEMBL	33	blocker	0.5834185692854944	VERNAKALANT HYDROCHLORIDE	ncit:C152865	VERNAKALANT HYDROCHLORIDE	FALSE	FALSE	FALSE
CA12	hgnc:1371	CA12	ChEMBL	33	inhibitor	0.8036888454443035	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.047647615	PAZOPANIB HYDROCHLORIDE	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.3182283105193605	RALTEGRAVIR POTASSIUM	rxcui:1235585	RALTEGRAVIR POTASSIUM	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.2151953739167807	HYDROXYPROGESTERONE CAPROATE	rxcui:12488	HYDROXYPROGESTERONE CAPROATE (USP)	TRUE	FALSE	FALSE
CA14	hgnc:1372	CA14	ChEMBL	33	inhibitor	0.8751278539282417	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
CA4	hgnc:1375	CA4	ChEMBL	33	inhibitor	0.2917092846427472	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.035574303	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.029766254	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
PSMB6	hgnc:9543	PSMB6	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.02875557	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.029106248	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.033701971	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.031631127	VINBLASTINE SULFATE	rxcui:11199	VINBLASTINE SULFATE	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.042689164	VINORELBINE TARTRATE	rxcui:114527	VINORELBINE TARTRATE	TRUE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.080781033	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.063415062	ARRY-614	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1071585127259071	AMANTADINE HYDROCHLORIDE	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2275522047050683	CLONIDINE HYDROCHLORIDE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.087222045	TETRAHYDROZOLINE HYDROCHLORIDE	rxcui:57983	TETRAHYDROZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.1154014752432845	TETRAHYDROZOLINE HYDROCHLORIDE	rxcui:57983	TETRAHYDROZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.042073455	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
RRM2	hgnc:10452	RRM2	ChEMBL	33	inhibitor	0.1187956362798518	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.487687349	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2035181055647073	ESMOLOL HYDROCHLORIDE	rxcui:203222	ESMOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2652	hgnc:4206	OPN1MW	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7015	iuphar.ligand:7015	UNC0638	FALSE	FALSE	FALSE
LAMB1	hgnc:6486	LAMB1	ChEMBL	33	cleavage	0.6908904109959803	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:9918	ncit:C104732	SAVOLITINIB	FALSE	FALSE	TRUE
LAMC3	hgnc:6494	LAMC3	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
LAMB4	hgnc:6491	LAMB4	ChEMBL	33	cleavage	1.381780822	OCRIPLASMIN	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.028498058	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.7160136986685613	ETODOLAC	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	agonist	0.251232877	SUCCINYLCHOLINE CHLORIDE	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	negative modulator	0.02804897	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.075442056	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	CHLORDIAZEPOXIDE HYDROCHLORIDE	rxcui:203173	CHLORDIAZEPOXIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.056500364	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	METHOHEXITAL SODIUM	rxcui:91185	METHOHEXITAL SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.053361455	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	MyCancerGenome	20-Jun-17	inhibitor	0.033232703	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.100976291	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.036770078	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.096758608	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1750255707856483	CHLORTETRACYCLINE HYDROCHLORIDE	rxcui:42545	CHLORTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	QUINUPRISTIN	rxcui:229367	QUINUPRISTIN	TRUE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	modulator	0.1852122442176172	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
PSMD10	hgnc:9555	PSMD10	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	modulator	0.045226246	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	modulator	0.2778183663264259	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
KCNK10	hgnc:6273	KCNK10	ChEMBL	33	potentiator	0.3387591692625452	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	modulator	0.2160809515872201	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	modulator	0.092606122	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	modulator	0.2160809515872201	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	modulator	0.2160809515872201	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	modulator	0.046303061	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	modulator	0.1495945049449985	GABAPENTIN ENACARBIL	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.067317527	CHLOROPROCAINE HYDROCHLORIDE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	PROCAINE HYDROCHLORIDE	rxcui:106558	PROCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.067317527	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.054243462	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.03591496	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	ABAMECTIN	ncit:C95196	ABAMECTIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.047886613	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
KCNK2	hgnc:6277	KCNK2	ChEMBL	33	potentiator	0.2419708351875322	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.006811217	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNK9	hgnc:6283	KCNK9	ChEMBL	33	potentiator	0.2822993077187876	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.008395854	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PTGIR	hgnc:9602	PTGIR	ChEMBL	33	agonist	3.750547945	TREPROSTINIL DIOLAMINE	rxcui:1927409	TREPROSTINIL DIOLAMINE	TRUE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	3.580068493342807	SUVOREXANT	rxcui:1547099	SUVOREXANT	TRUE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	0.3977853881492008	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.2386712328895204	OXTRIPHYLLINE	rxcui:20976	OXTRIPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.1442518440541057	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
PSMD14	hgnc:16889	PSMD14	ChEMBL	33	inhibitor	0.1035654265003836	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
PSMB6	hgnc:9543	PSMB6	ChEMBL	33	inhibitor	0.2243917574174978	IXAZOMIB CITRATE	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	CEP-7055	chembl:CHEMBL346631	CEP-7055	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.048083948	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.032055965	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1825	iuphar.ligand:1825	[ILE5]PTHRP-(1-36)	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1000146118775133	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.089756703	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	1.000146118775133	EMD-1204831	chembl:CHEMBL3545053	EMD-1204831	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.089756703	FIMEPINOSTAT	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	ChEMBL	33	inhibitor	0.180026301	RAVOXERTINIB	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.053854022	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.064190307	HMPL-306	ncit:C175602	IDH1/IDH2 DUAL INHIBITOR HMPL-306	FALSE	FALSE	FALSE
PRKD1	hgnc:9407	PRKD1	ChEMBL	33	inhibitor	0.3088686543276147	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	THELIATINIB	chembl:CHEMBL3545180	THELIATINIB	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.1143957978991165	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	OLMUTINIB	ncit:C101791	OLMUTINIB	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.043502627	GSK-690693	drugbank:DB12745	GSK-690693	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.1112450661773188	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.08914715	CRYSTAL VIOLET	rxcui:1546369	GENTIAN VIOLET CATION	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1416573864272333	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	2.019525817	RG-7376	chembl:CHEMBL3545082	RG-7376	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	2.763561643983921	SCH-900776	chembl:CHEMBL2386889	SCH-900776	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	1.381780822	RG-7741	chembl:CHEMBL3545199	RG-7741	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.6250913242344582	RO-4987655	drugbank:DB12933	RO-4987655	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.1315981735230438	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005297384	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.044878351	SF-1126	chembl:CHEMBL2326966	SF-1126	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	MUBRITINIB	ncit:C66212	MUBRITINIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.006495259	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	LAS190792	chembl:CHEMBL3545272	LAS190792	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.013299815	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	2.143170254518142	Siltuximab	rxcui:1535218	SILTUXIMAB	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.010440977	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.2778183663264258	ALPELISIB	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.060772768	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1682938180631233	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.052090944	VOXTALISIB	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PRKCH	hgnc:9403	PRKCH	ChEMBL	33	inhibitor	0.2386712328895204	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	ChEMBL	33	inhibitor	0.1312691780892362	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	ChEMBL	33	inhibitor	0.091159151	TG100-801	chembl:CHEMBL403989	TG100-801	FALSE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.3454452054979901	OXYBUPROCAINE	rxcui:18889	BENOXINATE	TRUE	FALSE	FALSE
UTS2R	hgnc:4468	UTS2R	ChEMBL	33	inhibitor	3.621218705909965	PALOSURAN	ncit:C66298	PALOSURAN	FALSE	FALSE	FALSE
NPY5R	hgnc:7958	NPY5R	ChEMBL	33	inhibitor	15.00219178	VELNEPERIT	ncit:C152850	VELNEPERIT	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Pepinemab	ncit:C96222	PEPINEMAB	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.3365876361262467	TRELANSERIN	ncit:C90946	TRELANSERIN	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	inhibitor	0.3431873936973497	RELCOVAPTAN	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.3621218705909966	HONOKIOL	rxcui:2562546	HONOKIOL	FALSE	FALSE	FALSE
NPY4R	hgnc:9329	NPY4R	ChEMBL	33	agonist	52.50767123569449	TM30339	drugbank:DB05085	TM30339	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	agonist	0.8751278539282416	DAVALINTIDE	ncit:C83650	DAVALINTIDE	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.108711535	GW468816	chembl:CHEMBL1207366	GW468816	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	1.117184494376478	ISPRONICLINE	ncit:C65986	ISPRONICLINE	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1651184630053286	AZD1305	chembl:CHEMBL3545169	AZD1305	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1530835896084387	GW468816	chembl:CHEMBL1207366	GW468816	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SKF-75670 HYDROBROMIDE	chembl:CHEMBL1256698	CHEMBL:CHEMBL1256698	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.5585922471882393	POZANICLINE	ncit:C81045	POZANICLINE	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.016156207	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.018423744	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.4688184931758437	NSC-628113	chembl:CHEMBL176599	CHEMBL:CHEMBL176599	FALSE	FALSE	FALSE
KCNC3	hgnc:6235	KCNC3	ChEMBL	33	blocker	0.1750255707856483	NERISPIRDINE	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	positive modulator	0.3125456621172291	MK-8777	chembl:CHEMBL3707401	MK-8777	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	ChEMBL	33	inhibitor	4.375639269641208	GRC-17536	chembl:CHEMBL3707318	GRC-17536	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.1973972602845657	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.04464938	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.035800685	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.1187956362798518	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.1562728310586145	ESMIRTAZAPINE MALEATE	ncit:C76940	ESMIRTAZAPINE MALEATE	FALSE	FALSE	FALSE
GRM3	hgnc:4595	GRM3	ChEMBL	33	agonist	2.625383561784724	POMAGLUMETAD METHIONIL	ncit:C170541	POMAGLUMETAD METHIONIL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.7395446652914718	RIVOCERANIB MESYLATE	ncit:C74012	RIVOCERANIB MESYLATE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007479725	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	inhibitor	0.8751278539282416	OTENABANT	ncit:C84034	OTENABANT	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	1.312691780892362	APLAVIROC HYDROCHLORIDE	ncit:C76492	APLAVIROC HYDROCHLORIDE	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.070574827	ESMIRTAZAPINE MALEATE	ncit:C76940	ESMIRTAZAPINE MALEATE	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.010923169	IUPHAR.LIGAND:5679	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.1640864726115453	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.033658764	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.097236428	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.038049037	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.031254566	RALFINAMIDE	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	inhibitor	1.458546423213736	DEXMECAMYLAMINE	ncit:C166871	DEXMECAMYLAMINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.013259513	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ITGB7	hgnc:6162	ITGB7	ChEMBL	33	inhibitor	17.50255707856483	ETROLIZUMAB	ncit:C97944	ETROLIZUMAB	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	ChEMBL	33	inhibitor	1.810609352954982	ODULIMOMAB	ncit:C188506	ODULIMOMAB	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.043003826	IUPHAR.LIGAND:7317	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
SOST	hgnc:13771	SOST	ChEMBL	33	inhibitor	13.12691780892362	ROMOSOZUMAB	rxcui:2123126	ROMOSOZUMAB	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	ChEMBL	33	other/unknown	2.386712328895204	LYM-1	chembl:CHEMBL2109447	LYM-1	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	1.250182648468916	AZD8330	iuphar.ligand:8474	AZD8330	FALSE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.042689164	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.042174836	CROLIBULIN	ncit:C66938	CROLIBULIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	negative modulator	0.042689164	FOSBRETABULIN TROMETHAMINE	ncit:C83721	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.640864726115453	REMOGLIFLOZIN ETABONATE	ncit:C91023	REMOGLIFLOZIN ETABONATE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.037666909	FOSBRETABULIN DISODIUM	ncit:C2503	FOSBRETABULIN DISODIUM	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.055563673	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
MYH6	hgnc:7576	MYH6	ChEMBL	33	activator	2.187819634820604	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
MYH7B	hgnc:15906	MYH7B	ChEMBL	33	activator	2.187819634820604	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	modulator	0.9723642821424906	ERTUMAXOMAB	ncit:C2658	ERTUMAXOMAB	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	ALCLOFENAC	ncit:C174701	ALCLOFENAC	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.021519537	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	FENOTEROL	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	METHAQUALONE HYDROCHLORIDE	ncit:C2484	METHAQUALONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.046965717	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	blocker	0.1442518440541058	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.048083948	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.096167896	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.046965717	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	blocker	0.2243917574174979	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	THENALIDINE	ncit:C84198	THENALIDINE	TRUE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	blocker	0.1553481397505754	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	blocker	0.2243917574174979	SULOCTIDIL	ncit:C152466	SULOCTIDIL	TRUE	FALSE	FALSE
HTR5A	hgnc:5300	HTR5A	ChEMBL	33	inhibitor	0.7721716358190368	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	3.443125982668491	TOVETUMAB	ncit:C82684	TOVETUMAB	FALSE	TRUE	TRUE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.2206204673768676	ZIMELDINE HYDROCHLORIDE	ncit:C152955	ZIMELDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1F	hgnc:5292	HTR1F	ChEMBL	33	inhibitor	0.1835932560688619	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.111481255	ALFACALCIDOL	rxcui:12062	ALFACALCIDOL	TRUE	FALSE	FALSE
CD70	hgnc:11937	CD70	ChEMBL	33	binder	4.039051633514961	VORSETUZUMAB MAFODOTIN	ncit:C88315	VORSETZUMAB MAFODOTIN	FALSE	FALSE	FALSE
CALCR	hgnc:1440	CALCR	ChEMBL	33	agonist	2.187819634820604	CALCITONIN	rxcui:1311287	CALCITONIN	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.1495945049449985	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.1296485709523321	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.4167275494896389	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.3431873936973497	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.4167275494896389	CLOTHIAPINE	rxcui:2620	CLOTHIAPINE	TRUE	FALSE	FALSE
MSLN	hgnc:7371	MSLN	ChEMBL	33	binder	5.834185692854944	SS1(DSFV)-PE38	drugbank:DB17579	SS1(DSFV)-PE38	FALSE	FALSE	FALSE
BSG	hgnc:1116	BSG	ChEMBL	33	inhibitor	6.563458904461812	ZIRALIMUMAB	ncit:C188597	ZIRALIMUMAB	FALSE	FALSE	FALSE
CD5	hgnc:1685	CD5	ChEMBL	33	binder	5.250767123569449	TELIMOMAB ARITOX	ncit:C2358	TELIMOMAB ARITOX	FALSE	FALSE	FALSE
TNFRSF18	hgnc:11914	TNFRSF18	ChEMBL	33	agonist	26.25383561784724	TRX-518	drugbank:DB17534	TRX-518	FALSE	FALSE	FALSE
HCN4	hgnc:16882	HCN4	ChEMBL	33	blocker	2.917092846427472	IVABRADINE	rxcui:1649480	IVABRADINE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.028413242	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.2035181055647073	LOFEXIDINE HYDROCHLORIDE	rxcui:235853	LOFEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.029766254	BREXANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	NARLAPREVIR	ncit:C166554	NARLAPREVIR	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.07631929	AVIPTADIL	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
PORCN	hgnc:17652	PORCN	ChEMBL	33	inhibitor	26.25383561784724	WNT-974	drugbank:DB12561	WNT-974	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.4070362111294147	SELITRECTINIB	ncit:C138160	SELITRECTINIB	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	ChEMBL	33	inhibitor	1.250182648468916	OPICAPONE	rxcui:2362167	OPICAPONE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.2500365296937833	NITRENDIPINE	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
TNKS	hgnc:11941	TNKS	ChEMBL	33	inhibitor	13.12691780892362	2X-121	drugbank:DB16063	2X-121	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	1.050153425	2X-121	drugbank:DB16063	2X-121	FALSE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	positive modulator	0.729273212	OLINCIGUAT	ncit:C153148	OLINCIGUAT	FALSE	FALSE	FALSE
PDE9A	hgnc:8795	PDE9A	ChEMBL	33	inhibitor	6.563458904461812	PF-04447943	drugbank:DB11953	PF-04447943	FALSE	FALSE	FALSE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	2.187819634820604	ROMILKIMAB	ncit:C174791	ROMILKIMAB	FALSE	FALSE	FALSE
HAVCR2	hgnc:18437	HAVCR2	ChEMBL	33	inhibitor	8.751278539282415	COBOLIMAB	ncit:C128627	COBOLIMAB	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	ChEMBL	33	agonist	1.544343271638073	TILSOTOLIMOD	ncit:C152632	TILSOTOLIMOD	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	AUMOLERTINIB	ncit:C133691	AUMOLERTINIB	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	2.282942227638891	JNJ-41443532	drugbank:DB12632	JNJ-41443532	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	negative modulator	0.8468979231563628	DEUCRAVACITINIB	rxcui:2612087	DEUCRAVACITINIB	TRUE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.8468979231563628	DEUCRAVACITINIB	rxcui:2612087	DEUCRAVACITINIB	TRUE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	1.640864726115453	PF-00489791	drugbank:DB11736	PF-00489791	FALSE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	ChEMBL	33	inhibitor	1.810609352954982	AT-1501	chembl:CHEMBL4594460	AT-1501	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	positive modulator	0.5585922471882393	MK-7622	drugbank:DB12897	MK-7622	FALSE	FALSE	FALSE
KDM1A	hgnc:29079	KDM1A	ChEMBL	33	inhibitor	2.625383561784724	BOMEDEMSTAT	ncit:C131827	BOMEDEMSTAT	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.061055432	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
LGALS1	hgnc:6561	LGALS1	ChEMBL	33	inhibitor	26.25383561784724	DAVANAT	drugbank:DB15311	DAVANAT	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.037213091	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	SAMIDORPHAN L-MALATE	rxcui:2570387	SAMIDORPHAN L-MALATE	TRUE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.7721716358190367	RUNCACIGUAT	ncit:C166842	RUNCACIGUAT	FALSE	FALSE	FALSE
MMP14	hgnc:7160	MMP14	ChEMBL	33	inhibitor	1.071585127259071	CTS-1027	drugbank:DB08490	CTS-1027	FALSE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	ChEMBL	33	agonist	4.922594178346359	RESIQUIMOD	ncit:C63958	RESIQUIMOD	FALSE	FALSE	FALSE
IL1RL1	hgnc:5998	IL1RL1	ChEMBL	33	inhibitor	17.50255707856483	ASTEGOLIMAB	ncit:C171824	ASTEGOLIMAB	FALSE	FALSE	FALSE
IL1RAP	hgnc:5995	IL1RAP	ChEMBL	33	inhibitor	5.834185692854944	ASTEGOLIMAB	ncit:C171824	ASTEGOLIMAB	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	agonist	0.7001022831425933	PUMOSETRAG	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	1.750255707856483	ZALUNFIBAN	ncit:C180665	ZALUNFIBAN	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	3.500511415712966	ZANSECIMAB	ncit:C177075	ZANSECIMAB	FALSE	FALSE	FALSE
NPY2R	hgnc:7957	NPY2R	ChEMBL	33	agonist	6.563458904461812	PEPTIDE YY HUMAN (3-36)	chembl:CHEMBL4297971	PEPTIDE YY HUMAN (3-36)	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.3547815624033412	ULOTARONT	ncit:C179130	ULOTARONT	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	agonist	0.5048814541893701	PSILOCYBINE	ncit:C62529	PSILOCYBINE	FALSE	FALSE	FALSE
PARP3	hgnc:273	PARP3	ChEMBL	33	inhibitor	2.917092846427472	E-7016	chembl:CHEMBL3527000	E-7016	FALSE	FALSE	FALSE
GCK	hgnc:4195	GCK	ChEMBL	33	activator	7.001022831425932	LY-2608204	drugbank:DB12284	LY-2608204	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.037213091	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	binder	3.043922970185188	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
S1PR3	hgnc:3167	S1PR3	ChEMBL	33	binder	2.625383561784725	FINGOLIMOD LAURYL SULFATE	rxcui:2610292	FINGOLIMOD LAURYL SULFATE	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.022099188	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3088686543276147	E7449	ncit:C102746	PARP/TANKYRASE INHIBITOR 2X-121	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.443726799	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.9845188356692719	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2778183663264258	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.088396753	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1400204566285186	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
AKT3	hgnc:393	AKT3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3076621361466474	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	2.341819737097098	GSK 2118436	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
ERBB5	hgnc:3430	ERBB2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ERBB6	hgnc:3430	ERBB2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
PRKAA2	hgnc:9377	PRKAA2	ClearityFoundationClinicalTrial	15-Jun-13	activator	0.2557191780959147	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PREDNICARBATE	rxcui:34369	PREDNICARBATE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.090821275	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.011171845	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	FUROXAN	chembl:CHEMBL336467	FUROXAN	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.1131630845596864	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	NSC-83217	chembl:CHEMBL120806	CHEMBL:CHEMBL120806	FALSE	FALSE	FALSE
ARG1	hgnc:663	ARG1	DTC	9/2/20	NULL	5.000730593875666	L-2-AMINOHISTIDINE	chembl:CHEMBL1099167	CHEMBL:CHEMBL1099167	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.056826484	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1274458039701322	HELIOMYCIN	ncit:C75147	HELIOMYCIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002258977	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
PSMC5	hgnc:9552	PSMC5	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.3070624048871023	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012794267	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.2051080907644316	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006756874	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008176218	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.038693936	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.02321294	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	5-NITRO-[1,10]PHENANTHROLINE	chembl:CHEMBL101815	CHEMBL:CHEMBL101815	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.036337489	ALEXIDINE HYDROCHLORIDE	chembl:CHEMBL1487183	ALEXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	SL-327	iuphar.ligand:6008	MEK1/2 INHIBITOR	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.066297565	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	ISONIAZID	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	NSC-636948	chembl:CHEMBL1998001	CHEMBL:CHEMBL1998001	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.041672755	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	BISPHENOL A	rxcui:1433347	BISPHENOL A	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.008460791	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	DNDI1417457	chembl:CHEMBL1530911	CHEMBL:CHEMBL1530911	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	ETIDRONIC ACID	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	SB-203186	iuphar.ligand:255	SB 203186	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SYROSINGOPINE	ncit:C152485	SYROSINGOPINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	ESCULIN	rxcui:1314351	ESCULIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004698673	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	TETROQUINONE	chembl:CHEMBL1329029	TETROQUINONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	METHOXYVONE	chembl:CHEMBL1591080	METHOXYVONE	FALSE	FALSE	FALSE
MAPK7	hgnc:6880	MAPK7	DTC	9/2/20	NULL	52.50767123569449	XMD8-85	chembl:CHEMBL1673039	CHEMBL:CHEMBL1673039	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	IRETOL	chembl:CHEMBL1606248	IRETOL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-5478	chembl:CHEMBL586982	CHEMBL:CHEMBL586982	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.037884323	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.2019525816757481	TANNIC ACID	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	2-PHENYLPHENOL	rxcui:236677	2-PHENYLPHENOL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	RS-67506	iuphar.ligand:3230	RS67506	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	GNF-PF-1872	chembl:CHEMBL600103	CHEMBL:CHEMBL600103	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1060761035064535	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.3062196950280639	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	4-(HEXYLOXY)PHENOL	chembl:CHEMBL225563	CHEMBL:CHEMBL225563	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.6563458904461813	DNDI1416917	chembl:CHEMBL1335833	CHEMBL:CHEMBL1335833	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1141471113819445	4-NONYLPHENOL	rxcui:1788868	4-NONYLPHENOL	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.012582715	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	CEAROIN	chembl:CHEMBL1613209	CEAROIN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	NITIDINE CHLORIDE	chembl:CHEMBL8443	NITIDINE CHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	BINOSPIRONE	ncit:C79884	BINOSPIRONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	DAIDZIN	drugbank:DB02115	DAIDZIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	MK-571	iuphar.ligand:10346	MK-571	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	ETICLOPRIDE	ncit:C65572	ETICLOPRIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	PHENAMIPHOS	chembl:CHEMBL1313005	PHENAMIPHOS	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.4773424657790409	E163	chembl:CHEMBL443095	E163	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	SECAUBRYOLIDE	chembl:CHEMBL2332132	SECAUBRYOLIDE	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.421837528	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
CXCR2	hgnc:6027	CXCR2	DTC	9/2/20	NULL	4.375639269641208	NAVARIXIN	ncit:C156730	NAVARIXIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005864158	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.008033609	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.057700738	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001798824	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.037425282	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	GNF-PF-521	chembl:CHEMBL580071	CHEMBL:CHEMBL580071	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.015806042	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	CORTICOSTERONE	drugbank:DB04652	CORTICOSTERONE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.6819178082557726	S-METHYL-D-THIOCITRULLINE	chembl:CHEMBL1161525	S-METHYL-D-THIOCITRULLINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	Y-27632	drugbank:DB08756	Y-27632	FALSE	FALSE	FALSE
CA12	hgnc:1371	CA12	DTC	9/2/20	NULL	7.501095891	TRIFLUOROMETHANESULFONAMIDE	chembl:CHEMBL67511	TRIFLUOROMETHANESULFONAMIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	BISSALICYL FUMARATE	chembl:CHEMBL1374986	BISSALICYL FUMARATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	TCMDC-125575	chembl:CHEMBL587620	CHEMBL:CHEMBL587620	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	10-IODOEVODIAMINE	chembl:CHEMBL2171807	CHEMBL:CHEMBL2171807	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.3500511415712966	TEGASEROD MALEATE	rxcui:339270	TEGASEROD MALEATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.007737647	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PIPERILATE ETHOBROMIDE	chembl:CHEMBL1909073	PIPERILATE ETHOBROMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.029170928	ZM-39923 HCL	chembl:CHEMBL538798	CHEMBL:CHEMBL538798	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL199592	CHEMBL:CHEMBL199592	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.085796848	OXITRIPTAN	rxcui:94	5-HYDROXYTRYPTOPHAN	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.011968924	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.1835932560688619	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.03124062	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.014024485	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.3977853881492006	TERTATOLOL	rxcui:37840	TERTATOLOL	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.095122593	DIPYRONE SODIUM	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.031822831	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	NCI-17383	chembl:CHEMBL188641	CHEMBL:CHEMBL188641	FALSE	FALSE	FALSE
CASP9	hgnc:1511	CASP9	DTC	9/2/20	NULL	0.8204323630577265	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	SK&F-86002	iuphar.ligand:6040	SKF-86002	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004579424	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	HERNANDEZINE	chembl:CHEMBL504936	HERNANDEZINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
VCP	hgnc:12666	VCP	DTC	9/2/20	NULL	2.187819634820604	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.025244073	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.012971263	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	CEPHARANTHINE	ncit:C83611	CEPHARANTHINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	NSC-125296	chembl:CHEMBL311489	CHEMBL:CHEMBL311489	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	NSC-50690	chembl:CHEMBL1388703	CHEMBL:CHEMBL1388703	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	ONONETIN	chembl:CHEMBL241858	ONONETIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	ROSE BENGAL	rxcui:9471	ROSE BENGAL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	LOFEPRAMINE HYDROCHLORIDE	rxcui:6294	LOFEPRAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005402024	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.051885051	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	CGP-55845	iuphar.ligand:1088	CGP 55845	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	MAYTANSINOL	chembl:CHEMBL214154	MAYTANSINOL	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.011474579	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.009787078	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW621970X	chembl:CHEMBL179465	GW621970X	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1060761035064535	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1193356164447602	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007496384	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.007252441	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.1816874437221263	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1810609352954982	NSC-125296	chembl:CHEMBL311489	CHEMBL:CHEMBL311489	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	CID 1540545	chembl:CHEMBL259784	CHEMBL:CHEMBL259784	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	CID 1540545	chembl:CHEMBL259784	CHEMBL:CHEMBL259784	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.01141223	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001165077	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	ISOCONAZOLE	rxcui:27901	ISOCONAZOLE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.032982206	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	NCI-13239	chembl:CHEMBL187216	CHEMBL:CHEMBL187216	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	0.2917092846427472	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.007561589	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.036162308	CID 1245272	chembl:CHEMBL408850	CHEMBL:CHEMBL408850	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.06466462	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.1508841127462485	MEN-10376	iuphar.ligand:2116	MEN 10376	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.007395447	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.070197421	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	TCMDC-123904	chembl:CHEMBL586061	CHEMBL:CHEMBL586061	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	DNDI1417254	chembl:CHEMBL2094567	CHEMBL:CHEMBL2094567	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.020391329	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	PTEROSTILBENE	ncit:C153353	PTEROSTILBENE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.016605842	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.023004456	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.023284998	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004409815	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006193403	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.06697407	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004409815	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	5-NITRO-[1,10]PHENANTHROLINE	chembl:CHEMBL101815	CHEMBL:CHEMBL101815	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-738482	chembl:CHEMBL103098	CHEMBL:CHEMBL103098	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	TCMDC-125298	chembl:CHEMBL581152	CHEMBL:CHEMBL581152	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	RIMEXOLONE	rxcui:55681	RIMEXOLONE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.5707355569097228	GW775608X	chembl:CHEMBL476351	GW775608X	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	GNF-PF-2893	chembl:CHEMBL312032	CHEMBL:CHEMBL312032	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007529925	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	TYRPHOSTIN 1	iuphar.ligand:5917	AG 9	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006077277	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.006548724	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.3079628811477683	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.031784305	SB-206553	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.041085815	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	CORONOPILIN	chembl:CHEMBL248564	CORONOPILIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008916229	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	MESNA	rxcui:1546354	2-MERCAPTOETHANESULFONIC ACID	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	GNF-PF-1211	chembl:CHEMBL600968	CHEMBL:CHEMBL600968	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.023759127	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.105015342	TETRADECYLTHIOACETIC ACID	chembl:CHEMBL187734	TETRADECYLTHIOACETIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	SJ000001516	chembl:CHEMBL592316	CHEMBL:CHEMBL592316	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007378818	PIRIBEDIL	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.053038052	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	STEARIC ACID	rxcui:1310551	STEARIC ACID	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	DTC	9/2/20	NULL	2.692701089009974	L-655708	chembl:CHEMBL52030	CHEMBL:CHEMBL52030	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	TCMDC-125353	chembl:CHEMBL547924	CHEMBL:CHEMBL547924	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	EVANS BLUE	rxcui:4191	EVANS BLUE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123535	chembl:CHEMBL527730	CHEMBL:CHEMBL527730	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	CRYPTOTANSHINONE	drugbank:DB15579	CRYPTOTANSHINONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	GNF-PF-107	chembl:CHEMBL578675	CHEMBL:CHEMBL578675	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	FUROXAN	chembl:CHEMBL336467	FUROXAN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002258977	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:12577	iuphar.ligand:12577	MK-912	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.8751278539282416	QUINALPHOS	ncit:C163697	QUINALPHOS	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.182318303	SJ000124275	chembl:CHEMBL602150	CHEMBL:CHEMBL602150	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.066047385	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.097236428	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.089756703	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006397133	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.026372512	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:5601	iuphar.ligand:5601	MRS3558	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	0.364636606	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.030598876	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	TCMDC-124425	chembl:CHEMBL548681	CHEMBL:CHEMBL548681	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.018071819	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.005293112	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
BRDT	hgnc:1105	BRDT	DTC	9/2/20	NULL	0.2206204673768676	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.069638821	IUPHAR.LIGAND:1059	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008503267	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DEMECOLCINE	ncit:C419	DEMECOLCINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	0.1312691780892362	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.1341192113299987	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	1-NAPHTHYLISOTHIOCYANATE	chembl:CHEMBL1381098	1-NAPHTHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00988845	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	0.6250913242344582	ICI-164384	drugbank:DB03860	ICI-164384	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007937668	EMBELIN	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	MyCancerGenome	20-Jun-17	other/unknown	0.4773424657790409	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	1,5-DINITRO-NAPHTHALENE	chembl:CHEMBL167316	CHEMBL:CHEMBL167316	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.073437302	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	DTC	9/2/20	NULL	4.039051633514961	22(S)-HYDROXYCHOLESTEROL	chembl:CHEMBL1243244	CHEMBL:CHEMBL1243244	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	VALERENIC ACID	chembl:CHEMBL1545045	VALERENIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	PIMETHIXENE MALEATE	ncit:C97703	PIMETHIXENE MALEATE	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.1074020548002842	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.05814803	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.035418328	NEOSTIGMINE BROMIDE	rxcui:82055	NEOSTIGMINE BROMIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	FPL-64176	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1363835616511545	GNF-PF-107	chembl:CHEMBL578675	CHEMBL:CHEMBL578675	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	E1501	chembl:CHEMBL1233714	E1501	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.031032903	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002657809	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.005995395	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	INDAPAMIDE	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	BENZOQUINONE	iuphar.ligand:6307	BENZOQUINONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.007979889	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.011205222	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.2778183663264259	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	0.4730420832044549	MOCLOBEMIDE	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.095468493	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NR2F2	hgnc:7976	NR2F2	DTC	9/2/20	NULL	0.092118721	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.072927321	midazolam	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.037505479	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.01495945	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-1692	chembl:CHEMBL582055	CHEMBL:CHEMBL582055	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.048083948	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.048394167	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.049256727	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	THUNBERGINOL E	chembl:CHEMBL421486	THUNBERGINOL E	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.044878351	VINORELBINE BASE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	NSC-16736	chembl:CHEMBL1728978	CHEMBL:CHEMBL1728978	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.046343929	GNF-PF-1852	chembl:CHEMBL533293	CHEMBL:CHEMBL533293	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.01763778	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	2.333674277141977	KOBOPHENOL A	chembl:CHEMBL397488	KOBOPHENOL A	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.051885051	PALIPERIDONE PALMITATE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1640864726115453	CY-208243	chembl:CHEMBL313737	CHEMBL:CHEMBL313737	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.1442518440541058	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.027929612	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	CANDIDIN	chembl:CHEMBL454843	CANDIDIN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.2800409132570373	ABIETIC ACID	chembl:CHEMBL71893	ABIETIC ACID	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	MITONAFIDE	ncit:C66165	MITONAFIDE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.020778659	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.046221542	BIX-01294	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
MCOLN3	hgnc:13358	MCOLN3	DTC	9/2/20	NULL	0.8204323630577265	GNF-PF-3084	chembl:CHEMBL601135	CHEMBL:CHEMBL601135	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	NCI-13239	chembl:CHEMBL187216	CHEMBL:CHEMBL187216	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.062808219	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.073540156	2-CHLORO-ADENOSINETRIPHOSPHATE	iuphar.ligand:1716	2-CHLOROADENOSINE-5-TRIPHOSPHATE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	5,8,11,14-EICOSATETRAYNOIC ACID	iuphar.ligand:2669	EICOSATETRANOIC ACID	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.00519107	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.079197091	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002356506	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	EPIPODOPHYLLOTOXIN 4-(MORPHOLINE)CARBAMATE	chembl:CHEMBL1773343	CHEMBL:CHEMBL1773343	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	CancerCommons	25-Jul-13	inhibitor	2.080014029626545	LDK378	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.093763699	DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE	chembl:CHEMBL1569494	CHEMBL:CHEMBL1569494	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.1944728564284981	4-PHENYLAMINO-[1,2]NAPHTHOQUINONE	chembl:CHEMBL299853	CHEMBL:CHEMBL299853	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	TCMDC-124336	chembl:CHEMBL527271	CHEMBL:CHEMBL527271	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	PURVALANOLA	chembl:CHEMBL23327	PURVALANOLA	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	SJ000066425	chembl:CHEMBL600255	CHEMBL:CHEMBL600255	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	L-741742	iuphar.ligand:3302	L741742	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.027855529	ZAPRINAST	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.068324881	BUTANOIC ACID	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.022632617	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	GNF-PF-2357	chembl:CHEMBL578257	CHEMBL:CHEMBL578257	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	GNF-PF-4579	chembl:CHEMBL584626	CHEMBL:CHEMBL584626	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CGI	2/1/22	NULL	0.019261802	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	GYROPHORIC ACID	chembl:CHEMBL470648	GYROPHORIC ACID	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.1535312024435511	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	7,3'-DIMETHOXYFLAVONE	chembl:CHEMBL1326944	7,3'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW580509X	chembl:CHEMBL179311	GW580509X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	OXENDOLONE	ncit:C174717	OXENDOLONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003405608	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	chembl:CHEMBL571700	BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.002879341	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.057700738	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	CGI	2/1/22	NULL	0.079557078	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.024861587	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.046881849	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	1,7-O-DIACETYLMETHYLGEOPYXIN A	chembl:CHEMBL1889303	CHEMBL:CHEMBL1889303	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003099626	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
MGLL	hgnc:17038	MGLL	DTC	9/2/20	NULL	8.751278539282415	N-PHENYLMALEIMIDE	chembl:CHEMBL76012	CHEMBL:CHEMBL76012	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.031069628	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002949869	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.013025967	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	GW405833	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.022839352	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004149492	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	MANGOSTIN	rxcui:2619910	MANGOSTIN	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	DTC	9/2/20	NULL	0.2375912725597036	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	CHLOROPYRAMINE	rxcui:20861	CHLOROPYRAMINE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.039598545	ROTTLERIN	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.018819954	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
ERCC4	hgnc:3436	ERCC4	CGI	2/1/22	NULL	0.045265234	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	NSC-638080	chembl:CHEMBL136344	CHEMBL:CHEMBL136344	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.02287916	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	BUTAMBEN	rxcui:19861	BUTAMBEN	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	GNF-PF-4283	chembl:CHEMBL606166	CHEMBL:CHEMBL606166	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	OXITRIPTAN	rxcui:94	5-HYDROXYTRYPTOPHAN	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011810092	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	RO-410960	chembl:CHEMBL1256291	CHEMBL:CHEMBL1256291	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.9053046764774912	TERBUTALINE SULFATE	rxcui:10369	TERBUTALINE SULFATE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.045579576	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	METHYL 2-(4-FLUOROBENZAMIDO)BENZOATE	chembl:CHEMBL250428	CHEMBL:CHEMBL250428	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.044198376	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.033148782	SU-4312	chembl:CHEMBL328710	CHEMBL:CHEMBL328710	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.099446347	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	CGI	2/1/22	NULL	0.290901226	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	TCMDC-124685	chembl:CHEMBL587579	CHEMBL:CHEMBL587579	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	SJ000120449	chembl:CHEMBL609027	CHEMBL:CHEMBL609027	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	LASALOCID A SODIUM	chembl:CHEMBL1489769	LASALOCID A SODIUM	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	LOFEPRAMINE	rxcui:6465	LOFEPRAMINE	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.4526523382387456	METHYLCURCUMIN	chembl:CHEMBL494826	METHYLCURCUMIN	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	DTC	9/2/20	NULL	4.200613699	CARBOXYLATED GLUCOSAMINE	chembl:CHEMBL1161830	CARBOXYLATED GLUCOSAMINE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.070574827	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.3088686543276147	3,4,5,6-TETRACHLORO-[1,2]BENZOQUINONE	chembl:CHEMBL364729	CHEMBL:CHEMBL364729	FALSE	FALSE	FALSE
MAPKAPK2	hgnc:6887	MAPKAPK2	DTC	9/2/20	NULL	0.6035364509849942	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1396480617970598	DIMETHYL YELLOW	chembl:CHEMBL263116	DIMETHYL YELLOW	FALSE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	5.834185692854944	AMOPYROQUINE	ncit:C73000	AMOPYROQUINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	13-EPI-SCLOREOL	chembl:CHEMBL464176	CHEMBL:CHEMBL464176	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.010670122	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	PROTOCATECHUIC ACID	chembl:CHEMBL37537	PROTOCATECHUIC ACID	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.3117023117067671	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	2.019525817	KMI-1795	chembl:CHEMBL2047666	CHEMBL:CHEMBL2047666	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	TCMDC-124381	chembl:CHEMBL579919	CHEMBL:CHEMBL579919	FALSE	FALSE	FALSE
POLL	hgnc:9184	POLL	DTC	9/2/20	NULL	8.751278539282415	1-DEOXYRUBRALACTONE	chembl:CHEMBL260980	CHEMBL:CHEMBL260980	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	SJ000119988	chembl:CHEMBL589694	CHEMBL:CHEMBL589694	FALSE	FALSE	FALSE
LGALS3	hgnc:6563	LGALS3	DTC	9/2/20	NULL	8.751278539282415	LACTOSE, ANHYDROUS	chembl:CHEMBL417016	LACTOSE, ANHYDROUS	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.1312691780892362	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-221466	chembl:CHEMBL95502	CHEMBL:CHEMBL95502	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	0.4487835148349958	TOREMIFENE CITRATE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	1.500219178	TRIACETIN	rxcui:10756	TRIACETIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	1.312691780892362	BETULINIC ACID	ncit:C38126	BETULINIC ACID	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	BENZOTHIAZOL-2-YLAMINE	chembl:CHEMBL329785	CHEMBL:CHEMBL329785	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(-)-THYSANONE	chembl:CHEMBL596082	CHEMBL:CHEMBL596082	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV001241	chembl:CHEMBL601492	CHEMBL:CHEMBL601492	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.041214813	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.06970816	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	ETIDRONIC ACID	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	U-0126	ncit:C1825	U-0126	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2580229544751573	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2892984641085096	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2447910080918158	2-ENE-VALPROATE	chembl:CHEMBL117487	CHEMBL:CHEMBL117487	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	(+)-TAXIFOLIN	chembl:CHEMBL66	(+)-TAXIFOLIN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.078958904	ISOCONAZOLE	rxcui:27901	ISOCONAZOLE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.009629135	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	CATECHIN	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	ETRETINATE	rxcui:4182	ETRETINATE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.030176823	PROPYLPYRAZOLETRIOL	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TIBOLONE	rxcui:38260	TIBOLONE	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.061412481	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	ALX-5407	iuphar.ligand:4618	(R)-NFPS	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.02505137	T091317	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	(D)-SERINE	rxcui:1742747	SERINE, D-	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.012713722	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.7095631248066824	PARTHENOLIDE	rxcui:32941	PARTHENOLIDE	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.2011788169949981	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	FLOCTAFENINE	rxcui:4444	FLOCTAFENINE	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.2430910705356227	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.1643432589536604	1-DEOXYRUBRALACTONE	chembl:CHEMBL260980	CHEMBL:CHEMBL260980	FALSE	FALSE	FALSE
PHOSPHO1	hgnc:16815	PHOSPHO1	DTC	9/2/20	NULL	0.750109589	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.013631275	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	TCMDC-124381	chembl:CHEMBL579919	CHEMBL:CHEMBL579919	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CGI	2/1/22	NULL	0.4254093734373397	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	DTC	9/2/20	NULL	1.058622403945453	AZELASTINE	rxcui:18603	AZELASTINE	TRUE	FALSE	FALSE
RAC1	hgnc:9801	RAC1	DTC	9/2/20	NULL	5.834185692854944	ZU-3594419	chembl:CHEMBL562095	CHEMBL:CHEMBL562095	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004339477	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	CGI	2/1/22	NULL	0.8444216134395313	Tipifarnib	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	5-MEO-DMT	iuphar.ligand:145	5-MEO-DMT	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.036162308	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006397133	MORIN	drugbank:DB16770	MORIN	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.048935388	SB-203580	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.025244073	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.01715937	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.080781033	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.01495945	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	1.193356164447602	AMODIAQUINE HYDROCHLORIDE	rxcui:314495	AMODIAQUINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.3571950424196904	DIPHENYLUREA	chembl:CHEMBL354676	DIPHENYLUREA	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.052090944	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	NSC-155693	chembl:CHEMBL68096	CHEMBL:CHEMBL68096	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	CGI	2/1/22	NULL	0.5125748858722557	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.024674658	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	TCMDC-124522	chembl:CHEMBL526776	CHEMBL:CHEMBL526776	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	DTC	9/2/20	NULL	0.2001054544043235	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00317843	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.018385039	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1017590527823536	IMIDOCARB DIPROPIONATE	rxcui:1740238	IMIDOCARB DIPROPIONATE	TRUE	FALSE	FALSE
MLL	hgnc:7132	KMT2A	CGI	2/1/22	NULL	0.1491695205559502	Belinostat	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
PRKAG2	hgnc:9386	PRKAG2	DTC	9/2/20	NULL	1.346350544504987	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.03505185	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.057197899	MRS-1220	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	1.591141552596803	BMS-687453	chembl:CHEMBL1089501	CHEMBL:CHEMBL1089501	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006100578	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.023080295	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	CGI	2/1/22	NULL	0.4055851016423223	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.061197752	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	BENZO(K)FLUORANTHENE	chembl:CHEMBL1441574	BENZO(K)FLUORANTHENE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.049442252	FPL-64176	iuphar.ligand:2518	FPL64176	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	SB-242084	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
MGAM	hgnc:7043	MGAM	DTC	9/2/20	NULL	0.3671865121377238	BAICALEIN	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	LY-294002	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	ACRIDIN-1-YLAMINE	chembl:CHEMBL146525	CHEMBL:CHEMBL146525	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.057574201	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1019566431761058	DIBENZ[A,H]ANTHRACENE	chembl:CHEMBL1346946	DIBENZ[A,H]ANTHRACENE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	2-(STYRYL)-BENZIMIDAZOLE	chembl:CHEMBL473721	CHEMBL:CHEMBL473721	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.1666910197958555	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1320947704042629	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	DNDI1417076	chembl:CHEMBL1526167	CHEMBL:CHEMBL1526167	FALSE	FALSE	FALSE
CA7	hgnc:1381	CA7	ChEMBL	33	inhibitor	1.750255707856483	METHAZOLAMIDE	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	CID 1225609	chembl:CHEMBL444376	CHEMBL:CHEMBL444376	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	QUINOLINIC ACID	drugbank:DB01796	QUINOLINIC ACID	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.071148606	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.099446347	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013825085	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	LOMOFUNGIN	ncit:C170125	LOMOFUNGIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.011000979	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
P2RY4	hgnc:8542	P2RY4	DTC	9/2/20	NULL	35.00511415712966	5-OME-UTP	chembl:CHEMBL601439	CHEMBL:CHEMBL601439	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	TOLONIUM CHLORIDE	rxcui:10638	TOLONIUM CHLORIDE	FALSE	FALSE	FALSE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	1.050153425	METHAZOLAMIDE	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
ADCY9	hgnc:240	ADCY9	DTC	9/2/20	NULL	5.250767123569449	NSC-270718	chembl:CHEMBL401844	CHEMBL:CHEMBL401844	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	RO-106-9920	chembl:CHEMBL271023	CHEMBL:CHEMBL271023	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	AZASERINE	ncit:C289	AZASERINE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.063034419	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	HEXOCYCLIUM METHYLSULFATE	rxcui:235430	HEXOCYCLIUM METHYLSULFATE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	CIS-RESVERATROL	chembl:CHEMBL87333	CIS-RESVERATROL	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.02804897	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003968834	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002623285	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	CEFOTAXIME	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.1154014752432845	2-CHLORO-ADENOSINETRIPHOSPHATE	iuphar.ligand:1716	2-CHLOROADENOSINE-5-TRIPHOSPHATE	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.4257378748840094	FESOTERODINE FUMARATE	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
CASP8	hgnc:1509	CASP8	DTC	9/2/20	NULL	1.312691780892362	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.072324616	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003689409	NOCODAZOLE	ncit:C75228	NOCODAZOLE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004540615	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	NSC-133896	chembl:CHEMBL512908	CHEMBL:CHEMBL512908	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-743899	chembl:CHEMBL101804	CHEMBL:CHEMBL101804	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.010902756	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV000340	chembl:CHEMBL592044	CHEMBL:CHEMBL592044	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004716823	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	1.093909817410302	PASIREOTIDE DIASPARTATE	rxcui:1364104	PASIREOTIDE DIASPARTATE	TRUE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.3621218705909966	GUANABENZ	rxcui:5033	GUANABENZ	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012763168	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	GRINIMIBINE	chembl:CHEMBL1477760	GRINIMIBINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	CARBENDAZIM	ncit:C1154	CARBENDAZIM	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.3409589041278864	2-CHLOROADENOSINE	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.058602312	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	PYRITHIONE	rxcui:35100	PYRITHIONE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	UMBELLIFERONE	chembl:CHEMBL51628	UMBELLIFERONE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.004191225	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.014145386	MITOXANTRONE HYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.02505934	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.039778539	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.065145994	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	GNF-PF-5029	chembl:CHEMBL1198140	CHEMBL:CHEMBL1198140	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00575742	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	NSC-699479	chembl:CHEMBL1701915	CHEMBL:CHEMBL1701915	FALSE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	2.019525817	DORZOLAMIDE HYDROCHLORIDE	rxcui:236065	DORZOLAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.073437302	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.010417155	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.006173741	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.013716738	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	STICTIC ACID	chembl:CHEMBL173530	STICTIC ACID	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.00423449	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.1535312024435511	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.049256727	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GITOXIN	chembl:CHEMBL109317	GITOXIN	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.2083637747448194	CIS-RESVERATROL	chembl:CHEMBL87333	CIS-RESVERATROL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003279475	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.025929714	NICLOSAMIDE	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.043109746	ROSE BENGAL	rxcui:9471	ROSE BENGAL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	INDIRUBIN-3-MONOXIME	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	EPINASTINE HYDROCHLORIDE	rxcui:236961	EPINASTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.7955707762984014	SINENSETIN	chembl:CHEMBL226507	SINENSETIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TCMDC-123457	chembl:CHEMBL285157	CHEMBL:CHEMBL285157	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	NSC-62406	chembl:CHEMBL1332182	CHEMBL:CHEMBL1332182	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DEMETON-S-METHYL	chembl:CHEMBL1898805	DEMETON-S-METHYL	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.054187483	ZM-447439	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	ANGUSTIBALIN	chembl:CHEMBL486196	ANGUSTIBALIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	GNF-PF-107	chembl:CHEMBL578675	CHEMBL:CHEMBL578675	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	SULCONAZOLE NITRATE	rxcui:56798	SULCONAZOLE NITRATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	TETROQUINONE	chembl:CHEMBL1329029	TETROQUINONE	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.750109589	APTIGANEL HYDROCHLORIDE	ncit:C142929	APTIGANEL HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	CHELERYTHRINE CHLORIDE	chembl:CHEMBL258893	CHELERYTHRINE CHLORIDE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.034453853	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	KAINIC ACID	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	SJ000001516	chembl:CHEMBL592316	CHEMBL:CHEMBL592316	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2446009529613098	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2678962818147679	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.03261346	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	6-AZAURIDINE	ncit:C291	6-AZAURIDINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	IMETIT	iuphar.ligand:1250	IMETIT	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	TDR78109	chembl:CHEMBL1304363	CHEMBL:CHEMBL1304363	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-3237	chembl:CHEMBL602206	CHEMBL:CHEMBL602206	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.043902735	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
TTR	hgnc:12405	TTR	DTC	9/2/20	NULL	8.751278539282415	BENZYL CAFFEATE	chembl:CHEMBL133714	BENZYL CAFFEATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DIHYDROERGOCRISTINE	rxcui:3416	DIHYDROERGOCRISTINE	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.100589408	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NSC-128437	chembl:CHEMBL1370698	CHEMBL:CHEMBL1370698	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.024030971	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.071439008	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	TCMDC-123748	chembl:CHEMBL530609	CHEMBL:CHEMBL530609	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	DTC	9/2/20	NULL	0.1017590527823536	ISONIPECOTIC ACID	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.027135747	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	NSC-748118	chembl:CHEMBL2063681	CHEMBL:CHEMBL2063681	FALSE	FALSE	FALSE
LRRC59	hgnc:28817	LRRC59	DTC	9/2/20	NULL	15.00219178162699	MELAGATRAN	ncit:C66077	MELAGATRAN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.039628431	PYROGALLOL RED	chembl:CHEMBL210208	PYROGALLOL RED	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.033204682	Galantamine	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	10.50153424713889	Sofosbuvir	rxcui:1484911	SOFOSBUVIR	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.047734247	Tetracaine	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.021149706	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.008240375	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	MyCancerGenome	20-Jun-17	inhibitor	0.1037701012563132	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	MyCancerGenome	20-Jun-17	inhibitor	1.467605717767858	TOFACITINIB CITRATE	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	inhibitor	0.9907107780319716	LINSITINIB	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.1725334213659184	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.079236928	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	0.3443125982668492	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	0.089046362	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.06697407	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547592	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1008469998124734	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2273059360852575	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2275522047050683	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
PARP2	hgnc:272	PARP2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3977853881492008	AZD 2281	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1591141552596803	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.088396753	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.6721614540713904	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3241214273808303	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.082043236	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1582152052299645	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.049864835	ATAZANAVIR	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
AANAT	hgnc:19	AANAT	NCI	14-Sep-17	NULL	0.022949157	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.049864835	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.1442518440541057	RU 486	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
ALDH2	hgnc:404	ALDH2	NCI	14-Sep-17	NULL	0.028898003	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	NCI	14-Sep-17	NULL	0.1795134059339982	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
AKR1B1	hgnc:381	AKR1B1	NCI	14-Sep-17	NULL	8.078103267029922	GROWTH AGENTS	ncit:C530	RECOMBINANT GROWTH FACTOR	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.025563618	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.1187956362798518	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
APP	hgnc:620	APP	NCI	14-Sep-17	NULL	0.089756703	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
AQP1	hgnc:633	AQP1	NCI	14-Sep-17	NULL	0.1973972602845657	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.2134458180312784	CYCLOOXYGENASE INHIBITOR	ncit:C1323	CYCLOOXYGENASE INHIBITOR	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.6403374540938354	ZD1694	ncit:C1804	RALTITREXED	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.032837818	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.071148606	COMPLETE FREUND&APOS;S ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.018560506	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.2845944240417045	THYROGLOBULIN	rxcui:10565	THYROGLOBULIN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.2134458180312784	MEDICATION	ncit:C459	MEDICATION	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.1669560293662782	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.02587222	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.022099188	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.035098711	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
CA2	hgnc:1373	CA2	NCI	14-Sep-17	NULL	0.1187956362798518	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
C8ORF4	hgnc:1357	TCIM	NCI	14-Sep-17	NULL	8.751278539282415	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.042619863	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.010344301	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.018019105	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.059667808	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
CARD9	hgnc:16391	CARD9	NCI	14-Sep-17	NULL	7.001022831425933	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
CA3	hgnc:1374	CA3	NCI	14-Sep-17	NULL	1.875273972703374	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
CALR	hgnc:1455	CALR	NCI	14-Sep-17	NULL	1.093909817410302	ANTIANGIOGENIC	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	NCI	14-Sep-17	NULL	0.1750255707856483	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
CALR	hgnc:1455	CALR	NCI	14-Sep-17	NULL	0.4234489615781814	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	NCI	14-Sep-17	NULL	0.06714536	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CDKN2D	hgnc:1790	CDKN2D	NCI	14-Sep-17	NULL	1.312691780892362	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
CGA	hgnc:1885	CGA	NCI	14-Sep-17	NULL	0.3365876361262467	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
CGA	hgnc:1885	CGA	NCI	14-Sep-17	NULL	0.3860858179095184	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
CNR1	hgnc:2159	CNR1	NCI	14-Sep-17	NULL	0.6177373086552295	TETRAHYDROCANNABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.2885036881082116	VITAMIN C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	1.750255707856483	ANTIMALARIALS	ncit:C271	ANTIMALARIAL AGENT	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.2500365296937833	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	1.060761035064535	ISOPROPANOL	rxcui:797541	ISOPROPYL ALCOHOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	NCI	14-Sep-17	NULL	0.011049594	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.009788902	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	ChEMBL	33	agonist	1.050153425	DEXTROMETHORPHAN HYDROBROMIDE	rxcui:102490	DEXTROMETHORPHAN HYDROBROMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.018071819	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
CYP3A43	hgnc:17450	CYP3A43	NCI	14-Sep-17	NULL	7.501095891	POMEGRANATE JUICE	rxcui:1358975	POMEGRANATE JUICE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.01715937	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.005873341	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	1.750255707856483	SR 4233	ncit:C1464	TIRAPAZAMINE	FALSE	FALSE	FALSE
CYP3A7	hgnc:2640	CYP3A7	NCI	14-Sep-17	NULL	0.2273059360852576	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.042845917	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.8140724222588294	PHOTOSENSITIZER	ncit:C1420	PHOTOSENSITIZING AGENT	FALSE	FALSE	FALSE
DKK1	hgnc:2891	DKK1	NCI	14-Sep-17	NULL	0.5834185692854945	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
DHPS	hgnc:2869	DHPS	NCI	14-Sep-17	NULL	52.50767123569449	DEOXYSPERGUALIN	drugbank:DB12991	DEOXYSPERGUALIN	FALSE	FALSE	FALSE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	0.5114383561918295	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	ChEMBL	33	modulator	2.100306849	PENTAZOCINE HYDROCHLORIDE	rxcui:104973	PENTAZOCINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DTYMK	hgnc:3061	DTYMK	NCI	14-Sep-17	NULL	0.1103102336884338	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.057479662	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ELA2	hgnc:3309	ELANE	NCI	14-Sep-17	NULL	0.099258358	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
EIF2AK2	hgnc:9437	EIF2AK2	NCI	14-Sep-17	NULL	1.875273972703374	IFN ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.046425881	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.1187956362798518	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
FADD	hgnc:3573	FADD	NCI	14-Sep-17	NULL	8.751278539282415	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.283060222	ANTI CD3	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.093596562	EPO	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.07767407	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.1022544717345559	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.2083637747448194	FREUND&APOS;S ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.6731752722524935	COMPLETE FREUND&APOS;S ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.4321619031744403	TPN	drugsatfda.nda:008378	DRUGSATFDA.NDA:008378	FALSE	FALSE	FALSE
GHRH	hgnc:4265	GHRH	NCI	14-Sep-17	NULL	7.001022831425934	INTRALIPID	rxcui:1309980	SOYBEAN SEED OIL	TRUE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.1905904582057876	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
GRM1	hgnc:4593	GRM1	NCI	14-Sep-17	NULL	0.2524407270946851	ANTIDEPRESSANT	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.4565884455277783	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.022155136	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.089527146	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	AZIRIDINE	chembl:CHEMBL540990	AZIRIDINE	FALSE	FALSE	FALSE
IRS1	hgnc:6125	IRS1	NCI	14-Sep-17	NULL	0.8751278539282417	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
INHBE	hgnc:24029	INHBE	NCI	14-Sep-17	NULL	13.12691780892362	GNRH	chembl:CHEMBL1200511	GONADORELIN ACETATE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.1400204566285186	ROSIGLITAZONE MALEATE	rxcui:253198	ROSIGLITAZONE MALEATE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.036925226	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	NCI	14-Sep-17	NULL	0.2075402025126264	DFMO	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
KCNJ3	hgnc:6264	KCNJ3	NCI	14-Sep-17	NULL	5.250767124	THYROTROPIN	rxcui:10579	THYROTROPIN	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	NCI	14-Sep-17	NULL	0.2075402025126264	ALPHA-DIFLUOROMETHYLORNITHINE	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	ChEMBL	33	inhibitor	5.250767123569449	WARFARIN SODIUM	rxcui:114194	WARFARIN SODIUM	TRUE	FALSE	FALSE
JUND	hgnc:6206	JUND	NCI	14-Sep-17	NULL	1.082632396612257	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
IVL	hgnc:6187	IVL	NCI	14-Sep-17	NULL	0.8468979231563628	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
KCNJ3	hgnc:6264	KCNJ3	NCI	14-Sep-17	NULL	0.2706580991530644	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
KRT18	hgnc:6430	KRT18	NCI	14-Sep-17	NULL	0.6908904109959803	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.051478109	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.1992701	ANTIBIOTICS	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.2258394461750301	NAC	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.5707355569097228	MISTLETOE LECTIN	ncit:C2703	MISTLETOE EXTRACT	FALSE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.7501095890813498	MEDROXYPROGESTERONE	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
MIRN125B2	hgnc:31507	MIR125B2	NCI	14-Sep-17	NULL	13.12691780892362	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	0.8334550989792776	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	ChEMBL	33	agonist	13.12691780892362	COSYNTROPIN	rxcui:2890	COSYNTROPIN	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	NCI	14-Sep-17	NULL	3.889457128569962	MONOCLONAL ANTIBODY 1F5	ncit:C29198	MONOCLONAL ANTIBODY 1F5	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.2991890098899971	SERMS	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1296485709523321	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	NCI	14-Sep-17	NULL	0.364636606	FAS LIGAND	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.047561296	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	NCI	14-Sep-17	NULL	0.030202859	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PCNA	hgnc:8729	PCNA	NCI	14-Sep-17	NULL	0.600087671	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.1635752997996713	DEXTROAMPHETAMINE ADIPATE	chembl:CHEMBL1200782	DEXTROAMPHETAMINE ADIPATE	TRUE	FALSE	FALSE
PDHX	hgnc:21350	PDHX	NCI	14-Sep-17	NULL	17.50255707856483	AUTOANTIGEN	ncit:C20972	AUTOANTIGEN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1211715490054488	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.031069628	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.080781033	IL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.01495945	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.089756703	SERMS	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	NCI	14-Sep-17	NULL	0.052639269	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.043866058	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.3125456621172291	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.8334550989792776	NYSTATIN	rxcui:7597	NYSTATIN	TRUE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	0.057574201	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
RBP3	hgnc:9921	RBP3	NCI	14-Sep-17	NULL	0.9053046764774914	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.1442518440541057	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	NCI	14-Sep-17	NULL	0.090064616	ANTISENSE AGENT	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.2273059360852575	DIFFERENTIATION AGENTS	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.5125748858722557	TRAMETINIB DIMETHYL SULFOXIDE	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
S100A12	hgnc:10489	S100A12	NCI	14-Sep-17	NULL	0.1875273972703374	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
RLN2	hgnc:10027	RLN2	NCI	14-Sep-17	NULL	4.039051633514962	AMPHOTERICIN B	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
RNF112	hgnc:12968	RNF112	NCI	14-Sep-17	NULL	1.329308132549227	ETHANOL	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
RLN2	hgnc:10027	RLN2	NCI	14-Sep-17	NULL	6.563458904461812	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.09963505	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.1193356164447602	TRAMETINIB DIMETHYL SULFOXIDE	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.5385402178019948	NYSTATIN	rxcui:7597	NYSTATIN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.201952582	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.080781033	UCN-01	chembl:CHEMBL574737	UCN-01	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.048958202	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	NCI	14-Sep-17	NULL	0.2917092846427472	ANESTHETICS	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	NCI	14-Sep-17	NULL	0.2557191780959147	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	NCI	14-Sep-17	NULL	2.187819634820604	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.4251633298436801	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.5000730593875666	SODIUM BUTYRATE	ncit:C2337	SODIUM BUTYRATE	FALSE	FALSE	FALSE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	0.7001022831425934	ANTIESTROGENS	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
CA4	hgnc:1375	CA4	ChEMBL	33	inhibitor	0.8751278539282418	METHAZOLAMIDE	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
TEC	hgnc:11719	TEC	NCI	14-Sep-17	NULL	0.5385402178019949	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.041426171	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
TLR3	hgnc:11849	TLR3	NCI	14-Sep-17	NULL	0.5834185692854945	HYDROXYCHLOROQUINE	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	0.8078103267029924	HSP70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
WWOX	hgnc:12799	WWOX	NCI	14-Sep-17	NULL	2.333674277141977	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.4303907478335614	NORETHYNODREL	rxcui:7515	NORETHYNODREL	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	OncoKB	23-Jul-20	NULL	0.1995646288518794	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	OncoKB	23-Jul-20	NULL	2.407466349146467	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	OncoKB	23-Jul-20	NULL	0.8290684931951763	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	OncoKB	23-Jul-20	NULL	0.5303805175322677	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	OncoKB	23-Jul-20	NULL	0.384671584	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	OncoKB	23-Jul-20	NULL	0.1750255707856483	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	OncoKB	23-Jul-20	NULL	0.2275522047050683	Temsirolimus	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	OncoKB	23-Jul-20	NULL	1.831662950082366	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.08607815	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.045658845	ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.021697385	androstenedione	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	PharmGKB	4/5/24	NULL	0.036451004	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.068637479	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SH2D1A	hgnc:10820	SH2D1A	PharmGKB	4/5/24	NULL	13.12691780892362	emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
RAB27A	hgnc:9766	RAB27A	PharmGKB	4/5/24	NULL	13.12691780892362	emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	PharmGKB	4/5/24	NULL	0.1567393171214761	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	PharmGKB	4/5/24	NULL	0.4906052389860809	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
SLC28A3	hgnc:16484	SLC28A3	PharmGKB	4/5/24	NULL	0.5000730593875666	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.1457197166578015	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.290901226	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.021309932	dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.023813003	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
FCGR2A	hgnc:3616	FCGR2A	PharmGKB	4/5/24	NULL	0.7778914257139925	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.1392776425349987	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.2641895408085258	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
KLRD1	hgnc:6378	KLRD1	PharmGKB	4/5/24	NULL	0.6775183385250904	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.010685322	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
CYP2A7P1	hgnc:2612	CYP2A7P1	PharmGKB	4/5/24	NULL	1.093909817410302	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	PharmGKB	4/5/24	NULL	0.097236428	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
ARRB2	hgnc:712	ARRB2	PharmGKB	4/5/24	NULL	0.1508841127462485	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
HLA-DRA	hgnc:4947	HLA-DRA	PharmGKB	4/5/24	NULL	1.666910197958555	flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.1172046232939609	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.007792334	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
ARHGAP12	hgnc:16348	ARHGAP12	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	PharmGKB	4/5/24	NULL	0.015118823	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.009756163	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
IL18	hgnc:5986	IL18	PharmGKB	4/5/24	NULL	0.145450613	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	PharmGKB	4/5/24	NULL	0.062695727	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.2243917574174978	grapefruit juice	rxcui:1431224	GRAPEFRUIT JUICE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.02926849	doxycycline	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.013199515	naproxen	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.017260904	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.00380325	progesterone	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
AOX1	hgnc:553	AOX1	PharmGKB	4/5/24	NULL	0.7001022831425934	allopurinol	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
CARD16	hgnc:33701	CARD16	PharmGKB	4/5/24	NULL	1.381780822	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	inhibitor	0.3889457128569962	NALTREXONE HYDROCHLORIDE	rxcui:105069	NALTREXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	PharmGKB	4/5/24	NULL	0.1669560293662782	exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
SLC22A5	hgnc:10969	SLC22A5	PharmGKB	4/5/24	NULL	0.7143900848393808	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	PharmGKB	4/5/24	NULL	0.049841169	sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	2.500365296937833	tolcapone	rxcui:72937	TOLCAPONE	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.1472865953315413	propofol	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.1605739181519709	NALTREXONE HYDROCHLORIDE	rxcui:105069	NALTREXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	PharmGKB	4/5/24	NULL	0.087077398	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	PharmGKB	4/5/24	NULL	0.218327115	lenalidomide	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.078136416	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
CACNB4	hgnc:1404	CACNB4	PharmGKB	4/5/24	NULL	0.1205687054780585	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PTGES	hgnc:9599	PTGES	PharmGKB	4/5/24	NULL	0.2612321952024602	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CACNA1A	hgnc:1388	CACNA1A	PharmGKB	4/5/24	NULL	0.104492878	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	CODEINE SULFATE	rxcui:91104	CODEINE SULFATE	TRUE	FALSE	FALSE
KCNQ3	hgnc:6297	KCNQ3	PharmGKB	4/5/24	NULL	0.1119566550867686	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.081030357	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ATP2A1	hgnc:811	ATP2A1	PharmGKB	4/5/24	NULL	0.1567393171214761	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
BCHE	hgnc:983	BCHE	PharmGKB	4/5/24	NULL	2.148041096005684	succinylcholine	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	PharmGKB	4/5/24	NULL	0.8204323630577265	ethosuximide	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	PharmGKB	4/5/24	NULL	0.7369497717290455	erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.1110098757625676	phenoxybenzamine	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	PharmGKB	4/5/24	NULL	0.013788779	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1090879596309442	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	PharmGKB	4/5/24	NULL	0.8649519486500064	erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.1383601350084176	phenoxybenzamine	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.075896417	o-desmethyltramadol	chembl:CHEMBL4650315	DESMETRAMADOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.04427291	desvenlafaxine	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
XRCC3	hgnc:12830	XRCC3	PharmGKB	4/5/24	NULL	0.2206204673768676	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CLMN	hgnc:19972	CLMN	PharmGKB	4/5/24	NULL	1.29648571	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
FIP1L1	hgnc:19124	FIP1L1	PharmGKB	4/5/24	NULL	0.7001022831425933	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.05853698	carvedilol	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	PharmGKB	4/5/24	NULL	0.2917092846427472	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
CHRNA5	hgnc:1959	CHRNA5	PharmGKB	4/5/24	NULL	0.9723642821424908	efgartigimod alfa	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PCYT1A	hgnc:8754	PCYT1A	PharmGKB	4/5/24	NULL	2.187819634820604	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
NLGN1	hgnc:14291	NLGN1	PharmGKB	4/5/24	NULL	0.8824818695074705	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.053038052	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.2187819634820604	nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.011112735	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC22A3	hgnc:10967	SLC22A3	PharmGKB	4/5/24	NULL	0.546954909	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
CMPK1	hgnc:18170	CMPK1	PharmGKB	4/5/24	NULL	2.187819634820604	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.01235184	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.025003653	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.008136519	indomethacin	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	0.2778183663264258	alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
CHRNA6	hgnc:15963	CHRNA6	PharmGKB	4/5/24	NULL	0.9723642821424908	ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.1074020548002842	indomethacin	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.039553801	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
YAP1	hgnc:16262	YAP1	PharmGKB	4/5/24	NULL	1.779921058837101	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TWIST1	hgnc:12428	TWIST1	PharmGKB	4/5/24	NULL	0.8824818695074705	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.025304902	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
CYP2R1	hgnc:20580	CYP2R1	PharmGKB	4/5/24	NULL	0.921187215	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.076263865	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
IFIT1	hgnc:5407	IFIT1	PharmGKB	4/5/24	NULL	1.381780822	ribavirin	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.071341945	norepinephrine	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.080781033	vitamin c	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.6482428547616605	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.1881995384791917	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
CYP27B1	hgnc:2606	CYP27B1	PharmGKB	4/5/24	NULL	2.019525817	tenofovir disoproxil fumarate	rxcui:322248	TENOFOVIR DISOPROXIL FUMARATE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
EYA4	hgnc:3522	EYA4	PharmGKB	4/5/24	NULL	0.5645986154375753	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
TXNRD2	hgnc:18155	TXNRD2	PharmGKB	4/5/24	NULL	0.5707355569097228	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
RFPL4B	hgnc:33264	RFPL4B	PharmGKB	4/5/24	NULL	7.501095890813499	o-desmethyltramadol	chembl:CHEMBL4650315	DESMETRAMADOL	FALSE	FALSE	FALSE
RPP30	hgnc:17688	RPP30	PharmGKB	4/5/24	NULL	1.000146118775133	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
SULT1A3	hgnc:11455	SULT1A3	PharmGKB	4/5/24	NULL	3.750547945406749	o-desmethyltramadol	chembl:CHEMBL4650315	DESMETRAMADOL	FALSE	FALSE	FALSE
FCER2	hgnc:3612	FCER2	PharmGKB	4/5/24	NULL	1.615620653405984	budesonide	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.097236428	buprenorphine	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.044878351	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
CHUK	hgnc:1974	CHUK	PharmGKB	4/5/24	NULL	0.375054795	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	PharmGKB	4/5/24	NULL	0.4375639269641209	ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
TAOK3	hgnc:18133	TAOK3	PharmGKB	4/5/24	NULL	2.282942227638891	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.2403097081725148	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.1442518440541058	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
ABCC10	hgnc:52	ABCC10	PharmGKB	4/5/24	NULL	1.250182648468916	tenofovir	rxcui:117466	TENOFOVIR	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.1094923635591405	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
GP6	hgnc:14388	GP6	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCF4	hgnc:7662	NCF4	PharmGKB	4/5/24	NULL	1.312691780892362	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
NQO2	hgnc:7856	NQO2	PharmGKB	4/5/24	NULL	0.1286952726365061	idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.325124899	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.6819178082557726	vildagliptin	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.3684748858645228	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.3684748858645228	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.011352028	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.001924909	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.2075402025126264	mycophenolic acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
ABI1	hgnc:11320	ABI1	PharmGKB	4/5/24	NULL	0.1704794520639432	dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.096167896	ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	TALC	12-May-16	inhibitor	0.079197091	MOMELOTINIB	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.026572708	MOMELOTINIB	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.1244847587380144	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.086007651	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.062833272	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	0.9907107780319716	AMG-479	hemonc:241	GANITUMAB	FALSE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	HYDROCHLOROTHIAZIDE	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P48023	hgnc:11936	FASLG	TdgClinicalTrial	Jan-14	NULL	0.6908904109959803	APG101	ncit:C90562	ASUNERCEPT	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.5357925636295356	ANTIHEMOPHILIC FACTOR	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.2075402025126264	APLINDORE	ncit:C77563	APLINDORE	FALSE	FALSE	FALSE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.1121958787087489	AR-42	drugbank:DB12707	AR-42	FALSE	FALSE	TRUE
UNIPROT:Q02641	hgnc:1401	CACNB1	TdgClinicalTrial	Jan-14	NULL	0.375054795	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.5181678082469852	ARRY-334543	ncit:C62530	VARLITINIB	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.061197752	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.054243462	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O43497	hgnc:1394	CACNA1G	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	ARVERAPAMIL	drugbank:DB06669	ARVERAPAMIL	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.053038052	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.060423097	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	AV-412	drugbank:DB06021	AV-412	FALSE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.2273059360852575	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1000146118775133	CARIPRAZINE	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P24394	hgnc:6015	IL4R	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	CINTREDEKIN BESUDOTOX	ncit:C2599	CINTREDEKIN BESUDOTOX	FALSE	FALSE	FALSE
UNIPROT:Q16654	hgnc:8812	PDK4	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
UNIPROT:P33681	hgnc:1700	CD80	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	RG-2077	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	ESMIRTAZAPINE	ncit:C76963	ESMIRTAZAPINE	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.032899543	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	1.432027397337122	ETORICOXIB	rxcui:307296	ETORICOXIB	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.032899543	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.035430277	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	FIPAMEZOLE	ncit:C65684	FIPAMEZOLE	FALSE	FALSE	FALSE
UNIPROT:P19022	hgnc:1759	CDH2	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	ADH-1	ncit:C53399	ADH-1	FALSE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	0.2625383561784725	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.068369364	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.080781033	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1615620653405984	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	3.889457128569962	LFB-R603	chembl:CHEMBL2109348	LFB-R603	FALSE	FALSE	FALSE
UNIPROT:P17752	hgnc:12008	TPH1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	LX1031	drugbank:DB05199	LX1031	FALSE	FALSE	FALSE
UNIPROT:P09467	hgnc:3606	FBP1	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	MB07803	chembl:CHEMBL4297400	MB-07803	FALSE	FALSE	FALSE
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.1037701012563132	LY3009104	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.84012274	MBX-2044	chembl:CHEMBL3545020	MBX-2044	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
UNIPROT:Q8TDV5	hgnc:19060	GPR119	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	MBX-2982	drugbank:DB12345	MBX-2982	FALSE	FALSE	FALSE
UNIPROT:O43614	hgnc:4849	HCRTR2	TdgClinicalTrial	Jan-14	NULL	3.580068493342807	SUVOREXANT	rxcui:1547099	SUVOREXANT	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.4000584475100533	PRAMIPEXOLE	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
UNIPROT:P20839	hgnc:6052	IMPDH1	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.062262061	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1000146118775133	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	inhibitor	0.057700738	CARVEDILOL PHOSPHATE	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:P16471	hgnc:9446	PRLR	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	SOMATROPIN RECOMBINANT	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1137761023525341	HYDROMORPHONE	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14784	hgnc:6009	IL2RB	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	INTERLEUKIN-2	ncit:C587	RECOMBINANT INTERLEUKIN-2	FALSE	FALSE	FALSE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.086007651	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.088396753	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P50579	hgnc:16672	METAP2	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	PPI-2458	drugbank:DB05864	PPI-2458	FALSE	FALSE	FALSE
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.3409589041278863	PIRFENIDONE	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TdgClinicalTrial	Jan-14	NULL	1.050153425	OPC-14523	drugbank:DB05422	OPC-14523	FALSE	FALSE	FALSE
UNIPROT:P54284	hgnc:1403	CACNB3	TdgClinicalTrial	Jan-14	NULL	0.252440727	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P05107	hgnc:6155	ITGB2	TdgClinicalTrial	Jan-14	NULL	0.729273212	SAR 1118	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	FIRATEGRAST	ncit:C76692	FIRATEGRAST	FALSE	FALSE	FALSE
UNIPROT:P24530	hgnc:3180	EDNRB	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	SPI-1620	ncit:C74027	SOVATELTIDE	FALSE	FALSE	FALSE
UNIPROT:P00790	hgnc:8885	PGA3	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	SUCRALFATE	rxcui:10156	SUCRALFATE	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1232574442152452	TABERMINOGENE VADENOVEC	drugbank:DB05011	TABERMINOGENE VADENOVEC	FALSE	FALSE	FALSE
UNIPROT:Q03431	hgnc:9608	PTH1R	TdgClinicalTrial	Jan-14	NULL	2.812910959055062	TERIPARATIDE	rxcui:32915	TERIPARATIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.024416494	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
UNIPROT:P61812	hgnc:11768	TGFB2	TdgClinicalTrial	Jan-14	NULL	7.501095891	TRABEDERSEN	ncit:C80066	TRABEDERSEN	FALSE	FALSE	FALSE
UNIPROT:Q15761	hgnc:7958	NPY5R	TdgClinicalTrial	Jan-14	NULL	15.00219178	VELNEPERIT	ncit:C152850	VELNEPERIT	FALSE	FALSE	FALSE
UNIPROT:O15496	hgnc:9029	PLA2G10	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	VARESPLADIB	ncit:C152832	VARESPLADIB	FALSE	FALSE	FALSE
UNIPROT:P29459	hgnc:5969	IL12A	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	VIRULIZIN	ncit:C26677	VIRULIZIN	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2465148884304905	APRACLONIDINE HYDROCHLORIDE	rxcui:91350	APRACLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q3KQW3	hgnc:9253	PPIA	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	VOCLOSPORIN	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
UNIPROT:O43451	hgnc:7043	MGAM	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	VOGLIBOSE	ncit:C95221	VOGLIBOSE	TRUE	FALSE	FALSE
UNIPROT:P68366	hgnc:12407	TUBA4A	TdgClinicalTrial	Jan-14	NULL	0.039527003	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.6789785073581185	VORELOXIN	ncit:C95148	VOSAROXIN	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.2234368988752957	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	agonist	0.021036727	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.082429625	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.05814803	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	CHLOPHEDIANOL	rxcui:21254	CHLOPHEDIANOL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.08334551	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.1603287671318916	CLOCORTOLONE	rxcui:21249	CLOCORTOLONE	TRUE	FALSE	FALSE
UNIPROT:P08709	hgnc:3544	F7	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	COAGULATION FACTOR VIIA	rxcui:2386863	COAGULATION FACTOR VIIA (RECOMBINANT)-JNCW	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.1411496538593938	CYPROHEPTADINE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.033412454	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.084146909	CYPROHEPTADINE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1262203635473425	ERGOLOID MESYLATE	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.088248187	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1630673019742065	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.077827576	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	0.7292732116068681	GOSERELIN	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.097236428	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.100976291	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	2.461297089173179	INTERFERON ALFA-N1	rxcui:202912	INTERFERON ALFA-N1	FALSE	TRUE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.070010228	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
DRD5	hgnc:3026	DRD5	ChEMBL	33	agonist	0.2019525816757481	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.075010959	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.069240885	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1077080435603989	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.045226246	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.077789143	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.081830137	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:Q8TDS4	hgnc:24827	HCAR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	MEPENZOLATE	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.041182487	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.097236428	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.1067229090156392	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.096167896	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.090452491	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1406455479527531	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TdgClinicalTrial	Jan-14	NULL	0.9546849315580819	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.2035181055647073	APRACLONIDINE HYDROCHLORIDE	rxcui:91350	APRACLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9GZZ6	hgnc:13800	CHRNA10	TdgClinicalTrial	Jan-14	NULL	0.4565884455277782	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TdgClinicalTrial	Jan-14	NULL	0.9546849315580819	PAMIDRONATE	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.187193124	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	TESTOLACTONE	rxcui:10378	TESTOLACTONE	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.056601873	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.3535870116881784	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.3547815624033412	CAFFEINE, CITRATED	rxcui:20033	CAFFEINE CITRATE	TRUE	FALSE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	2.800409132570373	TIROFIBAN	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.1790034246671403	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.067883221	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.070197421	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.073540156	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.079197091	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	inhibitor	0.2763561643983921	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.2375912725597036	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.07182992	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P00390	hgnc:4623	GSR	TEND	1-Aug-11	NULL	0.6509215442441467	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.1411496538593938	CYPROHEPTADINE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.084146909	CYPROHEPTADINE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.729273212	CAFFEINE, CITRATED	rxcui:20033	CAFFEINE CITRATE	TRUE	FALSE	FALSE
UNIPROT:P15260	hgnc:5439	IFNGR1	TEND	1-Aug-11	NULL	39.38075342677087	INTERFERON GAMMA-1B	rxcui:5882	INTERFERON GAMMA-1B	TRUE	TRUE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TEND	1-Aug-11	NULL	0.4102161815288632	DILTIAZEM	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.406619897	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
UNIPROT:P34995	hgnc:9593	PTGER1	TEND	1-Aug-11	NULL	0.9376369863516875	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.075496292	DULOXETINE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.1535312024435511	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	OXAPROZIN POTASSIUM	rxcui:660767	OXAPROZIN POTASSIUM	TRUE	FALSE	FALSE
UNIPROT:P07098	hgnc:6622	LIPF	TEND	1-Aug-11	NULL	2.692701089009974	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.048172175	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	1.432027397337122	ETORICOXIB	rxcui:307296	ETORICOXIB	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1583941817064691	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.076263865	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.038765353	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.060984519	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	INDOMETHACIN SODIUM	rxcui:1294612	INDOMETHACIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P47712	hgnc:9035	PLA2G4A	TEND	1-Aug-11	NULL	0.8751278539282418	FLUOCINOLONE ACETONIDE	rxcui:4461	FLUOCINOLONE ACETONIDE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.079197091	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.2206204673768676	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.059532507	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.4565884455277783	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.046881849	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.1154014752432846	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.09814518	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TEND	1-Aug-11	NULL	1.381780822	LEPIRUDIN	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	0.112919723	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.2678962818147678	LOFEXIDINE	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.090452491	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.065092154	MESALAZINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
UNIPROT:P20839	hgnc:6052	IMPDH1	TEND	1-Aug-11	NULL	0.4773424657790409	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.05814803	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.011143394	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.018672714	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
SCNN1A	hgnc:10599	SCNN1A	ChEMBL	33	blocker	2.917092846427472	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.059532507	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.020320306	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.051177067	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.020025809	OLANZAPINE	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.042619863	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.2408608772279564	PROPOXYPHENE	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1346350544504987	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TEND	1-Aug-11	NULL	2.051080907644316	TADALAFIL	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TEND	1-Aug-11	NULL	0.095122593	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 2	hgnc:6871	MAPK1	TTD	2020.06.01	NULL	0.060008767	BVD-523	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
RRM2	hgnc:10452	RRM2	ChEMBL	33	inhibitor	0.577007376	GALLIUM NITRATE	rxcui:25544	GALLIUM NITRATE	TRUE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.347732922	Thioureidobutyronitrile	ncit:C102881	THIOUREIDOBUTYRONITRILE	FALSE	FALSE	FALSE
PROHEPARIN-BINDING EGF-LIKE GROWTH FACTOR	hgnc:3059	HBEGF	TTD	2020.06.01	NULL	1.693795846312725	U3-1565	ncit:C95736	ANTI-HBEGF MONOCLONAL ANTIBODY U3-1565	FALSE	FALSE	FALSE
SOLUBLE GUANYLATE CYCLASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	1.050153425	IW-1973	ncit:C174906	PRALICIGUAT	FALSE	FALSE	FALSE
MITOCHONDRIAL ALDEHYDE DEHYDROGENASE	hgnc:404	ALDH2	TTD	2020.06.01	NULL	1.141471113819445	FP-045	ncit:C200589	ALDH2 ACTIVATOR FP-045	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.1162960603226899	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE ATR	hgnc:882	ATR	TTD	2020.06.01	NULL	1.166837138570988	BAY1895344	ncit:C146807	ELIMUSERTIB	FALSE	FALSE	TRUE
EXTRACELLULAR SIGNAL-REGULATED KINASE 1	hgnc:6877	MAPK3	TTD	2020.06.01	NULL	0.9907107780319716	ASN007	chembl:CHEMBL4650280	ASN007	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	1.944728564284981	BLU-667	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	4.039051633514961	FT-1101	drugbank:DB17553	FT-1101	FALSE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	agonist	0.7501095890813501	DECAMETHONIUM BROMIDE	ncit:C65365	DECAMETHONIUM BROMIDE	TRUE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	4.039051633514961	CC-90010	ncit:C151951	TROTABRESIB	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.1704794520639431	CYC065	ncit:C123902	FADRACICLIB	FALSE	FALSE	TRUE
TGF-BETA RECEPTOR TYPE I	hgnc:11772	TGFBR1	TTD	2020.06.01	NULL	7.501095891	LY3200882	ncit:C132013	TGFBETA INHIBITOR LY3200882	FALSE	FALSE	FALSE
SERINE/THREONINE PP2A	hgnc:9308	PTPA	TTD	2020.06.01	NULL	10.50153425	LB-100	drugbank:DB15412	LB-100	FALSE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	agonist	0.5527123287967842	DECAMETHONIUM BROMIDE	ncit:C65365	DECAMETHONIUM BROMIDE	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR 8	hgnc:15632	TLR8	TTD	2020.06.01	NULL	6.563458904461812	MEDI9197	ncit:C124653	TELRATOLIMOD	FALSE	FALSE	FALSE
FASCIN	hgnc:11148	FSCN1	TTD	2020.06.01	NULL	52.50767123569449	NP-G2-044	drugbank:DB14995	NP-G2-044	FALSE	FALSE	FALSE
PDE8B	hgnc:8794	PDE8B	ChEMBL	33	inhibitor	0.5000730593875666	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	1.050153425	SY-1365	ncit:C139552	MEVOCICLIB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.2218633995874415	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
EPHRIN TYPE-B RECEPTOR 2	hgnc:3393	EPHB2	TTD	2020.06.01	NULL	0.069089041	BVD-523	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.078682824	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
MITOCHONDRIAL PROTEIN UNSPECIFIC	hgnc:9282	PPP1CB	TTD	2020.06.01	NULL	2.019525816757481	EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN CD47	hgnc:1682	CD47	TTD	2020.06.01	NULL	6.563458904461812	TTI-621	ncit:C125718	ONTORPACEPT	FALSE	FALSE	FALSE
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	0.8468979231563628	BMS-986165	rxcui:2612087	DEUCRAVACITINIB	TRUE	FALSE	FALSE
LUTEINIZING HORMONE RECEPTOR	hgnc:6585	LHCGR	TTD	2020.06.01	NULL	1.640864726115453	TAK-385	rxcui:2472778	RELUGOLIX	TRUE	FALSE	FALSE
ANGIOPOIETIN 1 RECEPTOR	hgnc:11724	TEK	TTD	2020.06.01	NULL	1.640864726115453	AKB-9778	ncit:C152161	RAZUPROTAFIB	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.092988792	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
ANGIOPOIETIN-RELATED PROTEIN 3	hgnc:491	ANGPTL3	TTD	2020.06.01	NULL	26.25383561784724	Evinacumab	rxcui:2478335	EVINACUMAB	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR 8	hgnc:15632	TLR8	TTD	2020.06.01	NULL	13.12691780892362	VTX-2337	ncit:C80521	MOTOLIMOD	FALSE	FALSE	TRUE
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	2.763561643983921	CF102	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.059085902	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	0.2749092734853114	BMS-908662	drugbank:DB12854	BMS-908662	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.1888765152363111	DCC-2036	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.017295017	Levodopa	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	1.521961485092594	ASP3026	ncit:C116727	ALK INHIBITOR ASP3026	FALSE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.4861821410712454	Tivozanib	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	0.5147810905460245	GSK2849330	ncit:C111997	ANTI-HER3 MONOCLONAL ANTIBODY GSK2849330	FALSE	FALSE	TRUE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.1130007271930297	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
INTERLEUKIN 6 RECEPTOR	hgnc:6019	IL6R	TTD	2020.06.01	NULL	4.039051633514961	Sirukumab	ncit:C152371	SIRUKUMAB	FALSE	FALSE	FALSE
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	1.250182648468916	Factor viia	rxcui:2386863	COAGULATION FACTOR VIIA (RECOMBINANT)-JNCW	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.057574201	Flumazenil	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-5	hgnc:4079	GABRA5	TTD	2020.06.01	NULL	0.099446347	Flumazenil	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.087629625	Afimoxifene	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.040112812	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
MELANOCYTES LINEAGE-SPECIFIC ANTIGEN GP100	hgnc:10880	PMEL	TTD	2020.06.01	NULL	6.563458904461812	IMCgp100	rxcui:2590743	TEBENTAFUSP	TRUE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.591141552596803	AEZS-108	ncit:C74025	ZOPTARELIN DOXORUBICIN	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	1.875273972703375	bimatoprost (free acid form)	iuphar.ligand:1959	BIMATOPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	0.375054795	Berberine	rxcui:1437	BERBERINE	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.1470803115845784	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	3.281729452230906	Vardenafil	rxcui:306674	VARDENAFIL	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.084146909	Ocaperidone	ncit:C76441	OCAPERIDONE	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.252440727	MIN-101	chembl:CHEMBL4298043	ROLUPERIDONE HYDROCHLORIDE	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	2.386712328895204	NCX-4016	iuphar.ligand:9018	NCX-4016	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.1187956362798518	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
MONOCYTE CHEMOTACTIC AND ACTIVATING FACTOR	hgnc:10618	CCL2	TTD	2020.06.01	NULL	1.093909817410302	MCP-1	ncit:C1393	RECOMBINANT MONOCYTE CHEMOATTRACTANT PROTEIN-1	FALSE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA4.2	hgnc:18866	KCNT2	TTD	2020.06.01	NULL	1.166837138570988	phorbol 12-myristate 13-acetate	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	5.250767123569449	MOTILIN	iuphar.ligand:1457	MOTILIN	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.2983390411119005	Tianeptine	rxcui:38252	TIANEPTINE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.015434354	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.1682938180631233	Blonanserin	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.6241137025199848	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.069180068	Blonanserin	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	2.625383561784724	Isatoribine	ncit:C90811	ISATORIBINE	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.9723642821424906	Andolast	ncit:C74213	ANDOLAST	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.03394161	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN 1	hgnc:51	ABCC1	TTD	2020.06.01	NULL	0.053798843	Benzbromarone	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV4.3	hgnc:6239	KCND3	TTD	2020.06.01	NULL	3.281729452230906	Sodium bicarbonate	rxcui:36676	SODIUM BICARBONATE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	GSK233705	chembl:CHEMBL2308782	DAROTROPIUM BROMIDE	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
SECRETIN RECEPTOR	hgnc:10607	SCT	TTD	2020.06.01	NULL	26.25383561784724	Secretin	rxcui:9627	SECRETIN	TRUE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.1228249619548409	NVP-LAQ824	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	1.029562181092049	Elisidepsin	ncit:C66949	ELISIDEPSIN	FALSE	FALSE	FALSE
FERROCHELATASE	hgnc:3647	FECH	TTD	2020.06.01	NULL	10.50153424713889	Methyl aminolevulinate	ncit:C76305	METHYL AMINOLEVULINATE	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.4375639269641208	GSK461364	ncit:C70948	POLO-LIKE KINASE 1 INHIBITOR GSK461364	FALSE	FALSE	TRUE
INTERLEUKIN 4 RECEPTOR ALPHA	hgnc:6015	IL4R	TTD	2020.06.01	NULL	17.50255707856483	PRX-321	chembl:CHEMBL4298027	PRX-321	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.4070362111294147	ZALEPLON	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	3.043922970185188	Terlipressin	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	1.419126249613364	Aminoguanidine	rxcui:1311670	PIMAGEDINE	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.3337351985319565	PHA-739358	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	0.050879526	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NEURONAL PENTRAXIN-2	hgnc:7953	NPTX2	TTD	2020.06.01	NULL	52.50767123569449	PRM-151	ncit:C113177	ZINPENTRAXIN ALFA	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.1544343271638073	M100907	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.021449212	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.041182487	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
INTERLEUKIN-29	hgnc:18363	IFNL1	TTD	2020.06.01	NULL	17.50255707856483	Peginterferon lambda-1a	ncit:C166435	PEGINTERFERON LAMBDA-1A	FALSE	FALSE	FALSE
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	0.3947945205691315	SCH-442416	iuphar.ligand:3283	SCH442416	FALSE	FALSE	FALSE
PHOSPHOLIPASE D2	hgnc:9068	PLD2	TTD	2020.06.01	NULL	8.751278539282415	VU0364739	iuphar.ligand:5287	VU0364739	FALSE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	modulator	0.192335792	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
HLA-DR ANTIGENS-ASSOCIATED INVARIANT	hgnc:1697	CD74	TTD	2020.06.01	NULL	52.50767123569449	Milatuzumab	ncit:C66983	MILATUZUMAB	FALSE	TRUE	TRUE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.2201579506737715	CHR-3996	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
REACTIVE OXYGEN SPECIES	hgnc:10261	ROS1	TTD	2020.06.01	NULL	1.093909817410302	Procysteine	chembl:CHEMBL442218	PROCYSTEINE	FALSE	FALSE	FALSE
POLD3	hgnc:20932	POLD3	ChEMBL	33	inhibitor	0.094099769	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	0.2047082699247349	RGB-286638	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.053854022	DS-7423	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
SOLUBLE GUANYLYL CYCLASE	hgnc:4689	GUCY2D	TTD	2020.06.01	NULL	3.500511415712967	Riociguat	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
PRIM2	hgnc:9370	PRIM2	ChEMBL	33	inhibitor	0.094099769	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
UBIQUITIN-LIKE PROTEIN NEDD8	hgnc:7732	NEDD8	TTD	2020.06.01	NULL	10.50153425	MLN4924	ncit:C77906	PEVONEDISTAT	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.2302968036653267	NERATINIB MALEATE	rxcui:1940642	NERATINIB MALEATE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.004616194	Flufenamic Acid	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
POLE	hgnc:9177	POLE	ChEMBL	33	inhibitor	0.056459862	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M4	hgnc:1953	CHRM4	TTD	2020.06.01	NULL	0.1944728564284981	ACECLIDINE	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.729273212	BAY 1067197	iuphar.ligand:11222	NELADENOSON	FALSE	FALSE	FALSE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.6731752722524935	AMG 386	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.2019525816757481	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.4167275494896388	LIRIMILAST	ncit:C82304	LIRIMILAST	FALSE	FALSE	FALSE
PARATHYROID HORMONE 1 RECEPTOR	hgnc:9608	PTH1R	TTD	2020.06.01	NULL	3.750547945	Abaloparatide	rxcui:1921069	ABALOPARATIDE	TRUE	FALSE	FALSE
TNF ALPHA CONVERTING ENZYME	hgnc:195	ADAM17	TTD	2020.06.01	NULL	4.375639269641208	Aderbasib	ncit:C76115	ADERBASIB	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.9723642821424906	RTI-336	chembl:CHEMBL1186581	RTI-336	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	3.281729452230906	PF-489791	iuphar.ligand:8377	PF-00489791	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.9546849315580818	Albiglutide	rxcui:1534763	ALBIGLUTIDE	TRUE	FALSE	FALSE
CAMBRIDGE PATHOLOGY 1 ANTIGEN	hgnc:1804	CD52	TTD	2020.06.01	NULL	70.01022831425932	Alemtuzumab	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
PHOSPHODIESTERASE 3A	hgnc:8778	PDE3A	TTD	2020.06.01	NULL	0.4773424657790409	Aminophylline	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.3580068493342807	Apremilast	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.1233298208706858	Budesonide	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	0.9131768910555564	Chenodiol	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.4773424657790409	Fenoprofen	rxcui:4331	FENOPROFEN	TRUE	FALSE	FALSE
PROTEIN KINASE C GAMMA	hgnc:9402	PRKCG	TTD	2020.06.01	NULL	0.1268301237577161	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	0.6177373086552295	Marinol	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
CATECHOL-O-METHYL-TRANSFERASE	hgnc:2228	COMT	TTD	2020.06.01	NULL	2.500365296937833	Tolcapone	rxcui:72937	TOLCAPONE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.9546849315580819	Timolol	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.1861974157294131	ANAVEX 2-73	ncit:C171846	BLARCAMESINE	FALSE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DL1	hgnc:6329	KIR2DL1	TTD	2020.06.01	NULL	10.50153424713889	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DL3	hgnc:6331	KIR2DL3	TTD	2020.06.01	NULL	7.876150685354174	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	0.7095631248066824	LANEPITANT	ncit:C79124	LANEPITANT	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	LE-SN38	ncit:C95717	LIPOSOMAL SN-38	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	4.039051633514961	JNJ-54861911	ncit:C166553	ATABECESTAT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.6326225450083675	IUPHAR.LIGAND:108	iuphar.ligand:108	BMS 181,101	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:122	iuphar.ligand:122	DIPROPYL-5-CT	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:8422	iuphar.ligand:8422	5-BODMT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:165	iuphar.ligand:165	MK-212	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.5527123287967841	IUPHAR.LIGAND:282	iuphar.ligand:282	DIHYDROERGOCRYPTINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:188	iuphar.ligand:188	RS-127445	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:231	iuphar.ligand:231	LY334362	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:234	iuphar.ligand:234	BIMU 8	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:185	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
NCBIGENE:778	hgnc:1393	CACNA1F	GuideToPharmacology	2024.1	NULL	1.250182648468916	IUPHAR.LIGAND:4545	iuphar.ligand:4545	GLYCOCHENODEOXYCHOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1784	ncbigene:1784	DNCM	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:9916	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:4450	iuphar.ligand:4450	(+)-ADRENALINE	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.091796628	IUPHAR.LIGAND:7302	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:482	iuphar.ligand:482	HEAT (BE2254)	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.1988926940746003	IUPHAR.LIGAND:483	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:491	iuphar.ligand:491	A-123189	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1259176768242074	IUPHAR.LIGAND:525	iuphar.ligand:525	BRL 44408	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.1259176768242074	IUPHAR.LIGAND:7117	rxcui:14845	APRACLONIDINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.011804782	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1259176768242074	IUPHAR.LIGAND:524	iuphar.ligand:524	ARC-239	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.044198376	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:525	iuphar.ligand:525	BRL 44408	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:517	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.1084869240406911	IUPHAR.LIGAND:7268	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.03729238	IUPHAR.LIGAND:505	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:525	iuphar.ligand:525	BRL 44408	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:12575	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:517	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:1560	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9669	iuphar.ligand:9669	BTB07018	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2856	drugbank:DB02901	STANOLONE	FALSE	FALSE	FALSE
NCBIGENE:1560	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:9091	iuphar.ligand:9091	COMPOUND 1A [PMID: 25692029]	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.022353202	IUPHAR.LIGAND:413	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:3286	iuphar.ligand:3286	PSB1115	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:11153	ncit:C148039	IMARADENANT	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:386	iuphar.ligand:386	DPCPX	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:374	iuphar.ligand:374	CCPA	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:9942	iuphar.ligand:9942	AZD0156	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:465	iuphar.ligand:465	MRE 3010F20	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:6901	rxcui:1091642	AZILSARTAN MEDOXOMIL	TRUE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:7332	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8855	iuphar.ligand:8855	SM-122	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.068369364	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:2792	hgnc:4411	GNGT1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8855	iuphar.ligand:8855	SM-122	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:6163	iuphar.ligand:6163	NEUROMEDIN B (1-30) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11262	iuphar.ligand:11262	AM-37	FALSE	FALSE	FALSE
NCBIGENE:2844	hgnc:4476	GPR21	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:8319	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
NCBIGENE:2845	hgnc:4477	GPR22	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:8319	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:5387	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:5387	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.4234489615781814	IUPHAR.LIGAND:5387	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:11413	iuphar.ligand:11413	NEMTABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1789	hgnc:2979	DNMT3B	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7797	ncit:C116891	GALUNISERTIB	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:5681	iuphar.ligand:5681	GDC-0879	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:10073	iuphar.ligand:10073	COMPOUND 6 [PMID: 30125504]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:10564	iuphar.ligand:10564	ARV-771	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:7033	iuphar.ligand:7033	MOLIBRESIB	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:12143	iuphar.ligand:12143	WNY0824	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3791	iuphar.ligand:3791	[125I]HPP-DESARG10HOE140	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:672	ncit:C1606	LABRADIMIL	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:3831	iuphar.ligand:3831	[3H]NPC17731	FALSE	FALSE	FALSE
NCBIGENE:2471	hgnc:3881	FRA20A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6601	rxcui:18751	BAMBUTEROL	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:658	iuphar.ligand:658	NPC 18565	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:10227	iuphar.ligand:10227	ORYZATENSIN	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:6797	rxcui:194881	BRINZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:4224	iuphar.ligand:4224	INS(3,4,5,6)P4	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:6920	iuphar.ligand:6920	BENZOLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1558	hgnc:2622	CYP2C8	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8157	iuphar.ligand:8157	COMPOUND 15B [PMID: 18334293]	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.3281729452230906	IUPHAR.LIGAND:4319	rxcui:10328	TANNIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1618	hgnc:2685	DAZL	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:5299	iuphar.ligand:5299	Z-VDVAD-FMK	FALSE	FALSE	FALSE
NCBIGENE:1995	hgnc:3314	ELAVL3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8154	iuphar.ligand:8154	COMPOUND 14 [PMID: 24900428]	FALSE	FALSE	FALSE
NCBIGENE:1997	hgnc:3316	ELF1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:5985	iuphar.ligand:5985	IC261	FALSE	FALSE	FALSE
NCBIGENE:1597	hgnc:2312	CPN1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8656	iuphar.ligand:8656	SQ-24,798	FALSE	FALSE	FALSE
NCBIGENE:1998	hgnc:3317	ELF2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5985	iuphar.ligand:5985	IC261	FALSE	FALSE	FALSE
NCBIGENE:3273	hgnc:5181	HRG	GuideToPharmacology	2024.1	modulator	13.12691780892362	IUPHAR.LIGAND:9978	iuphar.ligand:9978	ONC201	FALSE	FALSE	FALSE
NCBIGENE:2345	ncbigene:2345	FNZ	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8634	iuphar.ligand:8634	COMPOUND 3 [PMID: 8410973]	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.4070362111294147	IUPHAR.LIGAND:7720	iuphar.ligand:7720	ML218	FALSE	FALSE	FALSE
NCBIGENE:2351	ncbigene:2351	FOLR2L	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10883	iuphar.ligand:10883	GC-376	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:736	iuphar.ligand:736	[3H]WIN55212-2	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:888	iuphar.ligand:888	YM-022	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:769	iuphar.ligand:769	CCL11	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	modulator	0.7955707762984014	IUPHAR.LIGAND:7825	iuphar.ligand:7825	AZD2423	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.5000730593875666	IUPHAR.LIGAND:765	iuphar.ligand:765	[125I]CCL7 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:835	iuphar.ligand:835	CXCL10	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:11598	iuphar.ligand:11598	BMS-741672	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:769	iuphar.ligand:769	CCL11	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4338	iuphar.ligand:4338	UCCF-853	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1426838892274307	IUPHAR.LIGAND:7124	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1630673019742065	IUPHAR.LIGAND:4795	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:10240	iuphar.ligand:10240	SC-560	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.081533651	IUPHAR.LIGAND:2593	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:918	iuphar.ligand:918	SAUVAGINE	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	antibody	0.750109589	IUPHAR.LIGAND:9161	iuphar.ligand:9161	ULOCUPLUMAB	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:5707	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:5951	iuphar.ligand:5951	CDK4 INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:5938	iuphar.ligand:5938	BOHEMINE	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:12881	iuphar.ligand:12881	TIBREMCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:10313	ncit:C138165	LEROCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	0.1615620653405984	IUPHAR.LIGAND:5890	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:9405	iuphar.ligand:9405	BS-181	FALSE	FALSE	FALSE
NCBIGENE:1982	hgnc:3297	EIF4G2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8160	iuphar.ligand:8160	COMPOUND 9B [PMID: 18986805]	FALSE	FALSE	FALSE
NCBIGENE:2027	hgnc:3354	ENO3	GuideToPharmacology	2024.1	inhibitor	0.9053046764774914	IUPHAR.LIGAND:5269	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
NCBIGENE:1365	hgnc:2045	CLDN3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8852	iuphar.ligand:8852	COMPOUND 4D [PMID: 20655626]	FALSE	FALSE	FALSE
NCBIGENE:1332	hgnc:2272	COX5BP3	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:2608	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
NCBIGENE:1321	ncbigene:1321	CORD4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8756	iuphar.ligand:8756	COMPOUND 23 [PMID: 17125252]	FALSE	FALSE	FALSE
NCBIGENE:1327	hgnc:2265	COX4I1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8833	iuphar.ligand:8833	COMPOUND 9 [PMID: 11606127]	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:3322	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:5861	ncit:C77981	IRALUKAST	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3414	iuphar.ligand:3358	ICI198615	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:3322	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.051629962	IUPHAR.LIGAND:1663	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1548898856510162	IUPHAR.LIGAND:1641	iuphar.ligand:1641	NALTRINDOLE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:1612	iuphar.ligand:1612	[3H]DIPRENORPHINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.077444943	IUPHAR.LIGAND:7563	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
NCBIGENE:1397	hgnc:2361	CRIP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10244	iuphar.ligand:10244	DH376	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11554	iuphar.ligand:11554	DSM705	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.004068785	IUPHAR.LIGAND:940	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.055563673	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8626	iuphar.ligand:8626	COMPOUND 4G [PMID: 22595175]	FALSE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:6476	ncit:C125714	ALVELESTAT	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9881	iuphar.ligand:9881	EBI-2511	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:11948	iuphar.ligand:11948	TIGOZERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:12380	iuphar.ligand:12380	MIFANERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.016131389	IUPHAR.LIGAND:5692	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:12612	iuphar.ligand:12612	PIROTINIB	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3156	iuphar.ligand:3156	COMPOUND 2 [PMID: 18295483]	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:5235	iuphar.ligand:5235	OL135	FALSE	FALSE	FALSE
NCBIGENE:2608	hgnc:3594	FASN	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8605	iuphar.ligand:8605	GSK2194069	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6487	iuphar.ligand:6487	CATPB	FALSE	FALSE	FALSE
PRIM1	hgnc:9369	PRIM1	ChEMBL	33	inhibitor	0.080656945	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2806	drugbank:DB08231	MYRISTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1062	rxcui:34658	PROPIONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2024	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:227	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1062	rxcui:34658	PROPIONIC ACID	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	modulator	0.046965717	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
NCBIGENE:227	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:6500	iuphar.ligand:6500	1-METHYLCYCLOPROPANECARBOXYLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:8138	iuphar.ligand:8138	COMPOUND 2C [PMID: 24900538]	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:7649	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
NCBIGENE:2365	hgnc:3873	FRA1F	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8563	iuphar.ligand:8563	ARI-3099	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:9767	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:11414	iuphar.ligand:11414	TASURGRATINIB	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	modulator	0.042968634	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
NCBIGENE:2609	hgnc:4145	GAPDHP67	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:5433	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NCBIGENE:3176	hgnc:5028	HNMT	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:11480	iuphar.ligand:11480	SLF	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.054695491	IUPHAR.LIGAND:9383	iuphar.ligand:9383	OSI-930	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.017092341	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:8108	iuphar.ligand:8108	DENFIVONTINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:7969	iuphar.ligand:7969	AKN-028	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.020836377	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	modulator	0.096167896	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:5689	iuphar.ligand:5689	JNJ-28312141	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:610	rxcui:3194	DEOXYCHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5831	iuphar.ligand:5831	PYRAZOLONE, 1	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6240	iuphar.ligand:6240	MMK-1	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.42006137	IUPHAR.LIGAND:1894	ncit:C79571	CLOPROSTENOL	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:6263	iuphar.ligand:6263	COMPOUND 1754-31 [PMID: 23788657]	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1030	iuphar.ligand:1030	T-BOC-FLFLF	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:7451	rxcui:1244607	TAFLUPROST	TRUE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.2625383561784725	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	modulator	0.048083948	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
NCBIGENE:253	ncbigene:253	ALS3	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:3780	iuphar.ligand:3780	[125I]FSH (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4094	iuphar.ligand:4094	&ALPHA;3IA	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.060077427	IUPHAR.LIGAND:4322	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6104	iuphar.ligand:6104	M1153	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:4685	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1743	hgnc:2911	DLST	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:4851	iuphar.ligand:4851	[125I]GDNF (RAT)	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	inhibitor	0.1172046232939609	IUPHAR.LIGAND:4264	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	NULL	0.6563458904461812	IUPHAR.LIGAND:4081	iuphar.ligand:4081	[3H]CNQX	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:4264	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:451	hgnc:769	ASS1P6	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:4181	drugbank:DB02852	DOMOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	blocker	0.051782713	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.1767935058440892	IUPHAR.LIGAND:3879	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
NCBIGENE:936	hgnc:1647	CD24P2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4767	iuphar.ligand:4767	ALX 1405	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	0.2430910705356226	IUPHAR.LIGAND:1015	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1184	iuphar.ligand:1184	T-98475	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:5582	iuphar.ligand:5582	WAY-207024	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1191	iuphar.ligand:1191	CYCLORELIX	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.054020238	IUPHAR.LIGAND:7005	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.084553416	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.08914715	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.2430910705356227	IUPHAR.LIGAND:8391	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.2403097081725148	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:9891	iuphar.ligand:9891	MARBOSTAT-100	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.1400204566285186	IUPHAR.LIGAND:7495	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.212581665	IUPHAR.LIGAND:7497	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.054695491	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.4861821410712454	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.2333674277141978	IUPHAR.LIGAND:7505	iuphar.ligand:7505	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.031765076	IUPHAR.LIGAND:34	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:11579	ncit:C73045	BILASTINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:1206	iuphar.ligand:1206	(&PLUSMN;)-CIS-H2-PAT	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.027433475	IUPHAR.LIGAND:85	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:10103	ncit:C73055	RUPATADINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.050294704	IUPHAR.LIGAND:277	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:4819	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.060353645	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1200	iuphar.ligand:1200	UR-PG146	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.059667808	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:8924	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
NCBIGENE:3222	hgnc:5127	HOXC5	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12478	iuphar.ligand:12478	BI-3231	FALSE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.047518255	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3006	iuphar.ligand:3006	COMPOUND 41 [PMID: 17574411]	FALSE	FALSE	FALSE
NCBIGENE:83	hgnc:155	ACTG1P10	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:4839	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5847	iuphar.ligand:5847	2-HYDROXY CAPRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:156	hgnc:289	GRK2	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:5535	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.1029562181092048	LOXAPINE SUCCINATE	rxcui:6476	LOXAPINE SUCCINATE	TRUE	FALSE	FALSE
NCBIGENE:3019	hgnc:27269	IDO2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10126	iuphar.ligand:10126	TRYPTANTHRIN 5I	FALSE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12988	iuphar.ligand:12988	ERAS-5024	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.2344092465879218	IUPHAR.LIGAND:1893	iuphar.ligand:1893	CARBACYCLIN	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:12437	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:10148	iuphar.ligand:10148	JAK INHIBITOR 17B	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:10147	iuphar.ligand:10147	JAK INHIBITOR 20A	FALSE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.1235474617310458	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1621	iuphar.ligand:1621	DYNORPHIN A-(1-8)	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1644	iuphar.ligand:1644	&BETA;-NEOENDORPHIN	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.076765601	IUPHAR.LIGAND:7591	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:1669	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	1.500219178	ETHOSUXIMIDE	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.023060023	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.013836014	IUPHAR.LIGAND:7649	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.02075402	IUPHAR.LIGAND:7707	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.012971263	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1280	iuphar.ligand:1280	[125I]TYR45-KISSPEPTIN-15	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:12870	iuphar.ligand:12870	LABUXTINIB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:7969	iuphar.ligand:7969	AKN-028	FALSE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	1.750255707856483	ETHOSUXIMIDE	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
NCBIGENE:520	hgnc:844	ATP5MC2P1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
NCBIGENE:437	hgnc:6266	KCNJ5	GuideToPharmacology	2024.1	blocker	5.834185692854944	IUPHAR.LIGAND:2408	iuphar.ligand:2408	NIP-142	FALSE	FALSE	FALSE
NCBIGENE:386	hgnc:18866	KCNT2	GuideToPharmacology	2024.1	blocker	0.4861821410712454	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.091159151	IUPHAR.LIGAND:2608	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	ChEMBL	33	inhibitor	2.019525817	VORAPAXAR SULFATE	rxcui:1537050	VORAPAXAR SULFATE	TRUE	FALSE	FALSE
NCBIGENE:539	hgnc:850	ATP5PO	GuideToPharmacology	2024.1	blocker	17.50255707856483	IUPHAR.LIGAND:11476	iuphar.ligand:11476	&KAPPA;M-CONOTOXIN RIIIK	FALSE	FALSE	FALSE
NCBIGENE:540	hgnc:870	ATP7B	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:9582	iuphar.ligand:9582	HSTX1[R14A]	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	2.019525817	IUPHAR.LIGAND:12650	ncit:C188540	AZETUKALNER	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.079718124	ARIPIPRAZOLE LAUROXIL	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2596	iuphar.ligand:2596	XE991	FALSE	FALSE	FALSE
NCBIGENE:552	hgnc:895	AVPR1A	GuideToPharmacology	2024.1	blocker	0.1268301237577161	IUPHAR.LIGAND:2343	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	inhibitor	0.577007376	IUPHAR.LIGAND:2599	ncit:C82306	LINOPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	activator	0.9723642821424906	IUPHAR.LIGAND:2600	iuphar.ligand:2600	(S)-N-[1-(3-MORPHOLIN-4-YL-PHENYL)-ETHYL]-3-PHENYL-ACRYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8209	iuphar.ligand:8209	COMPOUND 35 [PMID: 20684608]	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8073	iuphar.ligand:8073	GNE-7915	FALSE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12663	iuphar.ligand:12663	TRULI	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:10108	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8118	iuphar.ligand:8118	COMPOUND 30 [PMID: 22902653]	FALSE	FALSE	FALSE
NCBIGENE:1391	hgnc:6719	LTC4S	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9555	iuphar.ligand:9555	EXAMPLE 36 [WO2016177845]	FALSE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9091	iuphar.ligand:9091	COMPOUND 1A [PMID: 25692029]	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.078136416	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
NCBIGENE:2593	hgnc:4136	GAMT	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6702	iuphar.ligand:6702	COMPOUND 41 [PMID: 15026062]	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:2742	iuphar.ligand:2742	22R-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:2907	iuphar.ligand:2907	KI16425	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:5450	iuphar.ligand:5450	VPC32179	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:2905	iuphar.ligand:2905	AM966	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	1.693795846312725	GLPG-0555	chembl:CHEMBL3545249	GLPG-0555	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7024	iuphar.ligand:7024	NCL-1	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.2430910705356227	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:2675	hgnc:4244	GFRA2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9584	iuphar.ligand:9584	ML324	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1335	iuphar.ligand:1335	AGOUTI-RELATED PROTEIN	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6215	iuphar.ligand:6215	COMPOUND 11S [PMID: 19433355]	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.1544343271638073	IUPHAR.LIGAND:1365	iuphar.ligand:1365	(1S,3R)-ACPD	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6356	iuphar.ligand:6356	COMPOUND 9A [PMID: 22266036]	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:1377	iuphar.ligand:1377	DCG-IV	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:1402	iuphar.ligand:1402	4-MPPTS	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	0.036087747	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1407	iuphar.ligand:1407	(S)-3,4-DCPG	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1399	iuphar.ligand:1399	[3H]LY341495	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:6008	iuphar.ligand:6008	MEK1/2 INHIBITOR	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.1458546423213736	GSK-461364	iuphar.ligand:5684	GSK-461364A	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	0.5303805175322677	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:299	ncit:C76041	FURTRETHONIUM IODIDE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.050246575	IUPHAR.LIGAND:359	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:318	iuphar.ligand:318	[3H]QNB	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.035098711	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:308	iuphar.ligand:308	P-F-HHSID	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:318	iuphar.ligand:318	[3H]QNB	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:309	iuphar.ligand:309	OTENZEPAD	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1136529680426287	IUPHAR.LIGAND:297	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1562728310586145	SURUFATINIB	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.079557078	IUPHAR.LIGAND:288	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.046798281	IUPHAR.LIGAND:57	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:7549	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:7774	iuphar.ligand:7774	EFPPEA	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:11196	iuphar.ligand:11196	ICOA-13	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1348	iuphar.ligand:1348	GR 128107	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:10726	iuphar.ligand:10726	3F-MT-45	FALSE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:2613	iuphar.ligand:2613	AFT-II	FALSE	FALSE	FALSE
NCBIGENE:970	hgnc:11937	CD70	GuideToPharmacology	2024.1	inhibitor	0.08780547	IUPHAR.LIGAND:4836	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:2613	iuphar.ligand:2613	AFT-II	FALSE	FALSE	FALSE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	inhibitor	0.1400204566285186	IUPHAR.LIGAND:10119	iuphar.ligand:10119	AM-6120	FALSE	FALSE	FALSE
NCBIGENE:1888	hgnc:3143	EBVS1	GuideToPharmacology	2024.1	NULL	13.12691780892362	IUPHAR.LIGAND:5026	iuphar.ligand:5026	NGF	FALSE	FALSE	FALSE
NCBIGENE:476	hgnc:799	ATP1A1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8883	iuphar.ligand:8883	PHTX-11	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2101	iuphar.ligand:2101	SUBSTANCE P-OME	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11810	iuphar.ligand:11810	CP-424,174	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:2129	iuphar.ligand:2129	N&#8242;,2-DIPHENYLQUINOLINE-4-CARBOHYDRAZIDE	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1469	iuphar.ligand:1469	NEUROMEDIN U-23	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:7925	iuphar.ligand:7925	HAS-NMU	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:11490	iuphar.ligand:11490	CPN-116	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1469	iuphar.ligand:1469	NEUROMEDIN U-23	FALSE	FALSE	FALSE
NCBIGENE:310	hgnc:545	ANXA7	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1569	iuphar.ligand:1569	JMV431	FALSE	FALSE	FALSE
NCBIGENE:2129	hgnc:14311	NUAK1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11085	iuphar.ligand:11085	HTH-02-006	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	NULL	0.3804903712731485	IUPHAR.LIGAND:4687	iuphar.ligand:4687	[3H]ESTRADIOL-17&BETA;-GLUCURONIDE	FALSE	FALSE	FALSE
NCBIGENE:2964	hgnc:4654	GTF2F2P1	GuideToPharmacology	2024.1	blocker	10.50153424713889	IUPHAR.LIGAND:10041	iuphar.ligand:10041	CRAC CHANNEL INHIBITOR 1 [PMID: 26256403]	FALSE	FALSE	FALSE
NCBIGENE:3101	hgnc:4925	HK3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:11953	iuphar.ligand:11953	LY3372689	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	0.2822993077187876	IUPHAR.LIGAND:1711	iuphar.ligand:1711	2MESATP	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:1711	iuphar.ligand:1711	2MESATP	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1726	iuphar.ligand:1726	[32P]MRS2500	FALSE	FALSE	FALSE
NCBIGENE:2390	hgnc:3902	FRA4C	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8634	iuphar.ligand:8634	COMPOUND 3 [PMID: 8410973]	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:12493	iuphar.ligand:12493	ISOX-CHA-CHG-ARK(SULFO-CY5)-NH2	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:4061	iuphar.ligand:4061	AYPGKF-NH2	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:2678	iuphar.ligand:2678	NS-220	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:11137	ncit:C167015	SELADELPAR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:11137	ncit:C167015	SELADELPAR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.034727296	IUPHAR.LIGAND:3322	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:8701	iuphar.ligand:8701	TAGITININ A	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:9888	iuphar.ligand:9888	MDG 548	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:9997	iuphar.ligand:9997	AZD3458	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.065552648	IUPHAR.LIGAND:6741	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:11699	iuphar.ligand:11699	AMDIZALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:10233	iuphar.ligand:10233	AZ2	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:10441	iuphar.ligand:10441	COMPOUND 5D [PMID: 31335136]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:11699	iuphar.ligand:11699	AMDIZALISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:10233	iuphar.ligand:10233	AZ2	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:10627	ncit:C123925	ZANDELISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.051478109	IUPHAR.LIGAND:12616	iuphar.ligand:12616	DS-7423	FALSE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:10627	ncit:C123925	ZANDELISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:9997	iuphar.ligand:9997	AZD3458	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.3431873936973496	POSELTINIB	ncit:C141273	POSELTINIB	FALSE	FALSE	FALSE
NCBIGENE:1296	hgnc:2216	COL8A2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11099	iuphar.ligand:11099	COMPOUND 3M [PMID: 32603117]	FALSE	FALSE	FALSE
NCBIGENE:1297	hgnc:2217	COL9A1	GuideToPharmacology	2024.1	activator	2.100306849	IUPHAR.LIGAND:2347	iuphar.ligand:2347	CYCLIC GMP	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8377	iuphar.ligand:8377	PF-00489791	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	1.009762908	LGX-806	chembl:CHEMBL3545263	LGX-806	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:6558	ncit:C83728	GISADENAFIL	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:11099	iuphar.ligand:11099	COMPOUND 3M [PMID: 32603117]	FALSE	FALSE	FALSE
NCBIGENE:1305	hgnc:2190	COL13A1	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:9151	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:12781	iuphar.ligand:12781	TPN171	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:12518	iuphar.ligand:12518	NERANDOMILAST	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:9367	iuphar.ligand:9367	LGB321	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1041818873724097	KRN-633	iuphar.ligand:6057	VEGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:6978	iuphar.ligand:6978	SEMAGACESTAT	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:8664	iuphar.ligand:8664	WAY-255348	FALSE	FALSE	FALSE
NCBIGENE:2167	hgnc:3559	FABP4	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12072	iuphar.ligand:12072	(S)-RP-6306	FALSE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1871	iuphar.ligand:1871	PRRP-20	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:1827	iuphar.ligand:1827	TIP39-(7-39) (HUMAN/BOVINE)	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:10658	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9389	iuphar.ligand:9389	SB590885	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1041818873724097	KRN-633	iuphar.ligand:6057	VEGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:599	hgnc:995	BCL2L2	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:8906	iuphar.ligand:8906	CD2314	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:9867	iuphar.ligand:9867	TAK-828F	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10144	iuphar.ligand:10144	SR2211	FALSE	FALSE	FALSE
NCBIGENE:599	hgnc:995	BCL2L2	GuideToPharmacology	2024.1	agonist	0.072125922	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:599	hgnc:995	BCL2L2	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:598	hgnc:992	BCL2L1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:3432	iuphar.ligand:3432	7-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8911	ncit:C152866	VEROSUDIL	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1250182648468916	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.046303061	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
NCBIGENE:1856	hgnc:3086	DVL2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8831	iuphar.ligand:8831	COMPOUND 1 [PMID: 21882820]	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	inhibitor	0.8078103267029922	IUPHAR.LIGAND:4371	iuphar.ligand:4371	B-R13/17K H2 RELAXIN	FALSE	FALSE	FALSE
NCBIGENE:1525	hgnc:2559	CXADR	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8181	iuphar.ligand:8181	COMPOUND 1 [PMID: 20005102]	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:12501	iuphar.ligand:12501	SA10SC-RLX	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:9889	iuphar.ligand:9889	RP-101075	FALSE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	inhibitor	0.5048814541893702	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.092606122	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:9496	iuphar.ligand:9496	A-971432	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.3431873936973497	IUPHAR.LIGAND:911	iuphar.ligand:911	SPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:2924	iuphar.ligand:2924	FINGOLIMOD-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:3103	hgnc:10721	SELP	GuideToPharmacology	2024.1	NULL	5.250767123569449	IUPHAR.LIGAND:10014	iuphar.ligand:10014	SELECTIN P LIGAND	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.2465148884304905	SR-13668	chembl:CHEMBL245030	SR-13668	FALSE	FALSE	FALSE
NCBIGENE:2219	hgnc:3623	FCN1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11812	iuphar.ligand:11812	XMU-MP-1	FALSE	FALSE	FALSE
NCBIGENE:1517	hgnc:2540	CTSLP2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8209	iuphar.ligand:8209	COMPOUND 35 [PMID: 20684608]	FALSE	FALSE	FALSE
NCBIGENE:2632	hgnc:4180	GBE1	GuideToPharmacology	2024.1	activator	1.500219178162699	IUPHAR.LIGAND:6803	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	Y-39983	chembl:CHEMBL571948	Y-39983	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3120	iuphar.ligand:3120	COMPOUND 15 [PMID: 19456099]	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3122	iuphar.ligand:3122	COMPOUND 35 [PMID: 19191557]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5632	iuphar.ligand:5632	[GA-DOTA,TYR3,THR8]OCTREOTIDE	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2013	iuphar.ligand:2013	KE 108	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2040	iuphar.ligand:2040	BIM 23068	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2047	iuphar.ligand:2047	L-363,301	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2013	iuphar.ligand:2013	KE 108	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2003	iuphar.ligand:2003	BIM 23050	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.1861974157294131	IUPHAR.LIGAND:2007	iuphar.ligand:2007	CORTISTATIN-14	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:7763	iuphar.ligand:7763	ANALOG 32 [PMID:18543899]	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2019	iuphar.ligand:2019	SRIF-14	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	2.838252499226729	FIGOPITANT	ncit:C81498	FIGOPITANT	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2041	iuphar.ligand:2041	BIM 23197	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2059	iuphar.ligand:2059	[111IN,90Y]DOTA-TOC	FALSE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:10128	iuphar.ligand:10128	STING AGONIST 3	FALSE	FALSE	FALSE
NCBIGENE:3241	hgnc:5145	HPCAL1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12814	iuphar.ligand:12814	GNE-7883	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.2548916079402645	IUPHAR.LIGAND:6951	rxcui:3292	DEXTROTHYROXINE	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	inhibitor	1.458546423213736	TC-2216	chembl:CHEMBL504652	TC-2216	FALSE	FALSE	FALSE
NCBIGENE:614	hgnc:7972	NR2C2	GuideToPharmacology	2024.1	agonist	0.2885036881082115	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:1795	hgnc:2989	DOCK3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8194	iuphar.ligand:8194	COMPOUND 15B [PMID: 16539403]	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:10287	iuphar.ligand:10287	TONANTZITLOLONE	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:4206	iuphar.ligand:4206	GSMTX-4	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.172722603	PYROTINIB	ncit:C111895	PYROTINIB	FALSE	FALSE	FALSE
NCBIGENE:499	ncbigene:499	ATP5A2	GuideToPharmacology	2024.1	blocker	1.591141552596803	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.033615667	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	modulator	6.563458904461812	IUPHAR.LIGAND:12541	iuphar.ligand:12541	APV207095A	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.1875273972703375	IUPHAR.LIGAND:2432	iuphar.ligand:2432	RUTHENIUM RED	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	1.944728564284981	IUPHAR.LIGAND:12554	iuphar.ligand:12554	QUINAZOLIN-4(3H) DERIVATIVE 36	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4109	iuphar.ligand:4109	5'-IODORESINIFERATOXIN	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.5585922471882393	IUPHAR.LIGAND:8073	iuphar.ligand:8073	GNE-7915	FALSE	FALSE	FALSE
NCBIGENE:1836	hgnc:10994	SLC26A2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12320	iuphar.ligand:12320	SLC-391	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1223955040459079	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
NCBIGENE:1870	hgnc:3114	E2F2	GuideToPharmacology	2024.1	NULL	5.250767123569449	IUPHAR.LIGAND:5073	iuphar.ligand:5073	TUMOUR NECROSIS FACTOR MEMBRANE FORM	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:9803	iuphar.ligand:9803	SAR-20347	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2153	iuphar.ligand:2153	UROTENSIN-II	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.022099188	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
NCBIGENE:2426	hgnc:3936	FRA9B	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8661	iuphar.ligand:8661	LDN-91946	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2155	iuphar.ligand:2155	UROTENSIN-II	FALSE	FALSE	FALSE
NCBIGENE:2528	hgnc:4017	FUT6	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:4841	rxcui:402316	MIGLUSTAT	TRUE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	0.1553481397505754	IUPHAR.LIGAND:4823	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2280	iuphar.ligand:2280	HELODERMIN	FALSE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:11413	iuphar.ligand:11413	NEMTABRUTINIB	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	1.712206670729168	BMS-911543	drugbank:DB12591	BMS-911543	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:3762	iuphar.ligand:3762	[125I][LEU31,PRO34]NPY	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1549	iuphar.ligand:1549	NPY-(2-36)	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1507	iuphar.ligand:1507	NPY-(13-36) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1507	iuphar.ligand:1507	NPY-(13-36) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:2289	hgnc:3721	FKBP5	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8194	iuphar.ligand:8194	COMPOUND 15B [PMID: 16539403]	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	CIViC	10-Apr-24	NULL	0.022730594	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	0.3472729579080323	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	CIViC	10-Apr-24	NULL	0.064347636	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.012154554	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
BCL2L11	hgnc:994	BCL2L11	CIViC	10-Apr-24	NULL	1.458546423213736	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
CD274	hgnc:17635	CD274	CIViC	10-Apr-24	NULL	0.561579372	DURVALUMAB	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	CIViC	10-Apr-24	NULL	0.9883796938483671	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.039420174	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.8325740682192574	FUTIBATINIB	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
BLK	hgnc:1057	BLK	CIViC	10-Apr-24	NULL	0.037884323	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.024309107	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.030868707	PACRITINIB	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
SMARCA4	hgnc:11100	SMARCA4	CIViC	10-Apr-24	NULL	0.089910396	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.040515178	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.022995101	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.047127304	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
MYD88	hgnc:7562	MYD88	CIViC	10-Apr-24	NULL	1.591141552596803	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.049275217	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
ASNS	hgnc:753	ASNS	CIViC	10-Apr-24	NULL	14.58546423213736	ASPARAGINASE	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
CIC	hgnc:14214	CIC	CIViC	10-Apr-24	NULL	0.5303805175322677	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
SOX10	hgnc:11190	SOX10	CIViC	10-Apr-24	NULL	1.458546423213736	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.078958904	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PREX2	hgnc:22950	PREX2	CIViC	10-Apr-24	NULL	1.458546423213736	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
DNMT3A	hgnc:2978	DNMT3A	CIViC	10-Apr-24	NULL	0.040515178	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.006439499	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	CIViC	10-Apr-24	NULL	0.9053046764774912	PIXANTRONE	ncit:C26663	PIXANTRONE	TRUE	FALSE	TRUE
CREBBP	hgnc:2348	CREBBP	CIViC	10-Apr-24	NULL	0.070197421	THERAPEUTIC GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.2217384765020882	AKT INHIBITOR MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	0.1875273972703375	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
KIT	hgnc:6342	KIT	DoCM	10-Apr-24	NULL	0.4906052389860809	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	DoCM	10-Apr-24	NULL	0.1752202599633854	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	DoCM	10-Apr-24	NULL	0.1900426678745596	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	DoCM	10-Apr-24	NULL	0.5672124979164529	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	DoCM	10-Apr-24	NULL	0.1372749574789398	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.01037701	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.065226921	Ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1099637093941246	Toripalimab-tpzi	rxcui:2669407	TORIPALIMAB-TPZI	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.032616354	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.003665457	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	SAR405838	ncit:C106120	P53-HDM2 INTERACTION INHIBITOR MI-773	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.030545475	Hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.3977853881492007	BMS-906024	ncit:C116872	OSUGACESTAT	FALSE	FALSE	TRUE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.6731752722524935	Pyridone 6	drugbank:DB04716	2-TERT-BUTYL-9-FLUORO-1,6-DIHYDROBENZO[H]IMIDAZO[4,5-F]ISOQUINOLIN-7-ONE	FALSE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	1.902451856365742	ASP3026	ncit:C116727	ALK INHIBITOR ASP3026	FALSE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	7.533709351208341	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.017737081	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.016729292	Carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.061773731	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.2333674277141978	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.2210849315187136	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.079077818	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.3472729579080323	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	1.230648544586589	Revumenib	ncit:C165776	REVUMENIB	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.3241214273808303	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.5385402178019949	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	1.083491628673061	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.7778914257139926	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	XL888	ncit:C79835	HSP90 INHIBITOR XL888	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.066860362	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1693795846312726	Toripalimab-tpzi	rxcui:2669407	TORIPALIMAB-TPZI	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	PF-4708671	iuphar.ligand:8036	PF-4708671	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.054020238	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.4861821410712453	HS-10352	ncit:C179330	PI3K-ALPHA INHIBITOR HS-10352	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.060772768	Voxtalisib	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2217384765020882	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.039420174	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	0.1250182648468916	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.070956312	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.037345428	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2365210416022274	Onatasertib	ncit:C92575	ONATASERTIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CancerCommons	25-Jul-13	inhibitor	1.282909942931453	LGX818	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.05387244	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.051478109	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.062608511	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.059397818	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.033658764	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.030527716	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.030527716	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.033658764	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	BUTABARBITAL SODIUM	rxcui:91109	BUTABARBITAL SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.026586163	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.025003653	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.025929714	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.054020238	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.05913026	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.096050618	PENTOBARBITAL SODIUM	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.03394161	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.087318744	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.039598545	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.02091106	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.019695301	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	ChEMBL	33	agonist	1.250182648468916	LYPRESSIN	rxcui:6531	LYPRESSIN	TRUE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	agonist	0.760980743	LYPRESSIN	rxcui:6531	LYPRESSIN	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	inhibitor	1.715936968486748	BASILIXIMAB	rxcui:196102	BASILIXIMAB	TRUE	TRUE	FALSE
IL12A	hgnc:5969	IL12A	ChEMBL	33	inhibitor	1.050153425	USTEKINUMAB	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
POLD2	hgnc:9176	POLD2	ChEMBL	33	inhibitor	0.4605936073306535	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
POLA2	hgnc:30073	POLA2	ChEMBL	33	inhibitor	0.3947945205691315	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
POLA1	hgnc:9173	POLA1	ChEMBL	33	inhibitor	0.5791287268642776	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLE2	hgnc:9178	POLE2	ChEMBL	33	inhibitor	0.4605936073306535	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
POLE	hgnc:9177	POLE	ChEMBL	33	inhibitor	0.064824285	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
PRIM2	hgnc:9370	PRIM2	ChEMBL	33	inhibitor	0.2573905452730122	FLUDARABINE PHOSPHATE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLD1	hgnc:9175	POLD1	ChEMBL	33	inhibitor	0.2302968036653267	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
POLD3	hgnc:20932	POLD3	ChEMBL	33	inhibitor	0.4605936073306535	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
POLE3	hgnc:13546	POLE3	ChEMBL	33	inhibitor	0.4605936073306535	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
PRIM2	hgnc:9370	PRIM2	ChEMBL	33	inhibitor	0.4605936073306535	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.051277023	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	QUINIDINE SULFATE	rxcui:9069	QUINIDINE SULFATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.043180651	DRONEDARONE HYDROCHLORIDE	rxcui:736680	DRONEDARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	TETRACAINE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.039068208	MEPIVACAINE HYDROCHLORIDE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	ETIDOCAINE HYDROCHLORIDE	rxcui:227221	ETIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.065799087	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	PROPOXYCAINE HYDROCHLORIDE	ncit:C66493	PROPOXYCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	PROPARACAINE HYDROCHLORIDE	rxcui:227778	PROPARACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.042619863	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	INDECAINIDE HYDROCHLORIDE	ncit:C65911	INDECAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	TOCAINIDE HYDROCHLORIDE	ncit:C47761	TOCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1037701012563132	LURASIDONE HYDROCHLORIDE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.2365210416022274	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	ChEMBL	33	inhibitor	1.193356164447602	AVAGACESTAT	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
PSEN1	hgnc:9508	PSEN1	ChEMBL	33	inhibitor	1.009762908	AVAGACESTAT	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.8751278539282416	ETIRINOTECAN PEGOL	ncit:C74069	ETIRINOTECAN PEGOL	FALSE	FALSE	TRUE
DGAT1	hgnc:2843	DGAT1	ChEMBL	33	inhibitor	21.00306849427779	PRADIGASTAT	ncit:C166592	PRADIGASTAT	FALSE	FALSE	FALSE
BIRC3	hgnc:591	BIRC3	ChEMBL	33	inhibitor	0.6250913242344582	BIRINAPANT	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
CHEK2	hgnc:16627	CHEK2	ChEMBL	33	inhibitor	0.5147810905460244	PREXASERTIB	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
CASP9	hgnc:1511	CASP9	ChEMBL	33	inhibitor	2.187819634820604	NIVOCASAN	ncit:C98213	NIVOCASAN	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.07631929	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	binder	3.231241306811969	ADUCANUMAB	rxcui:2557217	ADUCANUMAB	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.069180068	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
TNFRSF12A	hgnc:18152	TNFRSF12A	ChEMBL	33	agonist	105.0153424713889	ENAVATUZUMAB	ncit:C80045	ENAVATUZUMAB	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	1.129197231	PEGSUNERCEPT	ncit:C90875	PEGSUNERCEPT	FALSE	FALSE	FALSE
MSTN	hgnc:4223	MSTN	ChEMBL	33	inhibitor	2.187819634820604	STAMULUMAB	ncit:C95795	STAMULUMAB	FALSE	FALSE	FALSE
ITGA2	hgnc:6137	ITGA2	ChEMBL	33	inhibitor	26.25383561784724	VATELIZUMAB	ncit:C152838	VATELIZUMAB	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	binder	2.423430980108977	GSK933776	chembl:CHEMBL2109300	GSK933776	FALSE	FALSE	FALSE
S1PR5	hgnc:14299	S1PR5	ChEMBL	33	modulator	2.625383561784725	AMISELIMOD HYDROCHLORIDE	ncit:C142922	AMISELIMOD HYDROCHLORIDE	FALSE	FALSE	FALSE
IFNA4	hgnc:5425	IFNA4	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
IFNA16	hgnc:5421	IFNA16	ChEMBL	33	inhibitor	2.019525816757481	RONTALIZUMAB	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
HTR5A	hgnc:5300	HTR5A	ChEMBL	33	inhibitor	0.5048814541893702	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.1442518440541058	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	inhibitor	0.081872668	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
ACE1	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.1271372184883643	CARBARIL	ncit:C76389	CARBARIL	TRUE	FALSE	FALSE
TNNI3	hgnc:11947	TNNI3	ChEMBL	33	positive modulator	1.875273972703374	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	agonist	0.091159151	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.057700738	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	ChEMBL	33	binder	2.917092846427472	MIRVETUXIMAB	ncit:C166766	MIRVETUXIMAB	FALSE	FALSE	FALSE
CD33	hgnc:1659	CD33	ChEMBL	33	binder	4.039051633514961	AVE-9633	chembl:CHEMBL2109266	AVE-9633	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	2.917092846427472	EPRATUZUMAB 90Y	chembl:CHEMBL2108357	EPRATUZUMAB 90Y	FALSE	FALSE	FALSE
CD28	hgnc:1653	CD28	ChEMBL	33	agonist	3.500511415712966	TGN-1412	chembl:CHEMBL2109250	TGN-1412	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	modulator	0.729273212	SOLITOMAB	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
MSTN	hgnc:4223	MSTN	ChEMBL	33	inhibitor	2.187819634820604	TREVOGRUMAB	ncit:C152733	TREVOGRUMAB	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	2.187819634820604	CMB-401	chembl:CHEMBL2109284	CMB-401	FALSE	FALSE	FALSE
NECTIN4	hgnc:19688	NECTIN4	ChEMBL	33	binder	4.118248724368196	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
GPA33	hgnc:4445	GPA33	ChEMBL	33	binder	39.38075342677087	KRN-330	chembl:CHEMBL2109293	KRN-330	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.5147810905460245	ELSUBRUTINIB	ncit:C175777	ELSUBRUTINIB	FALSE	FALSE	FALSE
LTB4R	hgnc:6713	LTB4R	ChEMBL	33	inhibitor	3.281729452230906	CP-195543	drugbank:DB13053	CP-195543	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.041672755	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.035719504	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.6563458904461812	RUBITECAN	ncit:C1485	RUBITECAN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.042689164	PACLITAXEL DOCOSAHEXAENOIC ACID	drugbank:DB05297	PACLITAXEL DOCOSAHEXAENOIC ACID	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.042174836	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.042689164	PATUPILONE	ncit:C1623	PATUPILONE	FALSE	FALSE	FALSE
SELE	hgnc:10718	SELE	ChEMBL	33	inhibitor	4.773424657790408	UPROLESELAN	ncit:C119743	UPROLESELAN	FALSE	FALSE	FALSE
GCK	hgnc:4195	GCK	ChEMBL	33	activator	3.500511415712966	DORZAGLIATIN	ncit:C169919	DORZAGLIATIN	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	ChEMBL	33	inhibitor	0.2243917574174978	TANZISERTIB	ncit:C152510	TANZISERTIB	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1190650141398968	NEMIRALISIB	ncit:C174798	NEMIRALISIB	FALSE	FALSE	FALSE
KLB	hgnc:15527	KLB	ChEMBL	33	agonist	6.563458904461812	FAZPILODEMAB	ncit:C188644	FAZPILODEMAB	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.064033745	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inverse agonist	0.7721716358190367	SUVN-G3031	drugbank:DB14835	SUVN-G3031	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.1635752997996713	HMPL-453	chembl:CHEMBL4650297	HMPL-453	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.037666909	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	RG-7600	chembl:CHEMBL2109281	RG-7600	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	SOFITUZUMAB VEDOTIN	ncit:C106119	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.1286952726365061	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
MSLN	hgnc:7371	MSLN	ChEMBL	33	binder	1.944728564284981	LMB-100	drugbank:DB18591	LMB-100	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	ELRANATAMAB	rxcui:2644880	ELRANATAMAB	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	SISOMICIN	rxcui:9806	SISOMICIN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.04182212	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	ChEMBL	33	inhibitor	0.07699072	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.099446347	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
TIGIT	hgnc:26838	TIGIT	ChEMBL	33	inhibitor	6.563458904461812	IBI-939	chembl:CHEMBL4650473	IBI-939	FALSE	FALSE	FALSE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	0.8334550989792776	VODOBATINIB	ncit:C174748	VODOBATINIB	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.1435420208739598	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
HSD11B1	hgnc:5208	HSD11B1	ChEMBL	33	inhibitor	3.088686543276147	BI-187004	chembl:CHEMBL3669417	BI-187004	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	agonist	0.3070624048871023	TALSACLIDINE	ncit:C96885	TALSACLIDINE	FALSE	FALSE	FALSE
NPR3	hgnc:7945	NPR3	ChEMBL	33	agonist	4.375639269641208	CARPERITIDE	ncit:C169829	CARPERITIDE	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	ChEMBL	33	inhibitor	7.501095891	SAR-113945	chembl:CHEMBL3544945	SAR-113945	FALSE	FALSE	FALSE
GP6	hgnc:14388	GP6	ChEMBL	33	inhibitor	26.25383561784724	GLENZOCIMAB	ncit:C166827	GLENZOCIMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	0.926605963	ERFONRILIMAB	ncit:C157632	ERFONRILIMAB	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.061628722	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.078136416	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	SPIRAMYCIN	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
TIGIT	hgnc:26838	TIGIT	ChEMBL	33	inhibitor	6.563458904461812	DOMVANALIMAB	ncit:C162875	DOMVANALIMAB	FALSE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.729273212	RUNCACIGUAT	ncit:C166842	RUNCACIGUAT	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1988926940746003	FAXELADOL	ncit:C80579	FAXELADOL	FALSE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	2.917092846427472	ORN-0829 HYDRATE	chembl:CHEMBL4650522	ORN-0829 HYDRATE	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.7955707762984014	OLSALAZINE	rxcui:32385	OLSALAZINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.038808331	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.03409589	AG-538	chembl:CHEMBL56393	CHEMBL:CHEMBL56393	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.038467158	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	ChEMBL	33	inhibitor	0.9376369863516875	NELIVAPTAN	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1944728564284981	GNF-PF-4864	chembl:CHEMBL583558	CHEMBL:CHEMBL583558	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.012573676	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002359895	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.09669921	TCMDC-125180	chembl:CHEMBL586163	CHEMBL:CHEMBL586163	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.043466615	MMV009085	chembl:CHEMBL581225	CHEMBL:CHEMBL581225	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.086789539	NSC-180246	chembl:CHEMBL484640	CHEMBL:CHEMBL484640	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	DEXBROMPHENIRAMINE MALEATE	rxcui:48936	DEXBROMPHENIRAMINE MALEATE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	1.419126249613364	TARAFENACIN	ncit:C87644	TARAFENACIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	NANAOMYCIN	chembl:CHEMBL1212972	NANAOMYCIN	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	1.280674908	VOACANGINE	chembl:CHEMBL182120	VOACANGINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.030038714	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	BETUNOLIC ACID	chembl:CHEMBL431525	BETUNOLIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000053346	chembl:CHEMBL590201	CHEMBL:CHEMBL590201	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.061412481	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002553627	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NSC-116702	chembl:CHEMBL1477383	CHEMBL:CHEMBL1477383	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	inhibitor	1.750255707856483	DRINABANT	ncit:C166890	DRINABANT	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	NSC-99550	chembl:CHEMBL1288014	CHEMBL:CHEMBL1288014	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.022632617	MICONAZOLE NITRATE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.050879526	GAMOLENIC ACID	rxcui:25605	GAMMA-LINOLENIC ACID	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.087952548	IRETOL	chembl:CHEMBL1606248	IRETOL	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	PURVALANOLA	chembl:CHEMBL23327	PURVALANOLA	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	CLOFAZIMINE	rxcui:2592	CLOFAZIMINE	TRUE	FALSE	FALSE
PTGER4	hgnc:9596	PTGER4	ChEMBL	33	agonist	3.088686543276147	RIVENPROST	ncit:C87384	RIVENPROST	FALSE	FALSE	FALSE
BBOX1	hgnc:964	BBOX1	DTC	9/2/20	NULL	1.000146118775133	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.2885036881082116	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.026253836	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	EMODIC ACID	chembl:CHEMBL290914	EMODIC ACID	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.047561296	CARMINE	chembl:CHEMBL1366408	CARMINE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.075442056	PROSTAGLANDIN B1	chembl:CHEMBL1561148	PROSTAGLANDIN B1	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.042516333	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.033148782	681640	chembl:CHEMBL379975	CHEMBL:CHEMBL379975	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	0.7095631248066824	EZLOPITANT	ncit:C97962	EZLOPITANT	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1875273972703374	PROTOAPIGENONE	chembl:CHEMBL414890	PROTOAPIGENONE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	ORTHOTOLIDINE	chembl:CHEMBL85109	ORTHOTOLIDINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	WAY-100,635	iuphar.ligand:3251	[3H]WAY100635	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.012433737	HEXACHLOROPHENE	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.037884323	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.29374921	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
MC4R	hgnc:6932	MC4R	ChEMBL	33	agonist	1.250182648468916	SETMELANOTIDE	rxcui:2469247	SETMELANOTIDE	TRUE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.2545826484154885	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2917092846427472	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ZWITTERGENT 3-12	chembl:CHEMBL1235854	CHEMBL:CHEMBL1235854	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	TCMDC-124355	chembl:CHEMBL531401	CHEMBL:CHEMBL531401	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1166837138570988	TRICLOSAN	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	GALLIC ACID	rxcui:1311389	GALLIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	METHAPHIT	chembl:CHEMBL41541	METHAPHIT	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	NORTRIPTYLINE HYDROCHLORIDE	rxcui:203130	NORTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	DNDI1417941	chembl:CHEMBL2095095	CHEMBL:CHEMBL2095095	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FENAMIDONE	chembl:CHEMBL1232792	FENAMIDONE	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	1.193356164447602	SYROSINGOPINE	ncit:C152485	SYROSINGOPINE	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	agonist	0.2778183663264258	APIMOSTINEL	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	(-)-HERDMANINE K	chembl:CHEMBL2208195	CHEMBL:CHEMBL2208195	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	10-(4-PYRIDYL)CAMPTOTHECIN HCL	chembl:CHEMBL1762594	CHEMBL:CHEMBL1762594	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GITOXIGENIN	chembl:CHEMBL464658	GITOXIGENIN	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	SULFISOXAZOLE	rxcui:10207	SULFISOXAZOLE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	DNDI1416955	chembl:CHEMBL1327172	CHEMBL:CHEMBL1327172	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	positive modulator	0.096167896	NEBOGLAMINE	ncit:C66222	NEBOGLAMINE	FALSE	FALSE	FALSE
GGPS1	hgnc:4249	GGPS1	DTC	9/2/20	NULL	26.25383561784724	DIGERANYL BISPHOSPHONATE	iuphar.ligand:3187	DIGERANYL BISPHOSPHONATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	HEMICHOLINIUM-3	iuphar.ligand:4494	HEMICHOLINIUM-3	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.08780547	AZAKENPAULLONE	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.002506094	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.096521454	SULFURETIN	chembl:CHEMBL490355	SULFURETIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	THUNBERGINOL E	chembl:CHEMBL421486	THUNBERGINOL E	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	GNF-PF-1134	chembl:CHEMBL600694	CHEMBL:CHEMBL600694	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	agonist	0.2778183663264258	RAPASTINEL	ncit:C152156	RAPASTINEL	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIK	chembl:CHEMBL1094689	AESCULIOSIDE IIK	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	DICYCLOMINE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.009840268	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.028810794	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	EQUILIN	ncit:C29020	EQUILIN	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.018106094	NSC-95397	chembl:CHEMBL429095	CHEMBL:CHEMBL429095	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.078136416	PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE	chembl:CHEMBL114544	CHEMBL:CHEMBL114544	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	agonist	0.096167896	RAPASTINEL	ncit:C152156	RAPASTINEL	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	1.029562181092048	GNF-PF-4665	chembl:CHEMBL601744	CHEMBL:CHEMBL601744	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005905046	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.016008436	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	DINALINE	ncit:C79870	DINALINE	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	positive modulator	0.1530835896084387	NEBOGLAMINE	ncit:C66222	NEBOGLAMINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	TYRPHOSTIN 51	chembl:CHEMBL78257	TYRPHOSTIN 51	FALSE	FALSE	FALSE
SLC6A15	hgnc:13621	SLC6A15	DTC	9/2/20	NULL	5.527123287967842	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	GNF-PF-3407	chembl:CHEMBL602990	CHEMBL:CHEMBL602990	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.010620484	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	agonist	0.2586584789935689	APIMOSTINEL	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	NSC-74429	chembl:CHEMBL1269022	CHEMBL:CHEMBL1269022	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	DNDI1340257	chembl:CHEMBL1702181	CHEMBL:CHEMBL1702181	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	TIZANIDINE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.052090944	DNDI1417181	chembl:CHEMBL1537417	CHEMBL:CHEMBL1537417	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	NECROSTATIN	iuphar.ligand:9750	NECROSTATIN-1	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-125734	chembl:CHEMBL586195	CHEMBL:CHEMBL586195	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	agonist	0.096167896	APIMOSTINEL	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
SIRT5	hgnc:14933	SIRT5	DTC	9/2/20	NULL	0.2187819634820604	GW7647	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	2-MERCAPTONICOTINIC ACID	chembl:CHEMBL1521174	2-MERCAPTONICOTINIC ACID	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.1912847768149162	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	BUTAMBEN	rxcui:19861	BUTAMBEN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	GNF-PF-159	chembl:CHEMBL599924	CHEMBL:CHEMBL599924	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DROSPIRENONE	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	SALICYLAMIDE	rxcui:9518	SALICYLAMIDE	TRUE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	DTC	9/2/20	NULL	4.039051633514961	ETHYL 2,4,6-TRIHYDROXYBENZOATE	chembl:CHEMBL2204435	CHEMBL:CHEMBL2204435	FALSE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.6250913242344582	RG3487	chembl:CHEMBL2151439	RG3487	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1112450661773188	CYSTAMINE DIHYDROCHLORIDE	ncit:C97356	CYSTAMINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	HYPOTAURINE	rxcui:2597523	HYPOTAURINE	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.094608417	HINOKITIOL	chembl:CHEMBL48310	HINOKITIOL	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.2734774543525755	QUINOLINIC ACID	drugbank:DB01796	QUINOLINIC ACID	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.049723174	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	PHENAMIL METHANESULFONATE	chembl:CHEMBL1256775	PHENAMIL METHANESULFONATE	FALSE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.5834185692854944	RG3487	chembl:CHEMBL2151439	RG3487	FALSE	FALSE	FALSE
RARG	hgnc:9866	RARG	DTC	9/2/20	NULL	0.3633748874442526	RO-137410	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.2500365296937833	QUINOLINIC ACID	drugbank:DB01796	QUINOLINIC ACID	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.027855529	NITROXOLINE	rxcui:31901	NITROXOLINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.018619742	CEFOTAXIME	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.072826174	ROSE BENGAL	rxcui:9471	ROSE BENGAL	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.096167896	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	IRIGINOL HEXAACEATATE	chembl:CHEMBL1440119	IRIGINOL HEXAACEATATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	NSC-668394	chembl:CHEMBL336095	CHEMBL:CHEMBL336095	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007699637	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.068369364	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	DNDI1417388	chembl:CHEMBL1528359	CHEMBL:CHEMBL1528359	FALSE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.6250913242344582	RG3487	chembl:CHEMBL2151439	RG3487	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.060984519	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	RESCINNAMINE	rxcui:9259	RESCINNAMINE	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.1121958787087489	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	chembl:CHEMBL1556914	METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	GNF-PF-1295	chembl:CHEMBL579837	CHEMBL:CHEMBL579837	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.055504938	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.5303805175322676	TCMDC-123591	chembl:CHEMBL588234	CHEMBL:CHEMBL588234	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.026927011	GW441756X	chembl:CHEMBL1516890	GW441756X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	NEFAZODONE HYDROCHLORIDE	rxcui:236082	NEFAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	blocker	0.3061671792168775	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	VANIPREVIR	ncit:C152828	VANIPREVIR	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.063415062	E-GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	PLICAMYCIN	rxcui:6995	PLICAMYCIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	PROCHLORAZ	chembl:CHEMBL522782	PROCHLORAZ	FALSE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	ChEMBL	33	agonist	0.3977853881492007	SIMPINICLINE	ncit:C179121	SIMPINICLINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	8,2'-DIMETHOXYFLAVONE	chembl:CHEMBL1516007	8,2'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	CID 727725	chembl:CHEMBL259422	CHEMBL:CHEMBL259422	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.3860858179095183	ISOQUINOLINE-1,3(2H,4H)-DIONE	chembl:CHEMBL1210769	CHEMBL:CHEMBL1210769	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	NIFLUMIC ACID	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	TCMDC-123748	chembl:CHEMBL530609	CHEMBL:CHEMBL530609	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	KAMEBANIN	chembl:CHEMBL472437	KAMEBANIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00575742	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124834	chembl:CHEMBL545880	CHEMBL:CHEMBL545880	FALSE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	DTC	9/2/20	NULL	0.9334697108567911	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.045461187	CGP-7930	iuphar.ligand:1079	CGP7930	FALSE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.182318303	GNF-PF-2272	chembl:CHEMBL601757	CHEMBL:CHEMBL601757	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.3535870116881784	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.036413087	NSC-66209	chembl:CHEMBL175266	CHEMBL:CHEMBL175266	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	GNF-PF-1654	chembl:CHEMBL602776	CHEMBL:CHEMBL602776	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.1187956362798518	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	GNF-PF-3464	chembl:CHEMBL602213	CHEMBL:CHEMBL602213	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	GNF-PF-3084	chembl:CHEMBL601135	CHEMBL:CHEMBL601135	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008432935	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
ADAM10	hgnc:188	ADAM10	DTC	9/2/20	NULL	0.4375639269641208	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	TCMDC-124307	chembl:CHEMBL546865	CHEMBL:CHEMBL546865	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	CYSTEINE METHYL-ESTER HCL	chembl:CHEMBL1426508	CHEMBL:CHEMBL1426508	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.019724895	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
CYTH2	hgnc:9502	CYTH2	DTC	9/2/20	NULL	1.419126249613364	CLOTRIMAZOLE	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1479089330582944	EVANS BLUE	rxcui:4191	EVANS BLUE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	NSC-720622	chembl:CHEMBL1287980	CHEMBL:CHEMBL1287980	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.093098708	TCMDC-124307	chembl:CHEMBL546865	CHEMBL:CHEMBL546865	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2561349816375342	APICIDIN	iuphar.ligand:7495	APICIDIN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.016764901	ASTERRIC ACID	chembl:CHEMBL469424	ASTERRIC ACID	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.023420014	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.023620185	SANGUINARINE SULFATE	chembl:CHEMBL1565133	SANGUINARINE SULFATE	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.2125816649218401	LITHOCHOLIC ACID	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
MMP14	hgnc:7160	MMP14	DTC	9/2/20	NULL	0.9376369863516875	CARMINIC ACID	rxcui:1368643	CARMINIC ACID	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	BITHIONOLOXIDE	ncit:C78040	BITHIONOLOXIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005412046	GW7074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.7395446652914718	CARBENICILLIN INDANYL	ncit:C76219	CARBENICILLIN INDANYL	FALSE	FALSE	FALSE
ME3	hgnc:6985	ME3	DTC	9/2/20	NULL	17.50255707856483	GLUTACONATE	chembl:CHEMBL557347	GLUTACONATE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	TETROQUINONE	chembl:CHEMBL1329029	TETROQUINONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	DNDI1417457	chembl:CHEMBL1530911	CHEMBL:CHEMBL1530911	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	TCMDC-124522	chembl:CHEMBL526776	CHEMBL:CHEMBL526776	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	DESOGESTREL	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.018430211	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.2536602475154323	GAMBOGIC ACID	chembl:CHEMBL555017	GAMBOGIC ACID	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.029783137	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.060492709	CEFAMANDOLE SODIUM	ncit:C47967	CEFAMANDOLE SODIUM	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	GUANABENZ ACETATE	rxcui:227225	GUANABENZ ACETATE	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.064824285	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.015443433	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.002674596	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.2386712328895204	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW301888X	chembl:CHEMBL531804	GW301888X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002421494	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.212581665	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.007623618	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	chembl:CHEMBL464433	4',7-DIMETHOXY-5-HYDROXYGENISTEIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.007110043	EBSELEN	ncit:C65503	EBSELEN	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.2206204673768676	GNF-PF-5029	chembl:CHEMBL1198140	CHEMBL:CHEMBL1198140	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01323278	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	DEQUALINIUM CHLORIDE	rxcui:3120	DEQUALINIUM CHLORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	OXITRIPTAN	rxcui:94	5-HYDROXYTRYPTOPHAN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.04339477	NEOSTIGMINE BROMIDE	rxcui:82055	NEOSTIGMINE BROMIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	METHAPYRILENE HYDROCHLORIDE	rxcui:235721	METHAPYRILENE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	CUCURBITACIN D	chembl:CHEMBL493646	CUCURBITACIN D	FALSE	FALSE	FALSE
HNRNPA1	hgnc:5031	HNRNPA1	DTC	9/2/20	NULL	3.000438356	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	2.838252499226729	CASOPITANT	ncit:C71635	CASOPITANT	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	BMS-777607	drugbank:DB12064	BMS-777607	FALSE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	GNF-PF-2260	chembl:CHEMBL601351	CHEMBL:CHEMBL601351	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	BENZOFURAN	drugbank:DB04179	BENZOFURAN	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.1100789753368857	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.065964411	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	GNF-PF-3084	chembl:CHEMBL601135	CHEMBL:CHEMBL601135	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	FLUAZINAM	chembl:CHEMBL1878267	FLUAZINAM	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.01090502	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
PRKAB1	hgnc:9378	PRKAB1	DTC	9/2/20	NULL	1.009762908	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.027811267	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	PEFLOXACINE MESYLATE	chembl:CHEMBL1428564	PEFLOXACIN MESYLATE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.027347745	N-DESMETHYLCLOZAPINE	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	ICI-164384	drugbank:DB03860	ICI-164384	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.010742159	RABEPRAZOLE SODIUM	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
GRIK3	hgnc:4581	GRIK3	ChEMBL	33	inhibitor	0.8334550989792778	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	3-METHOXYFLAVONOL	chembl:CHEMBL272005	CHEMBL:CHEMBL272005	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	BUTACAINE	rxcui:1829	BUTACAINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DITIOCARB SODIUM	ncit:C80963	DITIOCARB SODIUM	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.99446347	BETAXOLOL	rxcui:1520	BETAXOLOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	OLEOYLETHANOLAMIDE	iuphar.ligand:2661	N-OLEOYLETHANOLAMIDE	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.010332088	PHA-767491	drugbank:DB17043	PHA-767491	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004287741	HAEMATOXYLIN	chembl:CHEMBL1479103	HAEMATOXYLIN	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	PTEROSTILBENE	ncit:C153353	PTEROSTILBENE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007592202	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BATILOL	rxcui:1306190	BATILOL	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.013159817	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	BRONOPOL	rxcui:1114345	BRONOPOL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000171111	chembl:CHEMBL598279	CHEMBL:CHEMBL598279	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	agonist	0.040515178	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.052824619	BRIVANIB ALANINATE	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.089298761	BRIVANIB ALANINATE	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	2-(2'-METHOXYPHENYL)-1H-INDOLE	chembl:CHEMBL1449007	2-(2'-METHOXYPHENYL)-1H-INDOLE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	N-(4-CARBOXYMETHENE)PHENYLPYRROLE	chembl:CHEMBL258756	CHEMBL:CHEMBL258756	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.005294179	SURAMIN	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.021519537	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.035800685	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.025567767	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	4.773424657790408	AC-55541	iuphar.ligand:9456	AC-55541	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	RO-194603	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	DOCEBENONE	ncit:C76761	DOCEBENONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	GNF-PF-1295	chembl:CHEMBL579837	CHEMBL:CHEMBL579837	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	3-(PHENYLAMINO)PHENOL	chembl:CHEMBL1523215	CHEMBL:CHEMBL1523215	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	MICHLER'S KETONE	chembl:CHEMBL15137	MICHLER'S KETONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	N',N'-DIMETHYLARGININE HCL	chembl:CHEMBL1255836	CHEMBL:CHEMBL1255836	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	3-(PHENYLAMINO)PHENOL	chembl:CHEMBL1523215	CHEMBL:CHEMBL1523215	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1025540453822158	NSC-317605	chembl:CHEMBL1312050	CHEMBL:CHEMBL1312050	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.043902735	ZEARALENONE	chembl:CHEMBL454173	ZEARALENONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	PD-153035	chembl:CHEMBL29197	CHEMBL:CHEMBL29197	FALSE	FALSE	FALSE
PRDX5	hgnc:9355	PRDX5	DTC	9/2/20	NULL	26.25383561784724	2-(2-HYDROXYBENZYL)PHENOL	chembl:CHEMBL148831	CHEMBL:CHEMBL148831	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.5147810905460244	NSC-50690	chembl:CHEMBL1388703	CHEMBL:CHEMBL1388703	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	TCMDC-124176	chembl:CHEMBL588038	CHEMBL:CHEMBL588038	FALSE	FALSE	FALSE
TEK	hgnc:11724	TEK	DTC	9/2/20	NULL	0.9376369863516874	CETIRIZINE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.4102161815288632	CYCLIRAMINE MALEATE	ncit:C65355	CYCLIRAMINE MALEATE	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	2.282942227638891	AVOSENTAN	ncit:C79485	AVOSENTAN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	BIX-01294	iuphar.ligand:7014	BIX-01294	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	DNDI1417260	chembl:CHEMBL2094573	CHEMBL:CHEMBL2094573	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	TRIPROLIDINE	rxcui:10849	TRIPROLIDINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	DNDI1417260	chembl:CHEMBL2094573	CHEMBL:CHEMBL2094573	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	METHOXSALEN	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.1172046232939609	AMENTOFLAVONE	rxcui:2643210	AMENTOFLAVONE	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.01598407	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.2163777660811586	LUMATEPERONE	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	APTIGANEL HYDROCHLORIDE	ncit:C142929	APTIGANEL HYDROCHLORIDE	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	DTC	9/2/20	NULL	0.3454452054979901	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	2.917092846427472	OCRELIZUMAB	rxcui:1876366	OCRELIZUMAB	TRUE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.046881849	MYRICETIN	rxcui:1368374	MYRICETIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005130207	NSC-348401	chembl:CHEMBL515505	CHEMBL:CHEMBL515505	FALSE	FALSE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	11.66837138570988	DIETHYL-2-TRIDECYLIDENEMALONATE	chembl:CHEMBL1797709	CHEMBL:CHEMBL1797709	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006182465	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	SJ000072340	chembl:CHEMBL592813	CHEMBL:CHEMBL592813	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	3-METHOXYFLAVONOL	chembl:CHEMBL272005	CHEMBL:CHEMBL272005	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.055504938	GO-6976	drugbank:DB17029	GO-6976	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	2.187819634820604	INOTUZUMAB OZOGAMICIN	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.012794267	NSC-71033	chembl:CHEMBL116548	CHEMBL:CHEMBL116548	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.2263261691193728	DIMETHYLPHENYLPIPERAZINIUM IODIDE	chembl:CHEMBL47814	DIMETHYLPHENYLPIPERAZINIUM IODIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.014299475	Dronabinol	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.013021444	Pimozide	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.029515273	Protriptyline	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	FDA	10-Apr-24	NULL	0.1367387271762877	Prasugrel	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.9723642821424906	OTELIXIZUMAB	ncit:C95790	OTELIXIZUMAB	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	FDA	10-Apr-24	NULL	0.032899543	Phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.008681824	Phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
TTR	hgnc:12405	TTR	FDA	10-Apr-24	NULL	17.50255707856483	Tafamidis	rxcui:1545063	TAFAMIDIS	TRUE	FALSE	FALSE
RHD	hgnc:10009	RHD	ChEMBL	33	inhibitor	13.12691780892362	ROZROLIMUPAB	ncit:C152271	ROZROLIMUPAB	FALSE	FALSE	FALSE
F5	hgnc:3542	F5	FDA	10-Apr-24	NULL	0.1311052964686504	Rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.2263261691193728	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
NAGS	hgnc:17996	NAGS	FDA	10-Apr-24	NULL	26.25383561784724	Carglumic Acid	rxcui:401713	CARGLUMIC ACID	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.042174836	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.1172046232939609	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.088248187	PF-4691502	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.1442518440541057	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.1172046232939609	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.2083637747448194	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
ARAF	hgnc:646	ARAF	MyCancerGenome	20-Jun-17	inhibitor	0.1060761035064535	LGX818	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.038894571	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	MyCancerGenome	20-Jun-17	inhibitor	0.7778914257139926	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	MyCancerGenome	20-Jun-17	inhibitor	0.2187819634820604	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1232574442152452	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
MS4A1	hgnc:7315	MS4A1	MyCancerGenome	20-Jun-17	antibody	4.861821410712453	OFATUMUMAB	rxcui:712566	OFATUMUMAB	TRUE	TRUE	TRUE
IL6ST	hgnc:6021	IL6ST	ChEMBL	33	inhibitor	5.834185692854944	SATRALIZUMAB	rxcui:2391541	SATRALIZUMAB	TRUE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	MyCancerGenome	20-Jun-17	antibody	17.50255707856483	LBY135	chembl:CHEMBL2109247	LBY-135	FALSE	TRUE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	MyCancerGenome	20-Jun-17	antibody	29.17092846427472	LEXATUMUMAB	ncit:C64621	LEXATUMUMAB	FALSE	TRUE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	MyCancerGenome	20-Jun-17	antibody	5.834185692854944	CONATUMUMAB	ncit:C71015	CONATUMUMAB	FALSE	TRUE	TRUE
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.105015342	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1312691780892362	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.105015342	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
IL6R	hgnc:6019	IL6R	ChEMBL	33	inhibitor	5.385402178019948	SATRALIZUMAB	rxcui:2391541	SATRALIZUMAB	TRUE	FALSE	FALSE
PRRT2	hgnc:30500	PRRT2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	4.375639269641208	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.074850565	ERYTHROMYCIN	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1012684112549556	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.009899636	ZD1839	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.3443125982668492	NOVOBIOCIN	rxcui:7538	NOVOBIOCIN	FALSE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	NCI	14-Sep-17	NULL	0.027577558	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ARNT	hgnc:700	ARNT	NCI	14-Sep-17	NULL	0.1193356164447602	PROTEASOME INHIBITOR	ncit:C2160	PROTEASOME INHIBITOR	FALSE	FALSE	FALSE
ATP7B	hgnc:870	ATP7B	NCI	14-Sep-17	NULL	0.1988926940746004	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.077789143	INTERLEUKIN-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	NCI	14-Sep-17	NULL	0.2386712328895204	INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
CCL22	hgnc:10621	CCL22	NCI	14-Sep-17	NULL	17.50255707856483	SECONDARY LYMPHOID-TISSUE CHEMOKINE	ncit:C1792	RECOMBINANT HUMAN 6CKINE	FALSE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	inhibitor	3.281729452230906	CLENOLIXIMAB	ncit:C188527	CLENOLIXIMAB	FALSE	FALSE	FALSE
CD2	hgnc:1639	CD2	NCI	14-Sep-17	NULL	0.6482428547616605	SMS 201-995	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	3.500511415712966	IL-12 GENE	ncit:C2222	INTERLEUKIN-12 GENE	FALSE	FALSE	FALSE
CD2	hgnc:1639	CD2	NCI	14-Sep-17	NULL	0.7778914257139926	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	0.305277158	STEROID HORMONE	ncit:C1636	THERAPEUTIC STEROID HORMONE	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	1.363835616511545	AGM-1470	ncit:C1298	O-CHLOROACETYLCARBAMOYLFUMAGILLOL	FALSE	FALSE	FALSE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	0.6731752722524936	TOREMIFENE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.03849536	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
INHBA	hgnc:6066	INHBA	ChEMBL	33	inhibitor	8.751278539282415	SOTATERCEPT	ncit:C80038	SOTATERCEPT	FALSE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.130291988	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.012628108	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CHAT	hgnc:1912	CHAT	NCI	14-Sep-17	NULL	0.3535870116881784	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	0.729273212	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	1.166837138570989	TUMOR NECROSIS FACTOR	ncit:C1941	RECOMBINANT TUMOR NECROSIS FACTOR FAMILY PROTEIN	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1235474617310459	EGCG	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1400204566285186	BECLOMETHASONE DIPROPIONATE	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	ROQUINIMEX	ncit:C1519	ROQUINIMEX	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1400204566285186	MPA	iuphar.ligand:4595	MPA	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.2800409132570373	TGF-BETA 2	ncit:C1286	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA-2	FALSE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.092118721	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.1442518440541057	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
CTAG1B	hgnc:2491	CTAG1B	NCI	14-Sep-17	NULL	6.563458904461812	TUMOR ANTIGEN	ncit:C912	TUMOR ANTIGEN	FALSE	FALSE	FALSE
CTAG1B	hgnc:2491	CTAG1B	NCI	14-Sep-17	NULL	0.2344092465879218	FR901228	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	6.177373086552294	PLATELET FACTOR 4	ncit:C2251	IROPLACT	FALSE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	2.187819634820604	BB-94	ncit:C1529	BATIMASTAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.003849818	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.033529803	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.024674658	FR901228	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.007428929	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ETV6	hgnc:3495	ETV6	NCI	14-Sep-17	NULL	1.093909817410302	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
FCGR1A	hgnc:3613	FCGR1A	ChEMBL	33	modulator	5.250767123569449	MDX-210	drugbank:DB17250	MDX-210	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.069638821	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
SLC1A1	hgnc:10939	SLC1A1	NCI	14-Sep-17	NULL	0.4018444227221517	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1248696105486195	BUTYRATE	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
TAC3	hgnc:11521	TAC3	NCI	14-Sep-17	NULL	3.182283105193606	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	1.400204566285186	INCOMPLETE FREUNDS ADJUVANT	ncit:C1573	INCOMPLETE FREUND'S ADJUVANT	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.2419708351875322	ADENOVIRUS VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	1.779921058837101	IUDR	rxcui:5653	IDOXURIDINE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.080656945	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.057416808	RETINOID	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.045639002	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.6731752722524935	LEVAMISOLE	rxcui:6371	LEVAMISOLE	TRUE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.2778183663264259	DHEA	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
THRSP	hgnc:11800	THRSP	NCI	14-Sep-17	NULL	0.7955707762984016	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
KIR2DL3	hgnc:6331	KIR2DL3	ChEMBL	33	inhibitor	3.281729452230906	LIRILUMAB	ncit:C103820	LIRILUMAB	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.5645986154375752	PCB	rxcui:66925	PROCARBAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.011591097	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.016558711	INTERFERON ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	0.093763699	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.046446414	5-FU	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.055681518	NDGA	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	1.750255707856483	ACTH	iuphar.ligand:1331	ACTH	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.071148606	L-DOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
UCP2	hgnc:12518	UCP2	NCI	14-Sep-17	NULL	0.7955707762984016	TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.004743883	17 BETA-ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.007962947	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	NCI	14-Sep-17	NULL	0.084553416	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
ICAM1	hgnc:5344	ICAM1	ChEMBL	33	inhibitor	13.12691780892362	BI-505	chembl:CHEMBL2109482	BI-505	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.1000146118775133	paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	0.068458502	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.025588534	talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
GAA	hgnc:4065	GAA	PharmGKB	4/5/24	NULL	0.2430910705356226	alglucosidase alfa	rxcui:2475360	LYSOSOMAL ALPHA-GLUCOSIDASE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.064347636	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
CYB5R4	hgnc:20147	CYB5R4	PharmGKB	4/5/24	NULL	0.9546849315580819	isosorbide dinitrate	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.093763699	GLAFENINE	ncit:C72119	GLAFENINE	TRUE	FALSE	FALSE
B4GALT2	hgnc:925	B4GALT2	PharmGKB	4/5/24	NULL	0.5585922471882393	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.28382525	NIALAMIDE	rxcui:7394	NIALAMIDE	TRUE	FALSE	FALSE
CYB5R2	hgnc:24376	CYB5R2	PharmGKB	4/5/24	NULL	0.9546849315580819	isosorbide dinitrate	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.02550154	dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.063568609	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	2.100306849	ombitasvir / paritaprevir / ritonavir	wikidata:Q19858657	OMBITASVIR/PARITAPREVIR/RITONAVIR	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.041150213	dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	PharmGKB	4/5/24	NULL	0.03233231	dopamine	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.1341192113299987	pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.1411496538593938	lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	PharmGKB	4/5/24	NULL	0.1110098757625676	lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1161674142382621	cefradine	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1548898856510162	cefadroxil	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.007875757	progesterone	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.4102161815288632	cotinine	ncit:C70941	COTININE	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.013666755	vinblastine	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.021121348	rosiglitazone	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
PRF1	hgnc:9360	PRF1	PharmGKB	4/5/24	NULL	4.375639269641208	emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
JMJD8	hgnc:14148	JMJD8	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.058733413	sulfadiazine	rxcui:10171	SULFADIAZINE	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.6731752722524935	PHENOXYPROPAZINE	drugbank:DB09251	PHENOXYPROPAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.069043618	fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.054398002	propafenone	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.002642294	morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.005064397	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.020433651	fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.4366542306502661	fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	PharmGKB	4/5/24	NULL	0.4293851619741372	atomoxetine	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
COL1A1	hgnc:2197	COL1A1	PharmGKB	4/5/24	NULL	1.000146118775133	somatropin recombinant	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	PharmGKB	4/5/24	NULL	0.039553801	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CXCL12	hgnc:10672	CXCL12	PharmGKB	4/5/24	NULL	0.2917092846427472	rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	1.406455479527531	o-desmethyltramadol	chembl:CHEMBL4650315	DESMETRAMADOL	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.011218389	caffeine	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
GRAMD1B	hgnc:29214	GRAMD1B	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
BCHE	hgnc:983	BCHE	ChEMBL	33	inhibitor	0.6563458904461812	PROPANIDID	rxcui:8758	PROPANIDID	TRUE	FALSE	FALSE
SLC17A3	hgnc:10931	SLC17A3	PharmGKB	4/5/24	NULL	5.834185692854945	bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
SCARB1	hgnc:1664	SCARB1	PharmGKB	4/5/24	NULL	4.039051633514962	fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
SEPTIN3	hgnc:10750	SEPTIN3	PharmGKB	4/5/24	NULL	0.8751278539282416	tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
OR52J2P	hgnc:14797	OR52J2P	PharmGKB	4/5/24	NULL	2.500365296937833	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	REMOXIPRIDE HYDROCHLORIDE	rxcui:235832	REMOXIPRIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.016434326	amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.8334550989792776	lithium	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.039068208	nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
RRP7A	hgnc:24286	RRP7A	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
ZDHHC7	hgnc:18459	ZDHHC7	PharmGKB	4/5/24	NULL	2.282942227638891	methylphenidate	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT2B17	hgnc:12547	UGT2B17	PharmGKB	4/5/24	NULL	0.7721716358190368	diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.056888051	lenalidomide	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	1.944728564284981	benazepril	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.083016081	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	PharmGKB	4/5/24	NULL	0.7425327245451747	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.7095631248066824	PHENOXYPROPAZINE	drugbank:DB09251	PHENOXYPROPAZINE	TRUE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	PharmGKB	4/5/24	NULL	0.2117244807890907	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	0.1363835616511545	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.729273212	sulfamethazine	rxcui:10178	SULFAMETHAZINE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	5.966780822238011	elexacaftor	rxcui:2256951	ELEXACAFTOR	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.036025846	atorvastatin	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.6945459158160648	NIMOTUZUMAB	ncit:C2733	NIMOTUZUMAB	FALSE	TRUE	TRUE
CACNA1G	hgnc:1394	CACNA1G	PharmGKB	4/5/24	NULL	0.065308049	celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PCSK9	hgnc:20001	PCSK9	PharmGKB	4/5/24	NULL	6.058577450272442	evolocumab	rxcui:1665684	EVOLOCUMAB	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.325124899	ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.012822386	tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.068458502	etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
TAPBP	hgnc:11566	TAPBP	PharmGKB	4/5/24	NULL	0.7447896629176524	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	PharmGKB	4/5/24	NULL	0.004434582	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.2333674277141977	imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
FTO	hgnc:24678	FTO	PharmGKB	4/5/24	NULL	0.4375639269641208	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.055563673	mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
YBX1	hgnc:8014	YBX1	PharmGKB	4/5/24	NULL	8.751278539282415	abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
KRTAP10-4	hgnc:20521	KRTAP10-4	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
HLA-E	hgnc:4962	HLA-E	PharmGKB	4/5/24	NULL	0.5645986154375753	infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
PTGDR	hgnc:9591	PTGDR	PharmGKB	4/5/24	NULL	2.917092846427472	laropiprant	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.05413162	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.1902451856365742	ISOXSUPRINE HYDROCHLORIDE	rxcui:82033	ISOXSUPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	PharmGKB	4/5/24	NULL	0.098421127	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	PharmGKB	4/5/24	NULL	0.022554842	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
HNMT	hgnc:5028	HNMT	PharmGKB	4/5/24	NULL	0.1546617709446082	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	PharmGKB	4/5/24	NULL	0.063684259	clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.055859225	azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.3182283105193606	nevirapine	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
GALNT14	hgnc:22946	GALNT14	PharmGKB	4/5/24	NULL	0.3309307010653015	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP11B2	hgnc:2592	CYP11B2	PharmGKB	4/5/24	NULL	1.093909817410302	spironolactone	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	inhibitor	0.3547815624033412	ALVERINE	rxcui:17627	ALVERINE	TRUE	FALSE	FALSE
PPOX	hgnc:9280	PPOX	PharmGKB	4/5/24	NULL	17.50255707856483	givosiran	rxcui:2265712	GIVOSIRAN	TRUE	FALSE	FALSE
SLC22A16	hgnc:20302	SLC22A16	PharmGKB	4/5/24	NULL	1.323722804261206	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	PharmGKB	4/5/24	NULL	0.012606884	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	DEXTROMORAMIDE	rxcui:3290	DEXTROMORAMIDE	TRUE	FALSE	FALSE
PPP2R5D	hgnc:9312	PPP2R5D	PharmGKB	4/5/24	NULL	0.2941606231691568	fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.6509215442441467	pamidronate	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
TSPEAR	hgnc:1268	TSPEAR	PharmGKB	4/5/24	NULL	0.3723948314588262	aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1750255707856483	furazolidone	rxcui:4601	FURAZOLIDONE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.078136416	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.052507671	flutamide	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
NR1H3	hgnc:7966	NR1H3	PharmGKB	4/5/24	NULL	0.5556367326528519	laropiprant	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1215455352678113	COPANLISIB HYDROCHLORIDE	ncit:C138994	COPANLISIB HYDROCHLORIDE	TRUE	FALSE	FALSE
RFK	hgnc:30324	RFK	PharmGKB	4/5/24	NULL	3.000438356	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	1.154014752432846	glipizide	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.4167275494896389	clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
PTPRD	hgnc:9668	PTPRD	PharmGKB	4/5/24	NULL	2.625383561784725	trandolapril	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
NRP1	hgnc:8004	NRP1	ChEMBL	33	inhibitor	17.50255707856483	VESENCUMAB	ncit:C91728	VESENCUMAB	FALSE	FALSE	FALSE
IDO1	hgnc:6059	IDO1	PharmGKB	4/5/24	NULL	0.258658479	interferon alfa-2a, recombinant	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.9131768910555565	trandolapril	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	0.3621218705909965	interferon alfa-2a, recombinant	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	0.1620607136904151	buprenorphine	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
GLDC	hgnc:4313	GLDC	PharmGKB	4/5/24	NULL	1.000146118775133	escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.072927321	hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
ALDH3A1	hgnc:405	ALDH3A1	PharmGKB	4/5/24	NULL	0.300043836	thiotepa	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
UNIPROT:Q01668	hgnc:1391	CACNA1D	TdgClinicalTrial	Jan-14	NULL	0.3488881809680697	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
UNIPROT:Q9NPF7	hgnc:15488	IL23A	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	CNTO 1275	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
NGF	hgnc:7808	NGF	ChEMBL	33	inhibitor	7.501095891	PG-110	chembl:CHEMBL2109526	PG-110	FALSE	FALSE	FALSE
UNIPROT:P06241	hgnc:4037	FYN	TdgClinicalTrial	Jan-14	NULL	0.075768645	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:Q99665	hgnc:5972	IL12RB2	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
UNIPROT:P51692	hgnc:11367	STAT5B	TdgClinicalTrial	Jan-14	NULL	0.2727671233023091	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1293292394967845	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.069638821	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P20138	hgnc:1659	CD33	TdgClinicalTrial	Jan-14	NULL	2.423430980108977	GEMTUZUMAB OZOGAMICIN	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.069454592	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	modulator	0.525076712	FBT-A05	chembl:CHEMBL2109351	FBT-A05	FALSE	FALSE	FALSE
UNIPROT:P07814	hgnc:3418	EPRS1	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	HALOFUGINONE	ncit:C1120	HALOFUGINONE	FALSE	FALSE	FALSE
UNIPROT:P07333	hgnc:2433	CSF1R	TdgClinicalTrial	Jan-14	NULL	0.089103927	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:Q08345	hgnc:2730	DDR1	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	NEMIFITIDE	ncit:C90713	NEMIFITIDE	FALSE	FALSE	FALSE
UNIPROT:P05362	hgnc:5344	ICAM1	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	ALICAFORSEN	ncit:C169771	ALICAFORSEN	FALSE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.8751278539282416	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	3.842024724563012	MDX-1342	chembl:CHEMBL2109337	MDX-1342	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.5645986154375752	ISIS-104838	drugbank:DB16201	ISIS 104838	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.075010959	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.076840494	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.07160137	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	KARENITECIN	chembl:CHEMBL1743260	KARENITECIN	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.065125794	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.3006164383722967	LOTEPREDNOL ETABONATE	rxcui:237027	LOTEPREDNOL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.1166837138570989	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.1154014752432846	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.085239726	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	CHORIOGONADOTROPIN ALFA	rxcui:283550	CHORIOGONADOTROPIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.2027323213733378	DIPHENIDOL	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	1.186614039224734	PERINDOPRIL	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	PROGABIDE	rxcui:34568	PROGABIDE	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1962903597596056	QUINESTROL	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.021370644	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TEND	1-Aug-11	NULL	1.555782851427985	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TEND	1-Aug-11	NULL	0.3125456621172291	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:P26358	hgnc:2976	DNMT1	TEND	1-Aug-11	NULL	0.1790034246671403	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.091583148	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.100976291	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.007596596	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.032173818	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.096050618	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.034590034	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.1022876712383659	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1962903597596056	QUINESTROL	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	1.071585127259071	ROCURONIUM	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
UNIPROT:P30988	hgnc:1440	CALCR	TEND	1-Aug-11	NULL	13.12691780892362	SALMON CALCITONIN	rxcui:36118	SALMON CALCITONIN	TRUE	FALSE	FALSE
UNIPROT:P62942	hgnc:3711	FKBP1A	TEND	1-Aug-11	NULL	0.5373592085524291	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	1.071585127259071	MRA 003 US	chembl:CHEMBL2109615	MRA 003 US	FALSE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TEND	1-Aug-11	NULL	0.9334697108567911	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.2408608772279564	SUFENTANIL	rxcui:56795	SUFENTANIL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.055504938	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TEND	1-Aug-11	NULL	0.076934317	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.087318744	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TEND	1-Aug-11	NULL	0.8334550989792776	TAMIBAROTENE	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.1884246575443582	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.1591141552596803	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.085239726	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.2864054794674245	TENOXICAM	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
UNIPROT:O75762	hgnc:497	TRPA1	TEND	1-Aug-11	NULL	4.375639269641208	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
UNIPROT:P47901	hgnc:896	AVPR1B	TEND	1-Aug-11	NULL	3.750547945	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	1.250182648468916	TOLAZAMIDE	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	4.375639269641208	SAR-566658	chembl:CHEMBL2109635	SAR-566658	FALSE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TEND	1-Aug-11	NULL	0.1591141552596803	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.05073205	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.048260727	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.040703621	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.055504938	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	1.250182648468916	TORASEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.061628722	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
UNIPROT:P63027	hgnc:12643	VAMP2	TEND	1-Aug-11	NULL	17.50255707856483	BOTULINUM TOXIN TYPE B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
UNIPROT:O43497	hgnc:1394	CACNA1G	TEND	1-Aug-11	NULL	2.187819634820604	TRIMETHADIONE	rxcui:10827	TRIMETHADIONE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.077827576	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1136529680426288	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TEND	1-Aug-11	NULL	0.8204323630577265	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.1025540453822158	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.056826484	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.2302968036653267	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TEND	1-Aug-11	NULL	1.887530665335423	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	2.100306849	ANAVEX 2-73	ncit:C171846	BLARCAMESINE	FALSE	FALSE	FALSE
STEROL O-ACYLTRANSFERASE	hgnc:11177	SOAT1	TTD	2020.06.01	NULL	4.773424657790408	ATR-101	chembl:CHEMBL542103	NEVANIMIBE HYDROCHLORIDE	FALSE	FALSE	FALSE
CD37	hgnc:1666	CD37	ChEMBL	33	binder	35.00511415712966	NARATUXIMAB EMTANSINE	ncit:C100101	NARATUXIMAB EMTANSINE	FALSE	FALSE	FALSE
CERAMIDE GLUCOSYLTRANSFERASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	5.250767123569449	GZ402671	ncit:C152852	VENGLUSTAT	FALSE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 1	hgnc:6877	MAPK3	TTD	2020.06.01	NULL	0.2972132334095915	BVD-523	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	3.500511415712966	Zarnestra	hemonc:496	TIPIFARNIB	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	1.944728564284981	BMS-986104	drugbank:DB15214	BMS-986104	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.1143957978991165	Masitinib	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.062509132	ABBV-399	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	5.250767123569449	JNJ-42165279	drugbank:DB15173	JNJ-42165279	FALSE	FALSE	FALSE
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	1.591141552596802	MIN-202	iuphar.ligand:9308	SELTOREXANT	FALSE	FALSE	FALSE
FILAMIN A	hgnc:3754	FLNA	TTD	2020.06.01	NULL	26.25383561784724	PTI-125	chembl:CHEMBL4650230	SIMUFILAM	FALSE	FALSE	FALSE
MSTN	hgnc:4223	MSTN	ChEMBL	33	inhibitor	2.187819634820604	DOMAGROZUMAB	ncit:C166800	DOMAGROZUMAB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.2465148884304905	Tivozanib	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
TRAIL RECEPTOR 2	hgnc:11905	TNFRSF10B	TTD	2020.06.01	NULL	29.17092846427472	Lexatumumab	ncit:C64621	LEXATUMUMAB	FALSE	TRUE	TRUE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.3938075342677087	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	3.804903712731485	Sivelestat	ncit:C66539	SIVELESTAT	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.030746697	Apomorphine	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NIEMANN-PICK C1-LIKE PROTEIN 1	hgnc:7898	NPC1L1	TTD	2020.06.01	NULL	26.25383561784724	Ezetimibe	rxcui:341248	EZETIMIBE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.044611445	Diethylstilbestrol	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
SLC44A4	hgnc:13941	SLC44A4	ChEMBL	33	binder	6.563458904461812	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.075496292	Desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR-GAMMA	hgnc:10479	RXRG	TTD	2020.06.01	NULL	0.1767935058440892	Vitamin A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
NEUROPEPTIDE RECEPTOR	hgnc:7954	NPTXR	TTD	2020.06.01	NULL	17.50255707856483	NNZ-2566	rxcui:2632852	TROFINETIDE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.015407181	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.2983390411119005	Levomilnacipran	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.182318303	ASUNAPREVIR	rxcui:1652103	ASUNAPREVIR	FALSE	FALSE	FALSE
MYRISTOYLATED ALANINE-RICH C-KINASE SUBSTRATE	hgnc:6759	MARCKS	TTD	2020.06.01	NULL	105.0153424713889	BIO-11006	drugbank:DB14886	BIO-11006	FALSE	FALSE	FALSE
AGGRECANASE	hgnc:221	ADAMTS5	TTD	2020.06.01	NULL	17.50255707856483	AGG-523	drugbank:DB15460	AGG-523	FALSE	FALSE	FALSE
OSTEOCLAST DIFFERENTIATION FACTOR	hgnc:11926	TNFSF11	TTD	2020.06.01	NULL	43.75639269641208	Denosumab	rxcui:993449	DENOSUMAB	TRUE	FALSE	TRUE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	1.721562991334245	Ulipristal	rxcui:1005920	ULIPRISTAL ACETATE	TRUE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	agonist	2.625383561784724	TELRATOLIMOD	ncit:C124653	TELRATOLIMOD	FALSE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE	hgnc:1189	AHSA1	TTD	2020.06.01	NULL	0.364636606	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	2.282942227638891	AVL-3288	drugbank:DB18707	AVL-3288	FALSE	FALSE	FALSE
FAST SKELETAL MUSCLE TROPONIN COMPLEX	hgnc:11944	TNNC2	TTD	2020.06.01	NULL	11.66837138570988	CK-2127107	ncit:C166781	RELDESEMTIV	FALSE	FALSE	FALSE
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	3.281729452230906	MK-0731	drugbank:DB08037	MK-0731	FALSE	FALSE	FALSE
BROMODOMAIN TESTIS-SPECIFIC PROTEIN	hgnc:1105	BRDT	TTD	2020.06.01	NULL	0.7501095890813501	(+)-JQ1	iuphar.ligand:7511	(+)-JQ1	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.3697723326457359	Elpamotide	ncit:C74090	ELPAMOTIDE	FALSE	FALSE	FALSE
TGF-BETA RECEPTOR TYPE I	hgnc:11772	TGFBR1	TTD	2020.06.01	NULL	3.750547945	LY-2382770	chembl:CHEMBL2109585	LY-2382770	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.7160136986685613	Tiaprofenic acid	rxcui:38253	TIAPROFENIC ACID	FALSE	FALSE	FALSE
PROTO-ONCOGENE MAS	hgnc:6899	MAS1	TTD	2020.06.01	NULL	17.50255707856483	DSC-127	iuphar.ligand:8300	ACLERASTIDE	FALSE	FALSE	FALSE
HEPCIDIN	hgnc:15598	HAMP	TTD	2020.06.01	NULL	26.25383561784724	NOX-H94	ncit:C103195	LEXAPTEPID PEGOL	FALSE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	3.281729452230906	KAI-4169	rxcui:1876119	ETELCALCETIDE	TRUE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE	hgnc:1189	AHSA1	TTD	2020.06.01	NULL	1.458546423213736	BMS-582949	drugbank:DB12696	BMS-582949	FALSE	FALSE	FALSE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	5.834185692854944	LAS-101057	chembl:CHEMBL1672627	LAS101057	FALSE	FALSE	FALSE
SERINE/THREONINE PP2A-ALPHA	hgnc:9299	PPP2CA	TTD	2020.06.01	NULL	21.00306849	LB-100	drugbank:DB15412	LB-100	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	2.100306849	DP-b99	drugbank:DB05820	DP-B99	FALSE	FALSE	FALSE
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	3.889457128569962	VS-4718	drugbank:DB15273	VS-4718	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 1	hgnc:1602	CCR1	TTD	2020.06.01	NULL	11.66837138570988	BMS-817399	drugbank:DB14941	BMS-817399	FALSE	FALSE	FALSE
LEUCINE-RICH REPEAT NEURONAL PROTEIN 1	hgnc:21205	LINGO1	TTD	2020.06.01	NULL	13.12691780892362	BIIB-033	iuphar.ligand:8923	OPICINUMAB	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	0.789589041	RAMATROBAN	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
INTERFERON ALPHA/BETA RECEPTOR 1	hgnc:5432	IFNAR1	TTD	2020.06.01	NULL	1.458546423213736	MEDI-546	iuphar.ligand:8258	ANIFROLUMAB	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.1131630845596864	Nalidixic Acid	rxcui:7240	NALIDIXIC ACID	TRUE	FALSE	FALSE
INTERLEUKIN 17 RECEPTOR	hgnc:5985	IL17RA	TTD	2020.06.01	NULL	35.00511415712966	Brodalumab	rxcui:1872251	BRODALUMAB	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA 3	hgnc:4573	GRIA3	TTD	2020.06.01	NULL	0.9376369863516875	E-2007	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA 2	hgnc:4572	GRIA2	TTD	2020.06.01	NULL	1.193356164447602	E-2007	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA 1	hgnc:4571	GRIA1	TTD	2020.06.01	NULL	1.270346884734544	E-2007	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1B	hgnc:278	ADRA1B	TTD	2020.06.01	NULL	0.4565884455277782	Propericiazine	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	Ramosetron	ncit:C61921	RAMOSETRON	FALSE	FALSE	FALSE
KIF5B	hgnc:6324	KIF5B	ChEMBL	33	inhibitor	3.750547945406749	PRALSETINIB	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	1.795134059339982	Isocarboxazid	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.1346350544504987	MEDETOMIDINE	rxcui:52016	MEDETOMIDINE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.13086024	Amoxapine	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP1	hgnc:9593	PTGER1	TTD	2020.06.01	NULL	0.2344092465879218	PGF2alpha	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.1182605208011137	Urapidil	rxcui:39230	URAPIDIL	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	2.019525817	AZD3293	chembl:CHEMBL3989948	LANABECESTAT	FALSE	FALSE	FALSE
TUMOR SUSCEPTIBILITY GENE PROTEIN 101	hgnc:15971	TSG101	TTD	2020.06.01	NULL	8.078103267029922	FGI-101-1A6	chembl:CHEMBL2109593	FGI-101-1A6	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	CART-19 cells	ncit:C101258	CD19CAR-CD3ZETA-4-1BB-EXPRESSING ALLOGENEIC T-LYMPHOCYTE CELLS	FALSE	FALSE	FALSE
NEUROTROPHIC TYROSINE KINASE ROR1	hgnc:10256	ROR1	TTD	2020.06.01	NULL	26.25383561784724	ROR1 CAR-specific Autologous T-Lymphocytes	ncit:C117237	ROR1 CAR-SPECIFIC AUTOLOGOUS T-LYMPHOCYTES	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.034819411	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.020575106	IUPHAR.LIGAND:85	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.014601688	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.006521882	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.039538909	IUPHAR.LIGAND:37	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.3163112725041837	IUPHAR.LIGAND:126	iuphar.ligand:126	(+)-WAY 100135	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:123	iuphar.ligand:123	LYSERGOL	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.028413242	IUPHAR.LIGAND:85	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.027177884	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.085937269	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:185	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:212	rxcui:10510	THIOTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:188	iuphar.ligand:188	RS-127445	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.078958904	IUPHAR.LIGAND:192	iuphar.ligand:192	SB 228357	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.024030971	IUPHAR.LIGAND:88	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.01782943	IUPHAR.LIGAND:35	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.020320306	IUPHAR.LIGAND:34	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.077217164	IUPHAR.LIGAND:7241	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.8899605294185507	IUPHAR.LIGAND:8428	iuphar.ligand:8428	EMD-386088	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.070860555	IUPHAR.LIGAND:4	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	modulator	0.3070624048871023	IUPHAR.LIGAND:284	iuphar.ligand:284	OLEAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2435	hgnc:3833	FRA10E	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10150	iuphar.ligand:10150	K-604	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:6600	iuphar.ligand:6600	BW284C51	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:8181	iuphar.ligand:8181	COMPOUND 1 [PMID: 20005102]	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:8181	iuphar.ligand:8181	COMPOUND 1 [PMID: 20005102]	FALSE	FALSE	FALSE
PTGER2	hgnc:9594	PTGER2	ChEMBL	33	agonist	3.281729452230906	OMIDENEPAG ISOPROPYL	rxcui:2612690	OMIDENEPAG ISOPROPYL	TRUE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.094099769	IUPHAR.LIGAND:7397	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:497	iuphar.ligand:497	RO-70-0004	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.099071078	IUPHAR.LIGAND:53	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.076208521	IUPHAR.LIGAND:7302	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:599	iuphar.ligand:599	[PYR1]APELIN-13	FALSE	FALSE	FALSE
NCBIGENE:690	hgnc:1126	BTF3P11	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:10189	iuphar.ligand:10189	AUDIEN	FALSE	FALSE	FALSE
CCDC6	hgnc:18782	CCDC6	ChEMBL	33	inhibitor	3.750547945406749	PRALSETINIB	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:6187	iuphar.ligand:6187	E339-3D6	FALSE	FALSE	FALSE
NCBIGENE:690	hgnc:1126	BTF3P11	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10188	iuphar.ligand:10188	AUPHEN	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:4116	iuphar.ligand:4116	A-317567	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.5527123287967842	IUPHAR.LIGAND:2525	iuphar.ligand:2525	PB2+	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:379	iuphar.ligand:374	CCPA	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	0.280789686	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:861	iuphar.ligand:861	CCK-4	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:765	iuphar.ligand:765	[125I]CCL7 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:806	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	inhibitor	1.193356164447602	PECAVAPTAN	ncit:C166718	PECAVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:2764	hgnc:4373	GMFB	GuideToPharmacology	2024.1	antibody	1.312691780892362	IUPHAR.LIGAND:7384	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
NCBIGENE:65	ncbigene:65	ACTBP5	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:813	iuphar.ligand:813	ZK 756326	FALSE	FALSE	FALSE
PSMD8	hgnc:9566	PSMD8	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:12298	iuphar.ligand:12298	MOSUNETUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2766	hgnc:4376	GMPR	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:8719	iuphar.ligand:8719	ISATUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:8268	iuphar.ligand:8268	VELTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:13021	iuphar.ligand:13021	GOLCADOMIDE	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:7713	iuphar.ligand:7713	AZD7762	FALSE	FALSE	TRUE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	1.109316997937207	DIFELIKEFALIN	rxcui:2569089	DIFELIKEFALIN	TRUE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:6382	ncit:C66077	MELAGATRAN	FALSE	FALSE	FALSE
NCBIGENE:396	hgnc:678	ARHGDIA	GuideToPharmacology	2024.1	blocker	8.751278539282415	IUPHAR.LIGAND:2349	iuphar.ligand:2349	L-(CIS)-DILTIAZEM	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.1238388472539964	IUPHAR.LIGAND:5685	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.018012923	IUPHAR.LIGAND:5664	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:9383	iuphar.ligand:9383	OSI-930	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:11510	iuphar.ligand:11510	M4205	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.008643238	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:2334	hgnc:3776	AFF2	GuideToPharmacology	2024.1	inhibitor	4.773424657790409	IUPHAR.LIGAND:4262	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:607	hgnc:1008	BCL9	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:2758	iuphar.ligand:2758	CITCO	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.0230499	IUPHAR.LIGAND:2892	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:2897	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
RPS19	hgnc:10402	RPS19	ChEMBL	33	inhibitor	0.049864835	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:915	iuphar.ligand:915	[125I]CRF (OVINE)	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:918	iuphar.ligand:918	SAUVAGINE	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:916	iuphar.ligand:916	[125I]SAUVAGINE (FROG)	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:10335	iuphar.ligand:10335	ASTRESSIN 2B	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:925	iuphar.ligand:925	ASTRESSIN	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:759	iuphar.ligand:759	CCL7	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:842	iuphar.ligand:842	HYPOGLAUCIN A	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:848	iuphar.ligand:848	CXCL12-(1-9) DIMER	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5938	iuphar.ligand:5938	BOHEMINE	FALSE	FALSE	FALSE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9386	iuphar.ligand:9386	BMS-536924	FALSE	FALSE	TRUE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:2568	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3414	iuphar.ligand:3358	ICI198615	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:3327	ncit:C76576	SULUKAST	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9860	iuphar.ligand:9860	VIDOFLUDIMUS	FALSE	FALSE	FALSE
RPS15	hgnc:10388	RPS15	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:10658	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:1889	iuphar.ligand:1889	ZK110841	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:1876	iuphar.ligand:1876	&DELTA;12-PGJ2	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.013879903	IUPHAR.LIGAND:38	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:7670	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.025929714	IUPHAR.LIGAND:33	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
RPS6	hgnc:10429	RPS6	ChEMBL	33	inhibitor	0.108040476	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:2624	hgnc:4171	GATA2	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:6831	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
NCBIGENE:1455	hgnc:2455	CSNK1G2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9564	iuphar.ligand:9564	3 ALPHA-AMINOCHOLESTANE	FALSE	FALSE	FALSE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	0.2430910705356227	IUPHAR.LIGAND:7397	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492008	IUPHAR.LIGAND:7741	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:7423	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	agonist	0.082559232	IUPHAR.LIGAND:5012	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.037721028	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.3088686543276147	IUPHAR.LIGAND:12462	iuphar.ligand:12462	EPICATECHIN GALLATE	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.026626608	IUPHAR.LIGAND:2826	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
RPS2	hgnc:10404	RPS2	ChEMBL	33	inhibitor	0.108040476	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:661	hgnc:1080	POLR3D	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10362	iuphar.ligand:10362	ABSCISIC ACID	FALSE	FALSE	FALSE
NCBIGENE:664	hgnc:1084	BNIP3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12430	iuphar.ligand:12430	S7958	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:11878	drugbank:DB16756	IVARMACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:9991	rxcui:2591476	ABROCITINIB	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10147	iuphar.ligand:10147	JAK INHIBITOR 20A	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10148	iuphar.ligand:10148	JAK INHIBITOR 17B	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:11881	iuphar.ligand:11881	POVORCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.09869863	IUPHAR.LIGAND:11887	iuphar.ligand:11887	TINENGOTINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:10147	iuphar.ligand:10147	JAK INHIBITOR 20A	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:11883	iuphar.ligand:11883	SAFIMALTIB	FALSE	FALSE	FALSE
RPS3	hgnc:10420	RPS3	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:12384	iuphar.ligand:12384	ROVADICITINIB	FALSE	FALSE	FALSE
NCBIGENE:2865	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8489	iuphar.ligand:8489	EXAMPLE 131 [WO2009133348]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:9294	iuphar.ligand:9294	BU08028	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:9697	ncit:C152385	SOLCITINIB	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:1641	iuphar.ligand:1641	NALTRINDOLE	FALSE	FALSE	FALSE
F2R	hgnc:3537	F2R	ChEMBL	33	inhibitor	2.019525817	PZ-128	drugbank:DB11839	PZ-128	FALSE	FALSE	FALSE
NCBIGENE:968	hgnc:1693	CD68	GuideToPharmacology	2024.1	inhibitor	0.9723642821424908	IUPHAR.LIGAND:4839	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.041508041	IUPHAR.LIGAND:9921	iuphar.ligand:9921	TAFETINIB	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.012208247	IUPHAR.LIGAND:5056	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
NCBIGENE:521	hgnc:846	ATP5ME	GuideToPharmacology	2024.1	activator	1.071585127259071	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	2.625383561784724	IUPHAR.LIGAND:9312	iuphar.ligand:9312	SKA-20	FALSE	FALSE	FALSE
RPS18	hgnc:10401	RPS18	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2320	iuphar.ligand:2320	UCL1684	FALSE	FALSE	FALSE
NCBIGENE:429	hgnc:738	ASCL1	GuideToPharmacology	2024.1	blocker	13.12691780892362	IUPHAR.LIGAND:2383	iuphar.ligand:2383	TERTIAPIN-Q	FALSE	FALSE	FALSE
NCBIGENE:431	ncbigene:431	ASD1	GuideToPharmacology	2024.1	inhibitor	4.039051633514962	IUPHAR.LIGAND:708	iuphar.ligand:708	MG2+	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	2.500365296937833	IUPHAR.LIGAND:8492	iuphar.ligand:8492	SKA-121	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	TORIPALIMAB	rxcui:2669406	TORIPALIMAB	TRUE	FALSE	FALSE
NCBIGENE:442	hgnc:755	ASNSP2	GuideToPharmacology	2024.1	activator	2.625383561784725	IUPHAR.LIGAND:2411	rxcui:31748	NICORANDIL	FALSE	FALSE	FALSE
NCBIGENE:540	hgnc:870	ATP7B	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:9583	iuphar.ligand:9583	PSORA-4	FALSE	FALSE	FALSE
NCBIGENE:546	hgnc:886	ATRX	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:546	hgnc:886	ATRX	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:1052	iuphar.ligand:1052	LINOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11405	iuphar.ligand:11405	LP533401	FALSE	FALSE	FALSE
NCBIGENE:1872	hgnc:3116	E2F3P1	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:5070	iuphar.ligand:5070	LIGHT	FALSE	FALSE	FALSE
RPL38	hgnc:10349	RPL38	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:2679	hgnc:4252	GGT3P	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9584	iuphar.ligand:9584	ML324	FALSE	FALSE	FALSE
NCBIGENE:2717	hgnc:4296	GLA	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8949	iuphar.ligand:8949	A-196	FALSE	FALSE	FALSE
RPLP1	hgnc:10372	RPLP1	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:2681	hgnc:4253	GGTA1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10083	iuphar.ligand:10083	COMPOUND 9  [DOI:10.26434/CHEMRXIV.7072592.V1]	FALSE	FALSE	FALSE
NCBIGENE:2105	hgnc:7111	MKNK2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:6010	iuphar.ligand:6010	MNK1 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1320	iuphar.ligand:1320	&ALPHA;-MSH	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:9272	iuphar.ligand:9272	SETMELANOTIDE	FALSE	FALSE	FALSE
RPL36	hgnc:13631	RPL36	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.093931433	IUPHAR.LIGAND:7714	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.2059124362184097	IUPHAR.LIGAND:8143	iuphar.ligand:8143	COMPOUND 1O [PMID: 24210504]	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:10627	ncit:C123925	ZANDELISIB	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.1029562181092048	IUPHAR.LIGAND:7953	iuphar.ligand:7953	BMS-777607	FALSE	FALSE	TRUE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:7962	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.028078969	IUPHAR.LIGAND:5887	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:1573	hgnc:2634	CYP2J2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:6486	iuphar.ligand:6486	XMT-1191	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.5834185692854944	HT-0712	drugbank:DB11650	HT-0712	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:9920	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	0.3500511415712967	IUPHAR.LIGAND:1432	iuphar.ligand:1432	SIB-1893	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1428	iuphar.ligand:1428	MTEB	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	0.7001022831425934	IUPHAR.LIGAND:1365	iuphar.ligand:1365	(1S,3R)-ACPD	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.6250913242344582	HT-0712	drugbank:DB11650	HT-0712	FALSE	FALSE	FALSE
NCBIGENE:1512	hgnc:2535	CTSH	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8842	iuphar.ligand:8842	COMPOUND 35 [PMID: 23916259]	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1377	iuphar.ligand:1377	DCG-IV	FALSE	FALSE	FALSE
NCBIGENE:2099	hgnc:3467	ESR1	GuideToPharmacology	2024.1	inhibitor	0.061340737	IUPHAR.LIGAND:12936	iuphar.ligand:12936	PCC0105003	FALSE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	1.458546423213736	FILOREXANT	ncit:C169980	FILOREXANT	FALSE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:11674	iuphar.ligand:11674	TIZATERKIB	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	0.1646008502686348	IUPHAR.LIGAND:5269	iuphar.ligand:5269	SB203580	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.044198376	IUPHAR.LIGAND:9917	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1494	hgnc:6877	MAPK3	GuideToPharmacology	2024.1	inhibitor	0.2972132334095915	IUPHAR.LIGAND:9210	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9355	iuphar.ligand:9355	GNE-3511	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.4167275494896389	IUPHAR.LIGAND:10371	iuphar.ligand:10371	COMPOUND 20 [PMID: 30998356]	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.1483267549030917	IUPHAR.LIGAND:12057	iuphar.ligand:12057	TP0556351	FALSE	FALSE	FALSE
NCBIGENE:1628	hgnc:2697	DBP	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5220	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
NCBIGENE:1628	hgnc:2697	DBP	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8846	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:12057	iuphar.ligand:12057	TP0556351	FALSE	FALSE	FALSE
NCBIGENE:1630	hgnc:2701	DCC	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8259	iuphar.ligand:8259	CM-352	FALSE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:12057	iuphar.ligand:12057	TP0556351	FALSE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:7823	iuphar.ligand:7823	AZD6605	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1461	iuphar.ligand:1461	MOTILIN-(1-12) (HUMAN)	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	0.5303805175322677	IUPHAR.LIGAND:6639	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:7822	iuphar.ligand:7822	AZD6088	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:299	ncit:C76041	FURTRETHONIUM IODIDE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.5527123287967841	IUPHAR.LIGAND:365	iuphar.ligand:365	DIMETHYL-W84	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.035719504	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:308	iuphar.ligand:308	P-F-HHSID	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:10665	iuphar.ligand:10665	UCSF3384	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:9194	ncit:C170144	ATICAPRANT	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:12062	iuphar.ligand:12062	COMPOUND 27 [PMID: 35834807]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:9563	ncit:C125471	EGANELISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:10163	iuphar.ligand:10163	RV6153	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:10627	ncit:C123925	ZANDELISIB	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:9800	iuphar.ligand:9800	SELETALISIB	FALSE	FALSE	FALSE
NCBIGENE:2149	hgnc:3537	F2R	GuideToPharmacology	2024.1	inhibitor	0.2885036881082115	IUPHAR.LIGAND:8839	iuphar.ligand:8839	TORIN 2	FALSE	FALSE	FALSE
F2RL3	hgnc:3540	F2RL3	ChEMBL	33	inhibitor	8.751278539282415	BMS-986141	drugbank:DB14942	BMS-986141	FALSE	FALSE	FALSE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:7372	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9853	iuphar.ligand:9853	MK-0873	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:7372	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:5260	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9878	iuphar.ligand:9878	6-HYDROXY-5,7-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:5258	iuphar.ligand:5258	RO20-1724	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9878	iuphar.ligand:9878	6-HYDROXY-5,7-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:5258	iuphar.ligand:5258	RO20-1724	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:6557	iuphar.ligand:6557	RS-25344	FALSE	FALSE	FALSE
POLA2	hgnc:30073	POLA2	ChEMBL	33	inhibitor	0.6819178082557728	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:5658	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:9712	iuphar.ligand:9712	COMPOUND 5E [PMID: 28580438]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.075010959	IUPHAR.LIGAND:5695	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:9921	iuphar.ligand:9921	TAFETINIB	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:10672	iuphar.ligand:10672	COMPOUND 5 [TOMASSI ET AL., 2020]	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	1.779921058837101	DELAPRIL	ncit:C75022	DELAPRIL	FALSE	FALSE	FALSE
NCBIGENE:2383	hgnc:3895	FRA2K	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8658	iuphar.ligand:8658	PEPTIDE 18 [PMID: 24350995]	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.1422972120208522	IUPHAR.LIGAND:9061	iuphar.ligand:9061	PF-03882845	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:9606	iuphar.ligand:9606	PROGRAMMED CELL DEATH 1 LIGAND 1	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.1715936968486748	ABIVERTINIB	ncit:C147125	ABIVERTINIB	FALSE	FALSE	FALSE
NCBIGENE:2401	hgnc:3912	FRA6A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9819	iuphar.ligand:9819	COMPOUND 11 [PMID: 29442501]	FALSE	FALSE	FALSE
NCBIGENE:2408	hgnc:9545	PSMB8	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:8649	iuphar.ligand:8649	HT1042	FALSE	FALSE	FALSE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8287	iuphar.ligand:8287	EPZ015666	FALSE	FALSE	FALSE
NCBIGENE:2404	hgnc:3915	FRA6D	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8618	iuphar.ligand:8618	COMPOUND 3B [PMID: 24946214]	FALSE	FALSE	FALSE
NCBIGENE:1254	ncbigene:1254	CMTX3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:7032	iuphar.ligand:7032	COMPOUND 1 [PMID: 22795084]	FALSE	FALSE	FALSE
NCBIGENE:1257	ncbigene:1257	CNC2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7037	iuphar.ligand:7037	C21	FALSE	FALSE	FALSE
NCBIGENE:1487	hgnc:2494	CTBP1	GuideToPharmacology	2024.1	inhibitor	0.4303907478335614	IUPHAR.LIGAND:7946	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	agonist	0.040021091	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.053798843	IUPHAR.LIGAND:7946	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	agonist	0.040515178	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:10601	iuphar.ligand:10601	AZD7648	FALSE	FALSE	FALSE
NCBIGENE:1492	hgnc:9414	PRKG1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
NCBIGENE:1492	hgnc:9414	PRKG1	GuideToPharmacology	2024.1	modulator	4.773424657790408	IUPHAR.LIGAND:12071	iuphar.ligand:12071	ALLOSTERIC MODULATOR 33 [PMID: 35878399]	FALSE	FALSE	FALSE
NCBIGENE:2175	hgnc:3582	FANCA	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5196	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	agonist	0.038159645	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9698	iuphar.ligand:9698	CEP-37440	FALSE	FALSE	FALSE
NCBIGENE:3203	hgnc:5107	HOXA6	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12067	ncit:C155850	VOCIPROTAFIB	FALSE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	agonist	0.025439763	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	0.1615620653405984	IUPHAR.LIGAND:5890	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	agonist	0.036463661	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
NCBIGENE:2802	hgnc:4426	GOLGA3	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:7784	iuphar.ligand:7784	CCG-50014	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	0.095468493	IUPHAR.LIGAND:5890	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:2813	hgnc:4441	GP2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8033	iuphar.ligand:8033	RGS4 INHIBITOR 11B	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	agonist	0.039068208	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.038467158	IUPHAR.LIGAND:2644	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:2652	iuphar.ligand:2652	CD666	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:12792	iuphar.ligand:12792	KCL-286	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.077217164	IUPHAR.LIGAND:2646	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
NCBIGENE:2813	hgnc:4441	GP2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8034	iuphar.ligand:8034	CCG-203920	FALSE	FALSE	FALSE
CCKAR	hgnc:1570	CCKAR	ChEMBL	33	inhibitor	7.876150685354174	DEXLOXIGLUMIDE	ncit:C96871	DEXLOXIGLUMIDE	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.1930429089547592	IUPHAR.LIGAND:2646	drugbank:DB02877	AROTINOID ACID	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.2734774543525755	IUPHAR.LIGAND:5429	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:11416	ncit:C158093	ZETELETINIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1030909775569918	Navitoclax	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	Exarafenib	ncit:C180835	EXARAFENIB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.926605963	HX008	ncit:C160717	PUCOTENLIMAB	FALSE	FALSE	FALSE
SELPLG	hgnc:10722	SELPLG	ChEMBL	33	inhibitor	52.50767123569449	NEIHULIZUMAB	ncit:C121711	NEIHULIZUMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.235474617310458	BMS-936559	chembl:CHEMBL4297702	BMS-936559	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.3088686543276147	Cetrelimab	ncit:C129448	CETRELIMAB	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.5609793935437446	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	0.33338204	Melphalan	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.1802322811293861	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.3271505995993426	CPL304110	ncit:C173964	FGFR INHIBITOR CPL304110	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1526385791735305	Cetrelimab	ncit:C129448	CETRELIMAB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.07631929	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	1.221108633388244	Tinengotinib	ncit:C162532	TINENGOTINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.305277158	Zotatifin	ncit:C165746	ZOTATIFIN	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	PENPULIMAB	ncit:C155879	PENPULIMAB	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.031583562	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.033919684	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	PHI-101	drugbank:DB17237	PHI-101	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.8643238063488805	Lestaurtinib	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.108040476	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	FLX925	ncit:C120209	FLT3/CDK4/6 INHIBITOR FLX925	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.081030357	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.069089041	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.4605936073306534	SR9009	iuphar.ligand:8901	SR9009	FALSE	FALSE	FALSE
CTSK	hgnc:2536	CTSK	ChEMBL	33	inhibitor	11.66837138570988	BALICATIB	ncit:C79521	BALICATIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.028199609	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.004321619	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.1604757678352521	Vorasidenib	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.007336035	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2536602475154323	Pacritinib	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.652269208	Fedratinib	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.099220845	Dactolisib	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.008103036	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.2500365296937833	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.027010119	Infigratinib	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.097236428	Toripalimab-tpzi	rxcui:2669407	TORIPALIMAB-TPZI	TRUE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.2011788169949981	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.057574201	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.019318496	Abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.2318219480604613	SAR405838	ncit:C106120	P53-HDM2 INTERACTION INHIBITOR MI-773	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.012419033	Gedatolisib	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
NOS2	hgnc:7873	NOS2	ChEMBL	33	inhibitor	0.6081969641200136	TILARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	0.7143900848393808	OTAMIXABAN	ncit:C90704	OTAMIXABAN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.2035181055647073	FGFR INHIBITOR DEBIO 1347	chembl:CHEMBL3907479	FGFR INHIBITOR DEBIO 1347	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
FGB	hgnc:3662	FGB	ChEMBL	33	cleavage	2.333674277141977	ALFIMEPRASE	ncit:C79877	ALFIMEPRASE	FALSE	FALSE	FALSE
C3	hgnc:1318	C3	ChEMBL	33	inhibitor	5.834185692854944	AMY-101	drugbank:DB14803	AMY-101	FALSE	FALSE	FALSE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	1.750255707856483	MERIMEPODIB	ncit:C66097	MERIMEPODIB	FALSE	FALSE	FALSE
FAP	hgnc:3590	FAP	ChEMBL	33	binder	2.692701089009974	SIMLUKAFUSP ALFA	ncit:C129383	SIMLUKAFUSP ALFA	FALSE	FALSE	FALSE
GWT1	hgnc:23213	PIGW	ChEMBL	33	inhibitor	52.50767123569449	FOSMANOGEPIX	ncit:C155900	FOSMANOGEPIX	FALSE	FALSE	FALSE
IL2RG	hgnc:6010	IL2RG	ChEMBL	33	binder	1.750255707856483	SIMLUKAFUSP ALFA	ncit:C129383	SIMLUKAFUSP ALFA	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN [INJECTION], BIPHASIC	chembl:CHEMBL2108968	INSULIN [INJECTION], BIPHASIC	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN, ISOPHANE	chembl:CHEMBL2108964	INSULIN, ISOPHANE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	ChEMBL	33	inhibitor	0.7001022831425933	PLONMARLIMAB	ncit:C172653	PLONMARLIMAB	FALSE	FALSE	FALSE
FCGRT	hgnc:3621	FCGRT	ChEMBL	33	inhibitor	5.834185692854944	ORILANOLIMAB	ncit:C139561	ORILANOLIMAB	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN HUMAN, ISOPHANE	chembl:CHEMBL2108973	INSULIN HUMAN, ISOPHANE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
IL10RB	hgnc:5965	IL10RB	ChEMBL	33	agonist	4.375639269641208	PEGILODECAKIN	ncit:C113295	PEGILODECAKIN	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2287915957982331	BMN673	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1598407039138341	BMN673	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
APH1A	hgnc:29509	APH1A	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.7501095890813501	MK-0752	drugbank:DB12852	MK-0752	FALSE	FALSE	TRUE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1088116604009326	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.022122465	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2681242786503549	MLS003106905	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
RRM2B	hgnc:17296	RRM2B	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.112919723	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.080781033	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-2300	chembl:CHEMBL608855	CHEMBL:CHEMBL608855	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	0.3500511415712967	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	CID 5310655	chembl:CHEMBL408563	CHEMBL:CHEMBL408563	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	CLOCORTOLONE PIVALATE	rxcui:21249	CLOCORTOLONE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.020296742	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CLOMIPRAMINE HYDROCHLORIDE	rxcui:81984	CLOMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.02804897	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008916229	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.035964158	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.067664525	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.019889269	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.014985066	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-390523	chembl:CHEMBL157258	CHEMBL:CHEMBL157258	FALSE	FALSE	FALSE
PSMB3	hgnc:9540	PSMB3	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC3	hgnc:9549	PSMC3	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC2	hgnc:9548	PSMC2	DTC	9/2/20	NULL	0.729273212	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ADAM17	hgnc:195	ADAM17	DTC	9/2/20	NULL	0.9723642821424908	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
PSMC4	hgnc:9551	PSMC4	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD4	hgnc:9561	PSMD4	DTC	9/2/20	NULL	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	DESMETHOXYYANGONIN	chembl:CHEMBL254218	DESMETHOXYYANGONIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.030796288	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.004630306	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.029665351	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	TCMDC-123862	chembl:CHEMBL533074	CHEMBL:CHEMBL533074	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.027177884	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.1094923635591405	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	NSC-693571	chembl:CHEMBL1287983	CHEMBL:CHEMBL1287983	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	GUANIDINONALTRINDOLE	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1640864726115453	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.028598949	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	DEMETHYLENCECALIN	chembl:CHEMBL443462	DEMETHYLENCECALIN	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	inhibitor	0.051377369	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.072927321	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.011049594	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	STROPHANTHIDIN ACETATE	chembl:CHEMBL1981679	STROPHANTHIDIN ACETATE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.03251249	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.130616098	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	NSC-125910	chembl:CHEMBL1529609	CHEMBL:CHEMBL1529609	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	1.129197231	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	MEDRONIC ACID	rxcui:1314368	MEDRONIC ACID	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.009481342	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	FLUMEQUINE	rxcui:25112	FLUMEQUINE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.192335792	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PRULIFLOXACIN	ncit:C72637	PRULIFLOXACIN	FALSE	FALSE	FALSE
FPR2	hgnc:3827	FPR2	DTC	9/2/20	NULL	4.375639269641208	AG-26	iuphar.ligand:6268	AG-26	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006811217	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	BROMETHALIN	chembl:CHEMBL1901818	BROMETHALIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.019059046	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.093763699	DNDI1416975	chembl:CHEMBL1415851	CHEMBL:CHEMBL1415851	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.012888481	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	DTC	9/2/20	NULL	0.1642918374083057	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	ZK-164015	chembl:CHEMBL184074	CHEMBL:CHEMBL184074	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.009065551	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ELEMICIN	chembl:CHEMBL481044	ELEMICIN	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.1403948428761885	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.025827679	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.6819178082557726	IC261	drugbank:DB03083	IC261	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	N-PHENETHYLCINNAMAMIDE	chembl:CHEMBL1305393	CHEMBL:CHEMBL1305393	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.005562253	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.027840759	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	AM-251	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.015193192	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	ROCURONIUM BROMIDE	rxcui:32521	ROCURONIUM BROMIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
SF3B3	hgnc:10770	SF3B3	DTC	9/2/20	NULL	52.50767123569449	PLA D	chembl:CHEMBL1242564	PLA D	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1396480617970598	VITAMIN B2	chembl:CHEMBL1397833	VITAMIN B2	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	ONONIN	chembl:CHEMBL465980	ONONIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	0.1105424657593568	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	ETOFENAMATE	rxcui:24608	ETOFENAMATE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	MMV667491	chembl:CHEMBL1437888	CHEMBL:CHEMBL1437888	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	(S)-ROSCOVITINE	chembl:CHEMBL133342	(S)-ROSCOVITINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	DTC	9/2/20	NULL	0.729273212	SRIF-28	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.036847489	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	BUTACLAMOL	ncit:C81088	BUTACLAMOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BROMODICHLOROACETIC ACID	chembl:CHEMBL453528	BROMODICHLOROACETIC ACID	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.023202683	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	EUPAROTIN ACETATE	chembl:CHEMBL404627	EUPAROTIN ACETATE	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.090530468	FENOLDOPAM MESYLATE	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.2488515224440497	TCMDC-125561	chembl:CHEMBL526763	CHEMBL:CHEMBL526763	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DICOFOL	chembl:CHEMBL228511	DICOFOL	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	(R)-NIPHATENONE B	chembl:CHEMBL1946014	CHEMBL:CHEMBL1946014	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.029301156	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.034251579	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.049817525	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	1.394008970859145	SOLOMONSTEROL A	chembl:CHEMBL1649712	SOLOMONSTEROL A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	2-METHYL GRAMINE	chembl:CHEMBL1354316	2-METHYL GRAMINE	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.077789143	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	STROPHANTHIDIN ACETATE	chembl:CHEMBL1981679	STROPHANTHIDIN ACETATE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.020721259	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006210251	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	ETHAMSYLATE	rxcui:4112	ETHAMSYLATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	BISACODYL	rxcui:1596	BISACODYL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.005333977	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	GLABRANIN	chembl:CHEMBL253998	GLABRANIN	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.013120358	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	DTC	9/2/20	NULL	4.773424657790408	BENZO[B]THIOPHEN-2-YLMETHANAMINE	chembl:CHEMBL1770735	CHEMBL:CHEMBL1770735	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005208578	MIBEFRADIL	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	PYRILAMINE MALEATE	rxcui:82091	PYRILAMINE MALEATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	1R,9S-HYDRASTINE	chembl:CHEMBL475536	1R,9S-HYDRASTINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	5-(4-PHENYLBUTOXY)PSORALEN	iuphar.ligand:9583	PSORA-4	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.1119566550867686	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1367387271762877	BENZOXATHIAN	chembl:CHEMBL191044	BENZOXATHIAN	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	4.039051633514961	SJ000259188	chembl:CHEMBL592578	CHEMBL:CHEMBL592578	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.017114626	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.01609924	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.048935388	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	OCTAVERINE	ncit:C90894	OCTAVERINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SJ000160630	chembl:CHEMBL591404	CHEMBL:CHEMBL591404	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	DTC	9/2/20	NULL	0.2917092846427472	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003217973	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.022099188	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.008310806	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CID 650707	chembl:CHEMBL408653	CHEMBL:CHEMBL408653	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.023780648	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.1852122442176172	NSC-56452	chembl:CHEMBL1358137	CHEMBL:CHEMBL1358137	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1274458039701322	OXYCARBOXIN	chembl:CHEMBL1712057	OXYCARBOXIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.031822831	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001854084	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.008562895	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CTSK	hgnc:2536	CTSK	DTC	9/2/20	NULL	11.66837138570988	2-(1-CYCLODODECYLETHYLIDENE)HYDRAZINECARBOTHIOAMIDE	chembl:CHEMBL2316602	CHEMBL:CHEMBL2316602	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	1.193356164447602	BUFURALOL	ncit:C72613	BUFURALOL	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.2333674277141977	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	BENZO[E]PYRENE	chembl:CHEMBL1371125	BENZO[E]PYRENE	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.6482428547616604	OPHIOBOLIN O	chembl:CHEMBL1934283	OPHIOBOLIN O	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.7955707762984013	OPHIOBOLIN O	chembl:CHEMBL1934283	OPHIOBOLIN O	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.010348378	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.011355465	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
STAT1	hgnc:11362	STAT1	DTC	9/2/20	NULL	0.729273212	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.0136917	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	3.088686543276147	NSC-640583	chembl:CHEMBL1287895	CHEMBL:CHEMBL1287895	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	3,3'-DIMETHOXYBENZIDINE	chembl:CHEMBL398363	CHEMBL:CHEMBL398363	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1250182648468916	FAGARONINE	chembl:CHEMBL282622	FAGARONINE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.013588942	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.030886865	FENOLDOPAM MESYLATE	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	DEOXIEPINEPHRINE	chembl:CHEMBL31088	DEOXIEPINEPHRINE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.012466209	CYPROHEPTADINE HYDROCHLORIDE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-3314	chembl:CHEMBL582287	CHEMBL:CHEMBL582287	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.034229251	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	DNDI1417597	chembl:CHEMBL1330352	CHEMBL:CHEMBL1330352	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.012729132	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	SB-204070	iuphar.ligand:256	SB 204070	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00626658	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	DTC	9/2/20	NULL	0.062434805	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.051478109	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.2778183663264259	PD-174265	iuphar.ligand:6017	PD 174265	FALSE	FALSE	FALSE
RGS12	hgnc:9994	RGS12	DTC	9/2/20	NULL	0.525076712	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-2559	chembl:CHEMBL583584	CHEMBL:CHEMBL583584	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.008371759	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	IMAZODAN	ncit:C83787	IMAZODAN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003703461	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.1400204566285186	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.2625383561784725	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.015286076	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	3,6-DIMETHOXYFLAVONE	chembl:CHEMBL1331521	3,6-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.03219848	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	OXYQUINOLINE	rxcui:110	OXYQUINOLINE	TRUE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.014354202	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	2-HYDROXYESTRADIOL	ncit:C120474	2-HYDROXYESTRADIOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.01514062	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	PD-160170	chembl:CHEMBL422942	CHEMBL:CHEMBL422942	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	1.250182648468916	2,4-DIACETYL PHLOROGLUCINOL	chembl:CHEMBL276139	2,4-DIACETYLPHLOROGLUCINOL	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.040235763	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.015466177	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.9723642821424906	GW459057A	chembl:CHEMBL1909354	GW459057A	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.027476542	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	RESMETHRIN	rxcui:35380	RESMETHRIN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	DESLORATADINE	rxcui:275635	DESLORATADINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	FLUORESCEIN DIACETATE	chembl:CHEMBL1492044	FLUORESCEIN DIACETATE	FALSE	FALSE	FALSE
RHEB	hgnc:10011	RHEB	DTC	9/2/20	NULL	52.50767123569449	4,4'-HYDROXYBIPHENYL	chembl:CHEMBL76398	CHEMBL:CHEMBL76398	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	GNF-PF-628	chembl:CHEMBL1448140	CHEMBL:CHEMBL1448140	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW300660X	chembl:CHEMBL272028	GW300660X	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	4-METHYLDAPHNETIN	chembl:CHEMBL276618	4-METHYLDAPHNETIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	ALVERINE CITRATE	rxcui:71767	ALVERINE CITRATE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2580229544751573	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	DTC	9/2/20	NULL	2.187819634820604	LYCOBETAINE	chembl:CHEMBL253553	LYCOBETAINE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	SOFALCONE	ncit:C81118	SOFALCONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665830	chembl:CHEMBL602580	CHEMBL:CHEMBL602580	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	FLAVONE	rxcui:1536070	FLAVONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004919212	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.095122593	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	GNF-PF-4992	chembl:CHEMBL275177	CHEMBL:CHEMBL275177	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.096167896	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.060772768	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	7.501095891	MURABUTIDE	ncit:C175149	MURABUTIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.019724895	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00506733	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.011365297	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.045579576	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-238165	chembl:CHEMBL2059074	CHEMBL:CHEMBL2059074	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.027929612	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.022730594	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.042863405	NSC-11437	chembl:CHEMBL1814509	CHEMBL:CHEMBL1814509	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	GNF-PF-4832	chembl:CHEMBL601137	CHEMBL:CHEMBL601137	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	DTC	9/2/20	NULL	0.048260727	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FLUTOLANIL	chembl:CHEMBL487185	FLUTOLANIL	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.032982206	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.041344623	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.03070624	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.013415348	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.03043923	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.2476776945079929	GNF-PF-186	chembl:CHEMBL601140	CHEMBL:CHEMBL601140	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.040051618	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.007672074	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.012026494	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.006356861	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	4,4'-BIPYRIDINE	chembl:CHEMBL1374568	CHEMBL:CHEMBL1374568	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TRICHLOROMONOFLUOROMETHANE	chembl:CHEMBL348290	TRICHLOROMONOFLUOROMETHANE	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.056826484	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	SJ000111093	chembl:CHEMBL585045	CHEMBL:CHEMBL585045	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	DOCONEXENT	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	MEPANIPYRIM	chembl:CHEMBL2269513	MEPANIPYRIM	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.034251579	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	TCMDC-125473	chembl:CHEMBL535051	CHEMBL:CHEMBL535051	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010058941	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	3.500511415712966	HIRSUTINOLIDE-13-OACETATE	chembl:CHEMBL2062869	CHEMBL:CHEMBL2062869	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	RONNEL	drugbank:DB11456	RONNEL	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.3500511415712966	FERBAM	chembl:CHEMBL460100	FERBAM	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	FAMPROFAZONE	ncit:C65616	FAMPROFAZONE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1591141552596803	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.004602706	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.6908904109959803	NSC-628113	chembl:CHEMBL176599	CHEMBL:CHEMBL176599	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.016206071	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	1.458546423213736	SJ000033254	chembl:CHEMBL591148	CHEMBL:CHEMBL591148	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.017775109	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008103036	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	GNF-PF-4992	chembl:CHEMBL275177	CHEMBL:CHEMBL275177	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	GNF-PF-3286	chembl:CHEMBL581880	CHEMBL:CHEMBL581880	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	2-HYDROXY-NAPHTHALDEHYDE THIOSEMICARBAZONE	chembl:CHEMBL505209	CHEMBL:CHEMBL505209	FALSE	FALSE	FALSE
CAMK2A	hgnc:1460	CAMK2A	DTC	9/2/20	NULL	0.2344092465879218	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.020048748	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	6-METHOXY-HARMALAN	chembl:CHEMBL338115	CHEMBL:CHEMBL338115	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	EUPAROTIN ACETATE	chembl:CHEMBL404627	EUPAROTIN ACETATE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.020002922	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.055622533	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	PHOSMET	drugbank:DB11448	PHOSMET	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00399693	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	0.6731752722524935	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.029970132	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	NSC-26699	chembl:CHEMBL221721	CHEMBL:CHEMBL221721	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.015088411	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.020117882	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.5834185692854944	DIMPYLATE	ncit:C169912	DIMPYLATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00095957	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.02639903	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.021189536	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.038467158	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665852	chembl:CHEMBL10835	CHEMBL:CHEMBL10835	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TINORIDINE	ncit:C76821	TINORIDINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.017835486	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	MINOCYCLINE	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.009532983	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.2344092465879218	SB-242235	chembl:CHEMBL95692	SB-242235	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	NSC-56452	chembl:CHEMBL1358137	CHEMBL:CHEMBL1358137	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.034727296	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.014488872	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.012154554	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.1902451856365742	HYDRAMETHYLNON	chembl:CHEMBL464812	HYDRAMETHYLNON	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.019889269	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	2.019525817	BERKELEYAMIDE B	chembl:CHEMBL468640	BERKELEYAMIDE B	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	NORSTICTIC ACID	chembl:CHEMBL228281	NORSTICTIC ACID	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.3017682254924971	PEPSTATIN	ncit:C96295	PEPSTATIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.02617531	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.3387591692625452	SJ000114740	chembl:CHEMBL592068	CHEMBL:CHEMBL592068	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.010742159	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	AZELNIDIPINE	ncit:C73023	AZELNIDIPINE	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	CLORINDIONE	ncit:C81463	CLORINDIONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	GNF-PF-186	chembl:CHEMBL601140	CHEMBL:CHEMBL601140	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	FLAVOXATE	rxcui:4440	FLAVOXATE	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1902451856365742	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.035098711	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
HNF4A	hgnc:5024	HNF4A	DTC	9/2/20	NULL	0.1367387271762877	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
RPS8	hgnc:10441	RPS8	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
CSNK1E	hgnc:2453	CSNK1E	ChEMBL	33	inhibitor	4.375639269641208	UMBRALISIB TOSYLATE	rxcui:2478438	UMBRALISIB TOSYLATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	RAC-GONIOTHALAMIN	chembl:CHEMBL1170485	CHEMBL:CHEMBL1170485	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CETYLPYRIDINIUM CHLORIDE	rxcui:2287	CETYLPYRIDINIUM CHLORIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	N-HISTIDYL-2-AMINONAPHTHALENE (BETANA)	chembl:CHEMBL1489988	N-HISTIDYL-2-AMINONAPHTHALENE (BETANA)	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.3500511415712966	M-CSF	iuphar.ligand:4905	M-CSF	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:8304	iuphar.ligand:8304	COMPOUND 7D [PMID: 25703523]	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	3.580068493342807	IUPHAR.LIGAND:879	iuphar.ligand:3477	[3H]L365260	FALSE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	ChEMBL	33	inhibitor	19.69037671338543	BLISIBIMOD	ncit:C166445	BLISIBIMOD	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	TRIFLOXYSTROBIN	chembl:CHEMBL1897483	TRIFLOXYSTROBIN	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	COSMIC	4-Sep-20	NULL	0.5114383561918295	PD0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	6'-IODONONIVAMIDE	chembl:CHEMBL177809	CHEMBL:CHEMBL177809	FALSE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	blocker	0.1093909817410302	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	CARBETAPENTANE CITRATE	rxcui:283547	CARBETAPENTANE CITRATE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.034118045	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.1881995384791917	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11751	iuphar.ligand:11751	JNJ-67569762	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	NULL	0.2500365296937833	IUPHAR.LIGAND:5087	iuphar.ligand:5087	VEGFC	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.3513393859865807	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:3248	iuphar.ligand:3248	[3H]5-HT	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.6177373086552295	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CLOFOCTOL	rxcui:21264	CLOFOCTOL	FALSE	FALSE	FALSE
NRG2	hgnc:7998	NRG2	PharmGKB	4/5/24	NULL	1.312691780892362	panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	3,5-DIPHENYLISOXAZOLE	chembl:CHEMBL1374535	3,5-DIPHENYLISOXAZOLE	FALSE	FALSE	FALSE
AREG	hgnc:651	AREG	PharmGKB	4/5/24	NULL	0.3333820395917111	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.021697385	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	TALC	12-May-16	inhibitor	0.02617531	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	IODOPHENPROPIT	iuphar.ligand:1266	IODOPHENPROPIT	FALSE	FALSE	FALSE
INTERLEUKIN-13	hgnc:5973	IL13	TTD	2020.06.01	NULL	8.751278539282415	Lebrikizumab	ncit:C87767	LEBRIKIZUMAB	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.056826484	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.08334551	IUPHAR.LIGAND:147	iuphar.ligand:147	DOI	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	ChEMBL	33	inhibitor	0.1215455352678113	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	modulator	0.084146909	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	TAXIFOLIN	drugbank:DB02224	TAXIFOLIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	SAQUINAVIR	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	ETOXAZOLE	chembl:CHEMBL1881674	ETOXAZOLE	FALSE	FALSE	FALSE
LIPA	hgnc:6617	LIPA	NCI	14-Sep-17	NULL	1.591141552596803	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
NCBIGENE:2351	ncbigene:2351	FOLR2L	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9298	iuphar.ligand:9298	LHVS	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	MESOTRIONE	chembl:CHEMBL1873440	MESOTRIONE	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	TALC	12-May-16	inhibitor	0.1374032518317239	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9568	iuphar.ligand:9568	QWF	FALSE	FALSE	FALSE
NCBIGENE:281	hgnc:479	AMYP1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:7757	iuphar.ligand:7757	COMPOUND 38 [PMID: 22123324]	FALSE	FALSE	FALSE
RPL10	hgnc:10298	RPL10	NCI	14-Sep-17	NULL	0.7955707762984016	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:4201	iuphar.ligand:4201	GINKGOLIDE X	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.1959241464018451	IBCASERTIB	ncit:C115970	IBCASERTIB	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	8.751278539282417	ULIMORELIN HYDROCHLORIDE	ncit:C102755	ULIMORELIN HYDROCHLORIDE	FALSE	FALSE	FALSE
DPEP1	hgnc:3002	DPEP1	ChEMBL	33	inhibitor	17.50255707856483	CILASTATIN	rxcui:2540	CILASTATIN	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.011112735	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.138178082	(+)-EPITAXIFOLIN	chembl:CHEMBL9249	(+)-EPITAXIFOLIN	FALSE	FALSE	FALSE
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.1172046232939609	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.016408647	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004961042	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.021891879	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
NCBIGENE:1621	hgnc:2689	DBH	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5301	iuphar.ligand:5301	Z-WEHD-FMK	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:8897	iuphar.ligand:8897	AC-186	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.004214099	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
UNIPROT:P22748	hgnc:1375	CA4	TdgClinicalTrial	Jan-14	NULL	0.3977853881492008	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
CANCER/TESTIS ANTIGEN 1	hgnc:2491	CTAG1B	TTD	2020.06.01	NULL	2.187819634820604	CDX-1401	ncit:C170362	RASDEGAFUSP ALFA	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
GUCA2B	hgnc:4683	GUCA2B	NCI	14-Sep-17	NULL	10.50153425	POLYETHYLENE GLYCOL	rxcui:1310594	POLYETHYLENE GLYCOL 4000	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.1166837138570988	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	L-733060	chembl:CHEMBL1256740	CHEMBL:CHEMBL1256740	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.1481697953740938	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.093098708	ERDAFITINIB	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4600	iuphar.ligand:4600	ORG 24598	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	2-METHOXY-5 (6)EPOXY-TETRAHYDROCARYOPHYLLENE	chembl:CHEMBL1488390	2-METHOXY-5 (6)EPOXY-TETRAHYDROCARYOPHYLLENE	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.1333528158366844	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.099446347	IUPHAR.LIGAND:2667	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.012649403	nefazodone	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	DAZOXIBEN HYDROCHLORIDE	ncit:C169879	DAZOXIBEN HYDROCHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003890322	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	DTC	9/2/20	NULL	1.666910197958555	RO-0506220	chembl:CHEMBL1956069	CHEMBL:CHEMBL1956069	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.070129236	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.024354207	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.2703097618311171	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.052090944	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.014565235	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.2885036881082116	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	GW9662	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	L-655240	chembl:CHEMBL362223	CHEMBL:CHEMBL362223	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.024275391	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.017799211	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:2360	hgnc:3868	FRA1A	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:12417	iuphar.ligand:12417	ABELACIMAB	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:1631	iuphar.ligand:1631	&BETA;-FNA	FALSE	FALSE	FALSE
NTSR1	hgnc:8039	NTSR1	DTC	9/2/20	NULL	4.375639269641208	TCMDC-123851	chembl:CHEMBL548458	CHEMBL:CHEMBL548458	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TOLPERISONE HYDROCHLORIDE	ncit:C84220	TOLPERISONE HYDROCHLORIDE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.4278402841426959	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
TXNRD1	hgnc:12437	TXNRD1	ChEMBL	33	inhibitor	8.751278539282415	AUROTHIOGLUCOSE	rxcui:4980	AUROTHIOGLUCOSE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	IRL-2500	iuphar.ligand:3887	IRL 2500	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	BILIRUBIN	iuphar.ligand:4577	BILIRUBIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	BIMATOPROST	rxcui:283810	BIMATOPROST	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1084869240406911	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	0.8751278539282416	Lumefantrine	rxcui:847728	LUMEFANTRINE	TRUE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	agonist	0.1544343271638073	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1344	iuphar.ligand:1344	2-[125I]MELATONIN	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.070690956	ALPELISIB	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.272767123	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1341192113299987	Alpha 2 Interferon	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.151464436	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.002697266	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.017092341	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
UNIPROT:P47712	hgnc:9035	PLA2G4A	TEND	1-Aug-11	NULL	1.458546423213736	FLURANDRENOLIDE	rxcui:4500	FLURANDRENOLIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	TCMDC-123984	chembl:CHEMBL532909	CHEMBL:CHEMBL532909	FALSE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.8078103267029924	PENTAERYTHRITOL TETRANITRATE	rxcui:7992	PENTAERYTHRITOL TETRANITRATE	TRUE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9929	iuphar.ligand:9929	XILIERTINIB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	SIBUTRAMINE HYDROCHLORIDE	rxcui:1294535	SIBUTRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ACO1	hgnc:117	ACO1	NCI	14-Sep-17	NULL	1.000146118775133	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.03140411	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	5-METHOXYFLAVONE	chembl:CHEMBL16685	CHEMBL:CHEMBL16685	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006027051	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
DEPTOR	hgnc:22953	DEPTOR	MyCancerGenome	20-Jun-17	inhibitor	1.346350544504987	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:303	iuphar.ligand:303	OXOTREMORINE-M	FALSE	FALSE	FALSE
RPL11	hgnc:10301	RPL11	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.095642388	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SULT1A3	hgnc:11455	SULT1A3	PharmGKB	4/5/24	NULL	1.009762908	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.09969811	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q13200	hgnc:9559	PSMD2	TEND	1-Aug-11	NULL	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10528	iuphar.ligand:10528	COMPOUND 32 [PMID: 31638797]	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.017945205	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	2.763561643983921	DIC10	ncit:C29869	SN-1,2-DIDECANOYLGLYCEROL	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.014287802	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	GNF-PF-3286	chembl:CHEMBL581880	CHEMBL:CHEMBL581880	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:11676	ncit:C171059	TUXOBERTINIB	FALSE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	3.938075342677087	Measles vaccines	wikidata:Q6804161	MEASLES VACCINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	SJ000150791	chembl:CHEMBL600572	CHEMBL:CHEMBL600572	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.2408608772279564	acetaminophen / tramadol	wikidata:Q48564239	ACETAMINOPHEN/TRAMADOL	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.075768645	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.2573905452730122	IUPHAR.LIGAND:1394	iuphar.ligand:1394	LY379268	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.4773424657790409	IUPHAR.LIGAND:2178	iuphar.ligand:2178	[PHE3]OT	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.2500365296937833	GLESATINIB	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.041672755	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.09963505	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.008143249	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.010594768	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	BERGAMOTTIN	chembl:CHEMBL1078442	BERGAMOTTIN	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.025891357	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.3977853881492008	DIFFERENTIATION INDUCER	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.3977853881492008	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
UNIPROT:P01031	hgnc:1331	C5	TEND	1-Aug-11	NULL	1.591141552596803	ECULIZUMAB	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.021138354	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.1458546423213736	PERIFOSINE	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1657439117288336	Copanlisib	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.2302968036653267	IUPHAR.LIGAND:4321	iuphar.ligand:4321	TETRAHYDRODEOXYCORTICOSTERONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	PROROXAN HYDROCHLORIDE	ncit:C84120	PROROXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-2323	chembl:CHEMBL49055	CHEMBL:CHEMBL49055	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.093763699	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	1.186614039224734	Valsartan	rxcui:69749	VALSARTAN	TRUE	FALSE	FALSE
ESRRB	hgnc:3473	ESRRB	DTC	9/2/20	NULL	1.060761035064535	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	1.419126249613364	PRX-00023	ncit:C80775	NALUZOTAN	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.8950171233357017	ESMOLOL	rxcui:49737	ESMOLOL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.0296486	BROMOCRIPTINE MESYLATE	rxcui:142426	BROMOCRIPTINE MESYLATE	TRUE	FALSE	FALSE
TLR5	hgnc:11851	TLR5	ChEMBL	33	agonist	35.00511415712966	ENTOLIMOD	ncit:C99166	ENTOLIMOD	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	PharmGKB	4/5/24	NULL	0.1154014752432846	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.028630137	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.082043236	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.045304289	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.042073455	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.1121958787087489	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:12440	iuphar.ligand:12440	DATISCETIN	FALSE	FALSE	FALSE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.063722902	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.016669102	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	LANSOPRAZOLE SULFIDE	chembl:CHEMBL899	LANSOPRAZOLE SULFIDE	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	0.1091635576625665	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.5834185692854944	dimethyl fumarate	rxcui:1373478	DIMETHYL FUMARATE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.029301156	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.015017209	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
GATA4	hgnc:4173	GATA4	DTC	9/2/20	NULL	17.50255707856483	NSC-85661	chembl:CHEMBL1684098	CHEMBL:CHEMBL1684098	FALSE	FALSE	FALSE
RPS17	hgnc:10397	RPS17	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
GP	hgnc:18280	RNF130	ChEMBL	33	inhibitor	7.501095891	LARCAVIXIMAB	ncit:C166475	LARCAVIXIMAB	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.061055432	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.024651489	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	ChEMBL	33	inhibitor	0.7955707762984014	SNDX-5613	chembl:CHEMBL4650278	SNDX-5613	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	FOSFONET	drugbank:DB02823	PHOSPHONOACETIC ACID	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.015959778	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:8250	iuphar.ligand:8250	SOTULETINIB	FALSE	FALSE	FALSE
NCBIGENE:2225	hgnc:11408	STK4	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8768	iuphar.ligand:8768	COMPOUND 38 [PMID: 20817473]	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	CARNOSIC ACID	chembl:CHEMBL484853	CARNOSIC ACID	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:8372	iuphar.ligand:8372	(-)-ENGLERIN A	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.034590034	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.027752469	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8538	iuphar.ligand:8538	PF-04852946	FALSE	FALSE	FALSE
NCBIGENE:429	hgnc:738	ASCL1	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	1.518294108020081	RIPRETINIB	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.056826484	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	ALOE-EMODIN	chembl:CHEMBL40275	ALOE-EMODIN	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1415301111474245	FRENTIZOLE	ncit:C167023	FRENTIZOLE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.039353698	Tamsulosin	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	OncoKB	23-Jul-20	NULL	0.1535312024435511	Ado-Trastuzumab Emtansine	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	1.184383561707394	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.020446912	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.066591847	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	5.834185692854944	LITHOGLYCOCHOLATE	chembl:CHEMBL258818	LITHOGLYCOCHOLATE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.009349657	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	ACP-001	chembl:CHEMBL4297687	ACP-001	FALSE	FALSE	FALSE
SYNUCLEIN ALPHA	hgnc:11138	SNCA	TTD	2020.06.01	NULL	3.182283105193606	RG7935	chembl:CHEMBL4298077	PRASINEZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2615	hgnc:4161	LRRC32	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:300	iuphar.ligand:300	METHYLFURMETHIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009084372	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	3.889457128569962	UBLITUXIMAB	rxcui:2626349	UBLITUXIMAB	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.008572681	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	CGI	2/1/22	NULL	0.159436249	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	THIOINOSINE	ncit:C877	THIOINOSINE	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.482607272	Donepezil	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2078	iuphar.ligand:2078	&BETA;3-TETRAPEPTIDE	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.073540156	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:5837	iuphar.ligand:5837	FMET-MET-TRP-LEU-LEU	FALSE	FALSE	FALSE
NCBIGENE:1708	hgnc:6019	IL6R	GuideToPharmacology	2024.1	antibody	12.11715490054488	IUPHAR.LIGAND:7999	rxcui:1923319	SARILUMAB	TRUE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:8059	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.060077427	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	2.282942227638891	BETA-SITOSTEROL	ncit:C63662	BETA-SITOSTEROL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.375054795	Naldemedine Tosylate	rxcui:1876597	NALDEMEDINE	TRUE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:9600	iuphar.ligand:9600	MIVAVOTINIB	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BIAPENEM	ncit:C72620	BIAPENEM	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	GNF-PF-3418	chembl:CHEMBL582099	CHEMBL:CHEMBL582099	FALSE	FALSE	FALSE
UNIPROT:P18858	hgnc:6598	LIG1	TEND	1-Aug-11	NULL	6.563458904461812	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.1829535583125243	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.084281976	IUPHAR.LIGAND:8805	iuphar.ligand:8805	COMPOUND 82 [PMID: 21332118]	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	DNDI1417420	chembl:CHEMBL1546223	CHEMBL:CHEMBL1546223	FALSE	FALSE	FALSE
NCBIGENE:1578	hgnc:42418	CYP3A51P	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8803	iuphar.ligand:8803	APSTATIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.03409589	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
KCNG1	hgnc:6248	KCNG1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.005753635	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
GLA	hgnc:4296	GLA	ChEMBL	33	modulator	4.039051633514961	MIGALASTAT	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-2503	chembl:CHEMBL601358	CHEMBL:CHEMBL601358	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	PROPIONYLPROMAZINE HYDROCHLORIDE	chembl:CHEMBL1256661	PROPIONYLPROMAZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.025489161	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.035976479	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.031069628	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.051629962	saquinavir	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.088396753	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.2476776945079929	Scriptaid	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9242	iuphar.ligand:9242	TX2-121-1	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:310	iuphar.ligand:310	HEXAHYDROSILADIFENIDOL	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1374032518317239	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005581766	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008103036	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.027383401	VP-16	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
UOX	hgnc:12575	UOX	NCI	14-Sep-17	NULL	31.50460274141669	POLYETHYLENE GLYCOL	rxcui:1310594	POLYETHYLENE GLYCOL 4000	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.016669102	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	OXETHAZAINE	ncit:C81409	OXETHAZAINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:10129	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000408461	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	DNDI1417185	chembl:CHEMBL1549738	CHEMBL:CHEMBL1549738	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.135503668	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.090064616	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	3-HYDROXY-3',4'-DIMETHOXYFLAVONE	chembl:CHEMBL77098	3-HYDROXY-3',4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.066297565	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.012282496	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.9907107780319716	(+)-TUBERIFERIN	chembl:CHEMBL1940084	CHEMBL:CHEMBL1940084	FALSE	FALSE	FALSE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3241214273808303	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.9546849315580818	Carprofen	rxcui:20343	CARPROFEN	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	MM-302	ncit:C96038	HER2-TARGETED LIPOSOMAL DOXORUBICIN HYDROCHLORIDE MM-302	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.067317527	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.9131768910555564	TPX-0131	chembl:CHEMBL4802183	TPX-0131	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	DTC	9/2/20	NULL	0.6000876712650799	SULFOBROMOPHTHALEIN	rxcui:10212	SULFOBROMOPHTHALEIN	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.059667808	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	ETOXAZOLE	chembl:CHEMBL1881674	ETOXAZOLE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	CancerCommons	25-Jul-13	inhibitor	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CDH1	hgnc:1748	CDH1	CGI	2/1/22	NULL	1.312691780892362	Bicalutamide	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.01178888	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NCBIGENE:1225	hgnc:10952	SLCO3A1	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:4748	ncit:C47521	ESTROPIPATE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	THIOPHANATE METHYL	chembl:CHEMBL487187	THIOPHANATE METHYL	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	PharmGKB	4/5/24	NULL	0.033701971	polatuzumab vedotin	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1041818873724097	AM-404	iuphar.ligand:12556	AM404	FALSE	FALSE	FALSE
PSME3	hgnc:9570	PSME3	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.1591141552596803	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	PharmGKB	4/5/24	NULL	0.1417211099478933	interferons	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	0.6563458904461813	Dinoprostone	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:11743	drugbank:DB08577	3-[(3-(2-CARBOXYETHYL)-4-METHYLPYRROL-2-YL)METHYLENE]-2-INDOLINONE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	1.040600372117402	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	1.312691780892362	PF-04634817	drugbank:DB14955	PF-04634817	FALSE	FALSE	FALSE
E2F5	hgnc:3119	E2F5	ChEMBL	33	inhibitor	2.187819634820604	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	1.184383561707394	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.029498692	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.010417155	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.017329264	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.038159645	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1491695205559502	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.2778183663264259	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	0.1470803115845784	Gallium nitrate	rxcui:25544	GALLIUM NITRATE	TRUE	FALSE	FALSE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	3.281729452230906	INTERFERON ALFA-N3	rxcui:612937	INTERFERON ALFA-N3	TRUE	TRUE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.039778539	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	GRAMICIDIN S	ncit:C170034	GRAMICIDIN S	FALSE	FALSE	FALSE
CO-STIMULATORY MOLECULE 4-1BB	hgnc:11924	TNFRSF9	TTD	2020.06.01	NULL	78.76150685354175	Urelumab	ncit:C62449	URELUMAB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	TCMDC-125784	chembl:CHEMBL581574	CHEMBL:CHEMBL581574	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	PharmGKB	4/5/24	NULL	0.091796628	flunitrazepam	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.1252170220247087	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.008728004	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2875	hgnc:4552	GPT	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8608	iuphar.ligand:8608	ABL127	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	0.9723642821424906	HYDROFLUMETHIAZIDE	rxcui:5495	HYDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	NALMEFENE	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.016027983	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
NCBIGENE:2130	hgnc:3508	EWSR1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8047	iuphar.ligand:8047	WZ4003	FALSE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	ChEMBL	33	inhibitor	17.50255707856483	ONABOTULINUMTOXINA	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CancerCommons	25-Jul-13	antibody	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.066213961	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.056368944	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9	hgnc:20001	PCSK9	TTD	2020.06.01	NULL	4.039051633514961	REGN-727	rxcui:1659152	ALIROCUMAB	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.8468979231563628	DIMENHYDRINATE	rxcui:3444	DIMENHYDRINATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.059532507	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.087512785	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.012137696	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
CYB5R1	hgnc:13397	CYB5R1	PharmGKB	4/5/24	NULL	0.9546849315580819	primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 3A	hgnc:8778	PDE3A	TTD	2020.06.01	NULL	0.6819178082557726	Cilostazol	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FLUROGESTONE ACETATE	ncit:C77013	FLUROGESTONE ACETATE	FALSE	FALSE	FALSE
PISD	hgnc:8999	PISD	TALC	12-May-16	antibody	52.50767123569449	BAVITUXIMAB	ncit:C49088	BAVITUXIMAB	FALSE	FALSE	TRUE
PLAT	hgnc:9051	PLAT	NCI	14-Sep-17	NULL	0.1735790784651057	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	GLYCINE	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.034658529	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
CD80	hgnc:1700	CD80	ChEMBL	33	inhibitor	13.12691780892362	GALIXIMAB	ncit:C26447	GALIXIMAB	FALSE	FALSE	FALSE
ITGA4	hgnc:6140	ITGA4	ChEMBL	33	inhibitor	3.889457128569962	FIRATEGRAST	ncit:C76692	FIRATEGRAST	FALSE	FALSE	FALSE
RPL35A	hgnc:10345	RPL35A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.1539814405738841	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.057700738	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.011435427	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	antibody	2.972132334095915	CIXUTUMUMAB	ncit:C79828	CIXUTUMUMAB	FALSE	TRUE	TRUE
CSMD1	hgnc:14026	CSMD1	PharmGKB	4/5/24	NULL	0.5385402178019948	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.4773424657790409	JNJ-40346527	ncit:C101519	EDICOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:12974	iuphar.ligand:12974	MW01	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:1917	iuphar.ligand:1917	CICAPROST	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	0.9211872146613068	IUPHAR.LIGAND:1394	iuphar.ligand:1394	LY379268	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	LY-320135	iuphar.ligand:742	LY320135	FALSE	FALSE	FALSE
TMEM8A	hgnc:17205	PGAP6	PharmGKB	4/5/24	NULL	1.750255707856483	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	0.3394892536790592	PEGINTERFERON ALFA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.086551106	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
NCBIGENE:2339	hgnc:3782	FNTA	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10710	iuphar.ligand:10710	IPTACOPAN	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.6035364509849942	HYDROXYCAMPTOTHECIN	chembl:CHEMBL273862	HYDROXYCAMPTOTHECIN	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.099446347	METHIOTHEPIN MESYLATE	chembl:CHEMBL1256737	METHIOTHEPIN MESYLATE	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	DTC	9/2/20	NULL	1.400204566285186	SILYDIANIN	chembl:CHEMBL2397733	SILIDIANIN	FALSE	FALSE	FALSE
MTNR1B	hgnc:7464	MTNR1B	ChEMBL	33	agonist	10.50153424713889	RAMELTEON	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.054695491	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.09745299	NANDROLONE DECANOATE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:9725	ncit:C152764	TROPIFEXOR	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2984	iuphar.ligand:2984	COMPOUND 9 [PMID: 1992149]	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8225	iuphar.ligand:8225	1-METHYL-L-TRYPTOPHAN	FALSE	FALSE	FALSE
NCBIGENE:2285	hgnc:3717	FKBP1AP4	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:9600	iuphar.ligand:9600	MIVAVOTINIB	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	JWH-015	iuphar.ligand:5558	JWH015	FALSE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	PharmGKB	4/5/24	NULL	0.2592971419046642	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005308631	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	4.375639269641208	TCMDC-123910	chembl:CHEMBL528068	CHEMBL:CHEMBL528068	FALSE	FALSE	FALSE
REGENERATING HUMAN PRO-ISLET PEPTIDE	hgnc:8601	REG3A	TTD	2020.06.01	NULL	26.25383561784724	HIP-2B	chembl:CHEMBL4297978	BTI-410	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	PROTHIOFOS	chembl:CHEMBL1560680	PROTHIOFOS	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.3723948314588262	calcium channel blockers	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	0.1389091831632129	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.081092929	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.060984519	IUPHAR.LIGAND:2881	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	GW9662	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001461795	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
CCR6	hgnc:1607	CCR6	DTC	9/2/20	NULL	0.5645986154375753	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.014024485	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	QUAZINONE	ncit:C74347	QUAZINONE	FALSE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.1346350544504987	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	STANOLONE	ncit:C72098	STANOLONE	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.017444409	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.6945459158160648	NECITUMUMAB	rxcui:1723738	NECITUMUMAB	TRUE	TRUE	TRUE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.1744440904840348	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.071341945	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1422	iuphar.ligand:1422	CDPPB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	tipranavir	rxcui:190548	TIPRANAVIR	TRUE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	1.944728564284981	MACIMORELIN	rxcui:1999420	MACIMORELIN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.1374546367426557	LXH254	chembl:CHEMBL4583691	LXH254	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	0.9010915075351876	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.064033745	PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.6945459158160648	NECITUMUMAB	rxcui:1723738	NECITUMUMAB	TRUE	TRUE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.2465148884304905	DICLOXACILLIN	rxcui:3356	DICLOXACILLIN	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.005366139	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ME3	hgnc:6985	ME3	PharmGKB	4/5/24	NULL	0.4268916360625569	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inverse agonist	0.1411496538593938	EBASTINE	rxcui:23796	EBASTINE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	0.1816874437221263	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6122	iuphar.ligand:6122	GALP(3-32) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8071	iuphar.ligand:8071	GNF-5837	FALSE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1870	iuphar.ligand:1870	PRRP-(24-31) (HUMAN)	FALSE	FALSE	FALSE
PSORS1C3	hgnc:17203	PSORS1C3	PharmGKB	4/5/24	NULL	0.7143900848393808	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004149492	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
CAMK1	hgnc:1459	CAMK1	DTC	9/2/20	NULL	0.6250913242344582	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.015268296	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.05293112	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	ICILLIN	iuphar.ligand:2429	ICILIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016959842	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	0.1640864726115453	Peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	12-EPISCALARIN	chembl:CHEMBL269105	CHEMBL:CHEMBL269105	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.2734774543525755	THERAPEUTIC TUMOR INFILTRATING LYMPHOCYTES	ncit:C28699	THERAPEUTIC TUMOR INFILTRATING LYMPHOCYTES	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.1337207247088994	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
UNIPROT:Q14957	hgnc:4587	GRIN2C	TdgClinicalTrial	Jan-14	NULL	0.094099769	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.019304291	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.061412481	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:7793	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:4618	iuphar.ligand:4618	(R)-NFPS	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8172	iuphar.ligand:8172	COMPOUND 7 [PMID: 22464456]	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	TALC	12-May-16	inhibitor	0.2869271652223742	RAMUCIRUMAB	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
THPO	hgnc:11795	THPO	NCI	14-Sep-17	NULL	0.059297201	PROSTAGLANDIN E1	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	TRIDIHEXETHYL CHLORIDE	rxcui:54421	TRIDIHEXETHYL CHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1111665587205952	HYDROMORPHONE HYDROCHLORIDE	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P32970	hgnc:11937	CD70	TdgClinicalTrial	Jan-14	NULL	8.078103267029922	MDX-1203	ncit:C84855	ANTI-CD70 ANTIBODY-DRUG CONJUGATE MDX-1203	FALSE	FALSE	FALSE
NBEA	hgnc:7648	NBEA	PharmGKB	4/5/24	NULL	1.346350544504987	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SLC15A1	hgnc:10920	SLC15A1	NCI	14-Sep-17	NULL	3.500511415712966	ACYCLOVIR	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	3.500511415712966	TIVANTINIB	ncit:C62437	TIVANTINIB	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.010742159	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.182318303	LISDEXAMFETAMINE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:11751	iuphar.ligand:11751	JNJ-67569762	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.026045472	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.023295329	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:8275	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
RPL29	hgnc:10331	RPL29	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	BETA-CCM	chembl:CHEMBL453066	BETA-CCM	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00655895	ZIDOVUDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.025993897	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	0.7001022831425934	Artemether	rxcui:18343	ARTEMETHER	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1988926940746003	BROMOXYNIL	chembl:CHEMBL453905	BROMOXYNIL	FALSE	FALSE	FALSE
BTC	hgnc:1121	BTC	PharmGKB	4/5/24	NULL	0.3281729452230906	panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.002286123	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
SLC5A1	hgnc:11036	SLC5A1	NCI	14-Sep-17	NULL	0.4565884455277782	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.039531467	Iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004426918	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
ALDH5A1	hgnc:408	ALDH5A1	ChEMBL	33	inhibitor	0.6579908676152193	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
NCBIGENE:386	hgnc:18866	KCNT2	GuideToPharmacology	2024.1	blocker	0.8751278539282418	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
B2 BRADYKININ RECEPTOR	hgnc:1030	BDKRB2	TTD	2020.06.01	NULL	1.093909817410302	BRADYKININ	drugbank:DB12126	BRADYKININ	FALSE	FALSE	FALSE
UNIPROT:P18084	hgnc:6160	ITGB5	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	GLPG0187	ncit:C96223	INTEGRIN RECEPTOR ANTAGONIST GLPG0187	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.023620185	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.034229251	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.4321619031744403	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	0.035430277	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:4057	iuphar.ligand:4057	PAMP-20	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:292	iuphar.ligand:292	NNC 11-1585	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00337822	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.3281729452230906	ETODOLAC	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	2.045753424767318	E5501	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1029562181092049	AC-55649	iuphar.ligand:4055	AC55649	FALSE	FALSE	FALSE
AQP8	hgnc:642	AQP8	NCI	14-Sep-17	NULL	0.1280674908187671	ETHINYLESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.00962384	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	GAMMA-FAGARINE	chembl:CHEMBL252925	GAMMA-FAGARINE	FALSE	FALSE	FALSE
ENDOSIALIN	hgnc:18219	CD248	TTD	2020.06.01	NULL	157.5230137070835	Ontuxizumab	ncit:C82406	ONTUXIZUMAB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	MyCancerGenome	20-Jun-17	inhibitor	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.2273059360852575	CIGLITAZONE	ncit:C72726	CIGLITAZONE	FALSE	FALSE	FALSE
UNIPROT:P29274	hgnc:263	ADORA2A	TEND	1-Aug-11	NULL	0.1534190540122556	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	1.479089330582943	NP-506	chembl:CHEMBL480356	CHEMBL:CHEMBL480356	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	NCI	14-Sep-17	NULL	0.024041974	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	DTC	9/2/20	NULL	10.50153424713889	PF-04457845	drugbank:DB12012	PF-04457845	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003162351	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.012853775	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.5321723436050118	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.043629141	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.3182283105193606	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:771	iuphar.ligand:771	CCL2	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6076	iuphar.ligand:6076	J20 (GALANIN ANALOGUE)	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:5943	iuphar.ligand:5943	CDK/CRK INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2239	hgnc:4452	GPC4	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8117	iuphar.ligand:8117	COMPOUND 31 [PMID: 22902653]	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	1.017590527823536	E7090	ncit:C118672	TASURGRATINIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.037957353	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CETP	hgnc:1869	CETP	PharmGKB	4/5/24	NULL	0.3365876361262467	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
EFR3A	hgnc:28970	EFR3A	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FLUFENACET	chembl:CHEMBL1886718	FLUFENACET	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.043109746	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN CD47	hgnc:1682	CD47	TTD	2020.06.01	NULL	6.563458904461812	CC-90002	ncit:C121211	ANTI-CD47 MONOCLONAL ANTIBODY CC-90002	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:4090	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:1646	ncit:C80576	ENADOLINE	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:9929	iuphar.ligand:9929	XILIERTINIB	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:1804	iuphar.ligand:1804	[ILE5]PTHRP-(1-36) (HUMAN)	FALSE	FALSE	FALSE
ADH1C	hgnc:251	ADH1C	PharmGKB	4/5/24	NULL	0.1372749574789398	naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.011993529	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.004189553	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
APP	hgnc:620	APP	ChEMBL	33	vaccine	0.8078103267029922	AMILOMOTIDE	ncit:C166623	AMILOMOTIDE	FALSE	FALSE	FALSE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.192335792	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.067059606	IUPHAR.LIGAND:377	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.035719504	IUPHAR.LIGAND:5686	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	BRILLIANT GREEN OXALATE	chembl:CHEMBL1789985	BRILLIANT GREEN OXALATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.00414131	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
P2RX3	hgnc:8534	P2RX3	ChEMBL	33	inhibitor	26.25383561784724	GEFAPIXANT	ncit:C166945	GEFAPIXANT	FALSE	FALSE	FALSE
IFNA8	hgnc:5429	IFNA8	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	blocker	0.4861821410712453	TEGOPRAZAN	ncit:C152542	TEGOPRAZAN	FALSE	FALSE	FALSE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.070129236	PAZOPANI	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PTH1R	hgnc:9608	PTH1R	ChEMBL	33	agonist	3.750547945	TERIPARATIDE ACETATE	rxcui:114260	TERIPARATIDE ACETATE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.5738543304447485	NORELGESTROMIN	rxcui:326374	NORELGESTROMIN	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	PROPYLENE GLYCOL MONOSTEARATE	rxcui:1314411	PROPYLENE GLYCOL MONOSTEARATE	TRUE	FALSE	FALSE
INTERLEUKIN 4 RECEPTOR ALPHA	hgnc:6015	IL4R	TTD	2020.06.01	NULL	8.751278539282415	SAR231893	rxcui:1876376	DUPILUMAB	TRUE	FALSE	FALSE
AHRR	hgnc:346	AHRR	PharmGKB	4/5/24	NULL	0.4688184931758437	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
RPL3	hgnc:10332	RPL3	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:11434	iuphar.ligand:11434	[D-TYR6,&BETA;-ALA11,N-ME-ALA13,NLE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:2484	ncbigene:2484	FRV1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6041	iuphar.ligand:6041	SKI II	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:2640	iuphar.ligand:2640	AGN193109	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.036527076	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	IMG-7289	ncit:C131827	BOMEDEMSTAT	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
ME3	hgnc:6985	ME3	NCI	14-Sep-17	NULL	0.1241316104862754	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.596678082	4-HYDROXYESTRADIOL	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	SDZ-201106	chembl:CHEMBL314639	CHEMBL:CHEMBL314639	FALSE	FALSE	FALSE
GSR	hgnc:4623	GSR	ChEMBL	33	other/unknown	1.193356164447602	OXIGLUTATIONE	ncit:C62624	OXIGLUTATIONE	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.2442217266776488	ALTIRATINIB	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.5000730593875666	TEPOTINIB HYDROCHLORIDE	rxcui:2477104	TEPOTINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q09428	hgnc:59	ABCC8	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	MITIGLINIDE	ncit:C81699	MITIGLINIDE	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:9059	iuphar.ligand:9059	PF-04995274	FALSE	FALSE	FALSE
NCBIGENE:2022	hgnc:3349	ENG	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10367	iuphar.ligand:10367	DS21360717	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1169	iuphar.ligand:1169	[GLN8]GNRH	FALSE	FALSE	FALSE
NCBIGENE:1161	hgnc:3439	ERCC8	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:717	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:2038	iuphar.ligand:2038	BIM 23060	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.1403266238077355	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	TOLMETIN SODIUM	rxcui:42935	TOLMETIN SODIUM	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000310535	chembl:CHEMBL602940	CHEMBL:CHEMBL602940	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	2.625383561784724	AMG 853	ncit:C152874	VIDUPIPRANT	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.019418517	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.2628669398532891	felodipine	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.1500219178162699	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	modulator	0.048083948	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
HAMP	hgnc:15598	HAMP	ChEMBL	33	inhibitor	26.25383561784724	LY-2787106	chembl:CHEMBL2109440	LY-2787106	FALSE	FALSE	FALSE
UNIPROT:P11597	hgnc:1869	CETP	TdgClinicalTrial	Jan-14	NULL	6.058577450272442	ANACETRAPIB	ncit:C75251	ANACETRAPIB	FALSE	FALSE	FALSE
UNIPROT:Q96GD4	hgnc:11390	AURKB	TdgClinicalTrial	Jan-14	NULL	0.064413418	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
NR2F2	hgnc:7976	NR2F2	DTC	9/2/20	NULL	2.187819634820604	PYRIDABEN	chembl:CHEMBL225963	PYRIDABEN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	MMV006319	chembl:CHEMBL579105	CHEMBL:CHEMBL579105	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.025256215	durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.044498026	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	UNBS3157	chembl:CHEMBL244268	CHEMBL:CHEMBL244268	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	TCMDC-124327	chembl:CHEMBL581929	CHEMBL:CHEMBL581929	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	0.6731752722524935	RG7129	iuphar.ligand:9821	RO5508887	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.010554306	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.016027983	hydrocortisone	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	CGI	2/1/22	NULL	0.3174882446809434	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
GP	hgnc:18280	RNF130	ChEMBL	33	inhibitor	7.501095891	PORGAVIXIMAB	ncit:C175195	PORGAVIXIMAB	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.095904422	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.2678962818147678	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	ECHOTHIOPHATE IODIDE	rxcui:3740	ECHOTHIOPHATE IODIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.007396488	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	4.773424657790408	Cinalukast	ncit:C96709	CINALUKAST	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	CancerCommons	25-Jul-13	inhibitor	0.4861821410712453	SCH727965	hemonc:160	DINACICLIB	FALSE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	CancerCommons	25-Jul-13	inhibitor	0.3070624048871023	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.017170592	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.5223276196220918	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
EZH2	hgnc:3527	EZH2	CGI	2/1/22	NULL	2.917092846427472	EPZ-6438	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CGI	2/1/22	NULL	0.057841988	Bortezomib	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	0.179119736	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KCNJ5	hgnc:6266	KCNJ5	CGI	2/1/22	NULL	0.1296485709523321	Verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.017643707	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	0.1852122442176172	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	2.100306849	DICHLORPHENAMIDE	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.2386712328895204	4-METHYL-[1,10]PHENANTHROLINE	chembl:CHEMBL316589	CHEMBL:CHEMBL316589	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.016558711	Pramlintide	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1252170220247087	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.7119684235348407	TRANDOLAPRIL	rxcui:38454	TRANDOLAPRIL	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	2.500365296937833	RETEPLASE	rxcui:76895	RETEPLASE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	CLIDINIUM BROMIDE	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	2.917092846427472	METOLAZONE	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	OXPRENOLOL HYDROCHLORIDE	rxcui:203131	OXPRENOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	1.193356164447602	FLUVOXAMINE MALEATE	rxcui:203143	FLUVOXAMINE MALEATE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	CHOLINE FENOFIBRATE	rxcui:1433887	CHOLINE FENOFIBRATE	TRUE	FALSE	FALSE
ILES	NULL	NULL	ChEMBL	33	inhibitor	NULL	MUPIROCIN CALCIUM	rxcui:221128	MUPIROCIN CALCIUM	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	PHENMETRAZINE HYDROCHLORIDE	rxcui:203198	PHENMETRAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CA12	hgnc:1371	CA12	ChEMBL	33	inhibitor	0.7501095890813501	DICHLORPHENAMIDE	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
CA4	hgnc:1375	CA4	ChEMBL	33	inhibitor	1.750255707856483	DICHLORPHENAMIDE	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
TRPM8	hgnc:17961	TRPM8	ChEMBL	33	potentiator	4.836232876971861	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
PTGER3	hgnc:9595	PTGER3	ChEMBL	33	agonist	2.187819634820604	MISOPROSTOL	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
MMP13	hgnc:7159	MMP13	ChEMBL	33	inhibitor	1.640864726115453	DOXYCYCLINE CALCIUM	rxcui:82012	DOXYCYCLINE CALCIUM	TRUE	FALSE	FALSE
MMP8	hgnc:7175	MMP8	ChEMBL	33	inhibitor	1.875273972703375	DOXYCYCLINE CALCIUM	rxcui:82012	DOXYCYCLINE CALCIUM	TRUE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	2.282942227638891	BOSENTAN	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	0.3170753093942904	NICOTINE POLACRILEX	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
SLC22A11	hgnc:18120	SLC22A11	ChEMBL	33	inhibitor	4.773424657790409	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	NALBUPHINE HYDROCHLORIDE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.035145697	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.032412143	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.007621958	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.032055965	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.092606122	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.096167896	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.036237178	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.085239726	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.1534190540122556	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	inhibitor	0.074690855	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	0.094608417	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.2243917574174978	TEGASEROD MALEATE	rxcui:339270	TEGASEROD MALEATE	TRUE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAPENTINE	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAPENTINE	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAPENTINE	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAPENTINE	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	ChEMBL	33	inhibitor	0.5000730593875666	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD3	hgnc:9560	PSMD3	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD7	hgnc:9565	PSMD7	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ADRM1	hgnc:15759	ADRM1	ChEMBL	33	inhibitor	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD6	hgnc:9564	PSMD6	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PBP1A	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN POTASSIUM	rxcui:1299048	HETACILLIN POTASSIUM	TRUE	FALSE	FALSE
PBP1B	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN POTASSIUM	rxcui:1299048	HETACILLIN POTASSIUM	TRUE	FALSE	FALSE
PBP2A	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN POTASSIUM	rxcui:1299048	HETACILLIN POTASSIUM	TRUE	FALSE	FALSE
PBP2B	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN POTASSIUM	rxcui:1299048	HETACILLIN POTASSIUM	TRUE	FALSE	FALSE
PBP2X	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN POTASSIUM	rxcui:1299048	HETACILLIN POTASSIUM	TRUE	FALSE	FALSE
PBP3	NULL	NULL	ChEMBL	33	inhibitor	NULL	HETACILLIN POTASSIUM	rxcui:1299048	HETACILLIN POTASSIUM	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.2273059360852575	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.4167275494896388	ROCURONIUM BROMIDE	rxcui:32521	ROCURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.7501095890813501	TUBOCURARINE CHLORIDE	rxcui:82115	TUBOCURARINE CHLORIDE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.049723174	METHAMPHETAMINE HYDROCHLORIDE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
ATP1A2	hgnc:800	ATP1A2	ChEMBL	33	inhibitor	0.7501095890813501	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
ATP1A4	hgnc:14073	ATP1A4	ChEMBL	33	inhibitor	0.077217164	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
ATP1B1	hgnc:804	ATP1B1	ChEMBL	33	inhibitor	0.081281225	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
ATP1A4	hgnc:14073	ATP1A4	ChEMBL	33	inhibitor	0.2625383561784725	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
FXYD2	hgnc:4026	FXYD2	ChEMBL	33	inhibitor	0.4375639269641209	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
ATP1B2	hgnc:805	ATP1B2	ChEMBL	33	inhibitor	0.2573905452730122	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.033919684	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.045226246	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.039420174	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.064111931	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.037398626	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.037398626	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.085239726	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.034727296	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.087318744	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.019483366	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.016574391	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.013876234	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.014553124	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.014732792	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V POTASSIUM	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V POTASSIUM	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V POTASSIUM	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V POTASSIUM	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V POTASSIUM	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V POTASSIUM	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V POTASSIUM	rxcui:203195	PENICILLIN V POTASSIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME AXETIL	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME AXETIL	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME AXETIL	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME AXETIL	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME AXETIL	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME AXETIL	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME AXETIL	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOGLYCIN	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOGLYCIN	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOGLYCIN	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOGLYCIN	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOGLYCIN	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOGLYCIN	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALOGLYCIN	ncit:C65307	CEPHALOGLYCIN	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPROZIL	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPROZIL	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPROZIL	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPROZIL	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPROZIL	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPROZIL	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPROZIL	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOPERAZONE SODIUM	rxcui:227214	CEFOPERAZONE SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOPERAZONE SODIUM	rxcui:227214	CEFOPERAZONE SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOPERAZONE SODIUM	rxcui:227214	CEFOPERAZONE SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOPERAZONE SODIUM	rxcui:227214	CEFOPERAZONE SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOPERAZONE SODIUM	rxcui:227214	CEFOPERAZONE SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOPERAZONE SODIUM	rxcui:227214	CEFOPERAZONE SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOPERAZONE SODIUM	rxcui:227214	CEFOPERAZONE SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIRAMIDE SODIUM	ncit:C65304	CEFPIRAMIDE SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIRAMIDE SODIUM	ncit:C65304	CEFPIRAMIDE SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIRAMIDE SODIUM	ncit:C65304	CEFPIRAMIDE SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIRAMIDE SODIUM	ncit:C65304	CEFPIRAMIDE SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIRAMIDE SODIUM	ncit:C65304	CEFPIRAMIDE SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIRAMIDE SODIUM	ncit:C65304	CEFPIRAMIDE SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIRAMIDE SODIUM	ncit:C65304	CEFPIRAMIDE SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAROLINE FOSAMIL ACETATE	rxcui:1743286	CEFTAROLINE FOSAMIL ACETATE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAROLINE FOSAMIL ACETATE	rxcui:1743286	CEFTAROLINE FOSAMIL ACETATE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAROLINE FOSAMIL ACETATE	rxcui:1743286	CEFTAROLINE FOSAMIL ACETATE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAROLINE FOSAMIL ACETATE	rxcui:1743286	CEFTAROLINE FOSAMIL ACETATE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAROLINE FOSAMIL ACETATE	rxcui:1743286	CEFTAROLINE FOSAMIL ACETATE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAROLINE FOSAMIL ACETATE	rxcui:1743286	CEFTAROLINE FOSAMIL ACETATE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAROLINE FOSAMIL ACETATE	rxcui:1743286	CEFTAROLINE FOSAMIL ACETATE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN DISODIUM	rxcui:258332	CARBENICILLIN DISODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN DISODIUM	rxcui:258332	CARBENICILLIN DISODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN DISODIUM	rxcui:258332	CARBENICILLIN DISODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN DISODIUM	rxcui:258332	CARBENICILLIN DISODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN DISODIUM	rxcui:258332	CARBENICILLIN DISODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN DISODIUM	rxcui:258332	CARBENICILLIN DISODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN DISODIUM	rxcui:258332	CARBENICILLIN DISODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLACILLIN	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLACILLIN	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLACILLIN	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLACILLIN	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLACILLIN	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLACILLIN	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLACILLIN	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEZLOCILLIN SODIUM	rxcui:82048	MEZLOCILLIN SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEZLOCILLIN SODIUM	rxcui:82048	MEZLOCILLIN SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEZLOCILLIN SODIUM	rxcui:82048	MEZLOCILLIN SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEZLOCILLIN SODIUM	rxcui:82048	MEZLOCILLIN SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEZLOCILLIN SODIUM	rxcui:82048	MEZLOCILLIN SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEZLOCILLIN SODIUM	rxcui:82048	MEZLOCILLIN SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEZLOCILLIN SODIUM	rxcui:82048	MEZLOCILLIN SODIUM	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	blocker	0.1262203635473425	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	blocker	0.2243917574174979	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.046965717	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	blocker	0.2243917574174979	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NOVOBIOCIN SODIUM	rxcui:82057	NOVOBIOCIN SODIUM	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NOVOBIOCIN SODIUM	rxcui:82057	NOVOBIOCIN SODIUM	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.040051618	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.054695491	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.01924768	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.1235474617310458	OLANZAPINE PAMOATE	rxcui:1294588	OLANZAPINE PAMOATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.041508041	OLANZAPINE PAMOATE	rxcui:1294588	OLANZAPINE PAMOATE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.1000146118775133	LOXAPINE HYDROCHLORIDE	rxcui:91138	LOXAPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	FIDAXOMICIN	rxcui:1111103	FIDAXOMICIN	TRUE	FALSE	FALSE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	FIDAXOMICIN	rxcui:1111103	FIDAXOMICIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME2	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG1	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG2	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG3	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPME2	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMJ2	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
KCNA10	hgnc:6219	KCNA10	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNH5	hgnc:6254	KCNH5	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNC4	hgnc:6236	KCNC4	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNA7	hgnc:6226	KCNA7	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNS1	hgnc:6300	KCNS1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNS2	hgnc:6301	KCNS2	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	blocker	0.091476779	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEDIPASVIR	rxcui:1591922	LEDIPASVIR	TRUE	FALSE	FALSE
CYP51A	NULL	NULL	ChEMBL	33	inhibitor	NULL	ISAVUCONAZONIUM SULFATE	rxcui:1608321	ISAVUCONAZONIUM SULFATE	TRUE	FALSE	FALSE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	0.1930429089547591	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	modulator	0.1037701012563132	CARIPRAZINE HYDROCHLORIDE	rxcui:1721073	CARIPRAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SSTR3	hgnc:11332	SSTR3	ChEMBL	33	agonist	1.458546423213736	PASIREOTIDE PAMOATE	rxcui:1597818	PASIREOTIDE PAMOATE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.5000730593875666	BMS-698769	chembl:CHEMBL3545299	BMS-698769	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.2027323213733378	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.09869863	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.1785975212098452	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.1630673019742065	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	0.6563458904461813	ALTIRATINIB	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
MAP3K5	hgnc:6857	MAP3K5	ChEMBL	33	inhibitor	26.25383561784724	SELONSERTIB	ncit:C121943	SELONSERTIB	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.1000146118775133	ALTIRATINIB	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.201952582	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	2.800409132570373	GSK-1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.7395446652914718	DS-3078A	chembl:CHEMBL3544963	DS-3078A	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.052090944	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.6269572684859045	GSK-1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1682938180631233	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.030386384	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.050488145	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1223955040459079	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1363835616511545	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.2966535098061835	TTP-607	chembl:CHEMBL3545327	TTP-607	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.7160136986685613	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	1.166837138570988	TTP-607	chembl:CHEMBL3545327	TTP-607	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.030386384	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	0.6908904109959803	XL-844	chembl:CHEMBL3544936	XL-844	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.031479419	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1041818873724097	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	0.5048814541893701	SAD448	chembl:CHEMBL2397751	SAD448	FALSE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.2651902587661338	GS 6201	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	modulator	0.2075402025126264	ORDOPIDINE	ncit:C166429	ORDOPIDINE	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	5.527123287967842	MK-7246	chembl:CHEMBL561132	MK-7246	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.064624826	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.066676408	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1333528158366844	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.049302978	LUCITANIB	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.08334551	LUCITANIB	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.2944355396394084	LUCITANIB	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.6050266644442165	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
MAPK9	hgnc:6886	MAPK9	ChEMBL	33	inhibitor	0.546954909	CC-401	drugbank:DB12432	CC-401	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	ChEMBL	33	inhibitor	0.6863747873946993	CC-401	drugbank:DB12432	CC-401	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.2778183663264258	AFURESERTIB	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.2381300282797936	ACALISIB	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	1.141471113819445	DECERNOTINIB	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	modulator	5.834185692854944	AZD2066	drugbank:DB17078	AZD2066	FALSE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	ChEMBL	33	inhibitor	4.375639269641208	ANATIBANT	ncit:C79554	ANATIBANT	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	inhibitor	6.177373086552294	BARUSIBAN	ncit:C90866	BARUSIBAN	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.2734774543525755	DABUZALGRON	ncit:C75036	DABUZALGRON	FALSE	FALSE	FALSE
NPY5R	hgnc:7958	NPY5R	ChEMBL	33	inhibitor	7.501095891	S-237648	chembl:CHEMBL3545038	S-237648	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	1.141471113819445	ENRASENTAN	ncit:C87727	ENRASENTAN	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	1.280674908	SB-705498	drugbank:DB11883	SB-705498	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.2983390411119005	AZD7009	chembl:CHEMBL3545040	AZD7009	FALSE	FALSE	FALSE
SCNN1B	hgnc:10600	SCNN1B	ChEMBL	33	blocker	2.187819634820604	IDREVLORIDE	ncit:C184934	IDREVLORIDE	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.458546423213736	TEBANICLINE TOSYLATE	ncit:C75076	TEBANICLINE TOSYLATE	FALSE	FALSE	FALSE
PTGDR	hgnc:9591	PTGDR	ChEMBL	33	inhibitor	2.625383561784724	VIDUPIPRANT	ncit:C152874	VIDUPIPRANT	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1162317016838838	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.2991890098899972	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	ChEMBL	33	inhibitor	0.045579576	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	0.7095631248066824	APADENOSON	ncit:C74246	APADENOSON	FALSE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	1.250182648468916	DARUSENTAN	ncit:C75991	DARUSENTAN	FALSE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	ChEMBL	33	inhibitor	8.751278539282417	FARLETUZUMAB	ncit:C61503	FARLETUZUMAB	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOTAVIZUMAB	ncit:C88584	MOTAVIZUMAB	FALSE	FALSE	FALSE
BSG	hgnc:1116	BSG	ChEMBL	33	other/unknown	13.12691780892362	GAVILIMOMAB	ncit:C2621	GAVILIMOMAB	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	inhibitor	0.5834185692854945	VISILIZUMAB	ncit:C2229	VISILIZUMAB	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.5645986154375752	AFELIMOMAB	ncit:C166960	AFELIMOMAB	FALSE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	modulator	0.2243917574174979	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	modulator	0.2243917574174979	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	modulator	0.046965717	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	agonist	0.05309168	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	modulator	0.042968634	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	agonist	0.056368944	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	blocker	0.1312691780892362	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
KCNG3	hgnc:18306	KCNG3	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNS3	hgnc:6302	KCNS3	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNV2	hgnc:19698	KCNV2	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	agonist	0.1848861663228679	TELBERMIN	ncit:C152544	TELBERMIN	FALSE	FALSE	FALSE
KCNB1	hgnc:6231	KCNB1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNV1	hgnc:18861	KCNV1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.062808219	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	ChEMBL	33	inhibitor	2.917092846427472	VARESPLADIB METHYL	ncit:C152833	VARESPLADIB METHYL	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.042174836	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	inhibitor	3.281729452230906	IBALIZUMAB	rxcui:2043283	IBALIZUMAB	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.4234489615781814	ZONAMPANEL	ncit:C152963	ZONAMPANEL	FALSE	FALSE	FALSE
IL9	hgnc:6029	IL9	ChEMBL	33	inhibitor	17.50255707856483	ENOKIZUMAB	ncit:C97929	ENOKIZUMAB	FALSE	FALSE	FALSE
LTA	hgnc:6709	LTA	ChEMBL	33	inhibitor	6.563458904461812	BAMINERCEPT	ncit:C96762	BAMINERCEPT ALFA	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	1.750255707856483	TADOCIZUMAB	ncit:C88626	TADOCIZUMAB	FALSE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	PRO-542	drugbank:DB05793	PRO-542	FALSE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	ChEMBL	33	inhibitor	3.621218705909965	DAPIROLIZUMAB PEGOL	ncit:C174737	DAPIROLIZUMAB PEGOL	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	ChEMBL	33	inhibitor	2.187819634820604	BUTAMBEN PICRATE	rxcui:221067	BUTAMBEN PICRATE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.079557078	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.028413242	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.091796628	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.1056492378987816	MOXISYLYTE	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAMETHOXYPYRIDAZINE	rxcui:10181	SULFAMETHOXYPYRIDAZINE	TRUE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	ChEMBL	33	inhibitor	0.596678082	PROGLUMIDE	rxcui:8730	PROGLUMIDE	TRUE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	inhibitor	1.750255707856483	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	PYROVALERONE HYDROCHLORIDE	ncit:C73830	PYROVALERONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
HA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DIRIDAVUMAB	ncit:C169915	DIRIDAVUMAB	FALSE	FALSE	FALSE
M	NULL	NULL	ChEMBL	33	inhibitor	NULL	TCN-032	chembl:CHEMBL2109619	TCN-032	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	inhibitor	1.458546423213736	HOKT3	chembl:CHEMBL2109253	HOKT3	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	IMGATUZUMAB	ncit:C78838	IMGATUZUMAB	FALSE	FALSE	FALSE
TXNRD1	hgnc:12437	TXNRD1	ChEMBL	33	inhibitor	2.500365296937833	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
CD79B	hgnc:1699	CD79B	ChEMBL	33	binder	1.381780822	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	DEXKETOPROFEN	rxcui:237162	DEXKETOPROFEN	TRUE	FALSE	FALSE
UREB	NULL	NULL	ChEMBL	33	inhibitor	NULL	EBROTIDINE	ncit:C77440	EBROTIDINE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.085796848	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELAFLOXACIN MEGLUMINE	rxcui:1927662	DELAFLOXACIN MEGLUMINE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELAFLOXACIN MEGLUMINE	rxcui:1927662	DELAFLOXACIN MEGLUMINE	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	GLECAPREVIR	rxcui:1940635	GLECAPREVIR	TRUE	FALSE	FALSE
PAGA	hgnc:9352	PRDX1	ChEMBL	33	inhibitor	8.751278539282415	AVP-21D9	drugbank:DB17798	AVP-21D9	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	4.565884455277782	PLOZALIZUMAB	ncit:C88308	PLOZALIZUMAB	FALSE	FALSE	FALSE
TCDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ACTOXUMAB	ncit:C169762	ACTOXUMAB	FALSE	FALSE	FALSE
NOTCH1	hgnc:7881	NOTCH1	ChEMBL	33	inhibitor	19.69037671338543	BRONTICTUZUMAB	ncit:C103274	BRONTICTUZUMAB	FALSE	FALSE	TRUE
TPBG	hgnc:12004	TPBG	ChEMBL	33	modulator	10.50153424713889	NACOLOMAB TAFENATOX	ncit:C29328	NACOLOMAB TAFENATOX	FALSE	FALSE	FALSE
RPS9	hgnc:10442	RPS9	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006811217	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPS6	hgnc:10429	RPS6	ChEMBL	33	inhibitor	0.1093909817410302	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL8	hgnc:10368	RPL8	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS28	hgnc:10418	RPS28	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	HNK20	chembl:CHEMBL2109568	HNK20	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELAFLOXACIN MEGLUMINE	rxcui:1927662	DELAFLOXACIN MEGLUMINE	TRUE	FALSE	FALSE
RPL34	hgnc:10340	RPL34	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	DELAFLOXACIN MEGLUMINE	rxcui:1927662	DELAFLOXACIN MEGLUMINE	TRUE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.043756393	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
RPL30	hgnc:10333	RPL30	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL37A	hgnc:10348	RPL37A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.020257589	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	blocker	0.069454592	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2500365296937833	GLESATINIB	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	blocker	0.089298761	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNH7	hgnc:18863	KCNH7	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCND1	hgnc:6237	KCND1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNA6	hgnc:6225	KCNA6	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNH3	hgnc:6252	KCNH3	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNC1	hgnc:6233	KCNC1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	agonist	0.305277158	CENEGERMIN	rxcui:2104331	CENEGERMIN-BKBJ	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL	rxcui:2265702	CEFIDEROCOL	TRUE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.9053046764774912	SJ000290256	chembl:CHEMBL590666	CHEMBL:CHEMBL590666	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL	rxcui:2265702	CEFIDEROCOL	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL	rxcui:2265702	CEFIDEROCOL	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL	rxcui:2265702	CEFIDEROCOL	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL	rxcui:2265702	CEFIDEROCOL	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL	rxcui:2265702	CEFIDEROCOL	TRUE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.921012362281506	TISAGENLECLEUCEL	rxcui:1986438	TISAGENLECLEUCEL	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.03591496	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2917092846427472	DROTAVERINE	rxcui:23684	DROTAVERIN	FALSE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.088248187	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.035098711	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GARENOXACIN MESYLATE	ncit:C65801	GARENOXACIN MESYLATE	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GARENOXACIN MESYLATE	ncit:C65801	GARENOXACIN MESYLATE	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	GARENOXACIN MESYLATE	ncit:C65801	GARENOXACIN MESYLATE	FALSE	FALSE	FALSE
RPS11	hgnc:10384	RPS11	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	PHENAZINE-2,3-DIAMINE	chembl:CHEMBL274921	CHEMBL:CHEMBL274921	FALSE	FALSE	FALSE
RPL9P8	hgnc:30334	RPL9P8	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL27	hgnc:10328	RPL27	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS21	hgnc:10409	RPS21	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	GNF-PF-3542	chembl:CHEMBL598477	CHEMBL:CHEMBL598477	FALSE	FALSE	FALSE
RPL18A	hgnc:10311	RPL18A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL26	hgnc:10327	RPL26	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL8	hgnc:10368	RPL8	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	THIAMYLAL SODIUM	rxcui:203201	THIAMYLAL SODIUM	TRUE	FALSE	FALSE
RPL28	hgnc:10330	RPL28	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
PB2	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAVIPIRAVIR	ncit:C81605	FAVIPIRAVIR	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
CETP	hgnc:1869	CETP	ChEMBL	33	inhibitor	4.039051633514961	ROCACETRAPIB	ncit:C170369	ROCACETRAPIB	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.2917092846427472	AMORFRUTIN A	chembl:CHEMBL491820	AMORFRUTIN A	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.2500365296937833	LERCANIDIPINE HYDROCHLORIDE	rxcui:153679	LERCANIDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
L	NULL	NULL	ChEMBL	33	inhibitor	NULL	LUMICITABINE	ncit:C174641	LUMICITABINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	MALEIC ACID	rxcui:1426330	MALEIC ACID	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIVAMPICILLIN	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.4817217544559128	CP-866087	drugbank:DB12196	CP-866087	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	CAPRAVIRINE	ncit:C81612	CAPRAVIRINE	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	2.442217266776488	ABT-639	drugbank:DB15055	ABT-639	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	modulator	2.423430980108977	TRAMIPROSATE	rxcui:1374845	TRAMIPROSATE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	binder	1.029562181092049	CAMIDANLUMAB TESIRINE	ncit:C121949	CAMIDANLUMAB TESIRINE	FALSE	FALSE	FALSE
KLRC1	hgnc:6374	KLRC1	ChEMBL	33	inhibitor	105.0153424713889	MONALIZUMAB	ncit:C120208	MONALIZUMAB	FALSE	FALSE	FALSE
HLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUVRATOXUMAB	ncit:C152484	SUVRATOXUMAB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.729273212	VERICIGUAT	rxcui:2475830	VERICIGUAT	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2983390411119005	LOTAMILAST	ncit:C170131	LOTAMILAST	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2917092846427472	TRANIMILAST	ncit:C171863	TRANIMILAST	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.3125456621172291	TRANIMILAST	ncit:C171863	TRANIMILAST	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.596678082	TOFIMILAST	ncit:C76891	TOFIMILAST	FALSE	FALSE	FALSE
RPS9	hgnc:10442	RPS9	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS7	hgnc:10440	RPS7	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL21	hgnc:10313	RPL21	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.01635753	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
RPS20	hgnc:10405	RPS20	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL9P8	hgnc:30334	RPL9P8	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	5-(4-PHENYLBUTOXY)PSORALEN	iuphar.ligand:9583	PSORA-4	FALSE	FALSE	FALSE
RPL6	hgnc:10362	RPL6	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL4	hgnc:10353	RPL4	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.005007407	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
RPL27A	hgnc:10329	RPL27A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL35	hgnc:10344	RPL35	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENAMECILLIN	ncit:C170307	PENAMECILLIN	TRUE	FALSE	FALSE
TLR2	hgnc:11848	TLR2	DTC	9/2/20	NULL	7.501095891	2-PALMITAMIDOHEXADECANOIC ACID	chembl:CHEMBL1836411	CHEMBL:CHEMBL1836411	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENAMECILLIN	ncit:C170307	PENAMECILLIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENAMECILLIN	ncit:C170307	PENAMECILLIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENAMECILLIN	ncit:C170307	PENAMECILLIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENAMECILLIN	ncit:C170307	PENAMECILLIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENAMECILLIN	ncit:C170307	PENAMECILLIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENAMECILLIN	ncit:C170307	PENAMECILLIN	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
HA	NULL	NULL	ChEMBL	33	binder	NULL	MEDI-8852	chembl:CHEMBL4298034	MEDI-8852	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	negative modulator	0.8078103267029922	DONANEMAB	ncit:C166484	DONANEMAB	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	negative modulator	NULL	BECLABUVIR	ncit:C114983	BECLABUVIR	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	S-1360	chembl:CHEMBL218227	S-1360	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	2.917092846427472	CAPROMORELIN	rxcui:1986787	CAPROMORELIN	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	ADAFOSBUVIR	ncit:C169763	ADAFOSBUVIR	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NADIFLOXACIN	ncit:C166927	NADIFLOXACIN	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NADIFLOXACIN	ncit:C166927	NADIFLOXACIN	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NADIFLOXACIN	ncit:C166927	NADIFLOXACIN	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PEFLOXACIN	rxcui:7960	PEFLOXACIN	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.2282942227638891	GUSACITINIB	ncit:C166736	GUSACITINIB	FALSE	FALSE	FALSE
GRM4	hgnc:4596	GRM4	ChEMBL	33	positive modulator	7.501095891	FOLIGLURAX	ncit:C170000	FOLIGLURAX	FALSE	FALSE	FALSE
CTSC	hgnc:2528	CTSC	ChEMBL	33	inhibitor	7.501095891	BRENSOCATIB	ncit:C171778	BRENSOCATIB	FALSE	FALSE	FALSE
FABI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AFABICIN	ncit:C169766	AFABICIN	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	2.019525817	S-777469	drugbank:DB16321	S-777469	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	ChEMBL	33	inhibitor	0.4730420832044549	TILARGININE ACETATE	ncit:C90899	TILARGININE ACETATE	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	ChEMBL	33	inhibitor	0.2465148884304905	TILARGININE ACETATE	ncit:C90899	TILARGININE ACETATE	FALSE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	ChEMBL	33	inhibitor	13.12691780892362	ISPINESIB	ncit:C38131	ISPINESIB	FALSE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.5427149481725528	PROCATEROL	rxcui:34530	PROCATEROL	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	0.6250913242344582	PAMIPARIB	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.075333818	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
E2F7	hgnc:23820	E2F7	ChEMBL	33	inhibitor	2.187819634820604	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	ChEMBL	33	inhibitor	4.039051633514961	BELNACASAN	ncit:C171755	BELNACASAN	FALSE	FALSE	FALSE
TCDA	NULL	NULL	ChEMBL	33	binder	NULL	TOLEVAMER POTASSIUM SODIUM	ncit:C152682	TOLEVAMER POTASSIUM SODIUM	FALSE	FALSE	FALSE
TCDB	NULL	NULL	ChEMBL	33	binder	NULL	TOLEVAMER POTASSIUM SODIUM	ncit:C152682	TOLEVAMER POTASSIUM SODIUM	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	1.071585127259071	BEMIPARIN	rxcui:280611	BEMIPARIN	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	2.019525817	IZOKIBEP	ncit:C175101	IZOKIBEP	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.3547815624033412	REPINOTAN	ncit:C74388	REPINOTAN	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	0.7955707762984014	LEUPROLIDE MESYLATE	rxcui:2595041	LEUPROLIDE MESYLATE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.1666910197958555	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	0.1861974157294131	TEGAFUR	rxcui:10995	URACIL	TRUE	FALSE	TRUE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	SAMATASVIR	ncit:C152292	SAMATASVIR	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	2.187819634820604	K-134	drugbank:DB12685	K-134	FALSE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	1.591141552596802	ENOXIMONE	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
HLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOSATOXUMAB	ncit:C152701	TOSATOXUMAB	FALSE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.9723642821424906	ONZIGOLIDE	ncit:C88345	ONZIGOLIDE	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ZABOFLOXACIN	ncit:C82232	ZABOFLOXACIN	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEBTELOVIMAB	rxcui:2592360	BEBTELOVIMAB	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	ZABOFLOXACIN	ncit:C82232	ZABOFLOXACIN	FALSE	FALSE	FALSE
GROEL2	NULL	NULL	ChEMBL	33	vaccine	NULL	VERPASEP CALTESPEN	ncit:C2811	VERPASEP CALTESPEN	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	UPRIFOSBUVIR	ncit:C152805	UPRIFOSBUVIR	FALSE	FALSE	FALSE
UTRN	hgnc:12635	UTRN	ChEMBL	33	modulator	26.25383561784724	EZUTROMID	ncit:C166897	EZUTROMID	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	CS-1003	chembl:CHEMBL4594536	CS-1003	FALSE	FALSE	FALSE
RGMA	hgnc:30308	RGMA	ChEMBL	33	inhibitor	26.25383561784724	UNASNEMAB	ncit:C179131	UNASNEMAB	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
LAG3	hgnc:6476	LAG3	ChEMBL	33	vaccine	6.563458904461812	EFTILAGIMOD ALFA	ncit:C62509	EFTILAGIMOD ALPHA	FALSE	FALSE	FALSE
HBCAG	NULL	NULL	ChEMBL	33	inhibitor	NULL	VEBICORVIR	ncit:C175206	VEBICORVIR	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	1.693795846312725	MEQUITAZINE	rxcui:29528	MEQUITAZINE	TRUE	FALSE	FALSE
TNFSF14	hgnc:11930	TNFSF14	ChEMBL	33	inhibitor	26.25383561784724	QUISOVALIMAB	ncit:C184870	QUISOVALIMAB	FALSE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	4.039051633514961	LERODALCIBEP	ncit:C175808	LERODALCIBEP	FALSE	FALSE	FALSE
THYA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PEMETREXED TROMETHAMINE	ncit:C170306	PEMETREXED TROMETHAMINE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.093763699	XYLOMETAZOLINE	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.061055432	XYLOMETAZOLINE	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.054695491	XYLOMETAZOLINE	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.1479089330582944	XYLOMETAZOLINE	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
GART	hgnc:4163	GART	ChEMBL	33	inhibitor	0.6403374540938354	PEMETREXED TROMETHAMINE	ncit:C170306	PEMETREXED TROMETHAMINE	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3860858179095183	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
ATR	hgnc:882	ATR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1458546423213736	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.017664481	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CCND3	hgnc:1585	CCND3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.4286340509036285	PD 0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CCNE1	hgnc:1589	CCNE1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1166837138570988	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.031555091	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.042073455	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.205692444	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.093763699	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
NF1	hgnc:7765	NF1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2075402025126264	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.016352436	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.026789628	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3070624048871023	CS1229	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.039390601	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.070197421	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	COSMIC	4-Sep-20	NULL	0.3513393859865807	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.034544521	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.025003653	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	4-HYDROXYDERRICIN	chembl:CHEMBL458094	CHEMBL:CHEMBL458094	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	SJ000018300	chembl:CHEMBL590927	CHEMBL:CHEMBL590927	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	DNDI1417085	chembl:CHEMBL1522984	CHEMBL:CHEMBL1522984	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GLUTAMIC ACID HYDROCHLORIDE	rxcui:91269	GLUTAMIC ACID HYDROCHLORIDE	TRUE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.2917092846427472	SJ000032149	chembl:CHEMBL600778	CHEMBL:CHEMBL600778	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.043466615	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	PI-CLONIDINE	chembl:CHEMBL360803	PI-CLONIDINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.005174699	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	JWH-015	iuphar.ligand:5558	JWH015	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	FR-122047	chembl:CHEMBL275809	FR-122047	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	NAFRONYL OXALATE	ncit:C87286	NAFRONYL OXALATE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	CETRIMONIUM BROMIDE	rxcui:288999	CETRIMONIUM BROMIDE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.03292017	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.005310242	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.026830696	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.005655716	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	(R)-FLECAINIDE	chembl:CHEMBL398673	(R)-FLECAINIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.007906591	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	SJ000121257	chembl:CHEMBL592363	CHEMBL:CHEMBL592363	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.049723174	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.1450488155682168	NSC-67436	chembl:CHEMBL1331995	CHEMBL:CHEMBL1331995	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.040515178	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
FANCD2	hgnc:3585	FANCD2	DTC	9/2/20	NULL	0.7001022831425933	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	1-METHYLEVODIAMINE	chembl:CHEMBL2171778	CHEMBL:CHEMBL2171778	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	chembl:CHEMBL224214	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.072826174	NSC-663284	drugbank:DB17038	NSC-663284	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.059030547	TICRYNAFEN	ncit:C152613	TICRYNAFEN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	NSC-601359	chembl:CHEMBL1306524	CHEMBL:CHEMBL1306524	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	NSC-28081	chembl:CHEMBL512832	CHEMBL:CHEMBL512832	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	DNDI1417443	chembl:CHEMBL1553566	CHEMBL:CHEMBL1553566	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	SJ000082806	chembl:CHEMBL494668	CHEMBL:CHEMBL494668	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.017295017	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	NSC-695801	chembl:CHEMBL461193	CHEMBL:CHEMBL461193	FALSE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	DTC	9/2/20	NULL	3.580068493342807	L-365260	iuphar.ligand:3477	[3H]L365260	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	DIPHENHYDRAMINE HYDROCHLORIDE	rxcui:1362	DIPHENHYDRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	PHANQUONE	ncit:C90620	PHANQUONE	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.7395446652914718	KMN-21	chembl:CHEMBL570176	CHEMBL:CHEMBL570176	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.056826484	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.001444741	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.011355465	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.018962684	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002097622	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.073954467	BW-723C86	iuphar.ligand:161	BW723C86	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.090064616	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.031254566	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.007723988	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DYRK2	hgnc:3093	DYRK2	DTC	9/2/20	NULL	7.501095890813499	LEUCETTAMINE B	chembl:CHEMBL485053	LEUCETTAMINE B	FALSE	FALSE	FALSE
S1PR2	hgnc:3169	S1PR2	DTC	9/2/20	NULL	0.326134604	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.009192519	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.022249013	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	DTC	9/2/20	NULL	0.525076712	ELTROMBOPAG	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	GR-89696	iuphar.ligand:1649	GR 89696	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.072524408	SJ000071821	chembl:CHEMBL589924	CHEMBL:CHEMBL589924	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.035670972	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.007111006	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	GISENOSIDE RK1	chembl:CHEMBL251235	GISENOSIDE RK1	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-3736	chembl:CHEMBL583824	CHEMBL:CHEMBL583824	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	GRISEOFULVIN	rxcui:5021	GRISEOFULVIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	TCMDC-125000	chembl:CHEMBL579742	CHEMBL:CHEMBL579742	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.099446347	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	DNDI1417085	chembl:CHEMBL1522984	CHEMBL:CHEMBL1522984	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GNF-PF-1859	chembl:CHEMBL1520837	CHEMBL:CHEMBL1520837	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.025672984	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1981421556063943	CID 649849	chembl:CHEMBL405914	CHEMBL:CHEMBL405914	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.018712641	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.1268301237577161	NSC-172033	chembl:CHEMBL238624	CHEMBL:CHEMBL238624	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1141471113819445	METHOXYCHLOR	rxcui:2598123	METHOXYCHLOR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.5556367326528519	PD-168393	drugbank:DB07662	PD-168393	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	BUTYLPARABEN	rxcui:1306937	BUTYLPARABEN	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.003398555	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.001528608	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005366413	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
ALDH5A1	hgnc:408	ALDH5A1	DTC	9/2/20	NULL	0.6579908676152193	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	DTC	9/2/20	NULL	0.3977853881492006	RO-4882224	chembl:CHEMBL1077391	CHEMBL:CHEMBL1077391	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	1-O-ACETYLGEOPYXIN A	chembl:CHEMBL1902074	CHEMBL:CHEMBL1902074	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2117244807890907	AVOBENZONE	rxcui:45045	AVOBENZONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	DIGITOXIGENIN	drugbank:DB04177	DIGITOXIGENIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	DNDI1318925	chembl:CHEMBL1390716	CHEMBL:CHEMBL1390716	FALSE	FALSE	FALSE
TRHR	hgnc:12299	TRHR	DTC	9/2/20	NULL	1.750255707856483	GNF-PF-4227	chembl:CHEMBL585654	CHEMBL:CHEMBL585654	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1000146118775133	TRICLOCARBAN	rxcui:38609	TRICLOCARBAN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	GNF-PF-130	chembl:CHEMBL578890	CHEMBL:CHEMBL578890	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.276356164	(S)-MEXILETINE	chembl:CHEMBL146855	(S)-MEXILETINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TROPOLONE	rxcui:1368873	TROPOLONE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.3804903712731485	FLUSILAZOLE	chembl:CHEMBL1900522	FLUSILAZOLE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.009065551	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	PROADIFEN HYDROCHLORIDE	ncit:C66468	PROADIFEN HYDROCHLORIDE	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	0.056826484	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.013832369	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.040766825	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003106871	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW782612X	chembl:CHEMBL251549	GW782612X	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.6035364509849942	NSC-119236	chembl:CHEMBL458765	CHEMBL:CHEMBL458765	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	TCMDC-123579	chembl:CHEMBL533954	CHEMBL:CHEMBL533954	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.1232574442152452	SELEGILINE HYDROCHLORIDE	rxcui:203137	SELEGILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	SPICLOMAZINE	ncit:C66557	SPICLOMAZINE	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.019799273	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005135225	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	1.312691780892362	GNF-PF-231	chembl:CHEMBL601167	CHEMBL:CHEMBL601167	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	MALATHION	rxcui:6606	MALATHION	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.020041096	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FLUFENOXURON	drugbank:DB15006	FLUFENOXURON	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1810609352954983	SJ000040829	chembl:CHEMBL589711	CHEMBL:CHEMBL589711	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	PIPOBROMAN	rxcui:8347	PIPOBROMAN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV001230	chembl:CHEMBL589920	CHEMBL:CHEMBL589920	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.014249029	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.079557078	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.02726255	GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.1096651446025365	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.1842374429322613	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.1181009249565778	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006199253	ESCITALOPRAM	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	BP-897	iuphar.ligand:7625	BP 897	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	FENDILINE HYDROCHLORIDE	rxcui:236767	FENDILINE HYDROCHLORIDE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.04525223	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
SF3B3	hgnc:10770	SF3B3	DTC	9/2/20	NULL	52.50767123569449	PLADIENOLIDE B	chembl:CHEMBL1242745	PLADIENOLIDE B	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.025003653	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.052090944	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.013890918	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
TNNC1	hgnc:11943	TNNC1	DTC	9/2/20	NULL	0.2917092846427472	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
TNNT2	hgnc:11949	TNNT2	DTC	9/2/20	NULL	0.364636606	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	XCT790	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	3,3',4'-TRIHYDROXYFLAVONE	chembl:CHEMBL122701	CHEMBL:CHEMBL122701	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.2160809515872201	YANGONIN	chembl:CHEMBL1098658	YANGONIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ANCITABINE HYDROCHLORIDE	ncit:C403	ANCITABINE HYDROCHLORIDE	FALSE	FALSE	FALSE
GCK	hgnc:4195	GCK	DTC	9/2/20	NULL	3.500511415712966	RO-281675	chembl:CHEMBL1096435	RO-281675	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FANDOSENTAN POTASSIUM	ncit:C72774	FANDOSENTAN POTASSIUM	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.060772768	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.042344896	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
BCL2L1	hgnc:992	BCL2L1	DTC	9/2/20	NULL	0.1562728310586145	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.023274677	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006286838	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008279355	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001976425	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.060492709	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003668018	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CSNK1G3	hgnc:2456	CSNK1G3	DTC	9/2/20	NULL	0.1179947668217854	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.043109746	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	MEBENDAZOLE	rxcui:6672	MEBENDAZOLE	TRUE	FALSE	FALSE
CHUK	hgnc:1974	CHUK	DTC	9/2/20	NULL	7.501095891	AILANTHINONE	chembl:CHEMBL487194	AILANTHINONE	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	1.944728564284981	CINNAMTANNIN B1	iuphar.ligand:13186	CINNAMTANNIN B1	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.009954061	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.087512785	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.030598876	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.072324616	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	ETONOGESTREL	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.025298806	TACRINE	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.005541122	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.003667505	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ARG1	hgnc:663	ARG1	DTC	9/2/20	NULL	5.000730593875666	2-AMINOHOMOHISTIDINE	chembl:CHEMBL1099168	CHEMBL:CHEMBL1099168	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	1.250182648468916	LINOLEIC ACID	rxcui:6400	LINOLEIC ACID	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	CLIOXANIDE	ncit:C65338	CLIOXANIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	3,4-DIHYDROXYPHENYLACETIC ACID	chembl:CHEMBL1284	3,4-DIHYDROXYPHENYLACETIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SARCOLYSIN	ncit:C61936	SARCOLYSIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001008134	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.014853655	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.034318739	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	AMITHIOZONE	ncit:C85523	THIOACETAZONE	FALSE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	DTC	9/2/20	NULL	0.1097339001790898	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CLK3	hgnc:2071	CLK3	DTC	9/2/20	NULL	5.000730593875666	LEUCETTAMINE B	chembl:CHEMBL485053	LEUCETTAMINE B	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.018359326	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005899738	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	3-HYDROXY-3',4'-DIMETHOXYFLAVONE	chembl:CHEMBL77098	3-HYDROXY-3',4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	PROROXAN HYDROCHLORIDE	ncit:C84120	PROROXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.6604738520213144	QUERCETAGETIN	chembl:CHEMBL413552	QUERCETAGETIN	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	0.07767407	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	TRYPTANTHRIN	iuphar.ligand:8224	TRYPTANTHRIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008887554	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.2476776945079929	SJ000012773	chembl:CHEMBL589715	CHEMBL:CHEMBL589715	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.067231333	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	THIOTEPA	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.010193685	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	DTC	9/2/20	NULL	0.6563458904461813	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.006495259	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.035598421	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.055563673	DNDI1417031	chembl:CHEMBL1333049	CHEMBL:CHEMBL1333049	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1100789753368857	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.4953553890159858	ARTEANNUIN B	chembl:CHEMBL515516	ARTEANNUIN B	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.037398626	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ALCLOFENAC	ncit:C174701	ALCLOFENAC	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	CARINATIN G	chembl:CHEMBL2332131	CARINATIN G	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.055271233	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	EHNA	iuphar.ligand:5179	EHNA	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	DIPYRITHIONE	rxcui:1362743	DIPYRITHIONE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01823183	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CANRENONE	rxcui:1982	CANRENONE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.017611159	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1019566431761058	PYRACLOSTROBIN	chembl:CHEMBL519873	PYRACLOSTROBIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	GW9662	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.020737627	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.009515707	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.007540955	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	HYMECROMONE	rxcui:5556	HYMECROMONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	AM-281	iuphar.ligand:741	AM281	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.03261346	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.008245551	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	DTC	9/2/20	NULL	1.166837138570989	CID 100335	chembl:CHEMBL1520346	CHEMBL:CHEMBL1520346	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003185179	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	DTC	9/2/20	NULL	5.527123287967842	MRS-3481	chembl:CHEMBL382194	CHEMBL:CHEMBL382194	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	GERALDOL	chembl:CHEMBL509256	GERALDOL	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00279415	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.021240967	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.8140724222588294	CLENBUTEROL	rxcui:2580	CLENBUTEROL	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.034184682	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	NSC-209931	chembl:CHEMBL472656	CHEMBL:CHEMBL472656	FALSE	FALSE	FALSE
TSSK2	hgnc:11401	TSSK2	DTC	9/2/20	NULL	0.1019566431761058	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	1.810609352954982	2-(1-PHENYLETHYLIDENE)HYDRAZINECARBOXIMIDAMIDE	chembl:CHEMBL1644904	2-(1-PHENYLETHYLIDENE)HYDRAZINECARBOXIMIDAMIDE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.039361073	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	L-732138	iuphar.ligand:9461	L-732,138	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.019889269	HYDRALAZINE HYDROCHLORIDE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	1.009762908	N-[6-(4-CHLOROPHENYL)-7-(2,4-DICHLOROPHENYL)-2,2-DIMETHYL-3,4-DIHYDRO-2H-PYRANO[2,3-B]PYRIDINE-4-YL]-4,4,4-TRIFLUORO-3-HYDROXYBUTANAMIDE (DIASTEREOMERIC MIX)	chembl:CHEMBL1097456	N-[6-(4-CHLOROPHENYL)-7-(2,4-DICHLOROPHENYL)-2,2-DIMETHYL-3,4-DIHYDRO-2H-PYRANO[2,3-B]PYRIDINE-4-YL]-4,4,4-TRIFLUORO-3-HYDROXYBUTANAMIDE (DIASTEREOMERIC MIX)	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	TRIFLUSAL	rxcui:38655	TRIFLUSAL	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.011585982	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	TCMDC-125495	chembl:CHEMBL532412	CHEMBL:CHEMBL532412	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.010777437	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	ENNIATIN B	chembl:CHEMBL469036	ENNIATIN B	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.2651902587661338	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.003550214	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.015286076	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.024467694	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ERGONOVINE	rxcui:4021	ERGONOVINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1029562181092048	2,3,4-TRIHYDROXYBENZOPHENONE	chembl:CHEMBL1527	CHEMBL:CHEMBL1527	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	PT-103	chembl:CHEMBL398765	CHEMBL:CHEMBL398765	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	MIANSERIN HYDROCHLORIDE	rxcui:203127	MIANSERIN HYDROCHLORIDE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.017047945	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	DIHYDROXANTHOHUMOL	chembl:CHEMBL510279	DIHYDROXANTHOHUMOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV080034	chembl:CHEMBL1623028	CHEMBL:CHEMBL1623028	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.1835932560688619	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	GR-103545	iuphar.ligand:1649	GR 89696	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	TCMDC-138263	chembl:CHEMBL535307	CHEMBL:CHEMBL535307	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	TCMDC-125738	chembl:CHEMBL527585	CHEMBL:CHEMBL527585	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	TCMDC-123789	chembl:CHEMBL588859	CHEMBL:CHEMBL588859	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
TXN2	hgnc:17772	TXN2	DTC	9/2/20	NULL	17.50255707856483	BIOTINYLATED GAMBOGIC ACID	chembl:CHEMBL2205161	BIOTINYLATED GAMBOGIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003217382	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.005211162	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.1483267549030917	DNDI1318925	chembl:CHEMBL1390716	CHEMBL:CHEMBL1390716	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	1.750255707856483	AMAUROMINE	chembl:CHEMBL2022567	AMAUROMINE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.013777925	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PHENMEDIPHAM	chembl:CHEMBL1079421	PHENMEDIPHAM	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.008728004	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	4'-HYDROXYPHENYL-BENZO[D]THIAZOLE	chembl:CHEMBL47875	CHEMBL:CHEMBL47875	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BENOXACOR	chembl:CHEMBL2269059	BENOXACOR	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	HYMECROMONE	rxcui:5556	HYMECROMONE	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.9546849315580818	(Z)-16-NONADECENOIC ACID	chembl:CHEMBL2171117	CHEMBL:CHEMBL2171117	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005574063	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.173866461	LAURYL ISOQUINOLINIUM	chembl:CHEMBL1398631	LAURYL ISOQUINOLINIUM	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.029203377	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	BENSERAZIDE	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	CAPTAMINE	ncit:C83585	CAPTAMINE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	AC-55649	iuphar.ligand:4055	AC55649	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.00206886	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	2,3-DICHLORO-PROPENE	chembl:CHEMBL156075	CHEMBL:CHEMBL156075	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.017064567	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	METAPHIT METHANESULFONATE	chembl:CHEMBL1256971	METAPHIT METHANESULFONATE	FALSE	FALSE	FALSE
CDC37	hgnc:1735	CDC37	DTC	9/2/20	NULL	26.25383561784724	SODIUM MOLYBDATE	ncit:C1228	SODIUM MOLYBDATE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	NSC-309895	chembl:CHEMBL552439	CHEMBL:CHEMBL552439	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.040515178	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	1-(4-HYDROXYPHENYL)MALEIMIDE	chembl:CHEMBL565893	CHEMBL:CHEMBL565893	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.021661581	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	TAXIFOLIN	drugbank:DB02224	TAXIFOLIN	FALSE	FALSE	FALSE
HTR1E	hgnc:5291	HTR1E	DTC	9/2/20	NULL	2.625383561784724	SJ000189154	chembl:CHEMBL604664	CHEMBL:CHEMBL604664	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.025147352	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	0.7740688634254718	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009144492	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	BW-373U86	iuphar.ligand:9002	BW373U86	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	MALATHION	rxcui:6606	MALATHION	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	SJ000032081	chembl:CHEMBL590184	CHEMBL:CHEMBL590184	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.019107595	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.1944728564284981	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	NSC-663284	drugbank:DB17038	NSC-663284	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.018712641	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	PYRIDOSTIGMINE	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.028598949	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	SB-228357	iuphar.ligand:192	SB 228357	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	CANAVANINE	drugbank:DB01833	CANAVANINE	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.1367387271762877	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	GNF-PF-2954	chembl:CHEMBL582722	CHEMBL:CHEMBL582722	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665944	chembl:CHEMBL600030	CHEMBL:CHEMBL600030	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007699637	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	VANITIOLIDE	ncit:C74234	VANITIOLIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	LOPINAVIR	rxcui:195088	LOPINAVIR	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.012573676	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.013814173	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.021370644	DOMPERIDONE	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	NORADRENALINE	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.026372512	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
PADI1	hgnc:18367	PADI1	DTC	9/2/20	NULL	13.12691780892362	O-CL-AMIDINE	chembl:CHEMBL1910971	CHEMBL:CHEMBL1910971	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.3977853881492007	LACTOFEN	chembl:CHEMBL1243178	LACTOFEN	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	1.166837138570988	2',4,4',6-TETRAMETHOXYCHALCONE	chembl:CHEMBL140130	CHEMBL:CHEMBL140130	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	DNDI1417519	chembl:CHEMBL1402376	CHEMBL:CHEMBL1402376	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.182318303	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	DNDI1417083	chembl:CHEMBL1564100	CHEMBL:CHEMBL1564100	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.2318219480604613	PIFITHRIN-MU	chembl:CHEMBL1241268	CHEMBL:CHEMBL1241268	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1166837138570989	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.018385039	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL201761	SALINAZID	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.062808219	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-4857	chembl:CHEMBL584829	CHEMBL:CHEMBL584829	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	CHLORQUINALDOL	rxcui:2407	CHLORQUINALDOL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.013350539	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	DTC	9/2/20	NULL	0.038937836	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	UNOPROSTONE ISOPROPYL	ncit:C47778	UNOPROSTONE ISOPROPYL	TRUE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.053038052	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
CLCN3	hgnc:2021	CLCN3	DTC	9/2/20	NULL	26.25383561784724	DESACETYLBUFOTALIN	chembl:CHEMBL463065	DESACETYLBUFOTALIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.014114965	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.064347636	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	DNDI1417827	chembl:CHEMBL1363249	CHEMBL:CHEMBL1363249	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	ICILLIN	iuphar.ligand:2429	ICILIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FLUFENACET	chembl:CHEMBL1886718	FLUFENACET	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.022315202	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.048083948	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.070197421	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	HOE-33342	chembl:CHEMBL343002	CHEMBL:CHEMBL343002	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01256465	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004931224	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	DIHYDROXANTHOHUMOL	chembl:CHEMBL510279	DIHYDROXANTHOHUMOL	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.044955198	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	TCMDC-124377	chembl:CHEMBL531269	CHEMBL:CHEMBL531269	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	4,4'-METHYLENEDIANILINE	chembl:CHEMBL85728	4,4'-METHYLENEDIANILINE	FALSE	FALSE	FALSE
NR1D1	hgnc:7962	NR1D1	DTC	9/2/20	NULL	10.50153425	SR9011	iuphar.ligand:8900	SR9011	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.034704343	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.005562253	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	AMARANTH	chembl:CHEMBL1408927	AMARANTH	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.021869084	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	SJ000032149	chembl:CHEMBL600778	CHEMBL:CHEMBL600778	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	CAMBINOL	drugbank:DB15493	CAMBINOL	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.073954467	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	SKIMMIANINE	chembl:CHEMBL21396	SKIMMIANINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	SJ000147993	chembl:CHEMBL601618	CHEMBL:CHEMBL601618	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	BENSERAZIDE	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.051885051	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.081533651	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	1.193356164447602	CRYPTOLEPINE HYDROCHLORIDE	chembl:CHEMBL92129	CRYPTOLEPINE HYDROCHLORIDE	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.032776324	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	BP-897	iuphar.ligand:7625	BP 897	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	ISOXSUPRINE	rxcui:6066	ISOXSUPRINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	REL-CISAPRIDE	chembl:CHEMBL74656	REL-CISAPRIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.004831401	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.037398626	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	DTC	9/2/20	NULL	0.4526523382387456	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
HPGDS	hgnc:17890	HPGDS	DTC	9/2/20	NULL	26.25383561784724	HQL-79	drugbank:DB07917	4-(BENZHYDRYLOXY)-1-[3-(1H-TETRAAZOL-5-YL)PROPYL]PIPERIDINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002088278	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.056399217	TRICLOCARBAN	rxcui:38609	TRICLOCARBAN	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.009437037	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.021370644	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.030996264	IPRONIAZID	rxcui:5981	IPRONIAZID	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	NU-1025	chembl:CHEMBL123904	CHEMBL:CHEMBL123904	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-278539	chembl:CHEMBL275168	CHEMBL:CHEMBL275168	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	S-(2,4-DICHLOROBENZYL)ISOTHIOUREA HYDROBROMIDE	chembl:CHEMBL1224483	CHEMBL:CHEMBL1224483	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.002286123	PARAPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	PROSTAGLANDIN A2	iuphar.ligand:6279	PROSTAGLANDIN A2	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.1750255707856483	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.1223955040459079	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.036951211	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	ARCTIGENIN	drugbank:DB16880	ARCTIGENIN	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.5147810905460244	GNF-PF-4242	chembl:CHEMBL584514	CHEMBL:CHEMBL584514	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.0136917	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.008463519	TRIMIPRAMINE	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.01274458	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.011316308	ISOPRENALINE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.002414146	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.1930429089547591	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	DTC	9/2/20	NULL	0.3281729452230906	ANANDAMIDE	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1325951293830669	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	GNF-PF-5217	chembl:CHEMBL601970	CHEMBL:CHEMBL601970	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.025003653	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	0.2381300282797936	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.048083948	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005412046	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.078136416	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005363398	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.057385433	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.036873365	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.036770078	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE	chembl:CHEMBL457504	CHEMBL:CHEMBL457504	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	DILAZEP	ncit:C65389	DILAZEP	FALSE	FALSE	FALSE
F12	hgnc:3530	F12	DTC	9/2/20	NULL	1.250182648468916	PENTAMIDINE ISETHIONATE	rxcui:7995	PENTAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	SJ000082806	chembl:CHEMBL494668	CHEMBL:CHEMBL494668	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.061412481	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.099446347	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	AMBAZONE	ncit:C72627	AMBAZONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	GNF-PF-2588	chembl:CHEMBL578636	CHEMBL:CHEMBL578636	FALSE	FALSE	FALSE
POLR2A	hgnc:9187	POLR2A	DTC	9/2/20	NULL	35.00511415712966	PSI-7409	chembl:CHEMBL486231	GS-461203	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.022789788	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.010418189	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.07458476	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	PROPYLENE GLYCOL MONOSTEARATE	rxcui:1314411	PROPYLENE GLYCOL MONOSTEARATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	CHLORQUINALDOL	rxcui:2407	CHLORQUINALDOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	XANTHINE AMINE CONGENER	iuphar.ligand:404	XANTHINE AMINE CONGENER	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	GNF-PF-1656	chembl:CHEMBL579028	CHEMBL:CHEMBL579028	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01323278	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	GESTODENE	rxcui:25734	GESTODENE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.061628722	N-METHYLDOPAMINE HCL	chembl:CHEMBL1256484	CHEMBL:CHEMBL1256484	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	HYPEROSIDE	chembl:CHEMBL251254	HYPEROSIDE	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.056581542	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.046343929	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.027290889	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.051731696	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	(E)-DIBENZYLIDENEACETONE	chembl:CHEMBL17201	CHEMBL:CHEMBL17201	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003973038	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005581766	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.002932243	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	XANTHINE AMINE CONGENER	iuphar.ligand:404	XANTHINE AMINE CONGENER	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.028290771	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.074426182	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.2941606231691568	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.030814361	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.004855078	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.063034419	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	4'-O-ACETYLPATENTIFLORIN B	chembl:CHEMBL454803	4'-O-ACETYLPATENTIFLORIN B	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.013876234	MONTELUKAST SODIUM	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000093125	chembl:CHEMBL591641	CHEMBL:CHEMBL591641	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.039126432	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	CLOFENOXYDE	ncit:C78034	CLOFENOXYDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003981473	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	P-PHENYLENEDIAMINE	rxcui:1362740	4-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.009465958	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.1491695205559502	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	MEVASTATIN	ncit:C96285	MEVASTATIN	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.027361996	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	2-(4-HYDROXYBENZYLIDENE)MALONONITRILE	chembl:CHEMBL305695	CHEMBL:CHEMBL305695	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007946076	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
ELANE	hgnc:3309	ELANE	DTC	9/2/20	NULL	4.565884455277782	L-694458	chembl:CHEMBL310871	CHEMBL:CHEMBL310871	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	GNF-PF-5217	chembl:CHEMBL601970	CHEMBL:CHEMBL601970	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.07458476	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.021554873	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003483789	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.021878196	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.1902451856365742	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005677733	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.2983390411119005	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.021661581	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.010113188	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	DNDI1417776	chembl:CHEMBL1585652	CHEMBL:CHEMBL1585652	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.5527123287967842	HESPERIDIN	rxcui:5281	HESPERIDIN	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.046343929	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1121958787087489	DISOPYRAMIDE	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.019739726	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	DTC	9/2/20	NULL	7.001022831425932	3-[(4-ACETYLPHENYL)AMINO]BENZOIC ACID	chembl:CHEMBL1682201	CHEMBL:CHEMBL1682201	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.2917092846427472	HYMECROMONE	rxcui:5556	HYMECROMONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001573971	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002767057	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	1.193356164447602	ACEBUTOLOL	rxcui:149	ACEBUTOLOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003314878	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00575742	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	AMBAZONE	ncit:C72627	AMBAZONE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.04907259	ACETOCHLOR	chembl:CHEMBL1517425	ACETOCHLOR	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.091796628	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.007283628	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.031254566	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.049723174	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	ERUCIC ACID	chembl:CHEMBL1173380	ERUCIC ACID	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.1704794520639431	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.2375912725597036	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	CAPENSIN	chembl:CHEMBL1327256	CAPENSIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	DNQX	chembl:CHEMBL155265	DNQX	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.085796848	CAMBINOL	drugbank:DB15493	CAMBINOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	SODIUM AZIDE	chembl:CHEMBL89295	SODIUM AZIDE	FALSE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.2051080907644316	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.001253017	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.039068208	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003720782	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.012466209	LOPERAMIDE HYDROCHLORIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
CLK1	hgnc:2068	CLK1	DTC	9/2/20	NULL	3.000438356325399	LEUCETTAMINE B	chembl:CHEMBL485053	LEUCETTAMINE B	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	chembl:CHEMBL1256180	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DACTHAL	chembl:CHEMBL1888079	DACTHAL	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.007023498	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.1209854175937661	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	TRANSPLATIN	chembl:CHEMBL1386	TRANSPLATIN	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.032817295	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NLRP3	hgnc:16400	NLRP3	DTC	9/2/20	NULL	0.729273212	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	PENTETIC ACID	rxcui:3690	PENTETIC ACID	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.007759372	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.4817217544559128	ALFENTANIL HYDROCHLORIDE	rxcui:203203	ALFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	CID 649849	chembl:CHEMBL405914	CHEMBL:CHEMBL405914	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.040390516	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002956679	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	GNF-PF-4242	chembl:CHEMBL584514	CHEMBL:CHEMBL584514	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.07699072	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	DNDI1417263	chembl:CHEMBL1431115	CHEMBL:CHEMBL1431115	FALSE	FALSE	FALSE
CAMK2A	hgnc:1460	CAMK2A	DTC	9/2/20	NULL	0.1229687850953032	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	CARNOSIC ACID	chembl:CHEMBL484853	CARNOSIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GUAIAZULENE	rxcui:26290	GUAIAZULENE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.066803653	STANOLONE	ncit:C72098	STANOLONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.068191781	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1019566431761058	PHANQUONE	ncit:C90620	PHANQUONE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	EPIRUBICIN HYDROCHLORIDE	rxcui:203213	EPIRUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.1319288222002374	IOFETAMINE HYDROCHLORIDE	chembl:CHEMBL1255865	IOFETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	CINACALCET	rxcui:407990	CINACALCET	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.027563082	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.1835932560688619	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.027177884	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.2243917574174978	DIHYDRO-12-HYDROXY-2,2-DIMETHYL-2H,6H-PYRANO[3,2-B]XANTHEN-6-ONE	chembl:CHEMBL2387036	DIHYDRO-12-HYDROXY-2,2-DIMETHYL-2H,6H-PYRANO[3,2-B]XANTHEN-6-ONE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.013876234	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	CGP-60474	chembl:CHEMBL300389	CHEMBL:CHEMBL300389	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.004520678	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.016116535	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004386606	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.09741683	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.2027323213733378	FRENTIZOLE	ncit:C167023	FRENTIZOLE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004762601	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.1041818873724097	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	METHACHOLINE CHLORIDE	rxcui:40165	METHACHOLINE CHLORIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.019739726	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
CCR1	hgnc:1602	CCR1	DTC	9/2/20	NULL	1.458546423213736	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DNDI1417827	chembl:CHEMBL1363249	CHEMBL:CHEMBL1363249	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TETRANITROMETHANE	chembl:CHEMBL261663	TETRANITROMETHANE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	CETRIMIDE	rxcui:288088	CETRIMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	GERONTOXANTHONE H	chembl:CHEMBL514057	GERONTOXANTHONE H	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	EFLORNITHINE	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.053633985	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.014658758	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	TCMDC-125543	chembl:CHEMBL546170	CHEMBL:CHEMBL546170	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.016246185	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	CROMOLYN	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007244436	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	FDA	10-Apr-24	NULL	0.4947116523181093	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
HBB	hgnc:4827	HBB	FDA	10-Apr-24	NULL	NULL	Luspaterceptâaamt	NULL	NULL	NULL	NULL	NULL
PRKCI	hgnc:9404	PRKCI	DTC	9/2/20	NULL	0.044498026	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CYB5R	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	FDA	10-Apr-24	NULL	0.9842513760562132	Ivosidenib	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.031784305	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
HLA-A	hgnc:4931	HLA-A	FDA	10-Apr-24	NULL	0.1875273972703375	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.027635616	Methylene Blue	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
BRCA	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.010368813	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	FDA	10-Apr-24	NULL	0.3281729452230906	Ospemifene	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.006811217	Metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	0.060878459	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.028866229	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.037748146	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.2108741816694558	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.1860654544142257	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.019629036	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	3.500511415712966	TIVANTINIB	ncit:C62437	TIVANTINIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	0.047821194	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.1491695205559502	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.1491695205559502	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.1363835616511545	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.1657439117288336	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.1312691780892362	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.064624826	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.066676408	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.079197091	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.096521454	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.1583941817064691	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547592	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.095036509	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.073540156	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
MAPKAP1	hgnc:18752	MAPKAP1	MyCancerGenome	20-Jun-17	inhibitor	1.944728564284981	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.1704794520639432	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.039068208	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4930297768609811	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.8334550989792776	PD 0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.089298761	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.7501095890813498	PD 0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.065634589	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1403266238077355	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.184383561707394	BIBW 2992	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1607377690888607	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5114383561918295	PD 0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1275696580070323	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.9376369863516874	PD 0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005366413	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.020257589	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003541833	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.364636606	6-HYDROXYMELATONIN	iuphar.ligand:1347	6-HYDROXYMELATONIN	FALSE	FALSE	FALSE
PDGFC	hgnc:8801	PDGFC	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.071585127259071	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ABL	hgnc:76	ABL1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.7544205637312429	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3513393859865807	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.059667808	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.184383561707394	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	3.500511415712966	ARQ 197	ncit:C62437	TIVANTINIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3453256329104173	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.035560536	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.021715331	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
A2M	hgnc:7	A2M	NCI	14-Sep-17	NULL	0.1150222809106122	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.4055851016423223	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02804897	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.1154014752432846	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	0.067059606	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ADSS	hgnc:292	ADSS2	NCI	14-Sep-17	NULL	52.50767123569449	ALANOSINE	ncit:C994	ALANOSINE	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.063568609	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.068458502	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.4449802647092754	IDOXIFENE	ncit:C1406	IDOXIFENE	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.064724402	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
HRH4	hgnc:17383	HRH4	DTC	9/2/20	NULL	4.773424657790408	JNJ-7777120	iuphar.ligand:1278	JNJ 7777120	FALSE	FALSE	FALSE
ALPP	hgnc:439	ALPP	NCI	14-Sep-17	NULL	NULL	BISPHOSPHONATES	NULL	NULL	NULL	NULL	NULL
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	0.1403948428761885	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
ALDH3A1	hgnc:405	ALDH3A1	NCI	14-Sep-17	NULL	0.1046664542904209	ANTABUSE	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.1052961321571413	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
APP	hgnc:620	APP	NCI	14-Sep-17	NULL	NULL	TAXANES	NULL	NULL	NULL	NULL	NULL
KCNQ3	hgnc:6297	KCNQ3	DTC	9/2/20	NULL	2.678962818147678	EZOGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
APP	hgnc:620	APP	NCI	14-Sep-17	NULL	0.1242785118004603	AMB	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.091796628	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.069638821	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
APP	hgnc:620	APP	NCI	14-Sep-17	NULL	0.017754073	DAUNOMYCIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.032559532	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.064033745	PROTEASE INHIBITOR	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.005691888	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.065675636	ALPHA-METHYL-P-TYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.077616661	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.025111273	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.315361389	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.051604591	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	PARATHION	ncit:C163685	PARATHION	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.2386712328895204	AS101	iuphar.ligand:437	AS101	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.007955708	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.070197421	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	TDR77578	chembl:CHEMBL1364172	CHEMBL:CHEMBL1364172	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.1325951293830669	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.1988926940746003	MITHRAMYCIN	rxcui:6995	PLICAMYCIN	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	NULL	TAXANES	NULL	NULL	NULL	NULL	NULL
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.079557078	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-2491	chembl:CHEMBL577851	CHEMBL:CHEMBL577851	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	NCI	14-Sep-17	NULL	0.048550782	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.3723948314588262	IROFULVEN	ncit:C1717	IROFULVEN	FALSE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	DTC	9/2/20	NULL	0.7001022831425934	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.2792961235941196	PHYTOESTROGEN	ncit:C1194	PHYTOESTROGEN	FALSE	FALSE	FALSE
CAST	hgnc:1515	CAST	NCI	14-Sep-17	NULL	0.1000146118775133	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.3763990769583835	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.1268301237577161	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CEACAM6	hgnc:1818	CEACAM6	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.169927739	METHOCTRAMINE HYDROCHLORIDE	chembl:CHEMBL500996	METHOCTRAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	NULL	ANTIINFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.9376369863516875	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.6250913242344582	PHYTOESTROGEN	ncit:C1194	PHYTOESTROGEN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.022136455	IRBESARTAN	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.008432935	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010678802	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.009320613	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
CYP27A1	hgnc:2605	CYP27A1	NCI	14-Sep-17	NULL	0.2983390411119005	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.6250913242344582	TCMDC-125610	chembl:CHEMBL535315	CHEMBL:CHEMBL535315	FALSE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	NCI	14-Sep-17	NULL	0.3409589041278863	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
CYP2B	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.028290771	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CYP2B	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.063110182	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.004517955	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.004517955	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.069777636	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	GNF-PF-3542	chembl:CHEMBL598477	CHEMBL:CHEMBL598477	FALSE	FALSE	FALSE
DEFA1	hgnc:2761	DEFA1	NCI	14-Sep-17	NULL	2.500365296937833	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PENTACHLORONITROBENZENE	chembl:CHEMBL468759	PENTACHLORONITROBENZENE	FALSE	FALSE	FALSE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	0.292250489	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	1.591141552596802	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.087077398	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	AG1295	iuphar.ligand:5914	AG 1295	FALSE	FALSE	TRUE
EPHX1	hgnc:3401	EPHX1	NCI	14-Sep-17	NULL	0.5385402178019949	ANTICONVULSANT	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
EIF2AK2	hgnc:9437	EIF2AK2	NCI	14-Sep-17	NULL	2.917092846427472	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	NULL	ISOFLAVONES	NULL	NULL	NULL	NULL	NULL
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.172722603	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.072725306	AZA	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	4-HYDROXYESTRADIOL	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
F11	hgnc:3529	F11	NCI	14-Sep-17	NULL	0.9211872146613068	DEXTRAN SULFATE	rxcui:40068	DEXTRAN SULFATE	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.065799087	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
FCGR1A	hgnc:3613	FCGR1A	NCI	14-Sep-17	NULL	0.5385402178019948	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.6604738520213144	FLT3L	ncit:C1714	RECOMBINANT FLT3 LIGAND	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.055039488	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.02277496	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.3962843112127887	RECOMBINANT STEM CELL FACTOR	ncit:C1410	RECOMBINANT HUMAN STEM CELL FACTOR	FALSE	FALSE	FALSE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	0.1193356164447602	CBDCA	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.096167896	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.2287915957982331	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.502465753	DDS	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	NCI	14-Sep-17	NULL	0.1209854175937661	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	NCI	14-Sep-17	NULL	0.043502627	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
GPT	hgnc:4552	GPT	NCI	14-Sep-17	NULL	1.312691780892362	PROTEASE INHIBITOR	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.2125816649218401	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
GPD2	hgnc:4456	GPD2	NCI	14-Sep-17	NULL	2.625383561784725	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.042689164	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.4487835148349957	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1930429089547591	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.6141248097742047	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1029562181092049	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.546954909	DIETHYLSTILBESTROL DIPHOSPHATE	chembl:CHEMBL1200598	DIETHYLSTILBESTROL DIPHOSPHATE	TRUE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	0.1392776425349986	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.8204323630577265	TICARCILLIN	rxcui:10591	TICARCILLIN	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1491695205559502	PYRIMETHAMINE	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.082364974	DAC	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
ITGA2B	hgnc:6138	ITGA2B	NCI	14-Sep-17	NULL	0.093098708	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
INPP1	hgnc:6071	INPP1	NCI	14-Sep-17	NULL	2.500365296937833	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	NULL	OPIOIDS	NULL	NULL	NULL	NULL	NULL
ITGAV	hgnc:6150	ITGAV	NCI	14-Sep-17	NULL	0.09972967	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	2.386712328895204	LAK CELL	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	NULL	OPIOIDS	NULL	NULL	NULL	NULL	NULL
IVL	hgnc:6187	IVL	NCI	14-Sep-17	NULL	2.187819634820604	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
JAG1	hgnc:6188	JAG1	NCI	14-Sep-17	NULL	0.8334550989792776	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
LAMA5	hgnc:6485	LAMA5	NCI	14-Sep-17	NULL	NULL	RBC	NULL	NULL	NULL	NULL	NULL
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.025513932	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
KRT17	hgnc:6427	KRT17	NCI	14-Sep-17	NULL	1.346350544504987	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.019024519	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	(S)-ROSCOVITINE	chembl:CHEMBL133342	(S)-ROSCOVITINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	1.750255707856483	PC-SPES	ncit:C1828	CHRYSANTHEMUM MORIFOLIUM/GANODERMA LUCIDUM/GLYCYRRHIZA GLABRA/ISATIS INDIGOTICA/PANAX PSEUDOGINSENG/RABDOSIA RUBESCENS/SCUTELLARIA BAICALENSIS/SERONA REPENS SUPPLEMENT	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1591141552596803	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	3.387591692625451	COLESTIPOL HYDROCHLORIDE	rxcui:104485	COLESTIPOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.2083637747448194	METHOCTRAMINE HYDROCHLORIDE	chembl:CHEMBL500996	METHOCTRAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.1500219178162699	5-DEOXY-5-FLUOROURIDINE	ncit:C978	DOXIFLURIDINE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.1037701012563132	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.2000292237550266	QUINONE	rxcui:319868	1,4-BENZOQUINONE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.065854103	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.021215221	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.05486695	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.4773424657790409	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.151537291	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	N-2-NAPHTHYLIMIDODICARBONIMIDIC DIAMIDE	chembl:CHEMBL43078	CHEMBL:CHEMBL43078	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1041818873724097	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
MT1H	hgnc:7400	MT1H	NCI	14-Sep-17	NULL	0.3409589041278864	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.1271372184883644	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.5000730593875666	IL-9	iuphar.ligand:5000	IL-9	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.2983390411119005	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	NULL	ISOFLAVONES	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.07767407	APAP	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
NPPA	hgnc:7939	NPPA	NCI	14-Sep-17	NULL	26.25383561784724	INTRAVENOUS FLUID	ncit:C29107	IV FLUID	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.4730420832044549	OPIATE	ncit:C1657	OPIATE	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.1091635576625665	TYROSINE KINASE INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.2885036881082116	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	NULL	N-ETHYL-N-NITROSOUREA	NULL	NULL	NULL	NULL	NULL
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.1093909817410302	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.062509132	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	NCI	14-Sep-17	NULL	0.042344896	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.16256245	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.037721028	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.005385402	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.026927011	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.062139256	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.038467158	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.3029288725136221	FGF-1	iuphar.ligand:4923	FGF-1	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.009393143	PS341	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	NULL	ANTIINFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	NULL	BISPHOSPHONATES	NULL	NULL	NULL	NULL	NULL
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1666910197958555	ZOLEDRONATE	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.5000730593875667	OK-432	ncit:C745	PICIBANIL	FALSE	FALSE	FALSE
PLAUR	hgnc:9053	PLAUR	NCI	14-Sep-17	NULL	13.12691780892362	DIPHTHERIA TOXIN	ncit:C444	DIPHTHERIA TOXIN	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	1.640864726115453	ADENOSINE DEAMINASE INHIBITOR	ncit:C2157	ADENOSINE DEAMINASE INHIBITOR	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.1715936968486748	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	NULL	ISOFLAVONES	NULL	NULL	NULL	NULL	NULL
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	2.500365296937833	SOY PROTEIN ISOLATE	rxcui:196238	SOY PROTEIN ISOLATE	TRUE	FALSE	FALSE
REG3A	hgnc:8601	REG3A	NCI	14-Sep-17	NULL	1.875273972703374	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	DALBERGIONE, 4-METHOXY-4'-HYDROXY-	chembl:CHEMBL1374504	DALBERGIONE, 4-METHOXY-4'-HYDROXY-	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	NCI	14-Sep-17	NULL	0.1121958787087489	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.062434805	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	NCI	14-Sep-17	NULL	0.009334697	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.280789686	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
SFTPB	hgnc:10801	SFTPB	NCI	14-Sep-17	NULL	2.282942227638891	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	NULL	L6	NULL	NULL	NULL	NULL	NULL
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.024479101	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	NCI	14-Sep-17	NULL	0.1495945049449986	ALPHA-METHYL-P-TYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.062139256	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.2308029504865691	PENICILLAMINE	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.070244376	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	TRIBUTYLTIN-OXIDE	chembl:CHEMBL511667	TRIBUTYLTIN-OXIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	2-HYDROXY-NAPHTHALDEHYDE THIOSEMICARBAZONE	chembl:CHEMBL505209	CHEMBL:CHEMBL505209	FALSE	FALSE	FALSE
SMAD2	hgnc:6768	SMAD2	NCI	14-Sep-17	NULL	2.625383561784725	AMIFOSTINE	rxcui:1545987	AMIFOSTINE ANHYDROUS	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	INDIMITECAN	ncit:C95905	INDIMITECAN	FALSE	FALSE	FALSE
SMTN	hgnc:11126	SMTN	NCI	14-Sep-17	NULL	4.773424657790409	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	NCI	14-Sep-17	NULL	0.012964857	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	2.333674277141977	ESTRONE-SULFATE	ncit:C1091	ESTRONE SULFATE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.020470827	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
STAT4	hgnc:11365	STAT4	NCI	14-Sep-17	NULL	0.8751278539282418	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
SULT1A2	hgnc:11454	SULT1A2	NCI	14-Sep-17	NULL	0.760980743	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	NCI	14-Sep-17	NULL	3.125456621172291	LANREOTIDE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	NCI	14-Sep-17	NULL	0.2059124362184098	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV396632	chembl:CHEMBL1623897	CHEMBL:CHEMBL1623897	FALSE	FALSE	FALSE
TBP	hgnc:11588	TBP	NCI	14-Sep-17	NULL	0.5933070196123672	VP-16	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	ENPIROLINE	ncit:C75267	ENPIROLINE	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.030168154	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.3365876361262467	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
THBD	hgnc:11784	THBD	NCI	14-Sep-17	NULL	1.093909817410302	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
THBD	hgnc:11784	THBD	NCI	14-Sep-17	NULL	0.2651902587661338	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
THRSP	hgnc:11800	THRSP	NCI	14-Sep-17	NULL	0.5707355569097228	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	NCI	14-Sep-17	NULL	NULL	TAXANES	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	OncoKB	23-Jul-20	NULL	0.2917092846427472	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
FLT3	hgnc:3765	FLT3	OncoKB	23-Jul-20	NULL	NULL	High Dose Chemotherapy	NULL	NULL	NULL	NULL	NULL
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	[3H]-PHORBOL 12,13-DIBUTYRATE	chembl:CHEMBL27768	CHEMBL:CHEMBL27768	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	OncoKB	23-Jul-20	NULL	0.2917092846427472	Pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	OncoKB	23-Jul-20	NULL	0.4234489615781814	Iodine I 131-6-Beta-Iodomethyl-19-Norcholesterol	ncit:C74052	IODINE I 131-6-BETA-IODOMETHYL-19-NORCHOLESTEROL	FALSE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.021590325	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	OncoKB	23-Jul-20	NULL	4.702860988936115	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	OncoKB	23-Jul-20	NULL	0.040515178	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	OncoKB	23-Jul-20	NULL	0.082754407	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.035670972	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
TSC1	hgnc:12362	TSC1	OncoKB	23-Jul-20	NULL	2.625383561784725	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	0.9010915075351876	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	OncoKB	23-Jul-20	NULL	0.1657439117288336	Copanlisib	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
CDA	hgnc:1712	CDA	PharmGKB	4/5/24	NULL	NULL	ara-CTP	NULL	NULL	NULL	NULL	NULL
VKORC1	hgnc:23663	VKORC1	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
FPR2	hgnc:3827	FPR2	DTC	9/2/20	NULL	2.917092846427472	N-FORMYLMETHIONYL-LEUCYLPHENYLALANINE	iuphar.ligand:1022	FMET-LEU-PHE	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	NULL	latonduine a	NULL	NULL	NULL	NULL	NULL
ERCC1	hgnc:3433	ERCC1	PharmGKB	4/5/24	NULL	1.750255707856483	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
SLC28A1	hgnc:11001	SLC28A1	PharmGKB	4/5/24	NULL	NULL	ara-CTP	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	GRAMINE	ncit:C64181	GRAMINE	FALSE	FALSE	FALSE
ATP2B1	hgnc:814	ATP2B1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.010128795	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.06638138	troleandomycin	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.1017590527823536	doxazosin	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.2734774543525755	methoxamine	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
TLR3	hgnc:11849	TLR3	PharmGKB	4/5/24	NULL	2.625383561784724	Measles vaccines	wikidata:Q6804161	MEASLES VACCINE	FALSE	FALSE	FALSE
SLC28A3	hgnc:16484	SLC28A3	PharmGKB	4/5/24	NULL	NULL	ara-CTP	NULL	NULL	NULL	NULL	NULL
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.1315981735230438	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP3A43	hgnc:17450	CYP3A43	PharmGKB	4/5/24	NULL	0.8334550989792778	ticagrelor	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
FMO1	hgnc:3769	FMO1	PharmGKB	4/5/24	NULL	0.5385402178019949	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.067403943	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	PharmGKB	4/5/24	NULL	0.2108741816694558	midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.473042083	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
ZNF613	hgnc:25827	ZNF613	PharmGKB	4/5/24	NULL	0.5385402178019949	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-3792	chembl:CHEMBL582983	CHEMBL:CHEMBL582983	FALSE	FALSE	FALSE
BAG6	hgnc:13919	BAG6	PharmGKB	4/5/24	NULL	2.143170254518142	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.1215455352678113	aceclofenac	rxcui:16689	ACECLOFENAC	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.016206071	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	IPRONIAZID SULFATE	chembl:CHEMBL1534878	IPRONIAZID SULFATE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	LEVDOBUTAMINE	ncit:C166431	LEVDOBUTAMINE	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	PharmGKB	4/5/24	NULL	0.2983390411119005	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.066011799	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	NULL	thioxanthine	NULL	NULL	NULL	NULL	NULL
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	1.312691780892362	fenoterol	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	ECADOTRIL	ncit:C75238	ECADOTRIL	FALSE	FALSE	FALSE
PRSS53	hgnc:34407	PRSS53	PharmGKB	4/5/24	NULL	11.13799086817762	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.03729238	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
WWOX	hgnc:12799	WWOX	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.092933931	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
CFAP44	hgnc:25631	CFAP44	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	3.750547945	bacampicillin	rxcui:18687	BACAMPICILLIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.033243223	calcium channel blockers	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1166837138570989	atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
RBX1	hgnc:9928	RBX1	PharmGKB	4/5/24	NULL	0.4167275494896389	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
IL13	hgnc:5973	IL13	PharmGKB	4/5/24	NULL	NULL	Hepatitis vaccines	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.058733413	tenofovir alafenamide	rxcui:1721603	TENOFOVIR ALAFENAMIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	Melatonin receptor agonists	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.4487835148349957	daptomycin	rxcui:22299	DAPTOMYCIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.1121958787087489	elacridar	ncit:C73318	ELACRIDAR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.004315226	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.033658764	quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.024932417	teniposide	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.024932417	saquinavir	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
SERPINA3	hgnc:16	SERPINA3	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.039214094	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	PharmGKB	4/5/24	NULL	NULL	Iodine (131I) compounds	NULL	NULL	NULL	NULL	NULL
PBK	hgnc:18282	PBK	DTC	9/2/20	NULL	0.2561349816375341	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
SLC12A1	hgnc:10910	SLC12A1	PharmGKB	4/5/24	NULL	NULL	sulfonamides, plain	NULL	NULL	NULL	NULL	NULL
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CYP4B1	hgnc:2644	CYP4B1	PharmGKB	4/5/24	NULL	0.7095631248066824	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	PharmGKB	4/5/24	NULL	1.040600372117402	quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
PCSK9	hgnc:20001	PCSK9	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	0.1339481409073839	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	MENTHOFURAN	chembl:CHEMBL1522900	MENTHOFURAN	FALSE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.2838252499226729	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004557958	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.2134458180312784	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ADAM33	hgnc:15478	ADAM33	PharmGKB	4/5/24	NULL	1.280674908	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
FCER2	hgnc:3612	FCER2	PharmGKB	4/5/24	NULL	0.5122699632750682	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
TAAR6	hgnc:20978	TAAR6	PharmGKB	4/5/24	NULL	1.280674908	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.058602312	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
TRDN	hgnc:12261	TRDN	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ITPA	hgnc:6176	ITPA	PharmGKB	4/5/24	NULL	0.6403374540938354	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	PharmGKB	4/5/24	NULL	0.039939912	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CDK19	hgnc:19338	CDK19	DTC	9/2/20	NULL	0.047952211	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1312691780892362	norfloxacin	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
CSRNP3	hgnc:30729	CSRNP3	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	NULL	egfr inhibitors	NULL	NULL	NULL	NULL	NULL
SLCO1A2	hgnc:10956	SLCO1A2	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.033615667	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
CALM1	hgnc:1442	CALM1	PharmGKB	4/5/24	NULL	0.201178817	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
GCLC	hgnc:4311	GCLC	PharmGKB	4/5/24	NULL	0.7501095890813498	sulfamethoxazole	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	PharmGKB	4/5/24	NULL	0.1093909817410302	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	PharmGKB	4/5/24	NULL	0.5860231164698047	levetiracetam	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	NULL	hydroxybupropion	NULL	NULL	NULL	NULL	NULL
RGS5	hgnc:10001	RGS5	PharmGKB	4/5/24	NULL	0.9460841664089098	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
MIR4481	hgnc:41781	MIR4481	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
RALBP1	hgnc:9841	RALBP1	PharmGKB	4/5/24	NULL	0.1852122442176172	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.061737415	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.2160809515872201	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CXCL12	hgnc:10672	CXCL12	PharmGKB	4/5/24	NULL	0.1620607136904151	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.004216468	bromazepam	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.04427291	viloxazine	rxcui:11196	VILOXAZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.025298806	cevimeline	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.024130364	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
SLC22A6	hgnc:10970	SLC22A6	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	0.4118248724368196	naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
XRCC3	hgnc:12830	XRCC3	PharmGKB	4/5/24	NULL	0.4167275494896388	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CLMN	hgnc:19972	CLMN	PharmGKB	4/5/24	NULL	0.7001022831425933	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	0.4118248724368196	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.011279843	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
TBC1D32	hgnc:21485	TBC1D32	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	NULL	FOLFIRINOX	NULL	NULL	NULL	NULL	NULL
SLC22A6	hgnc:10970	SLC22A6	PharmGKB	4/5/24	NULL	0.4861821410712453	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.046840028	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
PRKCA	hgnc:9393	PRKCA	PharmGKB	4/5/24	NULL	0.1093909817410302	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
ITPA	hgnc:6176	ITPA	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
TGFB1	hgnc:11766	TGFB1	PharmGKB	4/5/24	NULL	NULL	Iodine (131I) compounds	NULL	NULL	NULL	NULL	NULL
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	NULL	ethinyl estradiol / norelgestromin	NULL	NULL	NULL	NULL	NULL
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.01763778	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	1.022876712383659	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.3125456621172291	hydrocortisone	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	DTC	9/2/20	NULL	3.750547945	METACETAMOL	ncit:C81395	METACETAMOL	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	PharmGKB	4/5/24	NULL	0.217423069	bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	PharmGKB	4/5/24	NULL	0.021340244	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
ZNF542P	hgnc:25393	ZNF542P	PharmGKB	4/5/24	NULL	2.100306849	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
F2	hgnc:3535	F2	PharmGKB	4/5/24	NULL	NULL	ethinyl estradiol / norelgestromin	NULL	NULL	NULL	NULL	NULL
F2	hgnc:3535	F2	PharmGKB	4/5/24	NULL	NULL	antithrombotic agents	NULL	NULL	NULL	NULL	NULL
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	DNDI1417777	chembl:CHEMBL1412002	CHEMBL:CHEMBL1412002	FALSE	FALSE	FALSE
CRP	hgnc:2367	CRP	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.1071585127259071	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CDH2	hgnc:1759	CDH2	PharmGKB	4/5/24	NULL	0.3125456621172291	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.036770078	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
DCTD	hgnc:2710	DCTD	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
DPYD	hgnc:3012	DPYD	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
ADORA2A	hgnc:263	ADORA2A	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	LENPERONE	ncit:C73287	LENPERONE	FALSE	FALSE	FALSE
GSTM5	hgnc:4637	GSTM5	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.078136416	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.7001022831425933	SJ000160630	chembl:CHEMBL591404	CHEMBL:CHEMBL591404	FALSE	FALSE	FALSE
SLC22A9	hgnc:16261	SLC22A9	PharmGKB	4/5/24	NULL	0.9376369863516874	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PPP2R5D	hgnc:9312	PPP2R5D	PharmGKB	4/5/24	NULL	0.9723642821424908	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	NULL	antithrombotic agents	NULL	NULL	NULL	NULL	NULL
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.3947945205691315	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
NFATC2	hgnc:7776	NFATC2	PharmGKB	4/5/24	NULL	0.201178817	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ITGA2B	hgnc:6138	ITGA2B	PharmGKB	4/5/24	NULL	3.500511415712967	tirofiban	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.019346968	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
EYS	hgnc:21555	EYS	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
SIK3	hgnc:29165	SIK3	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
HMGCR	hgnc:5006	HMGCR	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CELSR2	hgnc:3231	CELSR2	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CHRNA1	hgnc:1955	CHRNA1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.030147945	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
LPA	hgnc:6667	LPA	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
NPC1L1	hgnc:7898	NPC1L1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.002519804	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
SLC15A1	hgnc:10920	SLC15A1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
SREBF1	hgnc:11289	SREBF1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	3,7-DIMETHOXYFLAVONE	chembl:CHEMBL1449187	3,7-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
PRDM16	hgnc:14000	PRDM16	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
HLA-G	hgnc:4964	HLA-G	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00908123	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
CXCL5	hgnc:10642	CXCL5	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	MOMETASONE FUROATE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.044498026	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.1121958787087489	disopyramide	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
BCHE	hgnc:983	BCHE	PharmGKB	4/5/24	NULL	0.062509132	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.087585774	3,4-methylenedioxymethamphetamine	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.4039051633514962	edoxaban	rxcui:1599538	EDOXABAN	TRUE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.2885036881082115	amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	hydroxybupropion	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.027121731	dipyrone	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.004931224	flunitrazepam	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.019724895	3,4-methylenedioxymethamphetamine	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.014597629	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.024108205	rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	16alpha-hydroxytestosterone	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	11a-hydroxyprogesterone	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	NULL	egfr inhibitors	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	0.2083637747448194	capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
SELE	hgnc:10718	SELE	PharmGKB	4/5/24	NULL	0.2580229544751572	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	0.045226246	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	PharmGKB	4/5/24	NULL	0.056258219	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.760980743	ezetimibe / simvastatin	wikidata:Q48566705	EZETIMIBE / SIMVASTATIN	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	antithrombotic agents	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	CICHORIC ACID	chembl:CHEMBL282731	CICHORIC ACID	FALSE	FALSE	FALSE
SFRP5	hgnc:10779	SFRP5	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
POU5F1	hgnc:9221	POU5F1	PharmGKB	4/5/24	NULL	0.5357925636295356	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.596678082	disopyramide	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	0.6250913242344582	NORHARMANE	iuphar.ligand:8222	BETA-CARBOLINE	FALSE	FALSE	FALSE
EIF4E2	hgnc:3293	EIF4E2	PharmGKB	4/5/24	NULL	0.4861821410712453	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PRKAA2	hgnc:9377	PRKAA2	PharmGKB	4/5/24	NULL	0.4895820161836317	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.006705961	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
DSCAM	hgnc:3039	DSCAM	PharmGKB	4/5/24	NULL	0.4861821410712453	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	1.591141552596802	exenatide	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.021138354	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ARID5B	hgnc:17362	ARID5B	PharmGKB	4/5/24	NULL	5.000730593875666	Glucarpidase	rxcui:1242127	GLUCARPIDASE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.038049037	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
MLN	hgnc:7141	MLN	PharmGKB	4/5/24	NULL	2.143170254518142	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	NULL	amlodipine / atorvastatin / perindopril arginine	NULL	NULL	NULL	NULL	NULL
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.3804903712731485	viloxazine	rxcui:11196	VILOXAZINE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	PharmGKB	4/5/24	NULL	NULL	Iodine (131I) compounds	NULL	NULL	NULL	NULL	NULL
PROS1	hgnc:9456	PROS1	PharmGKB	4/5/24	NULL	NULL	ethinyl estradiol / norelgestromin	NULL	NULL	NULL	NULL	NULL
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	NULL	ethinyl estradiol / norelgestromin	NULL	NULL	NULL	NULL	NULL
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.1121958787087489	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
SEMA3C	hgnc:10725	SEMA3C	PharmGKB	4/5/24	NULL	1.666910197958555	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PROS1	hgnc:9456	PROS1	PharmGKB	4/5/24	NULL	NULL	estradiol / progesterone	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	PharmGKB	4/5/24	NULL	0.9842513760562132	ivosidenib	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
LIPC	hgnc:6619	LIPC	PharmGKB	4/5/24	NULL	0.3500511415712966	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	NULL	estradiol / progesterone	NULL	NULL	NULL	NULL	NULL
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.018619742	FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
KCNJ6	hgnc:6267	KCNJ6	PharmGKB	4/5/24	NULL	0.8751278539282417	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
ADCK1	hgnc:19038	ADCK1	PharmGKB	4/5/24	NULL	8.751278539282415	paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	NSC-693571	chembl:CHEMBL1287983	CHEMBL:CHEMBL1287983	FALSE	FALSE	FALSE
ADCY9	hgnc:240	ADCY9	PharmGKB	4/5/24	NULL	0.4039051633514962	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.1272913242077442	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	PharmGKB	4/5/24	NULL	0.2616661357260523	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TOFISOPAM	rxcui:38365	TOFISOPAM	FALSE	FALSE	FALSE
ANXA11	hgnc:535	ANXA11	PharmGKB	4/5/24	NULL	0.3281729452230906	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.2287915957982331	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
A2M	hgnc:7	A2M	PharmGKB	4/5/24	NULL	NULL	Enzymes	NULL	NULL	NULL	NULL	NULL
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.1047012387551236	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	0.088996053	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.3889457128569963	oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	NULL	Antifungals For Systemic Use	NULL	NULL	NULL	NULL	NULL
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	CLOMIPRAMINE HYDROCHLORIDE	rxcui:81984	CLOMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAGEA12	hgnc:6799	MAGEA12	TALC	12-May-16	vaccine	NULL	MAGE-12 PEPTIDE VACCINE (EMULSIFIED INMONTANIDE ISA-51)	NULL	NULL	NULL	NULL	NULL
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	GNF-PF-4046	chembl:CHEMBL600090	CHEMBL:CHEMBL600090	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	NULL	0.2465148884304905	VADIMEZAN	ncit:C2504	VADIMEZAN	FALSE	FALSE	TRUE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	1.184383561707394	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	NULL	ALITRETIONINE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10826	hgnc:9865	RARB	TdgClinicalTrial	Jan-14	NULL	NULL	ALITRETIONINE	NULL	NULL	NULL	NULL	NULL
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.028929846	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TdgClinicalTrial	Jan-14	NULL	NULL	ALITRETIONINE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P19793	hgnc:10477	RXRA	TdgClinicalTrial	Jan-14	NULL	NULL	ALITRETIONINE	NULL	NULL	NULL	NULL	NULL
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	D-TRYPTOPHAN	drugbank:DB03225	D-TRYPTOPHAN	FALSE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TdgClinicalTrial	Jan-14	NULL	NULL	ALITRETIONINE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48443	hgnc:10479	RXRG	TdgClinicalTrial	Jan-14	NULL	NULL	ALITRETIONINE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1605739181519709	ALKS 33	rxcui:2559612	SAMIDORPHAN	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	NULL	ALT-110	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08887	hgnc:6019	IL6R	TdgClinicalTrial	Jan-14	NULL	NULL	ALC-0061	NULL	NULL	NULL	NULL	NULL
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	(20S,21R)-FLUOROCAMPTOTHECIN	chembl:CHEMBL2435326	(20S,21R)-FLUOROCAMPTOTHECIN	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.2586584789935689	AM-101	chembl:CHEMBL2364609	ESKETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	NULL	ANHYDROVINBLASTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9UHF1	hgnc:20594	EGFL7	TdgClinicalTrial	Jan-14	NULL	NULL	ANTI-EGFL7	NULL	NULL	NULL	NULL	NULL
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.100976291	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
UNIPROT:O14786	hgnc:8004	NRP1	TdgClinicalTrial	Jan-14	NULL	NULL	ANTI-NRP1 MAB	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	NULL	ARI-2243	NULL	NULL	NULL	NULL	NULL
UNIPROT:P36507	hgnc:6842	MAP2K2	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	ARRY-300	chembl:CHEMBL3545359	ARRY-300	FALSE	FALSE	FALSE
UNIPROT:P04275	hgnc:12726	VWF	TdgClinicalTrial	Jan-14	NULL	5.527123287967842	ARC1779	ncit:C95742	EGAPTIVON PEGOL	FALSE	FALSE	FALSE
UNIPROT:P27361	hgnc:6877	MAPK3	TdgClinicalTrial	Jan-14	NULL	0.038104261	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
UNIPROT:P33681	hgnc:1700	CD80	TdgClinicalTrial	Jan-14	NULL	NULL	ASP2408	NULL	NULL	NULL	NULL	NULL
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.003155509	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P42081	hgnc:1705	CD86	TdgClinicalTrial	Jan-14	NULL	NULL	ASP2408	NULL	NULL	NULL	NULL	NULL
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	DERRUBONE	chembl:CHEMBL412010	DERRUBONE	FALSE	FALSE	FALSE
UNIPROT:Q92934	hgnc:936	BAD	TdgClinicalTrial	Jan-14	NULL	0.546954909	AT-101	ncit:C187300	ANTI-CD19 CAR T CELLS AT101	FALSE	FALSE	TRUE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	NULL	ATHX-105	NULL	NULL	NULL	NULL	NULL
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	NULL	AVN-101	NULL	NULL	NULL	NULL	NULL
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	NULL	AVN-211	NULL	NULL	NULL	NULL	NULL
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.034184682	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
UNIPROT:P42224	hgnc:11362	STAT1	TdgClinicalTrial	Jan-14	NULL	NULL	AVT-02 UE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48443	hgnc:10479	RXRG	TdgClinicalTrial	Jan-14	NULL	1.988926940746004	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.042898424	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
UNIPROT:P35408	hgnc:9596	PTGER4	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	BGC20-1531	iuphar.ligand:3380	BGC201531	FALSE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.693795846312725	BEPOTASTINE	rxcui:658552	BEPOTASTINE BESILATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	6.300920548	BMS 936564	ncit:C95755	ULOCUPLUMAB	FALSE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.030073122	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
UNIPROT:P43115	hgnc:9595	PTGER3	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	BIMATOPROST	rxcui:283810	BIMATOPROST	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	0.8078103267029922	CAPROSPINOL	drugbank:DB05263	CAPROSPINOL	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.066047385	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
UNIPROT:Q99788	hgnc:2121	CMKLR1	TdgClinicalTrial	Jan-14	NULL	NULL	CCX832	NULL	NULL	NULL	NULL	NULL
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	0.2524407270946851	HISTAMINE	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	NULL	CNDO101	NULL	NULL	NULL	NULL	NULL
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.5250767123569451	GW559768X	chembl:CHEMBL237347	GW559768X	FALSE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	2.972132334095915	CIXUTUMUMAB	ncit:C79828	CIXUTUMUMAB	FALSE	TRUE	TRUE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.09869863	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.034118045	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	NULL	CS-3030	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20648	hgnc:819	ATP4A	TdgClinicalTrial	Jan-14	NULL	0.729273212	ESOMEPRAZOLE	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
UNIPROT:P21453	hgnc:3165	S1PR1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	FINGOLIMOD	rxcui:1012892	FINGOLIMOD	TRUE	TRUE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	COLFORSIN	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
UNIPROT:P48544	hgnc:6266	KCNJ5	TdgClinicalTrial	Jan-14	NULL	0.364636606	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	SB-205384	chembl:CHEMBL1256667	CHEMBL:CHEMBL1256667	FALSE	FALSE	FALSE
UNIPROT:P04049	hgnc:9829	RAF1	TdgClinicalTrial	Jan-14	NULL	NULL	C-RAF ANTISENSE OLIGONUCLEOTIDE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P61812	hgnc:11768	TGFB2	TdgClinicalTrial	Jan-14	NULL	15.00219178	LERDELIMUMAB	ncit:C170107	LERDELIMUMAB	FALSE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	LGD-1550	drugbank:DB05785	LGD-1550	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.013909317	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
UNIPROT:Q969P6	hgnc:29787	TOP1MT	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	LE-SN38	ncit:C95717	LIPOSOMAL SN-38	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	LEVOCETIRIZINE	rxcui:356887	LEVOCETIRIZINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.099446347	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.041344623	GUANIDINONALTRINDOLE	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
UNIPROT:Q9Y275	hgnc:11929	TNFSF13B	TdgClinicalTrial	Jan-14	NULL	19.69037671338543	LY2127399	ncit:C91727	TABALUMAB	FALSE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	LY-2189265	rxcui:1551291	DULAGLUTIDE	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	0.8078103267029922	MABT5102A	iuphar.ligand:6934	CRENEZUMAB	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.1158257453728555	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	CINALUKAST	ncit:C96709	CINALUKAST	FALSE	FALSE	FALSE
UNIPROT:P20273	hgnc:1643	CD22	TdgClinicalTrial	Jan-14	NULL	14.58546423213736	EPRATUZUMAB	ncit:C1887	EPRATUZUMAB	FALSE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	NULL	MDAM	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	NULL	MEM 1003	NULL	NULL	NULL	NULL	NULL
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	NSC-695801	chembl:CHEMBL461193	CHEMBL:CHEMBL461193	FALSE	FALSE	FALSE
UNIPROT:Q01668	hgnc:1391	CACNA1D	TdgClinicalTrial	Jan-14	NULL	NULL	MEM 1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:O60840	hgnc:1393	CACNA1F	TdgClinicalTrial	Jan-14	NULL	NULL	MEM 1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13698	hgnc:1397	CACNA1S	TdgClinicalTrial	Jan-14	NULL	NULL	MEM 1003	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	1.050153425	MELOGLIPTIN	ncit:C87620	MELOGLIPTIN	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1448487482363986	EPICATECHIN GALLATE	iuphar.ligand:12462	EPICATECHIN GALLATE	FALSE	FALSE	FALSE
UNIPROT:P00749	hgnc:9052	PLAU	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	WX-671	ncit:C73985	UPAMOSTAT	FALSE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	MKC-253	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	ML-10302	iuphar.ligand:235	ML 10302	FALSE	FALSE	FALSE
UNIPROT:O15397	hgnc:9853	IPO8	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	0.048708415	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.068637479	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	VITAMIN K3H2	chembl:CHEMBL1405447	VITAMIN K3H2	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	IODINE	rxcui:5933	IODINE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	NULL	MU DELTA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	NULL	MU DELTA	NULL	NULL	NULL	NULL	NULL
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.044498026	GUANIDINONALTRINDOLE	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
UNIPROT:P51959	hgnc:1592	CCNG1	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	MX-DNG1	drugbank:DB05604	MX-DNG1	FALSE	FALSE	FALSE
UNIPROT:P33402	hgnc:4684	GUCY1A2	TdgClinicalTrial	Jan-14	NULL	NULL	NCX 1510	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	NULL	NCX 1510	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.030038714	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	NULL	NEU-2000	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	NULL	NEU-2000	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	NULL	NEU-2000	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14957	hgnc:4587	GRIN2C	TdgClinicalTrial	Jan-14	NULL	NULL	NEU-2000	NULL	NULL	NULL	NULL	NULL
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	SJ000108787	chembl:CHEMBL603130	CHEMBL:CHEMBL603130	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	NULL	NEU-2000	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	NULL	NEU-2000	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TCMDC-124557	chembl:CHEMBL530682	CHEMBL:CHEMBL530682	FALSE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	NULL	NEU-2000	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004172574	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
UNIPROT:Q99705	hgnc:4479	MCHR1	TdgClinicalTrial	Jan-14	NULL	NULL	NGD-4715	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ALPHA-TERTHIENYL	chembl:CHEMBL90017	ALPHA-TERTHIENYL	FALSE	FALSE	FALSE
UNIPROT:Q8TDS4	hgnc:24827	HCAR2	TdgClinicalTrial	Jan-14	NULL	NULL	NIACIN RECEPTOR AGONIST	NULL	NULL	NULL	NULL	NULL
UNIPROT:P49019	hgnc:16824	HCAR3	TdgClinicalTrial	Jan-14	NULL	NULL	NIACIN RECEPTOR AGONIST	NULL	NULL	NULL	NULL	NULL
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	NI-0401	chembl:CHEMBL1743020	FORALUMAB	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	NULL	NRP290	NULL	NULL	NULL	NULL	NULL
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	NULL	NRP290	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	NULL	NRP290	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1751715470748774	OXYMORPHONE	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.2333674277141978	XANTHOANGELOL B	chembl:CHEMBL494082	XANTHOANGELOL B	FALSE	FALSE	FALSE
UNIPROT:P09038	hgnc:3676	FGF2	TdgClinicalTrial	Jan-14	NULL	1.135300999690692	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.3017682254924971	PEGINTERFERON ALFA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
UNIPROT:P01138	hgnc:7808	NGF	TdgClinicalTrial	Jan-14	NULL	NULL	PG110	NULL	NULL	NULL	NULL	NULL
UNIPROT:P19838	hgnc:7794	NFKB1	TdgClinicalTrial	Jan-14	NULL	NULL	PG-490-88	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002188184	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
UNIPROT:Q00653	hgnc:7795	NFKB2	TdgClinicalTrial	Jan-14	NULL	NULL	PG-490-88	NULL	NULL	NULL	NULL	NULL
LDLR	hgnc:6547	LDLR	DTC	9/2/20	NULL	3.387591692625451	PF-429242	chembl:CHEMBL233611	CHEMBL:CHEMBL233611	FALSE	FALSE	FALSE
UNIPROT:P08842	hgnc:11425	STS	TdgClinicalTrial	Jan-14	NULL	NULL	PGL2001	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9Y251	hgnc:5164	HPSE	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	PG545	ncit:C95202	PIXATIMOD	FALSE	FALSE	FALSE
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	PH-797804	drugbank:DB07941	PH-797804	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	DESVENLAFAXINE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.6226206075378794	PRIDOPIDINE	ncit:C170349	PRIDOPIDINE	FALSE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	NULL	PRX-3140	NULL	NULL	NULL	NULL	NULL
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	NULL	SB-509	NULL	NULL	NULL	NULL	NULL
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	0.33338204	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P24941	hgnc:1771	CDK2	TdgClinicalTrial	Jan-14	NULL	0.292250489	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
UNIPROT:Q7L0J3	hgnc:20566	SV2A	TdgClinicalTrial	Jan-14	NULL	21.00306849427779	SELETRACETAM	ncit:C66534	SELETRACETAM	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.09055649	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1403266238077355	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P62942	hgnc:3711	FKBP1A	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	TC-5214	chembl:CHEMBL2103881	DEXMECAMYLAMINE	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.2641230947469542	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
UNIPROT:P42263	hgnc:4573	GRIA3	TdgClinicalTrial	Jan-14	NULL	0.2778183663264259	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.1229687850953032	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	TESOFENSINE	ncit:C66589	TESOFENSINE	FALSE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.3763990769583835	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TdgClinicalTrial	Jan-14	NULL	0.1376949420516464	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P20594	hgnc:7944	NPR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	CARDIODILATIN	drugbank:DB15591	ATRIAL NATRIURETIC PEPTIDE	FALSE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.084553416	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
UNIPROT:P49765	hgnc:12681	VEGFB	TdgClinicalTrial	Jan-14	NULL	NULL	VEGF-2	NULL	NULL	NULL	NULL	NULL
UNIPROT:P13639	hgnc:3214	EEF2	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	VB4-845	ncit:C61307	OPORTUZUMAB MONATOX	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.8468979231563628	VAPITADINE	ncit:C96721	VAPITADINE	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	1.202465753489187	FLUTICASONE FUROATE	rxcui:705022	FLUTICASONE FUROATE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	NULL	VI-0134	NULL	NULL	NULL	NULL	NULL
UNIPROT:O95264	hgnc:5298	HTR3B	TdgClinicalTrial	Jan-14	NULL	NULL	VI-0134	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8WXA8	hgnc:24003	HTR3C	TdgClinicalTrial	Jan-14	NULL	NULL	VI-0134	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q70Z44	hgnc:24004	HTR3D	TdgClinicalTrial	Jan-14	NULL	NULL	VI-0134	NULL	NULL	NULL	NULL	NULL
UNIPROT:A5X5Y0	hgnc:24005	HTR3E	TdgClinicalTrial	Jan-14	NULL	NULL	VI-0134	NULL	NULL	NULL	NULL	NULL
UNIPROT:P06756	hgnc:6150	ITGAV	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	VOLOCIXIMAB	ncit:C48426	VOLOCIXIMAB	FALSE	FALSE	TRUE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.5016656487486736	CALCIPOTRIOL	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.025827679	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.058341857	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.040703621	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.059667808	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.067317527	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1376949420516464	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TdgClinicalTrial	Jan-14	NULL	2.100306849	DICHLORPHENAMIDE	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2031244535229961	DICYCLOMINE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.2308029504865691	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.05814803	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.05814803	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.07699072	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.073089743	FLUOXYMESTERONE	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
UNIPROT:Q09470	hgnc:6218	KCNA1	TdgClinicalTrial	Jan-14	NULL	0.2419708351875322	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.039390601	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.032769506	LISURIDE	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.3211478363039418	LEVORPHANOL	rxcui:6378	LEVORPHANOL	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1132444383228493	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.074690855	LISURIDE	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.3211478363039418	LEVOMETHADYL ACETATE	rxcui:237005	LEVOMETHADYL	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.1117184494376478	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.1209854175937661	MECLIZINE	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
UNIPROT:P15538	hgnc:2591	CYP11B1	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	METYRAPONE	rxcui:6923	METYRAPONE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.056097939	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	METOCURINE IODIDE	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.09745299	NANDROLONE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
UNIPROT:Q9GZZ6	hgnc:13800	CHRNA10	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	PENTOLINIUM	ncit:C77367	PENTOLINIUM	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2004109589148645	PARAMETHASONE	rxcui:7910	PARAMETHASONE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	TRIDIHEXETHYL	rxcui:38617	TRIDIHEXETHYL	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.2308029504865691	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.2678962818147678	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.2220197515251353	DEXMEDETOMIDINE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.070197421	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TEND	1-Aug-11	NULL	1.790034246671403	ENPROFYLLINE	ncit:C74327	ENPROFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TEND	1-Aug-11	NULL	2.812910959055062	EPOPROSTENOL	rxcui:8814	EPOPROSTENOL	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	0.7001022831425934	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.08780547	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.084553416	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	2.917092846427472	ACETOHEXAMIDE	rxcui:173	ACETOHEXAMIDE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.082171629	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.4039051633514962	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TEND	1-Aug-11	NULL	0.086861325	ETANERCEPT	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.05309168	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.027276712	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
UNIPROT:P51787	hgnc:6294	KCNQ1	TEND	1-Aug-11	NULL	0.3977853881492006	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.079557078	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.1884246575443582	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.016161179	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.084383562	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
UNIPROT:P00519	hgnc:76	ABL1	TEND	1-Aug-11	NULL	0.1108075556053025	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TEND	1-Aug-11	NULL	3.281729452230906	INTERFERON ALFA-N3	rxcui:612937	INTERFERON ALFA-N3	TRUE	TRUE	TRUE
UNIPROT:P48551	hgnc:5433	IFNAR2	TEND	1-Aug-11	NULL	6.563458904461812	INTERFERON ALFACON-1	rxcui:59744	INTERFERON ALFACON-1	TRUE	TRUE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.4375639269641208	10-HYDROXYEVODIAMINE	chembl:CHEMBL2171812	CHEMBL:CHEMBL2171812	FALSE	FALSE	FALSE
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TEND	1-Aug-11	NULL	0.6563458904461812	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.015184405	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TEND	1-Aug-11	NULL	0.7343730242754476	ISOSORBIDE DINITRATE	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.1117184494376478	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.099446347	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1035654265003836	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TEND	1-Aug-11	NULL	0.2344092465879218	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.070448575	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TEND	1-Aug-11	NULL	1.166837138570988	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.07767407	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.066577774	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.074797252	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.083257407	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.091796628	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.1767935058440892	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-4998	chembl:CHEMBL585795	CHEMBL:CHEMBL585795	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.093596562	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.2234368988752957	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.1250182648468916	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P62942	hgnc:3711	FKBP1A	TEND	1-Aug-11	NULL	0.4688184931758437	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	BN-AO-014	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	BN-GU-005-DHP	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	AV-965	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	PF-885706	NULL	NULL	NULL	NULL	NULL
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	1.363835616511545	GOSSYPETIN-8-GLUCOSIDE	chembl:CHEMBL402915	CHEMBL:CHEMBL402915	FALSE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	NULL	HPP-851	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	ASP-3652	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Lu-02-750	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-8418	drugbank:DB13102	AZD-8418	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.000833098	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	NULL	CPP -15	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	U-73122	iuphar.ligand:5283	U73122	FALSE	FALSE	FALSE
PEPTIDE TYROSINE TYROSINE PYY	hgnc:9748	PYY	TTD	2020.06.01	NULL	NULL	Peptide YY 3-36	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	NULL	IMO-3100	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	IMO-3100	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
HEPATITIS C VIRUS DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	ChronVac-C hepatitis C DNA vaccine	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	WCK-1152	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-38093	drugbank:DB16893	S-38093	FALSE	FALSE	FALSE
MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN	hgnc:7467	MTTP	TTD	2020.06.01	NULL	NULL	KD020	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	DS-3078	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	NULL	PF-1228305	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	IL-2 XL	NULL	NULL	NULL	NULL	NULL
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	NULL	Talminogene laherparepvec	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005268681	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
LYASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	VT-464	ncit:C113652	SEVITERONEL	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	MIN-117	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	INX-189	chembl:CHEMBL1209734	BMS-986094	FALSE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.6563458904461812	COLFORSIN	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	EGFR/IGFR tandem adnectin	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	NULL	EGFR/IGFR tandem adnectin	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS MATURATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-955176	drugbank:DB15193	BMS-955176	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	3.281729452230906	Xmab-2513	chembl:CHEMBL4298133	XMAB-2513	FALSE	FALSE	FALSE
NEUROEPITHELIAL RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PH-80	NULL	NULL	NULL	NULL	NULL
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	NULL	BMS-933043	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 3	hgnc:8534	P2RX3	TTD	2020.06.01	NULL	NULL	AF-130	NULL	NULL	NULL	NULL	NULL
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
STROMAL CELL-DERIVED FACTOR 1	hgnc:10672	CXCL12	TTD	2020.06.01	NULL	NULL	REC-02	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	NULL	TD-0714	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006811217	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
HYDROXYCARBOXYLIC ACID RECEPTOR 3	hgnc:16824	HCAR3	TTD	2020.06.01	NULL	NULL	ARI-3037MO	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	NULL	BAY1193397	NULL	NULL	NULL	NULL	NULL
ADORA1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Neladenoson bialanate	ncit:C170208	NELADENOSON BIALANATE	FALSE	FALSE	FALSE
TTR	hgnc:12405	TTR	DTC	9/2/20	NULL	0.6250913242344582	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
IMMUNE CHECKPOINT	hgnc:2203	COL4A2	TTD	2020.06.01	NULL	NULL	AK107	NULL	NULL	NULL	NULL	NULL
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	0.6563458904461812	APG-115	ncit:C132991	ALRIZOMADLIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	0.1832728489902076	ASN003	ncit:C134967	BRAFV600/PI3K INHIBITOR ASN003	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.024605282	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	PHOSALONE	chembl:CHEMBL1528531	PHOSALONE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-2	hgnc:3676	FGF2	TTD	2020.06.01	NULL	0.7095631248066824	Bemarituzumab	ncit:C120040	BEMARITUZUMAB	FALSE	FALSE	FALSE
V-SET AND IMMUNOGLOBULIN DOMAIN-CONTAINING PROTEIN 9	hgnc:26838	TIGIT	TTD	2020.06.01	NULL	6.563458904461812	ASP8374	ncit:C141421	ANTI-TIGIT MONOCLONAL ANTIBODY ASP8374	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	DNDI1417722	chembl:CHEMBL1503190	CHEMBL:CHEMBL1503190	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CORT125281	ncit:C153309	EXICORILANT	FALSE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	FF-10101-01	drugbank:DB16050	FF-10101-01	FALSE	FALSE	FALSE
DNA SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	FF-10502-01	ncit:C125690	ANTIMETABOLITE FF-10502	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	0.6731752722524935	BMS-986158	drugbank:DB15435	BMS-986158	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.6177373086552295	ROEMERINE	chembl:CHEMBL36654	ROEMERINE	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IRX4204	ncit:C140551	RETINOID X RECEPTOR AGONIST IRX4204	FALSE	FALSE	FALSE
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	LXS196	ncit:C124796	DAROVASERTIB	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.009368006	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
DNA-DEPENDENT PROTEIN KINASE CATALYTIC	hgnc:9413	PRKDC	TTD	2020.06.01	NULL	NULL	M9831	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	MEDI4276	ncit:C126355	ANTI-HER2 ANTIBODY-DRUG CONJUGATE MEDI4276	FALSE	FALSE	FALSE
DNA-DEPENDENT PROTEIN KINASE CATALYTIC	hgnc:9413	PRKDC	TTD	2020.06.01	NULL	6.563458904461812	M3814	ncit:C120036	PEPOSERTIB	FALSE	FALSE	FALSE
SIGNAL TRANSDUCTION UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	OPB-111077	drugbank:DB16630	OPB-111077	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ORIC-101	iuphar.ligand:13167	ORIC-101	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	3.750547945	NLG802	ncit:C150393	INDOXIMOD PRODRUG NLG802	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.048260727	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	INCB57643	NULL	NULL	NULL	NULL	NULL
MAMMALIAN TARGET OF RAPAMYCIN COMPLEX 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
TARGET OF RAPAMYCIN COMPLEX 2 MAPKAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	BROMOCRIPTINE MESYLATE	rxcui:142426	BROMOCRIPTINE MESYLATE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE PIM	hgnc:8986	PIM1	TTD	2020.06.01	NULL	0.300043836	INCB53914	ncit:C124226	UZANSERTIB	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Annamycin liposomal	ncit:C25838	ANNAMYCIN LIPOSOMAL	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.9814517987980279	Debio 1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.034118045	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BBI503	ncit:C104745	AMCASERTIB	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.044498026	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
SOMATOSTATIN RECEPTOR TYPE 2	hgnc:11331	SSTR2	TTD	2020.06.01	NULL	2.917092846427472	PEN-221	ncit:C131562	NENDRATAREOTIDE UZATANSINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007149737	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
ADENOSINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NIR178	NULL	NULL	NULL	NULL	NULL
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	SJ000032154	chembl:CHEMBL591876	CHEMBL:CHEMBL591876	FALSE	FALSE	FALSE
PHOSPHORYLATED P68 RNA HELICASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RX-5902	ncit:C113293	P-P68 INHIBITOR RX-5902	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	NULL	VX-150	NULL	NULL	NULL	NULL	NULL
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	TCMDC-125310	chembl:CHEMBL582030	CHEMBL:CHEMBL582030	FALSE	FALSE	FALSE
CATERPILLER PROTEIN 1.1	hgnc:16400	NLRP3	TTD	2020.06.01	NULL	5.834185692854944	Dapansutrile	ncit:C166608	DAPANSUTRILE	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	DFD-11	NULL	NULL	NULL	NULL	NULL
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.027855529	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
ONCOSTATIN-M	hgnc:8506	OSM	TTD	2020.06.01	NULL	NULL	GSK2330811	NULL	NULL	NULL	NULL	NULL
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	NULL	JTE-451	NULL	NULL	NULL	NULL	NULL
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.045461187	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
CYTOKINE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06817024	NULL	NULL	NULL	NULL	NULL
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.009662803	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYTOSOLIC PHOSPHOLIPASE A2	NULL	NULL	TTD	2020.06.01	NULL	NULL	ZPL521	NULL	NULL	NULL	NULL	NULL
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALX-101	iuphar.ligand:9625	ROVAZOLAC	FALSE	FALSE	FALSE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cerdulatinib	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06700841	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	DIMERCAPROL	rxcui:3445	DIMERCAPROL	TRUE	FALSE	FALSE
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PRO22 topical gel	NULL	NULL	NULL	NULL	NULL
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.022554842	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
LANOSTEROL 14-ALPHA DEMETHYLASE	hgnc:2649	CYP51A1	TTD	2020.06.01	NULL	NULL	VT-1129	NULL	NULL	NULL	NULL	NULL
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.2430910705356227	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.017357908	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
OXYSTEROLS RECEPTOR LXR-BETA	hgnc:7965	NR1H2	TTD	2020.06.01	NULL	NULL	VTB-38543	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	OSAJIN	chembl:CHEMBL238188	OSAJIN	FALSE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nalbuphine extended release	NULL	NULL	NULL	NULL	NULL
OX40L RECEPTOR	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	3.500511415712966	GBR 830	chembl:CHEMBL4594546	TELAZORLIMAB	FALSE	FALSE	FALSE
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	0.1902451856365742	Cerdulatinib	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	2- (2,6-DIMETHOXYPHENOXYETHYL)AMINOMETHYL-1,4-BENZODIOXANE HYDROCHLORIDE (WB 4101)	chembl:CHEMBL556001	2- (2,6-DIMETHOXYPHENOXYETHYL)AMINOMETHYL-1,4-BENZODIOXANE HYDROCHLORIDE (WB 4101)	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	KX-01 ointment	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	NULL	Alpha-2c adrenergic receptor antagonist	NULL	NULL	NULL	NULL	NULL
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	1.029562181092048	SJ000120515	chembl:CHEMBL592314	CHEMBL:CHEMBL592314	FALSE	FALSE	FALSE
PLASMA KALLIKREIN	hgnc:6371	KLKB1	TTD	2020.06.01	NULL	NULL	KVD001	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	NULL	PMZ-2123	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-V/BETA-3	NULL	NULL	TTD	2020.06.01	NULL	NULL	SF0166	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	TF0023	NULL	NULL	NULL	NULL	NULL
DOPAMINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	EVK-001	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	RVT-103+RVT-104	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	LAM-001	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	OXYCARBOXIN	chembl:CHEMBL1712057	OXYCARBOXIN	FALSE	FALSE	FALSE
PROTEASOME	hgnc:9338	PRB2	TTD	2020.06.01	NULL	NULL	Marizomib IV	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAT 1004	chembl:CHEMBL3786673	EDASALONEXENT	FALSE	FALSE	FALSE
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	GBT440	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.1912847768149162	Goserelin	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.2641230947469542	BAY-57-9352	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	4.145342465975881	Finerenone	rxcui:2562811	FINERENONE	TRUE	FALSE	FALSE
SELECTIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	GMI-1070	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.025298806	Flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	S-110	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	DPV-001	ncit:C107681	ALLOGENEIC AUTOPHAGOSOME-ENRICHED VACCINE DPV-001	FALSE	FALSE	FALSE
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	VBY- 036	NULL	NULL	NULL	NULL	NULL
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	GK1-399	NULL	NULL	NULL	NULL	NULL
TPMT	hgnc:12014	TPMT	FDA	10-Apr-24	NULL	0.1666910197958555	Mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
INTERFERON ALPHA/BETA RECEPTOR 1	hgnc:5432	IFNAR1	TTD	2020.06.01	NULL	NULL	Belerofon	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GBL-310	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	2.763561643983921	AZD1981	iuphar.ligand:7680	AZD1981	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 5	hgnc:6933	MC5R	TTD	2020.06.01	NULL	NULL	MTC-896	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	FX-007	NULL	NULL	NULL	NULL	NULL
RECEPTOR UNSPECIFIC	hgnc:16147	MCM8	TTD	2020.06.01	NULL	NULL	BT-063	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.029515273	Nebivolol	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS 790052	rxcui:1606218	DACLATASVIR	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS 650032	rxcui:1652103	ASUNAPREVIR	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.5556367326528519	ICOTINIB	ncit:C138996	ICOTINIB	FALSE	FALSE	TRUE
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	2.333674277141978	GSK2816126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
PANCREATIC ALPHA-AMYLASE	hgnc:477	AMY2A	TTD	2020.06.01	NULL	NULL	Pancrecarb	NULL	NULL	NULL	NULL	NULL
PANCREATIC TRIACYLGLYCEROL LIPASE	hgnc:9155	PNLIP	TTD	2020.06.01	NULL	NULL	Pancrecarb	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	0.6783936852156912	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	MBO7133	drugbank:DB04999	MBO7133	FALSE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	XL652/XL014	NULL	NULL	NULL	NULL	NULL
G-PROTEIN COUPLED BILE ACID RECEPTOR 1	hgnc:19680	GPBAR1	TTD	2020.06.01	NULL	NULL	XL475	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US10022354, Example 152	NULL	NULL	NULL	NULL	NULL
G PROTEIN-COUPLED RECEPTOR KINASE 5	hgnc:4544	GRK5	TTD	2020.06.01	NULL	NULL	BDBM50173323	NULL	NULL	NULL	NULL	NULL
G PROTEIN-COUPLED RECEPTOR KINASE 5	hgnc:4544	GRK5	TTD	2020.06.01	NULL	NULL	BDBM50173327	NULL	NULL	NULL	NULL	NULL
G PROTEIN-COUPLED RECEPTOR KINASE 5	hgnc:4544	GRK5	TTD	2020.06.01	NULL	NULL	BDBM50173330	NULL	NULL	NULL	NULL	NULL
LEUCYL-CYSTEINYL AMINOPEPTIDASE	hgnc:6656	LNPEP	TTD	2020.06.01	NULL	NULL	US10023583, Example 24	NULL	NULL	NULL	NULL	NULL
LEUCYL-CYSTEINYL AMINOPEPTIDASE	hgnc:6656	LNPEP	TTD	2020.06.01	NULL	NULL	US10023583, Example 5	NULL	NULL	NULL	NULL	NULL
LEUCYL-CYSTEINYL AMINOPEPTIDASE	hgnc:6656	LNPEP	TTD	2020.06.01	NULL	NULL	US10023583, Example 8	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	4.773424657790408	Debio 0827	iuphar.ligand:7896	PL37	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.1124502911321247	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ACTIVIN RECEPTOR TYPE IB	hgnc:172	ACVR1B	TTD	2020.06.01	NULL	NULL	US10030004, Compound 19	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US10034861, Example 165	NULL	NULL	NULL	NULL	NULL
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	NULL	US10053465, 8	NULL	NULL	NULL	NULL	NULL
LEUCYL-CYSTEINYL AMINOPEPTIDASE	hgnc:6656	LNPEP	TTD	2020.06.01	NULL	NULL	US10059720, Example 84	NULL	NULL	NULL	NULL	NULL
KYNURENINE OXOGLUTARATE TRANSAMINASE II	hgnc:17929	AADAT	TTD	2020.06.01	NULL	NULL	US10065972, Example 281	NULL	NULL	NULL	NULL	NULL
KYNURENINE OXOGLUTARATE TRANSAMINASE II	hgnc:17929	AADAT	TTD	2020.06.01	NULL	NULL	US10065972, Example 396	NULL	NULL	NULL	NULL	NULL
CYTOMEGALOVIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	C06909	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10087167, Compound 3002	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10100051, Compound 1	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10100051, Compound 10	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US10092575, Example 141	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10149841, Compound 5	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10150740, Example 9	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.2546668357992238	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US10166249, Example 695	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9522888, 618	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US10174026, Example 99	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	AKOS020330656	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE C4 SYNTHASE	hgnc:6719	LTC4S	TTD	2020.06.01	NULL	NULL	US20160326143, 28	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE C4 SYNTHASE	hgnc:6719	LTC4S	TTD	2020.06.01	NULL	NULL	US20160326143, 3	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8481586, 15	NULL	NULL	NULL	NULL	NULL
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	1.250182648468916	AZD8330	iuphar.ligand:8474	AZD8330	FALSE	FALSE	TRUE
ACTIVATED CDC42 KINASE 1	hgnc:19297	TNK2	TTD	2020.06.01	NULL	NULL	US8481733, 106	NULL	NULL	NULL	NULL	NULL
ACTIVATED CDC42 KINASE 1	hgnc:19297	TNK2	TTD	2020.06.01	NULL	NULL	US8481733, 118	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8536181, A41	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8536181, C14	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ZAP-70	hgnc:12858	ZAP70	TTD	2020.06.01	NULL	NULL	US8546370, 102	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US8524917, 11	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 2	hgnc:3169	S1PR2	TTD	2020.06.01	NULL	NULL	US8975409, Example 13	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.1355619739303644	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8987457, 15	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8987457, 198	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 3B	hgnc:8779	PDE3B	TTD	2020.06.01	NULL	NULL	US8741907-compound-3	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE D1	hgnc:9067	PLD1	TTD	2020.06.01	NULL	NULL	US9127005, P2B	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	MHHFJYABEVJNEG-UHFFFAOYSA-N	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	YYDJCLCSBYCSCO-UHFFFAOYSA-N	NULL	NULL	NULL	NULL	NULL
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	US9156852, 83	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9187437, 8	NULL	NULL	NULL	NULL	NULL
AGGRECANASE-1	hgnc:220	ADAMTS4	TTD	2020.06.01	NULL	NULL	1607004-34-1	NULL	NULL	NULL	NULL	NULL
AGGRECANASE-1	hgnc:220	ADAMTS4	TTD	2020.06.01	NULL	NULL	US9206139, 4	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9216972, 132	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	US8614253, 29-1	NULL	NULL	NULL	NULL	NULL
DIBASIC-PROCESSING ENZYME	hgnc:8568	FURIN	TTD	2020.06.01	NULL	NULL	US9266828, E	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	BDBM50061601	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	BDBM50061608	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	BDBM50382283	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	CRWCYVOHVXAEMF-LBPRGKRZSA-N	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9346821, A-20	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	BDBM50363780	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9682991, 23	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9682991, 7	NULL	NULL	NULL	NULL	NULL
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	US9695118, 8	NULL	NULL	NULL	NULL	NULL
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	VAPBGCRAUJRZPO-UHFFFAOYSA-N	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9707205, 40	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9340511, 2	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9340511, 7	NULL	NULL	NULL	NULL	NULL
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	0.1377250393067396	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
CYSTATHIONINE GAMMA-LYASE	hgnc:2501	CTH	TTD	2020.06.01	NULL	NULL	5-Hydrazino-1H-tetrazole	NULL	NULL	NULL	NULL	NULL
CYSTATHIONINE GAMMA-LYASE	hgnc:2501	CTH	TTD	2020.06.01	NULL	NULL	Hydrazinoacetic acid	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	ZINC915379	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	BK7	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rosiglitazone + metformin	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rosiglitazone + simvastatin	NULL	NULL	NULL	NULL	NULL
ERBB4 TYROSINE KINASE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dacomitinib	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
ION CHANNEL UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-2927	iuphar.ligand:7704	AZD2927	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.4688184931758437	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
INHIBITOR OF APOPTOSIS PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
SRC TYROSINE KINASE SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
TUBULIN POLYMERIZATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	0.1229687850953032	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	RDEA-684	NULL	NULL	NULL	NULL	NULL
PROTON-COUPLED FOLATE TRANSPORTER	hgnc:30521	SLC46A1	TTD	2020.06.01	NULL	0.729273212	Folic Acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
CO-STIMULATORY MOLECULE 4-1BB	hgnc:11924	TNFRSF9	TTD	2020.06.01	NULL	NULL	Anti-CD137	NULL	NULL	NULL	NULL	NULL
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	NULL	LY2606368 MsOH H2O	NULL	NULL	NULL	NULL	NULL
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	NULL	CLR-1404	NULL	NULL	NULL	NULL	NULL
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.01495945	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
INTERLEUKIN 23 RECEPTOR	hgnc:19100	IL23R	TTD	2020.06.01	NULL	NULL	Anti-IL-23	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	NULL	F-7TG	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	NULL	Recombinant factor VIIa PEGylated liposomal	NULL	NULL	NULL	NULL	NULL
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	NULL	Pro-urokinase	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Selegiline	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	RWJ-416457	chembl:CHEMBL221877	CHEMBL:CHEMBL221877	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.055563673	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	NULL	CYT-013-IL1bQb	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	GZ402674	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	BAY-85-8102	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	EPI-12323 combination therapy	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.4953553890159858	OBP-801	drugbank:DB12279	OBP-801	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	0.1988926940746003	GnRH	chembl:CHEMBL1200511	GONADORELIN ACETATE	FALSE	FALSE	FALSE
PARATHYROID HORMONE RECEPTOR	hgnc:9609	PTH2R	TTD	2020.06.01	NULL	NULL	NPSP-795	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	NULL	Hypertension NCE	NULL	NULL	NULL	NULL	NULL
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.1215455352678113	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	NULL	T-2007	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	ZYH-7	NULL	NULL	NULL	NULL	NULL
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.049864835	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
CCR3 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASM8	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	ATD transdermal gel	NULL	NULL	NULL	NULL	NULL
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	BR-4628	NULL	NULL	NULL	NULL	NULL
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	NULL	MK-8342	NULL	NULL	NULL	NULL	NULL
SODIUM/GLUCOSE COTRANSPORTER 1	hgnc:11036	SLC5A1	TTD	2020.06.01	NULL	NULL	1614235 + 2330672	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	JNJ-17305600	NULL	NULL	NULL	NULL	NULL
ILEAL SODIUM/BILE ACID COTRANSPORTER	hgnc:10906	SLC10A2	TTD	2020.06.01	NULL	NULL	1614235 + 2330672	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	GW-42004	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.8334550989792777	ABT-806	ncit:C95206	DEPATUXIZUMAB	FALSE	TRUE	TRUE
TNFRSF8	hgnc:11923	TNFRSF8	MyCancerGenome	20-Jun-17	antibody	3.281729452230906	BRENTUXIMAB	ncit:C2007	BRENTUXIMAB	FALSE	TRUE	TRUE
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	GW-42004	NULL	NULL	NULL	NULL	NULL
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3314878234576672	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
HUMAN IMMUNODEFICIENCY VIRUS NUCLEOCAPSID P7	NULL	NULL	TTD	2020.06.01	NULL	NULL	HPH-116	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Zemab	NULL	NULL	NULL	NULL	NULL
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2917092846427472	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
ACTIVIN RECEPTOR-LIKE KINASE-1	hgnc:175	ACVRL1	TTD	2020.06.01	NULL	17.50255707856483	PF-03446962	ncit:C91073	ASCRINVACUMAB	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	V-950	NULL	NULL	NULL	NULL	NULL
DNA-DEPENDENT DNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CMX-001	rxcui:2599518	BRINCIDOFOVIR	TRUE	FALSE	FALSE
MACROPHAGE MIGRATION INHIBITORY FACTOR	hgnc:7097	MIF	TTD	2020.06.01	NULL	NULL	Anti-MIF antibodies	NULL	NULL	NULL	NULL	NULL
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.364636606	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	AGS-009	NULL	NULL	NULL	NULL	NULL
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDR-1018	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV1.3	hgnc:6221	KCNA3	TTD	2020.06.01	NULL	NULL	Debio-0824	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CMX-157	chembl:CHEMBL515564	TENOFOVIR EXALIDEX	FALSE	FALSE	FALSE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3241214273808303	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.4907258993990139	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	1.117184494376478	AZD-6088	chembl:CHEMBL5095221	AZD-6088	FALSE	FALSE	FALSE
INTERLEUKIN-5	hgnc:6016	IL5	TTD	2020.06.01	NULL	3.889457128569962	Benralizumab	rxcui:1989100	BENRALIZUMAB	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.2243917574174978	ANTIFUNGALS	ncit:C514	ANTIFUNGAL AGENT	FALSE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	3.182283105193605	S-888711	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
EGFR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	EGFR antisense DNA	ncit:C2617	EGFR ANTISENSE DNA	FALSE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	ARX-424	NULL	NULL	NULL	NULL	NULL
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	NU-100	NULL	NULL	NULL	NULL	NULL
HISTONE-LYSINE N-METHYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	EPZ-5676	ncit:C103179	PINOMETOSTAT	FALSE	FALSE	TRUE
AANAT	hgnc:19	AANAT	NCI	14-Sep-17	NULL	0.082300425	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
HEPATITIS B VIRUS REVERSE TRANSCRIPTASE PRIMING/DNA SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALAMIFOVIR	ncit:C77923	ALAMIFOVIR	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CD20Bi aATC	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD3	NULL	NULL	TTD	2020.06.01	NULL	NULL	CD20Bi aATC	NULL	NULL	NULL	NULL	NULL
GROWTH/DIFFERENTIATION FACTOR 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06252616	ncit:C166800	DOMAGROZUMAB	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	AD-03	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	NI-101	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	OMS824	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	AVE-8112	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	NULL	AVE-8112	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	NULL	AVE-8112	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	DCCCyB	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	Buprenorphine + naloxone	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.016829382	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
PARATHYROID HORMONE RECEPTOR	hgnc:9609	PTH2R	TTD	2020.06.01	NULL	26.25383561784724	BA-058	chembl:CHEMBL3301581	ABALOPARATIDE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4907258993990139	Hypericum	chemidplus:68917-49-7	ST. JOHN'S WORT	FALSE	FALSE	FALSE
PLASMODIUM DIHYDROOROTATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Avastin+/-Tarceva	NULL	NULL	NULL	NULL	NULL
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	NULL	TT-223	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	NS-7	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	DZ-2640	NULL	NULL	NULL	NULL	NULL
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	1.346350544504987	PEP	rxcui:34120	POLYESTRADIOL PHOSPHATE	TRUE	FALSE	FALSE
ADENOSINE DEAMINASE	hgnc:186	ADA	TTD	2020.06.01	NULL	0.06714536	Fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.1058622403945453	Mepivacaine	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.8607814956671229	Desogestrel	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Genaconazole	chembl:CHEMBL34139	GENACONAZOLE	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	SPH-1285	NULL	NULL	NULL	NULL	NULL
PRO-NEUREGULIN-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	GGF	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzphetamine	rxcui:1422	BENZPHETAMINE	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.4039051633514962	ANALGESICS	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
CANDIDA CHITIN SYNTHASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nikkomycin Z	drugbank:DB12939	NIKKOMYCIN Z	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	P32/98	NULL	NULL	NULL	NULL	NULL
AKR1C3	hgnc:386	AKR1C3	NCI	14-Sep-17	NULL	0.4118248724368196	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS TAT PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penicillamine	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PS-341	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	B-Lactams	NULL	NULL	NULL	NULL	NULL
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	8.751278539282415	FV-100	chembl:CHEMBL4297380	VALNIVUDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Olprinone	ncit:C90918	OLPRINONE	FALSE	FALSE	FALSE
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Methoxyestradiol	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	AjvW2	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Human neutral insulin	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.5933070196123671	Ramipril	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	RDP58	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.1405200835924027	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
MULTIDRUG RESISTANCE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzquinamide	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine	rxcui:8340	PIPERAZINE	TRUE	FALSE	FALSE
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	Human interferon alpha oral	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	BF-389	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.3006164383722967	Fluorometholone	rxcui:4491	FLUOROMETHOLONE	TRUE	FALSE	FALSE
INTRACELLULAR NITROREDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	SR-4554	NULL	NULL	NULL	NULL	NULL
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.3860858179095183	TRIBUTYRIN	ncit:C1260	TRIBUTYRIN	FALSE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetracycline	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	BrevaRex	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-24	hgnc:11346	IL24	TTD	2020.06.01	NULL	NULL	INGN-241	NULL	NULL	NULL	NULL	NULL
IMMUNOGLOBULIN E	hgnc:5522	IGHE	TTD	2020.06.01	NULL	NULL	AVP-13358	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SYN-1001	NULL	NULL	NULL	NULL	NULL
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.025563618	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfamylon	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	NULL	AWD-12-281	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	NULL	AWD-12-281	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TP-023	NULL	NULL	NULL	NULL	NULL
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.094665273	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.3697723326457359	Delphinidin	chembl:CHEMBL276780	DELPHINIDIN	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	NULL	L-651582	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefotiam	rxcui:2188	CEFOTIAM	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	Ciprofloxacin+dexamethasone	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.3431873936973496	Ispaghula	rxcui:104129	ISPAGHULA HUSK	TRUE	FALSE	FALSE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	2.187819634820604	Metoprine	ncit:C1161	METOPRINE	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	Y-25130	ncit:C73101	AZASETRON	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.8140724222588294	TA-2005	ncit:C171749	CARMOTEROL	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.3017682254924971	SOY PROTEIN	ncit:C1803	SOY PROTEIN ISOLATE	FALSE	FALSE	FALSE
PLASMODIUM BETA-HYDROXYACYL-ACP DEHYDRATASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
PLASMODIUM OXOACYL-[ACYL-CARRIER PROTEIN] REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.1553481397505754	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
STRYCHNINE-BINDING GLYCINE RECEPTOR	hgnc:4326	GLRA1	TTD	2020.06.01	NULL	0.3977853881492007	THIOCOLCHICOSIDE	rxcui:38085	THIOCOLCHICOSIDE	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.1131630845596864	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 47 MEMBER 1	hgnc:25588	SLC47A1	TTD	2020.06.01	NULL	0.5385402178019948	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Posaconazole	rxcui:282446	POSACONAZOLE	TRUE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	NULL	ARI-809	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	CT-102	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	HEGF	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.4579157375205915	Trafermin	ncit:C152708	TRAFERMIN	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.5585922471882393	Arecoline	ncit:C76610	ARECOLINE	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.2386712328895204	Ethotoin	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
AQP7	hgnc:640	AQP7	NCI	14-Sep-17	NULL	0.1801292323694494	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
PURINE NUCLEOSIDE PHOSPHORYLASE	hgnc:7892	PNP	TTD	2020.06.01	NULL	NULL	2'3'-Dideoxyinosine	NULL	NULL	NULL	NULL	NULL
PLASMODIUM ENOYL-ACP REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Plevitrexed	ncit:C1629	PLEVITREXED	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR-GAMMA	hgnc:10479	RXRG	TTD	2020.06.01	NULL	NULL	9cUAB-30	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	CpG-10101	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefditoren	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pfizer 10	NULL	NULL	NULL	NULL	NULL
LCK TYROSINE PROTEIN KINASE	hgnc:6524	LCK	TTD	2020.06.01	NULL	NULL	ISIS-CRP	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	ISIS-CRP	NULL	NULL	NULL	NULL	NULL
ARNT	hgnc:700	ARNT	NCI	14-Sep-17	NULL	0.2386712328895204	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
RIP2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-CRP	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 11 RECEPTOR ALPHA	hgnc:5967	IL11RA	TTD	2020.06.01	NULL	10.50153425	Oprelvekin	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
FUNGAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Natamycin	rxcui:7268	NATAMYCIN	TRUE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 1	hgnc:4593	GRM1	TTD	2020.06.01	NULL	NULL	NPS-2390	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefazolin	rxcui:2180	CEFAZOLIN	TRUE	FALSE	FALSE
PLASMODIUM DIHYDROOROTATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Artemisinin	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
AR	hgnc:644	AR	NCI	14-Sep-17	NULL	0.003654487	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	TG100801	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	NULL	Eptacog alfa intravenous	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfadiazine	rxcui:10171	SULFADIAZINE	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR BETA-4	hgnc:1964	CHRNB4	TTD	2020.06.01	NULL	0.8751278539282418	CYTISINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rolitetracycline	rxcui:9462	ROLITETRACYCLINE	FALSE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peginterferon beta	rxcui:1546168	PEGINTERFERON BETA-1A	TRUE	FALSE	FALSE
ESTRADIOL 17 BETA-DEHYDROGENASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	NK-314	NULL	NULL	NULL	NULL	NULL
BCR	hgnc:1014	BCR	NCI	14-Sep-17	NULL	0.6250913242344582	HERBIMYCIN A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-0249	drugbank:DB11910	MK-0249	FALSE	FALSE	FALSE
BACTERIAL DD-CARBOXYPEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TD-1792	chembl:CHEMBL4297645	CEFILAVANCIN	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE VI	hgnc:1380	CA6	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE XII	hgnc:1371	CA12	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE XIV	NULL	NULL	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	APN-201	NULL	NULL	NULL	NULL	NULL
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.1773907812016706	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.02075402	Dihydroergotamine	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
ONCHOCERCA GLUTAMATE-GATED CHLORIDE CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ivermectin	rxcui:6069	IVERMECTIN	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rilpivirine	rxcui:1102270	RILPIVIRINE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lexipafant	ncit:C170120	LEXIPAFANT	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	Mteron-F1	NULL	NULL	NULL	NULL	NULL
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	NULL	Epothilon	NULL	NULL	NULL	NULL	NULL
BACTERIAL DD-CARBOXYPEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	B-Lactams	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfonamides	ncit:C29739	SULFONAMIDE ANTI-INFECTIVE AGENT	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP120	NULL	NULL	TTD	2020.06.01	NULL	NULL	Multi-envelope HIV vaccine	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GLYCOPROTEIN 41	NULL	NULL	TTD	2020.06.01	NULL	NULL	Multi-envelope HIV vaccine	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Balapiravir	ncit:C87439	BALAPIRAVIR	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	0.1346350544504987	Orlistat	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	QVA-149	NULL	NULL	NULL	NULL	NULL
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	1.750255707856483	Albinterferon alfa-2b	ncit:C87296	ALBINTERFERON ALFA-2B	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.2386712328895204	CANCER VACCINE	ncit:C1663	ANTINEOPLASTIC VACCINE	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CYT-006-AngQb	NULL	NULL	NULL	NULL	NULL
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Linezolid	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	PSMA-targeted tubulysin B conjugates	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	6.177373086552294	Barusiban	ncit:C90866	BARUSIBAN	FALSE	FALSE	FALSE
INTERFERON ALPHA/BETA RECEPTOR 2	hgnc:5433	IFNAR2	TTD	2020.06.01	NULL	6.563458904461812	Interferon alfacon-1	rxcui:59744	INTERFERON ALFACON-1	TRUE	TRUE	TRUE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	NULL	C326	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	FENBUFEN	rxcui:24830	FENBUFEN	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	NULL	CYC-800	NULL	NULL	NULL	NULL	NULL
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.019261802	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mechlorethamine	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	Biferonex	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	NULL	GSK-706769	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	CGC-11047	drugbank:DB05722	CGC-11047	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.07458476	Epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clavulanate	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfamethazine	rxcui:10178	SULFAMETHAZINE	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Terconazole	rxcui:37806	TERCONAZOLE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sufentanil	rxcui:56795	SUFENTANIL	TRUE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	NCI	14-Sep-17	NULL	0.175610941	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
PLASMODIUM GLUTAMATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hexachlorophene	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
MYCOBACTERIUM ARABINOSYLTRANSFERASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ethambutol	rxcui:142435	ETHAMBUTOL HYDROCHLORIDE	TRUE	FALSE	FALSE
INTERLEUKIN-8	hgnc:6025	CXCL8	TTD	2020.06.01	NULL	0.016621612	Ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CARTPT	hgnc:24323	CARTPT	NCI	14-Sep-17	NULL	0.3962843112127886	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
MYELIN BASIC PROTEIN	hgnc:6925	MBP	TTD	2020.06.01	NULL	NULL	BHT-3009	NULL	NULL	NULL	NULL	NULL
CAMK2G	hgnc:1463	CAMK2G	NCI	14-Sep-17	NULL	0.065799087	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
KETOGENESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	AC-1202	chembl:CHEMBL1406148	TRICAPRILIN	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	CR-665	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	FST-201	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	0.1223955040459079	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flavanone	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
DICKKOPF-RELATED PROTEIN 1	hgnc:2891	DKK1	TTD	2020.06.01	NULL	NULL	PF-04840082	NULL	NULL	NULL	NULL	NULL
RIBOSOME	NULL	NULL	TTD	2020.06.01	NULL	NULL	TST-10088	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GLYCOPROTEIN 41	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gp41 HIV-1 vaccine	NULL	NULL	NULL	NULL	NULL
CAMK2B	hgnc:1461	CAMK2B	NCI	14-Sep-17	NULL	0.1419126249613364	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
MYCOBACTERIUM ANTIGEN COMPLEX 85A	NULL	NULL	TTD	2020.06.01	NULL	NULL	MVA-85A	NULL	NULL	NULL	NULL	NULL
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
STERYL-SULFATASE	hgnc:11425	STS	TTD	2020.06.01	NULL	NULL	COUMATE	NULL	NULL	NULL	NULL	NULL
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE BETA	hgnc:5960	IKBKB	TTD	2020.06.01	NULL	5.000730593875666	IMD-0354	chembl:CHEMBL3545089	IMD-0354	FALSE	FALSE	FALSE
AURORA KINASE C	hgnc:11391	AURKC	TTD	2020.06.01	NULL	2.800409132570373	GSK1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
CAST	hgnc:1515	CAST	NCI	14-Sep-17	NULL	0.7895890411382631	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	3.750547945	Pomaglumetad	chembl:CHEMBL375611	LY404039	FALSE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.6269572684859045	GSK1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	0.1785975212098452	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	SBS-1000	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.2401265452851882	Obatoclax	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	NULL	Amfetamine transdermal	NULL	NULL	NULL	NULL	NULL
GASTRIN-RELEASING PEPTIDE RECEPTOR	hgnc:4609	GRPR	TTD	2020.06.01	NULL	NULL	177Lu-AMBA	NULL	NULL	NULL	NULL	NULL
CETP	hgnc:1869	CETP	NCI	14-Sep-17	NULL	0.384671584	9-CIS RETINOIC ACID	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
REGULATORY PROTEIN UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Teplizumab	rxcui:2621880	TEPLIZUMAB	TRUE	FALSE	FALSE
CYCLOPHILIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alisporivir	ncit:C169774	ALISPORIVIR	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	JNJ-39220675	drugbank:DB12929	JNJ-39220675	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.3535870116881784	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
PROSTATE CANCE CELL	hgnc:2411	CRYGD	TTD	2020.06.01	NULL	13.12691780892362	HE3235	chembl:CHEMBL3545237	HE3235	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC KAINATE 1	hgnc:4579	GRIK1	TTD	2020.06.01	NULL	3.500511415712966	LY293558	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.4688184931758437	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lersivirine	ncit:C83872	LERSIVIRINE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	THRX-198321	NULL	NULL	NULL	NULL	NULL
LYSOPHOSPHATIDIC ACID RECEPTOR 1	hgnc:3166	LPAR1	TTD	2020.06.01	NULL	6.563458904461812	BMS-986202	iuphar.ligand:12723	BMS-986202	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	5.527123287967842	MK-7246	chembl:CHEMBL561132	MK-7246	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Irdabisant	ncit:C170078	IRDABISANT	FALSE	FALSE	FALSE
MYCOBACTERIUM MEMBRANE PROTEIN MMPL3	NULL	NULL	TTD	2020.06.01	NULL	NULL	BM-212	chembl:CHEMBL321077	BM-212	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	DA-1229	chembl:CHEMBL1779710	EVOGLIPTIN	FALSE	FALSE	FALSE
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	11C-GSK-215083	NULL	NULL	NULL	NULL	NULL
HYDROXY RADICAL ELIMINATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	HD-003	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bavisant	ncit:C171762	BAVISANT	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-5213	NULL	NULL	NULL	NULL	NULL
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.6250913242344582	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	TPI-1020	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	AP-301-IH	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR-2	hgnc:3676	FGF2	TTD	2020.06.01	NULL	NULL	DVC1-0101	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS ALPHA-HEMOLYSIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyrtominetin	chembl:CHEMBL1224646	CYRTOMINETIN	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.073694977	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
INTERFERON	hgnc:5417	IFNA1	TTD	2020.06.01	NULL	NULL	Low-dose oral interferon	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	3.088686543276147	N8-GP	ncit:C152786	TUROCTOCOG ALFA PEGOL	FALSE	FALSE	FALSE
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	2.625383561784724	RG7686	iuphar.ligand:8406	CODRITUZUMAB	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	TD-4208	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	99mTc-MIP-1405	NULL	NULL	NULL	NULL	NULL
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	NULL	S-PRAnt	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	AGN-208397	NULL	NULL	NULL	NULL	NULL
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	NULL	BIIB 028	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.9723642821424906	FBT-A05	chembl:CHEMBL2109351	FBT-A05	FALSE	FALSE	FALSE
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-8742	rxcui:1734628	ELBASVIR	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Selurampanel	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
CRP MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-CRPRx	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	EGS-21	NULL	NULL	NULL	NULL	NULL
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	HQK-1001	chembl:CHEMBL1650317	SODIUM 2,2-DIMETHYLBUTYRATE	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	EP-42675	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	EP-42675	NULL	NULL	NULL	NULL	NULL
FUNGAL 1,3-BETA-GLUCAN SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Micafungin	rxcui:325887	MICAFUNGIN	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NRX-1074	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.1207072901969988	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	EGFRvIII CAR	NULL	NULL	NULL	NULL	NULL
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	0.3431873936973496	MM-151	iuphar.ligand:9125	MM-151	FALSE	TRUE	TRUE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	CSL-362-AML	NULL	NULL	NULL	NULL	NULL
SODIUM/HYDROGEN EXCHANGER 3	hgnc:11073	SLC9A3	TTD	2020.06.01	NULL	NULL	AVE-0657	NULL	NULL	NULL	NULL	NULL
STERYL-SULFATASE	hgnc:11425	STS	TTD	2020.06.01	NULL	NULL	PGL-2001	NULL	NULL	NULL	NULL	NULL
HEPATITIS B VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Entecavir	rxcui:1546027	ENTECAVIR ANHYDROUS	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,2,4,5-tetra-substituted imidazole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,2,4-tri-substituted imidazoline derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Azetidine-1-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diaryl piperazine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diphenyl purine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diphenyl purine derivative 4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Hydrazide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazole derivative 5	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazole derivative 7	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazolidine-2,4-dione derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	N-(arylalkyl)-1H-indole-2-sulfonic acid amide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Piperazine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Purine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Purine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Purine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 20	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 21	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 23	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 27	NULL	NULL	NULL	NULL	NULL
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	1.250182648468916	ANTIFUNGAL AGENT	ncit:C514	ANTIFUNGAL AGENT	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 34	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 6	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 7	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 8	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazoline derivative 11	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazoline derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazoline derivative 4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrido[2,3-d]pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 6	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Sulfonylated piperazine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Tetra-hydro-1H-1,2,6-triazaazulene derivative 2	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	DSP-1053	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.1770916399180253	POLY I:POLY C	chembl:CHEMBL4297812	PREP-001	FALSE	FALSE	FALSE
ROTAMASE PIN1	hgnc:8988	PIN1	TTD	2020.06.01	NULL	NULL	Avastin+/-Tarceva	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.693795846312725	Methdilazine	rxcui:29648	METHDILAZINE	TRUE	FALSE	FALSE
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	NULL	HTU-PA	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mezlocillin	rxcui:6927	MEZLOCILLIN	FALSE	FALSE	FALSE
MAMMALIAN TARGET OF RAPAMYCIN COMPLEX 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	RBT-101	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.04427291	LACTOSE	rxcui:6211	LACTOSE	TRUE	FALSE	FALSE
ELECTRON TRANSPORT COMPLEX III	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tafenoquine	rxcui:2054023	TAFENOQUINE	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.1136529680426287	RIFAMPIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Eslicarbazepine	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetrodotoxin	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	CC8464	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.033487035	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
P2X PURINOCEPTOR 4	hgnc:8535	P2RX4	TTD	2020.06.01	NULL	NULL	P2X4 inhibitora	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAGE-718	iuphar.ligand:12050	SAGE-718	FALSE	FALSE	FALSE
GROWTH HORMONE SECRETION	NULL	NULL	TTD	2020.06.01	NULL	NULL	CIGB-500	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PT-304	chembl:CHEMBL253995	CHEMBL:CHEMBL253995	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.060772768	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.4487835148349957	BIMU-1	iuphar.ligand:233	BIMU 1	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Uracil mustard	rxcui:10996	URACIL MUSTARD	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS TAT PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALX-40-4C	NULL	NULL	NULL	NULL	NULL
CYP3A7	hgnc:2640	CYP3A7	NCI	14-Sep-17	NULL	0.258658479	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
ACETYL-COA:LYSO-PAF ACETYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	B-Lactams	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.4070362111294147	Tizanidine	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.006525935	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER A4	hgnc:34	ABCA4	TTD	2020.06.01	NULL	NULL	StarGen	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	INO-3510	NULL	NULL	NULL	NULL	NULL
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	NULL	KOS-2187	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.023336743	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE PIM-1	hgnc:8986	PIM1	TTD	2020.06.01	NULL	NULL	CXR-1002	NULL	NULL	NULL	NULL	NULL
CATHEPSIN A	hgnc:9251	CTSA	TTD	2020.06.01	NULL	NULL	SAR164653	NULL	NULL	NULL	NULL	NULL
BACTERIAL BOTULINUM TOXIN A	NULL	NULL	TTD	2020.06.01	NULL	NULL	RT-001	drugbank:DB16949	DEULINOLEATE ETHYL	FALSE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.2869271652223742	Androgen restored contraceptive	wikidata:Q85759692	ETHINYLESTRADIOL/DROSPIRENONE/PRASTERONE	FALSE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	7.001022831425932	ANTI-DIABETIC AGENT	ncit:C29711	ANTI-DIABETIC AGENT	FALSE	FALSE	FALSE
SCAVENGER DECAPPING ENZYME DCPS	hgnc:29812	DCPS	TTD	2020.06.01	NULL	105.0153424713889	RG3039	drugbank:DB16938	D-157495	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SMP-986	chembl:CHEMBL3545165	AFACIFENACIN	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Drug 2878175	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	VBY-129	NULL	NULL	NULL	NULL	NULL
BACTERIAL FATTY ACID SYNTHETASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	AFN-1720	ncit:C169766	AFABICIN	FALSE	FALSE	FALSE
CYP4B1	hgnc:2644	CYP4B1	NCI	14-Sep-17	NULL	1.050153425	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-759	NULL	NULL	NULL	NULL	NULL
BACTERIAL BOTULINUM TOXIN A	NULL	NULL	TTD	2020.06.01	NULL	NULL	XOMA-3AB	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Recombinant human Erbb3 fragment therapeutic tumor vaccine	NULL	NULL	NULL	NULL	NULL
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	NULL	Recombinant human Erbb3 fragment therapeutic tumor vaccine	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	ZY01	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	NULL	Sphingosine-1-phosphate receptor-1 agonist	NULL	NULL	NULL	NULL	NULL
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	NULL	JTT-654	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-20	hgnc:6002	IL20	TTD	2020.06.01	NULL	NULL	NN-8226	NULL	NULL	NULL	NULL	NULL
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1436598392221464	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
NKG2-A/B-ACTIVATING NK RECEPTOR	hgnc:6374	KLRC1	TTD	2020.06.01	NULL	105.0153424713889	NN8765	ncit:C120208	MONALIZUMAB	FALSE	FALSE	FALSE
CLOSTRIDIUM DIFFICILE TOXIN A	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-3415A	NULL	NULL	NULL	NULL	NULL
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1878628666751145	N-(4-HYDROXYPHENYL)RETINAMIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
CLOSTRIDIUM DIFFICILE TOXIN B	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-3415A	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	Anti-mesothelin CAR transduced PBL	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	CART-EGFR	NULL	NULL	NULL	NULL	NULL
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	9.546849315580817	CEPHALOSTATIN	ncit:C2052	CEPHALOSTATIN	FALSE	FALSE	FALSE
TUBULIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	OC-10X	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	CART-HER-2	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	GD2 T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART-19 T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-CAR and CD28-CAR T Cells	NULL	NULL	NULL	NULL	NULL
T-CELL-SPECIFIC SURFACE GLYCOPROTEIN CD28	hgnc:1653	CD28	TTD	2020.06.01	NULL	NULL	CD19-CAR and CD28-CAR T Cells	NULL	NULL	NULL	NULL	NULL
DLG4	hgnc:2903	DLG4	NCI	14-Sep-17	NULL	0.4605936073306535	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	CART-meso cells	NULL	NULL	NULL	NULL	NULL
PROSTATE STEM CELL ANTIGEN	hgnc:9500	PSCA	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting PSCA	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	GPC3 targeting CAR-T cells	NULL	NULL	NULL	NULL	NULL
DPP4	hgnc:3009	DPP4	NCI	14-Sep-17	NULL	0.1105424657593568	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
MYELOID INHIBITORY C-TYPE LECTIN-LIKE RECEPTOR	hgnc:31713	CLEC12A	TTD	2020.06.01	NULL	NULL	CLL1-specific gene-engineered T cells	NULL	NULL	NULL	NULL	NULL
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	NULL	CD38 CAR T cells	NULL	NULL	NULL	NULL	NULL
NEURAL CELL ADHESION MOLECULE 1	hgnc:7656	NCAM1	TTD	2020.06.01	NULL	NULL	CD56 CAR T cells	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	NULL	CART-10 cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CART-22 cells	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting BCMA	NULL	NULL	NULL	NULL	NULL
DPP4	hgnc:3009	DPP4	NCI	14-Sep-17	NULL	0.084012274	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
HLA-A02/AFP COMPLEX	NULL	NULL	TTD	2020.06.01	NULL	NULL	Autologous ET1402L1-CART cells	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	ICAR30 T cells	NULL	NULL	NULL	NULL	NULL
DPP4	hgnc:3009	DPP4	NCI	14-Sep-17	NULL	0.1615620653405984	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	C7R-GD2.CART cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	1.944728564284981	MB-CART20.1	ncit:C172063	AUTOLOGOUS ANTI-CD20 CAR TRANSDUCED CD4/CD8 ENRICHED T-CELLS MB-CART20.1	FALSE	FALSE	FALSE
SYNDECAN-1	hgnc:10658	SDC1	TTD	2020.06.01	NULL	NULL	CAR138 T Cells	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	Anti-CD123 CAR-T treatment	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	LCAR-B4822M CAR-T Cell	NULL	NULL	NULL	NULL	NULL
DRAM	hgnc:25645	DRAM1	NCI	14-Sep-17	NULL	0.7242437411819931	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19.CAR T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART19 cell	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	IC9-CAR19 T cells	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	CART123 cells	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	0.1556551518844698	Quisinostat	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pizotyline	rxcui:8373	PIZOTYLINE	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.3017682254924971	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	NULL	Terbutyline	NULL	NULL	NULL	NULL	NULL
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	T2c-001	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 2 RECEPTOR	hgnc:4325	GLP2R	TTD	2020.06.01	NULL	13.12691780892362	Teduglutide	rxcui:1364468	TEDUGLUTIDE	TRUE	FALSE	FALSE
EIF2AK2	hgnc:9437	EIF2AK2	NCI	14-Sep-17	NULL	13.12691780892362	RICIN	ncit:C809	RICIN	FALSE	FALSE	FALSE
ARYL HYDROCARBON RECEPTOR SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	AFP464	ncit:C48370	AMINOFLAVONE PRODRUG AFP464	FALSE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Auranofin	rxcui:1227	AURANOFIN	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beclomethasone	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
C-TYPE NATRIURETIC PEPTIDE	hgnc:7941	NPPC	TTD	2020.06.01	NULL	1.250182648468916	BMN-111	rxcui:2586354	VOSORITIDE	TRUE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	Cholic acid - Asklepion	NULL	NULL	NULL	NULL	NULL
ESRRG	hgnc:3474	ESRRG	NCI	14-Sep-17	NULL	0.5303805175322677	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cilostazol	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clozapine	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
GERANYLGERANYL TRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-778123	drugbank:DB07227	L-778123	FALSE	FALSE	FALSE
EZR	hgnc:12691	EZR	NCI	14-Sep-17	NULL	2.187819634820604	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
HEPATITIS C VIRUS NS3 HELICASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ACH-2684	chembl:CHEMBL3040582	DELDEPREVIR	FALSE	FALSE	FALSE
HAEMOPHILUS INFLUENZAE ACETYLGLUCOSAMINE DEACETYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ACHN-975	chembl:CHEMBL3939284	ACHN-975	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	AD-337	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	3.281729452230906	PF-04449913	rxcui:2105845	GLASDEGIB	TRUE	FALSE	TRUE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.3182283105193606	Tedatioxetine	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
FASLG	hgnc:11936	FASLG	NCI	14-Sep-17	NULL	0.6908904109959803	TUMOR NECROSIS FACTOR-BETA	ncit:C622	RECOMBINANT TUMOR NECROSIS FACTOR-BETA	FALSE	FALSE	FALSE
LEUTINIZING-HORMONE-RELEASING HORMONE	hgnc:4419	GNRH1	TTD	2020.06.01	NULL	NULL	CG201	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	ISIS-GCGRrx	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	JM216	rxcui:1733681	SATRAPLATIN	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.043074382	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.3777530304726222	Bafetinib	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	4.773424657790408	Masilukast	ncit:C83906	MASILUKAST	FALSE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pramiconazole	ncit:C72830	PRAMICONAZOLE	FALSE	FALSE	FALSE
INTEGRIN ALPHA-4/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRK-170	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-4/BETA-7	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRK-170	NULL	NULL	NULL	NULL	NULL
PRO-NEUREGULIN-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Neucardin	chembl:CHEMBL4594600	HUMAN NEUREGULIN-1 RECOMBINANT (177-237)	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	NCI	14-Sep-17	NULL	0.055300338	8-MOP	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1B	hgnc:7464	MTNR1B	TTD	2020.06.01	NULL	NULL	VLB-01	NULL	NULL	NULL	NULL	NULL
SERINE PALMITOYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	NA-808	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MURAGLITAZAR	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	F-15063	NULL	NULL	NULL	NULL	NULL
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.06757744	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	F-15063	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceftobiprole	ncit:C65306	CEFTOBIPROLE	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glufosfamide	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Apricitabine	ncit:C79871	APRICITABINE	FALSE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.092199598	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
ROOF PLATE-SPECIFIC SPONDIN-1	hgnc:21679	RSPO1	TTD	2020.06.01	NULL	NULL	NU-206	NULL	NULL	NULL	NULL	NULL
CHYMASE	hgnc:2097	CMA1	TTD	2020.06.01	NULL	NULL	SUN13834	NULL	NULL	NULL	NULL	NULL
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.325124899	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
INTEGRIN ALPHA-V/BETA-3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fluciclatide F-18	ncit:C74031	FLUCICLATIDE F 18	FALSE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.1165542091802319	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA3.1	hgnc:6293	KCNN4	TTD	2020.06.01	NULL	35.00511415712966	ICA-17043	ncit:C76882	SENICAPOC	FALSE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nemonaxacin	NULL	NULL	NULL	NULL	NULL
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zabofloxacin	ncit:C82232	ZABOFLOXACIN	FALSE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zabofloxacin	ncit:C82232	ZABOFLOXACIN	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	diclofenac sodium patch	NULL	NULL	NULL	NULL	NULL
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.1944728564284981	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	diclofenac sodium patch	NULL	NULL	NULL	NULL	NULL
MYCOBACTERIUM RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAS-106	drugbank:DB06656	TAS-106	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-00734200	ncit:C90616	GOSOGLIPTIN	FALSE	FALSE	FALSE
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Superoxide dismutase	rxcui:10245	SUPEROXIDE DISMUTASE	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Y-39983	chembl:CHEMBL571948	Y-39983	FALSE	FALSE	FALSE
FUNGAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amphotericin B inhalation powder	NULL	NULL	NULL	NULL	NULL
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	YH-4808	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR	hgnc:2436	CSF2RB	TTD	2020.06.01	NULL	NULL	TPI ASM8	NULL	NULL	NULL	NULL	NULL
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.3977853881492006	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SSTarbaclofen	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	NULL	OCV-101	NULL	NULL	NULL	NULL	NULL
IMMUNOGLOBULIN EPSILON FC RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Omalizumab	rxcui:302379	OMALIZUMAB	TRUE	FALSE	FALSE
INTERLEUKIN 4 RECEPTOR ALPHA	hgnc:6015	IL4R	TTD	2020.06.01	NULL	NULL	Altrakincept	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-13	hgnc:5973	IL13	TTD	2020.06.01	NULL	NULL	PEGylated pitrakinra	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-4	hgnc:6014	IL4	TTD	2020.06.01	NULL	NULL	PEGylated pitrakinra	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.1182605208011137	Ipratropium	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.251232877	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Ethinyl-pyrazole derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Heteroaryl-pyrazole derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	N-substituted pyrazole derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-22	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.018106094	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-22	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-37	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-39	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-40	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-42	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-43	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1591141552596803	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-44	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-46	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-51	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Tetra-hydro-imidazo[1,5-d][1,4]oxazepin-3-yl derivative 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Tetra-hydro-imidazo[1,5-d][1,4]oxazepin-3-yl derivative 6	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	Hydroxamate analog 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Hydroxamate analog 1	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1750255707856483	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Hydroxyqunoline analog 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-46	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-46	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-46	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-48	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-52	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1029562181092049	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Pyridine-2,4-dicarboxylic acid analog 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Pyridine-2,4-dicarboxylic acid analog 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridine-2,4-dicarboxylic acid derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Pyrido[1,2-a]indole-1.-carboxylic acid analog 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	Selenium compound 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	Selenium compound 3	NULL	NULL	NULL	NULL	NULL
5-HT 7 RECEPTOR	hgnc:5302	HTR7	TTD	2020.06.01	NULL	NULL	4-oxadiazole derivative 1	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	amidepsines	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Benzamide derivative 19	NULL	NULL	NULL	NULL	NULL
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	5.527123287967842	HPV-16 E6	ncit:C38726	SYNTHETIC HUMAN PAPILLOMAVIRUS 16 E6 PEPTIDE	FALSE	FALSE	FALSE
5-HT 7 RECEPTOR	hgnc:5302	HTR7	TTD	2020.06.01	NULL	NULL	Carbamide derivative 2	NULL	NULL	NULL	NULL	NULL
MANNOSIDE ACETYLGLUCOSAMINYLTRANSFERASE 2	hgnc:7045	MGAT2	TTD	2020.06.01	NULL	NULL	Dihydropyrimidinone derivative 3	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Lactam derivative 4	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-AZD3988	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Pyrazine carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 29	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminopiperidine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminopiperidine derivative 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-phe compound 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 46	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 49	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-12	NULL	NULL	NULL	NULL	NULL
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1367387271762877	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-37	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-56	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-6	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 33	NULL	NULL	NULL	NULL	NULL
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.546954909	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyrimidinedione derivative 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Xanthine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Xanthine/amino piperidine compound 1	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-10	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-Figure2-2	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-15	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-114	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-118	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-12	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-122	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-124	NULL	NULL	NULL	NULL	NULL
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.4375639269641209	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-125	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-130	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-134	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-135	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-137	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-14	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-143	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-148	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-150	NULL	NULL	NULL	NULL	NULL
IVL	hgnc:6187	IVL	NCI	14-Sep-17	NULL	5.834185692854944	PERILLYL ALCOHOL	ncit:C1461	PERILLYL ALCOHOL	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-153	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-156	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-158	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-19	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-28	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-36	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-37	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-38	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-40	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-43	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-46	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-49	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-51	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-54	NULL	NULL	NULL	NULL	NULL
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.087512785	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
KRT17	hgnc:6427	KRT17	NCI	14-Sep-17	NULL	2.100306849	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-56	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-57	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-62	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-69	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-7	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-71	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-76	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-80	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-84	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-85	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-86	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-91	NULL	NULL	NULL	NULL	NULL
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.1286952726365061	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-94	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-97	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-98	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	Buccal fentanyl	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 9	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 10	NULL	NULL	NULL	NULL	NULL
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.031583562	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 18	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 7	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 8	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 9	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Aromatic ring compound 3	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Biphenyl carboxamidopropanoic acid derivative 1	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Biphenyl carboxamidopropanoic acid derivative 4	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Heterocycle-containing compound 3	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Heterocycle-containing compound 5	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	PMID25828189-Compound-22	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 7	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Spiroimidazolone derivative 1	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Spiroimidazolone derivative 6	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Spiroimidazolone derivative 7	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-12	NULL	NULL	NULL	NULL	NULL
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.06697407	DEPSIPEPTIDE	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-13	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-14	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-17	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-20	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-20	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-29	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-33	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-39	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-4	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-4	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-44	NULL	NULL	NULL	NULL	NULL
MBP	hgnc:6925	MBP	NCI	14-Sep-17	NULL	0.283060222	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
CELLULAR INHIBITOR OF APOPTOSIS 2	hgnc:591	BIRC3	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-44	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-44	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 4	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 5	NULL	NULL	NULL	NULL	NULL
MDH2	hgnc:6971	MDH2	NCI	14-Sep-17	NULL	0.1810609352954982	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-D2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-D2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-E3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-E4	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-F2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-F2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-F2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-F2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-G1	NULL	NULL	NULL	NULL	NULL
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.2187819634820604	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-K1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	N-(pyridin-2-yl)pyrimidin-4-amine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Nitrogen mustard derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 3	hgnc:1772	CDK3	TTD	2020.06.01	NULL	NULL	Nitrogen mustard derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Nitrogen mustard derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	N-phenyl-pyrimidin-4-amine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	N-phenyl-pyrimidin-4-amine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Palbociclib/ribociclib analog 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	Palbociclib/ribociclib analog 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-34	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Pyrazolo-triazine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	NULL	Pyrazolo-triazine derivative 2	NULL	NULL	NULL	NULL	NULL
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1166837138570988	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Roscovitine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Roscovitine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	Roscovitine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	NULL	Roscovitine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Roscovitine derivative 1	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	PMID26293650-Compound-35	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl compound 3	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl compound 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 3	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 3	NULL	NULL	NULL	NULL	NULL
MT1H	hgnc:7400	MT1H	NCI	14-Sep-17	NULL	0.1034633915974275	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Gold-complexed thiosaccharide derivative 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 1	hgnc:11362	STAT1	TTD	2020.06.01	NULL	NULL	Oxazole derivative 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Oxazole derivative 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Peptide analog 7	NULL	NULL	NULL	NULL	NULL
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	15.00219178	GPI-0100	ncit:C2627	GPI-0100	FALSE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 1	hgnc:11362	STAT1	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 5	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 5	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 1	hgnc:11362	STAT1	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-10	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-10	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 5	hgnc:11366	STAT5A	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-10	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-11	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-13	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-51	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 65	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Salicylic acid derivative 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Salicylic acid derivative 4	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Salicylic acid derivative 5	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azetidine urea derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Benzyl pyrrolyloxoacetamide derivative 1	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.006627246	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Boronic acid derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 2	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 2	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	Carbamate derivative 2	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-46	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-47	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-49	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-50	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-54	NULL	NULL	NULL	NULL	NULL
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.218327115	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-8	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Pyrazolodiazepine derivative 1	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	Ampicidin analog 2	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 10	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 10	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 14	NULL	NULL	NULL	NULL	NULL
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.025439763	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 16	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 19	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 22	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 7	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 8	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-cyclodextrin conjugate derivative 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-cyclodextrin conjugate derivative 5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 10	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 14	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 22	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 27	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 6	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 8	NULL	NULL	NULL	NULL	NULL
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.201952582	LACTOSE	rxcui:6211	LACTOSE	TRUE	FALSE	FALSE
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 21	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 23	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	C-linked disaccharide biphenyl mannoside derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-126c	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5e	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5g	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-6a	NULL	NULL	NULL	NULL	NULL
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.031069628	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-6c	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-7d	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-8b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-9b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-9c	NULL	NULL	NULL	NULL	NULL
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.3125456621172291	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Aromatic hydrazine carboxyimidoamide derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzoic acid linked peptide analog 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzothiazole analog 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzothiazole analog 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 13	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 8	NULL	NULL	NULL	NULL	NULL
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.2500365296937833	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 2	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Aryl methoxyacrylate derivative 2	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 8	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Imidazo [1,2-a]pyridine compound 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Oligooxopiperazine derivative 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 7	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-14	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-2	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-8	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Tlouidine sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Aminocyclopentenone compound 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Aminocyclopentenone compound 4	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Aminocyclopentenone compound 5	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Aminocyclopentenone compound 6	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 10	NULL	NULL	NULL	NULL	NULL
REG1A	hgnc:9951	REG1A	NCI	14-Sep-17	NULL	0.9907107780319716	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.108040476	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 12	NULL	NULL	NULL	NULL	NULL
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.1315981735230438	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	NULL	Dihydropyrido pyrazinone compound 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 10	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-54	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-56	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrazole and thiophene derivative 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 3	hgnc:1104	BRD3	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 4	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 5	NULL	NULL	NULL	NULL	NULL
CREB-BINDING PROTEIN	hgnc:2348	CREBBP	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 6	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Amidine compound 2	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Amidine compound 5	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Amidine compound 6	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 9	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzothiazine-carboxamide compound 1	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzothiazine-carboxamide compound 4	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzothiazine-carboxamide compound 6	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	N6-cyclopropyllydine derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-20b	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-21b	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-21b	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-28	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-42b	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-44	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-26	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-26	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-28	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-28	NULL	NULL	NULL	NULL	NULL
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.6250913242344582	TRIBUTYRIN	ncit:C1260	TRIBUTYRIN	FALSE	FALSE	FALSE
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-31	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-31	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-33	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-41	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-43	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-44	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-6	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Isoxazoles and isoxazoline derivative 4	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID27172114-Compound-30	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	PMID27172114-Compound-30	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	PMID27172114-Compound-30	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	PMID27172114-Compound-47	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	PMID27172114-Compound-49	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Pyrimidine benzenesulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Pyrimidine benzenesulfonamide derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Cyano(dimethyl)methyl isoxazoles and [1,3,4]-thiadiazoles derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Cyano(dimethyl)methyl isoxazoles and [1,3,4]-thiadiazoles derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Isoquinoline derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Phytocannabinoid/aminoalkylindole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Phytocannabinoid/aminoalkylindole derivative 2	NULL	NULL	NULL	NULL	NULL
S100B	hgnc:10500	S100B	NCI	14-Sep-17	NULL	3.281729452230906	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-11	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-25	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo triazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo triazine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazotriazinone derivative 1	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-asCEBP-1HPE	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-asCEBP-2	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-CROs	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-miR-155-5p	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-423	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-423	NULL	NULL	NULL	NULL	NULL
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.1426838892274307	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3B	hgnc:2979	DNMT3B	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-423	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-434	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Table1Example8	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-3	hgnc:10431	RPS6KA2	TTD	2020.06.01	NULL	NULL	Indole-based analog 14	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-77	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 11	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 3	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 4	NULL	NULL	NULL	NULL	NULL
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.210030685	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 9	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Bidentate pyrazolopyrimidine acetamide analog 3	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine acetamide derivative 5	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 9	NULL	NULL	NULL	NULL	NULL
DUAL SPECIFICITY PROTEIN KINASE TTK	hgnc:10416	RPS27	TTD	2020.06.01	NULL	NULL	Tricyclic isoxazoloquinazoline derivative 2	NULL	NULL	NULL	NULL	NULL
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.3231241306811969	BETA-ADRENERGIC ANTAGONIST	ncit:C29576	BETA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Tricyclic isoxazoloquinazoline derivative 2	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Dihydropyridine compound 1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Dihydropyridine compound 4	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Isoindole 1,3-dione analog 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	PMID27724045-Compound-17	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Pyridazinone derivative 1	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	Biphenyl carboxylic acid derivative 2	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-18	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-W	hgnc:995	BCL2L2	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-18	NULL	NULL	NULL	NULL	NULL
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1615620653405984	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-18	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-18	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-19	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrole six-membered heteroaryl ring derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrole six-membered heteroaryl ring derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrole six-membered heteroaryl ring derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure12Example1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure12Example1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure8Example99	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 6	NULL	NULL	NULL	NULL	NULL
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	1.615620653405984	OMAPATRILAT	ncit:C1782	OMAPATRILAT	FALSE	FALSE	FALSE
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 6	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	Ruxolitinib derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ruxolitinib derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ruxolitinib derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Ruxolitinib derivative 2	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-133	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-135	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-144	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-145	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-156	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Fluorinated donepezil derivative 2	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-12	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-15	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-27	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-28	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-36	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-48	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-7	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-42	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-47	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-7	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-Figure4b	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-Figure6C	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Terpyridineplatinum(II) complexe 4	NULL	NULL	NULL	NULL	NULL
GLUTATHIONE REDUCTASE	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	Terpyridineplatinum(II) complexe 4	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Triazole gold complexe 2	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-13	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-19	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-5	NULL	NULL	NULL	NULL	NULL
SMAD2	hgnc:6768	SMAD2	NCI	14-Sep-17	NULL	0.3125456621172291	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
CATHEPSIN F	hgnc:2531	CTSF	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-5	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-5	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-5	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-5	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-6	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-6	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-8	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	Indazolyl-thiadiazolamine derivative 1	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoquinoline sulfonyl derivative 1	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-4	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-4	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	Tricyclic compound 4	NULL	NULL	NULL	NULL	NULL
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.1417211099478934	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	1,2,4-triazole derivative 4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 2	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Phenylpropylamine derivative 4	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Piperidine derivative 5	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperidine derivative 5	NULL	NULL	NULL	NULL	NULL
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.4118248724368196	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Piperidine derivative 6	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperidine derivative 6	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	2-(substituted ethynyl)quinoline derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	2-(substituted ethynyl)quinoline derivative 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	6-aryl-imidazopyridine and 6-aryl-triazolopyridine carboxamide analog 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	6-aryl-imidazopyridine and 6-aryl-triazolopyridine carboxamide analog 3	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Azaindazole derivative 1	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Azaindazole derivative 2	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Azaindazole derivative 3	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Fused thiophene derivative 1	NULL	NULL	NULL	NULL	NULL
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.3818739726232327	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
LEUCINE-RICH REPEAT KINASE 2 S935 PHOSPHORYLATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fused thiophene derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure16-b-2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 26	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 27	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 13	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 5	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 8	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	3-amino-5-benzyl-substituted indazole derivative 1	NULL	NULL	NULL	NULL	NULL
TDO2	hgnc:11708	TDO2	NCI	14-Sep-17	NULL	0.2442217266776488	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	3-amino-5-benzyl-substituted indazole derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	3-amino-5-benzyl-substituted indazole derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 7	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Five membered heterocyclic benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-(phenylpyrazolyl)benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpiperidine ether derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2010077680 481	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2010077680 495	NULL	NULL	NULL	NULL	NULL
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	5.527123287967842	CREMOPHOR	ncit:C28896	CREMOPHOR	FALSE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2013009582Example16	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2014129431Example8-1	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2016054807Example1	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2016054807Example1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2016054807Example1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-h]quinazoline-3-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-d]pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-b]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Six-membered heterocyclic benzamide derivative 5	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Triazolo[4,3-b]pyridazine derivative 2	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-18	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-20	NULL	NULL	NULL	NULL	NULL
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.2542744369767287	GALLIUM NITRATE	rxcui:25544	GALLIUM NITRATE	TRUE	FALSE	FALSE
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-24	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-25	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-30	NULL	NULL	NULL	NULL	NULL
EZH2 Y641F MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-10	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-13	NULL	NULL	NULL	NULL	NULL
EZH2 Y641F MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-13	NULL	NULL	NULL	NULL	NULL
TGFBR3	hgnc:11774	TGFBR3	NCI	14-Sep-17	NULL	0.8204323630577265	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-19	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-28	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-29	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-30	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	Pyridinone compound 1	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	Quinazolines and azaquinazoline derivative 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 14	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 22	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 23	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 13	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 16	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 11	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 5	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 7	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 8	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 14	NULL	NULL	NULL	NULL	NULL
TLR4	hgnc:11850	TLR4	NCI	14-Sep-17	NULL	0.3043922970185188	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 15	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 2	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 4	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 11	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 12	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 13	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Betais-sulfonylamino derivative 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Boswellia acid derivative 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Carboxylic acid derivative 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 7	NULL	NULL	NULL	NULL	NULL
TMSB10	hgnc:11879	TMSB10	NCI	14-Sep-17	NULL	1.207072901969988	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Methyl-piperidine compound 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Piperidine carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	PMID28627961-Compound-22	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	PMID28627961-Compound-44	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Benzodihydroisofuran derivative 3	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Benzodihydroisofuran derivative 4	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Imidazole derivative 9	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl pyrazole derivative 4	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl triazole derivative 3	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl triazole derivative 4	NULL	NULL	NULL	NULL	NULL
TICAM1	hgnc:18348	TICAM1	NCI	14-Sep-17	NULL	9.546849315580818	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl triazole derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 22	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 26	NULL	NULL	NULL	NULL	NULL
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 28	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 28	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 29	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 32	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme15-3	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme18	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-12	hgnc:7158	MMP12	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure17(10)	NULL	NULL	NULL	NULL	NULL
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.2692701089009974	IMMUNOMODULATORS	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure17(10)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-12	hgnc:7158	MMP12	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure17(12)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure17(12)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure17(13)	NULL	NULL	NULL	NULL	NULL
GELATINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure9(1)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-SB-3CT	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-SB-3CT	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID29166791-Compound-AMPCP	NULL	NULL	NULL	NULL	NULL
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzyl amine derivative 2	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-triazolopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Coumarin/resveratrol hybrid derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29324067-Compound-40	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Schiff base compound 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Schiff base compound 1	NULL	NULL	NULL	NULL	NULL
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.8975670296699914	HYPOXANTHINE	ncit:C29105	HYPOXANTHINE	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenoxypiperidine derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylsulfonyl derivative 4	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine carbamate/urea derivative 3	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine carbamate/urea derivative 6	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine carbamate/urea derivative 7	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	Piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	Piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.050805681	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-21	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-56	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-67	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-14	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-16	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-17	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-18	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-25	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-36	NULL	NULL	NULL	NULL	NULL
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.1583941817064691	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-37	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-46	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-47	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Acyl piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Benzimidazole and imadazopyridine carboximidamide compound 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Benzimidazole and imadazopyridine carboximidamide compound 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Biphenyl derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 13	NULL	NULL	NULL	NULL	NULL
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	2.692701089009974	STN	ncit:C1226	SIALYL TN ANTIGEN	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Five-membered heteroaromatic compound 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Hexahydro quinoline derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Hydoxyamidine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Hydroxy amidine derivative 1	NULL	NULL	NULL	NULL	NULL
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.1666910197958555	2-CDA	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Hydroxy amidine derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Imidazo[1,5-a]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Imidazo[1,5-a]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Indazole derivative 3	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	Indazole derivative 3	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Monofluorine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-10	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-74	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-74	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Di-substituted piperidine derivative 2	NULL	NULL	NULL	NULL	NULL
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.1666910197958555	CLADRIBINE	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Di-substituted piperidine derivative 2	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Di-substituted piperidine derivative 3	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Isochroman-4-ketone derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Isochroman-4-ketone derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-2a-i	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-2a-i	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-4	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-4	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-4	NULL	NULL	NULL	NULL	NULL
XRCC5	hgnc:12833	XRCC5	NCI	14-Sep-17	NULL	3.750547945	TRIBUTYRIN	ncit:C1260	TRIBUTYRIN	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 2	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 2	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 4	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 4	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 4	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 4	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 24	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 28	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 28	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 31	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 31	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 32	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 33	NULL	NULL	NULL	NULL	NULL
KDM6A	hgnc:12637	KDM6A	OncoKB	23-Jul-20	NULL	1.500219178162699	Tazemetostat	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 33	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 36	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 36	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 36	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 37	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 37	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 37	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 40	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	OncoKB	23-Jul-20	NULL	0.8444216134395313	Tipifarnib	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 43	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 9	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-41	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-53	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-53	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-53	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-53	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-55	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-55	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-55	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-55	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-56	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-58	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-59	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-61	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	Cyclic compound 3	NULL	NULL	NULL	NULL	NULL
CDKN2A	hgnc:1787	CDKN2A	OncoKB	23-Jul-20	NULL	0.9479406894984094	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclic peptidomimetic derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocyclic peptide analog 3	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-phenyl-pyridine-2-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 5	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 6	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example1	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example11	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example11	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example15	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Carbenicillin Indanyl Sodium	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	OncoKB	23-Jul-20	NULL	0.2243917574174978	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
BACTERIAL DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clofazimine	rxcui:2592	CLOFAZIMINE	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	OI362GT	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cerdulatinib	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	TAK-329	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	(S)-(+)-Dimethindene maleate	NULL	NULL	NULL	NULL	NULL
BACTERIAL UREASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acetohydroxamic Acid	rxcui:16728	ACETOHYDROXAMIC ACID	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	NULL	Befunolol hci	NULL	NULL	NULL	NULL	NULL
PTCH1	hgnc:9585	PTCH1	OncoKB	23-Jul-20	NULL	19.69037671338543	Vismodegib	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	1.250182648468916	Anistreplase	rxcui:40028	ANISTREPLASE	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA-2/DELTA-1	hgnc:1399	CACNA2D1	TTD	2020.06.01	NULL	0.3333820395917111	Amlodipine	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
BACTERIAL DD-CARBOXYPEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefotaxime	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	1.500219178	Bitolterol	rxcui:19499	BITOLTEROL	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.6482428547616605	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	13.12691780892362	Celiprolol hcl	chembl:CHEMBL1742424	CELIPROLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
ADENOSINE DEAMINASE	hgnc:186	ADA	TTD	2020.06.01	NULL	0.1521961485092594	Cladribine	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.1389091831632129	Conjugated Estrogens	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	NULL	Dihydroergotamine nasal	NULL	NULL	NULL	NULL	NULL
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	NULL	Dihydroergotamine nasal	NULL	NULL	NULL	NULL	NULL
TROPONIN C	hgnc:5318	TNC	TTD	2020.06.01	NULL	NULL	Dihydroxyaluminium	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dolutegravir	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1185944014357865	Domperidone	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Fluvirin A(H1N1)	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Focetria A(H1N1)	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gamma-Homolinolenic acid	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	GSK2592984A	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Ibopamine hci	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.072125922	Iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.5791287268642775	Galantamine	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.073089743	Fluoxymesterone	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mitomycin	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-1439	rxcui:2055755	DORAVIRINE	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Orphenadrine	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxiconazole	rxcui:32638	OXICONAZOLE	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.088248187	Naloxone	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NF1	hgnc:7765	NF1	OncoKB	23-Jul-20	NULL	0.2536602475154323	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	2.917092846427472	PITAVASTATIN CALCIUM	rxcui:861640	PITAVASTATIN CALCIUM	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Progabide	rxcui:34568	PROGABIDE	FALSE	FALSE	FALSE
ACETYL-COA:LYSO-PAF ACETYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quercetin	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Raltitrexed	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
BACTERIAL RNA POLYMERASE SWITCH REGION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	PharmGKB	4/5/24	NULL	0.010795163	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Salsalate	rxcui:36108	SALSALATE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.596678082	Roflumilast	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	2.500365296937833	Reteplase	rxcui:76895	RETEPLASE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tilidine	rxcui:10597	TILIDINE	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tranylcypromine	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
PLASMODIUM ENOYL-ACP REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triclosan	rxcui:10795	TRICLOSAN	TRUE	FALSE	FALSE
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
NKG2 D ACTIVATING NK RECEPTOR	hgnc:18788	KLRK1	TTD	2020.06.01	NULL	NULL	NKR-2 cells	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	NSC-639829	NULL	NULL	NULL	NULL	NULL
ABCB5	hgnc:46	ABCB5	PharmGKB	4/5/24	NULL	2.072671233	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	NULL	NV-52	NULL	NULL	NULL	NULL	NULL
STMN1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pbi-shRNA STMN1 LP	ncit:C99639	PBI-SHRNA STMN1 LIPOPLEX	FALSE	FALSE	FALSE
IMMUNOGLOBULIN E	hgnc:5522	IGHE	TTD	2020.06.01	NULL	NULL	PF-06444752	NULL	NULL	NULL	NULL	NULL
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	NULL	RG7741	NULL	NULL	NULL	NULL	NULL
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.2381300282797936	RP6530	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
ANKK1	hgnc:21027	ANKK1	PharmGKB	4/5/24	NULL	0.2960958904268486	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	1.184383561707394	OTX-015	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
VASOPRESSIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SKF-105494	iuphar.ligand:2229	SKF-105494	FALSE	FALSE	FALSE
ENDOTHELIN-CONVERTING ENZYME	hgnc:3146	ECE1	TTD	2020.06.01	NULL	NULL	SLV-338	NULL	NULL	NULL	NULL	NULL
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	NULL	SLV-338	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	NULL	TAK-202	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-targeting CAR T cells	NULL	NULL	NULL	NULL	NULL
GRB2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BP-100-1-01	NULL	NULL	NULL	NULL	NULL
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	0.09869863	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	BVT.28949	NULL	NULL	NULL	NULL	NULL
ERYTHROPOIETIN	hgnc:3415	EPO	TTD	2020.06.01	NULL	1.875273972703375	ARA 290	ncit:C171683	CIBINETIDE	FALSE	FALSE	FALSE
JUN N TERMINAL KINASE	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	0.6863747873946993	CC-401	drugbank:DB12432	CC-401	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	CROBENETINE HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	0.103633562	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
INFLUENZA NEURAMINIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	DAS-181	drugbank:DB15313	DAS-181	FALSE	FALSE	FALSE
ADENOSINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	DIADENOSINE TETRAPHOSPHATE	chembl:CHEMBL339385	DIADENOSINE TETRAPHOSPHATE	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	NULL	LM-1507.NA	NULL	NULL	NULL	NULL	NULL
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	13.12691780892362	Ispinesib	ncit:C38131	ISPINESIB	FALSE	FALSE	TRUE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	NULL	M-16209	NULL	NULL	NULL	NULL	NULL
MHC CLASS I NK CELL RECEPTOR 2DL1	hgnc:6329	KIR2DL1	TTD	2020.06.01	NULL	NULL	mab 1-7F9	NULL	NULL	NULL	NULL	NULL
SLC6A5	hgnc:11051	SLC6A5	PharmGKB	4/5/24	NULL	2.072671233	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
MHC CLASS I NK CELL RECEPTOR 2DL2	hgnc:6330	KIR2DL2	TTD	2020.06.01	NULL	NULL	mab 1-7F9	NULL	NULL	NULL	NULL	NULL
MHC CLASS I NK CELL RECEPTOR 2DL3	hgnc:6331	KIR2DL3	TTD	2020.06.01	NULL	NULL	mab 1-7F9	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.7395446652914718	Niravoline	ncit:C91012	NIRAVOLINE	FALSE	FALSE	FALSE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	1.009762908	MANOALIDE	chembl:CHEMBL463914	MANOALIDE	FALSE	FALSE	FALSE
MULTIDRUG RESISTANCE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ortataxel	ncit:C1867	ORTATAXEL	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	PharmGKB	4/5/24	NULL	0.9479406894984094	palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PICORNAVIRUS CAPSID PROTEIN VP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PLECONARIL	ncit:C81604	PLECONARIL	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	R-roscovitine	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	NULL	S-0509	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.292250489	R-roscovitine	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	T-82	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Talampanel	ncit:C38139	TALAMPANEL	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.095036509	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	BUCINDOLOL	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.028161797	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
SPHINGOSINE-1 PHOSPHATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAF312	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
INTEGRIN ALPHA-V/BETA-3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cilengitide	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	NULL	Claritin/Singulair	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	FARGLITAZAR	ncit:C81693	FARGLITAZAR	FALSE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	FK949E	NULL	NULL	NULL	NULL	NULL
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	1.166837138570988	lumiracoxib	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
SMAD7 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	GED-0301	iuphar.ligand:8277	MONGERSEN	FALSE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	ITF2357	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
O-6-METHYLGUANINE-DNA-ALKYLTRANSFERASE	hgnc:7059	MGMT	TTD	2020.06.01	NULL	NULL	O6-Benzylguanine alkylade	NULL	NULL	NULL	NULL	NULL
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	PC-DAC:Insulin	NULL	NULL	NULL	NULL	NULL
RORA	hgnc:10258	RORA	PharmGKB	4/5/24	NULL	0.750109589	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.028290771	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:3251	iuphar.ligand:3251	[3H]WAY100635	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.090374649	IUPHAR.LIGAND:51	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.052718545	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.081281225	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.1595977849109255	IUPHAR.LIGAND:3	iuphar.ligand:3	1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:168	iuphar.ligand:168	VER-3323	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:193	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.03070624	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.077217164	IUPHAR.LIGAND:210	ncit:C73158	SARPOGRELATE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.064347636	IUPHAR.LIGAND:28	iuphar.ligand:28	SB 216641	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:187	iuphar.ligand:187	RS-102221	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:8689	ncit:C166835	IDALOPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:8426	iuphar.ligand:8426	TD-8954	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.1483267549030917	IUPHAR.LIGAND:12	iuphar.ligand:12	EMDT	FALSE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.251232877	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.060772768	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.8899605294185507	IUPHAR.LIGAND:8429	iuphar.ligand:8429	WAY-208466	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:3241	iuphar.ligand:3241	SB399885	FALSE	FALSE	FALSE
NCBIGENE:2937	hgnc:4624	GSS	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10125	iuphar.ligand:10125	PFKFB3 KINASE INHIBITOR 69	FALSE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.1973972602845657	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
NCBIGENE:1658	hgnc:188	ADAM10	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8568	iuphar.ligand:8568	COMPOUND 25 [PMID: 18068976]	FALSE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.082494377	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:7791	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
NCBIGENE:1787	hgnc:2977	TRDMT1	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8107	iuphar.ligand:8107	VACTOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1264	hgnc:2155	CNN1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:5280	iuphar.ligand:5280	TOFA	FALSE	FALSE	FALSE
PGM1	hgnc:8905	PGM1	PharmGKB	4/5/24	NULL	10.50153425	acetaldehyde	rxcui:1311137	ACETALDEHYDE	TRUE	FALSE	FALSE
NCBIGENE:1658	hgnc:188	ADAM10	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:9687	iuphar.ligand:9687	GI254023X	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:12388	iuphar.ligand:12388	ZOTIZALKIB	FALSE	FALSE	FALSE
NCBIGENE:3070	hgnc:4861	HELLS	GuideToPharmacology	2024.1	inhibitor	2.019525816757481	IUPHAR.LIGAND:5277	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
NCBIGENE:2768	hgnc:4380	GNA12	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8637	iuphar.ligand:8637	AK198	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:8207	iuphar.ligand:8207	COMPOUND 5G [PMID: 20483621]	FALSE	FALSE	FALSE
NCBIGENE:2768	hgnc:4380	GNA12	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7418	ncit:C72879	ZENARESTAT	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.085378327	IUPHAR.LIGAND:503	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.040235763	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:7109	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:495	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:501	rxcui:5784	INDORAMIN	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:7170	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.053964719	IUPHAR.LIGAND:9868	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:7310	rxcui:10634	TOLAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.1392776425349987	IUPHAR.LIGAND:6812	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:7849	iuphar.ligand:7849	ANDARINE	FALSE	FALSE	FALSE
ADH7	hgnc:256	ADH7	PharmGKB	4/5/24	NULL	0.6646540662746139	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:1559	hgnc:2623	CYP2C9	GuideToPharmacology	2024.1	inhibitor	0.1215455352678113	IUPHAR.LIGAND:8677	iuphar.ligand:8677	COMPOUND 9 [PMID: 1738140]	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.086219493	IUPHAR.LIGAND:3283	iuphar.ligand:3283	SCH442416	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:11154	ncit:C159564	ETRUMADENANT	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:449	iuphar.ligand:449	MRS1754	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:8060	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6905	iuphar.ligand:6905	[SAR1,ILE8]ANG-II	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6909	iuphar.ligand:6909	LY301875	FALSE	FALSE	FALSE
COL26A1	hgnc:18038	COL26A1	PharmGKB	4/5/24	NULL	1.500219178	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:6166	iuphar.ligand:6166	PHYLLOLITORIN	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:616	iuphar.ligand:616	BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:1466	hgnc:2470	CSRP2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10946	iuphar.ligand:10946	CCG258747	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:10520	iuphar.ligand:10520	AM-6494	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:9816	iuphar.ligand:9816	LEVOSALBUTAMOL	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.06697407	IUPHAR.LIGAND:7297	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.066297565	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:562	iuphar.ligand:562	[125I]ICYP	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:5674	iuphar.ligand:5674	CHIR-265	FALSE	FALSE	TRUE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	0.280789686	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7516	iuphar.ligand:7516	COMPOUND 4D [PMID: 21851057]	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7522	iuphar.ligand:7522	COMPOUND 38 [PMID: 24000170]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:12141	iuphar.ligand:12141	XY-06-007	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.010375838	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:2726	hgnc:14310	BRD7	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8950	iuphar.ligand:8950	BI-9564	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:10457	ncit:C175851	REMIBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:637	iuphar.ligand:637	LYS-KALLIDIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.024309107	etrasimod	rxcui:2668045	ETRASIMOD	TRUE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:669	iuphar.ligand:669	FR191413	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:655	iuphar.ligand:655	B-9958	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11436	iuphar.ligand:11436	[125I]HPP-HOE140	FALSE	FALSE	FALSE
NCBIGENE:1949	hgnc:3228	EFNB3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8110	iuphar.ligand:8110	COMPOUND 2-3-2 [PMID: 24900824]	FALSE	FALSE	FALSE
NCBIGENE:1949	hgnc:3228	EFNB3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8109	iuphar.ligand:8109	COMPOUND 2-1-1 [PMID: 24900824]	FALSE	FALSE	FALSE
NCBIGENE:1949	hgnc:3228	EFNB3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8111	iuphar.ligand:8111	COMPOUND 2-3-1 [PMID: 24900824]	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:676	iuphar.ligand:676	NPC-567	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5762	iuphar.ligand:5762	PMX205	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:12516	iuphar.ligand:12516	EU-DTPA-[SER27, NLE70]HC5A	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:3529	iuphar.ligand:3529	SB290157	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:12257	iuphar.ligand:12257	CACCINH-A01	FALSE	FALSE	FALSE
NCBIGENE:1625	ncbigene:1625	DBIL3	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6515	iuphar.ligand:6515	ISATIN SULFONAMIDE 34 [PMID: 11384246]	FALSE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	blocker	5.834185692854944	IUPHAR.LIGAND:4149	iuphar.ligand:4149	CALCISEPTINE	FALSE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7724	iuphar.ligand:7724	TTA-A2	FALSE	FALSE	FALSE
NCBIGENE:2353	hgnc:3796	FOS	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:9298	iuphar.ligand:9298	LHVS	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.081281225	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:3502	iuphar.ligand:3502	GSK COMPOUND 34	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:788	iuphar.ligand:788	MET-CK&BETA;7	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:4359	iuphar.ligand:4359	VMIP-III	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:763	iuphar.ligand:763	[125I]CCL3 (HUMAN)	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.1215455352678113	lornoxicam	rxcui:20890	LORNOXICAM	TRUE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8115	iuphar.ligand:8115	COMPOUND 2 [PMID: 22560567]	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:9618	iuphar.ligand:9618	IBERDOMIDE	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	0.596678082	IUPHAR.LIGAND:4335	iuphar.ligand:4335	UCCF-029	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4337	iuphar.ligand:4337	UCCF-339	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	0.070197421	IUPHAR.LIGAND:2486	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	0.3977853881492006	IUPHAR.LIGAND:4271	iuphar.ligand:4271	NS004	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:10533	iuphar.ligand:10533	DTAG-13	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:6030	iuphar.ligand:6030	PURVALANOL A	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:8051	iuphar.ligand:8051	BMS-265246	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:7379	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:6045	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:10547	iuphar.ligand:10547	THAL-SNS-032	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:11065	drugbank:DB08463	(2R)-2-({9-(1-METHYLETHYL)-6-[(4-PYRIDIN-2-YLBENZYL)AMINO]-9H-PURIN-2-YL}AMINO)BUTAN-1-OL	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:6045	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:6045	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:8176	iuphar.ligand:8176	BS-194	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.2586584789935689	IUPHAR.LIGAND:8114	drugbank:DB07149	(7S)-2-(2-AMINOPYRIMIDIN-4-YL)-7-(2-FLUOROETHYL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.3621218705909966	IUPHAR.LIGAND:7934	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:10203	iuphar.ligand:10203	ENDOXIFEN	FALSE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.024490518	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1321	ncbigene:1321	CORD4	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8754	iuphar.ligand:8754	COMPOUND 39A [PMID: 15634016]	FALSE	FALSE	FALSE
NCBIGENE:1329	hgnc:2269	COX5B	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11353	iuphar.ligand:11353	BERBERINE	FALSE	FALSE	FALSE
NCBIGENE:1366	hgnc:2049	CLDN7	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:5210	ncit:C1433	LIAROZOLE	FALSE	FALSE	FALSE
KLRD1	hgnc:6378	KLRD1	PharmGKB	4/5/24	NULL	0.6364566210387212	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NCBIGENE:2743	hgnc:4329	GLRB	GuideToPharmacology	2024.1	antibody	2.625383561784724	IUPHAR.LIGAND:12966	iuphar.ligand:12966	CADONILIMAB	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:6195	iuphar.ligand:6195	[3H]LTC4	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	PharmGKB	4/5/24	NULL	0.009787078	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:902	hgnc:1594	CCNH	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:1372	drugbank:DB02999	QUISQUALIC ACID	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:9983	iuphar.ligand:9983	VANOXERINE	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:4792	rxcui:7500	NOMIFENSINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1161674142382621	IUPHAR.LIGAND:8868	iuphar.ligand:8868	SCH221510	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.2323348284765243	IUPHAR.LIGAND:1635	iuphar.ligand:1635	CTAP	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.027333509	IUPHAR.LIGAND:1638	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	5.527123287967842	IUPHAR.LIGAND:12106	iuphar.ligand:12106	FARUDODSTAT	FALSE	FALSE	FALSE
NCBIGENE:1396	hgnc:2360	CRIP1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5255	iuphar.ligand:5255	RHC80267	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.053854022	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.007866318	IUPHAR.LIGAND:968	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.058997383	IUPHAR.LIGAND:983	iuphar.ligand:983	NEMONAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.040766825	IUPHAR.LIGAND:7279	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.1141471113819445	IUPHAR.LIGAND:941	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.150021918	IUPHAR.LIGAND:941	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:5781	iuphar.ligand:5781	U101958	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.078958904	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
CRHR2	hgnc:2358	CRHR2	PharmGKB	4/5/24	NULL	0.2143170254518142	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:2833	hgnc:4540	CXCR3	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8230	iuphar.ligand:8230	IOX1	FALSE	FALSE	FALSE
NCBIGENE:2487	hgnc:3959	FRZB	GuideToPharmacology	2024.1	modulator	4.375639269641208	IUPHAR.LIGAND:10515	iuphar.ligand:10515	MAK683	FALSE	FALSE	FALSE
NCBIGENE:1825	hgnc:3037	DSC3	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:1823	hgnc:3035	DSC1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:7903	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9765	ncit:C120307	MAVELERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.033338204	IUPHAR.LIGAND:7719	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:7959	ncit:C143046	RALIMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12982	iuphar.ligand:12982	JBJ-04-125-02	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:9929	iuphar.ligand:9929	XILIERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8999	iuphar.ligand:8999	(S)-ARN2508	FALSE	FALSE	FALSE
NCBIGENE:1401	hgnc:2367	CRP	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10248	iuphar.ligand:10248	ASP8477	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.014206621	olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:2534	hgnc:4037	FYN	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8788	iuphar.ligand:8788	HM50316	FALSE	FALSE	FALSE
NCBIGENE:3017	hgnc:4747	H2BC5	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:10067	iuphar.ligand:10067	AFM13	FALSE	FALSE	FALSE
NCBIGENE:227	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1058	rxcui:164	ACETATE	TRUE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.051177067	IUPHAR.LIGAND:7877	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:8862	iuphar.ligand:8862	BLU-9931	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.092606122	IUPHAR.LIGAND:7877	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.003418468	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.019534104	IUPHAR.LIGAND:5671	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:7879	iuphar.ligand:7879	BMS-690514	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:5972	iuphar.ligand:5972	FLT-3 INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:10420	iuphar.ligand:10420	CHMFL-KIT-64	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.007196775	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.045461187	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
AMPD1	hgnc:468	AMPD1	PharmGKB	4/5/24	NULL	0.2430910705356226	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:5838	iuphar.ligand:5838	T20(DP178)	FALSE	FALSE	FALSE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1044	iuphar.ligand:1044	ANNEXIN I-(2-26)	FALSE	FALSE	FALSE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.16256245	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:2025	hgnc:3352	ENO1P1	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.1201548540862574	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:4367	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.049337723	IUPHAR.LIGAND:7313	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4257	iuphar.ligand:4257	MRK016	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.047886613	IUPHAR.LIGAND:7111	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.4070362111294147	IUPHAR.LIGAND:12917	iuphar.ligand:12917	ABBV-3373	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.305277158	IUPHAR.LIGAND:7078	rxcui:4462	FLUOCINONIDE	TRUE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:2361	drugbank:DB01931	5,7-DICHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
NCBIGENE:451	hgnc:769	ASS1P6	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:4075	iuphar.ligand:4075	[3H]SYM2081	FALSE	FALSE	FALSE
NCBIGENE:452	hgnc:4581	GRIK3	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:4075	iuphar.ligand:4075	[3H]SYM2081	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	blocker	0.1346350544504987	IUPHAR.LIGAND:4128	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1189	ncit:C132277	TEVERELIX	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	modulator	0.1136529680426287	IUPHAR.LIGAND:1192	iuphar.ligand:1192	5-(N,N-HEXAMETHYLENE)-AMILORIDE	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:9070	iuphar.ligand:9070	DENDROASPIS NATRIURETIC PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:9069	rxcui:1873752	PLECANATIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006525935	mianserin	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:401	hgnc:691	PHOX2A	GuideToPharmacology	2024.1	blocker	2.625383561784725	IUPHAR.LIGAND:2355	ncit:C81347	CILOBRADINE	FALSE	FALSE	FALSE
NCBIGENE:402	hgnc:693	ARL2	GuideToPharmacology	2024.1	blocker	2.100306849	IUPHAR.LIGAND:2355	ncit:C81347	CILOBRADINE	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:5800	iuphar.ligand:5800	COMPOUND 6O [PMID: 19524438]	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.081030357	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.025588534	IUPHAR.LIGAND:7009	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.1556551518844698	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	1.050153425	interferon beta-1b	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.112919723	IUPHAR.LIGAND:8365	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:7491	iuphar.ligand:7491	TMP269	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:11118	drugbank:DB14979	MARTINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:7500	iuphar.ligand:7500	RGFP966	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.2134458180312784	IUPHAR.LIGAND:11118	drugbank:DB14979	MARTINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.1988926940746004	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:67	iuphar.ligand:67	9-OH-RISPERIDONE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:7121	rxcui:18603	AZELASTINE	TRUE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:7491	iuphar.ligand:7491	TMP269	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:1265	iuphar.ligand:1265	CIPROXIFAN	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:10102	rxcui:61455	MIZOLASTINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:7151	rxcui:2977	CYCLIZINE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:4025	iuphar.ligand:4025	AMTHAMINE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.056097939	celiprolol	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:3957	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.037721028	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:1194	iuphar.ligand:1194	2-(3-BROMOPHENYL)HISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.062509132	IUPHAR.LIGAND:2954	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:3031	ncit:C96285	MEVASTATIN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.018699313	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
NCBIGENE:99	hgnc:4487	GPR32	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:5555	iuphar.ligand:5555	RVD1-ME	FALSE	FALSE	FALSE
NCBIGENE:104	hgnc:226	ADARB1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:6067	iuphar.ligand:6067	PROSAPTIDE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.012466209	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
NCBIGENE:83	hgnc:155	ACTG1P10	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:7802	iuphar.ligand:7802	DIPHENYLENEIODONIUM CHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5534	iuphar.ligand:5534	LAURIC ACID	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:5525	iuphar.ligand:5525	O-1602	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:10345	iuphar.ligand:10345	COMPOUND 3A [BADOLATO ET AL., 2019]	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.005753635	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:5231	iuphar.ligand:5231	NIL	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.074797252	itraconazole	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
NCBIGENE:2625	hgnc:4172	GATA3	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10741	ncit:C66097	MERIMEPODIB	FALSE	FALSE	FALSE
NCBIGENE:1402	hgnc:736	NAAA	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:10120	iuphar.ligand:10120	ARN19702	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.018193926	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	activator	0.3431873936973497	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.034521809	pyrazinamide	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.4375639269641209	IUPHAR.LIGAND:12424	iuphar.ligand:12424	L-TRP-TRP-TRP	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12447	drugbank:DB07928	N-(2-OXOTETRAHYDROFURAN-3-YL)OCTANAMIDE	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12448	iuphar.ligand:12448	SANTONIN	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:12446	iuphar.ligand:12446	NOBILETIN	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	NULL	0.172722603	IUPHAR.LIGAND:12310	iuphar.ligand:12310	SJ988497	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:10527	iuphar.ligand:10527	LASW1393	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:9387	iuphar.ligand:9387	CEP-33779	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:8123	iuphar.ligand:8123	COMPOUND 1D [PMID: 21493067]	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.074797252	sparfloxacin	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1647	iuphar.ligand:1647	DAMGO	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9191	iuphar.ligand:9191	PROBE 1.1 [PMID: 24187130]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:3475	ncit:C80576	ENADOLINE	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:8867	iuphar.ligand:8867	SR16835	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1622	iuphar.ligand:1622	DYNORPHIN B	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:1640	iuphar.ligand:1640	NALTRIBEN	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.002594253	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.041508041	IUPHAR.LIGAND:10136	ncit:C148147	LAZERTINIB	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	PharmGKB	4/5/24	NULL	0.2885036881082115	norclobazam	drugbank:DB17092	NORCLOBAZAM	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.004716823	IUPHAR.LIGAND:7881	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:7882	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
NCBIGENE:521	hgnc:846	ATP5ME	GuideToPharmacology	2024.1	activator	0.2083637747448194	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	activator	1.591141552596802	IUPHAR.LIGAND:4271	iuphar.ligand:4271	NS004	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9317	iuphar.ligand:9317	RA-2	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:10019	rxcui:50749	HALOFANTRINE	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:7664	iuphar.ligand:7664	NC00075159	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	1.050153425	sodium ascorbate	rxcui:267366	SODIUM ASCORBATE	TRUE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:11479	iuphar.ligand:11479	RETIGABINE DERIVATIVE 10G	FALSE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:11479	iuphar.ligand:11479	RETIGABINE DERIVATIVE 10G	FALSE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6709	iuphar.ligand:6709	COMPOUND 1 [PMID: 22533316]	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.013546871	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:2932	hgnc:4617	GSK3B	GuideToPharmacology	2024.1	antibody	1.141471113819445	IUPHAR.LIGAND:9536	iuphar.ligand:9536	RELATLIMAB	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9929	iuphar.ligand:9929	XILIERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1271	hgnc:2170	CNTFR	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:5159	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	PharmGKB	4/5/24	NULL	0.8178764989983567	pemigatinib	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:2913	hgnc:4595	GRM3	GuideToPharmacology	2024.1	antibody	5.250767123569449	IUPHAR.LIGAND:11762	iuphar.ligand:11762	LIVMONIPLIMAB	FALSE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8119	iuphar.ligand:8119	COMPOUND 35 [PMID: 22902653]	FALSE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6548	iuphar.ligand:6548	DG-051	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10035	iuphar.ligand:10035	COMPOUND 17L [PMID: 26288691]	FALSE	FALSE	FALSE
NCBIGENE:2055	hgnc:2079	CLN8	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8117	iuphar.ligand:8117	COMPOUND 31 [PMID: 22902653]	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	1.029562181092048	IUPHAR.LIGAND:11313	iuphar.ligand:11313	CPX	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:11798	iuphar.ligand:11798	BMS-986278	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	PharmGKB	4/5/24	NULL	0.093596562	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8980	iuphar.ligand:8980	RN-1	FALSE	FALSE	FALSE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	0.9376369863516874	IUPHAR.LIGAND:6999	iuphar.ligand:6999	ANACARDIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2680	hgnc:9886	KDM5A	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10141	iuphar.ligand:10141	KDM5 INHIBITOR N71	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:8587	iuphar.ligand:8587	MQ1	FALSE	FALSE	FALSE
STX4	hgnc:11439	STX4	PharmGKB	4/5/24	NULL	5.834185692854944	phenprocoumon	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	0.8751278539282418	IUPHAR.LIGAND:1324	rxcui:2262250	AFAMELANOTIDE	TRUE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	0.8751278539282418	IUPHAR.LIGAND:1324	rxcui:2262250	AFAMELANOTIDE	TRUE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:9133	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6259	iuphar.ligand:6259	THIIC	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	modulator	0.364636606	IUPHAR.LIGAND:7626	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:12334	iuphar.ligand:12334	COMPOUND 25C [PMID: 36649216]	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:12706	drugbank:DB15498	BOS172722	FALSE	FALSE	FALSE
MACROD2	hgnc:16126	MACROD2	PharmGKB	4/5/24	NULL	4.039051633514962	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:292	iuphar.ligand:292	NNC 11-1585	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.1262203635473425	IUPHAR.LIGAND:335	iuphar.ligand:335	G&OUML; 7874	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.026572708	IUPHAR.LIGAND:305	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.050488145	IUPHAR.LIGAND:298	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:310	iuphar.ligand:310	HEXAHYDROSILADIFENIDOL	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.055271233	IUPHAR.LIGAND:298	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.046059361	IUPHAR.LIGAND:325	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.07458476	IUPHAR.LIGAND:340	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:298	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:292	iuphar.ligand:292	NNC 11-1585	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:361	iuphar.ligand:361	TRIPITRAMINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.596678082	IUPHAR.LIGAND:12301	iuphar.ligand:12301	VU0467154	FALSE	FALSE	FALSE
TNFRSF1B	hgnc:11917	TNFRSF1B	PharmGKB	4/5/24	NULL	0.6058577450272442	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:348	iuphar.ligand:348	THIOCHROME	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:330	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:10129	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	1.419126249613364	IUPHAR.LIGAND:8289	iuphar.ligand:8289	AAE-M-PBP-AMINE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:8867	iuphar.ligand:8867	SR16835	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.096167896	IUPHAR.LIGAND:9002	iuphar.ligand:9002	BW373U86	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:7691	rxcui:1653781	ELUXADOLINE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:8868	iuphar.ligand:8868	SCH221510	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.2885036881082115	IUPHAR.LIGAND:9838	iuphar.ligand:9838	UFP-505	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.048083948	IUPHAR.LIGAND:7215	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2789	hgnc:4409	GNG5P1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7728	iuphar.ligand:7728	AZD5904	FALSE	FALSE	FALSE
CERS6	hgnc:23826	CERS6	PharmGKB	4/5/24	NULL	1.009762908	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NCBIGENE:2111	hgnc:27972	MYLK4	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12185	iuphar.ligand:12185	COMPOUND 17 [PMID: 36111834]	FALSE	FALSE	FALSE
NCBIGENE:970	hgnc:11937	CD70	GuideToPharmacology	2024.1	inhibitor	0.577007376	IUPHAR.LIGAND:4835	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
PTTG1	hgnc:9690	PTTG1	PharmGKB	4/5/24	NULL	4.039051633514962	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NCBIGENE:1847	hgnc:3071	DUSP5	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
NCBIGENE:3001	hgnc:4708	GZMA	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9933	iuphar.ligand:9933	NSC 780521	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7570	iuphar.ligand:7570	HUWENTOXIN IV	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	PharmGKB	4/5/24	NULL	0.076208521	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	blocker	0.9376369863516875	IUPHAR.LIGAND:2625	iuphar.ligand:2625	SAXITOXIN	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:2614	iuphar.ligand:2614	ATX-II	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	modulator	0.6035364509849942	IUPHAR.LIGAND:3986	iuphar.ligand:3986	A-867744	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2111	ncit:C152301	SAREDUTANT	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:5764	iuphar.ligand:5764	SB 218795	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:2111	ncit:C152301	SAREDUTANT	FALSE	FALSE	FALSE
CD84	hgnc:1704	CD84	PharmGKB	4/5/24	NULL	6.058577450272442	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1684	iuphar.ligand:1684	RO64-6198	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:1485	iuphar.ligand:1485	BIBP3226	FALSE	FALSE	FALSE
NCBIGENE:2871	hgnc:4547	GRK6P1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8702	iuphar.ligand:8702	KML110	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	PharmGKB	4/5/24	NULL	0.2019525816757481	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NCBIGENE:3220	hgnc:5121	HOXC@	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12352	iuphar.ligand:12352	COMPOUND 15A [PMID: 36642961]	FALSE	FALSE	FALSE
NCBIGENE:1020	hgnc:1774	CDK5	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:8482	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	NULL	0.3500511415712966	IUPHAR.LIGAND:4748	ncit:C47521	ESTROPIPATE	FALSE	FALSE	FALSE
NCBIGENE:3101	hgnc:4925	HK3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10509	iuphar.ligand:10509	THIAMET-G	FALSE	FALSE	FALSE
NCBIGENE:1222	hgnc:13819	SLCO1C1	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:4627	iuphar.ligand:4627	[125I]THYROXINE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.009471081	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NCBIGENE:1225	hgnc:10952	SLCO3A1	GuideToPharmacology	2024.1	NULL	0.8751278539282418	IUPHAR.LIGAND:1916	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2250	iuphar.ligand:2250	L-368,930	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5804	iuphar.ligand:5804	PFIZER COMPOUND 11 [PMID:18445527]	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	0.070197421	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6080	iuphar.ligand:6080	PCA 4248	FALSE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	PharmGKB	4/5/24	NULL	6.848826682916673	Pertussis vaccines	rxcui:8080	PERTUSSIS VACCINE	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2258	iuphar.ligand:2258	PACAP-38	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:4499	iuphar.ligand:4499	LYS[Z(NO2)]-LYS[Z(NO2)]	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	NULL	4.039051633514961	IUPHAR.LIGAND:12599	iuphar.ligand:12599	AC-[13C,15N]PGP	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:4499	iuphar.ligand:4499	LYS[Z(NO2)]-LYS[Z(NO2)]	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2656	iuphar.ligand:2656	GW409544	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2696	iuphar.ligand:2696	L-764406	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.028413242	IUPHAR.LIGAND:2700	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.2949869170544634	IUPHAR.LIGAND:10578	iuphar.ligand:10578	AS-252424	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.035418328	fesoterodine	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:9424	rxcui:2633005	LENIOLISIB	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.084281976	IUPHAR.LIGAND:7795	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1966579447029756	IUPHAR.LIGAND:10001	iuphar.ligand:10001	COMPOUND 52 [PMID: 28541707]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.034704343	IUPHAR.LIGAND:7936	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1966579447029756	IUPHAR.LIGAND:10162	iuphar.ligand:10162	RV1729	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.046303061	IUPHAR.LIGAND:8059	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:8244	iuphar.ligand:8244	TGX-221	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:8382	iuphar.ligand:8382	VS-5584	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.012054103	mavacamten	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:10001	iuphar.ligand:10001	COMPOUND 52 [PMID: 28541707]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:9907	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:10578	iuphar.ligand:10578	AS-252424	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:8244	iuphar.ligand:8244	TGX-221	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:10096	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.096521454	IUPHAR.LIGAND:8527	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:5225	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.029515273	terbinafine	rxcui:37801	TERBINAFINE	TRUE	FALSE	FALSE
NCBIGENE:1295	hgnc:2215	COL8A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12003	ncit:C177065	LENRISPODUN	FALSE	FALSE	FALSE
SCNN1A	hgnc:10599	SCNN1A	PharmGKB	4/5/24	NULL	2.917092846427472	triamterene	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
NCBIGENE:2145	hgnc:3526	EZH1	GuideToPharmacology	2024.1	inhibitor	2.019525816757481	IUPHAR.LIGAND:8204	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
NCBIGENE:2857	hgnc:4490	GPR34	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12185	iuphar.ligand:12185	COMPOUND 17 [PMID: 36111834]	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.2143170254518143	IUPHAR.LIGAND:7698	iuphar.ligand:7698	AZD1208	FALSE	FALSE	FALSE
NCBIGENE:3145	hgnc:4982	HMBS	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12019	iuphar.ligand:12019	GNF-1331	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.013622434	quinine	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:12141	iuphar.ligand:12141	XY-06-007	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.022467981	IUPHAR.LIGAND:7080	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.032837818	IUPHAR.LIGAND:7434	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
NCBIGENE:2385	hgnc:8747	PCSK5	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:8668	iuphar.ligand:8668	FURIN INHIBITOR PEPTIDE	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	PharmGKB	4/5/24	NULL	0.364636606	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
NCBIGENE:1213	hgnc:2092	CLTC	GuideToPharmacology	2024.1	inhibitor	0.1875273972703375	IUPHAR.LIGAND:1909	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:1787	iuphar.ligand:1787	PTHRP-(1-20)/TIP-(23-39) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1161	hgnc:3439	ERCC8	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1800	iuphar.ligand:1800	[ILE5,TRP23]PTHRP-(3-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:3006	hgnc:4716	H1-2	GuideToPharmacology	2024.1	modulator	2.500365296937833	IUPHAR.LIGAND:10473	rxcui:2594468	MITAPIVAT	TRUE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:12095	iuphar.ligand:12095	EXARAFENIB	FALSE	FALSE	FALSE
NCBIGENE:2631	hgnc:4179	NIPSNAP2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:6802	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
NCBIGENE:1866	ncbigene:1866	DYT7	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10109	iuphar.ligand:10109	7-BIA	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:2930	iuphar.ligand:2930	VPC44116	FALSE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	activator	0.3860858179095184	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:2926	iuphar.ligand:2926	SEW2871	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:9492	iuphar.ligand:9492	COMPOUND 43 [PMID: 26751273]	FALSE	FALSE	FALSE
NCBIGENE:840	hgnc:1508	CASP7	GuideToPharmacology	2024.1	modulator	3.088686543276147	IUPHAR.LIGAND:8822	iuphar.ligand:8822	TGN4	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	0.364636606	synthetic conjugated estrogens, A	rxcui:253166	SYNTHETIC CONJUGATED ESTROGENS, A	FALSE	FALSE	FALSE
CRY1	hgnc:2384	CRY1	PharmGKB	4/5/24	NULL	1.544343271638073	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.3561566847382379	brimonidine	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	20.00292237550266	paromomycin	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
SRPRB	hgnc:24085	SRPRB	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.081092929	dactinomycin	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.6250913242344582	venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
NCBIGENE:2211	hgnc:11388	STK10	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.048844345	IUPHAR.LIGAND:4790	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:1535	hgnc:2577	CYBA	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8040	iuphar.ligand:8040	GSK650394	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1356787370431382	IUPHAR.LIGAND:2586	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.2169738480813822	dapsone	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
NCBIGENE:833	hgnc:1493	CARS1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:6806	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	PharmGKB	4/5/24	NULL	0.2143170254518142	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:4754	rxcui:1545653	EMPAGLIFLOZIN	TRUE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3077	iuphar.ligand:3077	COMPOUND 4G [PMID: 17709461]	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.1029562181092049	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2038	iuphar.ligand:2038	BIM 23060	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	PharmGKB	4/5/24	NULL	0.2344092465879218	brimonidine	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:2027	iuphar.ligand:2027	BIM 23627	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2056	iuphar.ligand:2056	[111IN,90Y]DOTA-LAN	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:2149	iuphar.ligand:2149	OCTOPAMINE	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:2150	iuphar.ligand:2148	[3H]TYRAMINE	FALSE	FALSE	FALSE
NCBIGENE:2240	hgnc:11732	TESK2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8119	iuphar.ligand:8119	COMPOUND 35 [PMID: 22902653]	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:12768	drugbank:DB15137	VK-2809	FALSE	FALSE	FALSE
NCBIGENE:1754	hgnc:11850	TLR4	GuideToPharmacology	2024.1	agonist	4.565884455277782	IUPHAR.LIGAND:11150	iuphar.ligand:11150	GSK1795091	FALSE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	1.009762908	glimepiride	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6309	iuphar.ligand:6309	PF-4840154	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:10284	iuphar.ligand:10284	GSK2833503A	FALSE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	blocker	0.3860858179095184	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:511	hgnc:3145	TRPV5	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:12559	iuphar.ligand:12559	OXOGLAUCINE	FALSE	FALSE	FALSE
NCBIGENE:1871	hgnc:3115	E2F3	GuideToPharmacology	2024.1	NULL	4.375639269641208	IUPHAR.LIGAND:5064	iuphar.ligand:5064	LYMPHOTOXIN-&ALPHA;	FALSE	FALSE	FALSE
MYOCD	hgnc:16067	MYOCD	PharmGKB	4/5/24	NULL	3.088686543276147	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.1930429089547592	IUPHAR.LIGAND:6851	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	0.2885036881082116	IUPHAR.LIGAND:611	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:8707	rxcui:1876905	DEUTETRABENAZINE	TRUE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	2.019525817	phenprocoumon	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:7747	ncit:C83818	INECALCITOL	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2271	iuphar.ligand:2271	N-STEARYL-[NLE17]VIP	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2261	iuphar.ligand:2261	[125I]PACAP-27	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.008310806	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
NCBIGENE:2645	hgnc:4195	GCK	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:6808	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
NCBIGENE:2645	hgnc:4195	GCK	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:2645	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2257	iuphar.ligand:2257	PACAP-27	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.2083637747448194	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	NULL	2.625383561784724	IUPHAR.LIGAND:11726	iuphar.ligand:11726	COMPOUND 20 [PMID: 34432979]	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1545	iuphar.ligand:1545	[LEU31,PRO34]NPY	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.011162345	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.1374032518317239	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
EZH2	hgnc:3527	EZH2	CIViC	10-Apr-24	NULL	2.917092846427472	TAZEMETOSTAT	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	0.1093909817410302	REBASTINIB	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.4817217544559128	tianeptine	rxcui:38252	TIANEPTINE	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.272767123	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	3.000438356	ONARTUZUMAB	ncit:C82348	ONARTUZUMAB	FALSE	TRUE	TRUE
MITF	hgnc:7105	MITF	CIViC	10-Apr-24	NULL	0.036692992	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	0.637458239	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	0.1108075556053025	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	CIViC	10-Apr-24	NULL	0.1312691780892362	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
SMO	hgnc:11119	SMO	CIViC	10-Apr-24	NULL	5.104912481248077	SONIDEGIB	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	CIViC	10-Apr-24	NULL	0.010902756	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.040515178	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
TMX2	hgnc:30739	TMX2	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CALR	hgnc:1455	CALR	CIViC	10-Apr-24	NULL	0.2263261691193728	PEGINTERFERON ALFA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
AURKA	hgnc:11393	AURKA	CIViC	10-Apr-24	NULL	NULL	RADIATION THERAPY	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.015768069	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.1084869240406911	praziquantel	rxcui:8628	PRAZIQUANTEL	TRUE	FALSE	FALSE
ZEB1	hgnc:11642	ZEB1	CIViC	10-Apr-24	NULL	0.4268916360625569	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.1032937794800547	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.3241214273808302	FLT3/ABL/AURORA KINASE INHIBITOR KW-2449	ncit:C116858	FLT3/ABL/AURORA KINASE INHIBITOR KW-2449	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	AMG511	NULL	NULL	NULL	NULL	NULL
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	0.525076712	lorazepam	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	CIViC	10-Apr-24	NULL	NULL	ALK2 INHIBITOR LDN-193189	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	AGS324	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	KW2449	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.028360625	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	KG5	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.1374546367426557	MEK INHIBITOR TAK-733	iuphar.ligand:9911	TAK-733	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	CIViC	10-Apr-24	NULL	0.043629141	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.012676888	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	CIViC	10-Apr-24	NULL	0.2991890098899971	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1773907812016706	PI3K/BET INHIBITOR LY294002	ncit:C148229	PI3K/BET INHIBITOR LY294002	FALSE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.1861974157294131	QUARFLOXIN	ncit:C71726	QUARFLOXIN	FALSE	FALSE	TRUE
ATXN1L	hgnc:33279	ATXN1L	CIViC	10-Apr-24	NULL	0.6482428547616604	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.072324616	proguanil	rxcui:2382	PROGUANIL	TRUE	FALSE	FALSE
ASS1	hgnc:758	ASS1	CIViC	10-Apr-24	NULL	0.1172046232939609	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.013179636	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	NULL	HYPERTHERMIC INTRAPERITONEAL CHEMOTHERAPY	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.9842513760562132	IVOSIDENIB	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	0.010058941	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PML	hgnc:9113	PML	CIViC	10-Apr-24	NULL	0.8751278539282418	GEMTUZUMAB OZOGAMICIN	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	NULL	BPTES	NULL	NULL	NULL	NULL	NULL
NOS1	hgnc:7872	NOS1	PharmGKB	4/5/24	NULL	0.018037675	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NT5C2	hgnc:8022	NT5C2	CIViC	10-Apr-24	NULL	NULL	ARABINOSYLGUANINE	NULL	NULL	NULL	NULL	NULL
PTPRD	hgnc:9668	PTPRD	CIViC	10-Apr-24	NULL	NULL	IGF1R MONOCLONAL ANTIBODY	NULL	NULL	NULL	NULL	NULL
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.3580068493342807	meloxicam	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
CRLF2	hgnc:14281	CRLF2	CIViC	10-Apr-24	NULL	0.3070624048871023	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TOP2A	hgnc:11989	TOP2A	CIViC	10-Apr-24	NULL	NULL	MVT REGIMEN	NULL	NULL	NULL	NULL	NULL
MAFK	hgnc:6782	MAFK	PharmGKB	4/5/24	NULL	3.750547945406749	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	NULL	TAXANE COMPOUND	NULL	NULL	NULL	NULL	NULL
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	NULL	PCV REGIMEN	NULL	NULL	NULL	NULL	NULL
RRM1	hgnc:10451	RRM1	CIViC	10-Apr-24	NULL	0.3860858179095183	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	NULL	TAXANE COMPOUND	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	NULL	RADIATION THERAPY	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.006439499	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	DoCM	10-Apr-24	NULL	NULL	PRECLINICAL	NULL	NULL	NULL	NULL	NULL
RIPOR2	hgnc:13872	RIPOR2	PharmGKB	4/5/24	NULL	5.625821918110125	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
IL7R	hgnc:6024	IL7R	DoCM	10-Apr-24	NULL	NULL	RUXOLITINIB (IN SH2B3 DELETED)	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	NULL	PRECLINICAL	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	DoCM	10-Apr-24	NULL	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	DoCM	10-Apr-24	NULL	0.029244039	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
FGFR2	hgnc:3689	FGFR2	DoCM	10-Apr-24	NULL	NULL	PRECLINICAL	NULL	NULL	NULL	NULL	NULL
BACH1	hgnc:1282	GRIK1-AS2	PharmGKB	4/5/24	NULL	1.250182648468916	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	JAX-CKB	10-Apr-24	NULL	1.322135606654178	Asciminib	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	JAX-CKB	10-Apr-24	NULL	0.1766118064547324	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	JAX-CKB	10-Apr-24	NULL	0.1108075556053025	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	JAX-CKB	10-Apr-24	NULL	0.637458239	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	TASIN-1	NULL	NULL	NULL	NULL	NULL
CADM2	hgnc:29849	CADM2	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	XAV939	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.045658845	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.030996264	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	FH535	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	StAx-35	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	RAF709	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	C6-ceramide nanoliposome	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.016171134	Vinblastine	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	unspecified IGF-1R antibody	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	NULL	CHZ868	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.06109095	AZD6482	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.008854582	trifluoperazine	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1099637093941246	NVP-AEW541	iuphar.ligand:8067	NVP-AEW541	FALSE	FALSE	TRUE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.2885036881082115	Tofacitinib	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	BC21	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	PMED-1	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.095122593	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.3182283105193606	Triciribine	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
IAPP	hgnc:5329	IAPP	PharmGKB	4/5/24	NULL	7.501095890813499	rocuronium	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.1141471113819445	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	NULL	FIIN-1	NULL	NULL	NULL	NULL	NULL
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.029443554	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.2944355396394084	Lucitanib	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.3174882446809434	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.05387244	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	FIIN-2	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.048768735	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.1201548540862574	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	XAV939	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	PKF118-310	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.1581556362520918	Derazantinib	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.6563458904461812	RO6839921	ncit:C114980	MDM2 ANTAGONIST RO6839921	FALSE	FALSE	FALSE
PRORP	hgnc:19958	PRORP	PharmGKB	4/5/24	NULL	11.66837138570989	zileuton	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.054355767	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1296485709523321	hydroxyzine	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.053038052	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.760980743	caspofungin	rxcui:140108	CASPOFUNGIN	TRUE	FALSE	FALSE
IL6R	hgnc:6019	IL6R	PharmGKB	4/5/24	NULL	5.385402178019948	satralizumab	rxcui:2391541	SATRALIZUMAB	TRUE	FALSE	FALSE
KIRREL2	hgnc:18816	KIRREL2	PharmGKB	4/5/24	NULL	9.546849315580818	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.052507671	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MSH3	hgnc:7326	MSH3	JAX-CKB	10-Apr-24	NULL	NULL	Radiotherapy	NULL	NULL	NULL	NULL	NULL
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.6563458904461813	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	RAF709	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.033875917	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	IK-595	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.063517344	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1270346884734544	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	Rigosertib Sodium	ncit:C71355	RIGOSERTIB SODIUM	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2083637747448194	Capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.040515178	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified CTLA4 antibody	NULL	NULL	NULL	NULL	NULL
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	NULL	unspecified CTLA4 antibody	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.044347695	Panulisib	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.157680694	AZD6482	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1565212775308858	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.228073862	Capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	AR-mTOR-26	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	YU238259	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	GDC-0152	drugbank:DB12380	GDC-0152	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.044347695	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1419126249613365	NVP-AEW541	iuphar.ligand:8067	NVP-AEW541	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.048379304	Copanlisib	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1182605208011137	U0126	iuphar.ligand:5282	U0126	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.009336357	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	ONC201	iuphar.ligand:9978	ONC201	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.7095631248066824	GSK2256098	drugbank:DB16106	GSK2256098	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	unspecified IGF-1R antibody	NULL	NULL	NULL	NULL	NULL
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.1065064325267637	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	3.621218705909965	LY3295668	drugbank:DB18019	LY3295668	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	1.944728564284981	PRT1419	ncit:C176964	MYELOID CELL LEUKEMIA 1 INHIBITOR PRT1419	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.1383601350084176	estrone	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.921187215	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
IL6R	hgnc:6019	IL6R	ChEMBL	33	inhibitor	12.11715490054488	SARILUMAB	rxcui:1923319	SARILUMAB	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.012794267	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.052090944	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	ALFATRADIOL	rxcui:1926478	ALFATRADIOL	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.054020238	SERM	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.8401227397711121	DNA VACCINE	ncit:C39619	DNA VACCINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.039353698	tamsulosin	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NKAIN3	hgnc:26829	NKAIN3	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.5770073762164232	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
UMPS	hgnc:12563	UMPS	PharmGKB	4/5/24	NULL	3.281729452230906	tegafur	rxcui:10995	URACIL	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.020029629	palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
ACY3	hgnc:24104	ACY3	PharmGKB	4/5/24	NULL	19.69037671338543	bisoprolol	rxcui:19484	BISOPROLOL	TRUE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	14.58546423213736	Epratuzumab	ncit:C1887	EPRATUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:9308	iuphar.ligand:9308	SELTOREXANT	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	ChEMBL	33	inhibitor	6.563458904461812	AZD-4877	drugbank:DB11671	AZD-4877	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	ChEMBL	33	binder	1.071585127259071	ZILTIVEKIMAB	ncit:C171844	ZILTIVEKIMAB	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.006990459	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	CICLESONIDE	rxcui:274964	CICLESONIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	METHIOTHEPIN MESYLATE	chembl:CHEMBL1256737	METHIOTHEPIN MESYLATE	FALSE	FALSE	FALSE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.072125922	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.050294704	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
MTRR	hgnc:7473	MTRR	PharmGKB	4/5/24	NULL	0.8751278539282416	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
TRIM5	hgnc:16276	TRIM5	PharmGKB	4/5/24	NULL	0.4861821410712453	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.138178082	IUPHAR.LIGAND:335	iuphar.ligand:335	G&OUML; 7874	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	1.640864726115453	CDKI-73	ncit:C189967	ASNUCICLIB	FALSE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.046303061	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	1.040600372117402	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1591141552596802	APAZONE	rxcui:1029	APAZONE	TRUE	FALSE	FALSE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.095036509	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.005469549	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003528741	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	DTC	9/2/20	NULL	7.001022831425932	CYTOSPORONE B	iuphar.ligand:5424	CYTOSPORONE B	FALSE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.172722603	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
UNIPROT:P41180	hgnc:1514	CASR	TEND	1-Aug-11	NULL	3.281729452230906	CINACALCET	rxcui:407990	CINACALCET	TRUE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	PharmGKB	4/5/24	NULL	0.09972967	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
UNIPROT:Q14432	hgnc:8778	PDE3A	TEND	1-Aug-11	NULL	0.7955707762984013	MILRINONE	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	0.4487835148349958	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:946	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:1764	iuphar.ligand:1764	2MESAMP	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.082754407	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	CIViC	10-Apr-24	NULL	0.1682938180631234	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.018106094	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011738804	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.079197091	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.096167896	AM-101	chembl:CHEMBL2364609	ESKETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.9814517987980279	Debio 1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:12486	iuphar.ligand:12486	[3H]IPEROXO	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:26	iuphar.ligand:26	S-15535	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1534	iuphar.ligand:1534	C2-NPY (PIG)	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:2930	iuphar.ligand:2930	VPC44116	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	ChEMBL	33	inhibitor	0.6563458904461812	TACRINE HYDROCHLORIDE	rxcui:235972	TACRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.055563673	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	TCMDC-125814	chembl:CHEMBL533082	CHEMBL:CHEMBL533082	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.049817525	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.099446347	PHENOXYBENZAMINE	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.095399112	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.5834185692854944	OBP-801	drugbank:DB12279	OBP-801	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.9723642821424906	Tisagenlecleucel	rxcui:1986438	TISAGENLECLEUCEL	TRUE	FALSE	TRUE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.1244257612220248	IUPHAR.LIGAND:9578	iuphar.ligand:9578	SR8185	FALSE	FALSE	FALSE
P2RX7	hgnc:8537	P2RX7	ChEMBL	33	inhibitor	17.50255707856483	AZD9056	iuphar.ligand:7826	AZD9056	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TCMDC-123851	chembl:CHEMBL548458	CHEMBL:CHEMBL548458	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	GR-103545	iuphar.ligand:1649	GR 89696	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	KHELLIN	rxcui:6147	KHELLIN	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.035430277	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
NT5C2	hgnc:8022	NT5C2	PharmGKB	4/5/24	NULL	0.2160809515872201	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.1172046232939609	IUPHAR.LIGAND:5686	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:12721	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:7632	iuphar.ligand:7632	VU0119498	FALSE	FALSE	FALSE
GDF15	hgnc:30142	GDF15	NCI	14-Sep-17	NULL	0.2542744369767288	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.070956312	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.5609793935437446	Tariquidar	ncit:C2246	TARIQUIDAR	FALSE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TEND	1-Aug-11	NULL	0.4327555321623173	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
ITGA4	hgnc:6140	ITGA4	ChEMBL	33	inhibitor	5.834185692854944	UCB-1184197	chembl:CHEMBL4297363	UCB-1184197	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.1565057264849314	ABACAVIR	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1902451856365742	2,3,4,6-TETRACHLORO-PHENOL	chembl:CHEMBL320361	CHEMBL:CHEMBL320361	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.024932417	oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
KIAA2026	hgnc:23378	BRD10	PharmGKB	4/5/24	NULL	0.6482428547616604	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	1.117184494376478	MODUFOLIN	ncit:C157079	ARFOLITIXORIN	TRUE	FALSE	FALSE
UNIPROT:P47712	hgnc:9035	PLA2G4A	TEND	1-Aug-11	NULL	1.093909817410302	FLUOROMETHOLONE	rxcui:4491	FLUOROMETHOLONE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.4565884455277782	PLB1003	chembl:CHEMBL4650298	PLB1003	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.070574827	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	PharmGKB	4/5/24	NULL	0.5173169579871378	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
NCBIGENE:2135	hgnc:3516	EXTL2	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8937	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
NCBIGENE:947	hgnc:1662	CD34	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9484	iuphar.ligand:9484	YM-244769	FALSE	FALSE	FALSE
MART-1 MELANOMA ANTIGEN	hgnc:7124	MLANA	TTD	2020.06.01	NULL	2.917092846427472	MKC-1106-MT	ncit:C77971	IMMUNOTHERAPY REGIMEN MKC-1106-MT	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.076840494	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:481	iuphar.ligand:481	NS-49	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9330	iuphar.ligand:9330	CDP840	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.1835932560688619	sildenafil	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
PECAM1	hgnc:8823	PECAM1	NCI	14-Sep-17	NULL	2.143170254518142	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
RRP1B	hgnc:23818	RRP1B	PharmGKB	4/5/24	NULL	2.917092846427472	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	ChEMBL	33	inhibitor	0.085239726	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.4646696569530486	IUPHAR.LIGAND:1637	iuphar.ligand:1637	TIPP&PSI;	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	ChEMBL	33	negative modulator	1.458546423213736	ERLIZUMAB	ncit:C169959	ERLIZUMAB	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.6731752722524935	R101933	ncit:C28698	LANIQUIDAR	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.3697723326457359	Enadoline	ncit:C80576	ENADOLINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.01207443	fluphenazine	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:11096	iuphar.ligand:11096	MAPK13-IN-1	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2646556009863634	Pimasertib	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
SNAP25	hgnc:11132	SNAP25	ChEMBL	33	inhibitor	17.50255707856483	DAXIBOTULINUMTOXINA	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.030945115	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.1458546423213736	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	0.8078103267029924	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	1.346350544504987	IL-9	iuphar.ligand:5000	IL-9	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.062065805	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.3409589041278864	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	1.419126249613364	SONEDENOSON	ncit:C84176	SONEDENOSON	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	Anti-BCMA CAR T cells	ncit:C176023	ANTI-BCMA CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
NCBIGENE:1519	hgnc:2542	CTSO	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8005	iuphar.ligand:8005	OSU-03012	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:20	iuphar.ligand:151	[3H]LY334370	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.046303061	Tofacitinib	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
CA9	hgnc:1383	CA9	ChEMBL	33	binder	3.750547945	IODINE I 124 GIRENTUXIMAB	chembl:CHEMBL2108713	IODINE I 124 GIRENTUXIMAB	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.3500511415712966	GNF-PF-2347	chembl:CHEMBL579045	CHEMBL:CHEMBL579045	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	SB-228357	iuphar.ligand:192	SB 228357	FALSE	FALSE	FALSE
SLC25A31	hgnc:25319	SLC25A31	PharmGKB	4/5/24	NULL	0.9723642821424908	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
RPS14	hgnc:10387	RPS14	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	ChEMBL	33	inhibitor	0.3125456621172291	NIROGACESTAT	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
H19	hgnc:4713	H19	NCI	14-Sep-17	NULL	2.386712328895204	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
CHRNA6	hgnc:15963	CHRNA6	PharmGKB	4/5/24	NULL	0.7955707762984016	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
TNFRSF10A	hgnc:11904	TNFRSF10A	NCI	14-Sep-17	NULL	1.400204566285186	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.111481255	Seocalcitol	ncit:C26669	SEOCALCITOL	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.046549354	CAMBINOL	drugbank:DB15493	CAMBINOL	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.5834185692854945	MMF	rxcui:1546433	MONOMETHYL FUMARATE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.045898314	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	0.7001022831425934	Analgesics	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
SCNN1B	hgnc:10600	SCNN1B	PharmGKB	4/5/24	NULL	2.187819634820604	aldosterone	rxcui:1312358	ALDOSTERONE	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.2386712328895204	CT-1578	chembl:CHEMBL2035185	CT-1578	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	0.300043836	GUSACITINIB	ncit:C166736	GUSACITINIB	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018704642	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004762601	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.007043283	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	1.322135606654178	ABL 001	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.040515178	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.3860858179095183	TACRINE HYDROCHLORIDE	rxcui:235972	TACRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	modulator	4.375639269641208	BASIMGLURANT	ncit:C166619	BASIMGLURANT	FALSE	FALSE	FALSE
MYL2	hgnc:7583	MYL2	ChEMBL	33	activator	2.500365296937833	DANICAMTIV	ncit:C167013	DANICAMTIV	FALSE	FALSE	FALSE
CHRNA5	hgnc:1959	CHRNA5	PharmGKB	4/5/24	NULL	0.7955707762984016	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.2651902587661338	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.014749346	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.008821853	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1944728564284981	2,4-DIHYDROXYBENZOPHENONE	chembl:CHEMBL1392	2,4-DIHYDROXYBENZOPHENONE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	NSC-108783	chembl:CHEMBL1489812	CHEMBL:CHEMBL1489812	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.025942525	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.006324701	Metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.4751825451194073	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.088248187	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
UNIPROT:P04629	hgnc:8031	NTRK1	TEND	1-Aug-11	NULL	0.019180884	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	4.145342465975881	Chlormezanone	rxcui:2373	CHLORMEZANONE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	METIPRANOLOL HYDROCHLORIDE	rxcui:314731	METIPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	(E)-DIBENZYLIDENEACETONE	chembl:CHEMBL17201	CHEMBL:CHEMBL17201	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	NSC-93401	chembl:CHEMBL452954	CHEMBL:CHEMBL452954	FALSE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.5385402178019949	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	ETHYLENEDIAMINE	rxcui:4158	ETHYLENEDIAMINE	TRUE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.05853698	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CEACAM7	hgnc:1819	CEACAM7	NCI	14-Sep-17	NULL	2.692701089009974	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
NCBIGENE:2340	hgnc:2097	CMA1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9794	iuphar.ligand:9794	COMPOUND 7F [PMID: 29191554]	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.1422972120208523	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.084281976	IUPHAR.LIGAND:9907	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1527	iuphar.ligand:1527	[LEU31,PRO34]PYY (HUMAN)	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	1.693795846312725	METHDILAZINE	rxcui:29648	METHDILAZINE	TRUE	FALSE	FALSE
CA4	hgnc:1375	CA4	ChEMBL	33	inhibitor	0.3977853881492008	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GLCCI1	hgnc:18713	GLCCI1	PharmGKB	4/5/24	NULL	1.105424657593568	fluticasone propionate	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:8600	iuphar.ligand:8600	ALEXA-488-TELENZEPINE	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	ChEMBL	33	agonist	1.544343271638073	COBITOLIMOD	ncit:C166632	COBITOLIMOD	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.1860654544142257	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
PPAT	hgnc:9238	PPAT	ChEMBL	33	inhibitor	0.921187215	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.07458476	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.1712206670729168	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.002241666	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	ALPHA-NAPHTHOFLAVONE	drugbank:DB07453	ALPHA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.1535312024435511	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004195244	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	19.69037671338543	sipoglitazar	ncit:C87622	SIPOGLITAZAR	FALSE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	4.375639269641208	Dersalazine	ncit:C77949	DERSALAZINE	FALSE	FALSE	FALSE
CBR3	hgnc:1549	CBR3	PharmGKB	4/5/24	NULL	0.2592971419046642	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CRH	hgnc:2355	CRH	NCI	14-Sep-17	NULL	0.375054795	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	CancerCommons	25-Jul-13	inhibitor	0.4735540335109532	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	2-BFI	chembl:CHEMBL404505	CHEMBL:CHEMBL404505	FALSE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:9229	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.018305561	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.03409589	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.5834185692854944	4-hydroxycyclophosphamide	rxcui:2675983	4-HYDROXYCYCLOPHOSPHAMIDE	TRUE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.175610941	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
KCND3	hgnc:6239	KCND3	ChEMBL	33	blocker	0.1600843635234588	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	SALICYLANILIDE	ncit:C84142	SALICYLANILIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007232462	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.00770359	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	2.100306849	Elbasvir	rxcui:1734628	ELBASVIR	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.2785552850699974	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.1816874437221263	Atropine	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.2641230947469542	BAY-57-9352	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.2845944240417046	CHR-3996	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.08178765	BAZEDOXIFENE ACETATE	rxcui:1442171	BAZEDOXIFENE ACETATE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	0.358239472	amphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
ARGINASE	hgnc:77	ABL2	TTD	2020.06.01	NULL	1.009762908	BCT-100	ncit:C88286	PEGYLATED RECOMBINANT HUMAN ARGINASE I BCT-100	FALSE	FALSE	FALSE
P-SELECTIN	hgnc:10721	SELP	TTD	2020.06.01	NULL	8.751278539282417	GMI-1070	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	1.029066006546944	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.019318496	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.011766425	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CAPG	hgnc:1474	CAPG	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.9907107780319716	Depudecin	ncit:C1361	DEPUDECIN	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.2500365296937833	DIETHYLDITHIOCARBAMATE	rxcui:1427193	DIETHYLDITHIOCARBAMATE	FALSE	FALSE	FALSE
GCKR	hgnc:4196	GCKR	PharmGKB	4/5/24	NULL	0.4167275494896389	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.025439763	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1848861663228679	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.079557078	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:501	rxcui:5784	INDORAMIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	NSC-663284	drugbank:DB17038	NSC-663284	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00410569	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.005111728	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.1691068316769549	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	1.230648544586589	XL418	drugbank:DB05204	XL418	FALSE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	GTX-758	drugbank:DB14969	GTX-758	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.073540156	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8397	iuphar.ligand:8397	I-BRD9	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:12620	iuphar.ligand:12620	CIRTUVIVINT	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	5.834185692854944	AFQ056	ncit:C170154	MAVOGLURANT	FALSE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	0.2681242786503549	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
RPL18	hgnc:10310	RPL18	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.1539814405738841	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:402	hgnc:693	ARL2	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
UNIPROT:P05231	hgnc:6018	IL6	TdgClinicalTrial	Jan-14	NULL	4.286340509036285	ALD518	ncit:C82359	CLAZAKIZUMAB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.017295017	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:8947	iuphar.ligand:8947	JNJ-46281222	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.4817217544559128	KMN-21	chembl:CHEMBL570176	CHEMBL:CHEMBL570176	FALSE	FALSE	FALSE
UNIPROT:P08473	hgnc:7154	MME	TEND	1-Aug-11	NULL	4.773424657790408	CANDOXATRIL	ncit:C171870	CANDOXATRIL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DEXAMETHASONE VALARATE	chembl:CHEMBL1378167	DEXAMETHASONE VALARATE	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.6351734423672721	LEVOCETIRIZINE DIHYDROCHLORIDE	rxcui:356887	LEVOCETIRIZINE	TRUE	FALSE	FALSE
PSMA1	hgnc:9530	PSMA1	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
UNIPROT:P00797	hgnc:9958	REN	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	ALISKIREN	rxcui:325646	ALISKIREN	TRUE	FALSE	FALSE
ANKRD30B	hgnc:24165	ANKRD30B	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.086361301	IUPHAR.LIGAND:10458	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:9190	iuphar.ligand:9190	COMPOUND 3 [PMID: 23134120]	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	DTC	9/2/20	NULL	0.03849536	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.037884323	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	RONOMILAST	ncit:C97274	RONOMILAST	FALSE	FALSE	FALSE
UNIPROT:P04275	hgnc:12726	VWF	TdgClinicalTrial	Jan-14	NULL	8.290684931951763	ALX-0081	rxcui:2110604	CAPLACIZUMAB-YHDP	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	4'-HYDROXYPHENYL-BENZO[D]THIAZOLE	chembl:CHEMBL47875	CHEMBL:CHEMBL47875	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	MMV665817	chembl:CHEMBL590919	CHEMBL:CHEMBL590919	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	TABIMORELIN	ncit:C76887	TABIMORELIN	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.037134138	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.004118249	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
XRCC5	hgnc:12833	XRCC5	NCI	14-Sep-17	NULL	0.7501095890813501	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.055155117	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.1389091831632129	theophylline	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	agonist	0.1325951293830669	IUPHAR.LIGAND:4004	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN SUSP PROTAMINE ZINC PURIFIED PORK	chembl:CHEMBL1201638	INSULIN SUSP PROTAMINE ZINC PURIFIED PORK	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	XLCART001	ncit:C165551	ANTI-CD19 CAR T-CELLS XLCART001	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	SPICLOMAZINE	ncit:C66557	SPICLOMAZINE	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	3.000438356	Fostamatinib	rxcui:2044896	FOSTAMATINIB	TRUE	FALSE	TRUE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1187956362798518	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	6.563458904461812	INTERFERON ALFACON-1	rxcui:59744	INTERFERON ALFACON-1	TRUE	TRUE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.025489161	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	1.184383561707394	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenome	20-Jun-17	antibody	1.372749574789398	U3-1287	ncit:C78853	PATRITUMAB	FALSE	TRUE	TRUE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	0.9211872146613068	ABBV-744	iuphar.ligand:10730	ABBV-744	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.052648066	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.5303805175322677	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	1.521961485092594	ALVESPIMYCIN	ncit:C38142	ALVESPIMYCIN	FALSE	FALSE	TRUE
NCBIGENE:403	hgnc:694	ARL3	GuideToPharmacology	2024.1	blocker	1.250182648468916	IUPHAR.LIGAND:2357	rxcui:1649480	IVABRADINE	TRUE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:668	iuphar.ligand:668	FR190997	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.6049270879688307	Tofacitinib	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
TRANSFORMING GROWTH FACTOR BETA	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	0.2966535098061835	TEW-7197	ncit:C116357	VACTOSERTIB	FALSE	FALSE	FALSE
UNIPROT:P43116	hgnc:9594	PTGER2	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	ChEMBL	33	inhibitor	0.1187956362798518	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.084383562	Fluticasone	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	1.491695205559502	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.056500364	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
RPL36A	hgnc:10359	RPL36A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.01274458	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	MyCancerGenome	20-Jun-17	inhibitor	0.2991890098899972	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.032837818	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	AMEDIPLASE	ncit:C169777	AMEDIPLASE	FALSE	FALSE	FALSE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.1988926940746004	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.03729238	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	1.693795846312725	INCB-047986	chembl:CHEMBL3545225	INCB-047986	FALSE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.100976291	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	AMD-070	ncit:C126660	MAVORIXAFOR	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.100976291	OLANZAPINE PAMOATE	rxcui:1294588	OLANZAPINE PAMOATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	DIPYRITHIONE	rxcui:1362743	DIPYRITHIONE	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	1.944728564284981	GNF-PF-2133	chembl:CHEMBL578883	CHEMBL:CHEMBL578883	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-4674	chembl:CHEMBL584452	CHEMBL:CHEMBL584452	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.1693795846312726	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.2838252499226729	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
KLRD1	hgnc:6378	KLRD1	PharmGKB	4/5/24	NULL	0.1875273972703374	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.031929262	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
LRP1	hgnc:6692	LRP1	PharmGKB	4/5/24	NULL	1.060761035064535	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.3777530304726222	BAFETINIB	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	EP217609	drugbank:DB18393	EP-217609	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.2016939996249468	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:P45983	hgnc:6881	MAPK8	TdgClinicalTrial	Jan-14	NULL	0.5147810905460245	AM-111	iuphar.ligand:9101	BRIMAPITIDE	FALSE	FALSE	FALSE
SEMAPHORIN-4D	hgnc:10732	SEMA4D	TTD	2020.06.01	NULL	8.751278539282415	VX-15	chembl:CHEMBL4297884	PEPINEMAB	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.9546849315580818	CARPROFEN	rxcui:20343	CARPROFEN	TRUE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
DNTT	hgnc:2983	DNTT	NCI	14-Sep-17	NULL	0.3860858179095184	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.3580068493342807	SUPROFEN	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.093931433	IUPHAR.LIGAND:7434	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	1.458546423213736	HEPARIN CALCIUM	rxcui:20044	HEPARIN CALCIUM	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.018436682	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TdgClinicalTrial	Jan-14	NULL	1.406455479527531	MISOPROSTOL	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
FOLLICLE-STIMULATING HORMONE RECEPTOR	hgnc:3969	FSHR	TTD	2020.06.01	NULL	0.2763561643983921	Suramin	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	ALB-109564(a)	ncit:C78842	TUBULIN INHIBITOR ALB 109564 DIHYDROCHLORIDE	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	inhibitor	0.5834185692854944	IBIPINABANT	ncit:C174784	IBIPINABANT	FALSE	FALSE	FALSE
UNIPROT:Q15118	hgnc:8809	PDK1	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	AR-12	iuphar.ligand:8005	OSU-03012	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:3900	iuphar.ligand:3900	M871	FALSE	FALSE	FALSE
NCBIGENE:746	hgnc:1164	TMEM258	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	TORSEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.010966514	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:11747	iuphar.ligand:11747	BPR1R024	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.9546849315580818	APRICOXIB	ncit:C74021	APRICOXIB	FALSE	FALSE	FALSE
NCBIGENE:2896	hgnc:4601	GRN	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:9124	iuphar.ligand:9124	ANTI-ILT7 ANTIBODY	FALSE	FALSE	FALSE
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	ARRY-797	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.1319288222002374	PROPAZINE	chembl:CHEMBL1333189	PROPAZINE	FALSE	FALSE	FALSE
GAL	hgnc:4114	GAL	PharmGKB	4/5/24	NULL	0.6563458904461813	mirtazapine	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4078	iuphar.ligand:4078	[3H]CGP39653	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:5977	iuphar.ligand:5977	GSK-3BETA INHIBITOR I	FALSE	FALSE	FALSE
KCNH1	hgnc:6250	KCNH1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.023016221	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.041972559	ARRY-614	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	2-AMINOANTHRACENE	chembl:CHEMBL83154	2-AMINOANTHRACENE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CID 893238	chembl:CHEMBL473735	CHEMBL:CHEMBL473735	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.019404165	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	2.838252499226729	MULTIVITAMINS	ncit:C1654	MULTIVITAMIN	FALSE	FALSE	FALSE
ACTIVATION B7-1 ANTIGEN	hgnc:1700	CD80	TTD	2020.06.01	NULL	13.12691780892362	Galiximab	ncit:C26447	GALIXIMAB	FALSE	FALSE	FALSE
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	ARRY-797	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	0.6563458904461812	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.05309168	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
NCBIGENE:1998	hgnc:3317	ELF2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8050	iuphar.ligand:8050	PF-4800567	FALSE	FALSE	FALSE
NCBIGENE:94	hgnc:175	ACVRL1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:2910	drugbank:DB07780	FARNESYL DIPHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.108040476	ARRY-614	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
UNIPROT:Q06609	hgnc:9817	RAD51	TdgClinicalTrial	Jan-14	NULL	15.00219178162699	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.061055432	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P15941	hgnc:7508	MUC1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	AS1402	ncit:C38697	SONTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1605	hgnc:2666	DAG1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6538	iuphar.ligand:6538	UAMC00039	FALSE	FALSE	FALSE
SLC14A2	hgnc:10919	SLC14A2	PharmGKB	4/5/24	NULL	2.250328767	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2035181055647073	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
ADK	hgnc:257	ADK	PharmGKB	4/5/24	NULL	0.2763561643983921	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	TCMDC-125321	chembl:CHEMBL587449	CHEMBL:CHEMBL587449	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	ATRASENTAN	ncit:C61606	ATRASENTAN	FALSE	FALSE	FALSE
UNIPROT:P03952	hgnc:6371	KLKB1	TdgClinicalTrial	Jan-14	NULL	0.8334550989792778	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.8607814956671229	BECAPLERMIN	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344583	INTERFERON ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.1377250393067396	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
T-CELL ACTIVATION ANTIGEN CD27	hgnc:11922	CD27	TTD	2020.06.01	NULL	15.00219178	CDX-1127	ncit:C99127	VARLILUMAB	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:8334	iuphar.ligand:8334	MINIMISED INSL5 ANALOGUE 7	FALSE	FALSE	FALSE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	3.889457128569962	QUINAPRIL	rxcui:35208	QUINAPRIL	TRUE	FALSE	FALSE
UNIPROT:P05141	hgnc:10991	SLC25A5	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	CLODRONATE	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	0.251232877	IUPHAR.LIGAND:1054	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007330402	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	BROMPHENIRAMINE MALEATE	rxcui:142427	BROMPHENIRAMINE MALEATE	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.1480131676834235	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1666910197958555	GNF-PF-4464	chembl:CHEMBL600692	CHEMBL:CHEMBL600692	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.029498692	IUPHAR.LIGAND:9190	iuphar.ligand:9190	COMPOUND 3 [PMID: 23134120]	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.081365193	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.2453629496995069	BENZPHETAMINE HYDROCHLORIDE	rxcui:142425	BENZPHETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	blocker	0.096167896	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH3	hgnc:6252	KCNH3	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.055504938	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
KCNH6	hgnc:18862	KCNH6	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
RPL9P9	hgnc:30334	RPL9P8	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:7155	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.083257407	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1717	iuphar.ligand:1717	A2P5P	FALSE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7339	iuphar.ligand:7339	CHF-5074	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.1154014752432846	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.4234489615781814	misoprostol	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.112919723	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.008790837	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TdgClinicalTrial	Jan-14	NULL	21.00306849427779	CORIFOLLITROPIN ALFA	ncit:C169865	CORIFOLLITROPIN ALFA	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.029918901	quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Estrogen	chembl:CHEMBL592868	ESTROGEN	TRUE	FALSE	FALSE
NCBIGENE:2766	hgnc:4376	GMPR	GuideToPharmacology	2024.1	antibody	0.2917092846427472	IUPHAR.LIGAND:7395	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:7956	ncit:C82363	GOLVATINIB	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.023524942	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.064624826	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004252322	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	EPIRUBICIN HYDROCHLORIDE	rxcui:203213	EPIRUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P49354	hgnc:3782	FNTA	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	CP-609,754	ncit:C2551	CP-609,754	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.078840347	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.022439176	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006940869	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:12722	iuphar.ligand:12722	HU7691	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.3017682254924971	NSC-91340	chembl:CHEMBL1376091	CHEMBL:CHEMBL1376091	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.7395446652914718	CT-322	ncit:C62791	PEGDINETANIB	FALSE	FALSE	TRUE
RPS26	hgnc:10414	RPS26	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.1123399042269886	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW810372X	chembl:CHEMBL365248	GW810372X	FALSE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.3977853881492006	DESONIDE	rxcui:3254	DESONIDE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.079376676	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1600843635234588	IUPHAR.LIGAND:487	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
NCBIGENE:1998	hgnc:3317	ELF2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9371	iuphar.ligand:9371	PF-670462	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:10652	ncit:C170277	OXYCODEGOL	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:9010	iuphar.ligand:9010	COMPOUND NRA 4 [PMID: 25262941]	FALSE	FALSE	FALSE
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.2273059360852575	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
ANKK1	hgnc:21027	ANKK1	PharmGKB	4/5/24	NULL	1.184383561707394	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.015447976	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	PharmGKB	4/5/24	NULL	0.228073862	capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	TEROXIRONE	ncit:C2320	TEROXIRONE	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.1491695205559502	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.038256955	pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
SLC22A6	hgnc:10970	SLC22A6	ChEMBL	33	inhibitor	0.5966780822238011	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.1829535583125243	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.051027863	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613069	IUPHAR.LIGAND:3247	iuphar.ligand:3233	SB269970	FALSE	FALSE	FALSE
NCBIGENE:402	hgnc:693	ARL2	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:2357	rxcui:1649480	IVABRADINE	TRUE	FALSE	FALSE
B-CELL-ACTIVATING FACTOR	hgnc:11929	TNFSF13B	TTD	2020.06.01	NULL	19.69037671338543	Blisibimod	ncit:C166445	BLISIBIMOD	FALSE	FALSE	FALSE
BCL2L11	hgnc:994	BCL2L11	PharmGKB	4/5/24	NULL	0.305277158	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.1084869240406911	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	2,7-BIS[2-(DIMETHYLAMINO)ACETAMIDO]ANTHRAQUINONE	chembl:CHEMBL494283	CHEMBL:CHEMBL494283	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	4.200613699	PROTEIN KINASE A INHIBITOR	ncit:C2148	PROTEIN KINASE A INHIBITOR	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.039214094	QUININE	rxcui:9071	QUININE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.4257378748840094	FESOTERODINE	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
NCBIGENE:2601	hgnc:4153	GAPDHP60	GuideToPharmacology	2024.1	antibody	1.750255707856483	IUPHAR.LIGAND:6775	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
UNIPROT:Q9H6Z9	hgnc:14661	EGLN3	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	FG-2216	drugbank:DB08687	FG-2216	FALSE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	MyCancerGenome	20-Jun-17	other/unknown	0.5000730593875666	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.2917092846427472	pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
KCNC1	hgnc:6233	KCNC1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	0.2941606231691568	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1682938180631233	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
RPL23	hgnc:10316	RPL23	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.2051080907644316	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.035098711	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
NCBIGENE:2767	hgnc:4379	GNA11	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9753	iuphar.ligand:9753	PXS-4681A	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5926	iuphar.ligand:5926	ALSTERPAULLONE 2-CYANOETHYL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	TCMDC-124032	chembl:CHEMBL536375	CHEMBL:CHEMBL536375	FALSE	FALSE	FALSE
UNIPROT:Q00526	hgnc:1772	CDK3	TdgClinicalTrial	Jan-14	NULL	0.4375639269641209	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	GRISEOFULVIN	rxcui:5021	GRISEOFULVIN	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.013259513	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.08197919	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	PharmGKB	4/5/24	NULL	0.056826484	nirogacestat	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	PharmGKB	4/5/24	NULL	0.4953553890159858	flucytosine	rxcui:4451	FLUCYTOSINE	TRUE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.2678962818147679	FRUQUINTINIB	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	MyCancerGenome	20-Jun-17	inhibitor	0.3431873936973496	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001907844	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.07699072	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P11802	hgnc:1773	CDK4	TdgClinicalTrial	Jan-14	NULL	0.2083637747448194	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.2678962818147679	FRUQUINTINIB	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	0.1593072549626653	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TdgClinicalTrial	Jan-14	NULL	0.1403948428761885	MESALAZINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.1725334213659184	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	GARENOXACIN MESYLATE	ncit:C65801	GARENOXACIN MESYLATE	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.089501712	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
UNIPROT:P28908	hgnc:11923	TNFRSF8	TdgClinicalTrial	Jan-14	NULL	9.845188356692718	MDX-060	ncit:C26441	IRATUMUMAB	FALSE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.074797252	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.073643298	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	TOFIMILAST	ncit:C76891	TOFIMILAST	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.030688294	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001835419	ISOPRENALINE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
EIF4E	hgnc:3287	EIF4E	NCI	14-Sep-17	NULL	0.1392776425349987	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TdgClinicalTrial	Jan-14	NULL	0.1403948428761885	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.076934317	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.3680444245492605	ARZOXIFENE	ncit:C1805	ARZOXIFENE	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.019534104	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.012585731	sulfinpyrazone	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	MMV396705	chembl:CHEMBL1594640	CHEMBL:CHEMBL1594640	FALSE	FALSE	FALSE
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	MOD-4023	iuphar.ligand:12013	SOMATROGON	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.3804903712731485	ethambutol	rxcui:142435	ETHAMBUTOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	0.052181537	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	0.1376949420516464	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	NADIFLOXACIN	ncit:C166927	NADIFLOXACIN	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	ALKS 33	rxcui:2559612	SAMIDORPHAN	TRUE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:9188	iuphar.ligand:9188	PEPCAN-12	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:4023	iuphar.ligand:4023	A331440	FALSE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	MT-103	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
NCBIGENE:2174	hgnc:9408	PRKD3	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:9370	iuphar.ligand:9370	BPKDI	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.2864054794674245	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	SB-408124	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.3977853881492007	MURAGLITAZAR	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
TASTE RECEPTOR	hgnc:16713	SRSF10	TTD	2020.06.01	NULL	52.50767123569449	Cynarin	chembl:CHEMBL487258	CYNARIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	NEOSTIGMINE METHYLSULFATE	rxcui:7315	NEOSTIGMINE	TRUE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	1.093909817410302	PYRANTEL PAMOATE	rxcui:8985	PYRANTEL PAMOATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.018521224	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	1.050153425	MT110	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
SULT1C4	hgnc:11457	SULT1C4	PharmGKB	4/5/24	NULL	1.419126249613364	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.2357246744587856	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.4268916360625568	AT-101	ncit:C187300	ANTI-CD19 CAR T CELLS AT101	FALSE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.086361301	IUPHAR.LIGAND:8315	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.033701971	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
PNP	hgnc:7892	PNP	DTC	9/2/20	NULL	35.00511415712966	FORODESINE HYDROCHLORIDE	ncit:C26655	FORODESINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q8NER1	hgnc:12716	TRPV1	TdgClinicalTrial	Jan-14	NULL	2.561349816375341	NGD-8243	chembl:CHEMBL3545227	NGD-8243	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	DTC	9/2/20	NULL	3.750547945	PHENETHYL ISOCYANATE	chembl:CHEMBL2074871	PHENETHYL ISOCYANATE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.045461187	DIHYDROXANTHOHUMOL	chembl:CHEMBL510279	DIHYDROXANTHOHUMOL	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.011815408	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
HSPA1A	hgnc:5232	HSPA1A	PharmGKB	4/5/24	NULL	0.5357925636295356	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.096521454	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.066803653	PHENACYL CHLORIDE	iuphar.ligand:6285	OMEGA-CHLOROACETOPHENONE	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.033701971	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.032134438	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:P19838	hgnc:7794	NFKB1	TdgClinicalTrial	Jan-14	NULL	0.276356164	NF-KB DECOY	drugbank:DB05559	NF-KAPPAB DECOY	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.1902451856365742	CERDULATINIB	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
NCBIGENE:2016	hgnc:3340	EMX1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:1021	iuphar.ligand:1021	FMET-ILE-PHE-LEU	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:5904	iuphar.ligand:5904	PSB-0739	FALSE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.053633985	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.091796628	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.032252869	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.050978322	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-989	chembl:CHEMBL583150	CHEMBL:CHEMBL583150	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.086219493	IUPHAR.LIGAND:403	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:9551	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	SALAGEN	chembl:CHEMBL611494	SALAGEN	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.03070624	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
NPFFR1	hgnc:17425	NPFFR1	DTC	9/2/20	NULL	1.640864726115453	KISSPEPTIN-10	drugbank:DB16210	KISSPEPTIN-10	FALSE	FALSE	FALSE
KCNB1	hgnc:6231	KCNB1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
FCGRT	hgnc:3621	FCGRT	ChEMBL	33	inhibitor	5.834185692854944	BATOCLIMAB	ncit:C171826	BATOCLIMAB	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.6945459158160648	NIMOTUZUMAB	ncit:C2733	NIMOTUZUMAB	FALSE	TRUE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:2901	hgnc:4583	GRIK5	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11115	iuphar.ligand:11115	X-165	FALSE	FALSE	FALSE
UNIPROT:Q96RI1	hgnc:7967	NR1H4	TdgClinicalTrial	Jan-14	NULL	2.663432598912039	OBETICHOLIC ACID	rxcui:1798288	OBETICHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1999	hgnc:3318	ELF3	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:8163	iuphar.ligand:8163	COMPOUND 33 [PMID: 19364658]	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.010449288	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:876	hgnc:11006	SLC2A2	GuideToPharmacology	2024.1	NULL	4.375639269641208	IUPHAR.LIGAND:4643	iuphar.ligand:4643	[3H]2-DEOXYGLUCOSE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	METHANTHELINE	rxcui:6821	METHANTHELINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	PHYSOSTIGMINE	rxcui:8299	PHYSOSTIGMINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.205692444	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.000821138	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	OTELIXIZUMAB	ncit:C95790	OTELIXIZUMAB	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	2.000292237550266	LY2875358	ncit:C95732	EMIBETUZUMAB	FALSE	TRUE	TRUE
SLC28A3	hgnc:16484	SLC28A3	PharmGKB	4/5/24	NULL	0.1339481409073839	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.1223955040459079	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	PARECOXIB	rxcui:279950	PARECOXIB	TRUE	FALSE	FALSE
UNIPROT:P09211	hgnc:4638	GSTP1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	EZATIOSTAT	ncit:C83709	EZATIOSTAT	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:11226	iuphar.ligand:11226	NPS(1-4)NH2	FALSE	FALSE	FALSE
NCBIGENE:2841	hgnc:4472	GPR18	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8272	ncit:C65755	FORODESINE	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:2027	iuphar.ligand:2027	BIM 23627	FALSE	FALSE	FALSE
UNIPROT:P32745	hgnc:11332	SSTR3	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	PASIREOTIDE	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.030386384	SPERMINE	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
UNIPROT:P35346	hgnc:11334	SSTR5	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	PASIREOTIDE	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	3.281729452230906	Anti-CD30 CAR T cells	ncit:C201513	ANTI-CD30 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
UBE2I	hgnc:12485	UBE2I	PharmGKB	4/5/24	NULL	0.8334550989792777	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.1486416737033106	PARICALCITOL	rxcui:73710	PARICALCITOL	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	TCMDC-125625	chembl:CHEMBL549208	CHEMBL:CHEMBL549208	FALSE	FALSE	FALSE
UNIPROT:Q02156	hgnc:9401	PRKCE	TdgClinicalTrial	Jan-14	NULL	0.1640864726115453	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.055622533	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ChEMBL	33	inhibitor	4.375639269641208	OLOCROLIMUS	chembl:CHEMBL3545142	OLOCROLIMUS	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	ChEMBL	33	inhibitor	0.7721716358190367	XL-844	chembl:CHEMBL3544936	XL-844	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.16256245	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.072927321	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	EMETINE HYDROCHLORIDE	rxcui:82015	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.1725334213659184	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
INTERLEUKIN 13 RECEPTOR ALPHA-2	hgnc:5975	IL13RA2	TTD	2020.06.01	NULL	13.12691780892362	ABT-308	chembl:CHEMBL4297864	CENDAKIMAB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001835419	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.3088686543276147	PHYSOSTIGMINE	rxcui:8299	PHYSOSTIGMINE	TRUE	FALSE	FALSE
UNIPROT:Q07699	hgnc:10586	SCN1B	TdgClinicalTrial	Jan-14	NULL	2.100306849	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:P52732	hgnc:6388	KIF11	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	ISPINESIB	ncit:C38131	ISPINESIB	FALSE	FALSE	TRUE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.066297565	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	1.009762908	dolasetron	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ALFUZOSIN HYDROCHLORIDE	rxcui:46043	ALFUZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM1A	hgnc:29079	KDM1A	DTC	9/2/20	NULL	2.625383561784724	PARNATE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.070860555	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
UNIPROT:P01008	hgnc:775	SERPINC1	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	2-O, 3-O DESULFATED HEPARIN	drugbank:DB17569	2-O, 3-O DESULFATED HEPARIN	FALSE	FALSE	FALSE
MICROTUBULE-ASSOCIATED PROTEIN	hgnc:25228	SGSM3	TTD	2020.06.01	NULL	4.375639269641208	Demecolcine	ncit:C419	DEMECOLCINE	FALSE	FALSE	FALSE
KCNB2	hgnc:6232	KCNB2	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	inhibitor	3.281729452230906	SEMZUVOLIMAB	ncit:C188511	SEMZUVOLIMAB	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2381300282797936	PHENOXODIOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	ChEMBL	33	inhibitor	0.2692701089009974	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.2453629496995069	ESTETROL	rxcui:2539031	ESTETROL	TRUE	FALSE	FALSE
UNIPROT:P17252	hgnc:9393	PRKCA	TdgClinicalTrial	Jan-14	NULL	0.1367387271762877	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.2112984757975633	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.157680694	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:10490	iuphar.ligand:10490	SS-208	FALSE	FALSE	FALSE
NCBIGENE:630	hgnc:7981	NR4A2	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:12998	iuphar.ligand:12998	COMPOUND 108 [PMID: 37918435]	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.040390516	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.02321294	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.023080295	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.07699072	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.201952582	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.023630815	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SERPINB3	hgnc:10569	SERPINB3	NCI	14-Sep-17	NULL	15.00219178162699	GONADOTROPINS	ncit:C527	THERAPEUTIC GONADOTROPIN	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.029203377	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PSMD11	hgnc:9556	PSMD11	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.016764901	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.4773424657790409	EDICOTINIB	ncit:C101519	EDICOTINIB	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	1.381780822	RG-7602	chembl:CHEMBL3545007	RG-7602	FALSE	FALSE	FALSE
UNIPROT:Q9Y5Z0	hgnc:934	BACE2	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	POSIPHEN	drugbank:DB15317	POSIPHEN	FALSE	FALSE	FALSE
PSMD5	hgnc:9563	PSMD5	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:2833	hgnc:4540	CXCR3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8229	iuphar.ligand:8229	IOX2	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.3174882446809434	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.053145416	IUPHAR.LIGAND:7082	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TACR3	hgnc:11528	TACR3	ChEMBL	33	inhibitor	5.834185692854944	PAVINETANT	ncit:C166698	PAVINETANT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.04464938	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P01589	hgnc:6008	IL2RA	TdgClinicalTrial	Jan-14	NULL	0.1715936968486748	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	BERGAMOTTIN	chembl:CHEMBL1078442	BERGAMOTTIN	FALSE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TEND	1-Aug-11	NULL	1.312691780892362	ISOFLUROPHATE	rxcui:6027	ISOFLUROPHATE	TRUE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	1.193356164447602	Empagliflozin	rxcui:1545653	EMPAGLIFLOZIN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	BI-3406	iuphar.ligand:12061	BI-3406	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:4123	iuphar.ligand:4123	ACET	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.2885036881082116	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	modulator	1.875273972703375	IUPHAR.LIGAND:8343	iuphar.ligand:8343	135PAM1	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR	ncbigene:359995	mCR	TTD	2020.06.01	NULL	7.501095890813499	Bremelanotide	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1944728564284981	GALLIC ACID METHYL ESTER	chembl:CHEMBL65675	GALLIC ACID METHYL ESTER	FALSE	FALSE	FALSE
NAAA	hgnc:736	NAAA	DTC	9/2/20	NULL	21.00306849427779	CYCLOPENTYL PALMITATE	chembl:CHEMBL590884	CYCLOPENTYL PALMITATE	FALSE	FALSE	FALSE
UNIPROT:P15144	hgnc:500	ANPEP	TdgClinicalTrial	Jan-14	NULL	0.3860858179095183	PL37	iuphar.ligand:7896	PL37	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	(R)-FLECAINIDE	chembl:CHEMBL398673	(R)-FLECAINIDE	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.029833904	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	ChEMBL	33	inhibitor	0.074850565	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
CD28	hgnc:1653	CD28	ChEMBL	33	inhibitor	7.001022831425932	LULIZUMAB PEGOL	ncit:C175727	LULIZUMAB PEGOL	FALSE	FALSE	FALSE
RPL9P7	hgnc:30335	RPL9P7	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
UNIPROT:P28482	hgnc:6871	MAPK1	TdgClinicalTrial	Jan-14	NULL	0.011540148	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.099446347	BUDIODARONE	ncit:C83563	BUDIODARONE	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.087707691	CB-03-01	rxcui:2474340	CLASCOTERONE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.065226921	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:2746	hgnc:4335	GLUD1	GuideToPharmacology	2024.1	modulator	52.50767123569449	IUPHAR.LIGAND:8808	iuphar.ligand:8808	COMPOUND 13B [PMID: 19101153]	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005294179	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.094608417	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.192335792	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.4934931507114145	GW501516	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	NULL	0.1037701012563132	IUPHAR.LIGAND:5087	iuphar.ligand:5087	VEGFC	FALSE	FALSE	FALSE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	0.8334550989792778	Treprostinil	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	1.154014752432846	OTX-015	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.005397027	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.030518844	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P25025	hgnc:6027	CXCR2	TdgClinicalTrial	Jan-14	NULL	1.166837138570989	SCH-527123	iuphar.ligand:8497	NAVARIXIN	FALSE	FALSE	FALSE
PAH	hgnc:8582	PAH	ChEMBL	33	activator	8.751278539282415	SAPROPTERIN DIHYDROCHLORIDE	rxcui:753341	SAPROPTERIN DIHYDROCHLORIDE	TRUE	FALSE	FALSE
SCNN1A	hgnc:10599	SCNN1A	ChEMBL	33	blocker	2.625383561784724	AMILORIDE HYDROCHLORIDE	rxcui:142424	AMILORIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1389091831632129	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.1275696580070323	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:41	ncit:C169993	FLUPAROXAN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.014638325	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.2263261691193728	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.093763699	DNDI1417085	chembl:CHEMBL1522984	CHEMBL:CHEMBL1522984	FALSE	FALSE	FALSE
HLA-DRA	hgnc:4947	HLA-DRA	CIViC	10-Apr-24	NULL	0.2500365296937833	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.028850369	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.09055649	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.039939912	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.079557078	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:1704	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
UNIPROT:P24752	hgnc:93	ACAT1	TdgClinicalTrial	Jan-14	NULL	0.2083637747448194	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	NCI	14-Sep-17	NULL	0.6563458904461813	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.071585127259071	EP-217609	drugbank:DB18393	EP-217609	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.069240885	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	REL-CISAPRIDE	chembl:CHEMBL74656	REL-CISAPRIDE	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.019233579	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:341	iuphar.ligand:341	ALCURONIUM	FALSE	FALSE	FALSE
UNIPROT:P41180	hgnc:1514	CASR	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	STRONTIUM RANELATE	ncit:C93265	STRONTIUM RANELATE	FALSE	FALSE	FALSE
UNIPROT:Q99460	hgnc:9554	PSMD1	TEND	1-Aug-11	NULL	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.082754407	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	BETAINE HYDROCHLORIDE	rxcui:81965	BETAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.020936073	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	1.988926940746003	IUPHAR.LIGAND:1188	rxcui:301739	ABARELIX	TRUE	FALSE	TRUE
NCBIGENE:3180	hgnc:9479	LONP1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11505	iuphar.ligand:11505	COMPOUND 12D [PMID: 33821636]	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.039778539	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	Tunlametinib	ncit:C173437	TUNLAMETINIB	FALSE	FALSE	TRUE
GC	hgnc:4187	GC	PharmGKB	4/5/24	NULL	1.093909817410302	deferasirox	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.017502557	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	PharmGKB	4/5/24	NULL	0.1178623372293928	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:11853	iuphar.ligand:11853	COMPOUND 40 [PMID: 34982553]	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.012120884	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.059330702	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.9053046764774912	PLANT STEROL	ncit:C28178	PHYTOSTEROL	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	MSC-2364447	chembl:CHEMBL3545193	MSC-2364447	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	2.143170254518142	TAK-442	ncit:C96541	LETAXABAN	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	DTC	9/2/20	NULL	3.621218705909965	AMPKINONE	chembl:CHEMBL1271027	AMPKINONE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.03505185	DOMIPHEN BROMIDE	rxcui:49255	DOMIPHEN BROMIDE	FALSE	FALSE	FALSE
CDA	hgnc:1712	CDA	NCI	14-Sep-17	NULL	0.3704244884352345	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.09323095	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
DAO	hgnc:2671	DAO	DTC	9/2/20	NULL	10.50153424713889	BENZOIC ACID	rxcui:18989	BENZOIC ACID	TRUE	FALSE	FALSE
UNIPROT:Q15858	hgnc:10597	SCN9A	TdgClinicalTrial	Jan-14	NULL	0.062509132	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.375054795	DIPYRIDYL	chembl:CHEMBL39879	DIPYRIDYL	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.011152861	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	0.7573221812840553	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.055681518	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.06757744	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.8607814956671229	DESOGESTREL	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.3723948314588262	Pancuronium	rxcui:7883	PANCURONIUM	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.1785975212098452	Famitinib	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.053145416	IUPHAR.LIGAND:7791	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.035098711	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.012738397	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.021370644	MIBEFRADIL DIHYDROCHLORIDE	rxcui:83214	MIBEFRADIL DIHYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	SJ000244629	chembl:CHEMBL592115	CHEMBL:CHEMBL592115	FALSE	FALSE	FALSE
METTL21A	hgnc:30476	METTL21A	PharmGKB	4/5/24	NULL	1.514644363	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ARANIDIPINE	ncit:C73022	ARANIDIPINE	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	DTC	9/2/20	NULL	1.312691780892362	PHENMEDIPHAM	chembl:CHEMBL1079421	PHENMEDIPHAM	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.04464938	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	NAPROXCINOD	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
UNIPROT:P07202	hgnc:12015	TPO	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.1346350544504987	IUPHAR.LIGAND:941	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:1279	iuphar.ligand:1278	JNJ 7777120	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:12350	iuphar.ligand:12350	CEE321	FALSE	FALSE	FALSE
NCBIGENE:254	hgnc:6585	LHCGR	GuideToPharmacology	2024.1	agonist	16.40864726115453	IUPHAR.LIGAND:1159	rxcui:388084	LUTROPIN ALFA	TRUE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.053854022	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
SSTR1	hgnc:11330	SSTR1	PharmGKB	4/5/24	NULL	1.750255707856483	lutetium (177Lu) oxodotreotide	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
DEFA5	hgnc:2764	DEFA5	NCI	14-Sep-17	NULL	3.750547945406749	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
REPULSIVE GUIDANCE MOLECULE A	hgnc:30308	RGMA	TTD	2020.06.01	NULL	52.50767123569449	Elezanumab	ncit:C169936	ELEZANUMAB	FALSE	FALSE	FALSE
LYSOSOMAL ALPHA-GLUCOSIDASE	hgnc:4065	GAA	TTD	2020.06.01	NULL	0.729273212	BMN-701	chembl:CHEMBL3707295	REVEGLUCOSIDASE ALFA	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000043134	chembl:CHEMBL592332	CHEMBL:CHEMBL592332	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CIS-(Z)-FLUPENTHIXOL DIHYDROCHLORIDE	chembl:CHEMBL1256995	CHEMBL:CHEMBL1256995	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	BROMFENAC SODIUM	rxcui:47364	BROMFENAC SODIUM	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.2778183663264258	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P08183	hgnc:40	ABCB1	TdgClinicalTrial	Jan-14	NULL	0.02804897	TESMILIFENE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
RPS2	hgnc:10404	RPS2	ChEMBL	33	inhibitor	0.1093909817410302	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	GLYX-13	chembl:CHEMBL3544917	RAPASTINEL	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	TESOFENSINE	ncit:C66589	TESOFENSINE	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:8836	iuphar.ligand:8836	PP1	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.2134458180312784	IUPHAR.LIGAND:9702	iuphar.ligand:9702	TUBASTATIN A	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.3241214273808302	C225	ncit:C225	RECOMBINANT INTERFERON ALFA	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.2027323213733378	EHDP	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.035670972	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.2586584789935689	AZD8108	chembl:CHEMBL3707355	AZD8108	FALSE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.087512785	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O00254	hgnc:3539	F2RL2	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	RUSALATIDE	ncit:C152274	RUSALATIDE	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
PRKCI	hgnc:9404	PRKCI	DTC	9/2/20	NULL	0.1193356164447602	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	2.917092846427472	METOLAZONE	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	0.1339481409073839	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UNIPROT:O43174	hgnc:2603	CYP26A1	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	LIAROZOLE	ncit:C1433	LIAROZOLE	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:7360	iuphar.ligand:7360	AZD1283	FALSE	FALSE	FALSE
NCBIGENE:2428	hgnc:3938	FRA9D	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:7898	iuphar.ligand:7898	ML323	FALSE	FALSE	FALSE
IL2RG	hgnc:6010	IL2RG	ChEMBL	33	inhibitor	1.312691780892362	DACLIZUMAB	rxcui:190353	DACLIZUMAB	TRUE	TRUE	FALSE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FRK	hgnc:3955	FRK	ChEMBL	33	inhibitor	0.1562728310586145	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
UNIPROT:Q03405	hgnc:9053	PLAUR	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	1.544343271638073	IUPHAR.LIGAND:4489	iuphar.ligand:4489	[11C]GLYSAR	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.048379304	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1077080435603989	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	BUTYLPARABEN	rxcui:1306937	BUTYLPARABEN	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.6863747873946993	tiludronate	rxcui:11476	TILUDRONIC ACID	TRUE	FALSE	FALSE
DCK	hgnc:2704	DCK	NCI	14-Sep-17	NULL	1.712206670729168	DEOXYCYTIDINE	rxcui:2642208	DEOXYCYTIDINE	FALSE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.4375639269641208	ROCURONIUM BROMIDE	rxcui:32521	ROCURONIUM BROMIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1041818873724097	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.087512785	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9BZL6	hgnc:17293	PRKD2	TdgClinicalTrial	Jan-14	NULL	0.1286952726365061	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.09055649	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.096050618	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
HTRA1	hgnc:9476	HTRA1	NCI	14-Sep-17	NULL	2.625383561784725	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.1022876712383659	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P24723	hgnc:9403	PRKCH	TdgClinicalTrial	Jan-14	NULL	0.3409589041278863	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.066297565	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DES	hgnc:2770	DES	NCI	14-Sep-17	NULL	1.750255707856483	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.061055432	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	CancerCommons	25-Jul-13	inhibitor	0.2983390411119005	SCH727965	hemonc:160	DINACICLIB	FALSE	FALSE	TRUE
UNIPROT:Q01718	hgnc:6930	MC2R	TdgClinicalTrial	Jan-14	NULL	2.461297089173179	CORTICOTROPIN	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	CancerCommons	25-Jul-13	inhibitor	0.1704794520639431	SCH727965	hemonc:160	DINACICLIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	CancerCommons	25-Jul-13	inhibitor	0.272767123	COMETRIQ	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
CDK1	hgnc:1722	CDK1	CancerCommons	25-Jul-13	inhibitor	0.2573905452730122	SCH727965	hemonc:160	DINACICLIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	CancerCommons	25-Jul-13	inhibitor	0.1860654544142257	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	CGI	2/1/22	NULL	NULL	Tensirolimus	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	1.675776741564718	CYCRIMINE	rxcui:22037	CYCRIMINE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	CGI	2/1/22	NULL	NULL	Entrictinib	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	NULL	Tensirolimus	NULL	NULL	NULL	NULL	NULL
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	NULL	Tensirolimus	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	0.4278402841426959	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.00479785	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TSC2	hgnc:12363	TSC2	CGI	2/1/22	NULL	NULL	Tensirolimus	NULL	NULL	NULL	NULL	NULL
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.1411496538593938	TRIMEPRAZINE TARTRATE	rxcui:164308	TRIMEPRAZINE TARTRATE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	TRIPELENNAMINE CITRATE	rxcui:71533	TRIPELENNAMINE CITRATE	TRUE	FALSE	FALSE
UNIPROT:Q01718	hgnc:6930	MC2R	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	COSYNTROPIN	rxcui:2890	COSYNTROPIN	TRUE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	0.6177373086552295	DARBEPOETIN ALFA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.025942525	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.05293112	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.028645756	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
DDC	hgnc:2719	DDC	ChEMBL	33	inhibitor	5.250767123569449	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	0.064347636	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	2.692701089009974	ERYTHRITYL TETRANITRATE	rxcui:4040	ERYTHRITYL TETRANITRATE	TRUE	FALSE	FALSE
SCTR	hgnc:10608	SCTR	ChEMBL	33	agonist	10.50153424713889	SECRETIN SYNTHETIC PORCINE	chembl:CHEMBL1201616	SECRETIN SYNTHETIC PORCINE	TRUE	FALSE	FALSE
SCTR	hgnc:10608	SCTR	ChEMBL	33	agonist	15.75230137070834	SECRETIN	rxcui:9627	SECRETIN	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP EXTENDED PURIFIED BEEF	chembl:CHEMBL1201542	INSULIN ZINC SUSP EXTENDED PURIFIED BEEF	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN SUSP ISOPHANE BEEF/PORK	chembl:CHEMBL1201635	INSULIN SUSP ISOPHANE BEEF/PORK	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP PURIFIED BEEF	chembl:CHEMBL1201546	INSULIN ZINC SUSP PURIFIED BEEF	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.048859496	ZIPRASIDONE MESYLATE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.048859496	ZIPRASIDONE HYDROCHLORIDE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.048260727	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.077217164	OLANZAPINE PAMOATE	rxcui:1294588	OLANZAPINE PAMOATE	TRUE	FALSE	FALSE
MURA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FOSFOMYCIN TROMETHAMINE	rxcui:142135	FOSFOMYCIN TROMETHAMINE	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	agonist	2.763561643983921	DESOXYCORTICOSTERONE PIVALATE	rxcui:22537	DESOXYCORTICOSTERONE PIVALATE	TRUE	FALSE	FALSE
UNIPROT:P03886	hgnc:7455	MT-ND1	TdgClinicalTrial	Jan-14	NULL	0.3387591692625452	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	2.812910959055062	BIMATOPROST	rxcui:283810	BIMATOPROST	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	AMBENONIUM CHLORIDE	rxcui:624	AMBENONIUM CHLORIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	PARAMETHASONE ACETATE	rxcui:32895	PARAMETHASONE ACETATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	1.202465753489187	FLUTICASONE FUROATE	rxcui:705022	FLUTICASONE FUROATE	TRUE	FALSE	FALSE
UNIPROT:P20594	hgnc:7944	NPR2	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	ERYTHRITYL TETRANITRATE	rxcui:4040	ERYTHRITYL TETRANITRATE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.096521454	EPHEDRINE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
UNIPROT:O43497	hgnc:1394	CACNA1G	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	ETHOSUXIMIDE	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.133607306	DESOXIMETASONE	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.3059887601147698	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.084383562	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	1.750255707856483	ABCIXIMAB	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.2453629496995069	ESTROGENS, ESTERIFIED	rxcui:214549	ESTROGENS, ESTERIFIED (USP)	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344583	INTERFERON ALFA-2B, RECOMBINANT	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	1.419126249613364	ISOCARBOXAZID	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.4070362111294147	TIZANIDINE HYDROCHLORIDE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIK5	hgnc:4583	GRIK5	ChEMBL	33	inhibitor	0.1193356164447602	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.070197421	DICLOFENAC SODIUM	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	ChEMBL	33	agonist	1.215455352678113	OCTREOTIDE ACETATE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.4167275494896388	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
IMPDH2	hgnc:6053	IMPDH2	ChEMBL	33	inhibitor	0.1591141552596803	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	0.729273212	OCTREOTIDE ACETATE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	0.3182283105193606	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.07631929	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.6731752722524935	PARGYLINE HYDROCHLORIDE	rxcui:82069	PARGYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.2027323213733378	PHENELZINE SULFATE	rxcui:8124	PHENELZINE SULFATE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.4023576339899962	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
SCNN1B	hgnc:10600	SCNN1B	ChEMBL	33	blocker	1.640864726115453	AMILORIDE HYDROCHLORIDE	rxcui:142424	AMILORIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O60664	hgnc:16893	PLIN3	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	IDURSULFASE	rxcui:644101	IDURSULFASE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.066047385	VERAPAMIL HYDROCHLORIDE	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1320947704042629	AMLODIPINE BESYLATE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3125456621172291	DILTIAZEM MALATE	rxcui:81999	DILTIAZEM MALATE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.08334551	AMLODIPINE BESYLATE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.078136416	DILTIAZEM HYDROCHLORIDE	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	BOCEPREVIR	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	inhibitor	0.6731752722524935	ABCIXIMAB	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.1315981735230438	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
THRA	hgnc:11796	THRA	ChEMBL	33	agonist	0.7501095890813501	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
BCHE	hgnc:983	BCHE	ChEMBL	33	inhibitor	0.6563458904461812	RIVASTIGMINE TARTRATE	rxcui:994808	RIVASTIGMINE TARTRATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	BITOLTEROL MESYLATE	rxcui:47187	BITOLTEROL MESYLATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.029235897	TESTOSTERONE ENANTHATE	rxcui:37859	TESTOSTERONE ENANTHATE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.108711535	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.6819178082557726	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
TNFRSF8	hgnc:11923	TNFRSF8	ChEMBL	33	inhibitor	1.276228120312019	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	ChEMBL	33	inhibitor	0.7001022831425934	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.1013661606866689	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	ChEMBL	33	inhibitor	0.1166837138570989	COBICISTAT	rxcui:1306284	COBICISTAT	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.2778183663264258	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	1.591141552596803	ECULIZUMAB	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
CYP3A4	hgnc:2637	CYP3A4	ChEMBL	33	inhibitor	0.011746683	COBICISTAT	rxcui:1306284	COBICISTAT	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
PSMD13	hgnc:9558	PSMD13	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	MICONAZOLE NITRATE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.1470803115845784	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.4773424657790409	FOSAMPRENAVIR CALCIUM	rxcui:358262	FOSAMPRENAVIR	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.5250767123569451	RESCINNAMINE	rxcui:9259	RESCINNAMINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.9546849315580818	CARPROFEN	rxcui:20343	CARPROFEN	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.2386712328895204	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.5250767123569451	RAPACURONIUM BROMIDE	rxcui:228530	RAPACURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.6250913242344582	ATRACURIUM BESYLATE	rxcui:1219	ATRACURIUM BESYLATE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.6250913242344582	ROCURONIUM BROMIDE	rxcui:32521	ROCURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.5527123287967842	TUBOCURARINE CHLORIDE	rxcui:82115	TUBOCURARINE CHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.052090944	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
8238275	NULL	NULL	ChEMBL	33	agonist	NULL	SPINOSAD	rxcui:299081	SPINOSAD	TRUE	FALSE	FALSE
UNIPROT:O43451	hgnc:7043	MGAM	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	MIGLITOL	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
8238272	NULL	NULL	ChEMBL	33	agonist	NULL	SPINOSAD	rxcui:299081	SPINOSAD	TRUE	FALSE	FALSE
8238273	NULL	NULL	ChEMBL	33	agonist	NULL	SPINOSAD	rxcui:299081	SPINOSAD	TRUE	FALSE	FALSE
8232849	NULL	NULL	ChEMBL	33	agonist	NULL	SPINOSAD	rxcui:299081	SPINOSAD	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.056826484	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
8232852	NULL	NULL	ChEMBL	33	agonist	NULL	SPINOSAD	rxcui:299081	SPINOSAD	TRUE	FALSE	FALSE
8232002	NULL	NULL	ChEMBL	33	agonist	NULL	SPINOSAD	rxcui:299081	SPINOSAD	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.050879526	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
RXRB	hgnc:10478	RXRB	ChEMBL	33	agonist	0.8334550989792776	ETRETINATE	rxcui:4182	ETRETINATE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.8950171233357017	MORICIZINE	rxcui:40169	MORICIZINE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.078682824	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.096758608	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.022155136	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.031254566	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.061055432	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.080781033	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.076840494	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.018942161	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.1084869240406911	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	BESIFLOXACIN HYDROCHLORIDE	ncit:C76228	BESIFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ALATROFLOXACIN MESYLATE	rxcui:221054	ALATROFLOXACIN MESYLATE	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NORFLOXACIN	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPARFLOXACIN	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFADIAZINE, SILVER	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFANILAMIDE	rxcui:10184	SULFANILAMIDE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFACETAMIDE SODIUM	rxcui:82101	SULFACETAMIDE SODIUM	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAMETHOXAZOLE	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFISOXAZOLE	rxcui:10207	SULFISOXAZOLE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAPYRIDINE	rxcui:10188	SULFAPYRIDINE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFADIAZINE	rxcui:10171	SULFADIAZINE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAMETER	ncit:C66568	SULFAMETER	TRUE	FALSE	FALSE
BLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLAVULANATE POTASSIUM	rxcui:831418	CLAVULANATE POTASSIUM	TRUE	FALSE	FALSE
BLAT-3	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLAVULANATE POTASSIUM	rxcui:831418	CLAVULANATE POTASSIUM	TRUE	FALSE	FALSE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TdgClinicalTrial	Jan-14	NULL	0.9053046764774912	THIAMYLAL	rxcui:10464	THIAMYLAL	TRUE	FALSE	FALSE
BLAT-4	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLAVULANATE POTASSIUM	rxcui:831418	CLAVULANATE POTASSIUM	TRUE	FALSE	FALSE
BLAT-5	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLAVULANATE POTASSIUM	rxcui:831418	CLAVULANATE POTASSIUM	TRUE	FALSE	FALSE
BLAT-6	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLAVULANATE POTASSIUM	rxcui:831418	CLAVULANATE POTASSIUM	TRUE	FALSE	FALSE
BLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULBACTAM SODIUM	rxcui:82100	SULBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-3	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULBACTAM SODIUM	rxcui:82100	SULBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-4	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULBACTAM SODIUM	rxcui:82100	SULBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-5	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULBACTAM SODIUM	rxcui:82100	SULBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-6	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULBACTAM SODIUM	rxcui:82100	SULBACTAM SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME SODIUM	rxcui:221071	CEFTAZIDIME SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME SODIUM	rxcui:221071	CEFTAZIDIME SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME SODIUM	rxcui:221071	CEFTAZIDIME SODIUM	TRUE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	0.7292732116068681	TREPROSTINIL	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME SODIUM	rxcui:221071	CEFTAZIDIME SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME SODIUM	rxcui:221071	CEFTAZIDIME SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME SODIUM	rxcui:221071	CEFTAZIDIME SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME SODIUM	rxcui:221071	CEFTAZIDIME SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTRIAXONE SODIUM	rxcui:203172	CEFTRIAXONE SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTRIAXONE SODIUM	rxcui:203172	CEFTRIAXONE SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTRIAXONE SODIUM	rxcui:203172	CEFTRIAXONE SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTRIAXONE SODIUM	rxcui:203172	CEFTRIAXONE SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTRIAXONE SODIUM	rxcui:203172	CEFTRIAXONE SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTRIAXONE SODIUM	rxcui:203172	CEFTRIAXONE SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTRIAXONE SODIUM	rxcui:203172	CEFTRIAXONE SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFEPIME HYDROCHLORIDE	rxcui:236058	CEFEPIME HYDROCHLORIDE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFEPIME HYDROCHLORIDE	rxcui:236058	CEFEPIME HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.1136529680426287	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFEPIME HYDROCHLORIDE	rxcui:236058	CEFEPIME HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFEPIME HYDROCHLORIDE	rxcui:236058	CEFEPIME HYDROCHLORIDE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFEPIME HYDROCHLORIDE	rxcui:236058	CEFEPIME HYDROCHLORIDE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFEPIME HYDROCHLORIDE	rxcui:236058	CEFEPIME HYDROCHLORIDE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFEPIME HYDROCHLORIDE	rxcui:236058	CEFEPIME HYDROCHLORIDE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTAZIDIME	rxcui:1545984	CEFTAZIDIME ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDITOREN PIVOXIL	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDITOREN PIVOXIL	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDITOREN PIVOXIL	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDITOREN PIVOXIL	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDITOREN PIVOXIL	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDITOREN PIVOXIL	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFDITOREN PIVOXIL	rxcui:72611	CEFDITOREN PIVOXIL	TRUE	FALSE	FALSE
PBP4	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFCILLIN SODIUM	rxcui:9893	NAFCILLIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	TOLBUTAMIDE	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
PBPF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFCILLIN SODIUM	rxcui:9893	NAFCILLIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:Q9NYX4	hgnc:17938	CALY	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
MECA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFCILLIN SODIUM	rxcui:9893	NAFCILLIN SODIUM	TRUE	FALSE	FALSE
PBP2	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFCILLIN SODIUM	rxcui:9893	NAFCILLIN SODIUM	TRUE	FALSE	FALSE
PBPA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFCILLIN SODIUM	rxcui:9893	NAFCILLIN SODIUM	TRUE	FALSE	FALSE
PBP4	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXACILLIN SODIUM	rxcui:7773	OXACILLIN	TRUE	FALSE	FALSE
PBPF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXACILLIN SODIUM	rxcui:7773	OXACILLIN	TRUE	FALSE	FALSE
MECA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXACILLIN SODIUM	rxcui:7773	OXACILLIN	TRUE	FALSE	FALSE
PBP2	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXACILLIN SODIUM	rxcui:7773	OXACILLIN	TRUE	FALSE	FALSE
PBPA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXACILLIN SODIUM	rxcui:7773	OXACILLIN	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.1305078821102597	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TdgClinicalTrial	Jan-14	NULL	0.3512218811752141	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	ENFUVIRTIDE	rxcui:139896	ENFUVIRTIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	0.3671865121377238	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TEND	1-Aug-11	NULL	1.790034246671403	CONIVAPTAN	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	STREPTOMYCIN SULFATE	rxcui:10110	STREPTOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.2375912725597036	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.055504938	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.083257407	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.091796628	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.085239726	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TEND	1-Aug-11	NULL	2.625383561784724	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.6482428547616604	DIETHYLPROPION	rxcui:3389	DIETHYLPROPION	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	0.9376369863516874	INTERFERON ALFA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	1.312691780892362	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.3017682254924971	PEGINTERFERON ALFA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	inhibitor	1.029562181092049	DACLIZUMAB	rxcui:190353	DACLIZUMAB	TRUE	TRUE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	2.917092846427472	INTERFERON ALFA-N3	rxcui:612937	INTERFERON ALFA-N3	TRUE	TRUE	TRUE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	0.3394892536790592	PEGINTERFERON ALFA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BESIFLOXACIN HYDROCHLORIDE	ncit:C76228	BESIFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	BESIFLOXACIN HYDROCHLORIDE	ncit:C76228	BESIFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ALATROFLOXACIN MESYLATE	rxcui:221054	ALATROFLOXACIN MESYLATE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ALATROFLOXACIN MESYLATE	rxcui:221054	ALATROFLOXACIN MESYLATE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CINOXACIN	rxcui:2550	CINOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CINOXACIN	rxcui:2550	CINOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NORFLOXACIN	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NORFLOXACIN	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPARFLOXACIN	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SPARFLOXACIN	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GEMIFLOXACIN MESYLATE	rxcui:402429	GEMIFLOXACIN MESYLATE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GEMIFLOXACIN MESYLATE	rxcui:402429	GEMIFLOXACIN MESYLATE	TRUE	FALSE	FALSE
S1PR4	hgnc:3170	S1PR4	ChEMBL	33	agonist	1.166837138570989	FINGOLIMOD HYDROCHLORIDE	rxcui:1012891	FINGOLIMOD HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.042968634	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.017047945	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.017859752	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.062808219	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.2169738480813822	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.032899543	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.040328473	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.051478109	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RDL1	NULL	NULL	ChEMBL	33	negative modulator	NULL	LINDANE	rxcui:1388	LINDANE	TRUE	FALSE	FALSE
RDL2	NULL	NULL	ChEMBL	33	negative modulator	NULL	LINDANE	rxcui:1388	LINDANE	TRUE	FALSE	FALSE
RDL3	NULL	NULL	ChEMBL	33	negative modulator	NULL	LINDANE	rxcui:1388	LINDANE	TRUE	FALSE	FALSE
8239847	NULL	NULL	ChEMBL	33	negative modulator	NULL	LINDANE	rxcui:1388	LINDANE	TRUE	FALSE	FALSE
8232983	NULL	NULL	ChEMBL	33	negative modulator	NULL	LINDANE	rxcui:1388	LINDANE	TRUE	FALSE	FALSE
8233868	NULL	NULL	ChEMBL	33	negative modulator	NULL	LINDANE	rxcui:1388	LINDANE	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	GEMIFLOXACIN MESYLATE	rxcui:402429	GEMIFLOXACIN MESYLATE	TRUE	FALSE	FALSE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FIDAXOMICIN	rxcui:1111103	FIDAXOMICIN	TRUE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FIDAXOMICIN	rxcui:1111103	FIDAXOMICIN	TRUE	FALSE	FALSE
KCNK9	hgnc:6283	KCNK9	ChEMBL	33	potentiator	0.2917092846427472	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	GEMIFLOXACIN MESYLATE	rxcui:402429	GEMIFLOXACIN MESYLATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPME2	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMG1	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMG2	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMG3	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
KCNG2	hgnc:6249	KCNG2	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNF1	hgnc:6246	KCNF1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNG4	hgnc:19697	KCNG4	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNB2	hgnc:6232	KCNB2	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNA6	hgnc:6225	KCNA6	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNG1	hgnc:6248	KCNG1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNH6	hgnc:18862	KCNH6	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	LULICONAZOLE	rxcui:1482680	LULICONAZOLE	TRUE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	positive modulator	1.166837138570989	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	positive modulator	1.235474617310459	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.2083637747448194	BAZEDOXIFENE ACETATE	rxcui:1442171	BAZEDOXIFENE ACETATE	TRUE	FALSE	FALSE
KCNS2	hgnc:6301	KCNS2	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNG2	hgnc:6249	KCNG2	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.016927038	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.070197421	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
PDE9A	hgnc:8795	PDE9A	ChEMBL	33	inhibitor	0.046549354	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE7A	hgnc:8791	PDE7A	ChEMBL	33	inhibitor	0.074478966	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.297662535	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1442518440541057	BREXPIPRAZOLE	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.729273212	PASIREOTIDE PAMOATE	rxcui:1597818	PASIREOTIDE PAMOATE	TRUE	FALSE	FALSE
CD38	hgnc:1667	CD38	ChEMBL	33	inhibitor	0.3889457128569963	DARATUMUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.058799184	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	ChEMBL	33	inhibitor	0.1315981735230438	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.032134438	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	0.060353645	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
SRMS	hgnc:11298	SRMS	ChEMBL	33	inhibitor	0.1131630845596864	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.092443083	4SC-203	drugbank:DB12669	4SC-203	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.1411496538593938	CERDULATINIB	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.9546849315580818	ARRY-382	iuphar.ligand:9108	ARRY-382	FALSE	FALSE	FALSE
CDK10	hgnc:1770	CDK10	ChEMBL	33	inhibitor	0.4375639269641208	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.056826484	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.087512785	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK15	hgnc:14434	CDK15	ChEMBL	33	inhibitor	0.546954909	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
PIM1	hgnc:8986	PIM1	ChEMBL	33	inhibitor	0.5000730593875666	AZD-1208	chembl:CHEMBL3545423	AZD-1208	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	ChEMBL	33	inhibitor	1.029562181092048	AZD-1208	chembl:CHEMBL3545423	AZD-1208	FALSE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.1215455352678113	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK20	hgnc:21420	CDK20	ChEMBL	33	inhibitor	0.546954909	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	3.281729452230906	CE-245677	chembl:CHEMBL3545120	CE-245677	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.092606122	MP-412	chembl:CHEMBL5095024	MP-412	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.2966535098061835	MK-6592	chembl:CHEMBL3545378	MK-6592	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	1.166837138570988	MK-6592	chembl:CHEMBL3545378	MK-6592	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.364636606	MSC-2363318A	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1041818873724097	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.07463777	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.066297565	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1530835896084387	AZD8108	chembl:CHEMBL3707355	AZD8108	FALSE	FALSE	FALSE
UNIPROT:P03886	hgnc:7455	MT-ND1	TEND	1-Aug-11	NULL	0.3387591692625452	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	1.280674908	MAVATREP	ncit:C170153	MAVATREP	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.1209854175937661	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.042619863	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.062509132	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	4.145342465975881	FINERENONE	rxcui:2562811	FINERENONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.087707691	CLASCOTERONE	rxcui:2474340	CLASCOTERONE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.1315981735230438	INDEGLITAZAR	ncit:C98153	INDEGLITAZAR	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.1400204566285186	INDEGLITAZAR	ncit:C98153	INDEGLITAZAR	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.040703621	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.2651902587661338	INDEGLITAZAR	ncit:C98153	INDEGLITAZAR	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	DRF-10945	chembl:CHEMBL3545394	DRF-10945	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	ChEMBL	33	inhibitor	0.026899422	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.057574201	AEE-788	drugbank:DB12558	AEE-788	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.8468979231563628	PEFICITINIB	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.082559232	AXL-1717	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.317586721	EPINASTINE	rxcui:39684	EPINASTINE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.2187819634820604	JI-101	chembl:CHEMBL3545155	JI-101	FALSE	FALSE	FALSE
EPHB4	hgnc:3395	EPHB4	ChEMBL	33	inhibitor	4.375639269641208	JI-101	chembl:CHEMBL3545155	JI-101	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	1.312691780892362	DANUSERTIB	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	1.500219178	R-112	chembl:CHEMBL3545399	R-112	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1389091831632129	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	PG-760564	chembl:CHEMBL3545398	PG-760564	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	1.193356164447602	ENCAINIDE	rxcui:42368	ENCAINIDE	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	1.009762908	XL-281	chembl:CHEMBL3545027	XL-281	FALSE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	0.729273212	VABICASERIN HYDROCHLORIDE	ncit:C142993	VABICASERIN HYDROCHLORIDE	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.1988926940746003	LY377604	chembl:CHEMBL2012520	LY377604	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1084869240406911	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.099446347	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
GRM3	hgnc:4595	GRM3	ChEMBL	33	modulator	2.625383561784724	DECOGLURANT	ncit:C166865	DECOGLURANT	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	1.750255707856483	CENICRIVIROC	ncit:C166464	CENICRIVIROC	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	1.381780822	QAV680	iuphar.ligand:8996	QAV680	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	LY2624803	chembl:CHEMBL3545287	LY2624803	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.096521454	EPHEDRINE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	modulator	0.2243917574174979	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	modulator	0.1442518440541058	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	modulator	0.1187956362798518	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1226814748497534	ETHYNODIOL DIACETATE	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	modulator	0.2243917574174979	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	modulator	0.2243917574174979	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	modulator	0.2019525816757481	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	modulator	0.1346350544504987	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TEND	1-Aug-11	NULL	0.036977233	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.111481255	SEOCALCITOL	ncit:C26669	SEOCALCITOL	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.5303805175322676	IMIGLITAZAR	ncit:C83791	IMIGLITAZAR	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.040893825	DROLOXIFENE	ncit:C969	DROLOXIFENE	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	modulator	0.4303907478335614	ASOPRISNIL	ncit:C91054	ASOPRISNIL	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1111273465305703	CANERTINIB DIHYDROCHLORIDE	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.047821194	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.2108741816694558	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.046881849	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	modulator	0.2243917574174979	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	modulator	0.2243917574174979	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	modulator	0.1553481397505754	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	agonist	0.055681518	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.406619897	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	binder	1.009762908	BEVACIZUMAB 111IN	chembl:CHEMBL3707253	BEVACIZUMAB 111IN	FALSE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	GRAZOPREVIR	rxcui:1734630	GRAZOPREVIR	TRUE	FALSE	FALSE
KCNC3	hgnc:6235	KCNC3	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNB2	hgnc:6232	KCNB2	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNH8	hgnc:18864	KCNH8	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	1.640864726115453	BERUBICIN HYDROCHLORIDE	ncit:C61568	BERUBICIN HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P23921	hgnc:10451	RRM1	TEND	1-Aug-11	NULL	0.2725311655831894	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	ChEMBL	33	inhibitor	0.8751278539282416	EZATIOSTAT HYDROCHLORIDE	ncit:C61326	EZATIOSTAT HYDROCHLORIDE	FALSE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	ChEMBL	33	inhibitor	2.187819634820604	VARESPLADIB	ncit:C152832	VARESPLADIB	FALSE	FALSE	FALSE
RRM2	hgnc:10452	RRM2	ChEMBL	33	inhibitor	1.009762908	TEZACITABINE	ncit:C1539	TEZACITABINE	FALSE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TEND	1-Aug-11	NULL	2.187819634820604	FAMOTIDINE	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.2703097618311171	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.3659071166250487	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.8514757497680189	ISTRADEFYLLINE	rxcui:2199015	ISTRADEFYLLINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.4773424657790409	NAPROXEN ETEMESIL	ncit:C166529	NAPROXEN ETEMESIL	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.086551106	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	ChEMBL	33	other/unknown	3.750547945	MIFAMURTIDE	ncit:C1394	MIFAMURTIDE	TRUE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	0.2333674277141978	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
CNR1	hgnc:2159	CNR1	ChEMBL	33	negative modulator	0.1944728564284981	CANNABIDIOL	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.1785975212098452	CRISABOROLE	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
UNIPROT:P40238	hgnc:7217	MPL	TEND	1-Aug-11	NULL	2.983390411119005	ELTROMBOPAG	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	agonist	0.4579157375205915	TRAFERMIN	ncit:C152708	TRAFERMIN	FALSE	FALSE	FALSE
DDB1	hgnc:2717	DDB1	ChEMBL	33	inhibitor	1.009762908	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	3.088686543276147	ATRELEUTON	ncit:C64176	ATRELEUTON	FALSE	FALSE	FALSE
UNIPROT:P20594	hgnc:7944	NPR2	TEND	1-Aug-11	NULL	5.834185692854944	ERYTHRITYL TETRANITRATE	rxcui:4040	ERYTHRITYL TETRANITRATE	TRUE	FALSE	FALSE
NISCH	hgnc:18006	NISCH	ChEMBL	33	agonist	3.750547945406749	MOXONIDINE	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.2373228078449469	CANDESARTAN	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.3680444245492605	ARZOXIFENE	ncit:C1805	ARZOXIFENE	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	other/unknown	2.187819634820604	HUHMFG1	chembl:CHEMBL2109637	HUHMFG1	FALSE	FALSE	FALSE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	8.751278539282415	ANRUKINZUMAB	ncit:C95781	ANRUKINZUMAB	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1848861663228679	BUPRENORPHINE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
SELL	hgnc:10720	SELL	ChEMBL	33	inhibitor	17.50255707856483	ASELIZUMAB	ncit:C171823	ASELIZUMAB	FALSE	FALSE	FALSE
DKK1	hgnc:2891	DKK1	ChEMBL	33	inhibitor	11.66837138570988	BHQ-880	hemonc:57	BHQ-880	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.022789788	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
TNFSF4	hgnc:11934	TNFSF4	ChEMBL	33	inhibitor	26.25383561784724	OXELUMAB	ncit:C166910	OXELUMAB	FALSE	FALSE	FALSE
TCDB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEZLOTOXUMAB	rxcui:1855048	BEZLOTOXUMAB	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.1204304386139782	NALDEMEDINE TOSYLATE	rxcui:1876597	NALDEMEDINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1017590527823536	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	3.281729452230906	BRAZIKUMAB	ncit:C166795	BRAZIKUMAB	FALSE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	1.875273972703375	BRAZIKUMAB	ncit:C166795	BRAZIKUMAB	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.2294915700860773	METOPROLOL	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
RTN4	hgnc:14085	RTN4	ChEMBL	33	inhibitor	10.50153424713889	ATINUMAB	ncit:C97942	ATINUMAB	FALSE	FALSE	FALSE
CLFA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEFIBAZUMAB	ncit:C152538	TEFIBAZUMAB	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.3431873936973497	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
F12	hgnc:3530	F12	ChEMBL	33	activator	8.751278539282415	BISMUTH SUBGALLATE	rxcui:19476	BISMUTH SUBGALLATE	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	5.834185692854944	IBRITUMOMAB TIUXETAN	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.5147810905460244	NARATRIPTAN	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFSULODIN	rxcui:2190	CEFSULODIN	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFSULODIN	rxcui:2190	CEFSULODIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFSULODIN	rxcui:2190	CEFSULODIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFSULODIN	rxcui:2190	CEFSULODIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFSULODIN	rxcui:2190	CEFSULODIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFSULODIN	rxcui:2190	CEFSULODIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFSULODIN	rxcui:2190	CEFSULODIN	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.099446347	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
HSD11B2	hgnc:5209	HSD11B2	ChEMBL	33	inhibitor	13.12691780892362	CARBENOXOLONE	rxcui:2017	CARBENOXOLONE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.054886067	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	agonist	0.030386384	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.1447821817160693	AGOMELATINE	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	NETARSUDIL DIMESYLATE	chembl:CHEMBL4594251	NETARSUDIL DIMESYLATE	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.2983390411119005	PREDNICARBATE	rxcui:34369	PREDNICARBATE	TRUE	FALSE	FALSE
IFNA16	hgnc:5421	IFNA16	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
IFNA10	hgnc:5418	IFNA10	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	3.500511415712966	VILOBELIMAB	rxcui:2639620	VILOBELIMAB	TRUE	FALSE	FALSE
TNFRSF8	hgnc:11923	TNFRSF8	ChEMBL	33	binder	3.281729452230906	HEFI-1	chembl:CHEMBL2109255	HEFI-1	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.090739063	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
RPS5	hgnc:10426	RPS5	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.008751279	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL18A	hgnc:10311	RPL18A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
UNIPROT:Q9H2X9	hgnc:13818	SLC12A5	TEND	1-Aug-11	NULL	5.834185692854945	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
RPL24	hgnc:10325	RPL24	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL13A	hgnc:10304	RPL13A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL9P7	hgnc:30335	RPL9P7	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL9	hgnc:10369	RPL9	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	2.669881588255652	SAPRISARTAN	ncit:C152297	SAPRISARTAN	FALSE	FALSE	FALSE
RPL13	hgnc:10303	RPL13	ChEMBL	33	inhibitor	0.093763699	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TEND	1-Aug-11	NULL	0.4318065068724876	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	ChEMBL	33	inhibitor	0.9842513760562132	IVOSIDENIB	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.033295923	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1657439117288336	COPANLISIB	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1852122442176172	NERATINIB MALEATE	rxcui:1940642	NERATINIB MALEATE	TRUE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	ChEMBL	33	inhibitor	0.6819178082557726	APABETALONE	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	1.591141552596803	GFT14	drugbank:DB05061	GFT14	FALSE	FALSE	FALSE
MC1R	hgnc:6929	MC1R	ChEMBL	33	agonist	7.501095891	AFAMELANOTIDE ACETATE	rxcui:2278002	AFAMELANOTIDE ACETATE	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL	rxcui:2265702	CEFIDEROCOL	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAVUCONAZOLE	ncit:C38688	RAVUCONAZOLE	FALSE	FALSE	FALSE
L	NULL	NULL	ChEMBL	33	inhibitor	NULL	REMDESIVIR	rxcui:2284718	REMDESIVIR	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	CILUPREVIR	ncit:C76016	CILUPREVIR	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	0.7721716358190367	MIS-416	ncit:C127934	MICROPARTICLE MDP/BACTERIAL DNA-CONTAINING MIS416	FALSE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.7001022831425934	RAMOSETRON HYDROCHLORIDE	ncit:C88299	RAMOSETRON HYDROCHLORIDE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	PEMAFIBRATE	ncit:C166474	PEMAFIBRATE	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	ChEMBL	33	inhibitor	1.250182648468916	FADROZOLE HYDROCHLORIDE	ncit:C1044	FADROZOLE HYDROCHLORIDE	FALSE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	5.250767123569449	EPOETIN THETA	chembl:CHEMBL2108290	EPOETIN THETA	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	ChEMBL	33	inhibitor	4.039051633514961	OXYPURINOL	ncit:C87294	OXYPURINOL	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL SULFATE TOSYLATE	rxcui:2265863	CEFIDEROCOL SULFATE TOSYLATE	TRUE	FALSE	FALSE
PANCREATIC ALPHA-AMYLASE	hgnc:477	AMY2A	TTD	2020.06.01	NULL	0.8751278539282416	Liprotamase	chembl:CHEMBL2108703	LIPROTAMASE	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL SULFATE TOSYLATE	rxcui:2265863	CEFIDEROCOL SULFATE TOSYLATE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL SULFATE TOSYLATE	rxcui:2265863	CEFIDEROCOL SULFATE TOSYLATE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL SULFATE TOSYLATE	rxcui:2265863	CEFIDEROCOL SULFATE TOSYLATE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL SULFATE TOSYLATE	rxcui:2265863	CEFIDEROCOL SULFATE TOSYLATE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL SULFATE TOSYLATE	rxcui:2265863	CEFIDEROCOL SULFATE TOSYLATE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIDEROCOL SULFATE TOSYLATE	rxcui:2265863	CEFIDEROCOL SULFATE TOSYLATE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE MEDOCARIL	ncit:C70597	CEFTOBIPROLE MEDOCARIL	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE MEDOCARIL	ncit:C70597	CEFTOBIPROLE MEDOCARIL	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE MEDOCARIL	ncit:C70597	CEFTOBIPROLE MEDOCARIL	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE MEDOCARIL	ncit:C70597	CEFTOBIPROLE MEDOCARIL	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE MEDOCARIL	ncit:C70597	CEFTOBIPROLE MEDOCARIL	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE MEDOCARIL	ncit:C70597	CEFTOBIPROLE MEDOCARIL	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOBIPROLE MEDOCARIL	ncit:C70597	CEFTOBIPROLE MEDOCARIL	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.5164688974002737	RIPRETINIB	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	0.8537832721251137	TAFASITAMAB	rxcui:2387211	TAFASITAMAB	TRUE	FALSE	FALSE
REP	NULL	NULL	ChEMBL	33	inhibitor	NULL	REMDESIVIR	rxcui:2284718	REMDESIVIR	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	2.019525817	DOTINURAD	ncit:C166614	DOTINURAD	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
RPS3	hgnc:10420	RPS3	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS15A	hgnc:10389	RPS15A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS8	hgnc:10441	RPS8	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS16	hgnc:10396	RPS16	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPL27A	hgnc:10329	RPL27A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS28	hgnc:10418	RPS28	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL9P9	hgnc:30334	RPL9P8	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL34	hgnc:10340	RPL34	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL35A	hgnc:10345	RPL35A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL38	hgnc:10349	RPL38	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.2134458180312784	SINTILIMAB	ncit:C132992	SINTILIMAB	FALSE	FALSE	FALSE
CCKAR	hgnc:1570	CCKAR	ChEMBL	33	agonist	2.625383561784724	CE-326597	drugbank:DB12694	CE-326597	FALSE	FALSE	FALSE
PFATPASE4	NULL	NULL	ChEMBL	33	inhibitor	NULL	CIPARGAMIN	ncit:C169853	CIPARGAMIN	FALSE	FALSE	FALSE
RGMA	hgnc:30308	RGMA	ChEMBL	33	inhibitor	52.50767123569449	ELEZANUMAB	ncit:C169936	ELEZANUMAB	FALSE	FALSE	FALSE
LTB4R2	hgnc:19260	LTB4R2	ChEMBL	33	inhibitor	4.375639269641208	NOMACOPAN	ncit:C167012	NOMACOPAN	FALSE	FALSE	FALSE
L	NULL	NULL	ChEMBL	33	inhibitor	NULL	PC-786	chembl:CHEMBL4291143	PC-786	FALSE	FALSE	FALSE
RPL26	hgnc:10327	RPL26	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PEFLOXACIN	rxcui:7960	PEFLOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PEFLOXACIN	rxcui:7960	PEFLOXACIN	TRUE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	ODALASVIR	ncit:C174815	ODALASVIR	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	2.059124362184098	ELGEMTUMAB	ncit:C101895	ELGEMTUMAB	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	positive modulator	0.596678082	TAK-653	drugbank:DB16304	TAK-653	FALSE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	ChEMBL	33	agonist	3.281729452230906	SELGANTOLIMOD	ncit:C170376	SELGANTOLIMOD	FALSE	FALSE	FALSE
TNFRSF13C	hgnc:17755	TNFRSF13C	ChEMBL	33	binder	35.00511415712966	IANALUMAB	ncit:C116788	IANALUMAB	FALSE	FALSE	FALSE
DRD5	hgnc:3026	DRD5	ChEMBL	33	agonist	1.312691780892362	TAVAPADON	ncit:C174853	TAVAPADON	FALSE	FALSE	FALSE
PTPRB	hgnc:9665	PTPRB	ChEMBL	33	inhibitor	19.69037671338543	RAZUPROTAFIB	ncit:C152161	RAZUPROTAFIB	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.8334550989792777	PARSACLISIB	ncit:C113434	PARSACLISIB	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.094438258	SKLB1028	iuphar.ligand:12089	RUSERONTINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	agonist	0.3241214273808302	CDX-301	chembl:CHEMBL4650387	CDX-301	FALSE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	1.458546423213736	TRILACICLIB DIHYDROCHLORIDE	rxcui:2479691	TRILACICLIB DIHYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	ChEMBL	33	inhibitor	0.3851418428046051	DS-1001B	chembl:CHEMBL4650282	DS-1001B	FALSE	FALSE	FALSE
EPAS1	hgnc:3374	EPAS1	ChEMBL	33	inhibitor	1.750255707856483	BELZUTIFAN	rxcui:2567226	BELZUTIFAN	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.3500511415712967	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.056097939	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.042898424	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.6364566210387211	EFPEGLENATIDE	ncit:C166682	EFPEGLENATIDE	FALSE	FALSE	FALSE
N	NULL	NULL	ChEMBL	33	inhibitor	NULL	RSV-604	drugbank:DB15197	RSV-604	FALSE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	5.250767123569449	EFEPOETIN ALFA	ncit:C169930	EFEPOETIN ALFA	FALSE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	ChEMBL	33	inhibitor	3.281729452230906	TIBULIZUMAB	ncit:C152608	TIBULIZUMAB	FALSE	FALSE	FALSE
MYL7	hgnc:21719	MYL7	ChEMBL	33	activator	2.500365296937833	DANICAMTIV	ncit:C167013	DANICAMTIV	FALSE	FALSE	FALSE
MYL4	hgnc:7585	MYL4	ChEMBL	33	activator	2.500365296937833	DANICAMTIV	ncit:C167013	DANICAMTIV	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	4.565884455277782	MK-0812	drugbank:DB11990	MK-0812	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	negative modulator	0.042174836	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
GAG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LENACAPAVIR	rxcui:2625651	LENACAPAVIR	TRUE	FALSE	FALSE
DHOD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DSM-265	drugbank:DB12397	DSM-265	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.086361301	TARLOXOTINIB	drugbank:DB14944	TARLOXOTINIB	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	RIPASUDIL HYDROCHLORIDE DIHYDRATE	chembl:CHEMBL4594454	RIPASUDIL HYDROCHLORIDE DIHYDRATE	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.6731752722524935	RIPASUDIL HYDROCHLORIDE DIHYDRATE	chembl:CHEMBL4594454	RIPASUDIL HYDROCHLORIDE DIHYDRATE	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	ChEMBL	33	inhibitor	1.346350544504987	BRIMAPITIDE, C-TERMINAL ACID	chembl:CHEMBL4297348	BRIMAPITIDE, C-TERMINAL ACID	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	MOSUNETUZUMAB	rxcui:2625122	MOSUNETUZUMAB	TRUE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	MOSUNETUZUMAB	rxcui:2625122	MOSUNETUZUMAB	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	3.750547945	AL-12182	chembl:CHEMBL184999	AL-12182	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	TMC-647055	drugbank:DB11822	TMC-647055	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1635752997996713	NS-2359	drugbank:DB05805	NS-2359	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	1.009762908	TIBULIZUMAB	ncit:C152608	TIBULIZUMAB	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	BAMLANIVIMAB	rxcui:2463114	BAMLANIVIMAB	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	ChEMBL	33	inhibitor	1.640864726115453	OBEXELIMAB	ncit:C170236	OBEXELIMAB	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	1.009762908	EFLAPEGRASTIM	rxcui:2612526	EFLAPEGRASTIM	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	KN-026	chembl:CHEMBL4594568	KN-026	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.5000730593875666	MESDOPETAM	ncit:C175816	MESDOPETAM	FALSE	FALSE	FALSE
PSEN1	hgnc:9508	PSEN1	ChEMBL	33	inhibitor	0.2885036881082115	NIROGACESTAT	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
PKLR	hgnc:9020	PKLR	ChEMBL	33	activator	17.50255707856483	MITAPIVAT SULFATE	rxcui:2595574	MITAPIVAT SULFATE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	1.750255707856483	MITIGLINIDE	ncit:C81699	MITIGLINIDE	TRUE	FALSE	FALSE
GP	hgnc:18280	RNF130	ChEMBL	33	inhibitor	7.501095891	COSFROVIXIMAB	ncit:C171831	COSFROVIXIMAB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
E7	NULL	NULL	ChEMBL	33	vaccine	NULL	VERPASEP CALTESPEN	ncit:C2811	VERPASEP CALTESPEN	FALSE	FALSE	FALSE
GHR	hgnc:4263	GHR	ChEMBL	33	agonist	5.250767123569449	SOMATROGON	rxcui:2644503	SOMATROGON	TRUE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	modulator	0.8078103267029922	VALILTRAMIPROSATE	ncit:C186402	VALILTRAMIPROSATE	FALSE	FALSE	FALSE
ACACA	hgnc:84	ACACA	ChEMBL	33	inhibitor	0.5707355569097228	CLESACOSTAT	ncit:C177068	CLESACOSTAT	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	2.316514907	HUPERZINE A	rxcui:2267703	HUPERZINE A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	cleavage	0.011694359	DIMETHYLCURCUMIN	drugbank:DB06133	DIMETHYLCURCUMIN	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ZABOFLOXACIN	ncit:C82232	ZABOFLOXACIN	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ZABOFLOXACIN	ncit:C82232	ZABOFLOXACIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	MOBOCERTINIB SUCCINATE	rxcui:2570737	MOBOCERTINIB SUCCINATE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1666910197958555	PHENOXODIOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1101693521639275	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.312691780892362	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.075768645	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
XIAP	hgnc:592	XIAP	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2381300282797936	DEHYDROEQUOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	1.029562181092049	REGN1400	ncit:C103859	ANTI-ERBB3 MONOCLONAL ANTIBODY REGN1400	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	COSMIC	4-Sep-20	NULL	0.637458239	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	1.944728564284981	Senktide	iuphar.ligand:2127	SENKTIDE	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	COSMIC	4-Sep-20	NULL	15.31473744374422	Vismodegib	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.095122593	STANOLONE	ncit:C72098	STANOLONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	TCMDC-125784	chembl:CHEMBL581574	CHEMBL:CHEMBL581574	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	HALCINONIDE	rxcui:5084	HALCINONIDE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.2500365296937833	CMX-2043	drugbank:DB12795	CMX-2043	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	DTC	9/2/20	NULL	0.052350619	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	TCMDC-125602	chembl:CHEMBL580183	CHEMBL:CHEMBL580183	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.018219178	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
MYELOPEROXIDASE	hgnc:7218	MPO	TTD	2020.06.01	NULL	0.5834185692854944	AZD4831	iuphar.ligand:12154	MITIPERSTAT	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.002731502	ESTRADIOL VALERATE	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.5000730593875666	TCMDC-125543	chembl:CHEMBL546170	CHEMBL:CHEMBL546170	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	TCMDC-123579	chembl:CHEMBL533954	CHEMBL:CHEMBL533954	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.072424374	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009320613	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.3231241306811969	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	TCMDC-124536	chembl:CHEMBL580851	CHEMBL:CHEMBL580851	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	FUSARIC ACID	chembl:CHEMBL24510	FUSARIC ACID	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	0.6886251965336985	BLU-285	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-123884	chembl:CHEMBL580955	CHEMBL:CHEMBL580955	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	1.193356164447602	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1060761035064535	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DINOTERB	chembl:CHEMBL1994620	DINOTERB	FALSE	FALSE	FALSE
MGLL	hgnc:17038	MGLL	DTC	9/2/20	NULL	3.500511415712967	URB597	iuphar.ligand:4339	URB597	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	1.544343271638073	AST-008	ncit:C157771	CAVROTOLIMOD	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.061484393	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.03443126	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	1.981421556063943	1H-PYRROLO[2,3-B]PYRIDINE	chembl:CHEMBL389685	CHEMBL:CHEMBL389685	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DICHLOROTRIPHENYLBISMUTHANE	chembl:CHEMBL205061	DICHLOROTRIPHENYLBISMUTHANE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	DNDI1417031	chembl:CHEMBL1333049	CHEMBL:CHEMBL1333049	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	DTRMWXHS 12	ncit:C130001	BTK INHIBITOR DTRMWXHS-12	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	NSC-367089	chembl:CHEMBL1543865	CHEMBL:CHEMBL1543865	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.1159109740302306	COTI-2	drugbank:DB17507	COTI-2	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.021036727	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	PENTAMIDINE ISETHIONATE	rxcui:7995	PENTAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.1232574442152452	DNDI1417132	chembl:CHEMBL1492017	CHEMBL:CHEMBL1492017	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	MOFEBUTAZONE	rxcui:30202	MOFEBUTAZONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	chembl:CHEMBL1336287	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TOLVAPTAN	rxcui:358257	TOLVAPTAN	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.1190650141398968	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	BP-897	iuphar.ligand:7625	BP 897	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.054553425	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005795549	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.006137659	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002188184	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,7-BIS[3-(PROPYLAMINO)PROPIONAMIDO]ANTHRAQUINONE	chembl:CHEMBL481160	CHEMBL:CHEMBL481160	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.007561589	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008345148	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	3',4'-DIMETHOXYFLAVONE	chembl:CHEMBL91153	3',4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011205222	MONTELUKAST SODIUM	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	1.944728564284981	DS-3201	ncit:C127114	VALEMETOSTAT	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	DTC	9/2/20	NULL	0.3201687270469177	RO-229735	chembl:CHEMBL2170369	CHEMBL:CHEMBL2170369	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	HALAZONE	rxcui:59838	HALAZONE	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.1291172243500684	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.000775823	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.025244073	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.003961647	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	TCMDC-125580	chembl:CHEMBL528807	CHEMBL:CHEMBL528807	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.9460841664089098	DIOSMETIN	rxcui:1314347	DIOSMETIN	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE BETA-1	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	0.315361389	M2698	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.6604738520213144	DIOSMETIN	rxcui:1314347	DIOSMETIN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.034318739	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.2237542808339254	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.3684748858645227	DIOSMETIN	rxcui:1314347	DIOSMETIN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.020778659	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.1666910197958555	AC-480	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.207267123	AC-480	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.054243462	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.039688338	Rogaratinib	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
FOLR1	hgnc:3791	FOLR1	DTC	9/2/20	NULL	1.166837138570989	LOMETREXOL	ncit:C979	LOMETREXOL	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GR-89696	iuphar.ligand:1649	GR 89696	FALSE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.1458546423213736	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.05751114	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01823183	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.000793767	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	NAFRONYL OXALATE	ncit:C87286	NAFRONYL OXALATE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	RM-1929	ncit:C121850	CETUXIMAB SAROTALOCAN SODIUM	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	ANISINDIONE	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.072125922	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
ADM	hgnc:259	ADM	DTC	9/2/20	NULL	13.12691780892362	NSC-106221	chembl:CHEMBL2063510	CHEMBL:CHEMBL2063510	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.003641814	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
PROLYL ENDOPEPTIDASE FAP	hgnc:3590	FAP	TTD	2020.06.01	NULL	2.692701089009974	RG7461	ncit:C129383	SIMLUKAFUSP ALFA	FALSE	FALSE	FALSE
KHSRP	hgnc:6316	KHSRP	DTC	9/2/20	NULL	52.50767123569449	GO-Y030	chembl:CHEMBL598509	CHEMBL:CHEMBL598509	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.024513385	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.01644462	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.019107595	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
PROTEIN-TYROSINE PHOSPHATASE SHP-2	hgnc:9644	PTPN11	TTD	2020.06.01	NULL	5.000730593875666	TNO155	ncit:C139559	BATOPROTAFIB	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.08334551	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.090530468	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.3697723326457359	N-ACETYLGLUCOSAMINE THIAZOLINE	chembl:CHEMBL257158	CHEMBL:CHEMBL257158	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	SJ000244629	chembl:CHEMBL592115	CHEMBL:CHEMBL592115	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.2983390411119005	XCT790	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	N-METHYL-D-ASPARTIC ACID (NMDA)	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
SSTR3	hgnc:11332	SSTR3	DTC	9/2/20	NULL	3.500511415712966	SOMATOSTATIN	rxcui:9939	SOMATOSTATIN	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	0.8078103267029924	CPI-0610	ncit:C188265	PELABRESIB	FALSE	FALSE	FALSE
RHOB	hgnc:668	RHOB	DTC	9/2/20	NULL	11.66837138570988	TRIMETHYL-[3-(TETRADECANE-1-SULFONYLAMINO)-PROPYL]-AMMONIUM IODIDE	chembl:CHEMBL2436861	TRIMETHYL-[3-(TETRADECANE-1-SULFONYLAMINO)-PROPYL]-AMMONIUM IODIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	TRANSPLATIN	chembl:CHEMBL1386	TRANSPLATIN	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.5303805175322676	ESTROPIPATE	rxcui:33747	ESTROPIPATE	TRUE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.040390516	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001350193	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	3,3',4'-TRIHYDROXYFLAVONE	chembl:CHEMBL122701	CHEMBL:CHEMBL122701	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004350623	ZIDOVUDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	1.750255707856483	IMX-110	ncit:C154569	CURCUMIN/DOXORUBICIN-ENCAPSULATING NANOPARTICLE IMX-110	FALSE	FALSE	FALSE
PRKG1	hgnc:9414	PRKG1	DTC	9/2/20	NULL	0.046343929	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	1.071585127259071	PHOMOPSIN A	chembl:CHEMBL446991	PHOMOPSIN A	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	NORADRENALINE	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.042344896	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	TCMDC-125738	chembl:CHEMBL527585	CHEMBL:CHEMBL527585	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.012794267	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	0.364636606	TP-0903	ncit:C127116	DUBERMATINIB	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	chembl:CHEMBL1336287	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006265084	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SC-514	chembl:CHEMBL193093	CHEMBL:CHEMBL193093	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TEBUCONAZOLE	chembl:CHEMBL487186	TEBUCONAZOLE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	XANTHOXYLIN	chembl:CHEMBL450288	XANTHOXYLIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	EMETINE HYDROCHLORIDE	rxcui:82015	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	MMV006389	chembl:CHEMBL586000	CHEMBL:CHEMBL586000	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.040893825	STANOLONE	ncit:C72098	STANOLONE	FALSE	FALSE	FALSE
HEPATOCYTE GROWTH FACTOR	hgnc:4893	HGF	TTD	2020.06.01	NULL	0.9723642821424906	MP0250	ncit:C117236	VEGF/HGF-TARGETING DARPIN MP0250	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	S-(+)-FLUOXETINE HCL	chembl:CHEMBL1257031	CHEMBL:CHEMBL1257031	FALSE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.8204323630577265	CHLORQUINALDOL	rxcui:2407	CHLORQUINALDOL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006978691	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	DTC	9/2/20	NULL	0.056459862	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	GNF-PF-4464	chembl:CHEMBL600692	CHEMBL:CHEMBL600692	FALSE	FALSE	FALSE
MAPK SIGNAL-INTEGRATING KINASE 1	hgnc:7110	MKNK1	TTD	2020.06.01	NULL	26.25383561784724	EFT508	ncit:C125062	TOMIVOSERTIB	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW642138X	chembl:CHEMBL373073	GW642138X	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.063645662	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	1.458546423213736	DNDI1417169	chembl:CHEMBL2094499	CHEMBL:CHEMBL2094499	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	0.062808219	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.3697723326457359	ABI-009	ncit:C74065	SIROLIMUS ALBUMIN-BOUND NANOPARTICLES	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006324701	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	PYRILAMINE	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.014039484	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.03070624	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	PT-103	chembl:CHEMBL398765	CHEMBL:CHEMBL398765	FALSE	FALSE	FALSE
HEPATOCYTE GROWTH FACTOR	hgnc:4893	HGF	TTD	2020.06.01	NULL	9.723642821424907	Ficlatuzumab	ncit:C78844	FICLATUZUMAB	FALSE	TRUE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002060822	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	A-23187	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	DTC	9/2/20	NULL	0.212152207	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	SEP-363856	drugbank:DB15665	SEP-363856	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.03729238	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	IOFETAMINE HYDROCHLORIDE	chembl:CHEMBL1255865	IOFETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	CONICASTEROL E	chembl:CHEMBL1950810	CONICASTEROL E	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006811217	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
MCOLN3	hgnc:13358	MCOLN3	DTC	9/2/20	NULL	1.093909817410302	BUTACLAMOL HYDROCHLORIDE	ncit:C81089	BUTACLAMOL HYDROCHLORIDE	FALSE	FALSE	FALSE
GLUCAGON	hgnc:4191	GCG	TTD	2020.06.01	NULL	0.6731752722524935	JNJ-64565111	ncit:C169932	EFINOPEGDUTIDE	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.1093909817410302	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.018874073	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.2586584789935689	TETRAHYDROZOLINE HYDROCHLORIDE	rxcui:57983	TETRAHYDROZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	NORDEFRIN	ncit:C81340	NORDEFRIN	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.031555091	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.036873365	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	1,2-BIS(3-FLUOROBENZYLIDENE)HYDRAZINE	iuphar.ligand:1424	3,3'-DIFLUOROBENZALDAZINE	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	2.386712328895204	MAHANINE	chembl:CHEMBL590522	MAHANINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	GYKI-52466	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	ALPHA-NAPHTHOFLAVONE	drugbank:DB07453	ALPHA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.080781033	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	ROFECOXIB	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.00944043	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	chembl:CHEMBL1336287	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DNDI1417472	chembl:CHEMBL1563896	CHEMBL:CHEMBL1563896	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
CD40L RECEPTOR	hgnc:11919	CD40	TTD	2020.06.01	NULL	2.187819634820604	ASKP-1240	chembl:CHEMBL3990028	BLESELUMAB	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.012996948	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.011205222	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	NCG-C00093820-01	chembl:CHEMBL544115	CHEMBL:CHEMBL544115	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.001417211	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	TRIADIMENOL	chembl:CHEMBL520275	TRIADIMENOL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1293292394967844	GNF-PF-4464	chembl:CHEMBL600692	CHEMBL:CHEMBL600692	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	SJ000117462	chembl:CHEMBL590427	CHEMBL:CHEMBL590427	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW561436X	chembl:CHEMBL1885746	GW561436X	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	3.281729452230906	BGB-324	ncit:C121854	BEMCENTINIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	GNF-PF-4242	chembl:CHEMBL584514	CHEMBL:CHEMBL584514	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004520289	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.1325951293830669	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	METHOCARBAMOL	rxcui:6845	METHOCARBAMOL	TRUE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
EPAS1	hgnc:3374	EPAS1	DTC	9/2/20	NULL	8.751278539282415	NEOPETROFORMYNE A	chembl:CHEMBL2177350	NEOPETROFORMYNE A	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	FIDUXOSIN HYDROCHLORIDE	ncit:C81371	FIDUXOSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	Pegmusirudin	ncit:C175734	PEGMUSIRUDIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	TDR78834	chembl:CHEMBL1507526	CHEMBL:CHEMBL1507526	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.048618214	ZOXAZOLAMINE	ncit:C152966	ZOXAZOLAMINE	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1060761035064535	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	2-STYRYL-QUINOLINE	chembl:CHEMBL127579	CHEMBL:CHEMBL127579	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	NSC-158389	chembl:CHEMBL192626	CHEMBL:CHEMBL192626	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	JNJ-16259685	iuphar.ligand:1385	JNJ16259685	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.023060023	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.055155117	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.033615667	Salirasib	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.045579576	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.030386384	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007749066	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003483789	ISOPRENALINE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00747866	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TRICLABENDAZOLE	rxcui:2118525	TRICLABENDAZOLE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	PENTAMIDINE ISETHIONATE	rxcui:7995	PENTAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.005737289	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.2344092465879218	TDR77593	chembl:CHEMBL1510164	CHEMBL:CHEMBL1510164	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.015447976	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.039778539	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.005818669	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003789252	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	2,3,4-TRIHYDROXYBENZOPHENONE	chembl:CHEMBL1527	CHEMBL:CHEMBL1527	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.00777661	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.078958904	HYMECROMONE	rxcui:5556	HYMECROMONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002796829	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	3',4' DICHLOROBENZAMIL	iuphar.ligand:4597	3,4-DICHLOROBENZAMIL	FALSE	FALSE	FALSE
CYTOTOXIC T-LYMPHOCYTE PROTEIN 4	hgnc:2505	CTLA4	TTD	2020.06.01	NULL	0.9723642821424907	Tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
DCLK1	hgnc:2700	DCLK1	DTC	9/2/20	NULL	0.2548916079402645	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	TEROXIRONE	ncit:C2320	TEROXIRONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	TRIPHENYLSTANNANOL	chembl:CHEMBL506538	TRIPHENYLSTANNANOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001044139	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.031555091	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	DOMPERIDONE	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1A	hgnc:7463	MTNR1A	TTD	2020.06.01	NULL	2.500365296937833	Neu-P11	chembl:CHEMBL4297523	PIROMELATINE	FALSE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	DTC	9/2/20	NULL	0.2324817828272369	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.011611604	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1415301111474245	DNDI1417346	chembl:CHEMBL1490332	CHEMBL:CHEMBL1490332	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2083637747448194	GNF-PF-4464	chembl:CHEMBL600692	CHEMBL:CHEMBL600692	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	BW-373U86	iuphar.ligand:9002	BW373U86	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2447910080918158	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.014832675	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
P2Y PURINOCEPTOR 12	hgnc:18124	P2RY12	TTD	2020.06.01	NULL	4.375639269641208	Cangrelor	rxcui:1656052	CANGRELOR	TRUE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.2333674277141978	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.1458546423213736	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.1875273972703375	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1981421556063943	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	1.810609352954982	BETAINE ALDEHYDE CHLORIDE	chembl:CHEMBL1256576	BETAINE ALDEHYDE CHLORIDE	FALSE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	0.3671865121377238	Oxytocin	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	GNF-PF-3416	chembl:CHEMBL579550	CHEMBL:CHEMBL579550	FALSE	FALSE	FALSE
RARB	hgnc:9865	RARB	DTC	9/2/20	NULL	1.235474617310459	AC-55649	iuphar.ligand:4055	AC55649	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	1.579178082276526	CER-002	chembl:CHEMBL3544958	CER-002	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.01351201	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DNDI1417905	chembl:CHEMBL1449731	CHEMBL:CHEMBL1449731	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.009250823	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	2.386712328895204	GNF-PF-2976	chembl:CHEMBL579956	CHEMBL:CHEMBL579956	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	MMV006389	chembl:CHEMBL586000	CHEMBL:CHEMBL586000	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	L-694247	iuphar.ligand:15	L-694,247	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.014330696	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.066011799	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	ASARININ	chembl:CHEMBL43469	ASARININ	FALSE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.070197421	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	1.109316997937207	PF-00337210	chembl:CHEMBL3545136	PF-00337210	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.7192831676122533	SCHISANHENOL	chembl:CHEMBL490125	SCHISANHENOL	FALSE	FALSE	FALSE
IAPP	hgnc:5329	IAPP	DTC	9/2/20	NULL	0.3977853881492008	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	TRICLABENDAZOLE	rxcui:2118525	TRICLABENDAZOLE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.021309932	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
MYELIN BASIC PROTEIN	hgnc:6925	MBP	TTD	2020.06.01	NULL	7.501095891	NBI-5788	chembl:CHEMBL2108869	TIPLIMOTIDE	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1651184630053286	PECTOLINARIGENIN	chembl:CHEMBL78010	PECTOLINARIGENIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	1-(4-HYDROXYPHENYL)MALEIMIDE	chembl:CHEMBL565893	CHEMBL:CHEMBL565893	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.052455216	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-1030061A	chembl:CHEMBL518968	GSK-1030061A	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	4-CHLORO-BENZOIC ACID	chembl:CHEMBL618	4-CHLORO-BENZOIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	IRL-2500	iuphar.ligand:3887	IRL 2500	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	TCMDC-125606	chembl:CHEMBL536166	CHEMBL:CHEMBL536166	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
MAP KINASE P38	hgnc:6874	MAPK12	TTD	2020.06.01	NULL	0.108040476	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	RAC-ARISTOYUNNOLIN D	chembl:CHEMBL2333543	CHEMBL:CHEMBL2333543	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	PROTRIPTYLINE HYDROCHLORIDE	rxcui:203199	PROTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.011176601	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	HARMOL	chembl:CHEMBL486817	HARMOL	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	GNF-PF-2968	chembl:CHEMBL582473	CHEMBL:CHEMBL582473	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.073643298	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.004449803	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.029987248	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	1,8-DINITRO-NAPHTHALENE	chembl:CHEMBL167529	CHEMBL:CHEMBL167529	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.061484393	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2734774543525755	DIFLUFENICAN	chembl:CHEMBL1425995	DIFLUFENICAN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GALLIC ACID METHYL ESTER	chembl:CHEMBL65675	GALLIC ACID METHYL ESTER	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005903055	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.010650643	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-138263	chembl:CHEMBL535307	CHEMBL:CHEMBL535307	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	BUTACLAMOL HYDROCHLORIDE	ncit:C81089	BUTACLAMOL HYDROCHLORIDE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2134458180312784	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	1.154014752432846	Rizatriptan	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	CUCURBITACIN B	iuphar.ligand:12432	CUCURBITACIN B	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	OXYFLUORFEN	chembl:CHEMBL1871400	OXYFLUORFEN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	GNF-PF-3889	chembl:CHEMBL598270	CHEMBL:CHEMBL598270	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.1065064325267636	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	(R)-NIPHATENONE A	chembl:CHEMBL1946013	CHEMBL:CHEMBL1946013	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.032412143	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DESACETOXYMATRICARIN	chembl:CHEMBL517040	DESACETOXYMATRICARIN	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.5097832158805291	GNF-PF-3947	chembl:CHEMBL584508	CHEMBL:CHEMBL584508	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	0.7001022831425933	DITHIOLETHIONE	chembl:CHEMBL368700	DITHIOLETHIONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.005732279	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.041508041	Dapiprazole	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	DTC	9/2/20	NULL	1.944728564284981	6BIO	chembl:CHEMBL409450	6BIO	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.053038052	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.021129848	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.033529803	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.01117898	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BITERTANOL	chembl:CHEMBL1566634	BITERTANOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001914661	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.008468979	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	5.250767123569449	CP-80794	chembl:CHEMBL60550	TERLAKIREN	FALSE	FALSE	FALSE
S100A4	hgnc:10494	S100A4	DTC	9/2/20	NULL	0.1166837138570988	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005795549	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.2035181055647073	TALAROFLAVONE	chembl:CHEMBL408995	TALAROFLAVONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE	chembl:CHEMBL457504	CHEMBL:CHEMBL457504	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005953251	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
S100A4	hgnc:10494	S100A4	DTC	9/2/20	NULL	0.5303805175322677	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.072424374	L-655240	chembl:CHEMBL362223	CHEMBL:CHEMBL362223	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.033615667	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.027276712	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.036212187	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	3.938075342677087	Tak-220	iuphar.ligand:800	TAK-220	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00399693	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	NSC-353263	chembl:CHEMBL1383812	CHEMBL:CHEMBL1383812	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	1-(4-HYDROXYPHENYL)MALEIMIDE	chembl:CHEMBL565893	CHEMBL:CHEMBL565893	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	SODIUM LAURYL SULFATE	rxcui:9871	SODIUM DODECYL SULFATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	4-HYDROXYDERRICIN	chembl:CHEMBL458094	CHEMBL:CHEMBL458094	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	DIPHENHYDRAMINE HYDROCHLORIDE	rxcui:1362	DIPHENHYDRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV7.1	hgnc:6294	KCNQ1	TTD	2020.06.01	NULL	1.432027397337122	Indapamide	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	2,4-HEXADIENAL	chembl:CHEMBL1576086	2,4-HEXADIENAL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002951527	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	ANIRACETAM	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.024275391	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001392481	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	LEVOMEPROMAZINE MALEATE	rxcui:160372	LEVOMEPROMAZINE MALEATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2035181055647073	RACEPINEPHRINE HYDROCHLORIDE	rxcui:314610	RACEPINEPHRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	TRANSPLATIN	chembl:CHEMBL1386	TRANSPLATIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	chembl:CHEMBL224214	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.014484875	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.017679351	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FIPRONIL	rxcui:1433761	FIPRONIL	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	SCH-53020	chembl:CHEMBL66279	CHEMBL:CHEMBL66279	FALSE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.8975670296699914	Tegaserod	rxcui:139778	TEGASEROD	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.007946076	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	TRANSPLATIN	chembl:CHEMBL1386	TRANSPLATIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	DIETHYLCARBAMAZINE CITRATE	rxcui:203175	DIETHYLCARBAMAZINE CITRATE	TRUE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	0.9723642821424906	REL-CISAPRIDE	chembl:CHEMBL74656	REL-CISAPRIDE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010093747	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	ACETOCHLOR	chembl:CHEMBL1517425	ACETOCHLOR	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.1232574442152452	NSC-121858	chembl:CHEMBL483838	CHEMBL:CHEMBL483838	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	TIOPRONIN	rxcui:6765	TIOPRONIN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.1419126249613365	LAS-34273	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
MARK4	hgnc:13538	MARK4	DTC	9/2/20	NULL	0.086646322	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CALCIUM PANTOTHENATE	rxcui:1918	CALCIUM PANTOTHENATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TETRADIFON	chembl:CHEMBL437926	TETRADIFON	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
PHOSPHO1	hgnc:16815	PHOSPHO1	DTC	9/2/20	NULL	0.9053046764774914	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	Umespirone	ncit:C152798	UMESPIRONE	FALSE	FALSE	FALSE
AKR1B10	hgnc:382	AKR1B10	DTC	9/2/20	NULL	2.625383561784725	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	DNDI1417111	chembl:CHEMBL2094456	CHEMBL:CHEMBL2094456	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	AMINOQUINOL	ncit:C73273	AMINOQUINOL	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.014484875	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003840807	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	N-METHYL-D-ASPARTIC ACID (NMDA)	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	PENTAMIDINE ISETHIONATE	rxcui:7995	PENTAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
CASPASE-3	hgnc:1504	CASP3	TTD	2020.06.01	NULL	2.333674277141977	PAC1	iuphar.ligand:5238	PAC1	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.088396753	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.042481935	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.00629362	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.025588534	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	CLOFOCTOL	rxcui:21264	CLOFOCTOL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	DTC	9/2/20	NULL	0.061197752	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	4-{[([4-(TRIFLUOROMETHYL)PHENYL]AMINO}CARBONYL)AMINO]BENZENESULFONAMIDE	chembl:CHEMBL1337519	CHEMBL:CHEMBL1337519	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.063415062	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
ABAT	hgnc:23	ABAT	DTC	9/2/20	NULL	0.08470687	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.032572997	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	L-733060	chembl:CHEMBL1256740	CHEMBL:CHEMBL1256740	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009084372	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.014993624	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.02832129	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.009092237	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	TCMDC-124495	chembl:CHEMBL532452	CHEMBL:CHEMBL532452	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1988926940746003	RETUSIN 7-METHYL ETHER	chembl:CHEMBL1290347	RETUSIN 7-METHYL ETHER	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.2051080907644316	RETUSIN 7-METHYL ETHER	chembl:CHEMBL1290347	RETUSIN 7-METHYL ETHER	FALSE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	DTC	9/2/20	NULL	4.773424657790408	HL010183	chembl:CHEMBL2348411	CHEMBL:CHEMBL2348411	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	HARMOL	chembl:CHEMBL486817	HARMOL	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.082429625	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.3684748858645227	ANDROGRAPHOLIDE	ncit:C61637	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.1446492320542548	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1635752997996713	NSC-45174	iuphar.ligand:7028	AMI-1	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	DNDI1417132	chembl:CHEMBL1492017	CHEMBL:CHEMBL1492017	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.012137696	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	3',4' DICHLOROBENZAMIL	iuphar.ligand:4597	3,4-DICHLOROBENZAMIL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	4-PHENYLAZO-PHENYLAMINE	chembl:CHEMBL83761	CHEMBL:CHEMBL83761	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	CIANIDANOL	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	BETA-CCM	chembl:CHEMBL453066	BETA-CCM	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	TCMDC-123641	chembl:CHEMBL532849	CHEMBL:CHEMBL532849	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.093763699	CLOROPHENE	rxcui:21290	CLOROPHENE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.095468493	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	PROPICONAZOLE	ncit:C97997	PROPICONAZOLE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000389812	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.093098708	TCMDC-124327	chembl:CHEMBL581929	CHEMBL:CHEMBL581929	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	HAPLAMINE	chembl:CHEMBL1488010	HAPLAMINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.4907258993990139	BENZHYDRYL 4-HYDROXYBENZOATE	chembl:CHEMBL2071180	CHEMBL:CHEMBL2071180	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.015930725	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	2-MERCAPTOBENZIMIDAZOLE	chembl:CHEMBL70141	2-MERCAPTOBENZIMIDAZOLE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.031861451	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.002741629	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.008621949	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.079557078	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	U-50488	iuphar.ligand:1652	U50488	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003608031	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001914661	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.024861587	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.028536778	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.017578732	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.024309107	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.00777661	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.059667808	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.085239726	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	0.9053046764774912	SALERMIDE	chembl:CHEMBL597845	SALERMIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005085489	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	NORADRENALINE	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	BERGAMOTTIN	chembl:CHEMBL1078442	BERGAMOTTIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.000994897	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.3500511415712966	QUINOXYFEN	chembl:CHEMBL1869863	QUINOXYFEN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-124064	chembl:CHEMBL537045	CHEMBL:CHEMBL537045	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.051177067	NSC-172033	chembl:CHEMBL238624	CHEMBL:CHEMBL238624	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	HYDROXYPROGESTERONE CAPROATE	rxcui:12488	HYDROXYPROGESTERONE CAPROATE (USP)	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.000659926	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.006614723	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.4861821410712453	SJ000189154	chembl:CHEMBL604664	CHEMBL:CHEMBL604664	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	GNF-PF-3029	chembl:CHEMBL601554	CHEMBL:CHEMBL601554	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007003824	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.3750547945406749	DIHYDROXANTHOHUMOL	chembl:CHEMBL510279	DIHYDROXANTHOHUMOL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.003590023	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
FZD1	hgnc:4038	FZD1	DTC	9/2/20	NULL	26.25383561784724	TCMDC-124051	chembl:CHEMBL464249	CHEMBL:CHEMBL464249	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.007661998	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ETOCRYLENE	ncit:C80797	ETOCRYLENE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	DICLOFENAC SODIUM	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.100589408	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	LAWSONE	drugbank:DB04744	LAWSONE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DICHLORISONE ACETATE	chembl:CHEMBL1385514	DICHLORISONE ACETATE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	OLEANDEROLIDE	chembl:CHEMBL498230	OLEANDEROLIDE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.01644462	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	2.019525817	GNF-PF-1656	chembl:CHEMBL579028	CHEMBL:CHEMBL579028	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009144492	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.005235062	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.019024519	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1017590527823536	PORFIROMYCIN	ncit:C763	PORFIROMYCIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	GNF-PF-1549	chembl:CHEMBL227959	CHEMBL:CHEMBL227959	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	L-694247	iuphar.ligand:15	L-694,247	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005527705	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.038981196	NSC-45174	iuphar.ligand:7028	AMI-1	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.1438566335224507	TCMDC-125528	chembl:CHEMBL375673	CHEMBL:CHEMBL375673	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.047197907	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	NORETHINDRONE ACETATE	rxcui:31983	NORETHINDRONE ACETATE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.3125456621172291	GNF-PF-1500	chembl:CHEMBL577673	CHEMBL:CHEMBL577673	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.056826484	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
MCOLN3	hgnc:13358	MCOLN3	DTC	9/2/20	NULL	3.281729452230906	ARECOLINE HYDROBROMIDE	ncit:C72704	ARECOLINE HYDROBROMIDE	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.096167896	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.005663036	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.033211683	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005412046	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.006189023	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	CYCLOBENZAPRINE HYDROCHLORIDE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.026816992	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011311433	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013964806	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.018860514	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.050294704	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.053038052	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DICHLORODIMETHYLSTANNANE	chembl:CHEMBL1076891	DICHLORODIMETHYLSTANNANE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.009144492	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	SJ000200944	chembl:CHEMBL600173	CHEMBL:CHEMBL600173	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.033148782	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NITROSCANATE	ncit:C75226	NITROSCANATE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1033615575505797	TRIPHENYLSTANNYL ACETATE	chembl:CHEMBL474376	TRIPHENYLSTANNYL ACETATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	BERGAMOTTIN	chembl:CHEMBL1078442	BERGAMOTTIN	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.00961679	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.045461187	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.074850565	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.022315202	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.030996264	GLAFENINE	ncit:C72119	GLAFENINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003409146	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.061055432	SJ000014858	chembl:CHEMBL591628	CHEMBL:CHEMBL591628	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.010518364	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003162351	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	DINOSEB	chembl:CHEMBL1892987	DINOSEB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	0.7955707762984016	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	DTC	9/2/20	NULL	0.03729238	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00479785	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SJ000012773	chembl:CHEMBL589715	CHEMBL:CHEMBL589715	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.037721028	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	THIOGUANOSINE	chembl:CHEMBL283078	THIOGUANOSINE	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.064268875	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.3977853881492008	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ISATIN	drugbank:DB02095	ISATIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008103036	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.3697723326457359	CEP-5214	chembl:CHEMBL150894	CEP-5214	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	TRANILAST	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010629083	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.056157937	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	DTC	9/2/20	NULL	0.4861821410712453	NSC-79888	chembl:CHEMBL1939433	CHEMBL:CHEMBL1939433	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CGP-53353	iuphar.ligand:5163	CGP53353	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.022466607	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	3-CHLOROEVODIAMINE	chembl:CHEMBL2171782	CHEMBL:CHEMBL2171782	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.013720322	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.082171629	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	DTC	9/2/20	NULL	1.166837138570989	LOMETREXOL	ncit:C979	LOMETREXOL	FALSE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008027468	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	MECAMYLAMINE	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	TRIOXSALEN	rxcui:10844	TRIOXSALEN	TRUE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.100976291	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.002035181	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.007903021	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV020490	chembl:CHEMBL581187	CHEMBL:CHEMBL581187	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	DNDI1417185	chembl:CHEMBL1549738	CHEMBL:CHEMBL1549738	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.042619863	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.189216833	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PYRROLNITRIN	ncit:C81509	PYRROLNITRIN	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.2917092846427472	BERBERRUBINE	chembl:CHEMBL203135	BERBERRUBINE	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	1.166837138570988	KOLAVENIC ACID	chembl:CHEMBL1517738	KOLAVENIC ACID	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.032173818	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002016269	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.047561296	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.010620484	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.045382603	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005412046	MONTELUKAST SODIUM	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	TRIPHENYLSTANNYL ACETATE	chembl:CHEMBL474376	TRIPHENYLSTANNYL ACETATE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TRICYCLAZOLE	drugbank:DB02891	TRICYCLAZOLE	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.095399112	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.034727296	IPRONIAZID	rxcui:5981	IPRONIAZID	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	EPIANDROSTERONE	ncit:C61747	EPIANDROSTERONE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.013613604	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.05853698	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.020117882	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
MAPKAPK3	hgnc:6888	MAPKAPK3	DTC	9/2/20	NULL	1.875273972703374	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.056459862	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	TDR77593	chembl:CHEMBL1510164	CHEMBL:CHEMBL1510164	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	BENOXACOR	chembl:CHEMBL2269059	BENOXACOR	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.5000730593875666	CYTARABINE HYDROCHLORIDE	ncit:C71603	CYTARABINE HYDROCHLORIDE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.056157937	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002949869	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	METHIOTHEPIN MESYLATE	chembl:CHEMBL1256737	METHIOTHEPIN MESYLATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	CUCURBITACIN B	iuphar.ligand:12432	CUCURBITACIN B	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.7001022831425933	OCTADECYLAMINE	chembl:CHEMBL55860	OCTADECYLAMINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.015088411	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.005618798	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	DTC	9/2/20	NULL	0.044124093	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
SENP1	hgnc:17927	SENP1	DTC	9/2/20	NULL	5.834185692854944	DNDI1417884	chembl:CHEMBL1346025	CHEMBL:CHEMBL1346025	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.042863405	ALPHA-NAPHTHOFLAVONE	drugbank:DB07453	ALPHA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.091159151	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.013186256	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.5527123287967841	DYRENE	chembl:CHEMBL464135	DYRENE	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.013680998	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.00825852	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.028536778	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.016921583	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.2243917574174978	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	NALED	chembl:CHEMBL1887067	NALED	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000180366	chembl:CHEMBL609036	CHEMBL:CHEMBL609036	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.053579256	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	TYRPHOSTIN AG-112	iuphar.ligand:5913	AG 112	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.058602312	DNDI1417031	chembl:CHEMBL1333049	CHEMBL:CHEMBL1333049	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SJ000040829	chembl:CHEMBL589711	CHEMBL:CHEMBL589711	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.029698909	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TCMDC-125614	chembl:CHEMBL580609	CHEMBL:CHEMBL580609	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DIFENOCONAZOLE	chembl:CHEMBL466426	DIFENOCONAZOLE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	PENTAERYTHRITOL TETRANITRATE	rxcui:7992	PENTAERYTHRITOL TETRANITRATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.1093909817410302	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.03443126	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.018699313	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.3302369260106572	TCMDC-124032	chembl:CHEMBL536375	CHEMBL:CHEMBL536375	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	1.875273972703375	GNF-PF-3696	chembl:CHEMBL598885	CHEMBL:CHEMBL598885	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	NORARMEPAVINE	chembl:CHEMBL453038	NORARMEPAVINE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.016161179	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.033338204	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
SRD5A1	hgnc:11284	SRD5A1	DTC	9/2/20	NULL	8.751278539282415	BEXLOSTERIDE	ncit:C166644	BEXLOSTERIDE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.02234369	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.034184682	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001174668	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE	chembl:CHEMBL1214407	CHEMBL:CHEMBL1214407	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.024275391	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CASP9	hgnc:1511	CASP9	DTC	9/2/20	NULL	2.625383561784725	20(S)-PROTOPANAXADIOL	chembl:CHEMBL375563	CHEMBL:CHEMBL375563	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.038049037	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	DNDI1417132	chembl:CHEMBL1492017	CHEMBL:CHEMBL1492017	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-124315	chembl:CHEMBL532363	CHEMBL:CHEMBL532363	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.029465584	LAS38096	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.6177373086552295	GNF-PF-3352	chembl:CHEMBL600306	CHEMBL:CHEMBL600306	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	0.7143900848393808	NSC-663284	drugbank:DB17038	NSC-663284	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	THIOGUANOSINE	chembl:CHEMBL283078	THIOGUANOSINE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.078136416	1-O-ACETYLGEOPYXIN A	chembl:CHEMBL1902074	CHEMBL:CHEMBL1902074	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.00996918	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	0.729273212	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	3.088686543276147	NSC-640558	chembl:CHEMBL1288281	CHEMBL:CHEMBL1288281	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	0.7242437411819932	20(S)-PROTOPANAXADIOL	chembl:CHEMBL375563	CHEMBL:CHEMBL375563	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	CLOFOCTOL	rxcui:21264	CLOFOCTOL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	GNF-PF-5297	chembl:CHEMBL602575	CHEMBL:CHEMBL602575	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010569177	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	TCMDC-124377	chembl:CHEMBL531269	CHEMBL:CHEMBL531269	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.008081833	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	TETRAHYDROGAMBOGIC ACID	chembl:CHEMBL1605700	TETRAHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001727453	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	TRIPHENYLSTANNANOL	chembl:CHEMBL506538	TRIPHENYLSTANNANOL	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.002117672	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1232574442152452	2,3,4-TRIHYDROXYBENZOPHENONE	chembl:CHEMBL1527	CHEMBL:CHEMBL1527	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012325744	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.028199609	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	0.4102161815288632	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.038159645	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DIELDRIN	chembl:CHEMBL1873703	DIELDRIN	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.023630815	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	AG-99	chembl:CHEMBL296407	CHEMBL:CHEMBL296407	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002338872	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	GEOPYXIN A	chembl:CHEMBL1899565	GEOPYXIN A	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.007108118	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.032412143	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	2-NITRO-ETHANOL	chembl:CHEMBL324774	CHEMBL:CHEMBL324774	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.5303805175322676	LXR-623	chembl:CHEMBL456237	LXR-623	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	METHYL PARATHIONE	chembl:CHEMBL346516	METHYL PARATHIONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	AMIDATE	chembl:CHEMBL23731	AMIDATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003401858	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.004191225	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.090530468	BOLDINE	chembl:CHEMBL388342	BOLDINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.005903055	Amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1286952726365061	SALAGEN	chembl:CHEMBL611494	SALAGEN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	1.184383561707394	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	NULL	PEG-3350	NULL	NULL	NULL	NULL	NULL
TNFRSF8	hgnc:11923	TNFRSF8	FDA	10-Apr-24	NULL	1.276228120312019	Brentuximab Vedotin	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.01875274	Sodium Chloride	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.054243462	Carisoprodol	rxcui:2101	CARISOPRODOL	TRUE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	FDA	10-Apr-24	NULL	5.000730593875666	Dinutuximab	rxcui:1606274	DINUTUXIMAB	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.025298806	Cevimeline	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.1298891063344329	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.00402481	Doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.1766118064547324	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.3125456621172291	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.637458239	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.4102161815288633	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
CYB5R	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.003541833	Paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	0.070690956	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.066213961	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.002643159	Risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1500219178162699	Succimer	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.001362243	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.038382801	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	0.42006137	Telaprevir	rxcui:1102261	TELAPREVIR	TRUE	FALSE	FALSE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.027244868	Vortioxetine	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	NULL	ARQ736	NULL	NULL	NULL	NULL	NULL
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.1108075556053025	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	MyCancerGenome	20-Jun-17	inhibitor	2.800409132570373	GSK1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.3777530304726222	BAFETINIB	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.6269572684859045	GSK1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	MyCancerGenome	20-Jun-17	inhibitor	0.3409589041278863	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.092606122	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.172722603	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.070860555	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.021933029	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.038382801	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.1764963739014941	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenome	20-Jun-17	inhibitor	0.2357246744587856	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
AKT1S1	hgnc:28426	AKT1S1	MyCancerGenome	20-Jun-17	inhibitor	1.009762908	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
RPTOR	hgnc:30287	RPTOR	MyCancerGenome	20-Jun-17	inhibitor	0.5048814541893702	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
MAPKAP1	hgnc:18752	MAPKAP1	MyCancerGenome	20-Jun-17	inhibitor	1.346350544504987	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.2016939996249468	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
TNFRSF10A	hgnc:11904	TNFRSF10A	MyCancerGenome	20-Jun-17	antibody	15.75230137070834	DULANERMIN	ncit:C1685	DULANERMIN	FALSE	TRUE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	antibody	3.000438356	ONARTUZUMAB	ncit:C82348	ONARTUZUMAB	FALSE	TRUE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenome	20-Jun-17	antibody	1.544343271638073	MM-111	drugbank:DB17983	MM-111	FALSE	TRUE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenome	20-Jun-17	antibody	0.3431873936973496	AV203	ncit:C102535	ANTI-ERBB3 MONOCLONAL ANTIBODY AV-203	FALSE	TRUE	TRUE
PARP1	hgnc:270	PARP1	MyCancerGenome	20-Jun-17	other/unknown	0.900131507	MK4827	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	MyCancerGenome	20-Jun-17	other/unknown	4.200613699	INIPARIB	ncit:C62526	INIPARIB	FALSE	FALSE	TRUE
PSMD11	hgnc:9556	PSMD11	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD4P1	hgnc:9562	PSMD4P1	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD7	hgnc:9565	PSMD7	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD13	hgnc:9558	PSMD13	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC3IP	hgnc:17928	PSMC3IP	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD14	hgnc:16889	PSMD14	MyCancerGenome	20-Jun-17	other/unknown	0.2692701089009974	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA1	hgnc:9530	PSMA1	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD9	hgnc:9567	PSMD9	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD3	hgnc:9560	PSMD3	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD6	hgnc:9564	PSMD6	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD10P3	hgnc:30152	PSMD10P3	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD10	hgnc:9555	PSMD10	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSME2P2	hgnc:30160	PSME2P2	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	MyCancerGenome	20-Jun-17	other/unknown	5.104912481248077	ERISMODEGIB	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
PSMF1	hgnc:9571	PSMF1	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	5.104912481248077	LDE225	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1110098757625676	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
RAF-1	hgnc:9829	RAF1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1835932560688619	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1375060601009582	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
AKT3	hgnc:393	AKT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.546954909	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.049864835	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	0.2053085874318455	6-THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	0.4234489615781814	GANCICLOVIR	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1147708660889497	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.066011799	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.028290771	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	0.3860858179095183	GSK269962A	iuphar.ligand:8037	GSK269962A	FALSE	FALSE	FALSE
ACTB	hgnc:132	ACTB	NCI	14-Sep-17	NULL	1.500219178	ENVIRONMENTAL ESTROGEN	ncit:C1894	ENVIRONMENTAL ESTROGEN	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.2734774543525755	VORICONAZOLE	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
ABCG4	hgnc:13884	ABCG4	NCI	14-Sep-17	NULL	2.386712328895204	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.092606122	SKI-758	chembl:CHEMBL219557	CHEMBL:CHEMBL219557	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	1.544343271638073	RADIOSENSITIZERS	ncit:C798	RADIOSENSITIZING AGENT	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.1108075556053025	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
TOLL-LIKE RECEPTOR 3	hgnc:11849	TLR3	TTD	2020.06.01	NULL	5.250767123569449	Poly-ICLC	ncit:C1198	POLY ICLC	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	NCI	14-Sep-17	NULL	0.1483267549030917	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
ADK	hgnc:257	ADK	NCI	14-Sep-17	NULL	0.5527123287967842	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
ADRB2	hgnc:286	ADRB2	NCI	14-Sep-17	NULL	0.029074015	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	1.544343271638073	CEPHALOSPORINS	ncit:C357	CEPHALOSPORIN ANTIBIOTIC	FALSE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE 1	hgnc:1437	CALCA	TTD	2020.06.01	NULL	1.944728564284981	Cizolirtine	ncit:C77311	CIZOLIRTINE	FALSE	FALSE	FALSE
ALOX5AP	hgnc:436	ALOX5AP	NCI	14-Sep-17	NULL	1.666910197958555	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
ALDH3A1	hgnc:405	ALDH3A1	NCI	14-Sep-17	NULL	0.1046664542904209	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	NCI	14-Sep-17	NULL	0.021307461	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.1835932560688619	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
ATP7B	hgnc:870	ATP7B	NCI	14-Sep-17	NULL	0.2134458180312784	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.009334697	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Oxitropium bromide	rxcui:54270	OXITROPIUM BROMIDE	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1166837138570988	ANTHRACYCLINE	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1272913242077442	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1272913242077442	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	NULL	OPIOIDS	NULL	NULL	NULL	NULL	NULL
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	0.4922594178346359	DONEPEZIL	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.060984519	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
RIBONUCLEOTIDE REDUCTASE	hgnc:581	APBB1	TTD	2020.06.01	NULL	0.061412481	Clofarabine	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1829535583125243	INTERLEUKINS	ncit:C593	RECOMBINANT INTERLEUKIN	FALSE	FALSE	FALSE
CBL	hgnc:1541	CBL	NCI	14-Sep-17	NULL	1.750255707856483	FLT3-LIGAND	ncit:C1714	RECOMBINANT FLT3 LIGAND	FALSE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	6.563458904461812	LT-BETA	ncit:C1608	RECOMBINANT LYMPHOTOXIN BETA	FALSE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	NCI	14-Sep-17	NULL	0.7160136986685613	BENZODIAZEPINE	ncit:C1012	BENZODIAZEPINE	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.6168664383892681	HKI-272	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
CCL8	hgnc:10635	CCL8	NCI	14-Sep-17	NULL	0.8975670296699914	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.1041818873724097	URACIL	rxcui:10995	URACIL	TRUE	FALSE	TRUE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	0.2917092846427472	Hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
CCL28	hgnc:17700	CCL28	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.1136529680426287	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	0.7721716358190367	TENIDAP	ncit:C152558	TENIDAP	FALSE	FALSE	FALSE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
CD2	hgnc:1639	CD2	NCI	14-Sep-17	NULL	0.3889457128569963	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
CD244	hgnc:18171	CD244	NCI	14-Sep-17	NULL	3.500511415712966	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.053145416	Oxazepam	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
CD44	hgnc:1681	CD44	NCI	14-Sep-17	NULL	0.4251633298436802	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.1574442915613028	PROSTAGLANDIN E1	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
CD86	hgnc:1705	CD86	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
CDA	hgnc:1712	CDA	NCI	14-Sep-17	NULL	0.3704244884352345	CYTOSINE ARABINOSIDE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.082171629	Lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
CDH17	hgnc:1756	CDH17	NCI	14-Sep-17	NULL	4.375639269641208	SQUALAMINE	ncit:C143004	SQUALAMINE	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	0.093931433	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.052455216	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	1.129197231	ART621	chembl:CHEMBL2108739	PLACULUMAB	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.1190650141398968	CANCER DRUG	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.3889457128569963	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
CGA	hgnc:1885	CGA	NCI	14-Sep-17	NULL	0.6250913242344582	9-CIS-RETINOIC ACID	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	NULL	RED CELLS	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	0.1842374429322613	Trapidil	rxcui:10735	TRAPIDIL	FALSE	FALSE	FALSE
COL1A2	hgnc:2198	COL1A2	NCI	14-Sep-17	NULL	0.5303805175322677	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1000146118775133	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.077789143	INTERLEUKIN 1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	1.400204566285186	TRP-2	ncit:C38682	RECOMBINANT TYROSINASE-RELATED PROTEIN-2	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1400204566285186	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	MART1	ncit:C28724	MART-1 ANTIGEN	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.07699072	Lamotrigine	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.105015342	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.1682938180631233	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.1187956362798518	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	0.100589408	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	2.187819634820604	IL-13	iuphar.ligand:4980	IL-13	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	NULL	ISOFLAVONES	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.068436196	Adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.001174668	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.2187819634820604	Nicardipine	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.3409589041278864	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.018354192	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.7501095890813501	POLYETHYLENE GLYCOL	rxcui:1310594	POLYETHYLENE GLYCOL 4000	TRUE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.038894571	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.3889457128569963	ANTICONVULSANT	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.092064882	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	Nalfurafine hcl	chembl:CHEMBL490665	NALFURAFINE HYDROCHLORIDE	FALSE	FALSE	FALSE
EIF4E	hgnc:3287	EIF4E	NCI	14-Sep-17	NULL	0.1724389859957126	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
EPO	hgnc:3415	EPO	NCI	14-Sep-17	NULL	0.9376369863516875	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.2917092846427472	HERCEPTIN	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE XII	hgnc:1371	CA12	TTD	2020.06.01	NULL	0.9376369863516875	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.057291513	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.012841201	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.3621218705909966	AS101	iuphar.ligand:437	AS101	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.2011788169949981	VITAMIN K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.1591141552596803	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	NULL	BISPHOSPHONATES	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.9460841664089098	REBAMIPIDE	ncit:C29852	REBAMIPIDE	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	1.514644363	NABILONE	rxcui:31447	NABILONE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.179119736	BAY 43-9006	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FOLH1	hgnc:3788	FOLH1	NCI	14-Sep-17	NULL	3.889457128569962	PSMA PEPTIDE	ncit:C29340	PSMA PEPTIDE	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.1750255707856483	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.2210849315187136	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
GADD45A	hgnc:4095	GADD45A	NCI	14-Sep-17	NULL	0.1000146118775133	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.6731752722524935	TD-8954	iuphar.ligand:8426	TD-8954	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	NULL	BISPHOSPHONATES	NULL	NULL	NULL	NULL	NULL
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1315981735230438	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1250182648468916	PROTEASE INHIBITOR	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.5834185692854944	TOPOISOMERASE INHIBITORS	ncit:C1748	TOPOISOMERASE INHIBITOR	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.1848861663228679	BGT226	ncit:C74073	PI3K INHIBITOR BGT226	FALSE	FALSE	TRUE
BLOOD GROUP RH(D) POLYPEPTIDE	hgnc:10009	RHD	TTD	2020.06.01	NULL	26.25383561784724	Roledumab	ncit:C152241	ROLEDUMAB	FALSE	FALSE	FALSE
GZMA	hgnc:4708	GZMA	NCI	14-Sep-17	NULL	0.1724389859957126	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
GUCA2B	hgnc:4683	GUCA2B	NCI	14-Sep-17	NULL	3.750547945406749	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
H2AFX	hgnc:4739	H2AX	NCI	14-Sep-17	NULL	0.1000146118775133	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.061055432	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.1495945049449986	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.027584802	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
HIST3H2A	hgnc:20507	H2AC25	NCI	14-Sep-17	NULL	0.600087671	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	0.1875273972703375	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	NULL	VIRAL VECTOR	NULL	NULL	NULL	NULL	NULL
HPSE	hgnc:5164	HPSE	NCI	14-Sep-17	NULL	0.2430910705356226	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.3777530304726222	Flumatinib	hemonc:38662	FLUMATINIB	FALSE	FALSE	FALSE
HP	hgnc:5141	HP	NCI	14-Sep-17	NULL	0.326134604	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	NCI	14-Sep-17	NULL	0.3889457128569963	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.7343730242754476	DIFFERENTIATION INDUCER	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	NCI	14-Sep-17	NULL	0.096167896	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.1121958787087489	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	2.386712328895204	IMIQUIMOD	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	2.917092846427472	PF-3463275	iuphar.ligand:9057	PF-03463275	FALSE	FALSE	FALSE
IFI27	hgnc:5397	IFI27	NCI	14-Sep-17	NULL	1.250182648468916	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	NCI	14-Sep-17	NULL	1.009762908	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	9.546849315580817	CL 246,738	ncit:C1052	CL 246738	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	NULL	RBC	NULL	NULL	NULL	NULL	NULL
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.1562728310586145	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	1.093909817410302	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	0.087512785	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	2.763561643983921	MT-3995	chembl:CHEMBL3545392	MT-3995	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.6863747873946993	DNCB	ncit:C439	DINITROCHLOROBENZENE	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.1530835896084387	IFOSFAMIDE	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
IL7	hgnc:6023	IL7	NCI	14-Sep-17	NULL	3.500511415712967	DNA VACCINE	ncit:C39619	DNA VACCINE	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.3241214273808302	ALPHA INTERFERON	ncit:C225	RECOMBINANT INTERFERON ALFA	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	2.625383561784724	Cal-1	ncit:C165547	ANTI-HIV-1 LENTIVIRAL VECTOR-EXPRESSING SH5/C46 CAL-1	FALSE	FALSE	FALSE
IL8RB	hgnc:6027	CXCR2	NCI	14-Sep-17	NULL	0.100589408	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
LOH19CR1	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.1795134059339982	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	1.381780822	IL-13	iuphar.ligand:4980	IL-13	FALSE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	NCI	14-Sep-17	NULL	NULL	ANTIINFLAMMATORY AGENTS	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	1.944728564284981	MLN-591RL	chembl:CHEMBL2109557	MLN-591RL	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1442518440541058	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1442518440541058	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	NULL	BISPHOSPHONATES	NULL	NULL	NULL	NULL	NULL
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.1630673019742065	INTERLEUKINS	ncit:C593	RECOMBINANT INTERLEUKIN	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.2853677784548614	HMG-COA REDUCTASE INHIBITOR	ncit:C1655	HMG-COA REDUCTASE INHIBITOR	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.5357925636295356	Emicizumab	rxcui:1989794	EMICIZUMAB	TRUE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	11.66837138570988	RV-B7.1	ncit:C2237	RECOMBINANT VACCINIA-B7.1 VACCINE	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.05853698	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
MTAP	hgnc:7413	MTAP	NCI	14-Sep-17	NULL	26.25383561784724	L-ALANOSINE	ncit:C994	ALANOSINE	FALSE	FALSE	FALSE
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	1.367387271762877	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
MT1H	hgnc:7400	MT1H	NCI	14-Sep-17	NULL	0.5770073762164232	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	0.069225671	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MYB	hgnc:7545	MYB	NCI	14-Sep-17	NULL	0.1166837138570988	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1666910197958555	MNU	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.4375639269641209	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.057700738	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	NULL	L6	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.1215455352678113	Herbimycin A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
NAT1	hgnc:7645	NAT1	NCI	14-Sep-17	NULL	0.020688602	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NAT2	hgnc:7646	NAT2	NCI	14-Sep-17	NULL	0.031032903	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.006295884	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2958178661165888	BENZODIAZEPINE	ncit:C1012	BENZODIAZEPINE	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	0.7721716358190367	Tepoxalin	ncit:C76817	TEPOXALIN	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.052824619	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.3697723326457359	TIRAPAZAMINE	ncit:C1464	TIRAPAZAMINE	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.3697723326457359	IDOXIFENE	ncit:C1406	IDOXIFENE	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.1013661606866689	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	0.3947945205691315	T3D-959	chembl:CHEMBL3545176	DB959	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.2625383561784725	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.1186614039224734	VP-16	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.1154014752432846	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.018699313	TYROSINE KINASE INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.016206071	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
ENDOTHELIN B RECEPTOR	hgnc:3180	EDNRB	TTD	2020.06.01	NULL	1.250182648468916	ET-1	iuphar.ligand:989	ENDOTHELIN-1	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.060772768	UROKINASE-TYPE PLASMINOGEN ACTIVATOR	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.8334550989792777	TOPOISOMERASE-II INHIBITOR	ncit:C1968	TOPOISOMERASE-II INHIBITOR	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.005556367	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.032055965	TYROSINE KINASE INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.01468746	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.073437302	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
PLAT	hgnc:9051	PLAT	NCI	14-Sep-17	NULL	1.301843088488293	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
LEUKOTRIENE B4 RECEPTOR 2	hgnc:19260	LTB4R2	TTD	2020.06.01	NULL	6.563458904461812	Biomed 101	ncit:C2206	BIOMED 101	FALSE	FALSE	FALSE
POSTN	hgnc:16953	POSTN	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
PRDX1	hgnc:9352	PRDX1	NCI	14-Sep-17	NULL	0.8751278539282418	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	NULL	OPIOIDS	NULL	NULL	NULL	NULL	NULL
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.072927321	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
PTGDS	hgnc:9592	PTGDS	NCI	14-Sep-17	NULL	1.193356164447602	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	NCI	14-Sep-17	NULL	0.036718651	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
IMMUNOGLOBULIN E	hgnc:5522	IGHE	TTD	2020.06.01	NULL	17.50255707856483	MEMP1972A	ncit:C152116	QUILIZUMAB	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	NCI	14-Sep-17	NULL	0.1458546423213736	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.074797252	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.2243917574174978	TNX-102	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
PTHR1	hgnc:9608	PTH1R	NCI	14-Sep-17	NULL	2.500365296937833	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.2991890098899971	VITAMIN K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
CYCLIC PYRANOPTERIN MONOPHOSPHATE SYNTHASE	hgnc:7190	MOCS1	TTD	2020.06.01	NULL	26.25383561784724	ALXN1101	chembl:CHEMBL2338675	FOSDENOPTERIN	FALSE	FALSE	FALSE
PXN	hgnc:9718	PXN	NCI	14-Sep-17	NULL	1.009762908	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
RALBP1	hgnc:9841	RALBP1	NCI	14-Sep-17	NULL	0.1000146118775133	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.4167275494896388	ALPHA INTERFERON	ncit:C225	RECOMBINANT INTERFERON ALFA	FALSE	FALSE	FALSE
PYY	hgnc:9748	PYY	NCI	14-Sep-17	NULL	4.039051633514962	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
LYSOSOMAL ALPHA-GLUCOSIDASE	hgnc:4065	GAA	TTD	2020.06.01	NULL	0.729273212	GZ402666	chembl:CHEMBL4594320	AVALGLUCOSIDASE ALFA	FALSE	FALSE	FALSE
PZP	hgnc:9750	PZP	NCI	14-Sep-17	NULL	8.751278539282415	ESTRAMUSTINE PHOSPHATE	rxcui:105556	ESTRAMUSTINE PHOSPHATE	FALSE	FALSE	FALSE
SDHB	hgnc:10681	SDHB	NCI	14-Sep-17	NULL	0.2625383561784725	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	AVX901	ncit:C99903	HER2 ECD+TM VIRUS-LIKE REPLICON PARTICLES VACCINE AVX901	FALSE	FALSE	FALSE
SERPINA5	hgnc:8723	SERPINA5	NCI	14-Sep-17	NULL	1.093909817410302	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR B	hgnc:12681	VEGFB	TTD	2020.06.01	NULL	7.001022831425934	Aflibercept	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
SLC1A3	hgnc:10941	SLC1A3	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	NULL	VIRAL VECTOR	NULL	NULL	NULL	NULL	NULL
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.5834185692854944	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
TFAP2A	hgnc:11742	TFAP2A	NCI	14-Sep-17	NULL	1.750255707856483	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	NULL	ISOFLAVONES	NULL	NULL	NULL	NULL	NULL
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.8334550989792776	OPIATE	ncit:C1657	OPIATE	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	NULL	TAXANES	NULL	NULL	NULL	NULL	NULL
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	1.129197231	KW-2149	ncit:C1140	MITOMYCIN C ANALOG KW-2149	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR-ALPHA	hgnc:10477	RXRA	TTD	2020.06.01	NULL	0.4667348554283955	Bexarotene	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
TNFAIP1	hgnc:11894	TNFAIP1	NCI	14-Sep-17	NULL	3.500511415712966	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.074797252	Amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	NCI	14-Sep-17	NULL	NULL	NEW AGENTS	NULL	NULL	NULL	NULL	NULL
TNFRSF1B	hgnc:11917	TNFRSF1B	NCI	14-Sep-17	NULL	0.2500365296937833	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
TNFRSF8	hgnc:11923	TNFRSF8	NCI	14-Sep-17	NULL	0.1875273972703375	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	NCI	14-Sep-17	NULL	0.2917092846427472	TOPOISOMERASE INHIBITORS	ncit:C1748	TOPOISOMERASE INHIBITOR	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.019318496	R-FLURBIPROFEN	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.011591097	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	2.625383561784724	Alkavervir	chembl:CHEMBL1201658	ALKAVERVIR	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.055681518	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	NULL	KINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
TYK2	hgnc:12440	TYK2	NCI	14-Sep-17	NULL	0.056459862	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
GLIAL CELL LINE-DERIVED NEUROTROPHIC FACTOR	hgnc:4232	GDNF	TTD	2020.06.01	NULL	2.019525817	Liatermin	ncit:C1459	LIATERMIN	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.16256245	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	NCI	14-Sep-17	NULL	0.2125816649218401	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	NULL	ISOFLAVONES	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.035560536	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.01305187	tamsulosin	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.2430910705356227	atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.065634589	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
SORT1	hgnc:11186	SORT1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
TPH2	hgnc:20692	TPH2	PharmGKB	4/5/24	NULL	0.4375639269641209	mirtazapine	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
TPH2	hgnc:20692	TPH2	PharmGKB	4/5/24	NULL	0.1682938180631234	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	1.071585127259071	ALD-518	iuphar.ligand:9195	CLAZAKIZUMAB	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.3387591692625452	lomitapide	rxcui:1364478	LOMITAPIDE MESYLATE	TRUE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.3889457128569963	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.5645986154375752	inclisiran	rxcui:2588243	INCLISIRAN	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
SLC28A1	hgnc:11001	SLC28A1	PharmGKB	4/5/24	NULL	0.7778914257139926	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.022666813	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.2323348284765243	oxiconazole	rxcui:32638	OXICONAZOLE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.2323348284765243	ethambutol	rxcui:142435	ETHAMBUTOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.011914607	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.005736662	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CLCN6	hgnc:2024	CLCN6	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	NULL	Vitamin K antagonists	NULL	NULL	NULL	NULL	NULL
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	NULL	Enzyme inhibitors	NULL	NULL	NULL	NULL	NULL
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.8950171233357017	Measles vaccines	wikidata:Q6804161	MEASLES VACCINE	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	1.036335616	Measles vaccines	wikidata:Q6804161	MEASLES VACCINE	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	1.009762908	PRUVANSERIN	ncit:C72834	PRUVANSERIN	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	PharmGKB	4/5/24	NULL	0.086818239	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
KCNJ6	hgnc:6267	KCNJ6	PharmGKB	4/5/24	NULL	3.938075342677087	Analgesics	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
TCF7L2	hgnc:11641	TCF7L2	PharmGKB	4/5/24	NULL	1.500219178162699	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
IL22RA2	hgnc:14901	IL22RA2	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	NULL	Dopamine agonists	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.3860858179095183	Suronacrine maleate	ncit:C96776	SURONACRINE MALEATE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	4.150804050252529	nemonapride	ncit:C73036	NEMONAPRIDE	FALSE	FALSE	FALSE
SLC22A11	hgnc:18120	SLC22A11	PharmGKB	4/5/24	NULL	0.3125456621172291	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.010417155	yohimbine	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	NULL	ivacaftor / tezacaftor	NULL	NULL	NULL	NULL	NULL
CHRNA4	hgnc:1958	CHRNA4	PharmGKB	4/5/24	NULL	0.1241316104862754	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
HLA-DRA	hgnc:4947	HLA-DRA	PharmGKB	4/5/24	NULL	0.7895890411382631	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
CTPS1	hgnc:2519	CTPS1	PharmGKB	4/5/24	NULL	NULL	ara-CTP	NULL	NULL	NULL	NULL	NULL
CTPS1	hgnc:2519	CTPS1	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.1004611056805379	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.4688184931758437	tebentafusp	rxcui:2590743	TEBENTAFUSP	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
PPCDC	hgnc:28107	PPCDC	PharmGKB	4/5/24	NULL	NULL	FEC100	NULL	NULL	NULL	NULL	NULL
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.596678082	bucindolol	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
SUGCT	hgnc:16001	SUGCT	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	3.889457128569962	quinapril	rxcui:35208	QUINAPRIL	TRUE	FALSE	FALSE
SOLUBLE GUANYLATE CYCLASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	1.050153425	Sodium nitroprusside	rxcui:9895	SODIUM NITROPRUSSIDE	TRUE	FALSE	FALSE
LAMB3	hgnc:6490	LAMB3	PharmGKB	4/5/24	NULL	1.750255707856483	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
STAT4	hgnc:11365	STAT4	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	NULL	corr-4a	NULL	NULL	NULL	NULL	NULL
ANKK1	hgnc:21027	ANKK1	PharmGKB	4/5/24	NULL	0.8824818695074707	naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.1888765152363111	inotuzumab ozogamicin	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.08334551	cilostazol	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	0.036162308	curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	2-hydroxymethyl olanzapine	NULL	NULL	NULL	NULL	NULL
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.2403097081725148	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
GGH	hgnc:4248	GGH	PharmGKB	4/5/24	NULL	0.6563458904461813	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
PHB2	hgnc:30306	PHB2	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
ABCB11	hgnc:42	ABCB11	PharmGKB	4/5/24	NULL	0.3977853881492006	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
IGF2BP2	hgnc:28867	IGF2BP2	PharmGKB	4/5/24	NULL	1.875273972703374	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	0.1620607136904151	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ENOSF1	hgnc:30365	ENOSF1	PharmGKB	4/5/24	NULL	0.4688184931758437	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	NULL	acetaminophen sulfate	NULL	NULL	NULL	NULL	NULL
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
ACP1	hgnc:122	ACP1	PharmGKB	4/5/24	NULL	0.2328499833068492	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
INTERLEUKIN-5	hgnc:6016	IL5	TTD	2020.06.01	NULL	17.50255707856483	Reslizumab	rxcui:1746889	RESLIZUMAB	TRUE	FALSE	FALSE
KCNN1	hgnc:6290	KCNN1	PharmGKB	4/5/24	NULL	1.280674908	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
UHRF1	hgnc:12556	UHRF1	PharmGKB	4/5/24	NULL	0.5147810905460245	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ARF1	hgnc:652	ARF1	PharmGKB	4/5/24	NULL	0.5147810905460245	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	0.4773424657790409	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
C18ORF21	hgnc:28802	C18orf21	PharmGKB	4/5/24	NULL	1.312691780892362	quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NEDD4L	hgnc:7728	NEDD4L	PharmGKB	4/5/24	NULL	2.059124362184098	amiloride	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	PharmGKB	4/5/24	NULL	0.015416228	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
TAFA5	hgnc:21592	TAFA5	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
APOC1	hgnc:607	APOC1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
AQP2	hgnc:634	AQP2	PharmGKB	4/5/24	NULL	NULL	thiazolidinediones	NULL	NULL	NULL	NULL	NULL
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.324566649	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	NULL	raloxifene 6-glucuronide	NULL	NULL	NULL	NULL	NULL
ADH1A	hgnc:249	ADH1A	PharmGKB	4/5/24	NULL	0.5966780822238011	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
SLC22A2	hgnc:10966	SLC22A2	PharmGKB	4/5/24	NULL	0.546954909	fampridine	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	23.33674277141977	SAR-650984	rxcui:2282018	ISATUXIMAB	TRUE	FALSE	FALSE
FPGS	hgnc:3824	FPGS	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.1493817104856173	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.789589041	Glucarpidase	rxcui:1242127	GLUCARPIDASE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	2.100306849	voxilaprevir	rxcui:1939323	VOXILAPREVIR	TRUE	FALSE	FALSE
CDH13	hgnc:1753	CDH13	PharmGKB	4/5/24	NULL	0.3106962795011509	perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.5016656487486736	calcipotriol	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.4039051633514962	amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
KLC1	hgnc:6387	KLC1	PharmGKB	4/5/24	NULL	0.5556367326528519	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.011532544	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.2019525816757481	lomitapide	rxcui:1364478	LOMITAPIDE MESYLATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.01305187	rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.002669701	flunitrazepam	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.010541895	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	NULL	egfr inhibitors	NULL	NULL	NULL	NULL	NULL
UGT1A	hgnc:12529	UGT1A	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
F13A1	hgnc:3531	F13A1	PharmGKB	4/5/24	NULL	NULL	photodynamic therapy	NULL	NULL	NULL	NULL	NULL
DKK1	hgnc:2891	DKK1	PharmGKB	4/5/24	NULL	0.9723642821424906	alendronate	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.09814518	Bazedoxifene	rxcui:1441386	BAZEDOXIFENE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.091159151	ramucirumab	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
ACTG1	hgnc:144	ACTG1	PharmGKB	4/5/24	NULL	0.037042449	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TOMM40	hgnc:18001	TOMM40	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	6beta-hydroxyprogesterone	NULL	NULL	NULL	NULL	NULL
RBFOX1	hgnc:18222	RBFOX1	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2983390411119005	3,4-methylenedioxymethamphetamine	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.027347745	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.024861587	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.5357925636295356	Apixaban	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
ZNF100	hgnc:12880	ZNF100	PharmGKB	4/5/24	NULL	NULL	antineoplastic agents	NULL	NULL	NULL	NULL	NULL
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	NULL	Beta blocking agents, non-selective	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.078136416	sulfamethoxazole	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
LILRB5	hgnc:6609	LILRB5	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	13.12691780892362	Arepanrix	ncit:C88320	AS03-ADJUVANTED H1N1 PANDEMIC INFLUENZA VACCINE	FALSE	FALSE	FALSE
DMPK	hgnc:2933	DMPK	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
IGFBP7	hgnc:5476	IGFBP7	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	NULL	Hepatitis vaccines	NULL	NULL	NULL	NULL	NULL
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.3768493150887165	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
CSPG4	hgnc:2466	CSPG4	PharmGKB	4/5/24	NULL	0.3333820395917111	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.2333674277141977	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
CDKN2B-AS1	hgnc:34341	CDKN2B-AS1	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
PTGS1	hgnc:9604	PTGS1	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
IL10	hgnc:5962	IL10	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
KL	hgnc:6344	KL	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	0.1905904582057876	Amphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
MMP10	hgnc:7156	MMP10	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
ALOX15	hgnc:433	ALOX15	PharmGKB	4/5/24	NULL	NULL	Antiinflammatory agents, non-steroids	NULL	NULL	NULL	NULL	NULL
DCK	hgnc:2704	DCK	PharmGKB	4/5/24	NULL	NULL	ara-CTP	NULL	NULL	NULL	NULL	NULL
DCTD	hgnc:2710	DCTD	PharmGKB	4/5/24	NULL	NULL	ara-CTP	NULL	NULL	NULL	NULL	NULL
RRM1	hgnc:10451	RRM1	PharmGKB	4/5/24	NULL	NULL	ara-CTP	NULL	NULL	NULL	NULL	NULL
SPECC1L	hgnc:29022	SPECC1L	PharmGKB	4/5/24	NULL	0.9376369863516874	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.072125922	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	4.118248724368195	Carbetocin	ncit:C96858	CARBETOCIN	TRUE	FALSE	FALSE
NALCN	hgnc:19082	NALCN	PharmGKB	4/5/24	NULL	0.4688184931758437	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.093763699	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	2.187819634820604	solithromycin	ncit:C152386	SOLITHROMYCIN	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.072919531	Chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
MISP	hgnc:27000	MISP	PharmGKB	4/5/24	NULL	0.9723642821424908	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
ADAMTS1	hgnc:217	ADAMTS1	PharmGKB	4/5/24	NULL	NULL	hmg coa reductase inhibitors	NULL	NULL	NULL	NULL	NULL
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	NULL	ethinyl estradiol / norelgestromin	NULL	NULL	NULL	NULL	NULL
CBR3	hgnc:1549	CBR3	PharmGKB	4/5/24	NULL	0.3241214273808303	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
CCNK	hgnc:1596	CCNK	PharmGKB	4/5/24	NULL	0.9723642821424908	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	NULL	Iodine (131I) compounds	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.040390516	nitroglycerin	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
IL4R	hgnc:6015	IL4R	PharmGKB	4/5/24	NULL	NULL	Hepatitis vaccines	NULL	NULL	NULL	NULL	NULL
PIK3R1	hgnc:8979	PIK3R1	PharmGKB	4/5/24	NULL	NULL	egfr inhibitors	NULL	NULL	NULL	NULL	NULL
CYP2R1	hgnc:20580	CYP2R1	PharmGKB	4/5/24	NULL	4.375639269641208	calcidiol	rxcui:1855064	CALCIFEDIOL ANHYDROUS	TRUE	FALSE	FALSE
C20ORF194	hgnc:17721	DNAAF9	PharmGKB	4/5/24	NULL	1.640864726115453	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.1848861663228679	Dihydroergocristine	rxcui:3416	DIHYDROERGOCRISTINE	TRUE	FALSE	FALSE
ALDH1A2	hgnc:15472	ALDH1A2	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
NECAB1	hgnc:20983	NECAB1	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
APBB1IP	hgnc:17379	APBB1IP	PharmGKB	4/5/24	NULL	3.000438356	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
TSPEAR	hgnc:1268	TSPEAR	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	NULL	Antihypertensives And Diuretics In Combination	NULL	NULL	NULL	NULL	NULL
NIPAL2	hgnc:25854	NIPAL2	PharmGKB	4/5/24	NULL	7.001022831425933	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.015299438	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
PRRC2A	hgnc:13918	PRRC2A	PharmGKB	4/5/24	NULL	0.7143900848393808	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
FCGR2A	hgnc:3616	FCGR2A	PharmGKB	4/5/24	NULL	1.750255707856483	margetuximab	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
UGT2B@	ncbigene:7362	UGT2B@	PharmGKB	4/5/24	NULL	NULL	clozapine N+ glucuronide	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	1.334940794127826	Eprosartan	rxcui:83515	EPROSARTAN	TRUE	FALSE	FALSE
CYP2A13	hgnc:2608	CYP2A13	PharmGKB	4/5/24	NULL	2.187819634820604	coumarin	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
SLC29A4	hgnc:23097	SLC29A4	PharmGKB	4/5/24	NULL	1.346350544504987	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
PROC	hgnc:9451	PROC	PharmGKB	4/5/24	NULL	NULL	ethinyl estradiol / norelgestromin	NULL	NULL	NULL	NULL	NULL
PROC	hgnc:9451	PROC	PharmGKB	4/5/24	NULL	NULL	estradiol / progesterone	NULL	NULL	NULL	NULL	NULL
NEDD4	hgnc:7727	NEDD4	PharmGKB	4/5/24	NULL	3.182283105193606	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Prifinium	rxcui:236174	PRIFINIUM	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.8899605294185507	nitroprusside	rxcui:7476	NITROPRUSSIDE	TRUE	FALSE	FALSE
RBMS3	hgnc:13427	RBMS3	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	amlodipine / atorvastatin / perindopril arginine	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	toluidine blue	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1312691780892362	acetaminophen / tramadol	wikidata:Q48564239	ACETAMINOPHEN/TRAMADOL	FALSE	FALSE	FALSE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.1221108633388244	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
C18ORF21	hgnc:28802	C18orf21	PharmGKB	4/5/24	NULL	2.019525816757481	dofetilide	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
KCNT2	hgnc:18866	KCNT2	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.054187483	Pilocarpine	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HNF1A	hgnc:11621	HNF1A	PharmGKB	4/5/24	NULL	2.187819634820604	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
IL21R	hgnc:6006	IL21R	PharmGKB	4/5/24	NULL	1.093909817410302	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.2822993077187876	Tolperisone	rxcui:10639	TOLPERISONE	FALSE	FALSE	FALSE
KIF6	hgnc:21202	KIF6	PharmGKB	4/5/24	NULL	4.375639269641208	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
ERCC2	hgnc:3434	ERCC2	PharmGKB	4/5/24	NULL	2.386712328895204	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
MARCH1	hgnc:26077	MARCHF1	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	2.651902587661338	ticagrelor	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	2.282942227638891	RG7813	ncit:C141459	CERGUTUZUMAB AMUNALEUKIN	FALSE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.1346350544504987	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	PharmGKB	4/5/24	NULL	0.03591496	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
MEX3C	hgnc:28040	MEX3C	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	5.250767123569449	AMD-070	ncit:C126660	MAVORIXAFOR	FALSE	FALSE	FALSE
PKLR	hgnc:9020	PKLR	PharmGKB	4/5/24	NULL	NULL	Bisphosphonates	NULL	NULL	NULL	NULL	NULL
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.013890918	pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.01090502	pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
MIR107	hgnc:31496	MIR107	PharmGKB	4/5/24	NULL	26.25383561784724	acetaminophen / tramadol	wikidata:Q48564239	ACETAMINOPHEN/TRAMADOL	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.039628431	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CASP1	hgnc:1499	CASP1	PharmGKB	4/5/24	NULL	0.1262203635473425	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
CYP2R1	hgnc:20580	CYP2R1	PharmGKB	4/5/24	NULL	1.093909817410302	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.1041818873724097	alendronate	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
ANKS1B	hgnc:24600	ANKS1B	PharmGKB	4/5/24	NULL	1.009762908	amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.073540156	naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
MGAT4A	hgnc:7047	MGAT4A	PharmGKB	4/5/24	NULL	0.6563458904461813	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	4.375639269641208	coumarin	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	PharmGKB	4/5/24	NULL	0.048083948	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NOTCH2	hgnc:7882	NOTCH2	PharmGKB	4/5/24	NULL	1.250182648468916	odevixibat	rxcui:2563966	ODEVIXIBAT	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	0.2778183663264259	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.2853677784548614	donepezil	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
PEAR1	hgnc:33631	PEAR1	PharmGKB	4/5/24	NULL	17.50255707856483	ticagrelor	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	PharmGKB	4/5/24	NULL	0.032817295	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
F12	hgnc:3530	F12	PharmGKB	4/5/24	NULL	NULL	Enzymes	NULL	NULL	NULL	NULL	NULL
AKT1	hgnc:391	AKT1	TALC	12-May-16	inhibitor	0.443726799	PERIFOSINE	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	2.625383561784725	Apratastat	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.1704794520639432	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.3174882446809434	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.1275696580070323	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.1562728310586145	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.1829535583125243	FK-228	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.192335792	FK-228	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.192335792	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.6269572684859045	GSK1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.070129236	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	TALC	12-May-16	inhibitor	0.03337352	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	NULL	PD325901	NULL	NULL	NULL	NULL	NULL
AURKC	hgnc:11391	AURKC	TALC	12-May-16	inhibitor	2.800409132570373	GSK1070916	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
NAIP	hgnc:7634	NAIP	TALC	12-May-16	inhibitor	NULL	AEG40826	NULL	NULL	NULL	NULL	NULL
MTOR	hgnc:3942	MTOR	TALC	12-May-16	inhibitor	0.1232574442152452	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	TALC	12-May-16	inhibitor	0.020542907	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
CI MAN-6-P RECEPTOR	hgnc:5467	IGF2R	TTD	2020.06.01	NULL	52.50767123569449	Juvidex	drugbank:DB11848	MANNOSE 6-PHOSPHATE	FALSE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	TALC	12-May-16	inhibitor	0.5048814541893702	AZD 8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
RAD51	hgnc:9817	RAD51	TALC	12-May-16	inhibitor	15.00219178162699	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
BIRC2	hgnc:590	BIRC2	TALC	12-May-16	inhibitor	NULL	AEG40826	NULL	NULL	NULL	NULL	NULL
RPTOR	hgnc:30287	RPTOR	TALC	12-May-16	inhibitor	0.06697407	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
XIAP	hgnc:592	XIAP	TALC	12-May-16	inhibitor	NULL	AEG40826	NULL	NULL	NULL	NULL	NULL
BIRC3	hgnc:591	BIRC3	TALC	12-May-16	inhibitor	NULL	AEG40826	NULL	NULL	NULL	NULL	NULL
BIRC6	hgnc:13516	BIRC6	TALC	12-May-16	inhibitor	NULL	AEG40826	NULL	NULL	NULL	NULL	NULL
TNFRSF9	hgnc:11924	TNFRSF9	TALC	12-May-16	antibody	78.76150685354175	BMS-663513	ncit:C62449	URELUMAB	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	TALC	12-May-16	inhibitor	0.009603891	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	TALC	12-May-16	inhibitor	0.596678082	YM155	chembl:CHEMBL2105734	SEPANTRONIUM BROMIDE	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	NULL	3196	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	NULL	7A-METHYL-19-NORTESTOSTERONE,MENT	NULL	NULL	NULL	NULL	NULL
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.988926940746003	ABARELIX	rxcui:301739	ABARELIX	TRUE	FALSE	TRUE
UNIPROT:Q9Y275	hgnc:11929	TNFSF13B	TdgClinicalTrial	Jan-14	NULL	19.69037671338543	BLISIBIMOD	ncit:C166445	BLISIBIMOD	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	NULL	ABX-0401	NULL	NULL	NULL	NULL	NULL
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.028360625	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:Q02763	hgnc:11724	TEK	TdgClinicalTrial	Jan-14	NULL	0.041021618	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.039068208	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P07949	hgnc:9967	RET	TdgClinicalTrial	Jan-14	NULL	0.016206071	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	NULL	ADL7445	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	NULL	ADX415	NULL	NULL	NULL	NULL	NULL
UNIPROT:P98170	hgnc:592	XIAP	TdgClinicalTrial	Jan-14	NULL	NULL	AEG35156, GEM 640	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.1151484018326633	AE37	ncit:C171846	BLARCAMESINE	FALSE	FALSE	FALSE
UNIPROT:P19320	hgnc:12663	VCAM1	TdgClinicalTrial	Jan-14	NULL	NULL	AGI-1067, SUCCINOBUCOL	NULL	NULL	NULL	NULL	NULL
UNIPROT:P24394	hgnc:6015	IL4R	TdgClinicalTrial	Jan-14	NULL	NULL	AIR645	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	NULL	ALACIZUMAB PEGO	NULL	NULL	NULL	NULL	NULL
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	NULL	ALB109564(A)	NULL	NULL	NULL	NULL	NULL
UNIPROT:P18405	hgnc:11284	SRD5A1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	LEVONORGESTREL	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P10523	hgnc:10521	SAG	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	B27PD	drugbank:DB16289	B27PD	FALSE	FALSE	FALSE
UNIPROT:P01374	hgnc:6709	LTA	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	BAMINERCEPT	ncit:C96762	BAMINERCEPT ALFA	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.063858524	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
UNIPROT:P19113	hgnc:4855	HDC	TdgClinicalTrial	Jan-14	NULL	NULL	BF-DERM1	NULL	NULL	NULL	NULL	NULL
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.729273212	BF-1	iuphar.ligand:8424	BF-1	FALSE	FALSE	FALSE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	0.6908904109959803	LY2606368	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
UNIPROT:P43088	hgnc:9600	PTGFR	TdgClinicalTrial	Jan-14	NULL	2.812910959055062	BIMATOPROST	rxcui:283810	BIMATOPROST	TRUE	FALSE	FALSE
UNIPROT:Q02156	hgnc:9401	PRKCE	TdgClinicalTrial	Jan-14	NULL	0.3750547945406749	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:P05129	hgnc:9402	PRKCG	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:Q9NPF7	hgnc:15488	IL23A	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	BRIAKINUMAB	ncit:C95321	BRIAKINUMAB	FALSE	FALSE	FALSE
UNIPROT:Q9BZL6	hgnc:17293	PRKD2	TdgClinicalTrial	Jan-14	NULL	0.1103102336884338	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
NEURAL CELL ADHESION MOLECULE	hgnc:7656	NCAM1	TTD	2020.06.01	NULL	1.640864726115453	IMGN901	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
UNIPROT:Q04759	hgnc:9410	PRKCQ	TdgClinicalTrial	Jan-14	NULL	0.1875273972703374	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:O94806	hgnc:9408	PRKD3	TdgClinicalTrial	Jan-14	NULL	0.093763699	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.024932417	BUDIODARONE	ncit:C83563	BUDIODARONE	FALSE	FALSE	FALSE
UNIPROT:P02647	hgnc:600	APOA1	TdgClinicalTrial	Jan-14	NULL	4.565884455277782	CER-001	drugbank:DB18538	CER-001	FALSE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.217423069	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TdgClinicalTrial	Jan-14	NULL	1.712206670729168	CONIVAPTAN	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.106290832	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.034981793	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1111665587205952	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	NULL	CYTOFAB	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01589	hgnc:6008	IL2RA	TdgClinicalTrial	Jan-14	NULL	1.029562181092049	DACLIZUMAB	rxcui:190353	DACLIZUMAB	TRUE	TRUE	FALSE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.1223004764806549	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.08334551	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.1829535583125243	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:P43115	hgnc:9595	PTGER3	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	DG041	drugbank:DB05027	DG041	FALSE	FALSE	FALSE
UNIPROT:Q14957	hgnc:4587	GRIN2C	TdgClinicalTrial	Jan-14	NULL	0.2117244807890907	DIMIRACETAM	ncit:C79121	DIMIRACETAM	FALSE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	DIMIRACETAM	ncit:C79121	DIMIRACETAM	FALSE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.2430910705356226	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.096521454	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.018305561	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.030945115	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	NULL	DRF 10945	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31213	hgnc:11285	SRD5A2	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
UNIPROT:O43497	hgnc:1394	CACNA1G	TdgClinicalTrial	Jan-14	NULL	0.1750255707856483	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:O60939	hgnc:10589	SCN2B	TdgClinicalTrial	Jan-14	NULL	2.100306849	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	NULL	EP42675	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	NULL	EP42675	NULL	NULL	NULL	NULL	NULL
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	1.712206670729168	EVP-6124	ncit:C166844	ENCENICLINE	FALSE	FALSE	FALSE
UNIPROT:P18564	hgnc:6161	ITGB6	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	GLPG0187	ncit:C96223	INTEGRIN RECEPTOR ANTAGONIST GLPG0187	FALSE	FALSE	FALSE
UNIPROT:P23458	hgnc:6190	JAK1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	GLPG0634	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	1.166837138570989	SCH-527123	iuphar.ligand:8497	NAVARIXIN	FALSE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TdgClinicalTrial	Jan-14	NULL	7.876150685354174	HEMATIDE	rxcui:1248798	PEGINESATIDE	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.04464938	FACTOR IX	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
UNIPROT:P16422	hgnc:11529	EPCAM	TdgClinicalTrial	Jan-14	NULL	NULL	IGN101	NULL	NULL	NULL	NULL	NULL
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.8899605294185507	ILEPATRIL	ncit:C87731	ILEPATRIL	FALSE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	NULL	MPI-676	NULL	NULL	NULL	NULL	NULL
UNIPROT:P42701	hgnc:5971	IL12RB1	TdgClinicalTrial	Jan-14	NULL	NULL	INCELL-1001+ AD-1001	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q99665	hgnc:5972	IL12RB2	TdgClinicalTrial	Jan-14	NULL	NULL	INCELL-1001+ AD-1001	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20711	hgnc:2719	DDC	TdgClinicalTrial	Jan-14	NULL	NULL	IPX066	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.093098708	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	4.773424657790408	Sampatrilat	ncit:C132269	SAMPATRILAT	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.1389091831632129	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.8514757497680189	ISTRADEFYLLINE	rxcui:2199015	ISTRADEFYLLINE	TRUE	FALSE	FALSE
UNIPROT:P13591	hgnc:7656	NCAM1	TdgClinicalTrial	Jan-14	NULL	NULL	LORVOTUZUMAB	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	1.369765336583334	sparsentan	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	0.1093909817410302	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TdgClinicalTrial	Jan-14	NULL	0.056097939	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.2112984757975633	LOFEXIDINE	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.049723174	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.2616661357260523	LOFEXIDINE	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TdgClinicalTrial	Jan-14	NULL	NULL	LU AA24493	NULL	NULL	NULL	NULL	NULL
UNIPROT:P49069	hgnc:1471	CAMLG	TdgClinicalTrial	Jan-14	NULL	0.6035364509849942	CYCLOSPORINE A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.2	hgnc:1389	CACNA1B	TTD	2020.06.01	NULL	0.2344092465879218	Cilnidipine	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.2401265452851882	OBATOCLAX	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
UNIPROT:P04792	hgnc:5246	HSPB1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	OGX-427	ncit:C71740	APATORSEN	FALSE	FALSE	TRUE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.101562227	IUPHAR.LIGAND:150	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
UNIPROT:P28074	hgnc:9542	PSMB5	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.1442518440541057	OPC-34712	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	NULL	COMBRETASTATIN A1 DI-PHOSPHATE	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q99250	hgnc:10588	SCN2A	TdgClinicalTrial	Jan-14	NULL	0.053771297	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P35225	hgnc:5973	IL13	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	QAX576	iuphar.ligand:8714	DECTREKUMAB	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.8899605294185507	QUINAPRIL	rxcui:35208	QUINAPRIL	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.172950169	ROPINIROL	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
UNIPROT:P05019	hgnc:5464	IGF1	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT HUMAN INSULIN-LIKE GROWTH FACTOR BINDING PROTEIN-3	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.2631963470460877	ROCURONIUM	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.1666910197958555	ROCURONIUM	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
UNIPROT:P21452	hgnc:11527	TACR2	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	SAREDUTANT	ncit:C152301	SAREDUTANT	FALSE	FALSE	FALSE
UNIPROT:P02647	hgnc:600	APOA1	TdgClinicalTrial	Jan-14	NULL	0.326134604	RVX-208	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.035617739	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:8427	ncit:C152177	RELENOPRIDE	FALSE	FALSE	FALSE
UNIPROT:P32970	hgnc:11937	CD70	TdgClinicalTrial	Jan-14	NULL	8.078103267029922	SGN-70	chembl:CHEMBL2108673	VORSETUZUMAB	FALSE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.358239472	DEXTROAMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	NULL	SOU-003	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00797	hgnc:9958	REN	TdgClinicalTrial	Jan-14	NULL	NULL	SPP676	NULL	NULL	NULL	NULL	NULL
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:170	iuphar.ligand:170	ORG 12962	FALSE	FALSE	FALSE
UNIPROT:P09601	hgnc:5013	HMOX1	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	STANNSOPORFIN	ncit:C152424	STANNSOPORFIN	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.08178765	TAPENTADOL	rxcui:787390	TAPENTADOL	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.046303061	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
UNIPROT:P36897	hgnc:11772	TGFBR1	TdgClinicalTrial	Jan-14	NULL	NULL	TG-C	NULL	NULL	NULL	NULL	NULL
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:180	iuphar.ligand:180	LY215840	FALSE	FALSE	FALSE
UNIPROT:P37173	hgnc:11773	TGFBR2	TdgClinicalTrial	Jan-14	NULL	NULL	TG-C	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q03167	hgnc:11774	TGFBR3	TdgClinicalTrial	Jan-14	NULL	NULL	TG-C	NULL	NULL	NULL	NULL	NULL
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:186	iuphar.ligand:186	GLEMANSERIN	FALSE	FALSE	FALSE
UNIPROT:P39086	hgnc:4579	GRIK1	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.085796848	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.2128689374420047	TIOTROPIUM	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
UNIPROT:P48058	hgnc:4574	GRIA4	TdgClinicalTrial	Jan-14	NULL	0.5303805175322677	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P49356	hgnc:3785	FNTB	TdgClinicalTrial	Jan-14	NULL	2.333674277141978	TIPIFARNIB	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.2302968036653267	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.100976291	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.014369915	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5U5	hgnc:11914	TNFRSF18	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	TRX518	ncit:C95023	ANTI-HUMAN GITR MONOCLONAL ANTIBODY TRX518	FALSE	FALSE	FALSE
UNIPROT:Q9UQB9	hgnc:11391	AURKC	TdgClinicalTrial	Jan-14	NULL	0.1438566335224506	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	ETODOLAC	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	NULL	XP21279	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	NULL	XP21279	NULL	NULL	NULL	NULL	NULL
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.276356164	IUPHAR.LIGAND:169	iuphar.ligand:169	[125I]DOI	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	NULL	XP21279	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	NULL	XP21279	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	NULL	XP21279	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	ZYD1	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT HUMAN THROMBIN	NULL	NULL	NULL	NULL	NULL
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.061412481	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
UNIPROT:P12259	hgnc:3542	F5	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT HUMAN THROMBIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00451	hgnc:3546	F8	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT HUMAN THROMBIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	NULL	RFIX	NULL	NULL	NULL	NULL	NULL
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.050246575	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
UNIPROT:P08397	hgnc:4982	HMBS	TdgClinicalTrial	Jan-14	NULL	NULL	RAAV5-PBGD	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23458	hgnc:6190	JAK1	TdgClinicalTrial	Jan-14	NULL	0.8468979231563628	ASP015K	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:8423	rxcui:1791685	PIMAVANSERIN	TRUE	FALSE	FALSE
UNIPROT:O95749	hgnc:4249	GGPS1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	ZOLEDRONATE	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.076263865	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.2206204673768676	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:2941	rxcui:1300701	LORCASERIN	FALSE	FALSE	FALSE
UNIPROT:P08246	hgnc:3309	ELANE	TdgClinicalTrial	Jan-14	NULL	1.521961485092594	ALPHA-1-PROTEINASE INHIBITOR	rxcui:535	ALPHA 1-ANTITRYPSIN	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.078194596	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:186	iuphar.ligand:186	GLEMANSERIN	FALSE	FALSE	FALSE
UNIPROT:P05981	hgnc:5155	HPN	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	BENTIROMIDE	rxcui:18896	BENTIROMIDE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.201952582	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.159436249	CHLOROPROCAINE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	CARPHENAZINE	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.080225625	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.2206204673768676	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.038608582	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.596678082	DOBUTAMINE	rxcui:3616	DOBUTAMINE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.7143900848393808	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.596678082	DISOPYRAMIDE	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.2631963470460877	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.1884246575443582	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	PHENTERMINE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	PHENMETRAZINE	rxcui:8133	PHENMETRAZINE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.098884503	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
UNIPROT:Q9NSA0	hgnc:18120	SLC22A11	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	1.036335616	PROPARACAINE	rxcui:34905	PROPARACAINE	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.5933070196123671	RAMIPRIL	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.049442252	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.2234368988752957	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.029443554	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.1280674908187671	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	SALICYLIC ACID	rxcui:9525	SALICYLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.061055432	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.092118721	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TEND	1-Aug-11	NULL	0.729273212	ESOMEPRAZOLE	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.047886613	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.060169218	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:792	hgnc:74	ABCG2	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:10372	iuphar.ligand:10372	COMPOUND 14 [PMID: 30925062]	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.045898314	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.1816874437221263	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.4605936073306534	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P07355	hgnc:537	ANXA2	TEND	1-Aug-11	NULL	1.250182648468916	ANISTREPLASE	rxcui:40028	ANISTREPLASE	TRUE	FALSE	FALSE
UNIPROT:P48443	hgnc:10479	RXRG	TEND	1-Aug-11	NULL	1.988926940746004	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NCBIGENE:768	hgnc:1383	CA9	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11788	ncit:C76198	ZOSUQUIDAR	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.596678082	BEVANTOLOL	ncit:C79556	BEVANTOLOL	FALSE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TEND	1-Aug-11	NULL	1.944728564284981	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
UNIPROT:P05023	hgnc:799	ATP1A1	TEND	1-Aug-11	NULL	0.5834185692854944	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TEND	1-Aug-11	NULL	2.282942227638891	BOSENTAN	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.073266518	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.073266518	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.014977128	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.041639708	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:11888	ncit:C175551	ZILURGISERTIB	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TEND	1-Aug-11	NULL	0.2112984757975633	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.2983390411119005	DESVENLAFAXINE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.596678082	DOBUTAMINE	rxcui:3616	DOBUTAMINE	TRUE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:11875	iuphar.ligand:11875	FIDRISERTIB	FALSE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TEND	1-Aug-11	NULL	0.4375639269641208	DOLASETRON	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TEND	1-Aug-11	NULL	0.9376369863516874	INTERFERON ALFA-2B, RECOMBINANT	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P17181	hgnc:5432	IFNAR1	TEND	1-Aug-11	NULL	2.917092846427472	INTERFERON ALFA-N3	rxcui:612937	INTERFERON ALFA-N3	TRUE	TRUE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.3211478363039418	LEVOMETHADYL ACETATE	rxcui:237005	LEVOMETHADYL	TRUE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	modulator	0.6177373086552295	IUPHAR.LIGAND:5921	iuphar.ligand:5921	AKT INHIBITOR VIII	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.182318303	LISDEXAMFETAMINE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.025942525	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.2907401508067248	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.035083077	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
UNIPROT:Q9GZZ6	hgnc:13800	CHRNA10	TEND	1-Aug-11	NULL	10.50153424713889	PENTOLINIUM	ncit:C77367	PENTOLINIUM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1835932560688619	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.042619863	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TEND	1-Aug-11	NULL	0.058602312	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	modulator	0.7001022831425934	IUPHAR.LIGAND:5921	iuphar.ligand:5921	AKT INHIBITOR VIII	FALSE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TEND	1-Aug-11	NULL	1.346350544504987	RANIBIZUMAB	rxcui:595060	RANIBIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.029443554	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:11877	ncit:C154279	IRUPLINALKIB	FALSE	FALSE	FALSE
UNIPROT:P29274	hgnc:263	ADORA2A	TEND	1-Aug-11	NULL	0.9460841664089098	REGADENOSON	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.2386712328895204	RIMEXOLONE	rxcui:55681	RIMEXOLONE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.4375639269641208	SALICYLIC ACID	rxcui:9525	SALICYLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P40238	hgnc:7217	MPL	TEND	1-Aug-11	NULL	2.983390411119005	ROMIPLOSTIM	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.1280674908187671	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P25103	hgnc:11526	TACR1	TEND	1-Aug-11	NULL	2.838252499226729	APREPITANT	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.084146909	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:7739	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.11707396	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.2128689374420047	TIOTROPIUM	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.037721028	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TEND	1-Aug-11	NULL	0.1282238613814273	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.2282942227638891	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
DYSTROPHIN	hgnc:2928	DMD	TTD	2020.06.01	NULL	NULL	MyoDys	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2919	hgnc:4602	CXCL1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10062	iuphar.ligand:10062	ABX-1431	FALSE	FALSE	FALSE
LAMININ GAMMA-2 SUBUNIT	hgnc:6493	LAMC2	TTD	2020.06.01	NULL	NULL	BST-1005	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR IONOTROPIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	LY-545694	chembl:CHEMBL3545161	LY545694	FALSE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.106290832	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	WT-4869	NULL	NULL	NULL	NULL	NULL
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:500	iuphar.ligand:500	[125I]HEAT (BE2254)	FALSE	FALSE	FALSE
APOLIPOPROTEIN A-I	hgnc:600	APOA1	TTD	2020.06.01	NULL	NULL	CER-522	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	ABT-354	NULL	NULL	NULL	NULL	NULL
RESPIRATORY SYNCYTIAL VIRUS PROTEIN F	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAR438584	chembl:CHEMBL3707327	SUPTAVUMAB	FALSE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMAP-102	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	ANAVEX 1007	NULL	NULL	NULL	NULL	NULL
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.071148606	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	ANAVEX 1007	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	BN-OD-026	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	1.009762908	ABT-122	iuphar.ligand:9597	REMTOLUMAB	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	2.561349816375341	DWP-05195	chembl:CHEMBL3545229	DWP05195	FALSE	FALSE	FALSE
TGF-BETA RECEPTOR TYPE I	hgnc:11772	TGFBR1	TTD	2020.06.01	NULL	NULL	P-2745	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	NULL	ONO-4232	NULL	NULL	NULL	NULL	NULL
ERBB2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tucatinib	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
STEROID 17-ALPHA-MONOOXYGENASE	hgnc:2593	CYP17A1	TTD	2020.06.01	NULL	7.501095891	Seviteronel	ncit:C113652	SEVITERONEL	FALSE	FALSE	FALSE
DNA SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glufosfamide	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
HYDROXYCARBOXYLIC ACID RECEPTOR 3	hgnc:16824	HCAR3	TTD	2020.06.01	NULL	NULL	NIA-114	NULL	NULL	NULL	NULL	NULL
NICOTINIC ACID RECEPTOR	hgnc:24827	HCAR2	TTD	2020.06.01	NULL	NULL	NIA-114	NULL	NULL	NULL	NULL	NULL
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	NULL	ARN-6039	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	CTP-543	ncit:C175770	DEURUXOLITINIB	FALSE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	CTP-543	ncit:C175770	DEURUXOLITINIB	FALSE	FALSE	FALSE
INTERFERON ALPHA/BETA RECEPTOR 2	hgnc:5433	IFNAR2	TTD	2020.06.01	NULL	1.640864726115453	Anifrolumab	rxcui:2565265	ANIFROLUMAB	TRUE	FALSE	FALSE
SPHINGOSINE-1 PHOSPHATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	KPP203	NULL	NULL	NULL	NULL	NULL
T-CELL-SPECIFIC SURFACE GLYCOPROTEIN CD28	hgnc:1653	CD28	TTD	2020.06.01	NULL	7.001022831425932	Lulizumab pegol	ncit:C175727	LULIZUMAB PEGOL	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Trastuzumab biosimilar	NULL	NULL	NULL	NULL	NULL
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.2386712328895204	IUPHAR.LIGAND:5443	rxcui:5033	GUANABENZ	TRUE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMG 420	ncit:C159652	PACANALOTAMAB	FALSE	FALSE	FALSE
SLAM FAMILY MEMBER 7 SLAMF7	hgnc:21394	SLAMF7	TTD	2020.06.01	NULL	2.187819634820604	ABBV-838	ncit:C122816	AZINTUXIZUMAB VEDOTIN	FALSE	FALSE	FALSE
NEURAL CELL ADHESION MOLECULE L1	hgnc:6470	L1CAM	TTD	2020.06.01	NULL	NULL	JCAR023	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 13 RECEPTOR ALPHA-2	hgnc:5975	IL13RA2	TTD	2020.06.01	NULL	NULL	MB-101	NULL	NULL	NULL	NULL	NULL
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	BPX-501	ncit:C105395	RIVOGENLECLEUCEL	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:136	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	NULL	NY-ESO-TCR	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION GENE 3 PROTEIN	hgnc:6476	LAG3	TTD	2020.06.01	NULL	NULL	Anti-LAG3	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR-II	hgnc:5466	IGF2	TTD	2020.06.01	NULL	2.917092846427472	Xentuzumab	ncit:C106118	XENTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
DELTA-LIKE PROTEIN 4	hgnc:2910	DLL4	TTD	2020.06.01	NULL	5.250767123569449	Navicixizumab	ncit:C119620	NAVICIXIZUMAB	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NBTX-001	NULL	NULL	NULL	NULL	NULL
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	MIN-117	NULL	NULL	NULL	NULL	NULL
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:3930	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	NULL	MIN-117	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	MIN-117	NULL	NULL	NULL	NULL	NULL
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4907258993990139	SPN-812	chembl:CHEMBL2106483	VILOXAZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
TRANSFORMATION-SENSITIVE PROTEIN P120	hgnc:497	TRPA1	TTD	2020.06.01	NULL	NULL	HX-100	NULL	NULL	NULL	NULL	NULL
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:526	iuphar.ligand:526	RX821002	FALSE	FALSE	FALSE
LIPOXYGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ketoprofen topical	NULL	NULL	NULL	NULL	NULL
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.06466462	IUPHAR.LIGAND:2805	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	Ketoprofen topical	NULL	NULL	NULL	NULL	NULL
SYNUCLEIN ALPHA	hgnc:11138	SNCA	TTD	2020.06.01	NULL	NULL	NPT-200-11	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Radiprodil	ncit:C152143	RADIPRODIL	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	NULL	RTA-901	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	1.050153425	DNL201	iuphar.ligand:9393	GNE-0877	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Ropinirole subdermal implant	NULL	NULL	NULL	NULL	NULL
PATTERN RECOGNITION RECEPTOR NOD2	hgnc:5331	NOD2	TTD	2020.06.01	NULL	1.875273972703375	SB-9200	chembl:CHEMBL1076930	INARIGIVIR SOPROXIL	FALSE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	1.500219178	Vx-001	ncit:C111689	HLA-A*0201 RESTRICTED TERT(572Y)/TERT(572) PEPTIDES VACCINE VX-001	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	KRP-104	chembl:CHEMBL4297624	BISEGLIPTIN	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	AT001/r84	NULL	NULL	NULL	NULL	NULL
TRANSTHYRETIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Revusiran	ncit:C152204	REVUSIRAN	FALSE	FALSE	FALSE
KINESIN SPINDLE MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALN-VSP	NULL	NULL	NULL	NULL	NULL
PCSK9 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALN-PCS	rxcui:2588243	INCLISIRAN	TRUE	FALSE	FALSE
GHRELIN	hgnc:18129	GHRL	TTD	2020.06.01	NULL	NULL	Unacylated ghrelin	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Setrobuvir	ncit:C152351	SETROBUVIR	FALSE	FALSE	FALSE
IGF1R MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATL-1101	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL O-ACYLTRANSFERASE 2	hgnc:16940	DGAT2	TTD	2020.06.01	NULL	NULL	ARI-3037MO	NULL	NULL	NULL	NULL	NULL
GASTRIN-RELEASING PEPTIDE RECEPTOR	hgnc:4609	GRPR	TTD	2020.06.01	NULL	NULL	ASP-7147	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Crestor/TriLipix	NULL	NULL	NULL	NULL	NULL
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	AZD5658	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AT13148	ncit:C101786	MULTI-AGC KINASE INHIBITOR AT13148	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	AVA-101	NULL	NULL	NULL	NULL	NULL
C5A ANAPHYLATOXIN CHEMOTACTIC RECEPTOR	hgnc:1338	C5AR1	TTD	2020.06.01	NULL	0.9376369863516874	PMX-53	iuphar.ligand:579	PMX53	FALSE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	3.281729452230906	Cinacalcet	rxcui:407990	CINACALCET	TRUE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	0.5147810905460245	Anti-HER3/EGFR DAF	drugbank:DB12142	DULIGOTUZUMAB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1389091831632129	Anti-HER3/EGFR DAF	drugbank:DB12142	DULIGOTUZUMAB	FALSE	FALSE	FALSE
TRAIL RECEPTOR 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mapatumumab	ncit:C61502	MAPATUMUMAB	FALSE	TRUE	TRUE
CYTOMEGALOVIRUS 65KDA PHOSPHOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	CMVpp65-A0201	NULL	NULL	NULL	NULL	NULL
MACROPHAGE-STIMULATING PROTEIN RECEPTOR	hgnc:7381	MST1R	TTD	2020.06.01	NULL	NULL	RON mab	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-12 BETA	hgnc:5970	IL12B	TTD	2020.06.01	NULL	NULL	Ad-IL-12 DNA therapeutic	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Melphalan flufenamide	rxcui:2531369	MELPHALAN FLUFENAMIDE	TRUE	FALSE	FALSE
NEOPLASM ANTIGEN	hgnc:12811	XK	TTD	2020.06.01	NULL	0.8468979231563628	NPC-1C	ncit:C90532	ENSITUXIMAB	FALSE	FALSE	FALSE
HEMATOPOIETIC PROGENITOR CELL ANTIGEN CD34	hgnc:1662	CD34	TTD	2020.06.01	NULL	5.250767123569449	AMR-001	ncit:C103865	AUTOLOGOUS BONE MARROW-DERIVED CD34/CXCR4-POSITIVE STEM CELLS AMR-001	FALSE	FALSE	FALSE
NCBIGENE:2767	hgnc:4379	GNA11	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:7266	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE 2	hgnc:812	ATP2A2	TTD	2020.06.01	NULL	NULL	Mydicar	NULL	NULL	NULL	NULL	NULL
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Solithromycin oral	NULL	NULL	NULL	NULL	NULL
NITRIC-OXIDE SYNTHASE ENDOTHELIAL	hgnc:7876	NOS3	TTD	2020.06.01	NULL	NULL	ACCLAIM	NULL	NULL	NULL	NULL	NULL
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	NULL	DS-3801	NULL	NULL	NULL	NULL	NULL
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.2318219480604613	HDM201	ncit:C116325	SIREMADLIN	FALSE	FALSE	FALSE
APOLIPOPROTEIN A-I	hgnc:600	APOA1	TTD	2020.06.01	NULL	4.565884455277782	CER-001	drugbank:DB18538	CER-001	FALSE	FALSE	FALSE
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	N-{4	NULL	NULL	NULL	NULL	NULL
KYNURENINE OXOGLUTARATE TRANSAMINASE II	hgnc:17929	AADAT	TTD	2020.06.01	NULL	NULL	US8933095, 18	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US8609715, A-1	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US8609715, A-26	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US8609715, B-61	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	BB 0223767	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8669361, 105	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	EEA	NULL	NULL	NULL	NULL	NULL
GALECTIN-1	hgnc:6561	LGALS1	TTD	2020.06.01	NULL	NULL	US8703720, Reference Compound 1	NULL	NULL	NULL	NULL	NULL
CARBOXYPEPTIDASE B1	hgnc:2299	CPB1	TTD	2020.06.01	NULL	NULL	US8710232, 8	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8598210, Table XV, 5	NULL	NULL	NULL	NULL	NULL
ADAM METALLOPEPTIDASE 33	hgnc:15478	ADAM33	TTD	2020.06.01	NULL	NULL	US8772478, 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL NICOTINATE-NUCLEOTIDE ADENYLYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	DZ9	NULL	NULL	NULL	NULL	NULL
CASEIN KINASE II ALPHA PRIME	hgnc:2459	CSNK2A2	TTD	2020.06.01	NULL	NULL	US8791257, 17	NULL	NULL	NULL	NULL	NULL
REGULATOR OF G-PROTEIN SIGNALING 16	hgnc:9997	RGS16	TTD	2020.06.01	NULL	NULL	s2901	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C ZETA	hgnc:9412	PRKCZ	TTD	2020.06.01	NULL	NULL	US8889672, 252-036-001	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8921389, 22	NULL	NULL	NULL	NULL	NULL
BCL-2-RELATED PROTEIN A1	hgnc:991	BCL2A1	TTD	2020.06.01	NULL	NULL	US8937193-compound-6b	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9409892, 148	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US9434727, 63	NULL	NULL	NULL	NULL	NULL
PROKINETICIN RECEPTOR-1	hgnc:4524	PROKR1	TTD	2020.06.01	NULL	NULL	US9475795, 19	NULL	NULL	NULL	NULL	NULL
PROKINETICIN RECEPTOR-1	hgnc:4524	PROKR1	TTD	2020.06.01	NULL	NULL	US9475795, 80	NULL	NULL	NULL	NULL	NULL
PROKINETICIN RECEPTOR-1	hgnc:4524	PROKR1	TTD	2020.06.01	NULL	NULL	US9475795, 89	NULL	NULL	NULL	NULL	NULL
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6911	iuphar.ligand:6911	N,N`-BIS-ALKYL BUTYLIMMIDAZOLE 12B	FALSE	FALSE	FALSE
BETA-ADRENERGIC RECEPTOR KINASE 1	hgnc:289	GRK2	TTD	2020.06.01	NULL	NULL	US9493490, E	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9580418, Example 8	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9586945, 19a	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	BDBM50080570	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE EIF2AK2	hgnc:20932	POLD3	TTD	2020.06.01	NULL	NULL	US9650366, 9	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9656955, Example 351	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE C4 SYNTHASE	hgnc:6719	LTC4S	TTD	2020.06.01	NULL	NULL	US20160326143, 50	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 2	hgnc:3169	S1PR2	TTD	2020.06.01	NULL	NULL	Unii-R228S06soh	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9670220, 76	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Rituxan Immunology	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	G0-203-2c	NULL	NULL	NULL	NULL	NULL
HISTAMINE RECEPTOR	hgnc:5172	HR	TTD	2020.06.01	NULL	NULL	Votucalis ophthalmic	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	QAX-028	NULL	NULL	NULL	NULL	NULL
INTERFERON ALPHA/BETA RECEPTOR 1	hgnc:5432	IFNAR1	TTD	2020.06.01	NULL	NULL	EMZ701	NULL	NULL	NULL	NULL	NULL
GLUTATHIONE-DEPENDENT PGD SYNTHASE	hgnc:17890	HPGDS	TTD	2020.06.01	NULL	NULL	HF-0220	NULL	NULL	NULL	NULL	NULL
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	NULL	Revolade/Promacta	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	Iboctadekin + Doxil	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-18	hgnc:5986	IL18	TTD	2020.06.01	NULL	NULL	Iboctadekin + Doxil	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-18	hgnc:5986	IL18	TTD	2020.06.01	NULL	NULL	Iboctadekin + rituximab	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Iboctadekin + rituximab	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK1265744	rxcui:2475077	CABOTEGRAVIR	TRUE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	0.7001022831425933	CG-0070	ncit:C48412	CRETOSTIMOGENE GRENADENOREPVEC	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	NULL	Trametinib + 2141795	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	NULL	TRN-157	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	PSMA subunit vaccine	NULL	NULL	NULL	NULL	NULL
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	Leukemia cancer vaccine	NULL	NULL	NULL	NULL	NULL
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	NULL	RHuEPO	NULL	NULL	NULL	NULL	NULL
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	NULL	Peg-G-CSF	NULL	NULL	NULL	NULL	NULL
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	NULL	BVI-007	NULL	NULL	NULL	NULL	NULL
GUANYLYL CYCLASE C	hgnc:4688	GUCY2C	TTD	2020.06.01	NULL	NULL	ISIS-GCCRrx	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	NULL	CRX-675	NULL	NULL	NULL	NULL	NULL
TGF-BETA RECEPTOR TYPE II	hgnc:11773	TGFBR2	TTD	2020.06.01	NULL	NULL	TGF-BR2 mab	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7732	iuphar.ligand:7732	SM-337	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.596678082	HT-0712	drugbank:DB11650	HT-0712	FALSE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR ACETYLHYDROLASE	hgnc:9040	PLA2G7	TTD	2020.06.01	NULL	13.12691780892362	GSK2647544	chembl:CHEMBL3634561	GSK-2647544	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	IMO-2134	NULL	NULL	NULL	NULL	NULL
NUCLEOPHOSMIN	hgnc:7910	NPM1	TTD	2020.06.01	NULL	3.750547945	IPP-204106	ncit:C103297	NUCLEOLIN ANTAGONIST IPP-204106N	FALSE	FALSE	FALSE
APOB MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mipomersen	rxcui:1367839	MIPOMERSEN	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REV MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	HGTV43	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	NULL	0.364636606	IUPHAR.LIGAND:4935	iuphar.ligand:4935	GROWTH ARREST SPECIFIC PROTEIN 6	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS TAT MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	HGTV43	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS TRANS-ACTIVATION RESPONSE ELEMENT	NULL	NULL	TTD	2020.06.01	NULL	NULL	HGTV43	NULL	NULL	NULL	NULL	NULL
INFLUENZA HEMAGGLUTININ	NULL	NULL	TTD	2020.06.01	NULL	NULL	VGX-3400	NULL	NULL	NULL	NULL	NULL
SOD1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-SOD1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	ChronSeal	NULL	NULL	NULL	NULL	NULL
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	KUR-211	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vaniprevir	ncit:C152828	VANIPREVIR	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MBX-700	NULL	NULL	NULL	NULL	NULL
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	NULL	M118	NULL	NULL	NULL	NULL	NULL
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	PRX-3140	NULL	NULL	NULL	NULL	NULL
RIBONUCLEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	NTO-1151	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	NULL	Somatomedin-1	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AKB-6548	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	AMG 151	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR RXR-GAMMA	hgnc:10479	RXRG	TTD	2020.06.01	NULL	NULL	NRX-4204	NULL	NULL	NULL	NULL	NULL
PLASMODIUM THROMBOSPONDIN RELATE ANONYMOUS PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PlaMavax	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	FRM-0962	NULL	NULL	NULL	NULL	NULL
PHOSPHOFRUCTOKINASE 2	hgnc:8874	PFKFB3	TTD	2020.06.01	NULL	NULL	INGAP peptide	NULL	NULL	NULL	NULL	NULL
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:617	iuphar.ligand:617	LITORIN	FALSE	FALSE	FALSE
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	EDP-420	ncit:C174586	MODITHROMYCIN	FALSE	FALSE	FALSE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	NULL	RU-101	NULL	NULL	NULL	NULL	NULL
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PolyHeme	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	BN-2629	chembl:CHEMBL16498	SJG-136	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	OBE-101	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	BVT-74316	NULL	NULL	NULL	NULL	NULL
ADVANCED GLYCOSYLATION END PRODUCT RECEPTOR	hgnc:320	AGER	TTD	2020.06.01	NULL	NULL	TTP-4000	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	Tolamba	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiarabine	ncit:C92589	THIARABINE	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:3946	iuphar.ligand:3946	[D-TYR6,APA-4CL11,PHE13,NLE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
LONG TRANSIENT RECEPTOR POTENTIAL CHANNEL 8	hgnc:17961	TRPM8	TTD	2020.06.01	NULL	8.290684931951763	D-3263	chembl:CHEMBL3707315	D-3263	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	NULL	Rycals	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	ARI-2243	NULL	NULL	NULL	NULL	NULL
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	NULL	ALX-0651	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	FG-2216	drugbank:DB08687	FG-2216	FALSE	FALSE	FALSE
VASOPRESSIN V1B RECEPTOR	hgnc:896	AVPR1B	TTD	2020.06.01	NULL	NULL	ABT-436	NULL	NULL	NULL	NULL	NULL
CALCITONIN RECEPTOR	hgnc:1440	CALCR	TTD	2020.06.01	NULL	NULL	Calcitonin oral	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	NULL	AAV2-hFIX16	NULL	NULL	NULL	NULL	NULL
HUMAN PAPILLOMAVIRUS PROTEIN E7	NULL	NULL	TTD	2020.06.01	NULL	NULL	CIGB-228	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9823	iuphar.ligand:9823	COMPOUND 12 [PMID:28626832]	FALSE	FALSE	FALSE
PLASMODIAL PHOSPHOLIPID METABOLISM	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAR97276	ncit:C90735	ALBITIAZOLIUM BROMIDE	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	NULL	BI-44847	NULL	NULL	NULL	NULL	NULL
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	2.917092846427472	PMX-60056	chembl:CHEMBL2107820	DELPARANTAG	FALSE	FALSE	FALSE
BETA-CATENIN	hgnc:2514	CTNNB1	TTD	2020.06.01	NULL	2.386712328895204	CEQ-508	drugbank:DB17911	CEQ508	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	IBC-VS01	NULL	NULL	NULL	NULL	NULL
MART-1 MELANOMA ANTIGEN	hgnc:7124	MLANA	TTD	2020.06.01	NULL	NULL	Multi-epitope peptide melanoma vaccine	NULL	NULL	NULL	NULL	NULL
MELANOCYTES LINEAGE-SPECIFIC ANTIGEN GP100	hgnc:10880	PMEL	TTD	2020.06.01	NULL	NULL	Multi-epitope peptide melanoma vaccine	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Multi-epitope peptide melanoma vaccine	NULL	NULL	NULL	NULL	NULL
RAS-LIKE PROTEIN KIR	hgnc:4234	GEM	TTD	2020.06.01	NULL	1.312691780892362	Lirilumab	ncit:C103820	LIRILUMAB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.5556367326528519	IMGN289	ncit:C111906	LAPRITUXIMAB EMTANSINE	FALSE	FALSE	FALSE
T-CELL-SPECIFIC KINASE	hgnc:6171	ITK	TTD	2020.06.01	NULL	NULL	JTE-051	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	NULL	AR08	NULL	NULL	NULL	NULL	NULL
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	NULL	PAZ-320	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-2/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vatelizumab	ncit:C152838	VATELIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:6944	iuphar.ligand:6944	OXAZINE 89	FALSE	FALSE	FALSE
HAEMOPHILUS INFLUENZAE DNA GYRASE A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Inhaled liposomal ciprofloxacin	NULL	NULL	NULL	NULL	NULL
STREPTOCOCCUS TOPOISOMERASE IV A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Inhaled liposomal ciprofloxacin	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:12747	ncit:C166726	UMIBECESTAT	FALSE	FALSE	FALSE
CHOLESTEROL UPTAKE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PAMAQUESIDE	ncit:C170284	PAMAQUESIDE	FALSE	FALSE	FALSE
PTPN1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hydrogen peroxide	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
TRYPTASE ALPHA/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lactoferrin	rxcui:1425933	LACTOFERRIN	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Budipine	rxcui:19832	BUDIPINE	FALSE	FALSE	FALSE
VIRUS DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Idoxuridine	rxcui:5653	IDOXURIDINE	TRUE	FALSE	FALSE
ENDOTHELIN B RECEPTOR	hgnc:3180	EDNRB	TTD	2020.06.01	NULL	1.875273972703375	BQ788	iuphar.ligand:1010	BQ788	FALSE	FALSE	FALSE
INTERFERON ALPHA/BETA RECEPTOR 1	hgnc:5432	IFNAR1	TTD	2020.06.01	NULL	NULL	R-IFN-1a	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dactinomycin	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
P2Y PURINOCEPTOR 12	hgnc:18124	P2RY12	TTD	2020.06.01	NULL	NULL	ARL-67085	NULL	NULL	NULL	NULL	NULL
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.1172046232939609	IUPHAR.LIGAND:484	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
VASOPRESSIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Desmopressin	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
HISTAMINE N-METHYLTRANSFERASE	hgnc:5028	HNMT	TTD	2020.06.01	NULL	2.500365296937833	Metoprine	ncit:C1161	METOPRINE	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Naproxen	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
BACTERIAL FUMARATE REDUCTASE FLAVOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiabendazole	rxcui:10450	THIABENDAZOLE	TRUE	FALSE	FALSE
AROMATIC-L-AMINO-ACID DECARBOXYLASE	hgnc:2719	DDC	TTD	2020.06.01	NULL	NULL	Patrome	NULL	NULL	NULL	NULL	NULL
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:7445	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dirithromycin	rxcui:23437	DIRITHROMYCIN	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CALANOLIDE A	drugbank:DB04886	CALANOLIDE A	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:557	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
CASPASE-7	hgnc:1508	CASP7	TTD	2020.06.01	NULL	NULL	isatin sulfonamide 34	NULL	NULL	NULL	NULL	NULL
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:3401	iuphar.ligand:3401	15S-HETE	FALSE	FALSE	FALSE
CASPASE-9	hgnc:1511	CASP9	TTD	2020.06.01	NULL	NULL	isatin sulfonamide 34	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Eicosapentaenoic acid/docosa-hexaenoic acid	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	Eicosapentaenoic acid/docosa-hexaenoic acid	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfonamide	ncit:C29739	SULFONAMIDE ANTI-INFECTIVE AGENT	FALSE	FALSE	FALSE
AROMATIC-L-AMINO-ACID DECARBOXYLASE	hgnc:2719	DDC	TTD	2020.06.01	NULL	5.250767123569449	Carbidopa	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:1786	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:8144	iuphar.ligand:8144	COMPOUND 13R [PMID: 23639540]	FALSE	FALSE	FALSE
LOW-AFFINITY NERVE GROWTH FACTOR RECEPTOR	hgnc:7809	NGFR	TTD	2020.06.01	NULL	2.917092846427472	Voclosporin	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	HIF-1alpha	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	SUN N4057	NULL	NULL	NULL	NULL	NULL
CORE PROTEASOME 20S COMPLEX	NULL	NULL	TTD	2020.06.01	NULL	NULL	PS-341	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AjvW2	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	Antistasin	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	TA-7906	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	NULL	TA-7906	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	0.1446492320542548	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	NULL	TA-7906	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Muscimol	drugbank:DB12458	MUSCIMOL	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Methylscopolamine	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	L-751250	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	L-751250	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GLYCOPROTEIN 41	NULL	NULL	TTD	2020.06.01	NULL	NULL	T-1249	NULL	NULL	NULL	NULL	NULL
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	1.458546423213736	Phenmetrazine	rxcui:8133	PHENMETRAZINE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefuroxime	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
TNF-ALPHA/IL-1 BETA PRODUCTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Esonarimod	ncit:C65540	ESONARIMOD	FALSE	FALSE	FALSE
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	NULL	Ad-OC-hsvTK/valacyclovir	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:9977	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	NULL	ELND-002	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	NCX-6560	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Premarin/Pravachol	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	NULL	Premarin/Pravachol	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Premarin/Pravachol	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP120	NULL	NULL	TTD	2020.06.01	NULL	NULL	AIDSVAX	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CLX-0921	drugbank:DB05854	CLX-0921	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8876	iuphar.ligand:8876	MS363	FALSE	FALSE	FALSE
IRON	hgnc:4650	GTF2E1	TTD	2020.06.01	NULL	NULL	Soluble ferric pyrophosphate	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cephalexin	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	L-751250	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRYPTAMINE	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	AFTVac	NULL	NULL	NULL	NULL	NULL
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	2.282942227638891	CT84.66	ncit:C77885	YTTRIUM Y 90 ANTI-CEA MONOCLONAL ANTIBODY CT84.66	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.2692701089009974	Hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR BETA	hgnc:6009	IL2RB	TTD	2020.06.01	NULL	NULL	AFTVac	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2723	ncbigene:2723	GLC1C	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8876	iuphar.ligand:8876	MS363	FALSE	FALSE	FALSE
HORMONE SENSITIVE LIPASE	hgnc:6621	LIPE	TTD	2020.06.01	NULL	NULL	PMID15026062C41	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glyminox	NULL	NULL	NULL	NULL	NULL
PTPN1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRYPAN BLUE	rxcui:10878	TRYPAN BLUE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BRK	hgnc:9617	PTK6	TTD	2020.06.01	NULL	NULL	ISIS-CRP	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:9299	ncit:C116844	FENEBRUTINIB	FALSE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Meclocycline	rxcui:29418	MECLOCYCLINE	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Stavudine	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Daptomycin	rxcui:22299	DAPTOMYCIN	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	3.088686543276147	ONO-AE1-437	iuphar.ligand:8541	ONO-AE1-437	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	BCI-632	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SGS742	drugbank:DB05010	SGS-742	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Famciclovir	rxcui:68099	FAMCICLOVIR	TRUE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	JNJ-17216498	drugbank:DB17087	JNJ-17216498	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:10231	ncit:C136416	VECABRUTINIB	FALSE	FALSE	FALSE
SCHISTOSOMA PURINE NUCLEOSIDE PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	FP-253-GDEPT	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NS3 HELICASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BILN-2061	chembl:CHEMBL297884	CILUPREVIR	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:9285	iuphar.ligand:9285	PRN694	FALSE	FALSE	FALSE
FUCOSYLTRANSFERASE IV	hgnc:4015	FUT4	TTD	2020.06.01	NULL	NULL	99mTc-fanolesomab	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ki23819	NULL	NULL	NULL	NULL	NULL
NCBIGENE:939	hgnc:11922	CD27	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10256	ncit:C174684	CINROMIDE	FALSE	FALSE	FALSE
FUNGAL ISOLEUCYL T-RNA SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Icofungipen	ncit:C65880	ICOFUNGIPEN	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Trimegestone/ethinyl estradiol	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	NULL	Iboctadekin + rituximab	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefprozil	rxcui:1546020	CEFPROZIL ANHYDROUS	TRUE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.099446347	Methylergonovine	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE XIV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfamylon	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	MCD-386	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	CL-314698	NULL	NULL	NULL	NULL	NULL
DNA-BINDING FACTOR KBF1	hgnc:14372	SCYL1	TTD	2020.06.01	NULL	26.25383561784724	P54	drugbank:DB05451	P54	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3A	hgnc:8778	PDE3A	TTD	2020.06.01	NULL	1.591141552596802	Anagrelide	rxcui:236612	ANAGRELIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHOLECYSTOKININ RECEPTOR TYPE A	hgnc:1570	CCKAR	TTD	2020.06.01	NULL	NULL	FPL-14294	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	GCR-1087	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 1	hgnc:7956	NPY1R	TTD	2020.06.01	NULL	NULL	GI-264879A	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	L-751250	NULL	NULL	NULL	NULL	NULL
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:5768	iuphar.ligand:5768	C5A HEXAPEPTIDE ANALOGUE	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	NULL	MC-4 agonist	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 5	hgnc:7958	NPY5R	TTD	2020.06.01	NULL	NULL	NPY5RA-972	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	UC-781	drugbank:DB05871	UC-781	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	TKA-731	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	NULL	Micardis telmisartan	NULL	NULL	NULL	NULL	NULL
GALANIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	HT-2157	chembl:CHEMBL4297765	HT-2157	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	AWD-12-281	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1959	hgnc:3239	EGR2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12810	iuphar.ligand:12810	COMPOUND 26 [PMID: 34543009]	FALSE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Silver sulfadiazine	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	AN-1792	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	THIOCOLCHICOSIDE	rxcui:38085	THIOCOLCHICOSIDE	FALSE	FALSE	FALSE
GLYCINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	THIOCOLCHICOSIDE	rxcui:38085	THIOCOLCHICOSIDE	FALSE	FALSE	FALSE
GROWTH/DIFFERENTIATION FACTOR 5	NULL	NULL	TTD	2020.06.01	NULL	NULL	RhGDF-5	chembl:CHEMBL2108637	RADOTERMIN	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	activator	0.1035654265003836	IUPHAR.LIGAND:1204	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
CYTOMEGALOVIRUS DNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Guanosine	rxcui:1591890	GUANOSINE	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Guanosine	rxcui:1591890	GUANOSINE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Conjugated estrogens a	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valopicitabine dihydrochloride	ncit:C72874	VALOPICITABINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
FUNGAL 1,3-BETA-GLUCAN SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anidulafungin	rxcui:341018	ANIDULAFUNGIN	TRUE	FALSE	FALSE
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Diphtheria-tetanus vaccine	NULL	NULL	NULL	NULL	NULL
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	NULL	Rh-alphaglucosidase	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CX-1501	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRO-19622	ncit:C174604	OLESOXIME	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	(-)-3PPP, Maryland	NULL	NULL	NULL	NULL	NULL
DOPAMINE D5 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	LE-300	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	Organon-3	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-157533	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1956	hgnc:3236	EGFR	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:5274	iuphar.ligand:5274	STO609	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	NULL	RMG-40083	NULL	NULL	NULL	NULL	NULL
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SPI-376	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	H5N1 influenza vaccine	NULL	NULL	NULL	NULL	NULL
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	NULL	Atamestane-plus- Toremifene	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dornase Alfa	rxcui:337623	DORNASE ALFA	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	1.500219178	Amibegron	ncit:C77932	AMIBEGRON	FALSE	FALSE	FALSE
C-X-C MOTIF CHEMOKINE 2	hgnc:4603	CXCL2	TTD	2020.06.01	NULL	NULL	Laquinamod	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	activator	2.333674277141977	IUPHAR.LIGAND:5238	iuphar.ligand:5238	PAC1	FALSE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	ICA-17043	ncit:C76882	SENICAPOC	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Raltegravir	rxcui:1235585	RALTEGRAVIR POTASSIUM	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	ISIS-CRP	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Avastin+/-Tarceva	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
NCBIGENE:1550	hgnc:2612	CYP2A7P1	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8126	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	5.250767123569449	OZ277	chembl:CHEMBL404431	OZ277	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.033875917	HP-184	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	NULL	VER 50589	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 1 ALPHA	hgnc:4910	HIF1A	TTD	2020.06.01	NULL	NULL	HIF-1alpha	NULL	NULL	NULL	NULL	NULL
DUAL SPECIFICITY PROTEIN PHOSPHATASE 1	hgnc:3064	DUSP1	TTD	2020.06.01	NULL	NULL	Avastin+/-Tarceva	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1617	hgnc:2682	DAZ1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9901	iuphar.ligand:9901	URACIL 20	FALSE	FALSE	FALSE
M-PHASE INDUCER PHOSPHATASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Avastin+/-Tarceva	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	0.3365876361262467	Diflorasone	rxcui:23033	DIFLORASONE DIACETATE	TRUE	FALSE	FALSE
INFLUENZA NEURAMINIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CS-8958	chembl:CHEMBL467058	LANINAMIVIR OCTANOATE	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	Sphingosome Encapsulated Vinorelbine	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vildagliptin	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Melogliptin	ncit:C87620	MELOGLIPTIN	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASP8497	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	ER-319711-15	NULL	NULL	NULL	NULL	NULL
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	activator	0.305277158	IUPHAR.LIGAND:4065	iuphar.ligand:4065	(-)-(S)-BAYK8644	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	LY-2463665	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.045778266	Thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.8950171233357017	Esmolol	rxcui:49737	ESMOLOL	TRUE	FALSE	FALSE
NCBIGENE:2345	ncbigene:2345	FNZ	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:6541	iuphar.ligand:6541	COMPOUND 1 [PMID: 10498202]	FALSE	FALSE	FALSE
FOLLICLE STIMULATING HORMONE	hgnc:3964	FSHB	TTD	2020.06.01	NULL	NULL	AKP-501	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfamylon	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	2.917092846427472	Anamorelin	ncit:C52197	ANAMORELIN	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.2983390411119005	Desvenlafaxine	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE VI	hgnc:1380	CA6	TTD	2020.06.01	NULL	1.875273972703375	Sulfamylon	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	NULL	GRN163	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pargyline	rxcui:7930	PARGYLINE	FALSE	FALSE	FALSE
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dutasteride	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
NCBIGENE:2354	hgnc:3797	FOSB	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:6478	iuphar.ligand:6478	ODANACATIB	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dacarbazine	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ganciclovir	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
XIAP MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AEG35156	drugbank:DB06184	AEG35156	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	1.029562181092049	Glucosamine	rxcui:4845	GLUCOSAMINE	TRUE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.1333528158366844	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PI3-KINASE BETA	hgnc:8976	PIK3CB	TTD	2020.06.01	NULL	0.066676408	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
GLUCOSE-DEPENDENT INSULINOTROPIC RECEPTOR	hgnc:19060	GPR119	TTD	2020.06.01	NULL	NULL	SAR-260093	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1383	hgnc:1548	CBR1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984016	IUPHAR.LIGAND:5551	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR B	hgnc:8800	PDGFB	TTD	2020.06.01	NULL	NULL	GAM-501	NULL	NULL	NULL	NULL	NULL
CYCLOPHILIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	SCY-635	drugbank:DB12451	SCY-635	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	(S)-oxybutynin	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	RWJ-671818	chembl:CHEMBL1083499	CHEMBL:CHEMBL1083499	FALSE	FALSE	FALSE
ERBB2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
NCBIGENE:391	hgnc:672	RHOG	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:5412	iuphar.ligand:5412	PGF1&ALPHA;	FALSE	FALSE	FALSE
GALECTIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	GCS-100	drugbank:DB17566	GCS-100	FALSE	FALSE	FALSE
INTERFERON-GAMMA	hgnc:5438	IFNG	TTD	2020.06.01	NULL	NULL	VPM-4-001	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	VPM-4-001	NULL	NULL	NULL	NULL	NULL
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Eptifibatide	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.5048814541893701	Sulfamylon	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
MELANOCYTES LINEAGE-SPECIFIC ANTIGEN GP100	hgnc:10880	PMEL	TTD	2020.06.01	NULL	NULL	AE-08	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dutogliptin	ncit:C87492	DUTOGLIPTIN	FALSE	FALSE	FALSE
TRYPANOSOMA CRUZIPAIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRICLABENDAZOLE	rxcui:2118525	TRICLABENDAZOLE	TRUE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	S-110	NULL	NULL	NULL	NULL	NULL
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:8706	iuphar.ligand:8706	COMPOUND 70 [PMID: 26161824]	FALSE	FALSE	FALSE
OPIOID RECEPTOR ZETA	hgnc:15768	OGFR	TTD	2020.06.01	NULL	NULL	IRT-102	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Laromustine	ncit:C2653	LAROMUSTINE	FALSE	FALSE	FALSE
TREFOIL FACTOR-1	hgnc:11755	TFF1	TTD	2020.06.01	NULL	NULL	AG-013	NULL	NULL	NULL	NULL	NULL
MACROPHAGE-STIMULATING PROTEIN RECEPTOR	hgnc:7381	MST1R	TTD	2020.06.01	NULL	NULL	RON Monoclonal Antibody	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.596678082	TOFIMILAST	ncit:C76891	TOFIMILAST	FALSE	FALSE	FALSE
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Friulimicin topical	NULL	NULL	NULL	NULL	NULL
NCBIGENE:67	hgnc:140	ACTBP7	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9714	iuphar.ligand:9714	BI-6901	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	1.419126249613364	UK-432097	drugbank:DB12691	UK-432097	FALSE	FALSE	FALSE
CYTOTOXIC T-LYMPHOCYTE PROTEIN 4	hgnc:2505	CTLA4	TTD	2020.06.01	NULL	0.7001022831425934	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
TERATOCARCINOMA-DERIVED GROWTH FACTOR 1	hgnc:11701	CRIPTO	TTD	2020.06.01	NULL	NULL	BIIB 015	NULL	NULL	NULL	NULL	NULL
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:779	iuphar.ligand:779	RS-102895	FALSE	FALSE	FALSE
CI MAN-6-P RECEPTOR	hgnc:5467	IGF2R	TTD	2020.06.01	NULL	NULL	PXS-25	NULL	NULL	NULL	NULL	NULL
TNF ALPHA PRODUCTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	SH-529	NULL	NULL	NULL	NULL	NULL
MELANOCORTIN RECEPTOR 5	hgnc:6933	MC5R	TTD	2020.06.01	NULL	NULL	JNJ-10229570	NULL	NULL	NULL	NULL	NULL
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:753	iuphar.ligand:753	CCL14	FALSE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA1.1	hgnc:6284	KCNMA1	TTD	2020.06.01	NULL	NULL	CROMOGLYCATE LISETIL HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-3134	NULL	NULL	NULL	NULL	NULL
PI3-KINASE BETA	hgnc:8976	PIK3CB	TTD	2020.06.01	NULL	0.1041818873724097	CH-5132799	drugbank:DB13051	CH-5132799	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3530	iuphar.ligand:3530	SB328437	FALSE	FALSE	FALSE
CHORIOGONADOTROPIN BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CDX-1307	ncit:C77858	HUMAN MONOCLONAL ANTIBODY B11-HCG BETA FUSION PROTEIN CDX-1307	FALSE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	CIGB-M3	NULL	NULL	NULL	NULL	NULL
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	LTX-109	drugbank:DB12711	LTX-109	FALSE	FALSE	FALSE
RHINOVIRUS PROTEASE 3C	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rupintrivir	ncit:C82255	RUPINTRIVIR	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:7348	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
PANCREATIC HORMONE	hgnc:8582	PAH	TTD	2020.06.01	NULL	NULL	PP-1420	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
BACTERIAL RIBOSOME	NULL	NULL	TTD	2020.06.01	NULL	NULL	TP-434	rxcui:2055906	ERAVACYCLINE	TRUE	FALSE	FALSE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	2.386712328895204	JNJ-26070109	iuphar.ligand:6665	JNJ-26070109	FALSE	FALSE	FALSE
FRIZZLED-7 RECEPTOR	hgnc:4045	FZD7	TTD	2020.06.01	NULL	3.000438356325399	OMP-18R5	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:11725	iuphar.ligand:11725	MD-222	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CX-1739	chembl:CHEMBL3707399	CX1739	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	MEDl-551	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	AZD-2115	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-2115	NULL	NULL	NULL	NULL	NULL
ALPHA-1-ANTITRYPSIN	hgnc:8941	SERPINA1	TTD	2020.06.01	NULL	NULL	AGTC-0106	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Famitinib	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
ACTIN POLYMERIZATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Preverex	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	AN-019	NULL	NULL	NULL	NULL	NULL
INFLUENZA HEMAGGLUTININ	NULL	NULL	TTD	2020.06.01	NULL	NULL	ND-1.1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.023295329	IUPHAR.LIGAND:8741	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	Autologous T-cell therapy	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD3 EPSILON	hgnc:1674	CD3E	TTD	2020.06.01	NULL	NULL	Autologous T-cell therapy	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	NULL	Autologous T-cell therapy	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	0.2459375701906065	Famitinib	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.1807492985738192	Famitinib	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	NULL	LY-2189102	NULL	NULL	NULL	NULL	NULL
LUTEINIZING HORMONE RECEPTOR	hgnc:6585	LHCGR	TTD	2020.06.01	NULL	NULL	Org-43902	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	GED-0507-34-Levo	drugbank:DB16109	GED-0507-34-LEVO	FALSE	FALSE	FALSE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	6.177373086552294	GSK-557296	ncit:C99151	EPELSIBAN	FALSE	FALSE	FALSE
CHYMASE	hgnc:2097	CMA1	TTD	2020.06.01	NULL	NULL	ASB17061	NULL	NULL	NULL	NULL	NULL
CASEIN KINASE II	NULL	NULL	TTD	2020.06.01	NULL	NULL	CX-4945	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
INTERLEUKIN 21 RECEPTOR	hgnc:6006	IL21R	TTD	2020.06.01	NULL	NULL	ATR-107	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	BAY-1075553	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AIC-292	NULL	NULL	NULL	NULL	NULL
BACILLUS ANTHRACIS PROTECTIVE ANTIGEN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AIGIV	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BNC-210	chembl:CHEMBL4650452	BNC-210	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	NULL	ADC-3680	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.5048814541893701	Semagacestat	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	NULL	RO-14	NULL	NULL	NULL	NULL	NULL
MYOSIN-7	hgnc:7577	MYH7	TTD	2020.06.01	NULL	NULL	UshStat	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	PEGylated IFN beta 1-a	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-18	hgnc:5986	IL18	TTD	2020.06.01	NULL	0.9211872146613068	Iboctadekin	ncit:C1680	IBOCTADEKIN	FALSE	FALSE	FALSE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Baricitinib	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Baricitinib	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	AC430	iuphar.ligand:9177	AC430	FALSE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-779788	chembl:CHEMBL3545418	BMS-779788	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD4	hgnc:1678	CD4	TTD	2020.06.01	NULL	NULL	Fluoropeptide vaccine	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD8	hgnc:1706	CD8A	TTD	2020.06.01	NULL	NULL	Fluoropeptide vaccine	NULL	NULL	NULL	NULL	NULL
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sofinicline	ncit:C80527	SOFINICLINE	FALSE	FALSE	FALSE
NICOTINIC ACID RECEPTOR	hgnc:24827	HCAR2	TTD	2020.06.01	NULL	17.50255707856483	SCH-900271	drugbank:DB12433	SCH-900271	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	NeuVax	ncit:C117985	NELIPEPIMUT-S	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Her2-targeted autologous T-cell therapy	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1426838892274307	IUPHAR.LIGAND:4194	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
CASPASE 2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	QPI-1007	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMG 579	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	PF-06410293	NULL	NULL	NULL	NULL	NULL
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	YKP-GI	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Debio 1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	MK-2637	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS ALPHA-HEMOLYSIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	MEDI4893	chembl:CHEMBL3989997	SUVRATOXUMAB	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	1.141471113819445	AQW-051	iuphar.ligand:7371	AQW051	FALSE	FALSE	FALSE
INFLUENZA HEMAGGLUTININ	NULL	NULL	TTD	2020.06.01	NULL	NULL	CR8020 mab	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:10242	iuphar.ligand:10242	SC-236	FALSE	FALSE	FALSE
NCBIGENE:721	hgnc:1324	C4B	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
ENZYME UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	VT-1129	NULL	NULL	NULL	NULL	NULL
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	NULL	JTT-302	NULL	NULL	NULL	NULL	NULL
RESPIRATORY SYNCYTIAL VIRUS PROTEIN N	NULL	NULL	TTD	2020.06.01	NULL	NULL	RSV-604	drugbank:DB15197	RSV-604	FALSE	FALSE	FALSE
NCBIGENE:722	hgnc:1325	C4BPA	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV1.2	hgnc:1390	CACNA1C	TTD	2020.06.01	NULL	NULL	ARC029	NULL	NULL	NULL	NULL	NULL
NCBIGENE:717	hgnc:1248	C2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV1.3	hgnc:1391	CACNA1D	TTD	2020.06.01	NULL	NULL	ARC029	NULL	NULL	NULL	NULL	NULL
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	NULL	BI-831266	NULL	NULL	NULL	NULL	NULL
APOPTOSIS SIGNAL-REGULATING KINASE 1	hgnc:6857	MAP3K5	TTD	2020.06.01	NULL	26.25383561784724	GS-4997	ncit:C121943	SELONSERTIB	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	1.750255707856483	Cenicriviroc	ncit:C166464	CENICRIVIROC	FALSE	FALSE	FALSE
NCBIGENE:734	hgnc:1355	OSGIN2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
ENDOSIALIN	hgnc:18219	CD248	TTD	2020.06.01	NULL	157.5230137070835	MORAb-004	ncit:C82406	ONTUXIZUMAB	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	3.889457128569962	Ublituximab	rxcui:2626349	UBLITUXIMAB	TRUE	FALSE	FALSE
NCBIGENE:733	hgnc:1354	C8G	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
ADVANCED GLYCOSYLATION END PRODUCT RECEPTOR	hgnc:320	AGER	TTD	2020.06.01	NULL	NULL	PF-4494700	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tedizolid	rxcui:1540825	TEDIZOLID	TRUE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	5.834185692854944	CRS-207	drugbank:DB17323	CRS-207	FALSE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	HEV-239	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	CNTO-1959	rxcui:1928588	GUSELKUMAB	TRUE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:823	iuphar.ligand:823	MINI-TYRRS	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:8496	iuphar.ligand:8496	VCXCL1	FALSE	FALSE	FALSE
ACTIN	ncbigene:389036	ACT	TTD	2020.06.01	NULL	NULL	RGN-259 eye drops	NULL	NULL	NULL	NULL	NULL
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	NULL	BMS-936561	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	DSP-8658	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PRX-105	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	BAY 85-8501	NULL	NULL	NULL	NULL	NULL
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:837	iuphar.ligand:837	CXCL9	FALSE	FALSE	FALSE
IMMUNOGLOBULIN GAMMA FC RECEPTOR III	hgnc:3619	FCGR3A	TTD	2020.06.01	NULL	0.9907107780319716	AFM-13	drugbank:DB17404	AFM-13	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	PHN-131	NULL	NULL	NULL	NULL	NULL
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	Interferon alpha 2a	NULL	NULL	NULL	NULL	NULL
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:8535	iuphar.ligand:8535	CXCL122 (DIMER)	FALSE	FALSE	FALSE
MYCOBACTERIUM RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifamycin	rxcui:35616	RIFAMYCIN SV	TRUE	FALSE	FALSE
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cariprazine	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PSI-7977	rxcui:1484911	SOFOSBUVIR	TRUE	FALSE	FALSE
NFE2-RELATED FACTOR 2 PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	TECFIDERA	rxcui:1373478	DIMETHYL FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.089756703	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.921012362281506	Tisagenlecleucel	rxcui:1986438	TISAGENLECLEUCEL	TRUE	FALSE	TRUE
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	MAX-10129	NULL	NULL	NULL	NULL	NULL
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Omadacycline	rxcui:2059269	OMADACYCLINE	TRUE	FALSE	FALSE
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TP-434	rxcui:2055906	ERAVACYCLINE	TRUE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:11525	iuphar.ligand:11525	TAGTOCICLIB	FALSE	FALSE	FALSE
HEDGEHOG SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-04449913	rxcui:2105845	GLASDEGIB	TRUE	FALSE	TRUE
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ravulizumab	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	0.1037701012563132	Baricitinib	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-04958242	drugbank:DB11843	PF-04958242	FALSE	FALSE	FALSE
GABA(A) RECEPTOR DELTA	hgnc:4084	GABRD	TTD	2020.06.01	NULL	NULL	SAGE-217b	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAK-653	drugbank:DB16304	TAK-653	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefmenoxime	ncit:C65295	CEFMENOXIME	FALSE	FALSE	FALSE
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Azelaic Acid	rxcui:18602	AZELAIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1975	hgnc:3285	EIF4B	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
PLASMODIUM 80S RIBOSOME	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mefloquine	rxcui:6694	MEFLOQUINE	TRUE	FALSE	FALSE
SODIUM/POTASSIUM-TRANSPORTING ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sanguinarine	rxcui:1537755	SANGUINARINE	FALSE	FALSE	FALSE
FUNGAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Haloprogin	rxcui:26422	HALOPROGIN	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pipobroman	rxcui:8347	PIPOBROMAN	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Muscimol	drugbank:DB12458	MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefonicid	rxcui:2183	CEFONICID	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	NULL	HP-228	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfisoxazole	rxcui:10207	SULFISOXAZOLE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penicillin V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:5950	iuphar.ligand:5950	CDK4 INHIBITOR	FALSE	FALSE	FALSE
HISTAMINE RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CI-959	NULL	NULL	NULL	NULL	NULL
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	NULL	PAI-1	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS TAT PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ro-24-7429	chembl:CHEMBL2360841	RO-24-7429	FALSE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	3.938075342677087	Hexafluronium bromide	rxcui:26826	HEXAFLUORENIUM	FALSE	FALSE	FALSE
BACTERIAL DD-CARBOXYPEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefalotin	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	NULL	YM-16151-4	NULL	NULL	NULL	NULL	NULL
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	NULL	YM-16151-4	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfacytine	rxcui:78902	SULFACYTINE	TRUE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:10095	iuphar.ligand:10095	RO3306	FALSE	FALSE	FALSE
NEUROTRANSMITTER RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TN-871	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	SUN13834	NULL	NULL	NULL	NULL	NULL
INTERFERON RECEPTOR	hgnc:5447	IFNR	TTD	2020.06.01	NULL	NULL	HDV-interferon	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.2243917574174978	Cyclothiazide	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	KW-5092	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefadroxil	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	Avastin+/-Tarceva	NULL	NULL	NULL	NULL	NULL
CYCLIN D1 SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	GORALATIDE	ncit:C170033	GORALATIDE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.3663325900164732	Guanabenz	rxcui:5033	GUANABENZ	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.061725319	Mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
DNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifapentine	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
TUMOR-ASSOCIATED GLYCOPROTEIN 72	NULL	NULL	TTD	2020.06.01	NULL	NULL	Satumomab Pendetide	ncit:C1469	IN 111 SATUMOMAB PENDETIDE	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	CDT-fenofibrate	NULL	NULL	NULL	NULL	NULL
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	NULL	Radiosensitizer gene therapy	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Dexbrompheniramine	rxcui:1767	BROMPHENIRAMINE	TRUE	FALSE	FALSE
BACTERIAL RNA POLYMERASE SIGMA FACTOR SIGA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifamycin	rxcui:35616	RIFAMYCIN SV	TRUE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:11841	iuphar.ligand:11841	SY-5609	FALSE	FALSE	FALSE
STAPHYLOCOCCUS PLASTID RNA POLYMERASE BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifamycin	rxcui:35616	RIFAMYCIN SV	TRUE	FALSE	FALSE
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATG-Fresenius S	drugbank:DB05320	ATG-FRESENIUS S	FALSE	FALSE	FALSE
INTERLEUKIN 4 RECEPTOR ALPHA	hgnc:6015	IL4R	TTD	2020.06.01	NULL	NULL	Aerovant	NULL	NULL	NULL	NULL	NULL
REGULATORY PROTEIN UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	NI-0401	chembl:CHEMBL1743020	FORALUMAB	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	OI338GT	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR-2	hgnc:3676	FGF2	TTD	2020.06.01	NULL	0.3547815624033412	Squalamine	ncit:C143004	SQUALAMINE	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8945	iuphar.ligand:8945	CCT251545	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	SAR228810	NULL	NULL	NULL	NULL	NULL
CYCLOPHILIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	SCY-641	chembl:CHEMBL3707272	RUCLOSPORIN	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	NULL	S-474474	NULL	NULL	NULL	NULL	NULL
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	NULL	TK-DLI	NULL	NULL	NULL	NULL	NULL
RECEPTOR UNSPECIFIC	hgnc:16147	MCM8	TTD	2020.06.01	NULL	NULL	Epicardial angiogenesis patch	NULL	NULL	NULL	NULL	NULL
MELANOCYTES LINEAGE-SPECIFIC ANTIGEN GP100	hgnc:10880	PMEL	TTD	2020.06.01	NULL	NULL	Multi-epitope tyrosinase/gp100 vaccine	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Multi-epitope tyrosinase/gp100 vaccine	NULL	NULL	NULL	NULL	NULL
CYTOKINE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMEC-1217B	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP160	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad5-ENVA-48	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:7054	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
STAPHYLOCOCCUS CAPSULAR POLYSACCHARIDE CP5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06290510	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS CAPSULAR POLYSACCHARIDE CP8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06290510	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS CLUMPING FACTOR A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06290510	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1361	hgnc:2300	CPB2	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:11829	rxcui:2588846	LEVOKETOCONAZOLE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS MANGANESE TRANSPORTER C	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06290510	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-EGFRvIII CAR transduced PBL	NULL	NULL	NULL	NULL	NULL
CEREBROSIDE-SULFATASE	hgnc:713	ARSA	TTD	2020.06.01	NULL	2.187819634820604	HGT-1111	chembl:CHEMBL5095344	CEBSULFASE ALFA	FALSE	FALSE	FALSE
NKG2 D ACTIVATING NK RECEPTOR	hgnc:18788	KLRK1	TTD	2020.06.01	NULL	NULL	CM-CS1 T-cell	NULL	NULL	NULL	NULL	NULL
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	Anti-CEA-CAR T	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HER2-specific T cells	NULL	NULL	NULL	NULL	NULL
CHYMASE	hgnc:2097	CMA1	TTD	2020.06.01	NULL	NULL	BAY 11-42524	NULL	NULL	NULL	NULL	NULL
PROMININ-1	hgnc:9454	PROM1	TTD	2020.06.01	NULL	NULL	Anti-CD133-CAR vector-transduced T cells	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	Anti-meso-CAR T cells	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	Anti-MUC1 CAR T Cells	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	Anti-MUC1 CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19-CAR T cells	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	EGFRvIII CAR T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19-CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19 CAR-T	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Anti-HER2 CAR-T	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	TAI-GPC3-CART cells	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting Glypican-3 (GPC3)	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:8053	iuphar.ligand:8053	NVP-2	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	PCAR-019 (anti-CD19 CAR-T cells)	NULL	NULL	NULL	NULL	NULL
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	NULL	Anti-hCD70 CAR transduced PBL	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD19-TCRz-41BB and CD22-TCRz-41BB CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-TCRz-41BB and CD22-TCRz-41BB CAR-T Cells	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	Anti-CD123-CAR-transduced T cells	NULL	NULL	NULL	NULL	NULL
PROSTATE STEM CELL ANTIGEN	hgnc:9500	PSCA	TTD	2020.06.01	NULL	13.12691780892362	BPX-601	ncit:C128031	AUTOLOGOUS PROSTATE STEM CELL ANTIGEN-SPECIFIC CAR T CELLS BPX-601	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.9723642821424906	Anti-CD20 CAR-T cells	ncit:C201174	ANTI-CD20 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CEA	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting GPC3	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting mesothelin	NULL	NULL	NULL	NULL	NULL
CO-STIMULATORY MOLECULE 4-1BB	hgnc:11924	TNFRSF9	TTD	2020.06.01	NULL	NULL	CD137 CAR-T Cell	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CART20	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	Autologous T Cells Expressing MET scFv CAR	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:5209	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	CD123CAR-41BB-CD3zeta-EGFRt-expressing T cells	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	Anti-CD30 CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR123	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR123	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR22	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR22	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD22-CART	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	AntiCD19 CART	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD19/CD22 CAR T-Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19/CD22 CAR T-Cells	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD123	NULL	NULL	NULL	NULL	NULL
PROMININ-1	hgnc:9454	PROM1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD133	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD33	NULL	NULL	NULL	NULL	NULL
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting EpCAM	NULL	NULL	NULL	NULL	NULL
T-CELL RECEPTOR BETA CONSTANT 1	hgnc:12156	TRBC1	TTD	2020.06.01	NULL	NULL	TRBC1	NULL	NULL	NULL	NULL	NULL
PNEUMOCYSTIS CARINII DIHYDROPTEROATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dapsone	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
DNA REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dexlansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Doxycycline	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
HUMAN IMMUNODEFICIENCY VIRUS GLYCOPROTEIN 41	NULL	NULL	TTD	2020.06.01	NULL	NULL	Enfuvirtide	rxcui:139896	ENFUVIRTIDE	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fluocinonide	rxcui:4462	FLUOCINONIDE	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flurandrenolide	rxcui:4500	FLURANDRENOLIDE	TRUE	FALSE	FALSE
CYTOMEGALOVIRUS IE2 REGION MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fomivirsen sodium	rxcui:314633	FOMIVIRSEN SODIUM	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	2.100306849	Dichlorphenamide	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	7.501095891	Ethacrynate Sodium	rxcui:4108	ETHACRYNATE SODIUM	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gamma Hydroxybutyric Acid	NULL	NULL	NULL	NULL	NULL
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gemifloxacin	rxcui:138099	GEMIFLOXACIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gemifloxacin	rxcui:138099	GEMIFLOXACIN	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	Insulin-glargine	NULL	NULL	NULL	NULL	NULL
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Itraconazole	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Levofloxacin	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Levofloxacin	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	4.375639269641208	Insulin Susp Isophane Recombinant Human	chembl:CHEMBL1201540	INSULIN SUSP ISOPHANE RECOMBINANT HUMAN	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Loteprednol Etabonate	rxcui:237027	LOTEPREDNOL	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Medrysone	rxcui:29439	MEDRYSONE	TRUE	FALSE	FALSE
BACTERIAL ISOLEUCYL-TRNA SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mupirocin	rxcui:42372	MUPIROCIN	TRUE	FALSE	FALSE
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nifedipine	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pantoprazole	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.069180068	Piperacetazine	rxcui:8338	PIPERACETAZINE	TRUE	FALSE	FALSE
LOW-DENSITY LIPOPROTEIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Porfimer Sodium	rxcui:333848	PORFIMER SODIUM	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	1.779921058837101	Saralasin Acetate	rxcui:7830	SARALASIN ACETATE	TRUE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER A1	hgnc:29	ABCA1	TTD	2020.06.01	NULL	0.7573221812840553	Probucol	rxcui:8699	PROBUCOL	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.596678082	Seroxat	chembl:CHEMBL1708	PAROXETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	1.036335616	Proparacaine	rxcui:34905	PROPARACAINE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tipranavir	rxcui:190548	TIPRANAVIR	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASP-0777	NULL	NULL	NULL	NULL	NULL
ADENOSINE DEAMINASE	hgnc:186	ADA	TTD	2020.06.01	NULL	NULL	GSK2696273	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.1526385791735305	Thiamylal	rxcui:10464	THIAMYLAL	TRUE	FALSE	FALSE
PTPN1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-PTP1Brx	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Moxalactam Disodium	rxcui:258330	DISODIUM LATAMOXEF	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penicillin	wikidata:Q12190	PENICILLIN	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penicillin G Benzathine	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS NS3 HELICASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ombitasvir + paritaprevir + ritonavir	NULL	NULL	NULL	NULL	NULL
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SDZ-GPI-562	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Meclofenamate Sodium	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
BACTERIAL DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Furazolidone	rxcui:4601	FURAZOLIDONE	TRUE	FALSE	FALSE
BACTERIAL DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hydroxystilbamidine Isethionate	ncit:C65871	HYDROXYSTILBAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
FARNESYL PROTEIN TRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-778123	drugbank:DB07227	L-778123	FALSE	FALSE	FALSE
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	EDP-239	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	INS-117548	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	INS-117548	NULL	NULL	NULL	NULL	NULL
HEAT SHOCK PROTEIN 70	hgnc:5232	HSPA1A	TTD	2020.06.01	NULL	NULL	Minnelide 001	NULL	NULL	NULL	NULL	NULL
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	NULL	NsG-0202	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS ENVELOPE GLYCOPROTEIN E2	NULL	NULL	TTD	2020.06.01	NULL	NULL	XTL-6865	drugbank:DB06058	XTL-6865	FALSE	FALSE	FALSE
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	NULL	CXB-909	NULL	NULL	NULL	NULL	NULL
TGF-BETA RECEPTOR TYPE I	hgnc:11772	TGFBR1	TTD	2020.06.01	NULL	5.000730593875666	TEW-7197	ncit:C116357	VACTOSERTIB	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.4167275494896388	G1T28-1	chembl:CHEMBL3894860	TRILACICLIB	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR RECEPTOR TYPE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	VB-111	ncit:C71539	OFRANERGENE OBADENOVEC	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDX899	chembl:CHEMBL1652111	CHEMBL:CHEMBL1652111	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.1458546423213736	Daniquidone	ncit:C66984	DANIQUIDONE	FALSE	FALSE	FALSE
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 5	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 5	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 6	NULL	NULL	NULL	NULL	NULL
IMMUNOGLOBULIN GAMMA FC RECEPTOR IIIA	hgnc:3619	FCGR3A	TTD	2020.06.01	NULL	0.9907107780319716	AFM-13	drugbank:DB17404	AFM-13	FALSE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pargyline	rxcui:7930	PARGYLINE	FALSE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Selegiline	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tranylcypromine	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	AphanamgrandiolA	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzylcinnamate	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Coumaricacid	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PhyllanthoidA	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure1-Chukrasone A	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure2-Artoxanthochromane	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure3-Lycojaponicumin B	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 5-8	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-12	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-12	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-15	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-15	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 7-Vanillic acid	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 7-Vanillyl alcohol	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C11	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C13	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C15	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C17	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C5	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaromatic compound 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fused aromatic compound 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fused ring compound 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure2-J	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	H3K7T	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-EP20142759295NP-1	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-US2012165330(I)	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2012106509CAY10602	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-24	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-3	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-4	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-40	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-45	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-9	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 15	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 9	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Cyclopropyl-spiro piperidine derivative 4	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	NULL	Dihydrobenzoxazine and tetrahydroquinoxaline sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Dihydrobenzoxazine and tetrahydroquinoxaline sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Enzoxazolinone sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.3	hgnc:10590	SCN3A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 4	NULL	NULL	NULL	NULL	NULL
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydrothieno [2,3-e]indazole derivative 4	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Olenolic acid acetate derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2011788838110	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2011796857710	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2011806744710	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2012810604610	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US20130116324 2	NULL	NULL	NULL	NULL	NULL
POLYUBIQUITIN-C	hgnc:12468	UBC	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US20130237529 35	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2011127048 31	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2011127048 33	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2011152671 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2013082253 34	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoxaline derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tihotungstate derivative 1	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	PMID25623274-Compound-WO2014132220C2	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	6,6-fused nitrogenous heterocyclic compound 2	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkynyl-heteroaromatic ring compound 1	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indazole derivative 5	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indazole derivative 5	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-10	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-15c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-19b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-19b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-20a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-23a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-26a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-27	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-33a	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-33b	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-34c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-37c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-37c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-7	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-b]pyridine carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-10	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-105	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-107	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-108	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-113	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo quinoline derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2006015124	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2010127754	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2012135799 42(1.4)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridinone carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 10	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 15	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 17	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 23	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 25	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 6	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 8	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thieno[3,2-c]pyridine-7-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thieno[3,2-c]pyridine-7-carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Cyclic sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Cyclic sulfonamide derivative 2	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Cyclic sulfonamide derivative 3	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Cyclic sulfonamide derivative 4	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 4	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 7	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 8	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 9	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-15	NULL	NULL	NULL	NULL	NULL
SMOOTHENED D473H MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-17	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-17	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-22	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-25	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1361	hgnc:2300	CPB2	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12801	iuphar.ligand:12801	YXG-158	FALSE	FALSE	FALSE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-33	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-37	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-42	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-47	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-47	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-47	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-47	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1360	hgnc:2299	CPB1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:5224	rxcui:6923	METYRAPONE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-48	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-48	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-48	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-48	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-49	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-49	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-49	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-49	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-51	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-51	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-51	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-51	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-56	NULL	NULL	NULL	NULL	NULL
LAMININ RECEPTOR 37/67KDA	hgnc:36809	RPSA2	TTD	2020.06.01	NULL	NULL	PMID25747044-Compound-miRNA	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750TG6-129	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:11287	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750TG7-170	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750TG7-74	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-WO2012177618M4	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-WO2012177618M5	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	PMID25776143-Compound-3	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	Tetra-azabenzo[e]azulene derivative 1	NULL	NULL	NULL	NULL	NULL
JNK-INTERACTING PROTEIN 1 PEPTIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-N1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-N1	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-N2	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1332	hgnc:2272	COX5BP3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8832	iuphar.ligand:8832	COMPOUND 4 [PMID: 16495056]	FALSE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P5	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-Q2	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-U2014S0288042A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140309213A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140336177D	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2012058116B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2012058116C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013062892E	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014015495A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014015495C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014085210A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014085210B	NULL	NULL	NULL	NULL	NULL
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:6193	ncit:C96714	VERLUKAST	FALSE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014126944B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2015017305D	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2015017305E	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2015017305F	NULL	NULL	NULL	NULL	NULL
ZINC FINGER-CONTAINING UBIQUITIN PEPTIDASE 1	hgnc:21224	ZUP1	TTD	2020.06.01	NULL	NULL	Azepan-4-one derivative 1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1879	hgnc:3126	EBF1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:8889	iuphar.ligand:8889	SC-67655	FALSE	FALSE	FALSE
HERPESVIRUS UBIQUITIN-SPECIFIC PROTEASE	hgnc:12630	USP7	TTD	2020.06.01	NULL	NULL	PMID26077642-Compound-Vif2	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	2-pyrazinone derivative 1	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	2-pyrazinone derivative 2	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	2-pyrazinone derivative 6	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	2-pyrazinone derivative 7	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	4-pyridone derivative 1	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Dihydropyrimidinone derivative 1	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Dihydropyrimidinone derivative 2	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 55	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 55	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 58	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 58	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 61	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 61	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 62	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 62	NULL	NULL	NULL	NULL	NULL
NCBIGENE:3244	ncbigene:3244	HPE1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12815	iuphar.ligand:12815	COMPOUND 13 [PMID: 37465299]	FALSE	FALSE	FALSE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 63	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 68	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 34	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	1,5-di-substituted pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	1,5-di-substituted pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	4-(thiazol-5-yl)-pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	4-(thiazol-5-yl)-pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Aminoarylpyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Bipyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Flavopiridol analog 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Flavopiridol analog 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Indole-based analog 11	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	Indole-based analog 11	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Indole-based analog 13	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Indole-based analog 13	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	Indole-based analog 13	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Indole-based analog 13	NULL	NULL	NULL	NULL	NULL
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1161674142382621	IUPHAR.LIGAND:9003	iuphar.ligand:9003	ADL5747	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Isoquinoline 1,3-dione derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Isoquinoline 1,3-dione derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	Isoquinoline 1,3-dione derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	Isoquinoline 1,3-dione derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamide derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamide derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamoyl oxime derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Heteroaryl-substituted urea derivative 2	NULL	NULL	NULL	NULL	NULL
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1548898856510162	IUPHAR.LIGAND:10185	iuphar.ligand:10185	NFP	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Ketoheterocycle derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Piperazine urea derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Piperazine urea derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	PMID26413912-Compound-84	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	PMID26413912-Compound-84	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrimidinyl ethylenediamine derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrimidinyl ethylenediamine derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Tetra-hydro-naphthalene derivative 3	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2603	hgnc:2861	DHFR	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10820	ncit:C65877	ICLAPRIM	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Tetra-hydro-naphthyridine derivative 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	NULL	NPS-2390	NULL	NULL	NULL	NULL	NULL
PSEUDOMONAS LIPOPOLYSACCHARIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Panobacumab	ncit:C95791	PANOBACUMAB	FALSE	FALSE	FALSE
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	Imidazole derivative 11	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Acyl piperidine derivative 2	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Chalcone derivative 5	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1396	hgnc:2360	CRIP1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10243	iuphar.ligand:10243	DO34	FALSE	FALSE	FALSE
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Peptide analog 54	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-11	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-14	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-17	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-2	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-26	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-27	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 28	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 3	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 3	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 32	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 32	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8551	iuphar.ligand:8551	1G244	FALSE	FALSE	FALSE
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 33	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 33	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 8	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 8	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 10	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 8	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Chromene derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Diarylamine and arylheteroarylamine pyrazole derivative 3	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 11	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 12	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 15	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 5	NULL	NULL	NULL	NULL	NULL
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic-tetracyclic tetrahydrofuran derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	PMID26609882-Compound-34	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	PMID26609882-Compound-36	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 73	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolidine derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolidine derivative 2	NULL	NULL	NULL	NULL	NULL
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.019665794	IUPHAR.LIGAND:7295	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 7	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 9	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 10	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 11	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 13	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 2	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 7	NULL	NULL	NULL	NULL	NULL
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.011799477	IUPHAR.LIGAND:7427	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 8	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-109	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-111	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-11b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-11c	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-121	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-123	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure11Ala up	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure12bottommiddle01	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle10	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2833	hgnc:4540	CXCR3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8796	iuphar.ligand:8796	COMPOUND 6EE [PMID: 22364528]	FALSE	FALSE	FALSE
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle11	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle12	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle13	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	3-(phenoxymethyl) benzylamine derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	3-(phenoxymethyl) benzylamine derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Monoamine derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Monoamine derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-117	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-123	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-125	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-127	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-47	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-H	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2832	hgnc:4530	NPBWR2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8796	iuphar.ligand:8796	COMPOUND 6EE [PMID: 22364528]	FALSE	FALSE	FALSE
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Polyhydroxy benzamide derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Polyhydroxy benzamide derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 15	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 17	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 19	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 20	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 23	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 24	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 26	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 28	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 34	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 6	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	2,2-dimethylbenzopyran derivative 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-24	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1616	hgnc:2681	DAXX	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8620	iuphar.ligand:8620	S136492	FALSE	FALSE	FALSE
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 4	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 5	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Piperazine derivative 5	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Piperazine urea derivative 4	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Piperidine derivative 3	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	PMID26936077-Compound-34	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 11	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Aryl cyclopropylamine derivative 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Benzenamine derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 8	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-7	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 18	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1B	hgnc:21577	KDM1B	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-10	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-15	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-15	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-16	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-16	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-19	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-19	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 4	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 4	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 4	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 6	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 7	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 9	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-30	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-34	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-37	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-37	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Fused benzoheterocycle amide derivative 2	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Indazole amide derivative 1	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Macrolactam derivative 4	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Pyrazole N-1 aryl and heteroaryl derivative 1	NULL	NULL	NULL	NULL	NULL
IL-1 RECEPTOR-ASSOCIATED KINASE 1	hgnc:6112	IRAK1	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine and thienopyrimidine amide derivative 2	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine and thienopyrimidine amide derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [4,3-a]quinoxaline derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [4,3-a]quinoxaline derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	PMID27321640-Compound-76	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 3	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-12	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR BETA	hgnc:9865	RARB	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-7	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-1	hgnc:10430	RPS6KA1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Benzofurans derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Cycloalkyl acid derivative 1	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-101	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-95	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-96	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-98	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	PMID27537201-Compound-Figure15a	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	PMID27537201-Compound-Figure17	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Quinoline derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Quinoline derivative 17	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Sterol derivative 2	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Sterol derivative 3	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	Imidamide derivative 1	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	Methylbenzenesulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-3	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-7	NULL	NULL	NULL	NULL	NULL
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	PMID27551786-Compound-106	NULL	NULL	NULL	NULL	NULL
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	PMID27551786-Compound-138	NULL	NULL	NULL	NULL	NULL
RECEPTOR-INTERACTING PROTEIN 1	hgnc:10019	RIPK1	TTD	2020.06.01	NULL	NULL	Tricyclic compound 9	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Indole-based analog 5	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-76	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine acetamide analog 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine acetamide analog 5	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine acetamide analog 7	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1825	hgnc:3037	DSC3	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Phenylpurine acetamide analog 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Phenylpurine acetamide analog 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-4	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-61	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 3	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 11	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 2	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 15	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 15	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl amide derivative 2	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl amide derivative 3	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Chlorobenzamide derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Dihydroisoquinoline carboxamide analog 1	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-21	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	modulator	0.5000730593875666	IUPHAR.LIGAND:9222	iuphar.ligand:9222	EAI045	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-21	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-21	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-22	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-5	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:6015	iuphar.ligand:6015	PD 158780	FALSE	FALSE	FALSE
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloalkyl nitrile pyrazolo pyridone derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloalkyl nitrile pyrazolo pyridone derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoxazole derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoxazole derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Isoxazole derivative 1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:7944	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Example19	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Example19	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure2Example1-1left	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure2Example1-1left	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure2Example1-1right	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure2Example1-1right	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure3CompoundI-165	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure3CompoundI-165	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure6Example2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure7Example63	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure7Example63	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.015153729	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 1	NULL	NULL	NULL	NULL	NULL
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	NULL	1,2,4-triazolo[1,5a]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-triazolo[1,5a]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	1,2,4-triazolo[1,5a]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:12994	iuphar.ligand:12994	CAY10499	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	NULL	1,2,4-triazolo[1,5a]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-triazolo[1,5a]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 2	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3H)-one derivative 1	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Imidazo pyridine derivative 6	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Oxazolo[3,4-a]pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Oxazolo[3,4-a]pyrazine derivative 5	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-5	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indazole derivative 6	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2535	hgnc:4040	FZD2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8797	iuphar.ligand:8797	COMPOUND 13 [PMID: 17502136]	FALSE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indirubin derivative 2	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Maleimides derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Maleimides derivative 2	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Maleimides derivative 3	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-naphtyl-N-benzylurea derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-15	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-19	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazole and benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoline derivative 15	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Spiroquinolone derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic 5-quinolone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Aza-phenalene-3-ketone derivative 1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:10043	iuphar.ligand:10043	SETOGEPRAM	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Benzimidazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Dihydrodiazepinocarbazolone derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Dihydropyrido phthalazinone derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Phthalazine derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Phthalazine ketone derivative 3	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-23	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-37	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 2	hgnc:272	PARP2	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-37	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2024	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.092606122	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
TANKYRASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-37	NULL	NULL	NULL	NULL	NULL
TANKYRASE-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-37	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-38	NULL	NULL	NULL	NULL	NULL
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:6499	iuphar.ligand:6499	TRANS-2-METHYLCROTONIC ACID	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-V	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Quinazolinedione derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Tetra-cyclic pyridophthalazinone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 2	hgnc:272	PARP2	TTD	2020.06.01	NULL	NULL	Tetra-cyclic pyridophthalazinone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 13	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azaindole derivative 5	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azole benzene derivative 2	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azole benzene derivative 4	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 3	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 6	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-130	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	4-aryl quinol derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	4-aryl quinol derivative 7	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Bis-sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Bis-sulfonamide derivative 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Disulfide compound 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Metal complex derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Palmarumycin derivative 4	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-18	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-29	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-30	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-32	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Diazepinone derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Diazepinone derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Ethynyl compound 5	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-a]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyridine derivative 12	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyridine derivative 16	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 5	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-pyrazolopyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 11	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 4	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 5	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 9	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 1	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 10	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 2	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 5	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20100022547C87	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20100022547C88	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20120264760C80	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20120264760C86	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20120264760C87	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20120264760C88	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 2	hgnc:6053	IMPDH2	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 1	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 11	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 16	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 18	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 4	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 5	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 9	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 2	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 2	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 3	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 3	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32c	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32c	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32e	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32e	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32n	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32n	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32x	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32x	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32z	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32z	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33b	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridazine derivative 1	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2 G2019S MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
CLOSTRIDIUM DIFFICILE TOXIN B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bezlotoxumab	rxcui:1855048	BEZLOTOXUMAB	TRUE	FALSE	FALSE
DYSTROPHIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Eteplirsen	rxcui:1810569	ETEPLIRSEN	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 6	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-34	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-35	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-38	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-45	NULL	NULL	NULL	NULL	NULL
EZH2 Y641N MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-45	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-55	NULL	NULL	NULL	NULL	NULL
EZH2 Y641N MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-55	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-56	NULL	NULL	NULL	NULL	NULL
EZH2 Y641N MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-56	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-57	NULL	NULL	NULL	NULL	NULL
EZH2 Y641N MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-57	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-Figure3bI	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-Figure3bIII	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-Figure5aVIII	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazopyrimidinone derivative 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Octahydro-pyrrolo[3,4-c]-pyrrole derivative 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-11	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-22	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidinone derivative 5	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-carboline derivative 1	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DLG] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-phenyl-1,3,4-triazole derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	1-phenyl-1,3,4-triazole derivative 2	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DUAL DLG AND ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	3-phenyl propanoic derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	3-phenyl propanoic derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Benzamide derivative 5	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Benzamide derivative 6	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazole derivative 1	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DUAL DLG AND ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	Naphthalene derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Naphthalene derivative 1	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-12	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-12	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-35	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-35	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-36	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-36	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-50	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-50	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DUAL DLG AND ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-59	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-59	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-9	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-9	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-91	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-93	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Thiazole derivative 3	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vinyl sulfone derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Vinyl sulfone derivative 1	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	PMID28460551-Compound-2	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C ALPHA	hgnc:9393	PRKCA	TTD	2020.06.01	NULL	NULL	PMID28460551-Compound-3	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	N-(arylamino)sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	PMID28594589-Compound-TABLE3C1	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Right	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Right	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 2	hgnc:3093	DYRK2	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Right	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 3	hgnc:3094	DYRK3	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme21Right	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme24-11H-pyrido[4,3-a]carbazole	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme25-3	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme25-3	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme2WO2012/098065upper	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme2WO2012/098065upper	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme6Pyrrolo[2,3-d]pyrimidines	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme7WO2012/098070upper	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme7WO2012/098070upper	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT1610	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT1610	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT5372	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT5372	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-38	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-41	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-44	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-52	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-56	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-57	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-59	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-60	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-63	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-67	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-68	NULL	NULL	NULL	NULL	NULL
CASPASE-1	hgnc:1499	CASP1	TTD	2020.06.01	NULL	NULL	Ac-YVAD-FMK	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	Beta-naphthylacetic acids derivative 1	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	Indomethacin analog 1	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	N-(benzimidazole/indole) benzoic acid derivative 1	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	N-(naphthylamino)-benzoate derivative 1	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	N-(phenylamino)-benzoate derivative 1	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 12	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 9	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Triazole derivative 6	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidinyl-piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 12	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 13	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 14	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 15	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-14	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-14	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-7a	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-21	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-29	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-33	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-39	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-4	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-52	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-53	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-58	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-6	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-72	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-10	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-12	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-15	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-21	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-3	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-30	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-31	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-36	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-39	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-4	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-40	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-41	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-44	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-11	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-11	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-11	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-11	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-14	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-28	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-28	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 11	hgnc:19086	HDAC11	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-36	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-36	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-38a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-38a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-55	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-55	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-55	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-65a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-65a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 5	hgnc:14068	HDAC5	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-67	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-69	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 16	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30074415-Compound-12	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	1,2,4-oxadiazole derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-oxadiazole derivative 4	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-oxadiazole derivative 5	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	1,3,4-oxadiazole derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3,4-oxadiazole derivative 4	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3,4-thiadiazole derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3,4-thiadiazole derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3-dihydroxy phenyl derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3-dihydroxy phenyl derivative 2	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example3	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example44	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example54	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example59	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example8	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Benzamide derivative 8	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 8	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Benzamide derivative 9	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 9	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 3	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 3	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 3	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazinyl norbenzomorphane compound 2	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-14	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID30259754-Compound-LY2562175	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID30259754-Compound-WAY-362450	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-12	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-13	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-14	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-22b	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-41	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2005070959	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2013119856	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.2373228078449469	Candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Celtura	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.8468979231563628	Dimenhydrinate	rxcui:3444	DIMENHYDRINATE	TRUE	FALSE	FALSE
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fibrinolysin	ncit:C171921	FIBRINOLYSIN	FALSE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.8607814956671229	Ethynodiol Diacetate	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.085796848	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.3571950424196904	Fondaparinux sodium	rxcui:321208	FONDAPARINUX	TRUE	FALSE	FALSE
IMMUNOGLOBULIN UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Immune globulin intravenous	rxcui:42386	IMMUNOGLOBULINS, INTRAVENOUS	FALSE	FALSE	FALSE
ACETYLCHOLINE RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Incobotulinum toxin A	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoflurane	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
HEDGEHOG SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	Itraconazole	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
GLUTAMINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-alanyl-l-glutamine	rxcui:1359422	ALANYLGLUTAMINE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Levocetirizine dihydrochloride	rxcui:356887	LEVOCETIRIZINE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	0.9723642821424908	Minaprine	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	IM19 CAR-T	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1226814748497534	Nomegestrol acetate	rxcui:53744	NOMEGESTROL ACETATE	FALSE	FALSE	FALSE
TRYPTASE ALPHA/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pentamidine	rxcui:7994	PENTAMIDINE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pentazocine	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
STREPTOCOCCUS DIPHTHERIA PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Prevnar	ncit:C38141	PNEUMOCOCCAL 7-VALENT CONJUGATE VACCINE	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.016131389	Pentoxifylline	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.012208247	Pseudoephedrine	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfamethoxazole	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	TachoComb	NULL	NULL	NULL	NULL	NULL
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Teicoplanin	rxcui:57021	TEICOPLANIN	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Telithromycin	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
GROWTH HORMONE-RELEASING HORMONE RECEPTOR	hgnc:4266	GHRHR	TTD	2020.06.01	NULL	19.69037671338543	Sermorelin	rxcui:56188	SERMORELIN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M2	hgnc:1951	CHRM2	TTD	2020.06.01	NULL	0.1151484018326633	Scopolamine	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.063331621	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.1693795846312726	Tetrodotoxin	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zalcitabine	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
INFLUENZA NEURAMINIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zanamivir	rxcui:69722	ZANAMIVIR	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zopiclone	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
CHYMOTRYPSIN	hgnc:1440	CALCR	TTD	2020.06.01	NULL	NULL	Pancrecarb	NULL	NULL	NULL	NULL	NULL
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	NULL	[N-methyl-3H(3)]AZ-10419369	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	1069C	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	A-837093	chembl:CHEMBL469738	CHEMBL:CHEMBL469738	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	AST-005	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	NULL	BCI-632	NULL	NULL	NULL	NULL	NULL
THROMBOPOIETIN	hgnc:11795	THPO	TTD	2020.06.01	NULL	NULL	BVI-007	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 9	hgnc:1610	CCR9	TTD	2020.06.01	NULL	NULL	CCX-025	NULL	NULL	NULL	NULL	NULL
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	CJ-12255	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	CPC-212	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	CPC-250	NULL	NULL	NULL	NULL	NULL
TISSUE FACTOR PATHWAY INHIBITOR	hgnc:11760	TFPI	TTD	2020.06.01	NULL	2.763561643983921	BAX-499	chembl:CHEMBL4297890	ARC-19499	FALSE	FALSE	FALSE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	2.019525817	CJM112	ncit:C146808	ANTI-IL17A MONOCLONAL ANTIBODY CJM112	FALSE	FALSE	FALSE
CRP MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-CRP	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	LY-2334737	drugbank:DB12906	LY-2334737	FALSE	FALSE	FALSE
GLYCINAMIDE RIBONUCLEOTIDE FORMYLTRANSFERASE	hgnc:4163	GART	TTD	2020.06.01	NULL	NULL	LY309887	NULL	NULL	NULL	NULL	NULL
SERUM AMYLOID P-COMPONENT	hgnc:584	APCS	TTD	2020.06.01	NULL	13.12691780892362	GSK-2315698	ncit:C153209	MIRIDESAP	FALSE	FALSE	FALSE
EXTRACELLULAR MATRIX RECEPTOR III	hgnc:1681	CD44	TTD	2020.06.01	NULL	NULL	A-6	NULL	NULL	NULL	NULL	NULL
B2 BRADYKININ RECEPTOR	hgnc:1030	BDKRB2	TTD	2020.06.01	NULL	4.375639269641208	Anatibant	ncit:C79554	ANATIBANT	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	APH-0812	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	APH-0812	NULL	NULL	NULL	NULL	NULL
NICOTINIC ACID RECEPTOR	hgnc:24827	HCAR2	TTD	2020.06.01	NULL	NULL	ARI-3037MO	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	Girentuximab I-124	ncit:C53407	IODINE I-124 GIRENTUXIMAB	FALSE	FALSE	FALSE
SOLUBLE GUANYLYL CYCLASE	hgnc:4689	GUCY2D	TTD	2020.06.01	NULL	17.50255707856483	FK-409	chembl:CHEMBL173729	CHEMBL:CHEMBL173729	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	3.281729452230906	CRYPTOPHYCIN 52	ncit:C1826	CRYPTOPHYCIN 52	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IMO-8400	ncit:C114975	BAZLITORAN	FALSE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	Inecalcitol oral	NULL	NULL	NULL	NULL	NULL
AMINOPEPTIDASE N	hgnc:500	ANPEP	TTD	2020.06.01	NULL	NULL	IP10.C8-1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	IP10.C8-1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	K-134	drugbank:DB12685	K-134	FALSE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	WCK-771	ncit:C83879	LEVONADIFLOXACIN	FALSE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	WCK-771	ncit:C83879	LEVONADIFLOXACIN	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Xmab 5871	NULL	NULL	NULL	NULL	NULL
IMMUNOGLOBULIN GAMMA FC RECEPTOR IIB	hgnc:3618	FCGR2B	TTD	2020.06.01	NULL	NULL	Xmab 5871	NULL	NULL	NULL	NULL	NULL
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	NULL	Plasminogen concentrate	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	NULL	13-cis-retinoic acid, UCSD	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	modulator	1.250182648468916	IUPHAR.LIGAND:11622	ncit:C170744	ALOFANIB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Avastin+/-Tarceva	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED CALCIUM CHANNEL ALPHA-2/DELTA-1	hgnc:1399	CACNA2D1	TTD	2020.06.01	NULL	2.500365296937833	Mirogabalin	ncit:C170186	MIROGABALIN	FALSE	FALSE	FALSE
E-SELECTIN	hgnc:10718	SELE	TTD	2020.06.01	NULL	6.364566210387211	GMI-1070	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	NULL	Rosiglitazone + metformin	NULL	NULL	NULL	NULL	NULL
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	NULL	Rosiglitazone + metformin	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	NULL	Rosiglitazone + metformin	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	Rosiglitazone + metformin	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Rosiglitazone + metformin	NULL	NULL	NULL	NULL	NULL
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	NULL	SPD-465	NULL	NULL	NULL	NULL	NULL
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD38	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	Felbinac prodrug	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	2.100306849	Cutamesine	ncit:C83642	CUTAMESINE	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.028199609	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:1387	hgnc:2348	CREBBP	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8752	iuphar.ligand:8752	ML355	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.9907107780319716	SK-7068	chembl:CHEMBL152543	CHEMBL:CHEMBL152543	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:10454	iuphar.ligand:10454	ULOTARONT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:3925	iuphar.ligand:3925	[3H]NLX-112	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:1	ncit:C80760	FLESINOXAN	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.050294704	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:13	iuphar.ligand:13	FG-5893	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:9788	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:32	iuphar.ligand:26	S-15535	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.015608701	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.033295923	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.2108741816694558	IUPHAR.LIGAND:76	iuphar.ligand:76	SB 649915	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:218	iuphar.ligand:218	2-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.02875557	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.021554873	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.021554873	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:12313	iuphar.ligand:12313	COMPOUND 29 [PMID: 36356320]	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.034184682	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1025540453822158	IUPHAR.LIGAND:5691	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.026319635	IUPHAR.LIGAND:5679	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:12010	drugbank:DB15343	TUSPETINIB	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.2792961235941196	IUPHAR.LIGAND:3927	iuphar.ligand:3927	BRL-54443	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:175	iuphar.ligand:175	SPIRAMIDE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.021933029	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.018942161	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.069089041	IUPHAR.LIGAND:142	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:225	ncit:C74393	PIBOSEROD	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.016743518	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.078958904	IUPHAR.LIGAND:3	iuphar.ligand:3	1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.048260727	IUPHAR.LIGAND:109	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.032173818	IUPHAR.LIGAND:2	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.020320306	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:11660	iuphar.ligand:11660	COMPOUND 38K [PMID: 34351741]	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:247	iuphar.ligand:247	GR 113808	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.059397818	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.048483538	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:12	iuphar.ligand:12	EMDT	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.051177067	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1766118064547324	IUPHAR.LIGAND:5678	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.068369364	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
NCBIGENE:780	hgnc:2730	DDR1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8776	iuphar.ligand:8776	PAK-104P	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	NULL	3.750547945	IUPHAR.LIGAND:10074	iuphar.ligand:10074	ACHE REACTIVATOR 2	FALSE	FALSE	FALSE
NCBIGENE:80	hgnc:153	ACTG1P8	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:4358	iuphar.ligand:4358	CXCL12&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.008621949	IUPHAR.LIGAND:5698	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	modulator	0.9211872146613068	IUPHAR.LIGAND:9429	iuphar.ligand:9429	MIRANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:9429	iuphar.ligand:9429	MIRANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:7944	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
NCBIGENE:1662	hgnc:2735	DDX10	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9687	iuphar.ligand:9687	GI254023X	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:10437	iuphar.ligand:10437	COMPOUND E22 [PMID: 31298542]	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:7902	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	modulator	1.029562181092048	IUPHAR.LIGAND:9429	iuphar.ligand:9429	MIRANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:9429	iuphar.ligand:9429	MIRANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:12722	iuphar.ligand:12722	HU7691	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.055563673	IUPHAR.LIGAND:6058	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:7887	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:7887	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.1100789753368857	IUPHAR.LIGAND:495	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.045032308	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:11852	iuphar.ligand:11852	COMPOUND 39 [PMID: 34982553]	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.16256245	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:6057	iuphar.ligand:6057	VEGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:685	hgnc:1121	BTC	GuideToPharmacology	2024.1	blocker	0.3860858179095184	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	modulator	0.6035364509849942	IUPHAR.LIGAND:9445	iuphar.ligand:9445	PD81723	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.086219493	IUPHAR.LIGAND:422	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:3289	iuphar.ligand:3289	BAY 60-6583	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:5599	iuphar.ligand:5599	HEMADO	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:5599	iuphar.ligand:5599	HEMADO	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:403	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:1018	iuphar.ligand:1018	[3H]FMET-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:414	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:5599	iuphar.ligand:5599	HEMADO	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1136529680426287	IUPHAR.LIGAND:474	iuphar.ligand:474	MRS1523	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:5618	iuphar.ligand:5618	KF26777	FALSE	FALSE	FALSE
NCBIGENE:2720	hgnc:4298	GLB1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10445	iuphar.ligand:10445	COMPOUND 23 [PMID: 31398032]	FALSE	FALSE	FALSE
NCBIGENE:2719	hgnc:4451	GPC3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11939	iuphar.ligand:11939	AZ13824374	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12082	iuphar.ligand:12082	TUVUSERTIB	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:5827	iuphar.ligand:5827	GROUP E 1682-2106 [PMID:16118363]	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:8768	iuphar.ligand:8768	COMPOUND 38 [PMID: 20817473]	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:8060	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.076765601	IUPHAR.LIGAND:8353	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6242	iuphar.ligand:6242	SERUM AMYLOID A	FALSE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.1215455352678113	IUPHAR.LIGAND:6044	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2901	hgnc:4583	GRIK5	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9143	iuphar.ligand:9143	EXAMPLE 1.11 [WO2014139978]	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:11624	iuphar.ligand:11624	NINGETINIB	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:11665	iuphar.ligand:11665	XMD-12	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:6176	iuphar.ligand:6176	BANTAG-1	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:6166	iuphar.ligand:6166	PHYLLOLITORIN	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:4865	iuphar.ligand:4865	AMYLOID &BETA;	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:635	iuphar.ligand:635	D-NAL-CYS-TYR-D-TRP-LYS-VAL-CYS-NAL-NH2	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:11557	iuphar.ligand:11557	LY3202626	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9197	iuphar.ligand:9197	COMPOUND 9 [PMID: 26937601]	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7855	iuphar.ligand:7855	EXAMPLE 41 [WO2012028563]	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1031	iuphar.ligand:1031	ANNEXIN I	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.091796628	IUPHAR.LIGAND:2561	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.5645986154375752	IUPHAR.LIGAND:12578	iuphar.ligand:12578	CIMATEROL	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:563	rxcui:597	ALPRENOLOL	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:562	iuphar.ligand:562	[125I]ICYP	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.2206204673768676	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:9511	iuphar.ligand:9511	ACT-389949	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:8943	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.017715139	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2722	ncbigene:2722	GLC1B	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8306	iuphar.ligand:8306	COMPOUND 7 [PMID: 25719566]	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:8958	iuphar.ligand:8958	LIFIRAFENIB	FALSE	FALSE	FALSE
NCBIGENE:2599	hgnc:1375	CA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492008	IUPHAR.LIGAND:6849	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:7452	iuphar.ligand:7452	TAFLUPROST ACID	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:7046	iuphar.ligand:7046	INDISULAM	FALSE	FALSE	FALSE
NCBIGENE:3093	hgnc:4914	UBE2K	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:3310	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.030598876	IUPHAR.LIGAND:6849	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.1615620653405984	IUPHAR.LIGAND:7047	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	0.6731752722524935	IUPHAR.LIGAND:3308	rxcui:407990	CINACALCET	TRUE	FALSE	FALSE
NCBIGENE:1623	hgnc:2691	DBIP2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6515	iuphar.ligand:6515	ISATIN SULFONAMIDE 34 [PMID: 11384246]	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:713	iuphar.ligand:713	2-METHYL-3-PHENETHYL-3H-PYRIMIDIN-4-ONE	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:1958	rxcui:283810	BIMATOPROST	TRUE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:12647	iuphar.ligand:12647	ACT-709478	FALSE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7724	iuphar.ligand:7724	TTA-A2	FALSE	FALSE	FALSE
NCBIGENE:2345	ncbigene:2345	FNZ	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:11713	iuphar.ligand:11713	&BETA;-SECRETASE INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:10348	iuphar.ligand:10348	BAY-593074	FALSE	FALSE	FALSE
NCBIGENE:390	hgnc:671	RND3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:4269	iuphar.ligand:4269	NNC55-0396	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.018501646	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:391	hgnc:672	RHOG	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:4269	iuphar.ligand:4269	NNC55-0396	FALSE	FALSE	FALSE
NCBIGENE:391	hgnc:672	RHOG	GuideToPharmacology	2024.1	blocker	0.5147810905460245	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:9706	iuphar.ligand:9706	JWH-018	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:865	iuphar.ligand:865	GW-5823	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:8409	iuphar.ligand:8409	DESULFATED GASTRIN-34	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:891	ncit:C81601	LORGLUMIDE	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:878	ncit:C98235	DEVAZEPIDE	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:6667	iuphar.ligand:6667	[125I]-BDZ2	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.2386712328895204	IUPHAR.LIGAND:4156	iuphar.ligand:4156	CGS8216	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:767	iuphar.ligand:767	BX 471	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:10416	iuphar.ligand:10416	GSK2239633A	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.099446347	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6103	iuphar.ligand:6103	M1152	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6083	iuphar.ligand:6083	GALANIN(7-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:802	iuphar.ligand:802	[3H]ANCRIVIROC	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:783	iuphar.ligand:783	TAK-779	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6099	iuphar.ligand:6099	M242	FALSE	FALSE	FALSE
NCBIGENE:64	hgnc:137	ACTBP4	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:3655	iuphar.ligand:3655	[125I]CCL19 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2786	hgnc:4407	GNG4	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:7675	rxcui:2099295	MOXETUMOMAB PASUDOTOX	TRUE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8218	iuphar.ligand:8218	COMPOUND 1 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:11417	iuphar.ligand:11417	SPEXIN-1	FALSE	FALSE	FALSE
NCBIGENE:1508	hgnc:2527	CTSB	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8204	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:3861	iuphar.ligand:3861	C7	FALSE	FALSE	FALSE
NCBIGENE:2733	hgnc:4315	GLE1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8951	iuphar.ligand:8951	NVS-1	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3187	iuphar.ligand:3187	DIGERANYL BISPHOSPHONATE	FALSE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:12620	iuphar.ligand:12620	CIRTUVIVINT	FALSE	FALSE	FALSE
NCBIGENE:1990	hgnc:3308	CELA1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8115	iuphar.ligand:8115	COMPOUND 2 [PMID: 22560567]	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	NULL	0.2500365296937833	IUPHAR.LIGAND:4077	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
NCBIGENE:1993	hgnc:3313	ELAVL2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12974	iuphar.ligand:12974	MW01	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.2035181055647073	IUPHAR.LIGAND:7067	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:4182	iuphar.ligand:4182	DIPHENYLAMINE-2-CARBOXYLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:3248	hgnc:5154	HPGD	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:11729	iuphar.ligand:11729	MK-8262	FALSE	FALSE	FALSE
NCBIGENE:698	ncbigene:698	BTS1	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8760	iuphar.ligand:8760	DUP-714	FALSE	FALSE	FALSE
NCBIGENE:1255	ncbigene:1255	CNA1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8955	iuphar.ligand:8955	MS023	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.014198938	IUPHAR.LIGAND:2768	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:2364	hgnc:3872	FRA1E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:6550	iuphar.ligand:6550	COMPOUND 57 [PMID: 20121197]	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:11747	iuphar.ligand:11747	BPR1R024	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.070765056	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.090843722	IUPHAR.LIGAND:5230	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2335	hgnc:3778	FN1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:8619	iuphar.ligand:8619	COMPOUND 28 [PMID: 16460935]	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:924	iuphar.ligand:924	[125I]ASTRESSIN	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:2894	rxcui:278567	VALDECOXIB	TRUE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:919	iuphar.ligand:919	UROCORTIN 1	FALSE	FALSE	FALSE
NCBIGENE:2850	hgnc:4482	GPR27	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:8361	rxcui:1726104	ELOTUZUMAB	TRUE	FALSE	FALSE
NCBIGENE:3216	hgnc:5117	HOXB6	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12314	iuphar.ligand:12314	COMPOUND 27 [PMID: 36449304]	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:11065	drugbank:DB08463	(2R)-2-({9-(1-METHYLETHYL)-6-[(4-PYRIDIN-2-YLBENZYL)AMINO]-9H-PURIN-2-YL}AMINO)BUTAN-1-OL	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:10081	iuphar.ligand:10081	KINASE INHIBITOR 2 [PMID: 30199702]	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	0.251232877	IUPHAR.LIGAND:3329	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:8691	iuphar.ligand:8691	BEGELOMAB	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8402	ncit:C174662	OMARIGLIPTIN	FALSE	FALSE	FALSE
NCBIGENE:2005	hgnc:3326	ELK4	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8207	iuphar.ligand:8207	COMPOUND 5G [PMID: 20483621]	FALSE	FALSE	FALSE
NCBIGENE:2005	hgnc:3326	ELK4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11114	iuphar.ligand:11114	DCLK1-IN-1	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	0.052507671	IUPHAR.LIGAND:1909	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:1880	iuphar.ligand:1880	L-888,291	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:1897	iuphar.ligand:1897	BWA868C	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:1903	iuphar.ligand:1903	15(S)-15-METHYL-PGD2	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:1879	iuphar.ligand:1879	L-644,698	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:10169	ncit:C152874	VIDUPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.058341857	IUPHAR.LIGAND:2	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:9189	iuphar.ligand:9189	HS665	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:9190	iuphar.ligand:9190	COMPOUND 3 [PMID: 23134120]	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:951	iuphar.ligand:951	7-TRANS-OH-PIPAT	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.058997383	IUPHAR.LIGAND:3298	iuphar.ligand:3298	[3H]PD128907	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4079	iuphar.ligand:4079	[3H]CGP61594	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:956	iuphar.ligand:956	(+)-SCH-23390	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.2333674277141977	IUPHAR.LIGAND:44	iuphar.ligand:44	NAFADOTRIDE	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.011799477	IUPHAR.LIGAND:941	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:11959	iuphar.ligand:11959	EGIS-11150	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.001761116	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:983	iuphar.ligand:983	NEMONAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.5707355569097228	IUPHAR.LIGAND:7683	iuphar.ligand:7683	PF-592379	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.08780547	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.2734774543525755	IUPHAR.LIGAND:4084	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7003	iuphar.ligand:7003	PLUMBAGIN	FALSE	FALSE	FALSE
NCBIGENE:2012	hgnc:3333	EMP1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10081	iuphar.ligand:10081	KINASE INHIBITOR 2 [PMID: 30199702]	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.2734774543525755	IUPHAR.LIGAND:727	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
NCBIGENE:1832	hgnc:3052	DSP	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:4092	iuphar.ligand:4092	[3H]UBP310	FALSE	FALSE	FALSE
NCBIGENE:1833	hgnc:3053	EPYC	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7011	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	NULL	0.5000730593875666	IUPHAR.LIGAND:4917	iuphar.ligand:4917	EPIGEN	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:1922	iuphar.ligand:1922	SC-19220	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.064033745	IUPHAR.LIGAND:1916	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4208	iuphar.ligand:4208	GV196771A	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.2651902587661338	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:7903	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	NULL	0.4526523382387456	IUPHAR.LIGAND:5029	iuphar.ligand:5029	NEUREGULIN-2	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:9929	iuphar.ligand:9929	XILIERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.3621218705909966	IUPHAR.LIGAND:7647	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.053253216	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:9343	iuphar.ligand:9343	DESLORELIN	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:9711	rxcui:38260	TIBOLONE	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:10369	rxcui:10032	STANOZOLOL	TRUE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:8908	iuphar.ligand:8908	GSK5182	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	modulator	0.7955707762984014	IUPHAR.LIGAND:1179	iuphar.ligand:1179	CMPD-1	FALSE	FALSE	FALSE
NCBIGENE:2015	hgnc:3336	ADGRE1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3760	iuphar.ligand:3760	[125I][ALA1,3,11,15]ET-1	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1179	iuphar.ligand:1179	CMPD-1	FALSE	FALSE	FALSE
NCBIGENE:2017	hgnc:3338	CTTN	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9544	iuphar.ligand:9544	GSK2656157	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:11130	iuphar.ligand:11130	COMPOUND 25 [PMID: 32687365]	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	NULL	0.8334550989792776	IUPHAR.LIGAND:4075	iuphar.ligand:4075	[3H]SYM2081	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3179	iuphar.ligand:3179	NE58043	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	0.089756703	IUPHAR.LIGAND:1016	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:4197	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.062808219	IUPHAR.LIGAND:4193	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.040640612	IUPHAR.LIGAND:7111	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.1422972120208523	IUPHAR.LIGAND:4090	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:12118	iuphar.ligand:12118	COMPOUND 20 [PMID: 35584373]	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.2134458180312784	IUPHAR.LIGAND:4321	iuphar.ligand:4321	TETRAHYDRODEOXYCORTICOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.3017682254924971	IUPHAR.LIGAND:4321	iuphar.ligand:4321	TETRAHYDRODEOXYCORTICOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	agonist	0.2011788169949981	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	inhibitor	0.2586584789935689	IUPHAR.LIGAND:2312	iuphar.ligand:2312	BICUCULLINE	FALSE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:721	rxcui:1091	ARGININE	TRUE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.075442056	IUPHAR.LIGAND:4367	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:416	hgnc:721	ARSF	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:4184	iuphar.ligand:4184	DS2	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:4067	iuphar.ligand:4067	(&PLUSMN;)-CIS-2-CAMP	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6117	iuphar.ligand:6117	[125I][TYR26]GALANIN (PIG)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6122	iuphar.ligand:6122	GALP(3-32) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6109	iuphar.ligand:6109	[N-ME,DES-SAR]GAL-B2	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:1595	ncit:C81534	ACIFRAN	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:6128	iuphar.ligand:6128	SCH 202596	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3193	iuphar.ligand:3193	COMPOUND 19 [PMID: 18800762]	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:12413	iuphar.ligand:12413	PF-6870961	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.1023541349623674	IUPHAR.LIGAND:9745	rxcui:1999420	MACIMORELIN	TRUE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.4688184931758437	IUPHAR.LIGAND:4219	iuphar.ligand:4219	IDRA-21	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	0.078722146	IUPHAR.LIGAND:1059	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:4219	iuphar.ligand:4219	IDRA-21	FALSE	FALSE	FALSE
NCBIGENE:875	hgnc:1550	CBS	GuideToPharmacology	2024.1	NULL	2.625383561784724	IUPHAR.LIGAND:4643	iuphar.ligand:4643	[3H]2-DEOXYGLUCOSE	FALSE	FALSE	FALSE
NCBIGENE:878	ncbigene:878	CCA1	GuideToPharmacology	2024.1	NULL	13.12691780892362	IUPHAR.LIGAND:4643	iuphar.ligand:4643	[3H]2-DEOXYGLUCOSE	FALSE	FALSE	FALSE
NCBIGENE:2905	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:9827	iuphar.ligand:9827	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:875	hgnc:1550	CBS	GuideToPharmacology	2024.1	modulator	10.50153424713889	IUPHAR.LIGAND:8885	iuphar.ligand:8885	COMPOUND 30 [PMID: 22468970]	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:8643	iuphar.ligand:8643	ZK216348	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	modulator	0.760980743	IUPHAR.LIGAND:7846	iuphar.ligand:7846	TCN-201	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:4078	iuphar.ligand:4078	[3H]CGP39653	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:4078	iuphar.ligand:4078	[3H]CGP39653	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:4290	iuphar.ligand:4290	PREGNENOLONE SULPHATE	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:4072	iuphar.ligand:4072	(12E,20Z,18S)-8-HYDROXYVARIABILIN	FALSE	FALSE	FALSE
NCBIGENE:402	hgnc:693	ARL2	GuideToPharmacology	2024.1	blocker	2.625383561784724	IUPHAR.LIGAND:2358	ncit:C66687	ZATEBRADINE	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.059330702	IUPHAR.LIGAND:8015	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:5926	iuphar.ligand:5926	ALSTERPAULLONE 2-CYANOETHYL	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.1779921058837101	IUPHAR.LIGAND:5212	rxcui:42351	LITHIUM CARBONATE	TRUE	FALSE	FALSE
NCBIGENE:2029	hgnc:3360	ENSA	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1171	iuphar.ligand:1171	[SER8]GNRH	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:1599	iuphar.ligand:1599	5-METHYL-5-(5-METHYLTHIOPHEN-3-YL)-4-OXO-4,5-DIHYDROFURAN-2-CARBOXYLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:403	hgnc:694	ARL3	GuideToPharmacology	2024.1	blocker	1.875273972703375	IUPHAR.LIGAND:2358	ncit:C66687	ZATEBRADINE	FALSE	FALSE	FALSE
NCBIGENE:2031	ncbigene:2031	ENUR1	GuideToPharmacology	2024.1	activator	26.25383561784724	IUPHAR.LIGAND:9164	iuphar.ligand:9164	GUANYLYL CYCLASE-ACTIVATING PROTEIN 1	FALSE	FALSE	FALSE
NCBIGENE:401	hgnc:691	PHOX2A	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
NCBIGENE:2032	ncbigene:2032	ENUR2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:11120	iuphar.ligand:11120	ACY-738	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:1278	iuphar.ligand:1278	JNJ 7777120	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:1272	iuphar.ligand:1272	CCL16	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.026519026	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2968	iuphar.ligand:2968	COMPOUND 4I [PMID: 2296036]	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4352	iuphar.ligand:4352	7&BETA;-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4351	iuphar.ligand:4351	7&ALPHA;-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:11220	iuphar.ligand:11220	SUPRASTAT	FALSE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:12363	iuphar.ligand:12363	NCRW0105-E06	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	0.280789686	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.1037701012563132	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:717	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.150021918	IUPHAR.LIGAND:734	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:110	hgnc:13300	GPR61	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:12948	iuphar.ligand:12948	COMPOUND 1 [PMID: 37741852]	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5848	iuphar.ligand:5848	3-HYDROXY CAPRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:9994	iuphar.ligand:9994	BMS-509744	FALSE	FALSE	FALSE
NCBIGENE:150	hgnc:281	ADRA2A	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:7039	iuphar.ligand:7039	AR234960	FALSE	FALSE	FALSE
NCBIGENE:148	hgnc:277	ADRA1A	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:3700	iuphar.ligand:3700	R-SPONDIN-4	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:4971	rxcui:274403	MECASERMIN	TRUE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:5683	iuphar.ligand:5683	GSK-1838705A	FALSE	FALSE	FALSE
NCBIGENE:2448	hgnc:6145	ITGA9	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:12044	iuphar.ligand:12044	SVEP1	FALSE	FALSE	FALSE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9382	iuphar.ligand:9382	NVP-TAE 226	FALSE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8081	iuphar.ligand:8081	IRAK4 INHIBITOR RAC-45 [PMID: 18501603]	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1962	iuphar.ligand:1962	AFP-07	FALSE	FALSE	FALSE
NCBIGENE:1698	hgnc:6024	IL7R	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:9604	iuphar.ligand:9604	OSE-127	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.5147810905460244	IUPHAR.LIGAND:6412	iuphar.ligand:6412	VANILLIN	FALSE	FALSE	FALSE
NCBIGENE:676	hgnc:1105	BRDT	GuideToPharmacology	2024.1	agonist	0.3409589041278864	IUPHAR.LIGAND:10934	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:12468	iuphar.ligand:12468	GROSHEIMIN	FALSE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	0.8751278539282418	IUPHAR.LIGAND:12424	iuphar.ligand:12424	L-TRP-TRP-TRP	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:5716	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:9246	iuphar.ligand:9246	UPADACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2377	hgnc:3889	FRA2E	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8483	iuphar.ligand:8483	COMPOUND 4D [PMID: 25489658]	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	NULL	0.2263261691193728	IUPHAR.LIGAND:12310	iuphar.ligand:12310	SJ988497	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0296486	IUPHAR.LIGAND:7643	iuphar.ligand:7643	AEE788	FALSE	FALSE	TRUE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:1628	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0148243	IUPHAR.LIGAND:5671	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.1037701012563132	IUPHAR.LIGAND:10460	iuphar.ligand:10460	PAMUFETINIB	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.001820528	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10678	iuphar.ligand:10678	SOTORASIB	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12279	iuphar.ligand:12279	BI-0474	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:8250	iuphar.ligand:8250	SOTULETINIB	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12393	iuphar.ligand:12393	FULZERASIB	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	1.250182648468916	IUPHAR.LIGAND:12646	iuphar.ligand:12646	ASP-0819	FALSE	FALSE	FALSE
NCBIGENE:387	hgnc:667	RHOA	GuideToPharmacology	2024.1	blocker	0.375054795	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:438	hgnc:750	ASMT	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:2404	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:443	hgnc:756	ASPA	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	0.2386712328895204	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:385	hgnc:18865	KCNT1	GuideToPharmacology	2024.1	activator	0.8078103267029924	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:1242	hgnc:20692	TPH2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10647	ncit:C171780	RODATRISTAT	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:6044	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1816	hgnc:3026	DRD5	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NCBIGENE:2682	hgnc:11114	KDM5C	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8979	iuphar.ligand:8979	GSK-J4	FALSE	FALSE	FALSE
NCBIGENE:2853	hgnc:4486	GPR31	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10485	iuphar.ligand:10485	CCT365623	FALSE	FALSE	FALSE
NCBIGENE:2704	hgnc:29489	KMT5A	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:5952	iuphar.ligand:5952	CDK4 INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:2094	ncbigene:2094	ERVT4	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8178	iuphar.ligand:8178	COMPOUND 16 [PMID: 18945615]	FALSE	FALSE	FALSE
NCBIGENE:1816	hgnc:3026	DRD5	GuideToPharmacology	2024.1	NULL	2.625383561784724	IUPHAR.LIGAND:5023	iuphar.ligand:5023	MACROPHAGE STIMULATING PROTEIN 1	FALSE	FALSE	FALSE
NCBIGENE:2684	ncbigene:2684	GGTL1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10141	iuphar.ligand:10141	KDM5 INHIBITOR N71	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1296	iuphar.ligand:1296	[125I]MCH (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:3633	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1323	iuphar.ligand:1323	MT-II	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:1342	iuphar.ligand:1342	AC-C[CYS-GLU-HIS-D-PHE-ARG-TRP-D-CYS]-PRO-PRO-LYS-ASP-NH2	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1526385791735305	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.055504938	IUPHAR.LIGAND:7933	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:10151	iuphar.ligand:10151	NEOLYMPHOSTIN A	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.2059124362184097	IUPHAR.LIGAND:7904	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.077217164	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:3181	hgnc:5033	HNRNPA2B1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12894	iuphar.ligand:12894	STC-15	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	0.6403374540938354	IUPHAR.LIGAND:3953	iuphar.ligand:3953	A-841720	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6354	iuphar.ligand:6354	A-794278	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6435	iuphar.ligand:6435	GSK2210875	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6394	iuphar.ligand:6394	LSN2463359	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1368	iuphar.ligand:1368	L-CCG-I	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1394	iuphar.ligand:1394	LY379268	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6416	iuphar.ligand:6416	CPPZ	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6410	iuphar.ligand:6410	VU0404251	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	modulator	2.500365296937833	IUPHAR.LIGAND:10196	iuphar.ligand:10196	VU6012962	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:1398	iuphar.ligand:1398	&ALPHA;-METHYLSERINE-O-PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:11281	drugbank:DB15418	AZD-9977	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:8058	iuphar.ligand:8058	JNK-IN-8	FALSE	FALSE	FALSE
NCBIGENE:1502	hgnc:6875	MAPK13	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:11096	iuphar.ligand:11096	MAPK13-IN-1	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:9203	ncit:C166567	ACUMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:12334	iuphar.ligand:12334	COMPOUND 25C [PMID: 36649216]	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9377	iuphar.ligand:9377	JNK INHIBITOR 9L	FALSE	FALSE	FALSE
NCBIGENE:2093	ncbigene:2093	ERVT3	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11980	iuphar.ligand:11980	AX15836	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:9371	iuphar.ligand:9371	PF-670462	FALSE	FALSE	FALSE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8077	iuphar.ligand:8077	5Z-7-OXOZEAENOL	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:6482	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
NCBIGENE:2085	ncbigene:2085	ERV1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12336	iuphar.ligand:12336	COMPOUND 5I [PMID: 36542759]	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1464	iuphar.ligand:1464	MOTILIN-(2-22) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:988	hgnc:1743	CDC5L	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:10405	iuphar.ligand:10405	BAY-8002	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:6641	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:300	iuphar.ligand:300	METHYLFURMETHIDE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.042073455	IUPHAR.LIGAND:325	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:330	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1345	iuphar.ligand:1345	5-HEAT	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.096167896	IUPHAR.LIGAND:10651	rxcui:2559612	SAMIDORPHAN	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.03394161	IUPHAR.LIGAND:1638	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:1624	ncit:C65596	ETONITAZENE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.012543639	IUPHAR.LIGAND:1627	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
NCBIGENE:2125	hgnc:3503	EVPL	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
NCBIGENE:1749	hgnc:2918	DLX5	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:5020	iuphar.ligand:5020	M372049	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:8071	iuphar.ligand:8071	GNF-5837	FALSE	FALSE	FALSE
NCBIGENE:1251	hgnc:7872	NOS1	GuideToPharmacology	2024.1	inhibitor	0.2112984757975633	IUPHAR.LIGAND:11467	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
NCBIGENE:470	ncbigene:470	ATHS	GuideToPharmacology	2024.1	inhibitor	0.1630673019742065	IUPHAR.LIGAND:2585	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.2885036881082116	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:11656	drugbank:DB08040	KELATORPHAN	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278864	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	blocker	0.5303805175322676	IUPHAR.LIGAND:3986	iuphar.ligand:3986	A-867744	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	modulator	0.9053046764774912	IUPHAR.LIGAND:3991	iuphar.ligand:3991	PNU-120596	FALSE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	0.1268301237577161	IUPHAR.LIGAND:2585	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:10349	iuphar.ligand:10349	L760735	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2109	iuphar.ligand:2109	ZD6021	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2112	iuphar.ligand:2112	[&BETA;ALA8]NEUROKININ A-(4-10)	FALSE	FALSE	FALSE
NCBIGENE:2861	hgnc:4494	GPR37	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:11361	iuphar.ligand:11361	BRONTICTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6174	iuphar.ligand:6174	5-(6-CHLORO-2-HEXYL-1H-INDOL-1-YL)-5-OXO-VALERIC ACID	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:12603	ncit:C175783	FIRAZOREXTON	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:12605	iuphar.ligand:12605	T-516	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:8937	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:9466	iuphar.ligand:9466	[3H]CP-1	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	agonist	0.1930429089547592	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:4236	iuphar.ligand:4236	L-&BETA;&GAMMA;-MEATP	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:12567	iuphar.ligand:12567	BAY-1797	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3337	iuphar.ligand:3337	MRS2690	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	0.09963505	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	0.09963505	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:9468	iuphar.ligand:9468	PSB-416	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:9460	iuphar.ligand:9460	AC264613	FALSE	FALSE	FALSE
NCBIGENE:2878	hgnc:4555	GPX3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8684	iuphar.ligand:8684	COMPOUND 14B [PMID: 25742366]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9376	iuphar.ligand:9376	IC-87114	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:10162	iuphar.ligand:10162	RV1729	FALSE	FALSE	FALSE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9330	iuphar.ligand:9330	CDP840	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	modulator	1.640864726115453	IUPHAR.LIGAND:10451	iuphar.ligand:10451	BPN14770	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8128	iuphar.ligand:8128	COMPOUND 1A [PMID: 24900749]	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.2678962818147678	IUPHAR.LIGAND:9790	iuphar.ligand:9790	PIM447	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1866	iuphar.ligand:1866	PROKINETICIN-1	FALSE	FALSE	FALSE
NCBIGENE:2392	ncbigene:2392	FRA4E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8760	iuphar.ligand:8760	DUP-714	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:11747	iuphar.ligand:11747	BPR1R024	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:5656	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.070010228	IUPHAR.LIGAND:7882	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.087512785	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:6019	iuphar.ligand:6019	PDGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:12885	iuphar.ligand:12885	LERZEPARIB	FALSE	FALSE	FALSE
NCBIGENE:1257	ncbigene:1257	CNC2	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8955	iuphar.ligand:8955	MS023	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.2561349816375342	IUPHAR.LIGAND:11220	iuphar.ligand:11220	SUPRASTAT	FALSE	FALSE	FALSE
NCBIGENE:2401	hgnc:3912	FRA6A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9221	iuphar.ligand:9221	AZAPRO-3	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:5937	iuphar.ligand:5937	BISINDOLYLMALEIMIDE IV	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
NCBIGENE:1492	hgnc:9414	PRKG1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:7887	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2173	hgnc:3562	FABP7	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8048	iuphar.ligand:8048	CRT 0066101	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:5701	iuphar.ligand:5701	PI-103	FALSE	FALSE	FALSE
NCBIGENE:2181	hgnc:3570	ACSL3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5923	iuphar.ligand:5923	ALOISINE	FALSE	FALSE	FALSE
NCBIGENE:1521	hgnc:2546	CTSW	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8184	iuphar.ligand:8184	COMPOUND 32 [PMID: 20471253]	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:13005	iuphar.ligand:13005	COMPOUND 182 [PMID: 37500611]	FALSE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2648	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.42006137	IUPHAR.LIGAND:11220	iuphar.ligand:11220	SUPRASTAT	FALSE	FALSE	FALSE
NCBIGENE:2413	hgnc:3924	FRA7F	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4812	rxcui:325646	ALISKIREN	TRUE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:2811	iuphar.ligand:2811	AGN194204	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.063645662	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:612	hgnc:10479	RXRG	GuideToPharmacology	2024.1	agonist	0.9092237443410301	IUPHAR.LIGAND:2645	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:2815	iuphar.ligand:2815	PA451	FALSE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:8905	iuphar.ligand:8905	PA452	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9558	iuphar.ligand:9558	BELUMOSUDIL	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.1223955040459079	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:596	hgnc:990	BCL2	GuideToPharmacology	2024.1	agonist	0.1280674908187671	IUPHAR.LIGAND:8900	iuphar.ligand:8900	SR9011	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:11913	iuphar.ligand:11913	NANOLUC-INSL3	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:8336	iuphar.ligand:8336	MINIMISED RELAXIN-3 ANALOGUE 2	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:11460	iuphar.ligand:11460	COMPOUND 4 [PMID: 30824200]	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:1223	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11461	iuphar.ligand:11461	R3 B1-22R	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:11917	iuphar.ligand:11917	COMPOUND 7A [PMID: 33730669]	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1997	iuphar.ligand:1997	RELAXIN-3 (B CHAIN)	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:12504	iuphar.ligand:12504	HINSL5: A8-21 (T15K)	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:6679	iuphar.ligand:6679	NE-100	FALSE	FALSE	FALSE
NCBIGENE:2708	hgnc:10886	SIRT2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8099	iuphar.ligand:8099	AGK2	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:1250	iuphar.ligand:1250	IMETIT	FALSE	FALSE	FALSE
NCBIGENE:1416	hgnc:2399	CRYBB2P1	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:8787	iuphar.ligand:8787	COMPOUND 12E [PMID: 18605714]	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:2025	iuphar.ligand:2025	CYCLO(7-12) DES-AA1,2,5-[GLU7,D-TRP8,IAMP9,M-I-TYR11,HHLYS12]SRIF	FALSE	FALSE	FALSE
NCBIGENE:2210	hgnc:3614	FCGR1BP	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.2573905452730122	IUPHAR.LIGAND:1236	iuphar.ligand:1236	(R)-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2033	iuphar.ligand:2033	BIM 23027	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:2027	iuphar.ligand:2027	BIM 23627	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2022	iuphar.ligand:2022	[125I]CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2069	iuphar.ligand:2069	BIM 23295	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.059397818	IUPHAR.LIGAND:1204	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	0.3723948314588262	IUPHAR.LIGAND:2066	iuphar.ligand:2066	PRL-2915	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:2148	iuphar.ligand:2148	[3H]TYRAMINE	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:2146	ncit:C170114	LEVAMFETAMINE	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1246	iuphar.ligand:1246	VUF 8328	FALSE	FALSE	FALSE
NCBIGENE:1722	hgnc:7217	MPL	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:10657	iuphar.ligand:10657	HETROMBOPAG	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.061791905	IUPHAR.LIGAND:2634	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:11293	ncit:C169948	ENERISANT	FALSE	FALSE	FALSE
NCBIGENE:3189	hgnc:5043	HNRNPH3	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11683	ncit:C184931	SUCUNAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:8120	iuphar.ligand:8120	COMPOUND 13D [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.5707355569097228	IUPHAR.LIGAND:10285	iuphar.ligand:10285	CLEMIZOLE	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12895	iuphar.ligand:12895	GDC-6599	FALSE	FALSE	FALSE
NCBIGENE:2763	ncbigene:2763	GMFA	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:11264	rxcui:1311506	GLYCYRRHETINIC ACID	TRUE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.070197421	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	1.544343271638073	IUPHAR.LIGAND:4103	iuphar.ligand:4103	20-HETE	FALSE	FALSE	FALSE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	blocker	0.3860858179095184	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:493	hgnc:817	ATP2B4	GuideToPharmacology	2024.1	activator	5.250767124	IUPHAR.LIGAND:4290	iuphar.ligand:4290	PREGNENOLONE SULPHATE	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	activator	6.563458904461812	IUPHAR.LIGAND:12537	iuphar.ligand:12537	COMPOUND 39 [PMID: 36402081]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2972	iuphar.ligand:2972	COMPOUND 2T [PMID: 2296036]	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.088248187	IUPHAR.LIGAND:2486	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.1861974157294131	IUPHAR.LIGAND:12706	drugbank:DB15498	BOS172722	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1209854175937661	IUPHAR.LIGAND:5716	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:2918	iuphar.ligand:2918	KYNURENIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1031	hgnc:1789	CDKN2C	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11389	ncit:C166614	DOTINURAD	FALSE	FALSE	FALSE
NCBIGENE:2990	hgnc:4696	GUSB	GuideToPharmacology	2024.1	inhibitor	0.9723642821424907	IUPHAR.LIGAND:8804	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:2780	rxcui:291204	TACALCITOL	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2278	iuphar.ligand:2278	[ALA11,22,28]VIP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2169	ncit:C87380	ARGIPRESTOCIN	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2266	iuphar.ligand:2266	N-STEARYL-[NLE17] NEUROTENSIN-(6-11)/VIP-(7-28)	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:9565	iuphar.ligand:9565	PF-06840003	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:2202	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.014617949	IUPHAR.LIGAND:2175	iuphar.ligand:2175	[3H]AVP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:2173	iuphar.ligand:2173	OPC-51803	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:2184	iuphar.ligand:2184	D[D-PAL2]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2169	ncit:C87380	ARGIPRESTOCIN	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2175	iuphar.ligand:2175	[3H]AVP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9173	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
NCBIGENE:2285	hgnc:3717	FKBP1AP4	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:5923	iuphar.ligand:5923	ALOISINE	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.034184682	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	NULL	CARBOPLATIN/PACLITAXEL REGIMEN	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.00416199	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.012794267	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:9750	iuphar.ligand:9750	NECROSTATIN-1	FALSE	FALSE	FALSE
CD44	hgnc:1681	CD44	CIViC	10-Apr-24	NULL	NULL	RG7356	NULL	NULL	NULL	NULL	NULL
SMO	hgnc:11119	SMO	CIViC	10-Apr-24	NULL	15.31473744374422	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
NCBIGENE:156	hgnc:289	GRK2	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:4058	iuphar.ligand:4058	BOVINE ADRENAL MEDULLA PEPTIDE 8-22	FALSE	FALSE	FALSE
IKZF1	hgnc:13176	IKZF1	CIViC	10-Apr-24	NULL	0.093763699	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
SMARCB1	hgnc:11103	SMARCB1	CIViC	10-Apr-24	NULL	7.501095890813499	TAZEMETOSTAT	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
NCBIGENE:165	hgnc:303	AEBP1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:2917	iuphar.ligand:2917	JTE-013	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	CIViC	10-Apr-24	NULL	0.023813003	ALPELISIB	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	NULL	FGF/VEGF RECEPTOR TYROSINE KINASE INHIBITOR, PD173074	NULL	NULL	NULL	NULL	NULL
CD274	hgnc:17635	CD274	CIViC	10-Apr-24	NULL	NULL	RADIATION THERAPY	NULL	NULL	NULL	NULL	NULL
FANCC	hgnc:3584	FANCC	CIViC	10-Apr-24	NULL	1.050153425	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
NCBIGENE:745	hgnc:1181	MYRF	GuideToPharmacology	2024.1	activator	5.834185692854944	IUPHAR.LIGAND:4222	iuphar.ligand:4222	IP3	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	2.763561643983921	CTLA-4 INHIBITOR	ncit:C191738	CTLA-4-TARGETING AGENT	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.4234489615781814	BELVARAFENIB	ncit:C121646	BELVARAFENIB	FALSE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.069824031	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	NULL	RADIATION THERAPY	NULL	NULL	NULL	NULL	NULL
PTPRD	hgnc:9668	PTPRD	CIViC	10-Apr-24	NULL	NULL	JSI-124	NULL	NULL	NULL	NULL	NULL
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.043756393	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	0.080103236	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:646	hgnc:1081	BNC1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:3167	iuphar.ligand:3167	NE21650	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	CIViC	10-Apr-24	NULL	NULL	R-CHOP REGIMEN	NULL	NULL	NULL	NULL	NULL
FGFR4	hgnc:3691	FGFR4	CIViC	10-Apr-24	NULL	NULL	FGF/VEGF RECEPTOR TYROSINE KINASE INHIBITOR, PD173074	NULL	NULL	NULL	NULL	NULL
BIRC5	hgnc:593	BIRC5	CIViC	10-Apr-24	NULL	NULL	TAXANE COMPOUND	NULL	NULL	NULL	NULL	NULL
NCBIGENE:666	hgnc:1087	BOK	GuideToPharmacology	2024.1	agonist	1.500219178162699	IUPHAR.LIGAND:12432	iuphar.ligand:12432	CUCURBITACIN B	FALSE	FALSE	FALSE
MERTK	hgnc:7027	MERTK	CIViC	10-Apr-24	NULL	NULL	UNC1062	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	NULL	RADIATION THERAPY	NULL	NULL	NULL	NULL	NULL
TERT	hgnc:11730	TERT	CIViC	10-Apr-24	NULL	NULL	UO126	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2885	hgnc:4566	GRB2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10663	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	CIViC	10-Apr-24	NULL	0.033919684	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
EPOR	hgnc:3416	EPOR	CIViC	10-Apr-24	NULL	NULL	INHIBITOR	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:9619	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
FOXC2	hgnc:3801	FOXC2	CIViC	10-Apr-24	NULL	1.280674908	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.029244039	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	CCC-003	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	2.212697851403848	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1369765336583334	Belizatinib	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.072092912	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.3043922970185188	4SC-205	ncit:C90557	EG5 KINESIN-RELATED MOTOR PROTEIN INHIBITOR 4SC-205	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	PKF118-310	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	JW74	NULL	NULL	NULL	NULL	NULL
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.2447910080918158	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1603	iuphar.ligand:1603	(-)-BREMAZOCINE	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	NULL	Radiotherapy	NULL	NULL	NULL	NULL	NULL
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.2055094764606438	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.2075402025126264	IUPHAR.LIGAND:12782	ncit:C169761	ACRIZANIB	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	1.591141552596803	UNC1999	iuphar.ligand:8237	UNC1999	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	NULL	YU238259	NULL	NULL	NULL	NULL	NULL
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
ATR	hgnc:882	ATR	JAX-CKB	10-Apr-24	NULL	0.048282916	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.045668773	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.2877132670449014	AZD7648	iuphar.ligand:10601	AZD7648	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.5223276196220918	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.002207874	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.8751278539282416	PRT062607	iuphar.ligand:8070	P505-15	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.068637479	Ado-trastuzumab emtansine	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.069089041	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	1.050153425	Avapritinib	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.3088686543276147	Pegilodecakin	ncit:C113295	PEGILODECAKIN	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:5982	iuphar.ligand:5982	GTP-14564	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Pimivalimab	ncit:C157485	PIMIVALIMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	NULL	CTX-8371	NULL	NULL	NULL	NULL	NULL
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.2827336143460473	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.037064239	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11839	iuphar.ligand:11839	ASP2453	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified CTLA4 antibody	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	1.141471113819445	MTI-31	chembl:CHEMBL4594431	MTI-31	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.2282942227638891	Belizatinib	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.4565884455277783	Luminespib	ncit:C71467	LUMINESPIB	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.789589041	Birabresib	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	FIIN-1	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	3HP-2827	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	PRN1109	NULL	NULL	NULL	NULL	NULL
NCBIGENE:516	hgnc:841	ATP5MC1	GuideToPharmacology	2024.1	activator	1.141471113819445	IUPHAR.LIGAND:2326	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.2616661357260523	Brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.4579157375205915	Derazantinib	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	NULL	FIIN-2	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.7369497717290455	E7090	ncit:C118672	TASURGRATINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.179119736	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.014545061	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.017546423	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	TCS 359	iuphar.ligand:5970	FLT-3 INHIBITOR	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.4947116523181093	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	Zotiraciclib	ncit:C171725	ZOTIRACICLIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	LT-171-861	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.028360625	Linifanib	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:515	hgnc:840	ATP5PB	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.4278402841426959	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1296485709523321	Omacetaxine mepesuccinate	rxcui:27100	OMACETAXINE MEPESUCCINATE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1296485709523321	GTP-14564	iuphar.ligand:5982	GTP-14564	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	PI-273	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	NS1	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.172722603	LXH 254	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	NULL	Radiotherapy	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.053145416	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.106290832	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.001770767	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.011670965	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.546954909	LY3410738	iuphar.ligand:12340	LY3410738	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.038382801	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.081533651	Tenalisib	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.03357268	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.1037701012563132	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2634164108814105	Momelotinib	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	NULL	Radiotherapy	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.03849536	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.8468979231563628	Chelidonine	chembl:CHEMBL496867	CHELIDONINE	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	NS1	NULL	NULL	NULL	NULL	NULL
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified CTLA4 antibody	NULL	NULL	NULL	NULL	NULL
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	Radiotherapy	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.032412143	Lucitanib	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	YM-024	NULL	NULL	NULL	NULL	NULL
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	1.468746048550895	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	AZD0156	iuphar.ligand:9942	AZD0156	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.025672984	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	TY-1091	ncit:C199307	RET INHIBITOR TY-1091	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.2592971419046642	Volasertib	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-1 antibody	NULL	NULL	NULL	NULL	NULL
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	NULL	unspecified PD-L1 antibody	NULL	NULL	NULL	NULL	NULL
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.2586584789935689	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.1065064325267637	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	NULL	Radiotherapy	NULL	NULL	NULL	NULL	NULL
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.1136529680426288	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.009272878	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.1448487482363986	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	Radiotherapy	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	unspecified IGF-1R antibody	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	AZ32	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	Ad.p53-DC vaccine	NULL	NULL	NULL	NULL	NULL
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2318	iuphar.ligand:2318	NS8593	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.021074723	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.016558711	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.173866461	BI 907828	ncit:C156709	BRIGIMADLIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	MVAp53	NULL	NULL	NULL	NULL	NULL
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	modulator	0.1553481397505754	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
RPL36A	hgnc:10359	RPL36A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:2317	iuphar.ligand:2317	NS309	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	DTC	9/2/20	NULL	0.1058622403945453	BIPERIDEN	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
NCBIGENE:441	hgnc:6269	KCNJ8	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:2414	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK711701A	chembl:CHEMBL268885	GSK-711701A	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.5097832158805291	GNF-PF-2391	chembl:CHEMBL577415	CHEMBL:CHEMBL577415	FALSE	FALSE	FALSE
F5	hgnc:3542	F5	FDA	10-Apr-24	NULL	0.036306082	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.1143957978991165	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
CBL	hgnc:1541	CBL	NCI	14-Sep-17	NULL	0.1750255707856483	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.2983390411119005	levomilnacipran	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE	hgnc:1189	AHSA1	TTD	2020.06.01	NULL	1.458546423213736	ARRY-797	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
NCBIGENE:538	hgnc:869	ATP7A	GuideToPharmacology	2024.1	blocker	5.834185692854944	IUPHAR.LIGAND:7737	iuphar.ligand:7737	HELATX1	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.081365193	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.026319635	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.7192831676122533	GZ-389988	drugbank:DB16056	GZ-389988	FALSE	FALSE	FALSE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	1.200175343	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SJ000027778	chembl:CHEMBL592588	CHEMBL:CHEMBL592588	FALSE	FALSE	FALSE
NCBIGENE:547	hgnc:888	KIF1A	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11478	iuphar.ligand:11478	RY785	FALSE	FALSE	FALSE
PLCG1	hgnc:9065	PLCG1	DTC	9/2/20	NULL	2.917092846427472	PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER	iuphar.ligand:5092	&ALPHA;&BETA;-METHYLENEADP	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1933	iuphar.ligand:1933	ONO-AE1-329	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.3443125982668492	NORETHINDRONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
NCBIGENE:562	hgnc:6297	KCNQ3	GuideToPharmacology	2024.1	activator	2.678962818147678	IUPHAR.LIGAND:2601	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.010620484	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.018359326	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	4.039051633514961	IUPHAR.LIGAND:7667	iuphar.ligand:7667	ICA-27243	FALSE	FALSE	FALSE
PCBD1	hgnc:8646	PCBD1	NCI	14-Sep-17	NULL	2.019525816757481	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	PharmGKB	4/5/24	NULL	0.1752592497853621	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:5655	iuphar.ligand:5655	A-674563	FALSE	FALSE	FALSE
NCBIGENE:65	ncbigene:65	ACTBP5	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:815	iuphar.ligand:815	VMIP-I	FALSE	FALSE	FALSE
BRDT	hgnc:1105	BRDT	ChEMBL	33	inhibitor	0.5357925636295356	APABETALONE	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	GW770249X	iuphar.ligand:10133	COMPOUND 27 [PMID: 24900635]	FALSE	FALSE	FALSE
KCND2	hgnc:6238	KCND2	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.175610941	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:336	drugbank:DB02152	K-252A	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.2386712328895204	HOMOHARRINGTONINE	rxcui:27100	OMACETAXINE MEPESUCCINATE	TRUE	FALSE	FALSE
PVALB	hgnc:9704	PVALB	NCI	14-Sep-17	NULL	3.750547945406749	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
ACTIVATED CDC42 KINASE 1	hgnc:19297	TNK2	TTD	2020.06.01	NULL	0.042898424	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6718	iuphar.ligand:6718	COMPOUND 9 [PMID: 22533316]	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.1591141552596802	RWJ-67657	chembl:CHEMBL190333	RWJ-67657	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:8862	iuphar.ligand:8862	BLU-9931	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	CancerCommons	25-Jul-13	inhibitor	0.272767123	PLX3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.2375912725597036	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.3621218705909966	EPALRESTAT	ncit:C72762	EPALRESTAT	FALSE	FALSE	FALSE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	0.1615620653405984	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	0.1190650141398968	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CAMKK2	hgnc:1470	CAMKK2	PharmGKB	4/5/24	NULL	0.84012274	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.3777530304726222	Radotinib	ncit:C98110	RADOTINIB	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:1376	iuphar.ligand:1376	AIDA	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.010199625	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.017295017	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:292	iuphar.ligand:292	NNC 11-1585	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.1154014752432846	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
SMARCA2	hgnc:11098	SMARCA2	DTC	9/2/20	NULL	4.375639269641208	GNF-PF-3736	chembl:CHEMBL583824	CHEMBL:CHEMBL583824	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	CC-90006	chembl:CHEMBL4594467	CC-90006	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	5.834185692854944	STX-107	drugbank:DB16943	STX-107	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2853677784548614	IMG-7289	ncit:C131827	BOMEDEMSTAT	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9392	iuphar.ligand:9392	HG-10-102-01	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4605936073306534	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.4023576339899962	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	0.3860858179095183	Flavanone	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 1 ALPHA	hgnc:4910	HIF1A	TTD	2020.06.01	NULL	0.7242437411819931	EZN-2968	ncit:C68930	ANTI-HIF-1ALPHA LNA ANTISENSE OLIGONUCLEOTIDE EZN-2968	FALSE	FALSE	TRUE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:3498	iuphar.ligand:3498	CRA1000	FALSE	FALSE	FALSE
NCBIGENE:2055	hgnc:2079	CLN8	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8151	iuphar.ligand:8151	COMPOUND 14 [PMID: 19831390]	FALSE	FALSE	FALSE
NCBIGENE:1392	hgnc:2355	CRH	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:11402	ncit:C986	ACIVICIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	GNF-PF-2954	chembl:CHEMBL582722	CHEMBL:CHEMBL582722	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.7721716358190367	FLAVONE-8-ACETIC ACID	ncit:C1101	MITOFLAXONE	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:5613	iuphar.ligand:5613	ST-1535	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	1.810609352954982	P-IODOCLONIDINE HCL	chembl:CHEMBL1255758	CHEMBL:CHEMBL1255758	FALSE	FALSE	FALSE
NCBIGENE:1631	hgnc:7174	MMP7	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8629	iuphar.ligand:8629	SL422	FALSE	FALSE	FALSE
NCBIGENE:1838	hgnc:3058	DTNB	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.050246575	IUPHAR.LIGAND:7319	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.030038714	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
KCNA3	hgnc:6221	KCNA3	ChEMBL	33	blocker	0.1562728310586145	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11984	ncit:C169757	ACEBILUSTAT	FALSE	FALSE	FALSE
ACVRL1	hgnc:175	ACVRL1	ChEMBL	33	inhibitor	0.364636606	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	ChEMBL	33	blocker	0.093763699	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.3125456621172291	ZONAMPANEL	ncit:C152963	ZONAMPANEL	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	1.810609352954982	PHENACYLAMINE HYDROCHLORIDE	chembl:CHEMBL1213139	PHENACYLAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11205	iuphar.ligand:11205	LYS006	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.023110771	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PRIM1	hgnc:9369	PRIM1	NCI	14-Sep-17	NULL	7.501095891	3&APOS;-DEOXYADENOSINE	ncit:C1057	CORDYCEPIN	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:2755	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
RHOA	hgnc:667	RHOA	DTC	9/2/20	NULL	15.00219178	CLAUSINE E	chembl:CHEMBL235934	CLAUSINE E	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:2916	iuphar.ligand:2916	DIOCTANOYLGLYCEROL PYROPHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:Q92806	hgnc:6270	KCNJ9	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.1219218372345847	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	binder	2.100306849	IGN-101	chembl:CHEMBL2109259	IGN-101	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:2916	iuphar.ligand:2916	DIOCTANOYLGLYCEROL PYROPHOSPHATE	FALSE	FALSE	FALSE
RPL17	hgnc:10307	RPL17	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002188184	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.050707553	amphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	0.1268301237577161	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	0.2447910080918158	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.068637479	felodipine	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	0.577007376	IUPHAR.LIGAND:2906	iuphar.ligand:2906	LPA	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	TALC	12-May-16	vaccine	0.546954909	RAS PEPTIDE CANCER VACCINE	ncit:C2438	RAS PEPTIDE CANCER VACCINE	FALSE	FALSE	TRUE
RPS20	hgnc:10405	RPS20	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	SJ000260212	chembl:CHEMBL607138	CHEMBL:CHEMBL607138	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.034118045	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR-I	hgnc:5464	IGF1	TTD	2020.06.01	NULL	13.12691780892362	MEDI-573	ncit:C82683	DUSIGITUMAB	FALSE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	3.500511415712966	Tiazofurin	ncit:C1254	TIAZOFURIN	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:4031	iuphar.ligand:4031	DODECYLPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2034	hgnc:3374	EPAS1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8171	iuphar.ligand:8171	COMPOUND 5B [PMID: 24900464]	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.034727296	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11861	iuphar.ligand:11861	PRU-10	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1875273972703375	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
NCBIGENE:163	hgnc:563	AP2B1	GuideToPharmacology	2024.1	agonist	7.501095890813499	IUPHAR.LIGAND:2906	iuphar.ligand:2906	LPA	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.030211548	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
RPL39	hgnc:10350	RPL39	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00399693	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:2671	hgnc:4236	GFER	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:7025	iuphar.ligand:7025	DAMINOZIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	NSC-367089	chembl:CHEMBL1543865	CHEMBL:CHEMBL1543865	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.008479921	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.081533651	DOMIPHEN BROMIDE	rxcui:49255	DOMIPHEN BROMIDE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.03729238	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	PharmGKB	4/5/24	NULL	0.056826484	topiramate	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	0.1190650141398968	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1282238613814273	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1238388472539964	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	agonist	0.6563458904461813	IUPHAR.LIGAND:2910	drugbank:DB07780	FARNESYL DIPHOSPHATE	FALSE	FALSE	FALSE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	blocker	0.2243917574174979	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.082559232	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.1270346884734544	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
PANCREATIC TRIACYLGLYCEROL LIPASE	hgnc:9155	PNLIP	TTD	2020.06.01	NULL	6.563458904461812	Dalbavancin	rxcui:1539239	DALBAVANCIN	TRUE	FALSE	FALSE
PARP2	hgnc:272	PARP2	MyCancerGenome	20-Jun-17	other/unknown	2.187819634820604	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.07458476	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
HMOX1	hgnc:5013	HMOX1	NCI	14-Sep-17	NULL	2.333674277141978	NEUROTROPHIC FACTOR	ncit:C2259	RECOMBINANT NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.1902451856365742	misoprostol	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2226788432387383	MOMETASONE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.073437302	NIFLUMIC ACID	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:518	iuphar.ligand:518	SKF 105854	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	negative modulator	0.036463661	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.5801952622728673	ALPHA,BETA-METHYLENE-DCTP	chembl:CHEMBL1162298	CHEMBL:CHEMBL1162298	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.075442056	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	2.386712328895204	VA-106483	chembl:CHEMBL518043	FEDOVAPAGON	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.046303061	Amifampridine	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DNQX	chembl:CHEMBL155265	DNQX	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.3977853881492006	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.058602312	HOE-33342	chembl:CHEMBL343002	CHEMBL:CHEMBL343002	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.151537291	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
ELK1	hgnc:3321	ELK1	NCI	14-Sep-17	NULL	6.563458904461812	DHPG	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
P2RX7	hgnc:8537	P2RX7	ChEMBL	33	negative modulator	8.751278539282415	GSK1482160	iuphar.ligand:10504	GSK1482160	FALSE	FALSE	FALSE
NCBIGENE:2795	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:8825	iuphar.ligand:8825	COMPOUND III [PMID: 24080463]	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.021240967	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.050488145	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.026899422	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.053771297	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	agonist	0.2011788169949981	IUPHAR.LIGAND:4090	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.03999061	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.010819631	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	NCI	14-Sep-17	NULL	0.6177373086552295	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1875273972703375	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
GAL	hgnc:4114	GAL	PharmGKB	4/5/24	NULL	0.2524407270946851	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.015299438	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:9892	ncit:C48264	TALABOSTAT	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.007979889	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	0.561579372	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.062509132	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
BHMT2	hgnc:1048	BHMT2	ChEMBL	33	other/unknown	8.751278539282415	BETAINE HYDROCHLORIDE	rxcui:81965	BETAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.029106248	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:11959	iuphar.ligand:11959	EGIS-11150	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.7721716358190367	INIPARIB	ncit:C62526	INIPARIB	FALSE	FALSE	TRUE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	0.596678082	PD-170292	chembl:CHEMBL14153	PD-170292	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.4646696569530486	rifabutin	rxcui:55672	RIFABUTIN	TRUE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.072125922	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
GALR1	hgnc:4132	GALR1	PharmGKB	4/5/24	NULL	3.088686543276147	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	TALC	12-May-16	inhibitor	0.2333674277141978	VOLASERTIB	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.157680694	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:2668	hgnc:4232	GDNF	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:7488	iuphar.ligand:7488	MG149	FALSE	FALSE	FALSE
HSD11B2	hgnc:5209	HSD11B2	NCI	14-Sep-17	NULL	1.875273972703374	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2465148884304905	TIZANIDINE HYDROCHLORIDE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.059085902	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.037693949	TRANSPLATIN	chembl:CHEMBL1386	TRANSPLATIN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.047518255	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
RPL18	hgnc:10310	RPL18	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.092988792	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
DKK1	hgnc:2891	DKK1	CIViC	10-Apr-24	NULL	0.1422972120208523	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.009972967	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.079557078	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.003740928	Diazepam	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:2853	hgnc:4486	GPR31	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8412	iuphar.ligand:8412	SIMTUZUMAB	FALSE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.084758146	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.2500365296937833	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:657	iuphar.ligand:657	NPC 17731	FALSE	FALSE	FALSE
NCBIGENE:2104	hgnc:3474	ESRRG	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10167	iuphar.ligand:10167	TOMIVOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:3005	hgnc:4714	H1-0	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9932	iuphar.ligand:9932	SETANAXIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	1.221108633388244	KIN-3248	drugbank:DB17587	KIN-3248	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1545479653736408	CGM097	ncit:C104280	P53/HDM2 INTERACTION INHIBITOR CGM097	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	agonist	0.2792961235941196	CEVIMELINE HYDROCHLORIDE	rxcui:260036	CEVIMELINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:4231	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.1426838892274307	CT-1578	chembl:CHEMBL2035185	CT-1578	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.020164236	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.017456008	ISOPRENALINE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.8204323630577265	CLODRONATE DISODIUM	rxcui:1546871	CLODRONATE DISODIUM	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.3562257207306275	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1305	iuphar.ligand:1305	ATC0175	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.2900976311364336	SJ000118780	chembl:CHEMBL591836	CHEMBL:CHEMBL591836	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.017787152	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01150727	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DIELDRIN	chembl:CHEMBL1873703	DIELDRIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	PYRILAMINE	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
SLC9A9	hgnc:20653	SLC9A9	PharmGKB	4/5/24	NULL	1.750255707856483	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8227	iuphar.ligand:8227	AMG-1	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1311	iuphar.ligand:1311	S38151	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	GANGALEOIDIN	chembl:CHEMBL1491099	GANGALEOIDIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.030814361	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:12687	iuphar.ligand:12687	PTD10	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.276356164	IUPHAR.LIGAND:8600	iuphar.ligand:8600	ALEXA-488-TELENZEPINE	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	1.250182648468916	CHLOROTHIAZIDE	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
GNL3	hgnc:29931	GNL3	PharmGKB	4/5/24	NULL	0.9723642821424908	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1334	iuphar.ligand:1334	[D-TRP8]&GAMMA;-MSH	FALSE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	ChEMBL	33	blocker	0.1367387271762877	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.150021918	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.1041818873724097	DROLOXIFENE	ncit:C969	DROLOXIFENE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:10348	iuphar.ligand:10348	BAY-593074	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.070010228	IUPHAR.LIGAND:941	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.1693795846312726	IUPHAR.LIGAND:4128	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CRH	hgnc:2355	CRH	NCI	14-Sep-17	NULL	0.7721716358190368	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003874533	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.7395446652914718	RG7440	hemonc:278	IPATASERTIB	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:3927	iuphar.ligand:3927	BRL-54443	FALSE	FALSE	FALSE
NCBIGENE:531	hgnc:1393	CACNA1F	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:4488	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:1917	iuphar.ligand:1917	CICAPROST	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	HS-10365	ncit:C186653	RET INHIBITOR HS-10365	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	RIFAPENTINE	rxcui:35617	RIFAPENTINE	TRUE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.4773424657790409	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TdgClinicalTrial	Jan-14	NULL	0.9334697108567911	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	modulator	0.1346350544504987	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	2-BENZOYL-5-METHOXYBENZOQUINONE	chembl:CHEMBL1434057	2-BENZOYL-5-METHOXYBENZOQUINONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	SB-408124	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.08607815	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	3-HYDROXY-3',4'-DIMETHOXYFLAVONE	chembl:CHEMBL77098	3-HYDROXY-3',4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.021697385	SAHA	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TROPONIN C	hgnc:5318	TNC	TTD	2020.06.01	NULL	0.9376369863516874	Levosimendan	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	0.1426838892274307	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.9723642821424906	ARV-771	iuphar.ligand:10564	ARV-771	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.108711535	3,3',4'-TRIHYDROXYFLAVONE	chembl:CHEMBL122701	CHEMBL:CHEMBL122701	FALSE	FALSE	FALSE
RPL12	hgnc:10302	RPL12	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	0.081407242	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	activator	0.5048814541893701	IUPHAR.LIGAND:3310	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.1235474617310458	IUPHAR.LIGAND:8213	iuphar.ligand:8213	COMPOUND R-16 [PMID: 21967808]	FALSE	FALSE	FALSE
FZD8	hgnc:4046	FZD8	ChEMBL	33	inhibitor	26.25383561784724	IPAFRICEPT	ncit:C102565	IPAFRICEPT	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	0.054243462	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
PSMB1	hgnc:9537	PSMB1	ChEMBL	33	inhibitor	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
KCNC3	hgnc:6235	KCNC3	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	ChEMBL	33	inhibitor	0.3409589041278863	NIROGACESTAT	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.7001022831425934	ANTI-CD3 ANTIBODY	ncit:C2229	VISILIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.03251249	IUPHAR.LIGAND:5679	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.063110182	IUPHAR.LIGAND:340	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6363	iuphar.ligand:6363	FTIDC	FALSE	FALSE	FALSE
RARB	hgnc:9865	RARB	DTC	9/2/20	NULL	1.323722804261206	BMS-204493	iuphar.ligand:2641	BMS493	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.1646008502686348	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	1.458546423213736	CAPADENOSON	ncit:C87279	CAPADENOSON	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9885	iuphar.ligand:9885	CORTISTATIN A	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	GNF-PF-3889	chembl:CHEMBL598270	CHEMBL:CHEMBL598270	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	OncoKB	23-Jul-20	NULL	2.493675356344019	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.101562227	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:67	iuphar.ligand:67	9-OH-RISPERIDONE	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6916	iuphar.ligand:6916	[SAR1,GLY4,GLY8]ANG-II	FALSE	FALSE	FALSE
NCBIGENE:2343	ncbigene:2343	FNTBL1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10967	iuphar.ligand:10967	POSTSTATIN	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:9246	iuphar.ligand:9246	UPADACITINIB	FALSE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	PharmGKB	4/5/24	NULL	1.346350544504987	inclisiran	rxcui:2588243	INCLISIRAN	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.0095957	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.069180068	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	0.2333674277141977	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	DROTAVERINE	rxcui:23684	DROTAVERIN	FALSE	FALSE	FALSE
NCBIGENE:2522	ncbigene:2522	FUSE	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8465	iuphar.ligand:8465	COMPOUND 31 [PMID: 24809814]	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
SCAP	hgnc:30634	SCAP	PharmGKB	4/5/24	NULL	3.281729452230906	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	TAS-103	ncit:C1733	TAS-103	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.1785975212098452	Famitinib	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.07699072	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.093763699	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CYP17A1	hgnc:2593	CYP17A1	ChEMBL	33	inhibitor	30.00438356	ORTERONEL	ncit:C90582	ORTERONEL	FALSE	FALSE	TRUE
MTNR1B	hgnc:7464	MTNR1B	ChEMBL	33	agonist	5.250767123569449	PIROMELATINE	ncit:C170326	PIROMELATINE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.068369364	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	FLUNARIZINE HYDROCHLORIDE	rxcui:82019	FLUNARIZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.046303061	AEE-788	drugbank:DB12558	AEE-788	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.034363659	Chloroquine	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.801643836	DEXAMETHASONE-SPERMINE	chembl:CHEMBL1275761	CHEMBL:CHEMBL1275761	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.1363835616511545	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PTPRZ1	hgnc:9685	PTPRZ1	NCI	14-Sep-17	NULL	2.692701089009974	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.3409589041278863	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:1385	iuphar.ligand:1385	JNJ16259685	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	0.375054795	Trihexyphenidyl	rxcui:10811	TRIHEXYPHENIDYL	TRUE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.088396753	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	1.750255707856483	OK-432	ncit:C745	PICIBANIL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.013560866	chloramphenicol	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.017525925	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.077789143	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	SPLITOMICIN	iuphar.ligand:8101	SPLITOMICIN	FALSE	FALSE	FALSE
PYGL	hgnc:9725	PYGL	PharmGKB	4/5/24	NULL	0.305277158	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NRG3	hgnc:7999	NRG3	PharmGKB	4/5/24	NULL	0.1944728564284981	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:Q05655	hgnc:9399	PRKCD	TdgClinicalTrial	Jan-14	NULL	0.1172046232939609	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.4375639269641208	ATRACURIUM BESYLATE	rxcui:1219	ATRACURIUM BESYLATE	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.272767123	PEXIDARTINIB	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:1401	iuphar.ligand:1401	3-MPPTS	FALSE	FALSE	FALSE
PSMD12	hgnc:9557	PSMD12	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
GRIK2	hgnc:4580	GRIK2	ChEMBL	33	inhibitor	0.051885051	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6317	iuphar.ligand:6317	JNJ-42153605	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	AXOMADOL	ncit:C72138	AXOMADOL	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.012979279	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TdgClinicalTrial	Jan-14	NULL	5.625821918110125	SELEXIPAG	rxcui:1729002	SELEXIPAG	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.2536602475154323	LISDEXAMFETAMINE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.07963752	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
DEBRISOQUINE 4-HYDROXYLASE	hgnc:2625	CYP2D6	TTD	2020.06.01	NULL	0.005208578	Glutethimide	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:11614	iuphar.ligand:11614	LY395756	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:9836	ncit:C152510	TANZISERTIB	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12484	iuphar.ligand:12484	YL5084	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.006219814	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.2573905452730123	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:2065	hgnc:3431	ERBB3	GuideToPharmacology	2024.1	inhibitor	0.2059124362184098	IUPHAR.LIGAND:9989	iuphar.ligand:9989	COMPOUND 11 [PMID: 26431428]	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.6482428547616604	LT-BETA	ncit:C1608	RECOMBINANT LYMPHOTOXIN BETA	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.1442518440541057	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
UNIPROT:P20618	hgnc:9537	PSMB1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE ATR	hgnc:882	ATR	TTD	2020.06.01	NULL	0.9723642821424907	VX-970	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.1105424657593568	IUPHAR.LIGAND:349	rxcui:11201	VINCAMINE	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:6332	rxcui:1545989	ENALAPRILAT ANHYDROUS	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.052350619	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
TNFRSF4	hgnc:11918	TNFRSF4	ChEMBL	33	inhibitor	3.500511415712966	KHK-4083	chembl:CHEMBL4594567	KHK-4083	FALSE	FALSE	FALSE
NCBIGENE:2064	hgnc:3430	ERBB2	GuideToPharmacology	2024.1	NULL	0.3454452054979901	IUPHAR.LIGAND:12006	iuphar.ligand:12006	(R)-STU104	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.210030685	HARMOL	chembl:CHEMBL486817	HARMOL	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.2000292237550266	YUANHUADINE	chembl:CHEMBL1911631	YUANHUADINE	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.2187819634820604	SPIROXATRINE	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.053145416	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
PGD	hgnc:8891	PGD	NCI	14-Sep-17	NULL	0.921187215	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
ERCC2	hgnc:3434	ERCC2	PharmGKB	4/5/24	NULL	0.1909369863116163	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	0.4688184931758437	Isotretinoin	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	0.7955707762984014	NAFARELIN ACETATE	rxcui:203147	NAFARELIN ACETATE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.050879526	2,3,4-TRIHYDROXYBENZOPHENONE	chembl:CHEMBL1527	CHEMBL:CHEMBL1527	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1161674142382621	IUPHAR.LIGAND:1624	ncit:C65596	ETONITAZENE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00449706	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1458546423213736	sacituzumab govitecan-hziy	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.9053046764774912	ANTAZOLINE HYDROCHLORIDE	rxcui:81954	ANTAZOLINE HYDROCHLORIDE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	0.8334550989792778	Bumetanide	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
PLCB1	hgnc:15917	PLCB1	PharmGKB	4/5/24	NULL	1.666910197958555	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.006073762	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.016246185	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:6007	iuphar.ligand:6007	MEK INHIBITOR II	FALSE	FALSE	FALSE
XRCC5	hgnc:12833	XRCC5	PharmGKB	4/5/24	NULL	0.4054646427466756	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	CITRIC ACID	rxcui:21183	CITRIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:11867	drugbank:DB15254	AVUTOMETINIB	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.026519026	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	TESETAXEL	ncit:C37451	TESETAXEL	FALSE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	2.128689374420047	XALIPRODEN	ncit:C152924	XALIPRODEN	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:291	iuphar.ligand:291	NNC 11-1314	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.064033745	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6130	iuphar.ligand:6130	GALANIN(2-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	modulator	3.500511415712966	IUPHAR.LIGAND:10239	iuphar.ligand:10239	VU0422288	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:310	iuphar.ligand:310	HEXAHYDROSILADIFENIDOL	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	inhibitor	0.2678962818147678	IUPHAR.LIGAND:1712	iuphar.ligand:1712	ADP	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.028977744	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1166837138570988	STANOLONE	ncit:C72098	STANOLONE	FALSE	FALSE	FALSE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8761	iuphar.ligand:8761	COMPOUND 44 [PMID: 19748780]	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.095468493	LORNOXICAM	rxcui:20890	LORNOXICAM	TRUE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:11714	iuphar.ligand:11714	AZD7624	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9329	iuphar.ligand:9329	TAK-637	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:12349	iuphar.ligand:12349	ZIMBERELIMAB	FALSE	FALSE	FALSE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	1.000146118775133	PENICILLAMINE	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	DTC	9/2/20	NULL	11.66837138570988	4-(4-METHOXYPHENOXY)PHENOL	chembl:CHEMBL444161	CHEMBL:CHEMBL444161	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002421494	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.1651184630053286	ISOQUERCETIN	ncit:C117288	ISOQUERCETIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	GNF-PF-4464	chembl:CHEMBL600692	CHEMBL:CHEMBL600692	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012977675	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	1-(4-HYDROXYPHENYL)MALEIMIDE	chembl:CHEMBL565893	CHEMBL:CHEMBL565893	FALSE	FALSE	FALSE
TRHR	hgnc:12299	TRHR	DTC	9/2/20	NULL	0.5147810905460245	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.021661581	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NFATC1	hgnc:7775	NFATC1	PharmGKB	4/5/24	NULL	0.4526523382387457	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	NS-398	drugbank:DB14060	NS-398	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.100976291	IUPHAR.LIGAND:314	iuphar.ligand:314	MUSCARINIC TOXIN 7	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.3542686252046857	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.364636606	INK-1117	chembl:CHEMBL3545055	INK-1117	FALSE	FALSE	TRUE
HISTAMINE H4 RECEPTOR	hgnc:17383	HRH4	TTD	2020.06.01	NULL	9.546849315580817	UR-63325	chembl:CHEMBL3545345	UR-63325	FALSE	FALSE	FALSE
TNFRSF10C	hgnc:11906	TNFRSF10C	NCI	14-Sep-17	NULL	10.50153425	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.3977853881492007	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	1.438566335224506	SNA-120	ncit:C170295	PEGCANTRATINIB	FALSE	FALSE	FALSE
CCDC148	hgnc:25191	CCDC148	PharmGKB	4/5/24	NULL	2.917092846427472	letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.5527123287967841	IUPHAR.LIGAND:8595	iuphar.ligand:8595	[3H]OXOTREMORINE-M	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.021733308	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	1.381780822	Desoxycorticosterone Acetate	rxcui:258333	DESOXYCORTICOSTERONE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8117	iuphar.ligand:8117	COMPOUND 31 [PMID: 22902653]	FALSE	FALSE	FALSE
NCBIGENE:2244	hgnc:3662	FGB	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:12334	iuphar.ligand:12334	COMPOUND 25C [PMID: 36649216]	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ENNIATIN B	chembl:CHEMBL469036	ENNIATIN B	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	TRIADIMENOL	chembl:CHEMBL520275	TRIADIMENOL	FALSE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TEND	1-Aug-11	NULL	21.00306849427779	METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA	rxcui:729596	METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:367	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
UNIPROT:O00555	hgnc:1388	CACNA1A	TEND	1-Aug-11	NULL	0.4118248724368196	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.063784829	PD 0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.031254566	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:O43497	hgnc:1394	CACNA1G	TdgClinicalTrial	Jan-14	NULL	0.3977853881492008	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.2885036881082115	IUPHAR.LIGAND:1609	iuphar.ligand:1609	DSLET	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	ChEMBL	33	inhibitor	1.486066167047957	ENILURACIL	ncit:C1773	ENILURACIL	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2592971419046642	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.5527123287967841	IUPHAR.LIGAND:362	iuphar.ligand:362	W-84	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.037721028	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.048844345	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
ELANE	hgnc:3309	ELANE	DTC	9/2/20	NULL	4.565884455277782	SYMPLOSTATIN 5	chembl:CHEMBL2338554	SYMPLOSTATIN 5	FALSE	FALSE	FALSE
ATP8B1	hgnc:3706	ATP8B1	PharmGKB	4/5/24	NULL	8.751278539282415	odevixibat	rxcui:2563966	ODEVIXIBAT	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:7128	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
PIM2	hgnc:8987	PIM2	DTC	9/2/20	NULL	0.1474934585272317	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.069638821	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.5527123287967841	IUPHAR.LIGAND:363	iuphar.ligand:363	WDUO3	FALSE	FALSE	FALSE
MYD88	hgnc:7562	MYD88	PharmGKB	4/5/24	NULL	4.375639269641208	zanubrutinib	rxcui:2262435	ZANUBRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:367	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.075442056	PAZOPANI	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:2374	hgnc:3886	FRA2B	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8874	iuphar.ligand:8874	COMPOUND 33 [PMID: 19908842]	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.300043836	IUPHAR.LIGAND:2491	ncit:C1214	RESINIFERATOXIN	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.926605963	KN046	ncit:C157632	ERFONRILIMAB	FALSE	FALSE	FALSE
DNTT	hgnc:2983	DNTT	NCI	14-Sep-17	NULL	0.6250913242344582	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	0.6563458904461812	Volanesorsen	rxcui:2637345	VOLANESORSEN	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:324	iuphar.ligand:324	HIMBACINE	FALSE	FALSE	FALSE
UNIPROT:P49019	hgnc:16824	HCAR3	TEND	1-Aug-11	NULL	8.751278539282415	MEPENZOLATE	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1591141552596803	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.020465128	Flutamide	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.036162308	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.9546849315580818	CABIRALIZUMAB	ncit:C123831	CABIRALIZUMAB	FALSE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4167275494896388	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:7128	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.047049885	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.014849455	IUPHAR.LIGAND:209	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	DTC	9/2/20	NULL	5.250767123569449	OL-92	chembl:CHEMBL367966	CHEMBL:CHEMBL367966	FALSE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	Actimab-A	hemonc:10	ACTINIUM AC 225 LINTUZUMAB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	GYKI-52466	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	PharmGKB	4/5/24	NULL	0.9334697108567911	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
APOC1	hgnc:607	APOC1	PharmGKB	4/5/24	NULL	0.1440539677248134	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.034727296	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.022353202	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CALCITONIN RECEPTOR	hgnc:1440	CALCR	TTD	2020.06.01	NULL	13.12691780892362	Salmon Calcitonin	rxcui:36118	SALMON CALCITONIN	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	1.458546423213736	Paramethadione	rxcui:32894	PARAMETHADIONE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.031612084	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.027177884	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:301	ncit:C132273	MILAMELINE	FALSE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.3671865121377238	amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.072851434	Infliximab	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:438	iuphar.ligand:438	AS16	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:616	iuphar.ligand:616	BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1161674142382621	IUPHAR.LIGAND:1640	iuphar.ligand:1640	NALTRIBEN	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	inhibitor	0.05814803	IUPHAR.LIGAND:2312	iuphar.ligand:2312	BICUCULLINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	GNF-PF-4464	chembl:CHEMBL600692	CHEMBL:CHEMBL600692	FALSE	FALSE	FALSE
UNIPROT:Q14181	hgnc:30073	POLA2	TEND	1-Aug-11	NULL	1.000146118775133	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.003703461	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.7458476027797514	Bisoprolol	rxcui:19484	BISOPROLOL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	GNF-PF-4227	chembl:CHEMBL585654	CHEMBL:CHEMBL585654	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:75	iuphar.ligand:75	SB 272183	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.089298761	IUPHAR.LIGAND:3	iuphar.ligand:3	1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:6030	iuphar.ligand:6030	PURVALANOL A	FALSE	FALSE	FALSE
NCBIGENE:2608	hgnc:3594	FASN	GuideToPharmacology	2024.1	inhibitor	0.2991890098899972	IUPHAR.LIGAND:5277	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:367	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	1.750255707856483	QAW-039	ncit:C166588	FEVIPIPRANT	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.2778183663264259	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.043430663	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	SEMUSTINE	ncit:C827	SEMUSTINE	FALSE	FALSE	FALSE
SLC12A1	hgnc:10910	SLC12A1	ChEMBL	33	inhibitor	0.8334550989792778	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.084553416	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
PAPPA	hgnc:8602	PAPPA	NCI	14-Sep-17	NULL	2.386712328895204	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 3	hgnc:1104	BRD3	TTD	2020.06.01	NULL	0.7955707762984013	ABBV-744	iuphar.ligand:10730	ABBV-744	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:291	iuphar.ligand:291	NNC 11-1314	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.1651184630053286	ITF2357	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010687497	DEFEROXAMINE MESYLATE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.056399217	RETINAL	iuphar.ligand:2350	ALL-TRANS-RETINAL	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	LTT462	ncit:C126687	RINETERKIB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.3562257207306275	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.064347636	IUPHAR.LIGAND:129	iuphar.ligand:129	S33084	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:11934	iuphar.ligand:11934	ASP5878	FALSE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:6979	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	PHTHALAZINONE	chembl:CHEMBL124706	PHTHALAZINONE	FALSE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	8.751278539282415	Lexipafant	ncit:C170120	LEXIPAFANT	FALSE	FALSE	FALSE
PROLYL ENDOPEPTIDASE FAP	hgnc:3590	FAP	TTD	2020.06.01	NULL	4.039051633514961	BIBH 1	ncit:C2058	BIBH 1	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	5.250767123569449	Pyronaridine	ncit:C90737	PYRONARIDINE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.042073455	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.023482858	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.09669921	CALYCOSIN	chembl:CHEMBL241608	CALYCOSIN	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.2479701120930082	MILCICLIB	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	GNF-PF-1500	chembl:CHEMBL577673	CHEMBL:CHEMBL577673	FALSE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.2019525816757481	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.8204323630577265	adagrasib	rxcui:2625882	ADAGRASIB	TRUE	FALSE	TRUE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:295	iuphar.ligand:295	ARECAIDINE PROPARGYL ESTER	FALSE	FALSE	FALSE
PDE7A	hgnc:8791	PDE7A	DTC	9/2/20	NULL	7.001022831425932	ISOBUTYLMETHYLXANTHINE	drugbank:DB07954	3-ISOBUTYL-1-METHYL-7H-XANTHINE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	DTC	9/2/20	NULL	0.08334551	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.1238388472539964	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.03574382	IUPHAR.LIGAND:7082	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TdgClinicalTrial	Jan-14	NULL	0.5676504998453459	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.043976274	GALLIC ACID METHYL ESTER	chembl:CHEMBL65675	GALLIC ACID METHYL ESTER	FALSE	FALSE	FALSE
TAX TRANSCRIPTIONALLY-ACTIVATED GLYCOPROTEIN 1	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	3.500511415712966	RG7888	ncit:C121376	VONLEROLIZUMAB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.007366396	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.2778183663264259	DEHYDROEPIANDROSTERONE	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
GRB2	hgnc:4566	GRB2	NCI	14-Sep-17	NULL	0.4286340509036285	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.2651902587661338	CHLORHEXIDINE HYDROCHLORIDE	rxcui:2361	CHLORHEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:1896	iuphar.ligand:1896	AH6809	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.089756703	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:2018	hgnc:3341	EMX2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8169	iuphar.ligand:8169	COMPOUND A127 [WO2013110309]	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12706	drugbank:DB15498	BOS172722	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:3789	iuphar.ligand:3789	[125I]RELAXIN-3-B/INSL5 A CHIMERA	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.5147810905460245	D-ALANINE	drugbank:DB01786	D-ALANINE	FALSE	FALSE	FALSE
LIPOPROTEIN LIPASE	hgnc:6677	LPL	TTD	2020.06.01	NULL	0.1442518440541058	Gemfibrozil	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
CALR	hgnc:1455	CALR	NCI	14-Sep-17	NULL	0.5791287268642776	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.1600843635234588	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	DIALLYLDISULFIDE	chembl:CHEMBL366603	DIALLYLDISULFIDE	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	1.346350544504987	ABBV-744	iuphar.ligand:10730	ABBV-744	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:7354	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1164249916534246	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.053579256	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	PHENOXYBENZAMINE	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	BRL-54443	iuphar.ligand:3927	BRL-54443	FALSE	FALSE	FALSE
TPT1	hgnc:12022	TPT1	NCI	14-Sep-17	NULL	0.8824818695074705	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
SLC22A8	hgnc:10972	SLC22A8	DTC	9/2/20	NULL	2.500365296937833	DICLOXACILLIN	rxcui:3356	DICLOXACILLIN	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.099446347	IUPHAR.LIGAND:313	iuphar.ligand:313	MUSCARINIC TOXIN 3	FALSE	FALSE	FALSE
RPL5	hgnc:10360	RPL5	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.067897851	PAZOPANI	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:2598	hgnc:1372	CA14	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:6828	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.1037701012563132	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:10458	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	OncoKB	23-Jul-20	NULL	0.082043236	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.026372512	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	11.66837138570988	VEL-0230	chembl:CHEMBL1085282	CHEMBL:CHEMBL1085282	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.02926849	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:623	iuphar.ligand:623	[125I][TYR4]BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:2366	hgnc:3874	FRA1G	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8601	iuphar.ligand:8601	MI-1148	FALSE	FALSE	FALSE
NCBIGENE:936	hgnc:1647	CD24P2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7546	ncit:C174879	BITOPERTIN	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:313	iuphar.ligand:313	MUSCARINIC TOXIN 3	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:337	iuphar.ligand:337	KT 5720	FALSE	FALSE	FALSE
NCBIGENE:2996	hgnc:4705	GYPE	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9870	ncit:C95202	PIXATIMOD	FALSE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TEND	1-Aug-11	NULL	0.6731752722524935	TRANYLCYPROMINE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.027248402	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.2187819634820604	APAZONE	rxcui:1029	APAZONE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:291	iuphar.ligand:291	NNC 11-1314	FALSE	FALSE	FALSE
NCBIGENE:1878	ncbigene:1878	E11S	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:9311	iuphar.ligand:9311	URELUMAB	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.034567262	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:7128	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
RPLP0	hgnc:10371	RPLP0	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.033148782	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
LTF	hgnc:6720	LTF	NCI	14-Sep-17	NULL	1.009762908	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.017679351	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	1.640864726115453	n-desmethyltamoxifen	ncit:C64189	N-DESMETHYLTAMOXIFEN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.8008364246019593	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.020836377	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.2419708351875322	DNDI1417099	chembl:CHEMBL1565444	CHEMBL:CHEMBL1565444	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:7773	iuphar.ligand:7773	UCM 724	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.002631963	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	METHOXYCHLOR	rxcui:2598123	METHOXYCHLOR	FALSE	FALSE	FALSE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	0.1654653505326507	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
FOLR2	hgnc:3793	FOLR2	DTC	9/2/20	NULL	0.364636606	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1355	iuphar.ligand:1355	S26284	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.061041236	PERGOLIDE	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:2826	hgnc:4474	CCR10	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8030	iuphar.ligand:8030	L-739,750	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	1.029562181092048	IUPHAR.LIGAND:11314	iuphar.ligand:11314	CPY	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:10725	iuphar.ligand:10725	2F-MT-45	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1742	drugbank:DB04137	GUANOSINE-5'-TRIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10406	iuphar.ligand:10406	OD36	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2657	iuphar.ligand:2657	LY-510929	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	0.3542686252046857	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	2-BENZOYL-5-METHOXYBENZOQUINONE	chembl:CHEMBL1434057	2-BENZOYL-5-METHOXYBENZOQUINONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.025942525	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:9003	iuphar.ligand:9003	ADL5747	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.7001022831425933	NEUROPROTECTANTS	ncit:C1509	NEUROPROTECTIVE AGENT	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.082429625	IUPHAR.LIGAND:11691	iuphar.ligand:11691	ICI-199441	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	3.750547945	LY3381916	ncit:C143068	IDO-1 INHIBITOR LY3381916	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.2885036881082115	IUPHAR.LIGAND:9287	iuphar.ligand:9287	GSK1521498	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.3125456621172291	BALAMAPIMOD	ncit:C76769	BALAMAPIMOD	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1259176768242074	IUPHAR.LIGAND:12576	rxcui:18475	ATIPAMEZOLE	TRUE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:680	iuphar.ligand:680	BRADYZIDE	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:2361	drugbank:DB01931	5,7-DICHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1829	iuphar.ligand:1829	2-O-ETHYL-PAF C-16	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.071245144	LAS38096	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:7595	rxcui:6378	LEVORPHANOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.002796829	hydrocortisone	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.011585982	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00410569	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	0.036306082	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.038049037	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.076098074	ramucirumab	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.023014539	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
PSMC6	hgnc:9553	PSMC6	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.036062961	IUPHAR.LIGAND:7081	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.040703621	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
RPS24	hgnc:10411	RPS24	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	ChEMBL	33	inhibitor	0.789589041	APABETALONE	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
NCBIGENE:750	hgnc:1197	GAS8-AS1	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
RPL7	hgnc:10363	RPL7	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:5618	iuphar.ligand:5618	KF26777	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.2206204673768676	IUPHAR.LIGAND:7219	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.1166837138570989	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.1419126249613365	S-16924	iuphar.ligand:167	S 16924	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.3182283105193606	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:7571	iuphar.ligand:7571	PROTOXIN II	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00517674	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1363835616511545	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	1.230648544586589	elacridar	ncit:C73318	ELACRIDAR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003147942	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:10003	iuphar.ligand:10003	GNE-131	FALSE	FALSE	FALSE
UNIPROT:P62158	hgnc:1442	CALM1	TEND	1-Aug-11	NULL	0.7955707762984016	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.093763699	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CYSLTR1	hgnc:17451	CYSLTR1	PharmGKB	4/5/24	NULL	7.955707762984016	pranlukast	ncit:C96712	PRANLUKAST	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	activator	0.9376369863516875	IUPHAR.LIGAND:2626	iuphar.ligand:2626	VERATRIDINE	FALSE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:3635	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:12645	iuphar.ligand:12645	VIXOTRIGINE	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.072927321	IUPHAR.LIGAND:5893	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.082115757	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.089298761	TCMDC-125543	chembl:CHEMBL546170	CHEMBL:CHEMBL546170	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:5732	iuphar.ligand:5732	XEN907	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	FIPEXIDE HYDROCHLORIDE	chembl:CHEMBL1377408	FIPEXIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.006060442	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NOCICEPTIN RECEPTOR	hgnc:8155	OPRL1	TTD	2020.06.01	NULL	0.9376369863516874	PMX-53	iuphar.ligand:579	PMX53	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	0.3500511415712966	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007479725	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.046343929	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	L-689560	iuphar.ligand:4239	L689560	FALSE	FALSE	FALSE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1852122442176172	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	ALBUTROPIN	chembl:CHEMBL4298125	ALBUSOMATROPIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CIS/TRANS-ISOEUGENOL	chembl:CHEMBL2135887	CIS/TRANS-ISOEUGENOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TILIQUINOL	ncit:C72867	TILIQUINOL	FALSE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.050978322	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
NCBIGENE:585	hgnc:969	BBS4	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:12644	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
CYP20A1	hgnc:20576	CYP20A1	NCI	14-Sep-17	NULL	35.00511415712966	MBC	ncit:C1154	CARBENDAZIM	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.2983390411119005	JNJ-5207852	iuphar.ligand:1256	JNJ-5207852	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.1227531764715242	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	1.514644363	NELOTANSERIN	ncit:C83996	NELOTANSERIN	FALSE	FALSE	FALSE
TJP1	hgnc:11827	TJP1	NCI	14-Sep-17	NULL	0.4526523382387457	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
RETINOIC ACID RECEPTOR RXR-GAMMA	hgnc:10479	RXRG	TTD	2020.06.01	NULL	4.773424657790408	IRX4204	ncit:C140551	RETINOID X RECEPTOR AGONIST IRX4204	FALSE	FALSE	FALSE
NCBIGENE:3141	hgnc:4976	HLCS	GuideToPharmacology	2024.1	activator	26.25383561784724	IUPHAR.LIGAND:11143	iuphar.ligand:11143	LARGE PROLINE-RICH PROTEIN BAG6	FALSE	FALSE	FALSE
NOTCH1	hgnc:7881	NOTCH1	CancerCommons	25-Jul-13	inhibitor	3.938075342677087	RO4929097	iuphar.ligand:7338	RO4929097	FALSE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CGI	2/1/22	NULL	0.1269527834518725	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
ARAF	hgnc:646	ARAF	CGI	2/1/22	NULL	0.075369863	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:7697	iuphar.ligand:7697	AZD0328	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	CGI	2/1/22	NULL	0.007445784	Bortezomib	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CGI	2/1/22	NULL	0.1331836936859721	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KCNJ5	hgnc:6266	KCNJ5	CGI	2/1/22	NULL	0.3431873936973497	Amiloride	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CGI	2/1/22	NULL	0.3542686252046857	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.039361073	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.016131389	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.3547815624033412	ACETYLCHOLINE CHLORIDE	rxcui:20814	ACETYLCHOLINE CHLORIDE	TRUE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	0.8078103267029924	DICHLORPHENAMIDE	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
HTR1F	hgnc:5292	HTR1F	ChEMBL	33	agonist	0.5303805175322677	ELETRIPTAN HYDROBROMIDE	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	TRIHEXYPHENIDYL HYDROCHLORIDE	rxcui:1115	TRIHEXYPHENIDYL HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2792961235941196	TRIDIHEXETHYL CHLORIDE	rxcui:54421	TRIDIHEXETHYL CHLORIDE	TRUE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	0.3241214273808303	CYCLOTHIAZIDE	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.1988926940746003	TIMOLOL MALEATE	rxcui:42933	TIMOLOL MALEATE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	METOPROLOL TARTRATE	rxcui:203191	METOPROLOL TARTRATE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.041150213	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
NCBIGENE:2117	hgnc:3492	ETV3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8180	iuphar.ligand:8180	COMPOUND 31 [PMID: 20936789]	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.1491695205559502	PROPRANOLOL HYDROCHLORIDE	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	1.166837138570988	DOLASETRON MESYLATE	rxcui:29398	DOLASETRON MESYLATE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	ALOGLIPTIN BENZOATE	rxcui:1368000	ALOGLIPTIN BENZOATE	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.8975670296699915	ELETRIPTAN HYDROBROMIDE	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	1.009762908	FROVATRIPTAN SUCCINATE	rxcui:322249	FROVATRIPTAN SUCCINATE	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.2885036881082115	ERGOTAMINE TARTRATE	rxcui:42676	ERGOTAMINE TARTRATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.044611445	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2103	iuphar.ligand:2103	FK 224	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.047518255	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.057732459	PSEUDOEPHEDRINE HYDROCHLORIDE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	ELVITEGRAVIR	rxcui:1306286	ELVITEGRAVIR	TRUE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	agonist	3.850562557284263	PLERIXAFOR	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:3524	iuphar.ligand:3524	R-PSOP	FALSE	FALSE	FALSE
HSD3B2	hgnc:5218	HSD3B2	ChEMBL	33	inhibitor	13.12691780892362	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.2853677784548614	RUXOLITINIB PHOSPHATE	rxcui:1193325	RUXOLITINIB PHOSPHATE	TRUE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.8468979231563628	RUXOLITINIB PHOSPHATE	rxcui:1193325	RUXOLITINIB PHOSPHATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.0233679	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
NCBIGENE:1219	hgnc:10956	SLCO1A2	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:2765	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CA4	hgnc:1375	CA4	ChEMBL	33	inhibitor	1.093909817410302	ACETAZOLAMIDE SODIUM	rxcui:91406	ACETAZOLAMIDE SODIUM	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.6455861217503421	DROSPIRENONE	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.028413242	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	ChEMBL	33	potentiator	4.375639269641208	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	0.7425327245451747	ATORVASTATIN CALCIUM	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.029766254	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.034727296	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.035145697	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4570	rxcui:35616	RIFAMYCIN SV	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.006455332	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.007621958	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.1665148136438514	GUANFACINE HYDROCHLORIDE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1363835616511545	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	0.097236428	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.3017682254924971	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.1154014752432845	ERGOTAMINE TARTRATE	rxcui:42676	ERGOTAMINE TARTRATE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.1172046232939609	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.108711535	ERGOTAMINE TARTRATE	rxcui:42676	ERGOTAMINE TARTRATE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.081407242	VERAPAMIL HYDROCHLORIDE	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:2218	iuphar.ligand:2218	D(CH2)5[TYR(ME)2,THR4,PHE(3125I,4N3)-NH29]OVT	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2035181055647073	ISOETHARINE MESYLATE	rxcui:6024	ISOETHARINE MESYLATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2035181055647073	PENBUTOLOL SULFATE	rxcui:82070	PENBUTOLOL SULFATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2035181055647073	OXPRENOLOL HYDROCHLORIDE	rxcui:203131	OXPRENOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.8140724222588294	METAPROTERENOL SULFATE	rxcui:6804	METAPROTERENOL SULFATE	TRUE	FALSE	FALSE
PSMB8	hgnc:9545	PSMB8	ChEMBL	33	inhibitor	0.3182283105193606	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB7	hgnc:9544	PSMB7	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.5000730593875667	RAPACURONIUM BROMIDE	rxcui:228530	RAPACURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.4375639269641208	METOCURINE IODIDE	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:3870	iuphar.ligand:3870	DESGLYNH2-D(CH2)5[TYR(ME)2,THR4,ORN8]OT	FALSE	FALSE	FALSE
ATP1A3	hgnc:801	ATP1A3	ChEMBL	33	inhibitor	0.3281729452230906	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
ATP1B2	hgnc:805	ATP1B2	ChEMBL	33	inhibitor	0.8751278539282418	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.3182283105193605	IUPHAR.LIGAND:10444	iuphar.ligand:10444	LIT-001	FALSE	FALSE	FALSE
ATP1B3	hgnc:806	ATP1B3	ChEMBL	33	inhibitor	0.2573905452730122	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1718	iuphar.ligand:1718	ADENOSINE-3'-5'-BISPHOSPHATE	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.035574303	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.066297565	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.035574303	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.088396753	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:1725	iuphar.ligand:1725	PPADS	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.046518424	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.013560866	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.014206621	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.013876234	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:1734	drugbank:DB04005	URIDINE 5'-TRIPHOSPHATE	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.038894571	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.048083948	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	blocker	0.2019525816757481	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	blocker	0.1346350544504987	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	blocker	0.1553481397505754	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	0.084146909	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	blocker	0.2019525816757481	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	blocker	0.1553481397505754	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	blocker	0.1442518440541058	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1856	ncit:C65756	FOROPAFANT	FALSE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	blocker	0.2243917574174979	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	blocker	0.1442518440541058	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.063110182	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.051885051	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.050488145	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	modulator	0.9053046764774912	IUPHAR.LIGAND:12491	iuphar.ligand:12491	I-287	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.051277023	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.05293112	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.024197084	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.015702055	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.048260727	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.049026771	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inverse agonist	0.021846337	HALOPERIDOL DECANOATE	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.034590034	QUETIAPINE FUMARATE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.0296486	LEVOMEPROMAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.01858569	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inverse agonist	0.021846337	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	ChEMBL	33	inhibitor	0.063784829	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.2344092465879218	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.1136529680426287	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	0.1930429089547591	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.8899605294185507	PERINDOPRIL ARGININE	rxcui:1600711	PERINDOPRIL ARGININE	TRUE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.192335792	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.081030357	CT-1578	chembl:CHEMBL2035185	CT-1578	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1682938180631233	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.073954467	ALTIRATINIB	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	1.078924751	LAROTRECTINIB	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
PIM3	hgnc:19310	PIM3	ChEMBL	33	inhibitor	1.029562181092048	LGH-447	drugbank:DB14943	LGH-447	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	ChEMBL	33	inhibitor	5.000730593875666	MLN-0415	chembl:CHEMBL3545265	MLN-0415	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.052090944	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.3697723326457359	RG-7603	chembl:CHEMBL2331680	RG-7603	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.105947682	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.073437302	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	ChEMBL	33	inhibitor	0.085796848	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1875273972703375	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
GRM2	hgnc:4594	GRM2	ChEMBL	33	agonist	1.875273972703375	LY2969822	chembl:CHEMBL3545270	LY2969822	FALSE	FALSE	FALSE
P2RX7	hgnc:8537	P2RX7	ChEMBL	33	inhibitor	8.751278539282415	EVT401	chembl:CHEMBL3707396	EVT401	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	1.141471113819445	ABT-107	chembl:CHEMBL2151570	ABT-107	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.2917092846427472	CAFUSERTIB	chembl:CHEMBL3545354	CAFUSERTIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.099220845	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.440315901	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	ChEMBL	33	inhibitor	0.2972132334095915	ULIXERTINIB	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.091850154	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.034018575	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	1.438566335224506	PEGCANTRATINIB	ncit:C170295	PEGCANTRATINIB	FALSE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	3.889457128569962	LESOGABERAN	ncit:C166751	LESOGABERAN	FALSE	FALSE	FALSE
SCNN1A	hgnc:10599	SCNN1A	ChEMBL	33	blocker	3.500511415712966	IDREVLORIDE	ncit:C184934	IDREVLORIDE	FALSE	FALSE	FALSE
SCNN1G	hgnc:10602	SCNN1G	ChEMBL	33	blocker	1.944728564284981	IDREVLORIDE	ncit:C184934	IDREVLORIDE	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.5585922471882393	SOFINICLINE	ncit:C80527	SOFINICLINE	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.458546423213736	SOFINICLINE	ncit:C80527	SOFINICLINE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	modulator	0.2004109589148645	FOSDAGROCORAT	ncit:C170007	FOSDAGROCORAT	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.6326225450083675	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
MAP3K9	hgnc:6861	MAP3K9	ChEMBL	33	inhibitor	0.7292732116068681	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
PRKCI	hgnc:9404	PRKCI	ChEMBL	33	inhibitor	0.1458546423213736	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.2347585897273971	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2273059360852575	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	6.563458904461812	TRALOKINUMAB	rxcui:2589225	TRALOKINUMAB	TRUE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	ChEMBL	33	agonist	5.834185692854944	TIGATUZUMAB	ncit:C62482	TIGATUZUMAB	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	1.944728564284981	MOXETUMOMAB PASUDOTOX	rxcui:2099295	MOXETUMOMAB PASUDOTOX	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	agonist	0.050174554	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	modulator	0.038104261	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	modulator	0.1442518440541058	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CA9	hgnc:1383	CA9	ChEMBL	33	binder	3.750547945	CG250 111IN	chembl:CHEMBL3707280	CG250 111IN	FALSE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	modulator	0.2019525816757481	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
KCNA6	hgnc:6225	KCNA6	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.003739863	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNA10	hgnc:6219	KCNA10	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCND1	hgnc:6237	KCND1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNH5	hgnc:6254	KCNH5	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.2778183663264259	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
TPBG	hgnc:12004	TPBG	ChEMBL	33	other/unknown	21.00306849427779	NAPTUMOMAB ESTAFENATOX	ncit:C95789	NAPTUMOMAB ESTAFENATOX	FALSE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	negative modulator	3.281729452230906	KELIXIMAB	ncit:C188517	KELIXIMAB	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	inhibitor	0.7001022831425933	FORALUMAB	ncit:C95785	FORALUMAB	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	other/unknown	1.944728564284981	MDX-070	chembl:CHEMBL2109555	MDX-070	FALSE	FALSE	FALSE
TNC	hgnc:5318	TNC	ChEMBL	33	other/unknown	6.563458904461812	F16IL2	chembl:CHEMBL2109583	F16IL2	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.027752469	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.085239726	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.078136416	MOXISYLYTE	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.108711535	MOXISYLYTE	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	1.141471113819445	SITAXENTAN SODIUM	ncit:C152373	SITAXENTAN SODIUM	TRUE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	1.875273972703375	SITAXENTAN SODIUM	ncit:C152373	SITAXENTAN SODIUM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	binder	0.3454452054979901	T-DM1	chembl:CHEMBL2109399	T-DM1	FALSE	FALSE	FALSE
MTNR1A	hgnc:7463	MTNR1A	ChEMBL	33	agonist	1.875273972703375	AGOMELATINE	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
CD70	hgnc:11937	CD70	ChEMBL	33	binder	4.039051633514961	VORSETUZUMAB	ncit:C152916	VORSETUZUMAB	FALSE	FALSE	FALSE
MTNR1B	hgnc:7464	MTNR1B	ChEMBL	33	agonist	2.625383561784724	AGOMELATINE	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.032016873	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	ALOXIPRIN	rxcui:17393	ALOXIPRIN	TRUE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	KD-247	chembl:CHEMBL2109446	KD-247	FALSE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	binder	8.078103267029922	IMGN-388	chembl:CHEMBL2109633	IMGN-388	FALSE	FALSE	FALSE
IFNA6	hgnc:5427	IFNA6	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.6563458904461812	RINUCUMAB	ncit:C152224	RINUCUMAB	FALSE	FALSE	FALSE
RPS16	hgnc:10396	RPS16	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS3	hgnc:10420	RPS3	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS15A	hgnc:10389	RPS15A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RHD	hgnc:10009	RHD	ChEMBL	33	inhibitor	13.12691780892362	MOROLIMUMAB	ncit:C188621	MOROLIMUMAB	FALSE	FALSE	FALSE
RPS27A	hgnc:10417	RPS27A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS21	hgnc:10409	RPS21	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL37	hgnc:10347	RPL37	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL41	hgnc:10354	RPL41	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
HLA-DRB4	hgnc:4952	HLA-DRB4	ChEMBL	33	inhibitor	4.375639269641208	APOLIZUMAB	ncit:C2228	APOLIZUMAB	FALSE	FALSE	FALSE
HLA-DRB5	hgnc:4953	HLA-DRB5	ChEMBL	33	inhibitor	2.625383561784724	APOLIZUMAB	ncit:C2228	APOLIZUMAB	FALSE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	ChEMBL	33	blocker	0.1562728310586145	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	blocker	0.1250182648468916	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNA4	hgnc:6222	KCNA4	ChEMBL	33	blocker	0.1785975212098452	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNH1	hgnc:6250	KCNH1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	0.9845188356692718	GLESATINIB	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1479089330582944	GLESATINIB	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
KCNG3	hgnc:18306	KCNG3	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNC2	hgnc:6234	KCNC2	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNH4	hgnc:6253	KCNH4	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNH8	hgnc:18864	KCNH8	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNG2	hgnc:6249	KCNG2	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNV2	hgnc:19698	KCNV2	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNF1	hgnc:6246	KCNF1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNC4	hgnc:6236	KCNC4	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.3659071166250487	CEMIPLIMAB	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.4773424657790409	BRECANAVIR	ncit:C76908	BRECANAVIR	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.055155117	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.1093909817410302	TRASTUZUMAB DERUXTECAN	rxcui:2267574	FAM-TRASTUZUMAB DERUXTECAN-NXKI	TRUE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.047518255	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
RPS6	hgnc:10429	RPS6	ChEMBL	33	inhibitor	0.092118721	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPS5	hgnc:10426	RPS5	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPS2	hgnc:10404	RPS2	ChEMBL	33	inhibitor	0.092118721	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS20	hgnc:10405	RPS20	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL15	hgnc:10306	RPL15	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL21	hgnc:10313	RPL21	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL6	hgnc:10362	RPL6	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL23	hgnc:10316	RPL23	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NPR1	hgnc:7943	NPR1	ChEMBL	33	agonist	16.15620653405984	PL-3994	drugbank:DB15355	PL-3994	FALSE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	1.009762908	VERICIGUAT	rxcui:2475830	VERICIGUAT	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.5834185692854944	TOFIMILAST	ncit:C76891	TOFIMILAST	FALSE	FALSE	FALSE
RPS4X	hgnc:10424	RPS4X	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.6250913242344582	TOFIMILAST	ncit:C76891	TOFIMILAST	FALSE	FALSE	FALSE
RPS11	hgnc:10384	RPS11	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS4Y1	hgnc:10425	RPS4Y1	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS8	hgnc:10441	RPS8	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:3438	rxcui:21149	CIPROFIBRATE	TRUE	FALSE	FALSE
RPS27	hgnc:10416	RPS27	ChEMBL	33	modulator	0.091476779	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS10	hgnc:10383	RPS10	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.2651902587661338	IUPHAR.LIGAND:2666	iuphar.ligand:2666	PIRINIXIC ACID	FALSE	FALSE	FALSE
RPS25	hgnc:10413	RPS25	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS23	hgnc:10410	RPS23	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL3	hgnc:10332	RPL3	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2673	iuphar.ligand:2673	GW9578	FALSE	FALSE	FALSE
RPS16	hgnc:10396	RPS16	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL10A	hgnc:10299	RPL10A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL17	hgnc:10307	RPL17	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS15	hgnc:10388	RPS15	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS15A	hgnc:10389	RPS15A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS21	hgnc:10409	RPS21	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL9	hgnc:10369	RPL9	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL13	hgnc:10303	RPL13	ChEMBL	33	modulator	0.091476779	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:2497	hgnc:3989	FTH1P2	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8877	iuphar.ligand:8877	P6949	FALSE	FALSE	FALSE
RPL14	hgnc:10305	RPL14	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL32	hgnc:10336	RPL32	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.021850883	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
RPL31	hgnc:10334	RPL31	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL27	hgnc:10328	RPL27	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	EVOBRUTINIB	ncit:C141427	EVOBRUTINIB	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:9928	iuphar.ligand:9928	PUQUITINIB	FALSE	FALSE	FALSE
TLR3	hgnc:11849	TLR3	ChEMBL	33	activator	2.625383561784724	BEVASIRANIB	ncit:C169809	BEVASIRANIB	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.4375639269641208	7-ETHYL-10-HYDROXYCAMPTOTHECIN	ncit:C61618	7-ETHYL-10-HYDROXYCAMPTOTHECIN	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.596678082	BICIFADINE	ncit:C79930	BICIFADINE	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.1141471113819445	GUSACITINIB	ncit:C166736	GUSACITINIB	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.1693795846312726	GUSACITINIB	ncit:C166736	GUSACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.021070494	IUPHAR.LIGAND:7940	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PTGER2	hgnc:9594	PTGER2	ChEMBL	33	agonist	3.281729452230906	TAPRENEPAG ISOPROPYL	ncit:C152513	TAPRENEPAG ISOPROPYL	FALSE	FALSE	FALSE
ELANE	hgnc:3309	ELANE	ChEMBL	33	inhibitor	4.565884455277782	DEPELESTAT	ncit:C87386	DEPELESTAT	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:7743	iuphar.ligand:7743	IZORLISIB	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	ChEMBL	33	inhibitor	1.050153425	AZD-1236	drugbank:DB11961	AZD-1236	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	negative modulator	0.039538909	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.3517260274161354	FUTIBATINIB	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:8974	iuphar.ligand:8974	OMIPALISIB	FALSE	FALSE	FALSE
E2F3	hgnc:3115	E2F3	ChEMBL	33	inhibitor	1.640864726115453	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ChEMBL	33	inhibitor	1.458546423213736	ZOTAROLIMUS	ncit:C82294	ZOTAROLIMUS	FALSE	FALSE	FALSE
E2F6	hgnc:3120	E2F6	ChEMBL	33	inhibitor	2.187819634820604	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	ChEMBL	33	inhibitor	0.6563458904461812	APG115	chembl:CHEMBL4091801	APG115	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	ChEMBL	33	agonist	2.500365296937833	SETMELANOTIDE ACETATE	rxcui:2469248	SETMELANOTIDE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:1310	hgnc:2196	COL19A1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9617	ncit:C170150	MARDEPODECT	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	0.5048814541893701	BELVARAFENIB	ncit:C121646	BELVARAFENIB	FALSE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.2692701089009974	RIPASUDIL	ncit:C152226	RIPASUDIL	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.089756703	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
NCBIGENE:2858	ncbigene:2858	GPR34P	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11793	iuphar.ligand:11793	BAY-091	FALSE	FALSE	FALSE
WT1	hgnc:12796	WT1	ChEMBL	33	vaccine	4.039051633514961	OMBIPEPIMUT-S	chembl:CHEMBL4297235	OMBIPEPIMUT-S	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	DICLOFENAC ETALHYALURONATE SODIUM	ncit:C174668	DICLOFENAC ETALHYALURONATE SODIUM	FALSE	FALSE	FALSE
LGR4	hgnc:13299	LGR4	ChEMBL	33	inhibitor	26.25383561784724	ROSMANTUZUMAB	ncit:C122921	ROSMANTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:8784	iuphar.ligand:8784	SGI-1776	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:10676	iuphar.ligand:10676	AZ1366	FALSE	FALSE	FALSE
ERVW-1	hgnc:13525	ERVW-1	ChEMBL	33	inhibitor	52.50767123569449	TEMELIMAB	ncit:C170386	TEMELIMAB	FALSE	FALSE	FALSE
MAP3K8	hgnc:6860	MAP3K8	ChEMBL	33	inhibitor	3.500511415712966	TILPISERTIB	ncit:C175865	TILPISERTIB	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	ChEMBL	33	positive modulator	1.381780822	EFTRENONACOG ALFA	rxcui:1535944	COAGULATION FACTOR IX RECOMBINANT IMMUNOGLOBULIN G1 FUSION PROTEIN	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	2.500365296937833	SEPETAPROST	ncit:C152337	SEPETAPROST	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	1.207072901969988	MITIGLINIDE	ncit:C81699	MITIGLINIDE	TRUE	FALSE	FALSE
NCBIGENE:2388	hgnc:3900	FRA4A	GuideToPharmacology	2024.1	NULL	7.501095891	IUPHAR.LIGAND:10713	iuphar.ligand:10713	COMPOUND 16 [PMID: 31653597]	FALSE	FALSE	FALSE
UGCG	hgnc:12524	UGCG	ChEMBL	33	inhibitor	5.250767123569449	VENGLUSTAT	ncit:C152852	VENGLUSTAT	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:12347	iuphar.ligand:12347	PENPULIMAB	FALSE	FALSE	FALSE
MARCKS	hgnc:6759	MARCKS	ChEMBL	33	inhibitor	105.0153424713889	BIO-11006	drugbank:DB14886	BIO-11006	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	0.1367387271762877	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.076098074	XYLOMETAZOLINE	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
MYH7	hgnc:7577	MYH7	ChEMBL	33	inhibitor	1.944728564284981	MAVACAMTEN	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
CCND2	hgnc:1583	CCND2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.4286340509036285	PD 0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2041114528112516	PD 0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CCND3	hgnc:1585	CCND3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3750547945406749	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1190650141398968	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.066297565	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.097236428	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:1162	hgnc:18762	SLC36A2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4693	iuphar.ligand:4693	&ALPHA;-METHYL-D,L-TRYPTOPHAN	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.039420174	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1495945049449985	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.06335385	PF-05212384	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
CFLAR	hgnc:1876	CFLAR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.9376369863516874	DEHYDROEQUOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2465148884304905	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.06375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.05348829	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
VEGFB	hgnc:12681	VEGFB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6563458904461812	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1788	iuphar.ligand:1788	PTHRP-(1-21)/PTH-(22-34) (HUMAN)	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.097236428	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	2.019525817	CHAULMOSULFONE	ncit:C76257	CHAULMOSULFONE	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.082559232	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.092606122	RETINAL	iuphar.ligand:2350	ALL-TRANS-RETINAL	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	DTC	9/2/20	NULL	0.019468918	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.1093909817410302	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	MANEB	chembl:CHEMBL491517	MANEB	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	3.387591692625451	(-)-ZILEUTON	chembl:CHEMBL1164975	CHEMBL:CHEMBL1164975	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:5575	iuphar.ligand:5575	[ALA1,12,AIB3,GLN10,HARG11,TRP14,ARG19]PTH-(1-21)-NH2 (HUMAN)	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-236687	chembl:CHEMBL318892	CHEMBL:CHEMBL318892	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	DNDI1417827	chembl:CHEMBL1363249	CHEMBL:CHEMBL1363249	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.031317948	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.005697447	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1874	iuphar.ligand:1874	PRRP-31	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CETALKONIUM CHLORIDE	rxcui:47907	CETALKONIUM CHLORIDE	TRUE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.045579576	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1909369863116163	NSC-111847	chembl:CHEMBL1984884	CHEMBL:CHEMBL1984884	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	LECANORIC ACID	chembl:CHEMBL1451874	LECANORIC ACID	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.2143170254518142	FUSARIC ACID	chembl:CHEMBL24510	FUSARIC ACID	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	CID 649849	chembl:CHEMBL405914	CHEMBL:CHEMBL405914	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	DIFENOCONAZOLE	chembl:CHEMBL466426	DIFENOCONAZOLE	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.017352172	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.023233483	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.043756393	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.045778266	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:1816	iuphar.ligand:1816	TIP39-(3-39) (HUMAN/BOVINE)	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.024309107	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
PPIA	hgnc:9253	PPIA	DTC	9/2/20	NULL	0.4310974649892816	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:1815	iuphar.ligand:1815	TIP39	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	CETYLPYRIDINIUM CHLORIDE	rxcui:2287	CETYLPYRIDINIUM CHLORIDE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.073437302	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001967464	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.014299475	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.018860514	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:1810	iuphar.ligand:1810	[TYR34]PTH-(1-34) (HUMAN)	FALSE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	1.400204566285186	SILYDIANIN	chembl:CHEMBL2397733	SILIDIANIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	IBUFENAC	ncit:C96750	IBUFENAC	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	L-165041	drugbank:DB08078	{4-[3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPOXY]PHENOXY}ACETIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	MMV666022	chembl:CHEMBL599100	CHEMBL:CHEMBL599100	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.012466209	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	NSC-656158	chembl:CHEMBL280099	CHEMBL:CHEMBL280099	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:1788	iuphar.ligand:1788	PTHRP-(1-21)/PTH-(22-34) (HUMAN)	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.060353645	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.004410927	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1136529680426287	L-165041	drugbank:DB08078	{4-[3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPOXY]PHENOXY}ACETIC ACID	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.096937239	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005835482	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	ISOQUERCETIN	ncit:C117288	ISOQUERCETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ENILCONAZOLE	rxcui:1442172	ENILCONAZOLE	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1799	iuphar.ligand:1799	[ILE5,TRP23]PTHRP-(2-36) (HUMAN)	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.017295017	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.035358701	TRANILAST	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	SJ000014858	chembl:CHEMBL591628	CHEMBL:CHEMBL591628	FALSE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.1810609352954982	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
NCBIGENE:3006	hgnc:4716	H1-2	GuideToPharmacology	2024.1	activator	7.501095891	IUPHAR.LIGAND:10650	iuphar.ligand:10650	COMPOUND 16 [PMID: 31977207]	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.5000730593875666	DIHYDROXANTHOHUMOL	chembl:CHEMBL510279	DIHYDROXANTHOHUMOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	1.250182648468916	PIMARIC ACID	chembl:CHEMBL1410398	PIMARIC ACID	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1400204566285186	CLOROPHENE	rxcui:21290	CLOROPHENE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.006286838	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.028977744	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.00770359	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.1312691780892362	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013021444	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.2333674277141977	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:2412	hgnc:3923	FRA7E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8556	iuphar.ligand:8556	COMPOUND 3 [PMID: 17942791]	FALSE	FALSE	FALSE
NLRP1	hgnc:14374	NLRP1	DTC	9/2/20	NULL	2.019525816757481	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.2243917574174978	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.03043923	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	XANTHOANGELOL	chembl:CHEMBL494083	XANTHOANGELOL	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	2.763561643983921	TCMDC-125182	chembl:CHEMBL588143	CHEMBL:CHEMBL588143	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TRIBUTYLCHLOROSTANNANE	chembl:CHEMBL1088186	TRIBUTYLCHLOROSTANNANE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	L-733060	chembl:CHEMBL1256740	CHEMBL:CHEMBL1256740	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.051177067	DITHIOLETHIONE	chembl:CHEMBL368700	DITHIOLETHIONE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	N-METHYLCALOTHRIXIN B	chembl:CHEMBL560303	N-METHYLCALOTHRIXIN B	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:9661	iuphar.ligand:9661	GSK2981278	FALSE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.2651902587661338	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	3,5-DINITROCATECHOL (OR-486)	chembl:CHEMBL168276	3,5-DINITROCATECHOL (OR-486)	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	SRT-2183	chembl:CHEMBL403308	CHEMBL:CHEMBL403308	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-3445	chembl:CHEMBL582697	CHEMBL:CHEMBL582697	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	DNDI1417149	chembl:CHEMBL1622802	CHEMBL:CHEMBL1622802	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	CHLORHEXIDINE HYDROCHLORIDE	rxcui:2361	CHLORHEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.033985548	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	PYRIDOSTIGMINE	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:599	hgnc:995	BCL2L2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:2741	iuphar.ligand:2741	ALL-TRANS-4-OXO-RETINOIC ACID	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.091159151	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	GIPARMEN	ncit:C74115	GIPARMEN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.002851353	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.099446347	INDACATEROL	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	CIGLITAZONE	ncit:C72726	CIGLITAZONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004847011	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	GNF-PF-1549	chembl:CHEMBL227959	CHEMBL:CHEMBL227959	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.027433475	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007479725	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	SJ000014858	chembl:CHEMBL591628	CHEMBL:CHEMBL591628	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	CI-966	iuphar.ligand:4612	CI-966	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.059837802	GNF-PF-3889	chembl:CHEMBL598270	CHEMBL:CHEMBL598270	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1458546423213736	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007699637	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.022267884	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.005497034	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	TRYPTANTHRIN	iuphar.ligand:8224	TRYPTANTHRIN	FALSE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.051987793	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	IMIQUIMOD	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	CF102	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.097236428	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.01261294	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.001460169	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	CGP-74514A	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01715937	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	CHLORHEXIDINE HYDROCHLORIDE	rxcui:2361	CHLORHEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	PHANQUONE	ncit:C90620	PHANQUONE	FALSE	FALSE	FALSE
CAMK2A	hgnc:1460	CAMK2A	DTC	9/2/20	NULL	0.2273059360852576	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.089756703	MILTIRONE	chembl:CHEMBL45830	MILTIRONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	SJ000018300	chembl:CHEMBL590927	CHEMBL:CHEMBL590927	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	(S)-AMPA	drugbank:DB02057	(S)-AMPA	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.002543976	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.023274677	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
AKT2	hgnc:392	AKT2	DTC	9/2/20	NULL	0.069454592	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.1244847587380144	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	DTC	9/2/20	NULL	0.364636606	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.003708169	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.364636606	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	TAXIFOLIN	drugbank:DB02224	TAXIFOLIN	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	MAKALUVAMINE A	chembl:CHEMBL449905	MAKALUVAMINE A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
TNNI3	hgnc:11947	TNNI3	DTC	9/2/20	NULL	0.364636606	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.9053046764774912	FENOTEROL HBR	chembl:CHEMBL537445	FENOTEROL HBR	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.006250913	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.030996264	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	QUINESTROL	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	TORSEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.014537008	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	MALTOL	rxcui:1362894	MALTOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	PF-03715455	drugbank:DB12138	PF-03715455	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	METHYL ROBUSTONE	chembl:CHEMBL1403041	METHYL ROBUSTONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-242717	chembl:CHEMBL269450	CHEMBL:CHEMBL269450	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:10133	iuphar.ligand:10133	COMPOUND 27 [PMID: 24900635]	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.050294704	DNDI1318925	chembl:CHEMBL1390716	CHEMBL:CHEMBL1390716	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	6'-IODONONIVAMIDE	chembl:CHEMBL177809	CHEMBL:CHEMBL177809	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.364636606	METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE	chembl:CHEMBL1214407	CHEMBL:CHEMBL1214407	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.015858554	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.015127534	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	CID 5310801	chembl:CHEMBL260451	CHEMBL:CHEMBL260451	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	2-BENZOYL-5-METHOXYBENZOQUINONE	chembl:CHEMBL1434057	2-BENZOYL-5-METHOXYBENZOQUINONE	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:10695	iuphar.ligand:10695	SOVESUDIL	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2917092846427472	CID 100335	chembl:CHEMBL1520346	CHEMBL:CHEMBL1520346	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	GW9662	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	AMITRAZ	rxcui:17763	AMITRAZ	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007727398	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1991	iuphar.ligand:1991	[33P]RELAXIN (HUMAN)	FALSE	FALSE	FALSE
USP5	hgnc:12628	USP5	DTC	9/2/20	NULL	52.50767123569449	VIALININ A	iuphar.ligand:8669	VIALININ A	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.014658758	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	HYDROCORTISONE SODIUM PHOSPHATE	rxcui:235482	HYDROCORTISONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010678802	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.00825852	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.023171964	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.012325744	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.056399217	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.01274458	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.6819178082557726	LEUCETTAMINE B	chembl:CHEMBL485053	LEUCETTAMINE B	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	DICHLORORIBOBENZIMIDAZOLE	iuphar.ligand:5178	DRB	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:4372	iuphar.ligand:4372	INSL3 B CHAIN DIMER ANALOGUE 8	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.003687336	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:2917	iuphar.ligand:2917	JTE-013	FALSE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	DTC	9/2/20	NULL	0.5147810905460244	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.023493365	ZOXAZOLAMINE	ncit:C152966	ZOXAZOLAMINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	PROADIFEN HYDROCHLORIDE	ncit:C66468	PROADIFEN HYDROCHLORIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
DHRS9	hgnc:16888	DHRS9	DTC	9/2/20	NULL	15.00219178	(+)-ISOZONARONE	chembl:CHEMBL459574	CHEMBL:CHEMBL459574	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.023630815	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.008804103	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	SULFAQUINOXALINE	rxcui:1306111	SULFAQUINOXALINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:8709	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	DORSOMORPHIN	drugbank:DB08597	DORSOMORPHIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	IFENPRODIL	rxcui:27403	IFENPRODIL	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.03729238	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.000855871	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1017590527823536	THUNBERGINOL A	chembl:CHEMBL68810	THUNBERGINOL A	FALSE	FALSE	FALSE
NCBIGENE:2198	ncbigene:2198	FAUNA@	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8049	iuphar.ligand:8049	HG-9-91-01	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	SJ000066481	chembl:CHEMBL588749	CHEMBL:CHEMBL588749	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	PROROXAN HYDROCHLORIDE	ncit:C84120	PROROXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	ARACHIDONOYL DOPAMINE	iuphar.ligand:4261	NADA	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.01199079	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.3684748858645227	QUERCETAGETIN	chembl:CHEMBL413552	QUERCETAGETIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	NSC-50654	chembl:CHEMBL1372046	CHEMBL:CHEMBL1372046	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.045579576	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.034162441	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1367387271762877	JL-18	chembl:CHEMBL63329	CHEMBL:CHEMBL63329	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	P-PHENYLENEDIAMINE	rxcui:1362740	4-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	BMS-191011	chembl:CHEMBL45349	CHEMBL:CHEMBL45349	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.021697385	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
NCBIGENE:2511	hgnc:16253	SPTLC3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:6664	iuphar.ligand:6664	MYRIOCIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.025840389	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003874533	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	THIOPHANATE METHYL	chembl:CHEMBL487187	THIOPHANATE METHYL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-4803	chembl:CHEMBL585240	CHEMBL:CHEMBL585240	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	RAC-GONIOTHALAMIN	chembl:CHEMBL1170485	CHEMBL:CHEMBL1170485	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.055819636	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.4526523382387456	GNF-PF-1260	chembl:CHEMBL584849	CHEMBL:CHEMBL584849	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	RETINAL	iuphar.ligand:2350	ALL-TRANS-RETINAL	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.011171845	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.1238388472539964	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	SJ000260214	chembl:CHEMBL602740	CHEMBL:CHEMBL602740	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
NCBIGENE:2214	hgnc:3619	FCGR3A	GuideToPharmacology	2024.1	inhibitor	0.082559232	IUPHAR.LIGAND:7949	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.042436157	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01323278	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	OTILONIUM	rxcui:32311	OCTYLONIUM	FALSE	FALSE	FALSE
KLF5	hgnc:6349	KLF5	DTC	9/2/20	NULL	0.7292732116068681	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.1325951293830669	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	PHENYL BIGUANIDE	iuphar.ligand:2284	1-PHENYLBIGUANIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	PENTAMIDINE DIISETHIONATE	chembl:CHEMBL361506	PENTAMIDINE ISETHIONATE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.42006137	GLABROL	chembl:CHEMBL462721	GLABROL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	NSC-154983	chembl:CHEMBL227298	CHEMBL:CHEMBL227298	FALSE	FALSE	FALSE
NCBIGENE:2225	hgnc:11408	STK4	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.01905213	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	FOLPET	chembl:CHEMBL1883819	FOLPET	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.082429625	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.002126161	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	HYDROXYZINE	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.014160645	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.2853677784548614	TCMDC-123789	chembl:CHEMBL588859	CHEMBL:CHEMBL588859	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	METHYL ROBUSTONE	chembl:CHEMBL1403041	METHYL ROBUSTONE	FALSE	FALSE	FALSE
NCBIGENE:1538	hgnc:2582	CYLC1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8219	iuphar.ligand:8219	COMPOUND 74 [PMID: 24793884]	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	OXADIAZON	chembl:CHEMBL1080648	OXADIAZON	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.08334551	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.07767407	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	EPIRUBICIN HYDROCHLORIDE	rxcui:203213	EPIRUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.045304289	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.02804897	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.016992774	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	N-METHYL-D-ASPARTIC ACID (NMDA)	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.6250913242344582	LEUCETTAMINE B	chembl:CHEMBL485053	LEUCETTAMINE B	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	DNDI1417827	chembl:CHEMBL1363249	CHEMBL:CHEMBL1363249	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	2',4'-DIHYDROXYCHALCONE	chembl:CHEMBL105310	2',4'-DIHYDROXYCHALCONE	FALSE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.046343929	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.013957382	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	GERONTOXANTHONE H	chembl:CHEMBL514057	GERONTOXANTHONE H	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	SIDURON	chembl:CHEMBL1902120	SIDURON	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00389812	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.005602611	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.014243231	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:7435	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
PADI4	hgnc:18368	PADI4	DTC	9/2/20	NULL	6.563458904461812	O-CL-AMIDINE	chembl:CHEMBL1910971	CHEMBL:CHEMBL1910971	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001914661	ISOPRENALINE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00410569	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00317843	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	N6-2-PHENYLETHYLADENOSINE	chembl:CHEMBL1257013	CHEMBL:CHEMBL1257013	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	GNF-PF-2968	chembl:CHEMBL582473	CHEMBL:CHEMBL582473	FALSE	FALSE	FALSE
NCBIGENE:1534	hgnc:2571	CYB561	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9423	iuphar.ligand:9423	COMPOUND 14N [PMID: 25589934]	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	JNJ-16259685	iuphar.ligand:1385	JNJ16259685	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.6177373086552295	IRL-2500	iuphar.ligand:3887	IRL 2500	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.008275441	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.099446347	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	CALYCOSIN	chembl:CHEMBL241608	CALYCOSIN	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.072524408	NSC-353263	chembl:CHEMBL1383812	CHEMBL:CHEMBL1383812	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	CASTANOSPERMINE	drugbank:DB01816	CASTANOSPERMINE	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.023264365	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	TCMDC-124327	chembl:CHEMBL581929	CHEMBL:CHEMBL581929	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.085239726	MMV006513	chembl:CHEMBL585622	CHEMBL:CHEMBL585622	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.2430910705356226	HYPEROSIDE	chembl:CHEMBL251254	HYPEROSIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	CLIOXANIDE	ncit:C65338	CLIOXANIDE	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.090530468	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.034453853	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
NCBIGENE:1136	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	antibody	1.591141552596803	IUPHAR.LIGAND:8405	iuphar.ligand:8405	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	BAS-8770957	chembl:CHEMBL500812	CHEMBL:CHEMBL500812	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	DEFERASIROX	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.030176823	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	PYRIDOSTIGMINE	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.029301156	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.025489161	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.034118045	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	QUINAPRIL HYDROCHLORIDE	rxcui:235759	QUINAPRIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	RETINAL	iuphar.ligand:2350	ALL-TRANS-RETINAL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	THIOGUANOSINE	chembl:CHEMBL283078	THIOGUANOSINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	DROFENINE HYDROCHLORIDE	chembl:CHEMBL1368313	DROFENINE HYDROCHLORIDE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	LASSBIO-294	chembl:CHEMBL233194	CHEMBL:CHEMBL233194	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1367387271762877	CHLORHEXIDINE HYDROCHLORIDE	rxcui:2361	CHLORHEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	(R)-NITRENDIPINE	chembl:CHEMBL268609	(R)-NITRENDIPINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	THIOTHIXENE	rxcui:10510	THIOTHIXENE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.056888051	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.033529803	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
NPY1R	hgnc:7956	NPY1R	DTC	9/2/20	NULL	2.625383561784724	METOPROLOL TARTRATE	rxcui:203191	METOPROLOL TARTRATE	TRUE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.2430910705356227	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.069089041	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.1988926940746004	ABACAVIR	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.021301287	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124399	chembl:CHEMBL582180	CHEMBL:CHEMBL582180	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1325951293830669	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	PROPICONAZOLE	ncit:C97997	PROPICONAZOLE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	DIALLYLDISULFIDE	chembl:CHEMBL366603	DIALLYLDISULFIDE	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1325951293830669	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	CID 649849	chembl:CHEMBL405914	CHEMBL:CHEMBL405914	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.048083948	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-633825	iuphar.ligand:8642	SB-633825	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.026385764	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.042140988	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.2573905452730122	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	GLYASPERIN D	chembl:CHEMBL1563332	GLYASPERIN D	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	DTC	9/2/20	NULL	0.2041114528112516	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CCND1	hgnc:1582	CCND1	DTC	9/2/20	NULL	0.063784829	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.02617531	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.042481935	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	BROMOETHANE	chembl:CHEMBL156378	BROMOETHANE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.021554873	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1363835616511545	DILAZEP	ncit:C65389	DILAZEP	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.3281729452230906	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
AKR1B10	hgnc:382	AKR1B10	DTC	9/2/20	NULL	2.187819634820604	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.027361996	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.042344896	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.047561296	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	NU-1025	chembl:CHEMBL123904	CHEMBL:CHEMBL123904	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.085239726	DNDI1417346	chembl:CHEMBL1490332	CHEMBL:CHEMBL1490332	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.026519026	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003840807	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.016764901	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.097236428	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	A-77636 HCL	chembl:CHEMBL1256876	CHEMBL:CHEMBL1256876	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.003961647	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.011668371	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	THIOPHANATE METHYL	chembl:CHEMBL487187	THIOPHANATE METHYL	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.055622533	CGP-74514A	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.042073455	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.033401826	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.1084869240406911	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.012454381	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	3.500511415712966	HEMOPRESSIN	chembl:CHEMBL510801	HEMOPRESSIN	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.037639908	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.019687916	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	1.166837138570989	HESPERIDIN	rxcui:5281	HESPERIDIN	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.02804897	BX-795	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	GNF-PF-1549	chembl:CHEMBL227959	CHEMBL:CHEMBL227959	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.4234489615781814	SJ000018309	chembl:CHEMBL591363	CHEMBL:CHEMBL591363	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.032899543	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	GNF-PF-3265	chembl:CHEMBL581868	CHEMBL:CHEMBL581868	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	DTC	9/2/20	NULL	0.8140724222588294	BICUCULLINE	drugbank:DB11562	BICUCULLINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	TCMDC-123641	chembl:CHEMBL532849	CHEMBL:CHEMBL532849	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	CROMOLYN	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.014050755	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.030255068	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004426918	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	1.381780822	NSC-121858	chembl:CHEMBL483838	CHEMBL:CHEMBL483838	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	GNF-PF-2954	chembl:CHEMBL582722	CHEMBL:CHEMBL582722	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.03729238	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	DNDI1318925	chembl:CHEMBL1390716	CHEMBL:CHEMBL1390716	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.050048162	DICLOFENAC SODIUM	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
NPFFR2	hgnc:4525	NPFFR2	DTC	9/2/20	NULL	26.25383561784724	KISSPEPTIN-10	drugbank:DB16210	KISSPEPTIN-10	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001244081	ESTRADIOL VALERATE	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.068907705	DITHIOLETHIONE	chembl:CHEMBL368700	DITHIOLETHIONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.063110182	AZ628	iuphar.ligand:8475	AZ628	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	MELEVODOPA	ncit:C83927	MELEVODOPA	TRUE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.015930725	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.010058941	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	DNDI1417011	chembl:CHEMBL1386434	CHEMBL:CHEMBL1386434	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	SJ000032081	chembl:CHEMBL590184	CHEMBL:CHEMBL590184	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	CID 838877	chembl:CHEMBL405317	CHEMBL:CHEMBL405317	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.3621218705909966	TCMDC-124573	chembl:CHEMBL525826	CHEMBL:CHEMBL525826	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003720782	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIMETHISOQUIN HYDROCHLORIDE	ncit:C72742	DIMETHISOQUIN HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PYRIDABEN	chembl:CHEMBL225963	PYRIDABEN	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.047049885	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	R-N-PROPYLNORAPOMORPHINE	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	2.282942227638891	PALINURIN	chembl:CHEMBL464381	PALINURIN	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	DTC	9/2/20	NULL	3.621218705909965	CASEARINONE B	chembl:CHEMBL459014	CASEARINONE B	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004652461	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.012020987	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	3.500511415712966	OCHROMYCINONE	drugbank:DB15644	OCHROMYCINONE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.076098074	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.4688184931758437	TCMDC-125543	chembl:CHEMBL546170	CHEMBL:CHEMBL546170	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010687497	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1325951293830669	TRANILAST	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.2344092465879218	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.004554399	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.9723642821424906	CRYPTOLEPINE HYDROCHLORIDE	chembl:CHEMBL92129	CRYPTOLEPINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	SKIMMIANINE	chembl:CHEMBL21396	SKIMMIANINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	TRICLABENDAZOLE	rxcui:2118525	TRICLABENDAZOLE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	SB-204070A	iuphar.ligand:256	SB 204070	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	DIFFRACTAIC ACID	chembl:CHEMBL367741	DIFFRACTAIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	SARCOLYSIN	ncit:C61936	SARCOLYSIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.012683012	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1232574442152452	NSC-677438	chembl:CHEMBL118678	CHEMBL:CHEMBL118678	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.01875274	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.4861821410712453	2,3,4,4'-TETRAMETHOXYBIPHENYL	chembl:CHEMBL28250	2,3,4,4'-TETRAMETHOXYBIPHENYL	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.041150213	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.019799273	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	GNF-PF-4803	chembl:CHEMBL585240	CHEMBL:CHEMBL585240	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	DIGITOXIGENIN	drugbank:DB04177	DIGITOXIGENIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	AG-370	chembl:CHEMBL59150	CHEMBL:CHEMBL59150	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.063415062	GUGGULSTERONE	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	LISINOPRIL HYDRATE	chembl:CHEMBL1729579	LISINOPRIL HYDRATE	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	DTC	9/2/20	NULL	0.4054646427466756	CGS-21680	iuphar.ligand:375	CGS 21680	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	TCMDC-124440	chembl:CHEMBL547407	CHEMBL:CHEMBL547407	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	GNF-PF-3543	chembl:CHEMBL598679	CHEMBL:CHEMBL598679	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CYMOXANIL	chembl:CHEMBL59983	CYMOXANIL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	PROSTAGLANDIN A2	iuphar.ligand:6279	PROSTAGLANDIN A2	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.087512785	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.019059046	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	HYMECROMONE METHYL ETHER	chembl:CHEMBL12636	HYMECROMONE METHYL ETHER	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.5738543304447485	(S)-VERAPAMIL	chembl:CHEMBL36148	(S)-VERAPAMIL	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.030176823	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.023482858	CIANIDANOL	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.009430257	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.034888818	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	AMITRIPTYLINOXIDE	ncit:C72698	AMITRIPTYLINOXIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	PHENOXYBENZAMINE	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	OSM-S-85	chembl:CHEMBL1494650	CHEMBL:CHEMBL1494650	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.013411921	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.2853677784548614	GW8510	chembl:CHEMBL1276446	CHEMBL:CHEMBL1276446	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	GNF-PF-3165	chembl:CHEMBL581257	CHEMBL:CHEMBL581257	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006780433	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003559601	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	COCLAURINE	chembl:CHEMBL453291	COCLAURINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	AMARANTH	chembl:CHEMBL1408927	AMARANTH	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.094099769	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV396669	chembl:CHEMBL2028050	CHEMBL:CHEMBL2028050	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	RAC-GONIOTHALAMIN	chembl:CHEMBL1170485	CHEMBL:CHEMBL1170485	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00292359	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001359809	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.8204323630577265	THAPSIGARGIN	ncit:C128634	THAPSIGARGIN	FALSE	FALSE	FALSE
GLRA2	hgnc:4327	GLRA2	DTC	9/2/20	NULL	1.312691780892362	HU-308	ncit:C184881	ONTERNABEZ	FALSE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	1.000146118775133	SR9011	iuphar.ligand:8900	SR9011	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00479785	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.036013492	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.021070494	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.1615620653405984	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV000326	chembl:CHEMBL589723	CHEMBL:CHEMBL589723	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003418468	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.022439176	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.017811286	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.042107194	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	TCMDC-125606	chembl:CHEMBL536166	CHEMBL:CHEMBL536166	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	SJ000170251	chembl:CHEMBL603154	CHEMBL:CHEMBL603154	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.035865896	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	GNF-PF-4057	chembl:CHEMBL598903	CHEMBL:CHEMBL598903	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001835419	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.014916952	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.2263261691193728	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CYCLOASPEPTIDE A	chembl:CHEMBL473074	CYCLOASPEPTIDE A	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.16256245	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	5,7,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL242385	CHEMBL:CHEMBL242385	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.033487035	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.07458476	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006555265	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002669701	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.015516451	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	LANSOPRAZOLE SULFIDE	chembl:CHEMBL899	LANSOPRAZOLE SULFIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	FIPEXIDE HYDROCHLORIDE	chembl:CHEMBL1377408	FIPEXIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.025147352	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	BUNITROLOL	ncit:C72614	BUNITROLOL	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
HIF1AN	hgnc:17113	HIF1AN	DTC	9/2/20	NULL	17.50255707856483	L-3,4-DEHYDROPROLINE	chembl:CHEMBL78920	CHEMBL:CHEMBL78920	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.025814981	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CLOSTEBOL	rxcui:61686	CLOSTEBOL	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.019031414	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.011812749	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.1084869240406911	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.012996948	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.1250182648468916	A-77636 HCL	chembl:CHEMBL1256876	CHEMBL:CHEMBL1256876	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.005741681	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	INGLIFORIB	ncit:C75982	INGLIFORIB	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.3365876361262468	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	EPIRUBICIN HYDROCHLORIDE	rxcui:203213	EPIRUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003313623	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	QUININE ETHYLCARBONATE	chembl:CHEMBL3138665	QUININE ETHYLCARBONATE	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.1591141552596803	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.080164384	DIBUTYLDICHLOROSTANNANE	chembl:CHEMBL1088184	DIBUTYLDICHLOROSTANNANE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.032982206	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	SARCOLYSIN	ncit:C61936	SARCOLYSIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	IPRONIAZID PHOSPHATE	chembl:CHEMBL1256361	IPRONIAZID PHOSPHATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	CLOFIBRIC ACID	ncit:C81531	CLOFIBRIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003390216	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.021370644	DOMIPHEN BROMIDE	rxcui:49255	DOMIPHEN BROMIDE	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.036062961	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.079557078	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005669763	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
SLC9A1	hgnc:11071	SLC9A1	DTC	9/2/20	NULL	52.50767123569449	HOE-694	chembl:CHEMBL62231	CHEMBL:CHEMBL62231	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009084372	HYDRALAZINE HYDROCHLORIDE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.00962384	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	4'-HYDROXYPHENYL-BENZO[D]THIAZOLE	chembl:CHEMBL47875	CHEMBL:CHEMBL47875	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.011474579	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	GNF-PF-3561	chembl:CHEMBL599712	CHEMBL:CHEMBL599712	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.05814803	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	NSC-753574	chembl:CHEMBL2088730	CHEMBL:CHEMBL2088730	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	NSC-753574	chembl:CHEMBL2088730	CHEMBL:CHEMBL2088730	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	FIPEXIDE HYDROCHLORIDE	chembl:CHEMBL1377408	FIPEXIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	TCMDC-124573	chembl:CHEMBL525826	CHEMBL:CHEMBL525826	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	PROADIFEN HYDROCHLORIDE	ncit:C66468	PROADIFEN HYDROCHLORIDE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.3061671792168775	LEUCETTAMINE B	chembl:CHEMBL485053	LEUCETTAMINE B	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.023482858	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.006137659	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	TCMDC-124573	chembl:CHEMBL525826	CHEMBL:CHEMBL525826	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.019889269	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	ALPHA-NAPHTHOFLAVONE	drugbank:DB07453	ALPHA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	NALOXONE BENZOYLHYDRAZONE	iuphar.ligand:1664	NALOXONE BENZOYLHYDRAZONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	HYPEROSIDE	chembl:CHEMBL251254	HYPEROSIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	FLUORANTHENE	chembl:CHEMBL355014	FLUORANTHENE	FALSE	FALSE	FALSE
IDE	hgnc:5381	IDE	DTC	9/2/20	NULL	0.5250767123569451	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	METHYL ANTHRANILATE	rxcui:29742	METHYL ANTHRANILATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006937201	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	THIOGUANOSINE	chembl:CHEMBL283078	THIOGUANOSINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NICORANDIL	rxcui:31748	NICORANDIL	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	LUCIDUMOL A	chembl:CHEMBL1917739	LUCIDUMOL A	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NICORANDIL	rxcui:31748	NICORANDIL	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	ECHINATIN	chembl:CHEMBL141530	ECHINATIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004176557	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005424346	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.045265234	NORADRENALINE	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.020391329	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.077217164	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.004854629	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.012794267	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	NSC-172033	chembl:CHEMBL238624	CHEMBL:CHEMBL238624	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.023171964	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006027051	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
KDM1A	hgnc:29079	KDM1A	DTC	9/2/20	NULL	21.00306849427779	2-[N-(PHTHALIMIDO)]ETHYL CARBAMIMIDOTHIOATE HCL	chembl:CHEMBL2182009	CHEMBL:CHEMBL2182009	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.009935226	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TALIPEXOLE	ncit:C152496	TALIPEXOLE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.015930725	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.003785155	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.027290889	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.2763561643983921	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.2067231151011594	MERSALYL	rxcui:6774	MERSALYL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	(S)-ALAPROCLATE	chembl:CHEMBL251941	(S)-ALAPROCLATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	VINBURNINE	rxcui:57954	VINBURNINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	DEXEFAROXAN	ncit:C77943	DEXEFAROXAN	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.09741683	LAS38096	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	BENZOPHENONE	rxcui:18997	BENZOPHENONE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.028290771	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.044878351	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.042242696	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.010405801	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
PADI2	hgnc:18341	PADI2	DTC	9/2/20	NULL	5.834185692854944	O-F-AMIDINE	iuphar.ligand:8625	O-F-AMIDINE	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.1058622403945453	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	CILNIDIPINE	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.066297565	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.6250913242344582	VEGFRECINE	chembl:CHEMBL2332119	VEGFRECINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	DOMIPHEN BROMIDE	rxcui:49255	DOMIPHEN BROMIDE	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	DTC	9/2/20	NULL	0.062733179	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	CLOFENOXYDE	ncit:C78034	CLOFENOXYDE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.400821918	OUABAIN HYDRATE	chembl:CHEMBL1889436	OUABAIN	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.067897851	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.016429184	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
PPOX	hgnc:9280	PPOX	FDA	10-Apr-24	NULL	17.50255707856483	Givosiran	rxcui:2265712	GIVOSIRAN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.025298806	Lofexidine	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.016690296	Lacosamide	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
HPRT1	hgnc:5157	HPRT1	FDA	10-Apr-24	NULL	1.193356164447602	Mycophenolic Acid	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.3472729579080324	CO-1686	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	0.03591496	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.042516333	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.09753747	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.5903640284436551	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.075768645	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:9547	ncit:C166520	MIZAGLIFLOZIN	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.089501712	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.1894216134043813	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.1835932560688619	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.1166837138570988	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.047518255	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.085796848	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.073540156	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.085796848	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.1715936968486748	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3126	iuphar.ligand:3126	COMPOUND 3 [PMID: 19191557]	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.2375912725597036	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.2273059360852575	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.031254566	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2083637747448194	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:3065	iuphar.ligand:3065	COMPOUND 1 [OVERHAND ET AL., 1997]	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1442518440541057	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.8334550989792776	PD 0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3104	iuphar.ligand:3104	E5700	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.082115757	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3135	iuphar.ligand:3135	1-ALLYL-2-[3-(ISOPROPYLAMINO)PROPOXY]-9H-XANTHEN-9-ONE	FALSE	FALSE	FALSE
PDGFB	hgnc:8800	PDGFB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3571950424196904	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
VEGFB	hgnc:12681	VEGFB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	2.187819634820604	ENDOSTATIN (84-114)-NH2 (JKC367)	drugbank:DB06423	ENDOSTATIN	FALSE	FALSE	TRUE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2042	iuphar.ligand:2042	BOC-ATE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.027855529	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
VEGFC	hgnc:12682	VEGFC	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.458546423213736	ENDOSTATIN (84-114)-NH2 (JKC367)	drugbank:DB06423	ENDOSTATIN	FALSE	FALSE	TRUE
DDR2	hgnc:2731	DDR2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.9546849315580819	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:2026	iuphar.ligand:2026	BIM 23454	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
A2M	hgnc:7	A2M	NCI	14-Sep-17	NULL	0.052718545	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.081597003	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	0.6482428547616605	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.1187956362798518	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2043	iuphar.ligand:2043	DC 23-60	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.08780547	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
AIFM1	hgnc:8768	AIFM1	NCI	14-Sep-17	NULL	0.6035364509849942	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.068458502	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.030688294	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2024	iuphar.ligand:2024	[125I]TYR10-CST14	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.042107194	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
ATP7A	hgnc:869	ATP7A	NCI	14-Sep-17	NULL	0.2651902587661338	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1067229090156392	DONEPEZIL	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2063	iuphar.ligand:2063	[111IN]DOTA-BOC-ATE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.065675636	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.024393808	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10674	iuphar.ligand:10674	NVP‐TNKS656	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.2134458180312784	DDTC	ncit:C432	DITIOCARB	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.038808331	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.042361978	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.9460841664089098	ISOFLAVONE	drugbank:DB12007	ISOFLAVONE	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.05792352	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.032837818	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
BTF3L1	hgnc:1126	BTF3P11	NCI	14-Sep-17	NULL	1.193356164447602	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.042968634	VINORELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.011171845	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10676	iuphar.ligand:10676	AZ1366	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	NCI	14-Sep-17	NULL	0.2625383561784725	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
CAST	hgnc:1515	CAST	NCI	14-Sep-17	NULL	0.6250913242344582	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	NCI	14-Sep-17	NULL	0.2019525816757481	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
CA2	hgnc:1373	CA2	NCI	14-Sep-17	NULL	0.4487835148349957	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
CAST	hgnc:1515	CAST	NCI	14-Sep-17	NULL	0.375054795	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.8468979231563628	NIMUSTINE HYDROCHLORIDE	ncit:C693	NIMUSTINE	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.6482428547616605	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.1119566550867686	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:2639	ncit:C81539	SOBETIROME	FALSE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.2885036881082116	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.3125456621172291	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.025929714	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CUBN	hgnc:2548	CUBN	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
CTSG	hgnc:2532	CTSG	NCI	14-Sep-17	NULL	0.3365876361262467	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:9254	iuphar.ligand:9254	GSK2245035	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.2083637747448194	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.023336743	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.025298806	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.005712634	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	NCI	14-Sep-17	NULL	0.3231241306811969	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.07458476	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
NCBIGENE:3015	hgnc:4741	H2AZ1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5994	iuphar.ligand:5994	JAK3 INHIBITOR IV	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.2333674277141978	AMPRENAVIR	rxcui:228656	AMPRENAVIR	TRUE	FALSE	FALSE
CYP3A7	hgnc:2640	CYP3A7	NCI	14-Sep-17	NULL	0.1704794520639432	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
DCK	hgnc:2704	DCK	NCI	14-Sep-17	NULL	0.4565884455277783	CDA	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
DCN	hgnc:2705	DCN	NCI	14-Sep-17	NULL	0.384671584	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.05309168	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1275785139360852	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
DNTT	hgnc:2983	DNTT	NCI	14-Sep-17	NULL	2.187819634820604	2&APOS;,3&APOS;-DIDEOXYCYTIDINE	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
NCBIGENE:2252	hgnc:3685	FGF7	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:10536	iuphar.ligand:10536	DTRIM24	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.091732479	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	NCI	14-Sep-17	NULL	0.009882867	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.074927706	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.074927706	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
DNTT	hgnc:2983	DNTT	NCI	14-Sep-17	NULL	2.187819634820604	2,3-DIDEOXYCYTIDINE	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
EMP2	hgnc:3334	EMP2	NCI	14-Sep-17	NULL	1.193356164447602	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
EPHA8	hgnc:3391	EPHA8	NCI	14-Sep-17	NULL	2.019525817	PHYTOESTROGEN	ncit:C1194	PHYTOESTROGEN	FALSE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.1201548540862574	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:10275	iuphar.ligand:10275	JT010	FALSE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	NCI	14-Sep-17	NULL	0.6177373086552295	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.138178082	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.1136529680426287	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.036577967	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.596678082	IUPHAR.LIGAND:6306	rxcui:1227	AURANOFIN	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.051604591	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	0.057291513	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.3125456621172291	FADROZOLE	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.384671584	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.192335792	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.7721716358190367	IUPHAR.LIGAND:12525	iuphar.ligand:12525	OPTOBI-1	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1470803115845784	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
GDF15	hgnc:30142	GDF15	NCI	14-Sep-17	NULL	0.3061671792168775	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.4118248724368196	RHGH	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
GHRH	hgnc:4265	GHRH	NCI	14-Sep-17	NULL	1.000146118775133	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.4321619031744403	MNU	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.090452491	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
GPX1	hgnc:4553	GPX1	NCI	14-Sep-17	NULL	4.039051633514962	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.6908904109959803	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:10291	iuphar.ligand:10291	PICO145	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	NCI	14-Sep-17	NULL	0.6471015821300378	GLUTAMINE	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.1315981735230438	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
GPT	hgnc:4552	GPT	NCI	14-Sep-17	NULL	2.386712328895204	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.4339476961627644	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.5303805175322677	GOSERELIN ACETATE	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
GSTA1	hgnc:4626	GSTA1	NCI	14-Sep-17	NULL	0.2763561643983921	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:12463	iuphar.ligand:12463	SCUTELLAREIN	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	NCI	14-Sep-17	NULL	1.093909817410302	DHPG	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.069180068	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1346350544504987	AMB	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1250182648468916	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1262203635473425	ALPHA-METHYL-P-TYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1367387271762877	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.05293112	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	CEFEPIME	rxcui:20481	CEFEPIME	TRUE	FALSE	FALSE
NCBIGENE:502	hgnc:13357	MCOLN2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11860	iuphar.ligand:11860	ESTRADIOL 3-METHYL ETHER	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.058832125	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.031555091	PARACETAMOL	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.017303566	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.019065966	TAXOL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ITGA11	hgnc:6136	ITGA11	NCI	14-Sep-17	NULL	2.692701089009974	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.6789785073581185	GP39	ncit:C1437	RECOMBINANT CD40-LIGAND	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	1.591141552596802	IUPHAR.LIGAND:3048	drugbank:DB04714	ISOPENTENYL PYROPHOSPHATE	FALSE	FALSE	FALSE
INHA	hgnc:6065	INHA	NCI	14-Sep-17	NULL	1.500219178	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	2.386712328895204	IUPHAR.LIGAND:6239	iuphar.ligand:6239	ASPIRIN-TRIGGERED RESOLVIN D1	FALSE	FALSE	FALSE
ITGAX	hgnc:6152	ITGAX	NCI	14-Sep-17	NULL	1.750255707856483	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.1682938180631233	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	1.458546423213736	BUTEIN	ncit:C1028	BUTEIN	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.5834185692854945	ANTI-CD3 ANTIBODY	ncit:C2229	VISILIZUMAB	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	NCI	14-Sep-17	NULL	0.2991890098899971	ANXIOLYTIC	ncit:C28197	ANTIANXIETY AGENT	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.1041818873724097	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	blocker	0.5966780822238011	IUPHAR.LIGAND:6326	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	NCI	14-Sep-17	NULL	0.006365724	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
KRT20	hgnc:20412	KRT20	NCI	14-Sep-17	NULL	0.3500511415712966	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.029665351	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	1.117184494376478	IUPHAR.LIGAND:9238	iuphar.ligand:9238	COMPOUND 27F [PMID: 25625617]	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.2187819634820604	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.1411496538593938	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.3079628811477683	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.3763990769583835	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.2187819634820604	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
LIPC	hgnc:6619	LIPC	NCI	14-Sep-17	NULL	0.3182283105193606	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2160	iuphar.ligand:2160	[PEN5]U-(4-11) (HUMAN)	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.1795134059339982	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.6731752722524935	FGF-1	iuphar.ligand:4923	FGF-1	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.2000292237550266	REBAMIPIDE	ncit:C29852	REBAMIPIDE	FALSE	FALSE	FALSE
NCBIGENE:1013	hgnc:1754	CDH15	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4759	iuphar.ligand:4759	VESAMICOL	FALSE	FALSE	FALSE
MATK	hgnc:6906	MATK	NCI	14-Sep-17	NULL	2.143170254518142	IL-4	iuphar.ligand:4996	IL-4	FALSE	FALSE	FALSE
MBP	hgnc:6925	MBP	NCI	14-Sep-17	NULL	0.3488881809680698	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.096432821	6-THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:3842	iuphar.ligand:3842	[LYS15,ARG16,LEU27]VIP-(1-7)/GRF-(8-27)-NH2	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.08334551	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.054953083	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
MT-CO1	hgnc:7419	MT-CO1	NCI	14-Sep-17	NULL	0.7447896629176524	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1875273972703375	GLN	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.300043836	AMIFOSTINE	rxcui:1545987	AMIFOSTINE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1539	iuphar.ligand:1539	NPY-(22-36) (PIG)	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.1682938180631233	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
NFKBIL1	hgnc:7800	NFKBIL1	NCI	14-Sep-17	NULL	2.692701089009974	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.1493817104856173	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:1522	iuphar.ligand:1522	[ALA31,AIB32]NPY (PIG)	FALSE	FALSE	FALSE
NOTCH1	hgnc:7881	NOTCH1	NCI	14-Sep-17	NULL	0.3125456621172291	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.1785975212098452	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
NPPA	hgnc:7939	NPPA	NCI	14-Sep-17	NULL	0.6908904109959803	AZA	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
NCBIGENE:587	hgnc:977	BCAT2	GuideToPharmacology	2024.1	agonist	0.6731752722524936	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.094244538	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.036847489	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.2430910705356227	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.062509132	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.1458546423213736	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.015516451	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PCBD1	hgnc:8646	PCBD1	NCI	14-Sep-17	NULL	1.500219178	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	NCI	14-Sep-17	NULL	0.071245144	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PAPPA	hgnc:8602	PAPPA	NCI	14-Sep-17	NULL	1.500219178	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	NCI	14-Sep-17	NULL	0.2206204673768676	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
PGD	hgnc:8891	PGD	NCI	14-Sep-17	NULL	5.000730593875666	PENICILLAMINE	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
P2RY2	hgnc:8541	P2RY2	NCI	14-Sep-17	NULL	0.5000730593875666	9-CIS-RETINOIC ACID	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
PAPOLA	hgnc:14981	PAPOLA	NCI	14-Sep-17	NULL	1.779921058837101	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.048618214	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.073437302	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1154014752432845	GONADOTROPINS	ncit:C527	THERAPEUTIC GONADOTROPIN	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1510	iuphar.ligand:1510	NPY-(3-36) (PIG)	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.073437302	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.089756703	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.8078103267029922	THYROID STIMULATING HORMONE	ncit:C887	RECOMBINANT THYROID-STIMULATING HORMONE	FALSE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	0.6731752722524936	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
PLA2G7	hgnc:9040	PLA2G7	NCI	14-Sep-17	NULL	0.7721716358190368	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
PLD1	hgnc:9067	PLD1	NCI	14-Sep-17	NULL	1.166837138570988	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.2822993077187876	RETINOIC ACIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.2778183663264259	MNU	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.049864835	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
RNASEH2A	hgnc:18518	RNASEH2A	NCI	14-Sep-17	NULL	1.193356164447602	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	CIViC	10-Apr-24	NULL	0.1219690388750162	VENETOCLAX	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
S100A10	hgnc:10487	S100A10	NCI	14-Sep-17	NULL	7.501095890813499	GONADOTROPINS	ncit:C527	THERAPEUTIC GONADOTROPIN	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.3125456621172291	9-CIS-RETINOIC ACID	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.1562728310586145	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.1544343271638073	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1615620653405984	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.027855529	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.040390516	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.5385402178019948	ALPHA-ADRENERGIC ANTAGONIST	ncit:C29713	ALPHA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.036718651	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.5385402178019948	SORBITOL	rxcui:9945	SORBITOL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	NCI	14-Sep-17	NULL	0.030572152	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	NCI	14-Sep-17	NULL	0.1735790784651057	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.050764748	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
SMAD7	hgnc:6773	SMAD7	NCI	14-Sep-17	NULL	1.312691780892362	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	1.009762908	GANCICLOVIR	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
SREBF1	hgnc:11289	SREBF1	NCI	14-Sep-17	NULL	10.50153425	NEUROTROPHIC FACTOR	ncit:C2259	RECOMBINANT NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
SP3	hgnc:11208	SP3	NCI	14-Sep-17	NULL	0.7001022831425933	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.6213925590023018	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
BCL2L11	hgnc:994	BCL2L11	CIViC	10-Apr-24	NULL	0.525076712	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
STAT4	hgnc:11365	STAT4	NCI	14-Sep-17	NULL	15.55782851427985	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
STAT5B	hgnc:11367	STAT5B	NCI	14-Sep-17	NULL	1.400204566285186	RHGH	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
ST14	hgnc:11344	ST14	NCI	14-Sep-17	NULL	2.625383561784725	PROTEASE INHIBITOR	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.208916464	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.4118248724368196	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.1207072901969988	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.1842374429322614	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
TFF2	hgnc:11756	TFF2	NCI	14-Sep-17	NULL	0.3977853881492008	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.300043836	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
THBD	hgnc:11784	THBD	NCI	14-Sep-17	NULL	0.760980743	PROSTAGLANDIN E1	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	NCI	14-Sep-17	NULL	0.071780822	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	0.4751825451194073	DESFERRIOXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.079197091	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	2.692701089009974	POTASSIUM OXONATE	ncit:C2415	OTERACIL POTASSIUM	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	OncoKB	23-Jul-20	NULL	1.897867635025102	Avapritinib	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.03505185	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.064111931	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.033338204	STI-571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	OncoKB	23-Jul-20	NULL	0.1999620096341412	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
BRCA1	hgnc:1100	BRCA1	OncoKB	23-Jul-20	NULL	0.1269527834518725	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	OncoKB	23-Jul-20	NULL	0.5509279467829125	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	CIViC	10-Apr-24	NULL	0.09699693	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	OncoKB	23-Jul-20	NULL	0.2739530673166669	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CDK12	hgnc:24224	CDK12	OncoKB	23-Jul-20	NULL	0.1000146118775133	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
U2AF1	hgnc:12453	U2AF1	OncoKB	23-Jul-20	NULL	13.12691780892362	H3B-8800	drugbank:DB14017	H3B-8800	FALSE	FALSE	TRUE
CHRNA3	hgnc:1957	CHRNA3	PharmGKB	4/5/24	NULL	0.1767935058440892	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.3387591692625452	indinavir	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.1065064325267637	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
STMN1	hgnc:6510	STMN1	PharmGKB	4/5/24	NULL	1.750255707856483	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.8751278539282416	nabumetone	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
APOC3	hgnc:610	APOC3	PharmGKB	4/5/24	NULL	0.1875273972703375	protease inhibitors	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
PALB2	hgnc:26144	PALB2	CIViC	10-Apr-24	NULL	0.2983390411119005	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.093596562	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	PharmGKB	4/5/24	NULL	0.3947945205691315	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.067059606	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	0.057700738	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.092606122	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
LRMDA	hgnc:23405	LRMDA	PharmGKB	4/5/24	NULL	1.615620653405984	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.076934317	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.2430910705356226	sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
SLCO1A2	hgnc:10956	SLCO1A2	PharmGKB	4/5/24	NULL	0.1346350544504987	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.025588534	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.009349657	fosphenytoin	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.010058941	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	PharmGKB	4/5/24	NULL	0.048327355	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
EWSR1	hgnc:3508	EWSR1	CIViC	10-Apr-24	NULL	0.2263261691193728	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.065634589	topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.096521454	felodipine	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	1.050153425	sitamaquine	ncit:C73010	SITAMAQUINE	FALSE	FALSE	FALSE
SLC14A2	hgnc:10919	SLC14A2	PharmGKB	4/5/24	NULL	0.9376369863516874	nifedipine	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.041672755	nifedipine	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.009653033	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
TGFA	hgnc:11765	TGFA	PharmGKB	4/5/24	NULL	0.6563458904461813	panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.052090944	amifampridine	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.010199625	curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.017260904	amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.022439176	indinavir	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.013199515	felodipine	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.081597003	probenecid	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	1.930429089547592	deferasirox	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
ATIC	hgnc:794	ATIC	PharmGKB	4/5/24	NULL	1.680245479542224	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
FOLR3	hgnc:3795	FOLR3	PharmGKB	4/5/24	NULL	0.84012274	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.1346350544504987	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
EXO1	hgnc:3511	EXO1	PharmGKB	4/5/24	NULL	1.400204566285186	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
IGF2BP2	hgnc:28867	IGF2BP2	PharmGKB	4/5/24	NULL	0.7292732116068681	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.039598545	perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	0.1207072901969988	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	0.076098074	WHI-P154	iuphar.ligand:5993	JAK3 INHIBITOR II	FALSE	FALSE	TRUE
APOBEC3B	hgnc:17352	APOBEC3B	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ERCC1	hgnc:3433	ERCC1	CIViC	10-Apr-24	NULL	0.047049885	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NUP62	hgnc:8066	NUP62	PharmGKB	4/5/24	NULL	0.5147810905460245	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
HBEGF	hgnc:3059	HBEGF	PharmGKB	4/5/24	NULL	0.084689792	panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	1.750255707856483	bilirubin	iuphar.ligand:4577	BILIRUBIN	FALSE	FALSE	FALSE
NAGS	hgnc:17996	NAGS	PharmGKB	4/5/24	NULL	4.375639269641208	glycerol phenylbutyrate	rxcui:1368451	GLYCEROL PHENYLBUTYRATE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	CIViC	10-Apr-24	NULL	0.7059854956059763	AVELUMAB	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
NFIB	hgnc:7785	NFIB	PharmGKB	4/5/24	NULL	2.187819634820604	paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
PLA2G4A	hgnc:9035	PLA2G4A	PharmGKB	4/5/24	NULL	0.1682938180631234	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.1620607136904151	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.1909369863116163	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.2125816649218401	fosphenytoin	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.6364566210387212	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.022305723	ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	PharmGKB	4/5/24	NULL	0.1426838892274307	ropeginterferon alfa-2b	rxcui:2587059	ROPEGINTERFERON ALFA-2B	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.030202859	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.078252863	ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.019159887	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.046303061	tegafur	rxcui:10995	URACIL	TRUE	FALSE	TRUE
DHFR	hgnc:2861	DHFR	PharmGKB	4/5/24	NULL	0.037721028	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.007717177	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TLR4	hgnc:11850	TLR4	PharmGKB	4/5/24	NULL	0.061150238	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.05553429	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.1620607136904151	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.032412143	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
MRPL47	hgnc:16652	MRPL47	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
RAC2	hgnc:9802	RAC2	PharmGKB	4/5/24	NULL	0.3241214273808302	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.092606122	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.052560231	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.008854582	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.015325238	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ECHS1	hgnc:3151	ECHS1	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.00655895	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
PACSIN2	hgnc:8571	PACSIN2	PharmGKB	4/5/24	NULL	2.763561643983921	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
FTO	hgnc:24678	FTO	PharmGKB	4/5/24	NULL	0.5181678082469852	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
RAC1	hgnc:9801	RAC1	PharmGKB	4/5/24	NULL	0.3070624048871023	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
ITPA	hgnc:6176	ITPA	PharmGKB	4/5/24	NULL	1.312691780892362	protease inhibitors	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.048935388	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
DRD1	hgnc:3020	DRD1	PharmGKB	4/5/24	NULL	0.032173818	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1325951293830669	oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1666910197958555	medroxyprogesterone	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
CYP24A1	hgnc:2602	CYP24A1	PharmGKB	4/5/24	NULL	2.187819634820604	deferasirox	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.099446347	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	PharmGKB	4/5/24	NULL	0.034727296	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.1172046232939609	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
MSH3	hgnc:7326	MSH3	PharmGKB	4/5/24	NULL	0.7032277397637656	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.052090944	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
AGXT	hgnc:341	AGXT	PharmGKB	4/5/24	NULL	26.25383561784724	lumasiran	rxcui:2467140	LUMASIRAN	TRUE	FALSE	FALSE
EPHA6	hgnc:19296	EPHA6	PharmGKB	4/5/24	NULL	0.5834185692854945	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	2.651902587661338	Vitamin K1	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	CIViC	10-Apr-24	NULL	0.021554873	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
RBMS3	hgnc:13427	RBMS3	PharmGKB	4/5/24	NULL	0.9376369863516874	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ITGA2B	hgnc:6138	ITGA2B	PharmGKB	4/5/24	NULL	3.646366058	abciximab	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	0.1311052964686504	rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
NOC3L	hgnc:24034	NOC3L	PharmGKB	4/5/24	NULL	3.000438356	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.080550887	dofetilide	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
TGFBR3	hgnc:11774	TGFBR3	PharmGKB	4/5/24	NULL	0.2524407270946851	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
TGFBR2	hgnc:11773	TGFBR2	PharmGKB	4/5/24	NULL	0.8334550989792777	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SCNN1G	hgnc:10602	SCNN1G	PharmGKB	4/5/24	NULL	1.372749574789398	amiloride	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.2631963470460877	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
ATP10A	hgnc:13542	ATP10A	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	0.047049885	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.039449791	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.046528729	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.084214389	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
MTRR	hgnc:7473	MTRR	PharmGKB	4/5/24	NULL	0.5676504998453459	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
CYP2C18	hgnc:2620	CYP2C18	PharmGKB	4/5/24	NULL	1.060761035064535	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
F3	hgnc:3541	F3	PharmGKB	4/5/24	NULL	0.1400204566285186	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CXCL10	hgnc:10637	CXCL10	PharmGKB	4/5/24	NULL	0.1930429089547591	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
TAAR6	hgnc:20978	TAAR6	PharmGKB	4/5/24	NULL	2.763561643983921	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.1221108633388244	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
ACSS3	hgnc:24723	ACSS3	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.502465753	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
CYB5R2	hgnc:24376	CYB5R2	PharmGKB	4/5/24	NULL	0.9546849315580819	primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.3977853881492007	4-hydroxyestradiol	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
FASTKD3	hgnc:28758	FASTKD3	PharmGKB	4/5/24	NULL	2.917092846427472	tegafur	rxcui:10995	URACIL	TRUE	FALSE	TRUE
DDO	hgnc:2727	DDO	PharmGKB	4/5/24	NULL	0.7001022831425933	topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	CIViC	10-Apr-24	NULL	0.1798207919030633	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
IL2RA	hgnc:6008	IL2RA	PharmGKB	4/5/24	NULL	0.8579684842433742	denileukin diftitox	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	PharmGKB	4/5/24	NULL	0.021541609	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
CELF4	hgnc:14015	CELF4	PharmGKB	4/5/24	NULL	5.000730593875666	iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.7212592202705288	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.1660584163051692	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
RPP30	hgnc:17688	RPP30	PharmGKB	4/5/24	NULL	0.6731752722524936	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NRG3	hgnc:7999	NRG3	PharmGKB	4/5/24	NULL	0.5250767123569451	panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.044878351	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
PIN1	hgnc:8988	PIN1	PharmGKB	4/5/24	NULL	0.075768645	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
HLA-DPA1	hgnc:4938	HLA-DPA1	PharmGKB	4/5/24	NULL	3.281729452230906	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ETS2	hgnc:3489	ETS2	PharmGKB	4/5/24	NULL	0.1944728564284981	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	0.084012274	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	PharmGKB	4/5/24	NULL	0.2055094764606438	Glucarpidase	rxcui:1242127	GLUCARPIDASE	TRUE	FALSE	FALSE
PSORS1C1	hgnc:17202	PSORS1C1	PharmGKB	4/5/24	NULL	0.4286340509036285	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	PharmGKB	4/5/24	NULL	0.1530835896084387	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
NT5C2	hgnc:8022	NT5C2	PharmGKB	4/5/24	NULL	1.250182648468916	didanosine	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.034727296	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABL2	hgnc:77	ABL2	CIViC	10-Apr-24	NULL	0.013463505	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CXCR4	hgnc:2561	CXCR4	PharmGKB	4/5/24	NULL	0.105015342	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CNTF	hgnc:2169	CNTF	PharmGKB	4/5/24	NULL	5.000730593875666	iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	PharmGKB	4/5/24	NULL	0.020836377	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCG8	hgnc:13887	ABCG8	PharmGKB	4/5/24	NULL	2.100306849	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
SSTR5	hgnc:11334	SSTR5	PharmGKB	4/5/24	NULL	0.8751278539282418	lutetium (177Lu) oxodotreotide	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
PML	hgnc:9113	PML	CIViC	10-Apr-24	NULL	1.458546423213736	TAMIBAROTENE	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	PharmGKB	4/5/24	NULL	0.057073556	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
MTRR	hgnc:7473	MTRR	PharmGKB	4/5/24	NULL	1.750255707856483	tegafur	rxcui:10995	URACIL	TRUE	FALSE	TRUE
SHMT1	hgnc:10850	SHMT1	PharmGKB	4/5/24	NULL	0.8751278539282418	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CACNA1A	hgnc:1388	CACNA1A	PharmGKB	4/5/24	NULL	0.1346350544504987	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	PharmGKB	4/5/24	NULL	0.025563618	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	PharmGKB	4/5/24	NULL	1.078924751	larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
ASTN2	hgnc:17021	ASTN2	PharmGKB	4/5/24	NULL	1.750255707856483	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	2.500365296937833	omacetaxine	rxcui:1546446	OMACETAXINE	TRUE	FALSE	FALSE
SF3B1	hgnc:10768	SF3B1	CIViC	10-Apr-24	NULL	0.3977853881492008	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.5834185692854944	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
SLC15A2	hgnc:10921	SLC15A2	PharmGKB	4/5/24	NULL	0.2447910080918158	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	PharmGKB	4/5/24	NULL	3.889457128569962	afutuzumab	rxcui:974779	OBINUTUZUMAB	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.023744802	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
NME2	hgnc:7850	NME2	PharmGKB	4/5/24	NULL	0.7778914257139926	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.1773907812016706	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
ITGAV	hgnc:6150	ITGAV	TALC	12-May-16	NULL	4.039051633514961	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
NUDT15	hgnc:23063	NUDT15	CIViC	10-Apr-24	NULL	0.6908904109959803	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.016083624	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
KIF11	hgnc:6388	KIF11	TALC	12-May-16	inhibitor	3.281729452230906	MK0731	ncit:C49174	MK0731	FALSE	FALSE	TRUE
UNIPROT:P06213	hgnc:6091	INSR	TdgClinicalTrial	Jan-14	NULL	0.042459033	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.7955707762984014	ALEGLITAZAR	ncit:C72687	ALEGLITAZAR	FALSE	FALSE	FALSE
UNIPROT:O43614	hgnc:4849	HCRTR2	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	ALMOREXANT	ncit:C87423	ALMOREXANT	FALSE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	ALMOTRIPTAN	rxcui:279645	ALMOTRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1305078821102597	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.2059124362184098	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.108711535	AM-101	chembl:CHEMBL2364609	ESKETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q14957	hgnc:4587	GRIN2C	TdgClinicalTrial	Jan-14	NULL	0.1209854175937661	AM-101	chembl:CHEMBL2364609	ESKETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.1295419520617463	MEPIVACAINE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14778	hgnc:5993	IL1R1	TdgClinicalTrial	Jan-14	NULL	3.141484604	ANAKINRA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	ATAMESTANE	ncit:C1224	ATAMESTANE	FALSE	FALSE	FALSE
UNIPROT:Q96NY8	hgnc:19688	NECTIN4	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	ASG-22ME	chembl:CHEMBL3301589	ENFORTUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.06525008	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	AUS-131	chembl:CHEMBL198877	AUS-131	FALSE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TdgClinicalTrial	Jan-14	NULL	0.7425327245451747	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
UNIPROT:Q6P5Z2	hgnc:17999	PKN3	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	ATU027	ncit:C84847	ANTI-PKN3 SIRNA ATU027	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	CIViC	10-Apr-24	NULL	1.272913242077442	GSK126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	AVE-1625	drugbank:DB05750	AVE-1625	FALSE	FALSE	FALSE
UNIPROT:O43557	hgnc:11930	TNFSF14	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	BAMINERCEPT	ncit:C96762	BAMINERCEPT ALFA	FALSE	FALSE	FALSE
UNIPROT:Q9Y275	hgnc:11929	TNFSF13B	TdgClinicalTrial	Jan-14	NULL	32.81729452230906	BELIMUMAB	rxcui:1092437	BELIMUMAB	TRUE	TRUE	TRUE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.1715936968486748	BUPROPION	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	0.2812910959055062	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.037345428	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.801643836	CORT 108297	chembl:CHEMBL271220	CORT 108297	FALSE	FALSE	FALSE
UNIPROT:P13569	hgnc:1884	CFTR	TdgClinicalTrial	Jan-14	NULL	1.591141552596802	CROFELEMER	rxcui:1364449	CROFELEMER	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.025390557	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:Q07973	hgnc:2602	CYP24A1	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	CTA018	drugbank:DB05024	CTA018	FALSE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	0.046549354	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	1.032937794800547	ETONOGESTREL	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
UNIPROT:Q9GZT9	hgnc:1232	EGLN1	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	FG-4592	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.050174554	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.027177884	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	CIViC	10-Apr-24	NULL	0.061992528	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P04141	hgnc:2434	CSF2	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	KB002	drugbank:DB05194	KB002	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	LEVOMILNACIPRAN	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
UNIPROT:P12931	hgnc:11283	SRC	TdgClinicalTrial	Jan-14	NULL	0.1143957978991165	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	MEM 1414	drugbank:DB05888	MEM 1414	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	MEM3454	chembl:CHEMBL5095032	RG3487	FALSE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.037666909	MILATAXEL	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
UNIPROT:Q02763	hgnc:11724	TEK	TdgClinicalTrial	Jan-14	NULL	0.9845188356692718	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
UNIPROT:P14324	hgnc:3631	FDPS	TdgClinicalTrial	Jan-14	NULL	2.333674277141977	MINODRONATE	drugbank:DB06548	MINODRONIC ACID	FALSE	FALSE	FALSE
UNIPROT:Q13258	hgnc:9591	PTGDR	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
UNIPROT:Q8TEX9	hgnc:19426	IPO4	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
SMARCA4	hgnc:11100	SMARCA4	CIViC	10-Apr-24	NULL	0.364636606	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	3.850562557284263	PLERIXAFOR	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.4518732464345482	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.1875273972703374	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
UNIPROT:P07949	hgnc:9967	RET	TdgClinicalTrial	Jan-14	NULL	0.2778183663264259	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.1852122442176172	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.078252863	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1591141552596802	NAPROXCINOD	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
UNIPROT:P33402	hgnc:4684	GUCY1A2	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	NAPROXCINOD	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.546954909	NI-0401	chembl:CHEMBL1743020	FORALUMAB	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.1262203635473425	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.212152207	OXYMORPHONE	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.07631929	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	1.166837138570988	PALONOSETRON	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.072125922	PAGOCLONE	ncit:C74529	PAGOCLONE	FALSE	FALSE	FALSE
UNIPROT:P00813	hgnc:186	ADA	TdgClinicalTrial	Jan-14	NULL	3.043922970185188	PENTOSTATIN	rxcui:8011	PENTOSTATIN	TRUE	FALSE	TRUE
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.7778914257139926	PH-797804	drugbank:DB07941	PH-797804	FALSE	FALSE	FALSE
UNIPROT:P25092	hgnc:4688	GUCY2C	TdgClinicalTrial	Jan-14	NULL	19.69037671338543	PLECANATIDE	rxcui:1873752	PLECANATIDE	TRUE	FALSE	FALSE
UNIPROT:O00555	hgnc:1388	CACNA1A	TdgClinicalTrial	Jan-14	NULL	0.4039051633514961	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.8008364246019593	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.072125922	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	SB-681323	ncit:C96531	DILMAPIMOD	FALSE	FALSE	FALSE
UNIPROT:P50750	hgnc:1780	CDK9	TdgClinicalTrial	Jan-14	NULL	0.4167275494896389	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	2.128689374420047	TOZADENANT	ncit:C152704	TOZADENANT	FALSE	FALSE	FALSE
UNIPROT:P07949	hgnc:9967	RET	TdgClinicalTrial	Jan-14	NULL	0.3968833804663227	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.3571950424196904	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.1848861663228679	MTOR KINASE INHIBITOR AZD8055	ncit:C78856	MTOR KINASE INHIBITOR AZD8055	FALSE	FALSE	TRUE
UNIPROT:P00750	hgnc:9051	PLAT	TdgClinicalTrial	Jan-14	NULL	3.182283105193605	TRANEXAMIC ACID	rxcui:10691	TRANEXAMIC ACID	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	TOLVAPTAN	rxcui:358257	TOLVAPTAN	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.026045472	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	TLN-4601	ncit:C62508	DIAZEPINOMICIN	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	1.721562991334245	ULIPRISTAL	rxcui:1005920	ULIPRISTAL ACETATE	TRUE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TdgClinicalTrial	Jan-14	NULL	0.1495945049449985	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
UNIPROT:P16422	hgnc:11529	EPCAM	TdgClinicalTrial	Jan-14	NULL	4.200613699	VB4-845	ncit:C61307	OPORTUZUMAB MONATOX	FALSE	FALSE	FALSE
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	VOLOCIXIMAB	ncit:C48426	VOLOCIXIMAB	FALSE	FALSE	TRUE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.8514757497680189	BIIB014	ncit:C152892	VIPADENANT	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.2991890098899972	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
UNIPROT:P32238	hgnc:1570	CCKAR	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	CERULETIDE	ncit:C65309	CERULETIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.1270346884734544	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.066465407	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
CCNE2	hgnc:1590	CCNE2	CIViC	10-Apr-24	NULL	1.071585127259071	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1346350544504987	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.068191781	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.064824285	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q9UI33	hgnc:10583	SCN11A	TdgClinicalTrial	Jan-14	NULL	0.130291988	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.076934317	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	DEMECARIUM BROMIDE	rxcui:22482	DEMECARIUM BROMIDE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.133607306	DIFLORASONE	rxcui:23033	DIFLORASONE DIACETATE	TRUE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	0.5527123287967842	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.085239726	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.020465128	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.060984519	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.063300387	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	CIViC	10-Apr-24	NULL	0.054355767	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.064111931	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.061737415	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.064944553	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.021846337	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TdgClinicalTrial	Jan-14	NULL	0.8468979231563629	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.2047082699247349	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.2536602475154323	LISDEXAMFETAMINE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.006669123	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.086551106	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.059085902	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.093763699	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.067839369	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
UNIPROT:P04054	hgnc:9030	PLA2G1B	TdgClinicalTrial	Jan-14	NULL	0.1553481397505754	NIFLUMIC ACID	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	CIViC	10-Apr-24	NULL	0.1193356164447602	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.09814518	NORGESTIMATE	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
UNIPROT:P20273	hgnc:1643	CD22	TdgClinicalTrial	Jan-14	NULL	8.751278539282417	OSPA LIPOPROTEIN	rxcui:54214	OSPA PROTEIN	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.837888371	OXYPHENONIUM	rxcui:7818	OXYPHENONIUM	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.064347636	PERGOLIDE	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	0.5321723436050118	TRANYLCYPROMINE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.4605936073306534	TRIDIHEXETHYL	rxcui:38617	TRIDIHEXETHYL	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.7160136986685613	TIAPROFENIC ACID	rxcui:38253	TIAPROFENIC ACID	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1556551518844698	ZUCLOPENTHIXOL	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
SMAD4	hgnc:6770	SMAD4	CIViC	10-Apr-24	NULL	0.112919723	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
UNIPROT:Q8N0U8	hgnc:21492	VKORC1L1	TdgClinicalTrial	Jan-14	NULL	3.182283105193606	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.062608511	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.9376369863516875	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1562728310586145	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TEND	1-Aug-11	NULL	1.591141552596803	DEGARELIX	rxcui:475230	DEGARELIX	TRUE	FALSE	FALSE
CX3CL1	hgnc:10647	CX3CL1	CIViC	10-Apr-24	NULL	0.8334550989792776	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.3006164383722967	DIFLUPREDNATE	rxcui:23043	DIFLUPREDNATE	TRUE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TEND	1-Aug-11	NULL	0.5527123287967842	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TEND	1-Aug-11	NULL	0.040275444	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.175610941	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.086694009	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.083522277	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	CIViC	10-Apr-24	NULL	0.406619897	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.2386712328895204	FLECAINIDE	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
UNIPROT:O43451	hgnc:7043	MGAM	TEND	1-Aug-11	NULL	3.182283105193605	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
UNIPROT:Q9UHC9	hgnc:7898	NPC1L1	TEND	1-Aug-11	NULL	26.25383561784724	EZETIMIBE	rxcui:341248	EZETIMIBE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.078545507	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
UNIPROT:P49286	hgnc:7464	MTNR1B	TEND	1-Aug-11	NULL	1.086365611772989	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TEND	1-Aug-11	NULL	0.2344092465879218	ISOTRETINOIN	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	1.221108633388244	METHOHEXITAL	rxcui:6847	METHOHEXITAL	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.032003863	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.596678082	MEXILETINE	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
NF2	hgnc:7773	NF2	CIViC	10-Apr-24	NULL	0.030176823	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P28074	hgnc:9542	PSMB5	TEND	1-Aug-11	NULL	0.4273880216858854	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1305078821102597	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.2059124362184098	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.075732218	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TEND	1-Aug-11	NULL	4.039051633514961	NITROPRUSSIDE	rxcui:7476	NITROPRUSSIDE	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TEND	1-Aug-11	NULL	0.6213925590023018	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.07767407	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.076690854	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.073885091	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.091796628	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DoCM	10-Apr-24	NULL	1.346350544504987	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.083744292	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.1166837138570989	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1221108633388244	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	1.071585127259071	YSIL6	drugbank:DB05017	YSIL6	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	KTE-C19 CAR	ncit:C120309	AXICABTAGENE CILOLEUCEL	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.00731101	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CHEK2	hgnc:16627	CHEK2	CIViC	10-Apr-24	NULL	0.1754935535952356	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
MAP KINASE P38	hgnc:6874	MAPK12	TTD	2020.06.01	NULL	0.6482428547616604	ARRY-797	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
ANGIOPOIETIN-RELATED PROTEIN 3	hgnc:491	ANGPTL3	TTD	2020.06.01	NULL	26.25383561784724	AKCEA-ANGPTL3-LRX	chembl:CHEMBL4298197	VUPANORSEN	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.050488145	AZD8186	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.4773424657790409	BLZ-945	drugbank:DB16838	BLZ-945	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-RAF	hgnc:9829	RAF1	TTD	2020.06.01	NULL	0.6731752722524935	GDC-5573	iuphar.ligand:11544	BELVARAFENIB	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	3.088686543276147	E7046	ncit:C129689	PALUPIPRANT	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.3424413341458336	Dalantercept	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	1.312691780892362	HDM201	ncit:C116325	SIREMADLIN	FALSE	FALSE	FALSE
ATM SERINE/THREONINE KINASE	hgnc:795	ATM	TTD	2020.06.01	NULL	0.7192831676122533	M3541	ncit:C138076	ATM INHIBITOR M 3541	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	0.577007376	OTX-015	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
METHIONINE AMINOPEPTIDASE 2	hgnc:16672	METAP2	TTD	2020.06.01	NULL	6.563458904461812	SDX-7320	ncit:C128030	EVEXOMOSTAT	FALSE	FALSE	FALSE
CELL DIFFERENTIATION	hgnc:2505	CTLA4	TTD	2020.06.01	NULL	1.750255707856483	FF-10501-01	drugbank:DB17554	FF-10501-01	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	DoCM	10-Apr-24	NULL	0.084214389	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	1.105424657593568	Debio 1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
HEPATITIS A VIRUS CELLULAR RECEPTOR 2	hgnc:18437	HAVCR2	TTD	2020.06.01	NULL	17.50255707856483	MBG453	ncit:C124850	SABATOLIMAB	FALSE	FALSE	FALSE
CERAMIDE GLUCOSYLTRANSFERASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	5.250767123569449	Venglustat	ncit:C152852	VENGLUSTAT	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	Inebilizumab	rxcui:2373950	INEBILIZUMAB-CDON	TRUE	FALSE	FALSE
ACTIVIN RECEPTOR TYPE IIA	hgnc:173	ACVR2A	TTD	2020.06.01	NULL	13.12691780892362	BYM338	ncit:C116852	BIMAGRUMAB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.015477574	Etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
IL-1 RECEPTOR-LIKE 2	hgnc:5999	IL1RL2	TTD	2020.06.01	NULL	8.751278539282415	BI655130	iuphar.ligand:12169	SPESOLIMAB	FALSE	FALSE	FALSE
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	0.5081387538938177	PF-06700841	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	1.750255707856483	Setipiprant	ncit:C152348	SETIPIPRANT	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.041508041	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
GLUCAGON	hgnc:4191	GCG	TTD	2020.06.01	NULL	0.6731752722524935	SAR425899	chembl:CHEMBL3545269	SAR425899	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.9546849315580818	FPA-008	ncit:C123831	CABIRALIZUMAB	FALSE	FALSE	FALSE
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.9546849315580818	FPA-008	ncit:C123831	CABIRALIZUMAB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.059532507	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.4605936073306534	Dacomitinib	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.3043922970185188	PF-07284892	ncit:C178469	SHP2 INHIBITOR PF-07284892	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	0.750109589	VVP-808	chembl:CHEMBL19	METHAZOLAMIDE	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.2333674277141978	Volasertib	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
ESTROGEN-RELATED RECEPTOR-ALPHA	hgnc:3471	ESRRA	TTD	2020.06.01	NULL	1.750255707856483	Rimexolone	rxcui:55681	RIMEXOLONE	TRUE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.5834185692854944	ADL-5859	iuphar.ligand:9004	ADL5859	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.037149902	Leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.013860972	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
MEMBRANE GLYCOPROTEIN OX2	hgnc:7203	CD200	TTD	2020.06.01	NULL	157.5230137070835	ALXN6000	ncit:C77891	SAMALIZUMAB	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	1.064344687210023	XL418	drugbank:DB05204	XL418	FALSE	FALSE	FALSE
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	4.200613699	VB4-845	ncit:C61307	OPORTUZUMAB MONATOX	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.8078103267029924	Dichlorphenamide	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.7395446652914718	BRL-52656	chembl:CHEMBL433508	CHEMBL:CHEMBL433508	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	1.500219178	Insulin, porcine	rxcui:221109	INSULIN, REGULAR, PORK	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Trimeprazine	rxcui:10825	TRIMEPRAZINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1570910134201779	LY3214996	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	0.2282942227638891	CYTISINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	1.193356164447602	Arofylline	ncit:C74223	AROFYLLINE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR BETA-2	hgnc:4082	GABRB2	TTD	2020.06.01	NULL	0.1526385791735305	THIOCOLCHICOSIDE	rxcui:38085	THIOCOLCHICOSIDE	FALSE	FALSE	FALSE
FOLATE RECEPTOR	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	0.364636606	Folic Acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	PF-04217903	drugbank:DB12848	PF-04217903	FALSE	FALSE	TRUE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.4468737977505915	CYTISINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.024991752	Sapanisertib	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
GASTRIC TRIACYLGLYCEROL LIPASE	hgnc:6622	LIPF	TTD	2020.06.01	NULL	11.66837138570988	Cetilistat	ncit:C77404	CETILISTAT	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	2.100306849	Nicaraven	ncit:C76580	NICARAVEN	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.1017590527823536	AEE-788	drugbank:DB12558	AEE-788	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.5303805175322676	MPI-0479605	iuphar.ligand:9399	MPI-0479605	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	0.1579178082276526	BMS-582664	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.6482428547616604	DOV 21947	chembl:CHEMBL1818442	AMITIFADINE HYDROCHLORIDE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.046518424	Primidone	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.8607814956671229	Dydrogesterone	rxcui:3706	DYDROGESTERONE	TRUE	FALSE	FALSE
CALCINEURIN	hgnc:9314	PPP3CA	TTD	2020.06.01	NULL	6.563458904461812	Voclosporin	rxcui:2475166	VOCLOSPORIN	TRUE	FALSE	FALSE
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	6.563458904461812	SB-743921	drugbank:DB05546	SB-743921	FALSE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.068191781	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
AMIDOPHOSPHORIBOSYLTRANSFERASE	hgnc:9238	PPAT	TTD	2020.06.01	NULL	0.7778914257139925	Mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.8178764989983567	Pemigatinib	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
CARDIAC MYOSIN	hgnc:7551	MYBPC3	TTD	2020.06.01	NULL	6.563458904461812	Omecamtiv mecarbil	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.08178765	Lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
GUANYLATE CYCLASE SOLUBLE BETA-1	hgnc:4687	GUCY1B1	TTD	2020.06.01	NULL	1.544343271638073	Cinaciguat	ncit:C87280	CINACIGUAT	FALSE	FALSE	FALSE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	Palonosetron	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.2573905452730122	Tridihexethyl	rxcui:38617	TRIDIHEXETHYL	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.4773424657790409	FENBUFEN	rxcui:24830	FENBUFEN	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.4907258993990139	ODM-203	drugbank:DB16843	ODM-203	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA-2/DELTA-1	hgnc:1399	CACNA2D1	TTD	2020.06.01	NULL	0.1562728310586145	Diltiazem	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	0.4039051633514962	Reserpine	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M2	hgnc:1951	CHRM2	TTD	2020.06.01	NULL	0.1151484018326633	Methylscopolamine	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
PROLYL ENDOPEPTIDASE	hgnc:9358	PREP	TTD	2020.06.01	NULL	17.50255707856483	ALV-003	chembl:CHEMBL3137344	LATIGLUTENASE	FALSE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	2.187819634820604	AS-1402	chembl:CHEMBL2108341	SONTUZUMAB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.305277158	ABT-737	drugbank:DB17023	ABT-737	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	1.419126249613364	GW 597599	drugbank:DB05418	GW 597599	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.116943588	MK-0773	drugbank:DB16244	MK-0773	FALSE	FALSE	FALSE
CREB-BINDING PROTEIN	hgnc:2348	CREBBP	TTD	2020.06.01	NULL	2.386712328895204	PRI-724	drugbank:DB15034	PRI-724	FALSE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	2.386712328895204	Maltose	rxcui:1311261	MALTOSE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	0.4688184931758437	Obatoclax	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	0.1172046232939609	Obatoclax	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.5834185692854944	TOFIMILAST	ncit:C76891	TOFIMILAST	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	4.039051633514961	Tbo-Filgrastim	rxcui:1433764	TBO-FILGRASTIM	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.034567262	Carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.1154014752432845	IPI-145	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	1.346350544504987	CG-100649	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	2.493675356344019	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.3387591692625452	LIDOFLAZINE	rxcui:6390	LIDOFLAZINE	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.069180068	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
CTP SYNTHASE	hgnc:2519	CTPS1	TTD	2020.06.01	NULL	2.763561643983921	Cyclopentenylcytosine	ncit:C1359	CYCLOPENTENYL CYTOSINE	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.06525008	Prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	1.346350544504987	NXN-188	drugbank:DB06096	NXN-188	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	2.019525817	LY-2828360	iuphar.ligand:12751	LY2828360	FALSE	FALSE	FALSE
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	2.187819634820604	4SC-205	ncit:C90557	EG5 KINESIN-RELATED MOTOR PROTEIN INHIBITOR 4SC-205	FALSE	FALSE	FALSE
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	21.00306849427779	Mitemcinal fumarate	ncit:C170187	MITEMCINAL FUMARATE	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	1.693795846312725	SMP-986	chembl:CHEMBL3545165	AFACIFENACIN	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.2108741816694558	LY294002	ncit:C148229	PI3K/BET INHIBITOR LY294002	FALSE	FALSE	TRUE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	C-CAR088	ncit:C170747	AUTOLOGOUS ANTI-BCMA-CAR-4-1BB-CD3ZETA-EXPRESSING T-CELLS C-CAR088	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.035982643	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	0.8334550989792776	Ardeparin	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR ALPHA	hgnc:6008	IL2RA	TTD	2020.06.01	NULL	1.715936968486748	Basiliximab	rxcui:196102	BASILIXIMAB	TRUE	TRUE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.6250913242344582	TOFIMILAST	ncit:C76891	TOFIMILAST	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	AZD5312	ncit:C116326	ANDROGEN RECEPTOR ANTISENSE OLIGONUCLEOTIDE AZD5312	FALSE	FALSE	FALSE
5-HT 1F RECEPTOR	hgnc:5292	HTR1F	TTD	2020.06.01	NULL	1.591141552596802	LY-334370	iuphar.ligand:151	[3H]LY334370	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.1363835616511545	Meclofenamate Sodium	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
PYRUVATE KINASE M2	hgnc:9021	PKM	TTD	2020.06.01	NULL	1.458546423213736	CAP-232	ncit:C67087	PYRUVATE KINASE INHIBITOR TLN-232	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.4167275494896388	Varlitinib	ncit:C62530	VARLITINIB	FALSE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	2.917092846427472	Ipamorelin	ncit:C81120	IPAMORELIN	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.6403374540938354	Combotox	ncit:C67061	DEGLYCOSYLATED RICIN A CHAIN-CONJUGATED ANTI-CD19/ANTI-CD22 IMMUNOTOXINS	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.4217483633389116	FF-10101	chembl:CHEMBL4650283	FF-10101	FALSE	FALSE	FALSE
INTERLEUKIN 5 RECEPTOR ALPHA	hgnc:6017	IL5RA	TTD	2020.06.01	NULL	52.50767123569449	Benralizumab	rxcui:1989100	BENRALIZUMAB	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	1.265245090016735	Motesanib Diphosphate	ncit:C48374	MOTESANIB DIPHOSPHATE	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.607377690888607	BETRIXABAN	rxcui:1927851	BETRIXABAN	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.2117244807890907	Antazoline	rxcui:865	ANTAZOLINE	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.5585922471882393	Atracurium	rxcui:1218	ATRACURIUM	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.079077818	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
INTERLEUKIN 1 RECEPTOR TYPE 1	hgnc:5993	IL1R1	TTD	2020.06.01	NULL	3.141484604	Anakinra	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	0.7693431682885642	Anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.055740628	Calcidiol	rxcui:1855064	CALCIFEDIOL ANHYDROUS	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.1270346884734544	Clemastine	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	0.7249579855026854	Febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.2734774543525755	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	4.039051633514961	Filgrastim	rxcui:1433764	TBO-FILGRASTIM	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1962903597596056	Mazindol	rxcui:6664	MAZINDOL	TRUE	FALSE	FALSE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	11.66837138570988	Sargramostim	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.1331836936859721	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	0.3281729452230906	Ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.364636606	INK-1117	chembl:CHEMBL3545055	INK-1117	FALSE	FALSE	TRUE
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	23.33674277141977	Odanacatib	ncit:C66981	ODANACATIB	FALSE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	1.117184494376478	TAK-071	iuphar.ligand:12302	TAK-071	FALSE	FALSE	FALSE
SPHINGOMYELIN SYNTHASE	hgnc:11123	SMS	TTD	2020.06.01	NULL	52.50767123569449	2-hydroxyoleic acid	chembl:CHEMBL4594452	2-HYDROXYOLEIC ACID	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 5	hgnc:11851	TLR5	TTD	2020.06.01	NULL	17.50255707856483	CBLB-502	chembl:CHEMBL2108683	ENTOLIMOD	FALSE	FALSE	FALSE
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	1.875273972703375	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
MORTALIN	hgnc:5244	HSPA9	TTD	2020.06.01	NULL	157.5230137070835	MKT-077	ncit:C2731	RHODACYANINE ANALOG MKT-077	FALSE	FALSE	FALSE
E-SELECTIN	hgnc:10718	SELE	TTD	2020.06.01	NULL	4.773424657790408	Bimosiamose	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	1.419126249613364	LECOZOTAN HYDROCHLORIDE	ncit:C72813	LECOZOTAN HYDROCHLORIDE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.2035181055647073	BUCINDOLOL	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.006756005	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.020575106	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.1054370908347279	IUPHAR.LIGAND:28	iuphar.ligand:28	SB 216641	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.016674395	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.046425881	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:163	ncit:C80757	BROLAMFETAMINE	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.074797252	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.034727296	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:8182	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:195	iuphar.ligand:195	SDZ SER-082	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:250	iuphar.ligand:250	RS 100235	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:248	iuphar.ligand:248	GR 125487	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:8689	ncit:C166835	IDALOPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.046840028	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.055622533	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:1790	hgnc:18123	ACVR1C	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8216	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:12378	iuphar.ligand:12378	FICONALKIB	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.019114551	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:486	iuphar.ligand:486	(+)-CYCLAZOSIN	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.058212496	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.067403943	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:501	rxcui:5784	INDORAMIN	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.091796628	IUPHAR.LIGAND:516	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:487	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.017811286	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:7109	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1259176768242074	IUPHAR.LIGAND:527	iuphar.ligand:527	[3H]MK-912	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.062958838	IUPHAR.LIGAND:7308	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	modulator	0.053964719	IUPHAR.LIGAND:1192	iuphar.ligand:1192	5-(N,N-HEXAMETHYLENE)-AMILORIDE	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:527	iuphar.ligand:527	[3H]MK-912	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.1084869240406911	IUPHAR.LIGAND:521	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:503	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:527	iuphar.ligand:527	[3H]MK-912	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:509	rxcui:66887	RACEPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:5509	rxcui:7247	NAPHAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:8638	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
NCBIGENE:2767	hgnc:4379	GNA11	GuideToPharmacology	2024.1	antibody	5.250767123569449	IUPHAR.LIGAND:9097	iuphar.ligand:9097	TIMOLUMAB	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:6367	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6378	ncit:C65893	IMIDAPRILAT	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:369	iuphar.ligand:369	(R,S)-PHPNECA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1804387327687096	IUPHAR.LIGAND:369	iuphar.ligand:369	(R,S)-PHPNECA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.060146244	IUPHAR.LIGAND:448	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.032412143	IUPHAR.LIGAND:7790	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:3944	iuphar.ligand:3944	CGP42112	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:5931	drugbank:DB07545	N-{3-[(4-{[3-(TRIFLUOROMETHYL)PHENYL]AMINO}PYRIMIDIN-2-YL)AMINO]PHENYL}CYCLOPROPANECARBOXAMIDE	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.112919723	IUPHAR.LIGAND:6907	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:7914	iuphar.ligand:7914	BV-6	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:635	iuphar.ligand:635	D-NAL-CYS-TYR-D-TRP-LYS-VAL-CYS-NAL-NH2	FALSE	FALSE	FALSE
NCBIGENE:2844	hgnc:4476	GPR21	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:11086	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:633	iuphar.ligand:633	[D-TYR6,(R)-APA11,PHE13,NLE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:2845	hgnc:4477	GPR22	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11781	iuphar.ligand:11781	AZD4320	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:12578	iuphar.ligand:12578	CIMATEROL	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.031555091	IUPHAR.LIGAND:536	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
NCBIGENE:1789	hgnc:2979	DNMT3B	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8120	iuphar.ligand:8120	COMPOUND 13D [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11777	iuphar.ligand:11777	SIM1	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.023482858	IUPHAR.LIGAND:2367	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7517	iuphar.ligand:7517	COMPOUND 9 [PMID: 23517011]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:9520	iuphar.ligand:9520	N-METHYL-2-PYRROLIDONE	FALSE	FALSE	FALSE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8950	iuphar.ligand:8950	BI-9564	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9266	iuphar.ligand:9266	CNX-774	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:8249	iuphar.ligand:8249	RN486	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:638	iuphar.ligand:638	MET-LYS-BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:652	iuphar.ligand:652	B-10356	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:662	iuphar.ligand:662	SSR240612	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:10255	iuphar.ligand:10255	NG291	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.4102161815288632	Fingolimod	rxcui:1012892	FINGOLIMOD	TRUE	TRUE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:657	iuphar.ligand:657	NPC 17731	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:638	iuphar.ligand:638	MET-LYS-BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:12516	iuphar.ligand:12516	EU-DTPA-[SER27, NLE70]HC5A	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8384	iuphar.ligand:8384	COMPOUND 4 [PMID: 25259874]	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.1930429089547592	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	1.531473744374423	KRT-232	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
NCBIGENE:1550	hgnc:2612	CYP2A7P1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8140	iuphar.ligand:8140	COMPOUND 2C [PMID: 22115617]	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:718	ncit:C76682	TECALCET	FALSE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:2733	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:4488	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:2733	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:4488	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:12647	iuphar.ligand:12647	ACT-709478	FALSE	FALSE	FALSE
NCBIGENE:390	hgnc:671	RND3	GuideToPharmacology	2024.1	blocker	0.5147810905460245	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:907	iuphar.ligand:907	Z-360	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:4382	iuphar.ligand:4382	CCL18	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:793	iuphar.ligand:793	YM-355179	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:1272	iuphar.ligand:1272	CCL16	FALSE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:8114	drugbank:DB07149	(7S)-2-(2-AMINOPYRIMIDIN-4-YL)-7-(2-FLUOROETHYL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	0.1576806944014849	IUPHAR.LIGAND:7327	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:843	iuphar.ligand:843	KALLSTROEMIN D	FALSE	FALSE	FALSE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9886	iuphar.ligand:9886	JH-VIII-49	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:10461	iuphar.ligand:10461	FADRACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:10532	iuphar.ligand:10532	BSJ-03-123	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:10081	iuphar.ligand:10081	KINASE INHIBITOR 2 [PMID: 30199702]	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:6030	iuphar.ligand:6030	PURVALANOL A	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:11064	iuphar.ligand:11064	(S)-CR8	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:9886	iuphar.ligand:9886	JH-VIII-49	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:7379	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:5943	iuphar.ligand:5943	CDK/CRK INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:10547	iuphar.ligand:10547	THAL-SNS-032	FALSE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:7303	rxcui:10378	TESTOLACTONE	TRUE	FALSE	TRUE
NCBIGENE:1983	hgnc:3299	EIF5	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
NCBIGENE:1361	hgnc:2300	CPB2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8638	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
NCBIGENE:1358	hgnc:2297	CPA2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:6957	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:10547	iuphar.ligand:10547	THAL-SNS-032	FALSE	FALSE	FALSE
NCBIGENE:1365	hgnc:2045	CLDN3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11382	iuphar.ligand:11382	LUNACALCIPOL	FALSE	FALSE	FALSE
NCBIGENE:2743	hgnc:4329	GLRB	GuideToPharmacology	2024.1	antibody	0.2625383561784725	IUPHAR.LIGAND:6888	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
NCBIGENE:2004	hgnc:3325	ELK3	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.1736364789540161	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
NCBIGENE:3244	ncbigene:3244	HPE1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12816	iuphar.ligand:12816	YT47R	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.077444943	IUPHAR.LIGAND:9002	iuphar.ligand:9002	BW373U86	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1161674142382621	IUPHAR.LIGAND:9150	rxcui:1876597	NALDEMEDINE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:3819	iuphar.ligand:3819	[3H]DPDPE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.077444943	IUPHAR.LIGAND:1628	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
NCBIGENE:1396	hgnc:2360	CRIP1	GuideToPharmacology	2024.1	inhibitor	0.6731752722524936	IUPHAR.LIGAND:5277	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:10020	iuphar.ligand:10020	DSM421	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:8368	iuphar.ligand:8368	ML321	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.026927011	IUPHAR.LIGAND:209	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.058997383	IUPHAR.LIGAND:7683	iuphar.ligand:7683	PF-592379	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.058997383	IUPHAR.LIGAND:951	iuphar.ligand:951	7-TRANS-OH-PIPAT	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.058997383	IUPHAR.LIGAND:11288	iuphar.ligand:11288	R-VK4-40	FALSE	FALSE	FALSE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.024513385	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.095122593	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:3295	iuphar.ligand:3295	[125I]L750667	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.006210251	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:934	iuphar.ligand:934	N-PROPYLNORAPOMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:2010	hgnc:3331	EMD	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:2011	hgnc:3332	MARK2	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:8171	iuphar.ligand:8171	COMPOUND 5B [PMID: 24900464]	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.010675184	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NCBIGENE:1615	hgnc:2678	DARS1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:6506	ncit:C73039	DAGLUTRIL	FALSE	FALSE	FALSE
NCBIGENE:1249	hgnc:7876	NOS3	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:11467	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10967	iuphar.ligand:10967	POSTSTATIN	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.3024635439844153	LY3214996	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
NCBIGENE:1821	hgnc:3032	DRP2	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9273	iuphar.ligand:9273	EPZ011989	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	Dubermatinib	ncit:C127116	DUBERMATINIB	FALSE	FALSE	FALSE
NCBIGENE:1828	hgnc:3048	DSG1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:9204	iuphar.ligand:9204	NAZARTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:8183	iuphar.ligand:8183	PD166285	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:10634	iuphar.ligand:10634	MS39	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.055441823	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:7642	iuphar.ligand:7642	PKI166	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9012	iuphar.ligand:9012	JNJ-42165279	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.054020238	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
NCBIGENE:2023	hgnc:3350	ENO1	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:7476	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:5589	iuphar.ligand:5589	GRIFOLIC ACID METHYL ETHER	FALSE	FALSE	FALSE
NCBIGENE:227	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1060	drugbank:DB02531	ISOBUTYRIC ACID	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	Ipatasertib	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1060	drugbank:DB02531	ISOBUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:3176	hgnc:5028	HNMT	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:12610	iuphar.ligand:12610	COMPOUND 19B [PMID: 37058391]	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.022789788	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:8095	iuphar.ligand:8095	AC710	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.068369364	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1182605208011137	GSK2334470	iuphar.ligand:8008	GSK2334470	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.082043236	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:1044	iuphar.ligand:1044	ANNEXIN I-(2-26)	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:5825	iuphar.ligand:5825	BVT173187	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:5836	iuphar.ligand:5836	MET-MET-TRP-LEU-LEU	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.3889457128569962	IUPHAR.LIGAND:1044	iuphar.ligand:1044	ANNEXIN I-(2-26)	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6244	iuphar.ligand:6244	PRP106-126	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	BLZ945	chembl:CHEMBL4227505	BLZ945	FALSE	FALSE	FALSE
NCBIGENE:235	hgnc:4045	FZD7	GuideToPharmacology	2024.1	antibody	2.100306849	IUPHAR.LIGAND:10197	iuphar.ligand:10197	VANTICTUMAB	FALSE	FALSE	FALSE
NCBIGENE:235	hgnc:4045	FZD7	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12916	iuphar.ligand:12916	F7H	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.027290889	CUDC-907	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:233	ncbigene:233	ALDRL2	GuideToPharmacology	2024.1	antibody	10.50153425	IUPHAR.LIGAND:10197	iuphar.ligand:10197	VANTICTUMAB	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:4321	iuphar.ligand:4321	TETRAHYDRODEOXYCORTICOSTERONE	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.064505739	Sapanisertib	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4095	iuphar.ligand:4095	&ALPHA;5IA	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	ABT-737	drugbank:DB17023	ABT-737	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.1325951293830669	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.1988926940746003	IUPHAR.LIGAND:4296	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6086	iuphar.ligand:6086	GALANIN(1-15)	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.044347695	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6115	iuphar.ligand:6115	GAL-B2-C18	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:6124	iuphar.ligand:6124	DITHIIPIN-1,1,4,4-TETROXIDE ANALOGUE 7	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:6124	iuphar.ligand:6124	DITHIIPIN-1,1,4,4-TETROXIDE ANALOGUE 7	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.1389091831632129	IUPHAR.LIGAND:4133	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1984416902331613	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:4078	iuphar.ligand:4078	[3H]CGP39653	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.096167896	IUPHAR.LIGAND:2361	drugbank:DB01931	5,7-DICHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
NCBIGENE:936	hgnc:1647	CD24P2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11298	ncit:C174621	OPIRANSERIN	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:9344	iuphar.ligand:9344	HISTERELIN	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:3786	iuphar.ligand:3786	[125I]GNRH I (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1186	iuphar.ligand:1186	[125I]CETRORELIX	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	0.1241316104862754	IUPHAR.LIGAND:1012	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	CancerCommons	25-Jul-13	inhibitor	0.052824619	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:12906	iuphar.ligand:12906	COMPOUND 77A [PMID: 37639383]	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:5585	rxcui:475230	DEGARELIX	TRUE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	0.3671865121377238	IUPHAR.LIGAND:611	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:1185	ncit:C97486	SUFUGOLIX	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5788	iuphar.ligand:5788	MK 6892	FALSE	FALSE	FALSE
NCBIGENE:403	hgnc:694	ARL3	GuideToPharmacology	2024.1	blocker	7.501095891	IUPHAR.LIGAND:6262	iuphar.ligand:6262	EC18	FALSE	FALSE	FALSE
NCBIGENE:1887	ncbigene:1887	EBVM1	GuideToPharmacology	2024.1	NULL	17.50255707856483	IUPHAR.LIGAND:4891	iuphar.ligand:4891	B AND T LYMPHOCYTE ATTENUATOR	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:8365	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:11118	drugbank:DB14979	MARTINOSTAT	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.077827576	CABERGOLINE	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.1209854175937661	IUPHAR.LIGAND:8367	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.07699072	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.1215455352678113	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.094099769	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:8365	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:7374	iuphar.ligand:7374	TUBACIN	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:10490	iuphar.ligand:10490	SS-208	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1620607136904151	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.058212496	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.2134458180312784	IUPHAR.LIGAND:10490	iuphar.ligand:10490	SS-208	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.071148606	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:7057	iuphar.ligand:7057	COMPOUND 16 [PMID: 20947351]	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:7916	iuphar.ligand:7916	SANTACRUZAMATE A	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7491	iuphar.ligand:7491	TMP269	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.1835932560688619	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.2430910705356227	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:10490	iuphar.ligand:10490	SS-208	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.095468493	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	SJ000147784	chembl:CHEMBL590186	CHEMBL:CHEMBL590186	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:1194	iuphar.ligand:1194	2-(3-BROMOPHENYL)HISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1205	iuphar.ligand:1205	METHYLHISTAPRODIFEN	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:7176	rxcui:39684	EPINASTINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.02321294	IUPHAR.LIGAND:209	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:3959	ncit:C152643	TIOTIDINE	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1265	iuphar.ligand:1265	CIPROXIFAN	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1268	iuphar.ligand:1268	2-METHYLHISTAMINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	BAS-8770954	chembl:CHEMBL478324	CHEMBL:CHEMBL478324	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:1254	iuphar.ligand:1254	METHIMEPIP	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5849	iuphar.ligand:5849	2-HYDROXYLAURIC ACID	FALSE	FALSE	FALSE
MUCL3	hgnc:21666	MUCL3	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NCBIGENE:152	hgnc:283	ADRA2C	GuideToPharmacology	2024.1	agonist	0.7395446652914718	IUPHAR.LIGAND:2365	drugbank:DB03107	BETA-ALANINE	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10682	iuphar.ligand:10682	COMPOUND 8U [PMID: 31999451]	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
ADH1C	hgnc:251	ADH1C	PharmGKB	4/5/24	NULL	0.028459442	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:2884	hgnc:4561	GPX1P2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9217	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12450	drugbank:DB12709	TRIBUTYRIN	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.8537832721251137	PDR001	ncit:C121625	SPARTALIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:10136	ncit:C148147	LAZERTINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:12171	iuphar.ligand:12171	COMPOUND 8L [PMID: 36053746]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:8868	iuphar.ligand:8868	SCH221510	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.015019357	IUPHAR.LIGAND:1627	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:7956	ncit:C82363	GOLVATINIB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:8095	iuphar.ligand:8095	AC710	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	Indium-111	rxcui:90540	INDIUM-111	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.008690445	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.5834185692854944	Lintopride	ncit:C66018	LINTOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:517	hgnc:842	ATP5MC2	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:525	hgnc:853	ATP6V1B1	GuideToPharmacology	2024.1	blocker	1.050153425	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:571	hgnc:1282	GRIK1-AS2	GuideToPharmacology	2024.1	blocker	0.8751278539282418	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:2612	iuphar.ligand:2612	ERGTX-1	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	0.546954909	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
AP ENDONUCLEASE 1	hgnc:587	APEX1	TTD	2020.06.01	NULL	0.5277152888009498	APX-3330	chembl:CHEMBL578390	APX-3330	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:8610	iuphar.ligand:8610	3S,4R-293B	FALSE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:5702	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6711	iuphar.ligand:6711	COMPOUND 3 [PMID: 22533316]	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.1071585127259071	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	C-CAR011	ncit:C141050	AUTOLOGOUS ANTI-CD19 CHIMERIC ANTIGEN RECEPTOR T-CELLS C-CAR011	FALSE	FALSE	FALSE
NCBIGENE:1391	hgnc:6719	LTC4S	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8875	iuphar.ligand:8875	COMPOUND 39 [PMID: 23623673]	FALSE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:10402	iuphar.ligand:10402	ZAK INHIBITOR 6P	FALSE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11656	drugbank:DB08040	KELATORPHAN	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.1875273972703375	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
NCBIGENE:633	hgnc:1044	BGN	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:10483	iuphar.ligand:10483	COMPOUND 6N [PMID: 31419141]	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:2752	iuphar.ligand:2752	27-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:11314	iuphar.ligand:11314	CPY	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:2910	drugbank:DB07780	FARNESYL DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2675	hgnc:4244	GFRA2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10141	iuphar.ligand:10141	KDM5 INHIBITOR N71	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:2451	ncit:C87339	NADIDE	FALSE	FALSE	FALSE
NCBIGENE:2675	hgnc:4244	GFRA2	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:8744	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1297	iuphar.ligand:1297	[PHE13,TYR19]MCH	FALSE	FALSE	FALSE
NCBIGENE:2096	hgnc:3463	ESAT	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9848	iuphar.ligand:9848	GALAPAGOS MAPKAPK5 INHIBITOR D	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:3633	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
NCBIGENE:2847	hgnc:4479	MCHR1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:11783	iuphar.ligand:11783	AZD5991	FALSE	FALSE	FALSE
NCBIGENE:281	hgnc:479	AMYP1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:1307	iuphar.ligand:1307	[AVA9,10,AVA14,15]-AC-HMCH6-16-NH2	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:1314	iuphar.ligand:1314	T-226296	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6342	iuphar.ligand:6342	COMPOUND 2F [PMID: 17532216]	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6346	iuphar.ligand:6346	COMPOUND 23E [PMID: 17929793]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2004	iuphar.ligand:2004	BIM 23052	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:1368	iuphar.ligand:1368	L-CCG-I	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	modulator	0.5903640284436551	IUPHAR.LIGAND:7626	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:6006	iuphar.ligand:6006	MEK INHIBITOR I	FALSE	FALSE	FALSE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8875	iuphar.ligand:8875	COMPOUND 39 [PMID: 23623673]	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:307	iuphar.ligand:307	4-DAMP	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.02321294	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:361	iuphar.ligand:361	TRIPITRAMINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.5527123287967841	IUPHAR.LIGAND:7635	iuphar.ligand:7635	DUO3	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.069089041	IUPHAR.LIGAND:340	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.5527123287967841	IUPHAR.LIGAND:358	iuphar.ligand:358	LEVETIMIDE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:323	iuphar.ligand:323	HEXOCYCLIUM	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.025489161	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:300	iuphar.ligand:300	METHYLFURMETHIDE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:12486	iuphar.ligand:12486	[3H]IPEROXO	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.09814518	NOMIFENSINE MALEATE	rxcui:262302	NOMIFENSINE MALEATE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:303	iuphar.ligand:303	OXOTREMORINE-M	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:323	iuphar.ligand:323	HEXOCYCLIUM	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:335	iuphar.ligand:335	G&OUML; 7874	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:349	rxcui:11201	VINCAMINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.07458476	IUPHAR.LIGAND:340	iuphar.ligand:340	WIN 62,577	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:7483	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:361	iuphar.ligand:361	TRIPITRAMINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.1591141552596803	IUPHAR.LIGAND:332	iuphar.ligand:332	N-BENZYL BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1345	iuphar.ligand:1345	5-HEAT	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.043180651	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:9189	iuphar.ligand:9189	HS665	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1647	iuphar.ligand:1647	DAMGO	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:9190	iuphar.ligand:9190	COMPOUND 3 [PMID: 23134120]	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.044385183	IUPHAR.LIGAND:7082	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:3005	hgnc:4714	H1-0	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9933	iuphar.ligand:9933	NSC 780521	FALSE	FALSE	FALSE
NCBIGENE:2789	hgnc:4409	GNG5P1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9670	iuphar.ligand:9670	COMPOUND 28 [PMID: 28671460]	FALSE	FALSE	FALSE
NCBIGENE:2789	hgnc:4409	GNG5P1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10053	drugbank:DB11683	PF-06282999	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2614	iuphar.ligand:2614	ATX-II	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:9980	iuphar.ligand:9980	PF‐06526290	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:2614	iuphar.ligand:2614	ATX-II	FALSE	FALSE	FALSE
NCBIGENE:981	hgnc:23089	SLC13A5	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12852	iuphar.ligand:12852	COMPOUND 7 [PMID: 37428122]	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.052090944	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.1562728310586145	IUPHAR.LIGAND:2625	iuphar.ligand:2625	SAXITOXIN	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.1091635576625665	IUPHAR.LIGAND:2402	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:9537	iuphar.ligand:9537	ATRACURIUM	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2094	iuphar.ligand:2094	PHYSALAEMIN	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2104	iuphar.ligand:2104	L-703,606	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3901	iuphar.ligand:3901	MEN10627	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:13008	iuphar.ligand:13008	NT-0796	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:9747	iuphar.ligand:9747	AT-403	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:12419	iuphar.ligand:12419	MCOPPB	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1682	iuphar.ligand:1682	N/OFQ-(1-13)-NH2	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:7928	iuphar.ligand:7928	PEG40-NMU	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.1643432589536604	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
NCBIGENE:2696	hgnc:4271	GIPR	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12352	iuphar.ligand:12352	COMPOUND 15A [PMID: 36642961]	FALSE	FALSE	FALSE
NCBIGENE:2129	hgnc:14311	NUAK1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8047	iuphar.ligand:8047	WZ4003	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.2386712328895204	IUPHAR.LIGAND:2175	iuphar.ligand:2175	[3H]AVP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2278	iuphar.ligand:2278	[ALA11,22,28]VIP	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	2.625383561784724	BMS-813160	drugbank:DB16240	BMS-813160	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	1.544343271638073	IUPHAR.LIGAND:11370	iuphar.ligand:11370	(3,5)-[19F]2-PHE-&PSI;-ALA	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:4498	iuphar.ligand:4498	LYS[Z(NO2)]-PRO	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	3.088686543276147	IUPHAR.LIGAND:11368	iuphar.ligand:11368	[3H]-IPP	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.053038052	IUPHAR.LIGAND:2674	iuphar.ligand:2674	GW7647	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:11130	iuphar.ligand:11130	COMPOUND 25 [PMID: 32687365]	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:2686	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
UNIPROT:O14965	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.1582152052299645	MLN-8237	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2708	iuphar.ligand:2708	BADGE	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:2708	iuphar.ligand:2708	BADGE	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2709	iuphar.ligand:2709	PAT5A	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1562728310586146	IUPHAR.LIGAND:8527	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:10096	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:7795	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:10096	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:9907	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.034727296	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.070197421	IUPHAR.LIGAND:7951	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9852	iuphar.ligand:9852	MK-0359	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:9776	ncit:C169909	DIFAMILAST	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9790	iuphar.ligand:9790	PIM447	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.048618214	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
NCBIGENE:2864	hgnc:4498	FFAR1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8468	iuphar.ligand:8468	ME0328	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:11348	iuphar.ligand:11348	PJ34	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.076765601	IUPHAR.LIGAND:2804	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.2243917574174979	IUPHAR.LIGAND:611	iuphar.ligand:611	LITHOCHOLIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.007496384	TESTOSTERONE UNDECANOATE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
NCBIGENE:2384	hgnc:3896	FRA3A	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:8668	iuphar.ligand:8668	FURIN INHIBITOR PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:2395	hgnc:3951	FXN	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10967	iuphar.ligand:10967	POSTSTATIN	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:11518	iuphar.ligand:11518	DOSTARLIMAB	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.1881995384791917	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
NCBIGENE:3263	hgnc:5171	HPX	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4735	iuphar.ligand:4735	MICROCYSTIN-LR	FALSE	FALSE	FALSE
NCBIGENE:3264	hgnc:9281	PPP1CA	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5349	iuphar.ligand:5349	OKADAIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1213	hgnc:2092	CLTC	GuideToPharmacology	2024.1	NULL	7.501095891	IUPHAR.LIGAND:6689	iuphar.ligand:6689	[3H]N5-METHYLFOLATE	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3713	iuphar.ligand:3713	QRFP43	FALSE	FALSE	FALSE
NCBIGENE:3007	hgnc:4717	H1-3	GuideToPharmacology	2024.1	modulator	8.751278539282415	IUPHAR.LIGAND:10473	rxcui:2594468	MITAPIVAT	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.280789686	DONITRIPTAN	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:8943	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:11544	iuphar.ligand:11544	BELVARAFENIB	FALSE	FALSE	FALSE
NCBIGENE:1527	hgnc:2563	TEX28	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10437	iuphar.ligand:10437	COMPOUND E22 [PMID: 31298542]	FALSE	FALSE	FALSE
NCBIGENE:2631	hgnc:4179	NIPSNAP2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:6822	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
PSMD1	hgnc:9554	PSMD1	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1853	hgnc:9668	PTPRD	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10109	iuphar.ligand:10109	7-BIA	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.2692701089009974	IUPHAR.LIGAND:1989	iuphar.ligand:1989	RELAXIN	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:11465	iuphar.ligand:11465	NANOLUC R3/I5 CHIMERA	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1994	iuphar.ligand:1994	RELAXIN	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:11459	iuphar.ligand:11459	B1-27	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1000146118775133	OPHIOBOLIN O	chembl:CHEMBL1934283	OPHIOBOLIN O	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:11460	iuphar.ligand:11460	COMPOUND 4 [PMID: 30824200]	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:2922	iuphar.ligand:2922	PHYTOSPHINGOSINE 1-PHOSPHATE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	3-HYDROXYPHTHALIC ANHYDRIDE	chembl:CHEMBL2057864	CHEMBL:CHEMBL2057864	FALSE	FALSE	FALSE
NCBIGENE:2198	ncbigene:2198	FAUNA@	GuideToPharmacology	2024.1	inhibitor	0.4565884455277782	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2930	iuphar.ligand:2930	VPC44116	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:2407	rxcui:1012892	FINGOLIMOD	TRUE	TRUE	FALSE
NCBIGENE:2225	hgnc:11408	STK4	GuideToPharmacology	2024.1	inhibitor	0.326134604	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.035976479	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:2217	hgnc:3621	FCGRT	GuideToPharmacology	2024.1	inhibitor	0.2536602475154323	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1526385791735305	IUPHAR.LIGAND:7118	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.093931433	IUPHAR.LIGAND:7351	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.07631929	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NPM1	hgnc:7910	NPM1	FDA	10-Apr-24	NULL	0.4167275494896389	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NCBIGENE:3096	hgnc:4920	HIVEP1	GuideToPharmacology	2024.1	NULL	10.50153424713889	IUPHAR.LIGAND:10480	iuphar.ligand:10480	BAY-293	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5636	iuphar.ligand:5636	DEMOTATE 2	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2046	iuphar.ligand:2046	L-054,522	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.062065805	IUPHAR.LIGAND:2055	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2008	iuphar.ligand:2008	CST-17	FALSE	FALSE	FALSE
NCBIGENE:2418	hgnc:3929	FRA8A	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8483	iuphar.ligand:8483	COMPOUND 4D [PMID: 25489658]	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.03262504	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:2739	hgnc:4323	GLO1	GuideToPharmacology	2024.1	NULL	4.375639269641208	IUPHAR.LIGAND:12308	iuphar.ligand:12308	A947	FALSE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11600	iuphar.ligand:11600	COMPOUND 21 [PMID: 34141085]	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:9633	iuphar.ligand:9633	METHYLMALONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:615	hgnc:7973	NR2E1	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:2641	iuphar.ligand:2641	BMS493	FALSE	FALSE	FALSE
NCBIGENE:2421	hgnc:3931	FRA8C	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:10733	iuphar.ligand:10733	I-432	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	1.628144844517658	INDIPLON	ncit:C74385	INDIPLON	FALSE	FALSE	FALSE
NCBIGENE:2423	hgnc:3933	FRA8E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8581	iuphar.ligand:8581	EXAMPLE 8 [WO1999033801A1]	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.1988926940746003	IUPHAR.LIGAND:6285	iuphar.ligand:6285	OMEGA-CHLOROACETOPHENONE	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.7721716358190367	IUPHAR.LIGAND:10278	iuphar.ligand:10278	GSK1702934A	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	BROMODIPHENHYDRAMINE	rxcui:19759	BROMODIPHENHYDRAMINE	TRUE	FALSE	FALSE
NCBIGENE:499	ncbigene:499	ATP5A2	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:1640	iuphar.ligand:1640	NALTRIBEN	FALSE	FALSE	FALSE
NCBIGENE:502	hgnc:13357	MCOLN2	GuideToPharmacology	2024.1	activator	1.750255707856483	IUPHAR.LIGAND:2794	iuphar.ligand:2794	PHOSPHATIDYL (3,5) INOSITOL BISPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:498	hgnc:823	ATP5F1A	GuideToPharmacology	2024.1	activator	0.6563458904461812	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.2500365296937833	IUPHAR.LIGAND:4261	iuphar.ligand:4261	NADA	FALSE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:7575	rxcui:1599538	EDOXABAN	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4310	iuphar.ligand:4310	SB452533	FALSE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.108711535	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:6813	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
NCBIGENE:1870	hgnc:3114	E2F2	GuideToPharmacology	2024.1	NULL	3.500511415712966	IUPHAR.LIGAND:5064	iuphar.ligand:5064	LYMPHOTOXIN-&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:2367	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:10458	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
NCBIGENE:1031	hgnc:1789	CDKN2C	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9327	ncit:C152863	VERINURAD	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2151	iuphar.ligand:2151	AC-7954	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	ChEMBL	33	inhibitor	1.500219178	ENTACAPONE	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
NCBIGENE:2431	hgnc:12628	USP5	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8669	iuphar.ligand:8669	VIALININ A	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3501	iuphar.ligand:3501	FL104	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:9437	iuphar.ligand:9437	JNJ-39319202	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1524	iuphar.ligand:1524	[LEU31,PRO34]NPY (PIG)	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	modulator	3.500511415712966	IUPHAR.LIGAND:12607	iuphar.ligand:12607	TERT-BUTYLPHENOXYCYCLOHEXANOL	FALSE	FALSE	FALSE
PRPS1	hgnc:9462	PRPS1	CIViC	10-Apr-24	NULL	3.500511415712967	LOMETREXOL	ncit:C979	LOMETREXOL	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	DUP-697	chembl:CHEMBL42485	DUP-697	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.057878826	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.099446347	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.4167275494896388	SONIDEGIB	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.3697723326457359	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
IRS2	hgnc:6126	IRS2	CIViC	10-Apr-24	NULL	6.563458904461812	DUAL IGF-1R/INSR INHIBITOR BMS-754807	ncit:C74043	DUAL IGF-1R/INSR INHIBITOR BMS-754807	FALSE	FALSE	TRUE
MDM4	hgnc:6974	MDM4	CIViC	10-Apr-24	NULL	0.2917092846427472	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.032412143	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.8140724222588294	MN-221	chembl:CHEMBL2218893	BEDORADRINE SULFATE	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.546954909	SERIBANTUMAB	ncit:C78859	SERIBANTUMAB	FALSE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	CIViC	10-Apr-24	NULL	1.078924751	LAROTRECTINIB	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.1461794856227575	APALUTAMIDE	rxcui:1999574	APALUTAMIDE	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.108374966	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.099220845	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.1367387271762877	ZUCLOPENTHIXOL	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	CIViC	10-Apr-24	NULL	1.077080435603989	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.2592971419046642	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.068369364	RIGOSERTIB	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	0.1207072901969988	L-Alanine	rxcui:426	ALANINE	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1520492410300034	ALPELISIB	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
FLCN	hgnc:27310	FLCN	CIViC	10-Apr-24	NULL	0.4605936073306534	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
ARID1A	hgnc:11110	ARID1A	CIViC	10-Apr-24	NULL	0.1591141552596803	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
GNA11	hgnc:4379	GNA11	CIViC	10-Apr-24	NULL	0.2386712328895204	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.020465128	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12943	iuphar.ligand:12943	TOMINOSTAT	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	CIViC	10-Apr-24	NULL	0.009974862	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.002069839	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.299554767	AGI-5198	iuphar.ligand:9240	AGI-5198	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	CIViC	10-Apr-24	NULL	0.027390543	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.015272737	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
PTPRD	hgnc:9668	PTPRD	CIViC	10-Apr-24	NULL	3.281729452230906	CIXUTUMUMAB	ncit:C79828	CIXUTUMUMAB	FALSE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.053361455	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DoCM	10-Apr-24	NULL	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	JAX-CKB	10-Apr-24	NULL	0.8008364246019593	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.8334550989792776	LANREOTIDE ACETATE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1826353782111113	Luminespib	ncit:C71467	LUMINESPIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.024991752	Panobinostat	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	CC-90003	ncit:C119747	ERK INHIBITOR CC-90003	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.024991752	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.5527123287967842	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.3106962795011509	Momelotinib	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.1049104320393496	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.031822831	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.091317689	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.006768633	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1752592497853621	Brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1144789343801478	Aprutumab ixadotin	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.6848826682916673	Upadacitinib	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.1615620653405984	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	1.141471113819445	Ilginatinib	ncit:C98109	ILGINATINIB	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	NORSTICTIC ACID	chembl:CHEMBL228281	NORSTICTIC ACID	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	1.897867635025102	Avapritinib	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.2957715794844315	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.031317948	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.1331836936859721	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.4167275494896388	SCH772984	iuphar.ligand:8056	SCH772984	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.375054795	VX-11e	iuphar.ligand:9375	VTX-11E	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:10423	ncit:C152226	RIPASUDIL	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.2500365296937833	Ravoxertinib	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.2083637747448194	U0126	iuphar.ligand:5282	U0126	FALSE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	1.666910197958555	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.018572323	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.3387591692625452	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.044573575	Foretinib	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	inhibitor	0.036463661	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	Miransertib	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.069454592	Afuresertib	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1135300999690691	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	PKI-402	chembl:CHEMBL589258	CHEMBL:CHEMBL589258	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2365210416022274	MS417	iuphar.ligand:7512	MS417	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	Borussertib	chembl:CHEMBL4795065	BORUSSERTIB	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.022099188	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
KCNK18	hgnc:19439	KCNK18	ChEMBL	33	potentiator	0.2917092846427472	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.1750255707856483	ONVANSERTIB	ncit:C143162	ONVANSERTIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.010247399	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	0.1223955040459079	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
NCBIGENE:1385	hgnc:2345	CREB1	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:9054	iuphar.ligand:9054	PF-04191834	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.081872668	amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
NCBIGENE:452	hgnc:4581	GRIK3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:4185	iuphar.ligand:4185	DYSIHERBAINE	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:12356	iuphar.ligand:12356	SZUH280	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.025942525	IUPHAR.LIGAND:9769	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:2610	iuphar.ligand:2610	BEKM-1	FALSE	FALSE	FALSE
NCBIGENE:436	hgnc:747	ASLP1	GuideToPharmacology	2024.1	activator	6.563458904461812	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:8586	iuphar.ligand:8586	AE9C90CB	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	1.544343271638073	IUPHAR.LIGAND:4599	iuphar.ligand:4599	[14C]GLYSAR	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:2634	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.082043236	DIPYRONE	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002648692	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.1902451856365742	ELTROMBOPAG	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
TTR	hgnc:12405	TTR	FDA	10-Apr-24	NULL	8.751278539282415	Patisiran	rxcui:2053490	PATISIRAN	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	0.2347585897273971	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.4039051633514962	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.038894571	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	ChEMBL	33	inhibitor	0.053798843	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.4039051633514961	TYRPHOSTIN A25	ncit:C1484	TYRPHOSTIN A25	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	(R)-INDOPROFEN	chembl:CHEMBL264931	(R)-INDOPROFEN	FALSE	FALSE	FALSE
UNIPROT:P23415	hgnc:4326	GLRA1	TdgClinicalTrial	Jan-14	NULL	0.1290114772375786	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	1.544343271638073	DEMECARIUM BROMIDE	rxcui:22482	DEMECARIUM BROMIDE	TRUE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	0.4861821410712453	G-202	ncit:C90554	MIPSAGARGIN	FALSE	FALSE	FALSE
PANCREATIC TRIACYLGLYCEROL LIPASE	hgnc:9155	PNLIP	TTD	2020.06.01	NULL	3.029288725136221	Orlistat	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	A-007	ncit:C61305	SIVIFENE	FALSE	FALSE	FALSE
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	1.071585127259071	ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
TSC1	hgnc:12362	TSC1	CIViC	10-Apr-24	NULL	0.2302968036653267	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
MYH7B	hgnc:15906	MYH7B	ChEMBL	33	inhibitor	1.944728564284981	MAVACAMTEN	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DIFLUPREDNATE	rxcui:23043	DIFLUPREDNATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	TOMELUKAST	ncit:C74135	TOMELUKAST	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.1552333222045661	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.02896176	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.01535312	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.028598949	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.1715936968486748	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.075333818	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.086551106	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	2.059124362184098	BMS-986142	drugbank:DB15291	BMS-986142	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:1008	iuphar.ligand:1008	SARAFOTOXIN S6C	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.054243462	IUPHAR.LIGAND:4193	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:1093	iuphar.ligand:1093	GHRP-6	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1801	iuphar.ligand:1801	[ILE5,TRP23]PTHRP-(4-36) (HUMAN)	FALSE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	4.565884455277782	ZIBOTENTAN	ncit:C48430	ZIBOTENTAN	FALSE	FALSE	TRUE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.112036283	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	inhibitor	0.3547815624033412	ROBALZOTAN	ncit:C74143	ROBALZOTAN	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.016878069	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	PharmGKB	4/5/24	NULL	0.1235474617310458	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1262203635473425	ERGOLOID MESYLATE	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.072851434	INFLIXIMAB	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	2.734774543525755	10-PROPARGYL-10-DEAZAAMINOPTERIN	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.024309107	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.251232877	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.3977853881492006	DOV 21947	chembl:CHEMBL1818442	AMITIFADINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.082043236	OXYMETAZOLINE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.4070362111294147	IUPHAR.LIGAND:7724	iuphar.ligand:7724	TTA-A2	FALSE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:10435	iuphar.ligand:10435	COMPOUND 10A [PMID: 31283223]	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1367387271762877	IFENPRODIL	rxcui:27403	IFENPRODIL	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.089298761	IUPHAR.LIGAND:2711	ncit:C72726	CIGLITAZONE	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.4884434533552977	NEUROTROPHIC FACTOR	ncit:C2259	RECOMBINANT NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	0.2035181055647073	Citarinostat	ncit:C121641	CITARINOSTAT	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1419126249613365	BAY1125976	iuphar.ligand:10908	BAY1125976	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP SEMISYNTHETIC PURIFIED HUMAN	chembl:CHEMBL1201543	INSULIN ZINC SUSP SEMISYNTHETIC PURIFIED HUMAN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	GNF-PF-3736	chembl:CHEMBL583824	CHEMBL:CHEMBL583824	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.2386712328895204	IUPHAR.LIGAND:6307	iuphar.ligand:6307	BENZOQUINONE	FALSE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	PharmGKB	4/5/24	NULL	0.3088686543276147	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
PTPRD	hgnc:9668	PTPRD	CIViC	10-Apr-24	NULL	0.5048814541893702	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	CIViC	10-Apr-24	NULL	0.1582152052299645	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
PRTN3	hgnc:9495	PRTN3	NCI	14-Sep-17	NULL	1.640864726115453	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VIM	hgnc:12692	VIM	ChEMBL	33	other/unknown	10.50153424713889	PRITUMUMAB	ncit:C170350	PRITUMUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1570910134201779	E6201	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.173866461	TCMDC-125614	chembl:CHEMBL580609	CHEMBL:CHEMBL580609	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
CYP24A1	hgnc:2602	CYP24A1	PharmGKB	4/5/24	NULL	2.333674277141978	telaprevir	rxcui:1102261	TELAPREVIR	TRUE	FALSE	FALSE
ALDH1A2	hgnc:15472	ALDH1A2	PharmGKB	4/5/24	NULL	0.5834185692854945	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.1295419520617463	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:170	iuphar.ligand:170	ORG 12962	FALSE	FALSE	FALSE
UNIPROT:Q00653	hgnc:7795	NFKB2	TdgClinicalTrial	Jan-14	NULL	0.7095631248066824	NF-KB DECOY	drugbank:DB05559	NF-KAPPAB DECOY	FALSE	FALSE	FALSE
UNIPROT:Q9Y5Y4	hgnc:4502	PTGDR2	TdgClinicalTrial	Jan-14	NULL	4.145342465975881	OC000459	iuphar.ligand:9277	TIMAPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:9970	iuphar.ligand:9970	COMPOUND 11H [PMID: 29808961]	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.023823807	IUPHAR.LIGAND:5698	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:1490	hgnc:2500	CCN2	GuideToPharmacology	2024.1	inhibitor	0.1187956362798518	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.2059124362184098	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	0.6731752722524935	Neu-P11	chembl:CHEMBL4297523	PIROMELATINE	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	BNC-105	ncit:C162343	VASCULAR DISRUPTING AGENT BNC105	FALSE	FALSE	FALSE
UNIPROT:P26358	hgnc:2976	DNMT1	TdgClinicalTrial	Jan-14	NULL	0.1790034246671403	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	PROCAINE	rxcui:8701	PROCAINE	TRUE	FALSE	FALSE
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	4.039051633514961	SGN-CD70A	chembl:CHEMBL4594498	SGN-CD70A	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	SCH772984	iuphar.ligand:8056	SCH772984	FALSE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.024041974	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	LONCASTUXIMAB TESIRINE	rxcui:2540964	LONCASTUXIMAB TESIRINE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	PROPIONYLPROMAZINE HYDROCHLORIDE	chembl:CHEMBL1256661	PROPIONYLPROMAZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	ChEMBL	33	negative modulator	2.187819634820604	MECAMYLAMINE HYDROCHLORIDE	rxcui:91240	MECAMYLAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
B7 HOMOLOG 3	hgnc:19137	CD276	TTD	2020.06.01	NULL	10.50153424713889	MGD009	ncit:C136983	OBRINDATAMAB	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.5181678082469852	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	PharmGKB	4/5/24	NULL	1.009762908	lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
UNIPROT:P21397	hgnc:6833	MAOA	TdgClinicalTrial	Jan-14	NULL	2.692701089009974	CX157	drugbank:DB05205	CX157	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11799	iuphar.ligand:11799	SJ995973	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.027577558	NAPROXEN SODIUM	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1875273972703375	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.031254566	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2343	ncbigene:2343	FNTBL1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9298	iuphar.ligand:9298	LHVS	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	modulator	3.500511415712966	IUPHAR.LIGAND:10238	iuphar.ligand:10238	VU0155094	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.006811217	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	activator	1.944728564284981	IUPHAR.LIGAND:4222	iuphar.ligand:4222	IP3	FALSE	FALSE	FALSE
RICTOR	hgnc:28611	RICTOR	PharmGKB	4/5/24	NULL	0.7501095890813501	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.029090123	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	0.364636606	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ESTRAMUSTINE PHOSPHATE SODIUM	rxcui:4090	ESTRAMUSTINE PHOSPHATE SODIUM	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.034544521	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
DNTT	hgnc:2983	DNTT	NCI	14-Sep-17	NULL	2.187819634820604	ALPHA INTERFERON	ncit:C225	RECOMBINANT INTERFERON ALFA	FALSE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	2.019525817	ALUM	rxcui:221456	ALUM, POTASSIUM	TRUE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.036718651	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
SLC16A7	hgnc:10928	SLC16A7	PharmGKB	4/5/24	NULL	1.406455479527531	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NCBIGENE:1402	hgnc:736	NAAA	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:10121	iuphar.ligand:10121	F215	FALSE	FALSE	FALSE
DDX12P	hgnc:2737	DDX12P	PharmGKB	4/5/24	NULL	7.001022831425933	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:11815	iuphar.ligand:11815	SA-57	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	NULL	1.166837138570988	IUPHAR.LIGAND:4935	iuphar.ligand:4935	GROWTH ARREST SPECIFIC PROTEIN 6	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.300043836	DNQX	chembl:CHEMBL155265	DNQX	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009433646	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	GNF-PF-3696	chembl:CHEMBL598885	CHEMBL:CHEMBL598885	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-948	chembl:CHEMBL602158	CHEMBL:CHEMBL602158	FALSE	FALSE	FALSE
SLC2A2	hgnc:11006	SLC2A2	PharmGKB	4/5/24	NULL	0.8975670296699914	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:449	iuphar.ligand:449	MRS1754	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	BESIFLOXACIN HYDROCHLORIDE	ncit:C76228	BESIFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.1000146118775133	OLANZAPINE PAMOATE	rxcui:1294588	OLANZAPINE PAMOATE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.024354207	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CFI	hgnc:5394	CFI	NCI	14-Sep-17	NULL	5.000730593875666	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:10947	iuphar.ligand:10947	NIK INHIBITOR 12F	FALSE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.3182283105193606	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.028692717	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.06823609	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.068037151	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.2822993077187876	ABT-122	iuphar.ligand:9597	REMTOLUMAB	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	3.088686543276147	PF-4191834	drugbank:DB11645	PF-4191834	FALSE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	2.625383561784724	Flotetuzumab	ncit:C117238	FLOTETUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10582	iuphar.ligand:10582	COMPOUND 15B [PMID: 31811124]	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	1.831662950082366	Debio 1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.097236428	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
P4HTM	hgnc:28858	P4HTM	ChEMBL	33	inhibitor	4.375639269641208	ROXADUSTAT	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:1467	iuphar.ligand:1467	OHM-11526	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	0.8008364246019593	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.052229116	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	0.6141248097742047	Dabigatran	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	inhibitor	1.312691780892362	HYDROXYCHLOROQUINE SULFATE	rxcui:153972	HYDROXYCHLOROQUINE SULFATE	TRUE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.8751278539282416	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	DIPYRITHIONE	rxcui:1362743	DIPYRITHIONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008036068	ZIDOVUDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:12262	iuphar.ligand:12262	SRX246	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.729273212	1,4-BIS(2,6-DIFLUOROPHENYLSULFONYL)PIPERAZINE	chembl:CHEMBL1093369	CHEMBL:CHEMBL1093369	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.1396480617970598	TETRYDAMINE	ncit:C152580	TETRYDAMINE	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.3923362732430473	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PSMB5	hgnc:9542	PSMB5	MyCancerGenome	20-Jun-17	other/unknown	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
MASP2	hgnc:6902	MASP2	ChEMBL	33	inhibitor	105.0153424713889	NARSOPLIMAB	ncit:C119952	NARSOPLIMAB	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	DICOFOL	chembl:CHEMBL228511	DICOFOL	FALSE	FALSE	FALSE
BMP10	hgnc:20869	BMP10	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	26.25383561784724	DALANTERCEPT	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
PI3-KINASE BETA	hgnc:8976	PIK3CB	TTD	2020.06.01	NULL	0.1562728310586146	AZD8186	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:6223	iuphar.ligand:6223	COMPOUND 3 [PMID: 21105727]	FALSE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.070197421	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.004667349	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.03505185	RETINAL	iuphar.ligand:2350	ALL-TRANS-RETINAL	FALSE	FALSE	FALSE
NCBIGENE:1282	hgnc:2202	COL4A1	GuideToPharmacology	2024.1	activator	13.12691780892362	IUPHAR.LIGAND:10215	iuphar.ligand:10215	FD6	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.011110383	DEFEROXAMINE MESYLATE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.2282942227638891	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	0.070197421	Fluphenazine	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.020391329	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1767935058440892	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.009205412	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:785	iuphar.ligand:785	TEIJIN-LEAD_CMP_5	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	0.1211715490054488	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
UNIPROT:Q12809	hgnc:6251	KCNH2	TEND	1-Aug-11	NULL	0.021370644	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	NCI	14-Sep-17	NULL	0.760980743	NELFINAVIR	rxcui:134527	NELFINAVIR	TRUE	FALSE	TRUE
SERINE/THREONINE PP1-ALPHA	hgnc:9281	PPP1CA	TTD	2020.06.01	NULL	5.250767123569449	CANTHARIDIN	rxcui:1984	CANTHARIDIN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.011458303	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.036212187	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	HALAZONE	rxcui:59838	HALAZONE	FALSE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.6863747873946994	atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	MMV667491	chembl:CHEMBL1437888	CHEMBL:CHEMBL1437888	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.1584738568481725	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
NCBIGENE:276	hgnc:474	AMY1A	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:9492	iuphar.ligand:9492	COMPOUND 43 [PMID: 26751273]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2056	iuphar.ligand:2056	[111IN,90Y]DOTA-LAN	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:7578	iuphar.ligand:7578	COMPOUND 15A [PMID: 22464687]	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003262967	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
SNORD68	hgnc:32729	SNORD68	PharmGKB	4/5/24	NULL	1.419126249613364	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.2011788169949981	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	1.272913242077442	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.3125456621172291	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.2917092846427472	4-HYDROPEROXYCYCLOPHOSPHAMIDE	ncit:C1423	PERFOSFAMIDE	FALSE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.4150804050252529	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	modulator	0.2243917574174979	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
KCND2	hgnc:6238	KCND2	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.1842374429322614	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	ChEMBL	33	inhibitor	2.386712328895204	IMPLITAPIDE	ncit:C65901	IMPLITAPIDE	FALSE	FALSE	FALSE
PNLIP	hgnc:9155	PNLIP	DTC	9/2/20	NULL	13.12691780892362	HOOKEROSIDE A	chembl:CHEMBL505479	HOOKEROSIDE A	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
NCBIGENE:2197	hgnc:3597	FAU	GuideToPharmacology	2024.1	inhibitor	0.2282942227638891	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	3.088686543276147	INCB13739	drugbank:DB05064	INCB13739	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.3547815624033412	Methscopolamine Bromide	rxcui:56092	METHSCOPOLAMINE BROMIDE	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.1802322811293861	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	HYDROCORTISONE PROBUTATE	rxcui:27196	HYDROCORTISONE PROBUTATE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.4167275494896388	GSK-356278	drugbank:DB12542	GSK-356278	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.024593757	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.5834185692854944	MK-0873	drugbank:DB13029	MK-0873	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1635752997996713	LEVOMILNACIPRAN	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.1988926940746003	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	NOBILETIN	iuphar.ligand:12446	NOBILETIN	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	1.458546423213736	IUPHAR.LIGAND:12687	iuphar.ligand:12687	PTD10	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.1121958787087489	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.1408971500063358	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	0.3125456621172291	ALTEPLASE	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.5556367326528517	DIETHYLDITHIOCARBAMATE	rxcui:1427193	DIETHYLDITHIOCARBAMATE	FALSE	FALSE	FALSE
NCBIGENE:281	hgnc:479	AMYP1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1297	iuphar.ligand:1297	[PHE13,TYR19]MCH	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	1.381780822	NALOXONE METHIODIDE	chembl:CHEMBL1514361	NALOXONE METHIODIDE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.007995686	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	1.117184494376478	ATG002	drugbank:DB05068	ATG002	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	LAVENDUSTIN B	ncit:C1616	LAVENDUSTIN B	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.009285176	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.048958202	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	6.300920548	MSX-122	drugbank:DB12715	MSX-122	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.037438625	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.021608095	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TEND	1-Aug-11	NULL	0.097236428	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2580229544751573	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	0.046549354	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.02012945	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.5983780197799943	grepafloxacin	rxcui:83719	GREPAFLOXACIN	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	PharmGKB	4/5/24	NULL	0.6961244292611014	repotrectinib	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.1682938180631233	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:2116	hgnc:3491	ETV2	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	ERYTHROMYCIN LACTOBIONATE	rxcui:24347	ERYTHROMYCIN LACTOBIONATE	TRUE	FALSE	FALSE
FAU	hgnc:3597	FAU	ChEMBL	33	inhibitor	0.064824285	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.052090944	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
SEQUESTOSOME-1 P62	hgnc:11280	SQSTM1	TTD	2020.06.01	NULL	52.50767123569449	IMX-942	chembl:CHEMBL3545314	DUSQUETIDE	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1920	iuphar.ligand:1920	ONO-8711	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:11437	iuphar.ligand:11437	VU0409551	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:9005	iuphar.ligand:9005	AR-M1000390	FALSE	FALSE	FALSE
PLAUR	hgnc:9053	PLAUR	NCI	14-Sep-17	NULL	1.193356164447602	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
NCBIGENE:1827	hgnc:3040	RCAN1	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.082559232	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9706	iuphar.ligand:9706	JWH-018	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.085239726	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.1054370908347279	IUPHAR.LIGAND:67	iuphar.ligand:67	9-OH-RISPERIDONE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.021933029	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	0.6000876712650799	SULFOBROMOPHTHALEIN	rxcui:10212	SULFOBROMOPHTHALEIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.4375639269641209	3,5-DINITROCATECHOL (OR-486)	chembl:CHEMBL168276	3,5-DINITROCATECHOL (OR-486)	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3981	iuphar.ligand:3981	[3H]&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:4112	iuphar.ligand:4112	8-DEOXY-NEODYSIHERBAINE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.013025967	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.3431873936973497	PREMARIN	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	AMINACRINE	rxcui:645	AMINACRINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.006466462	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.030246354	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.1041818873724097	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.006258861	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.007023498	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	PharmGKB	4/5/24	NULL	0.029138552	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
MYOM2	hgnc:7614	MYOM2	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CLORGYLINE HYDROCHLORIDE	chembl:CHEMBL539507	CLORGYLINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.043180651	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.2734774543525755	GRAZOPREVIR	rxcui:1734630	GRAZOPREVIR	TRUE	FALSE	FALSE
POLL	hgnc:9184	POLL	DTC	9/2/20	NULL	1.312691780892362	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
PTPN12	hgnc:9645	PTPN12	DTC	9/2/20	NULL	4.375639269641208	GNF-PF-231	chembl:CHEMBL601167	CHEMBL:CHEMBL601167	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.072927321	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.2381300282797936	IPI-145	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
THYROID PEROXIDASE	hgnc:12015	TPO	TTD	2020.06.01	NULL	2.625383561784725	Propylthiouracil	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.030176823	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
FGF23	hgnc:3680	FGF23	ChEMBL	33	inhibitor	105.0153424713889	BUROSUMAB	rxcui:2043854	BUROSUMAB-TWZA	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	CBP501	ncit:C71529	SERINE/THREONINE KINASE INHIBITOR CBP501	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.016992774	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
LIPA	hgnc:6617	LIPA	NCI	14-Sep-17	NULL	0.7955707762984016	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
NCBIGENE:1274	hgnc:4855	HDC	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:5189	iuphar.ligand:5189	FMH	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.061055432	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.1411496538593938	CERDULATINIB	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.010082118	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.066297565	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:5683	iuphar.ligand:5683	GSK-1838705A	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	AZD-7762	drugbank:DB12242	AZD-7762	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.034658529	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.8468979231563628	PHYTOESTROGEN	ncit:C1194	PHYTOESTROGEN	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.086551106	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:4197	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	DIPHENHYDRAMINE	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.8468979231563628	ROPSACITINIB	ncit:C180657	ROPSACITINIB	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.546954909	deferasirox	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
CCR1	hgnc:1602	CCR1	ChEMBL	33	inhibitor	5.834185692854944	CCX354	iuphar.ligand:10164	CCX354	FALSE	FALSE	FALSE
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	KAPPAPROCT	chembl:CHEMBL5095448	COBITOLIMOD SODIUM	FALSE	FALSE	FALSE
RPS18	hgnc:10401	RPS18	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.05792352	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	2.282942227638891	lovastatin acid	ncit:C77442	LOVASTATIN ACID	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.058471794	HE3235	chembl:CHEMBL3545237	HE3235	FALSE	FALSE	FALSE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516874	IUPHAR.LIGAND:8937	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	12-HYDROXY-4,4-BISNOR-4,8,11,13-PODOCARPATETRAEN-3-ONE	chembl:CHEMBL1358735	12-HYDROXY-4,4-BISNOR-4,8,11,13-PODOCARPATETRAEN-3-ONE	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.596678082	COBIMETINIB FUMARATE	rxcui:1722380	COBIMETINIB FUMARATE	TRUE	FALSE	FALSE
ESRRG	hgnc:3474	ESRRG	ChEMBL	33	inhibitor	0.6250913242344582	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
RPL32	hgnc:10336	RPL32	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
A2M	hgnc:7	A2M	NCI	14-Sep-17	NULL	0.055010656	PROSTAGLANDIN E1	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.42006137	ALEGLITAZAR	ncit:C72687	ALEGLITAZAR	FALSE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.3251536612259921	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.087903467	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:11972	iuphar.ligand:11972	ULEVOSTINAG	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	CGI	2/1/22	NULL	0.108374966	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.085796848	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	MyCancerGenome	20-Jun-17	inhibitor	0.364636606	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
NCBIGENE:2010	hgnc:3331	EMD	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8127	iuphar.ligand:8127	COMPOUND 3B [PMID: 23454515]	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.016856395	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.008789366	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	TRICLOCARBAN	rxcui:38609	TRICLOCARBAN	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	0.7721716358190367	SAR-407899	iuphar.ligand:8910	SAR407899	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.091796628	IUPHAR.LIGAND:516	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	AVE-9940	chembl:CHEMBL3545117	AVE-9940	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	2.187819634820604	BECATECARIN	ncit:C1620	BECATECARIN	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.011284692	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	TCMDC-123828	chembl:CHEMBL588804	CHEMBL:CHEMBL588804	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.058602312	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	PharmGKB	4/5/24	NULL	0.029301156	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1479089330582944	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
FGF22	hgnc:3679	FGF22	DTC	9/2/20	NULL	0.4688184931758437	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
TTR	hgnc:12405	TTR	PharmGKB	4/5/24	NULL	17.50255707856483	inotersen	rxcui:2099289	INOTERSEN	TRUE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	3.750547945	BOSENTAN	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.1245241215075758	durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
ALPHA-GLUCOSIDASE	hgnc:4296	GLA	TTD	2020.06.01	NULL	2.019525817	Anamorelin	ncit:C52197	ANAMORELIN	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.049723174	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.03729238	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:11435	iuphar.ligand:11435	[125I]BANTAG-1	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:5944	iuphar.ligand:5944	CDK1 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.054695491	IUPHAR.LIGAND:7882	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.1325951293830669	IUPHAR.LIGAND:4090	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.2536602475154323	IUPHAR.LIGAND:4066	iuphar.ligand:4066	(+)-HA966	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4866	iuphar.ligand:4866	ANANTIN	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	activator	0.1041818873724097	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:8123	iuphar.ligand:8123	COMPOUND 1D [PMID: 21493067]	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	MS417	iuphar.ligand:7512	MS417	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DNDI1246786	chembl:CHEMBL1863271	CHEMBL:CHEMBL1863271	FALSE	FALSE	FALSE
CRP	hgnc:2367	CRP	PharmGKB	4/5/24	NULL	0.546954909	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278864	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:7399	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
UNIPROT:Q13370	hgnc:8779	PDE3B	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	NM-702	drugbank:DB05505	NM-702	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:7914	iuphar.ligand:7914	BV-6	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	0.059330702	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	inhibitor	4.200613699	CTCE-9908	drugbank:DB05625	CTCE-9908	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	TRANYLCYPROMINE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:4778	iuphar.ligand:4778	SSR-103800	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	TORSEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
KRTAP10-4	hgnc:20521	KRTAP10-4	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	(R)-FLECAINIDE	chembl:CHEMBL398673	(R)-FLECAINIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	TDR84367	chembl:CHEMBL1485420	CHEMBL:CHEMBL1485420	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	BIFEMELANE	rxcui:47111	BIFEMELANE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.013673873	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	TDR77593	chembl:CHEMBL1510164	CHEMBL:CHEMBL1510164	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.006643177	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.052090944	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	agonist	2.625383561784724	DASIGLUCAGON HYDROCHLORIDE	rxcui:2535234	DASIGLUCAGON HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TdgClinicalTrial	Jan-14	NULL	4.200613699	RISEDRONATE	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:12893	iuphar.ligand:12893	ZELNECIRNON	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.022789788	IUPHAR.LIGAND:5702	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:10151	iuphar.ligand:10151	NEOLYMPHOSTIN A	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.049723174	Panobinostat	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.013408496	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.082043236	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.069043618	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.1902451856365742	NSC-48300	chembl:CHEMBL1091971	CHEMBL:CHEMBL1091971	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	SJ000082806	chembl:CHEMBL494668	CHEMBL:CHEMBL494668	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	DTC	9/2/20	NULL	0.4375639269641208	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.012573676	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.029057925	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:2087	ncbigene:2087	ERVK2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12336	iuphar.ligand:12336	COMPOUND 5I [PMID: 36542759]	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	1.105424657593568	Debio 1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	1-O-ACETYLGEOPYXIN A	chembl:CHEMBL1902074	CHEMBL:CHEMBL1902074	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.04339477	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:8367	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
BIRC6	hgnc:13516	BIRC6	TALC	12-May-16	inhibitor	3.750547945406749	LCL161	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
HTR7	hgnc:5302	HTR7	ChEMBL	33	inhibitor	1.750255707856483	JNJ-18038683	iuphar.ligand:8432	JNJ-18038683	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	NULL	1.221108633388244	IUPHAR.LIGAND:9247	rxcui:2669799	VAMOROLONE	TRUE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	1.615620653405984	AS101	iuphar.ligand:437	AS101	FALSE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.100589408	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.4730420832044549	FAMOTIDINE	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.092118721	IUPHAR.LIGAND:168	iuphar.ligand:168	VER-3323	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1630673019742065	IUPHAR.LIGAND:7219	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	NULL	0.1268301237577161	IUPHAR.LIGAND:4748	ncit:C47521	ESTROPIPATE	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:5701	iuphar.ligand:5701	PI-103	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.2381300282797936	2,5-BIS(4-MORPHOLINOSTYRYL)PYRAZINE	chembl:CHEMBL2181041	CHEMBL:CHEMBL2181041	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.789589041	DIETHYLDITHIOCARBAMATE	rxcui:1427193	DIETHYLDITHIOCARBAMATE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	GNF-PF-310	chembl:CHEMBL600719	CHEMBL:CHEMBL600719	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.2778183663264258	AZD8108	chembl:CHEMBL3707355	AZD8108	FALSE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	ChEMBL	33	blocker	0.089298761	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.012695278	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:7250	rxcui:7688	METAPROTERENOL	TRUE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.4070362111294147	IUPHAR.LIGAND:12647	iuphar.ligand:12647	ACT-709478	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.596678082	mexiletine	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TEND	1-Aug-11	NULL	0.8334550989792776	ARDEPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
DNTT	hgnc:2983	DNTT	NCI	14-Sep-17	NULL	2.187819634820604	ACYCLOVIR	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.375054795	SU-11274	iuphar.ligand:5057	SU11274	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002737341	TRIAMCINOLONE ACETONIDE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	TCMDC-125000	chembl:CHEMBL579742	CHEMBL:CHEMBL579742	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.059532507	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	TCMDC-124573	chembl:CHEMBL525826	CHEMBL:CHEMBL525826	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.100976291	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.032016873	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
CDK18	hgnc:8751	CDK18	ChEMBL	33	inhibitor	0.4375639269641208	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.2717788366236775	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
MME	hgnc:7154	MME	ChEMBL	33	inhibitor	4.773424657790408	RACECADOTRIL	rxcui:16738	RACECADOTRIL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	(-)-U-50488 METHANE SULFONATE	chembl:CHEMBL1513237	(-)-U-50488 METHANE SULFONATE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.035502144	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	NCI	14-Sep-17	NULL	0.03821519	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
BTF3L1	hgnc:1126	BTF3P11	NCI	14-Sep-17	NULL	0.8751278539282417	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SPIPERONE HYDROCHLORIDE	chembl:CHEMBL1256875	SPIPERONE HYDROCHLORIDE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.8140724222588294	Metaproterenol Sulfate	rxcui:6804	METAPROTERENOL SULFATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	SB-408124	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.1209854175937661	AZD8108	chembl:CHEMBL3707355	AZD8108	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	2.838252499226729	CASOPITANT	ncit:C71635	CASOPITANT	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	ChEMBL	33	inhibitor	0.3182283105193606	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
UNIPROT:Q01344	hgnc:6017	IL5RA	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	BENRALIZUMAB	rxcui:1989100	BENRALIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P07948	hgnc:6735	LYN	TdgClinicalTrial	Jan-14	NULL	0.1544343271638073	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
CAMKK2	hgnc:1470	CAMKK2	DTC	9/2/20	NULL	0.1039755866053356	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.048394167	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.02804897	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.057878826	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	CID 100335	chembl:CHEMBL1520346	CHEMBL:CHEMBL1520346	FALSE	FALSE	FALSE
UNIPROT:O43497	hgnc:1394	CACNA1G	TEND	1-Aug-11	NULL	0.3977853881492008	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	NSC-353263	chembl:CHEMBL1383812	CHEMBL:CHEMBL1383812	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	ChEMBL	33	inhibitor	0.9723642821424907	BERZOSERTIB	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
RPS10	hgnc:10383	RPS10	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.375054795	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.3241214273808302	NS-2359	drugbank:DB05805	NS-2359	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.068037151	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.059481927	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:390	iuphar.ligand:390	MRE 2029F20	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	modulator	0.5413161983061289	IUPHAR.LIGAND:12483	iuphar.ligand:12483	MRS8054	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:10530	iuphar.ligand:10530	BSJ-03-204	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.028866229	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.3559842117674203	AMIFOSTINE	rxcui:1545987	AMIFOSTINE ANHYDROUS	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.577007376	PENICILLAMINE	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	0.8751278539282416	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	PharmGKB	4/5/24	NULL	0.6563458904461813	margetuximab	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
BIFUNCTIONAL AMINOACYL-TRNA SYNTHETASE	hgnc:3418	EPRS1	TTD	2020.06.01	NULL	17.50255707856483	HT-100	ncit:C1120	HALOFUGINONE	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE ENDOTHELIAL	hgnc:7876	NOS3	TTD	2020.06.01	NULL	1.875273972703375	VAS-203	ncit:C152249	RONOPTERIN	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	5.250767123569449	Pomaglumetad	chembl:CHEMBL375611	LY404039	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1060761035064535	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.041393513	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.1682938180631234	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	DIHYDROSPINGOSINE	iuphar.ligand:2453	DIHYDROSPHINGOSINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.008824819	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
TBP	hgnc:11588	TBP	NCI	14-Sep-17	NULL	0.7955707762984016	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	2.493675356344019	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1909369863116163	ETRAVIRINE	rxcui:475969	ETRAVIRINE	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.046965717	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	DILMAPIMOD	ncit:C96531	DILMAPIMOD	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.058471794	DAROLUTAMIDE	rxcui:2180325	DAROLUTAMIDE	TRUE	FALSE	TRUE
COCH	hgnc:2180	COCH	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.7395446652914718	INTERLEUKIN-1 RECEPTOR ANTAGONIST	ncit:C2486	RECOMBINANT INTERLEUKIN-1 RECEPTOR ANTAGONIST	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	GNF-PF-1577	chembl:CHEMBL600315	CHEMBL:CHEMBL600315	FALSE	FALSE	FALSE
NCBIGENE:2065	hgnc:3431	ERBB3	GuideToPharmacology	2024.1	inhibitor	1.029562181092049	IUPHAR.LIGAND:12376	iuphar.ligand:12376	DARIZMETINIB	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:12155	iuphar.ligand:12155	ZASOCITINIB	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2273059360852575	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.032412143	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	ChEMBL	33	blocker	0.085378327	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.0504235	SAPANISERTIB	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.084146909	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
RPL13A	hgnc:10304	RPL13A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.091850154	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:194	iuphar.ligand:194	SB 243213	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3889457128569963	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:10059	iuphar.ligand:10059	MIRICORILANT	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1988	iuphar.ligand:1988	RELAXIN-1	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.074426182	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	NSC-677438	chembl:CHEMBL118678	CHEMBL:CHEMBL118678	FALSE	FALSE	FALSE
KLC1	hgnc:6387	KLC1	PharmGKB	4/5/24	NULL	0.9460841664089098	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1734	drugbank:DB04005	URIDINE 5'-TRIPHOSPHATE	FALSE	FALSE	FALSE
ANXA5	hgnc:543	ANXA5	NCI	14-Sep-17	NULL	0.2019525816757481	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.018295356	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1981421556063943	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
MOTHERS AGAINST DECAPENTAPLEGIC HOMOLOG 7	hgnc:6773	SMAD7	TTD	2020.06.01	NULL	13.12691780892362	GED-0301	iuphar.ligand:8277	MONGERSEN	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:7416	ncit:C66578	TANAPROGET	FALSE	FALSE	FALSE
DBI	hgnc:2690	DBI	NCI	14-Sep-17	NULL	0.7955707762984016	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.043137707	Desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CANRENONE	rxcui:1982	CANRENONE	TRUE	FALSE	FALSE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	modulator	0.1442518440541058	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3856	iuphar.ligand:3856	AVA5	FALSE	FALSE	FALSE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	2.000292237550266	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.013792401	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016780975	IPRONIAZID	rxcui:5981	IPRONIAZID	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.4730420832044549	ARTESUNATE	rxcui:18346	ARTESUNATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.056826484	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:63	hgnc:136	ACTBP3	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:3648	iuphar.ligand:3648	BETA-DEFENSIN 4A	FALSE	FALSE	FALSE
NCBIGENE:682	hgnc:1116	BSG	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:12496	drugbank:DB03694	N-PHENYLTHIOUREA	FALSE	FALSE	FALSE
NCBIGENE:2055	hgnc:2079	CLN8	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8119	iuphar.ligand:8119	COMPOUND 35 [PMID: 22902653]	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.011971653	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1207072901969988	NSC-119236	chembl:CHEMBL458765	CHEMBL:CHEMBL458765	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.057700738	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.057912873	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.030176823	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
MISP	hgnc:27000	MISP	PharmGKB	4/5/24	NULL	0.3241214273808302	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:3143	ncbigene:3143	HMAA	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11264	rxcui:1311506	GLYCYRRHETINIC ACID	TRUE	FALSE	FALSE
F8	hgnc:3546	F8	PharmGKB	4/5/24	NULL	0.3431873936973497	desmopressin	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	4.286340509036285	CDP-6038	ncit:C172654	OLOKIZUMAB	FALSE	FALSE	FALSE
TP53AIP1	hgnc:29984	TP53AIP1	PharmGKB	4/5/24	NULL	0.9723642821424908	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.2287915957982331	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
HBA1	hgnc:4823	HBA1	ChEMBL	33	negative modulator	8.751278539282415	EFAPROXIRAL	ncit:C1435	EFAPROXIRAL	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	INEBILIZUMAB	rxcui:2373950	INEBILIZUMAB-CDON	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.3697723326457359	BAY-1125976	chembl:CHEMBL4751394	BAY-1125976	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	positive modulator	2.983390411119005	IVACAFTOR	rxcui:1243041	IVACAFTOR	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	ChEMBL	33	inhibitor	0.4487835148349957	CC-401	drugbank:DB12432	CC-401	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.49187514	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
NCBIGENE:2719	hgnc:4451	GPC3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8641	iuphar.ligand:8641	COMPOUND 60 [PMID: 26155854]	FALSE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	MyCancerGenome	20-Jun-17	other/unknown	0.4773424657790409	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:11064	iuphar.ligand:11064	(S)-CR8	FALSE	FALSE	FALSE
NCBIGENE:85	ncbigene:85	ACTL5	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:11514	iuphar.ligand:11514	CVN424	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.067317527	IUPHAR.LIGAND:7791	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	1.591141552596803	CPI-1205	drugbank:DB14581	CPI-1205	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.050294704	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.3454452054979901	FILGRASTIM	rxcui:1433764	TBO-FILGRASTIM	TRUE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.039331589	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
PAEP	hgnc:8573	PAEP	NCI	14-Sep-17	NULL	0.6035364509849942	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	(E)-DIBENZYLIDENEACETONE	chembl:CHEMBL17201	CHEMBL:CHEMBL17201	FALSE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.031822831	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	PharmGKB	4/5/24	NULL	0.041672755	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	MGBG	ncit:C661	MITOGUAZONE	FALSE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	0.077789143	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.08914715	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:5872	iuphar.ligand:5872	JMV3008	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1682938180631233	VABICASERIN HYDROCHLORIDE	ncit:C142993	VABICASERIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	modulator	0.2019525816757481	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	ChEMBL	33	inhibitor	6.563458904461812	ATACICEPT	ncit:C81166	ATACICEPT	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003262967	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:9387	iuphar.ligand:9387	CEP-33779	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	DIPHENYLSULFANE	chembl:CHEMBL219876	DIPHENYLSULFANE	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1640864726115453	BALSALAZIDE	rxcui:18747	BALSALAZIDE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.059397818	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.042276708	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.2573905452730122	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	BMS-817378	chembl:CHEMBL3545050	BMS-817378	FALSE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11365	iuphar.ligand:11365	DX-9065A	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	DICLOFENAC ETALHYALURONATE SODIUM	ncit:C174668	DICLOFENAC ETALHYALURONATE SODIUM	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.023110771	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.217423069	Glucarpidase	rxcui:1242127	GLUCARPIDASE	TRUE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.4688184931758437	AFURESERTIB	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	modulator	0.2243917574174979	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	CIViC	10-Apr-24	NULL	0.019138936	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:8958	iuphar.ligand:8958	LIFIRAFENIB	FALSE	FALSE	FALSE
NCBIGENE:515	hgnc:840	ATP5PB	GuideToPharmacology	2024.1	blocker	0.8751278539282418	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2266	iuphar.ligand:2266	N-STEARYL-[NLE17] NEUROTENSIN-(6-11)/VIP-(7-28)	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	TRIADIMEFON	chembl:CHEMBL520897	TRIADIMEFON	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.1182605208011137	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.038104261	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:746	hgnc:1164	TMEM258	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.222962511	ELDECALCITOL	ncit:C87291	ELDECALCITOL	FALSE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.4167275494896388	LGD-1550	drugbank:DB05785	LGD-1550	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1562728310586145	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:118	iuphar.ligand:118	[3H]ELETRIPTAN	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.061376588	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	5.250767123569449	CCR5 mab	drugbank:DB05906	CCR5 MAB	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.086361301	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.022789788	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.1785975212098452	MAPK INHIBITORS	ncit:C2149	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.008382451	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.001023541	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	CIS-(Z)-FLUPENTHIXOL DIHYDROCHLORIDE	chembl:CHEMBL1256995	CHEMBL:CHEMBL1256995	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	1.084869240406911	Montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	PF-03715455	drugbank:DB12138	PF-03715455	FALSE	FALSE	FALSE
ACACB	hgnc:85	ACACB	ChEMBL	33	negative modulator	0.4234489615781814	FIRSOCOSTAT	ncit:C169983	FIRSOCOSTAT	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10442	iuphar.ligand:10442	UDM-001651	FALSE	FALSE	FALSE
NCBIGENE:3171	hgnc:5023	FOXA3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11401	iuphar.ligand:11401	BJP-06-005-3	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:9368	iuphar.ligand:9368	CX-6258	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1014640990061729	Brentuximab vedotin	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.021286894	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2365210416022274	Miransertib	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	4-DODECYL-PHENOL	chembl:CHEMBL194881	CHEMBL:CHEMBL194881	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.041972559	HMAF	ncit:C1717	IROFULVEN	FALSE	FALSE	FALSE
UNIPROT:Q969P6	hgnc:29787	TOP1MT	TEND	1-Aug-11	NULL	0.84012274	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	TCMDC-125086	chembl:CHEMBL532504	CHEMBL:CHEMBL532504	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PENCONAZOLE	rxcui:2593184	PENCONAZOLE	FALSE	FALSE	FALSE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	3.088686543276147	Retosiban	ncit:C76681	RETOSIBAN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.008214592	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.1193356164447602	Tetrodotoxin	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
PYGL	hgnc:9725	PYGL	PharmGKB	4/5/24	NULL	0.2344092465879218	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	modulator	0.2243917574174979	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.091636424	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.091850154	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.085239726	GW9662	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.078252863	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.6105543166941221	AZD-3043	drugbank:DB12576	AZD-3043	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1232574442152452	KRN633	iuphar.ligand:6057	VEGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.4234489615781814	BENZYL SALICYLATE	rxcui:1362907	BENZYL SALICYLATE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1562728310586145	MEVASTATIN	ncit:C96285	MEVASTATIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:75	iuphar.ligand:75	SB 272183	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.065125794	IUPHAR.LIGAND:6963	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	0.1164249916534246	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GNF-PF-2713	chembl:CHEMBL578719	CHEMBL:CHEMBL578719	FALSE	FALSE	FALSE
UNIPROT:P61073	hgnc:2561	CXCR4	TEND	1-Aug-11	NULL	3.850562557284263	PLERIXAFOR	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.1526385791735305	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
TNFSF11	hgnc:11926	TNFSF11	ChEMBL	33	inhibitor	43.75639269641208	DENOSUMAB	rxcui:993449	DENOSUMAB	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.013560866	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1562728310586145	BLM	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	2.763561643983921	MART1	ncit:C28724	MART-1 ANTIGEN	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3659	iuphar.ligand:3659	[125I]CXCL5 (HUMAN)	FALSE	FALSE	FALSE
INTERLEUKIN-18	hgnc:5986	IL18	TTD	2020.06.01	NULL	5.527123287967842	MEDI-2338	chembl:CHEMBL2109604	CAMOTESKIMAB	FALSE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	DTC	9/2/20	NULL	0.2059124362184098	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.1795134059339982	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.1312691780892362	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	SJ000012773	chembl:CHEMBL589715	CHEMBL:CHEMBL589715	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.070574827	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	MMV006513	chembl:CHEMBL585622	CHEMBL:CHEMBL585622	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	DIFLORASONE DIACETATE	rxcui:23033	DIFLORASONE DIACETATE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:451	iuphar.ligand:451	XCC	FALSE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	1.346350544504987	TOLCAPONE	rxcui:72937	TOLCAPONE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.023080295	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006286838	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.3231241306811969	DAPIPRAZOLE	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1478	iuphar.ligand:1478	EFWSLAAPQRF-NH2	FALSE	FALSE	FALSE
PSMD2	hgnc:9559	PSMD2	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ITGA2B	hgnc:6138	ITGA2B	ChEMBL	33	inhibitor	2.187819634820604	TADOCIZUMAB	ncit:C88626	TADOCIZUMAB	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	DIETHYLCARBAMAZINE CITRATE	rxcui:203175	DIETHYLCARBAMAZINE CITRATE	TRUE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5563	iuphar.ligand:5563	CID1792197	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.008287196	TRIMIPRAMINE	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.027752469	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	BENOXINATE	rxcui:18889	BENOXINATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	BUFOGENIN	ncit:C77829	BUFOGENIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	CYCLOASPEPTIDE A	chembl:CHEMBL473074	CYCLOASPEPTIDE A	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	CancerCommons	25-Jul-13	inhibitor	0.4828291607879953	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
IMPDH2	hgnc:6053	IMPDH2	ChEMBL	33	inhibitor	1.312691780892362	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
FGR	hgnc:3697	FGR	ChEMBL	33	inhibitor	0.1315981735230438	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3596415838061266	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
UNIPROT:O43613	hgnc:4848	HCRTR1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	ALMOREXANT	ncit:C87423	ALMOREXANT	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.017549355	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:7923	iuphar.ligand:7923	UCM 765	FALSE	FALSE	FALSE
CALMODULIN	hgnc:14986	SNAP91	TTD	2020.06.01	NULL	0.5834185692854944	Trifluoperazine	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2689	iuphar.ligand:2689	L-796449	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	0.2734774543525755	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.021933029	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.729273212	TYRPHOSTIN A25	ncit:C1484	TYRPHOSTIN A25	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.060353645	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.2263261691193728	BERUBICIN HYDROCHLORIDE	ncit:C61568	BERUBICIN HYDROCHLORIDE	FALSE	FALSE	FALSE
RPS13	hgnc:10386	RPS13	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
UNIPROT:P33681	hgnc:1700	CD80	TEND	1-Aug-11	NULL	5.250767123569449	ABATACEPT	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	NORBINALTORPHIMINE	iuphar.ligand:1642	NOR-BINALTORPHIMINE	FALSE	FALSE	FALSE
RTN4	hgnc:14085	RTN4	ChEMBL	33	inhibitor	10.50153424713889	OZANEZUMAB	ncit:C166450	OZANEZUMAB	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.078194596	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TdgClinicalTrial	Jan-14	NULL	0.7095631248066824	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.130291988	IUPHAR.LIGAND:7476	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.030246354	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.021149706	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	PharmGKB	4/5/24	NULL	0.030483409	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
EPHX2	hgnc:3402	EPHX2	DTC	9/2/20	NULL	0.750109589	ALOE-EMODIN	chembl:CHEMBL40275	ALOE-EMODIN	FALSE	FALSE	FALSE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	0.4375639269641208	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
ETV6	hgnc:3495	ETV6	NCI	14-Sep-17	NULL	2.917092846427472	L-ASPARAGINASE	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.6543011991986852	PHENTERMINE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
NCBIGENE:2844	hgnc:4476	GPR21	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11781	iuphar.ligand:11781	AZD4320	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	inhibitor	0.038159645	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
NCBIGENE:932	hgnc:7317	MS4A3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4583	iuphar.ligand:4583	(R/S) EF-1500	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:4090	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.015521038	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	0.1014640990061729	Brentuximab Vedotin	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007063179	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.1715936968486748	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.05387244	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.026748686	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	FUSARIC ACID	chembl:CHEMBL24510	FUSARIC ACID	FALSE	FALSE	FALSE
AANAT	hgnc:19	AANAT	NCI	14-Sep-17	NULL	0.035098711	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.011786234	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	CIViC	10-Apr-24	NULL	0.060353645	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:6952	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.005184407	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	POTASSIUM DICHROMATE	rxcui:8595	POTASSIUM DICHROMATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	OLPRINONE	ncit:C90918	OLPRINONE	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.2108741816694558	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	1.381780822	ARGATROBAN	rxcui:15202	ARGATROBAN	TRUE	FALSE	FALSE
UNIPROT:O95373	hgnc:9852	IPO7	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.005864158	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
KIT	hgnc:6342	KIT	CancerCommons	25-Jul-13	inhibitor	0.2711239478607289	PLX3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CGI	2/1/22	NULL	0.035982643	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CGI	2/1/22	NULL	0.064318974	Bicalutamide	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.8008364246019593	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	CGI	2/1/22	NULL	0.2592971419046642	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CGI	2/1/22	NULL	0.018572323	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.4234489615781814	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CGI	2/1/22	NULL	0.099446347	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.083016081	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.020164236	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.0296486	PROCHLORPERAZINE MALEATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	ChEMBL	33	agonist	3.281729452230906	LH (MENOTROPINS)	chembl:CHEMBL1201697	LH (MENOTROPINS)	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.025942525	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.8899605294185507	OLMESARTAN MEDOXOMIL	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
CALCR	hgnc:1440	CALCR	ChEMBL	33	agonist	13.12691780892362	CALCITONIN SALMON RECOMBINANT	rxcui:36118	SALMON CALCITONIN	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.069454592	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	1.166837138570988	PALONOSETRON HYDROCHLORIDE	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ChEMBL	33	inhibitor	0.5373592085524291	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
ALDH5A1	hgnc:408	ALDH5A1	ChEMBL	33	inhibitor	7.501095891	VALPROATE SODIUM	rxcui:9919	SODIUM VALPROATE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.4243044140258141	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.7721716358190367	NARATRIPTAN HYDROCHLORIDE	rxcui:236690	NARATRIPTAN HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	agonist	0.3860858179095183	LORCASERIN HYDROCHLORIDE	rxcui:1300700	LORCASERIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.037363144	ZIPRASIDONE MESYLATE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.022606632	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1262203635473425	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.006643177	HALOPERIDOL DECANOATE	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.032173818	QUETIAPINE FUMARATE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.037363144	ZIPRASIDONE HYDROCHLORIDE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
KLKB1	hgnc:6371	KLKB1	ChEMBL	33	inhibitor	11.25164383622025	ECALLANTIDE	rxcui:658708	ECALLANTIDE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.1250182648468916	CHLOROTRIANISENE	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	4.039051633514961	FILGRASTIM	rxcui:1433764	TBO-FILGRASTIM	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.077217164	LOXAPINE HYDROCHLORIDE	rxcui:91138	LOXAPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	3.454452054979901	EPLERENONE	rxcui:298869	EPLERENONE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.042504861	METHADONE HYDROCHLORIDE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1715936968486748	BUPROPION HYDROBROMIDE	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	FENTANYL HYDROCHLORIDE	rxcui:1652097	FENTANYL HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	HYDROCORTAMATE HYDROCHLORIDE	ncit:C65863	HYDROCORTAMATE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	BETAMETHASONE SODIUM PHOSPHATE	rxcui:203220	BETAMETHASONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	1.029562181092048	NEOSTIGMINE METHYLSULFATE	rxcui:7315	NEOSTIGMINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	DEXAMETHASONE SODIUM PHOSPHATE	rxcui:48933	DEXAMETHASONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	BETAMETHASONE DIPROPIONATE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	CICLESONIDE	rxcui:274964	CICLESONIDE	TRUE	FALSE	FALSE
CD2	hgnc:1639	CD2	ChEMBL	33	inhibitor	11.66837138570988	ALEFACEPT	rxcui:299635	ALEFACEPT	TRUE	TRUE	FALSE
MGAM	hgnc:7043	MGAM	ChEMBL	33	inhibitor	3.182283105193605	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	0.9334697108567911	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.3125456621172291	ESTROGENS, ESTERIFIED	rxcui:214549	ESTROGENS, ESTERIFIED (USP)	TRUE	FALSE	FALSE
ITGA2B	hgnc:6138	ITGA2B	ChEMBL	33	inhibitor	3.646366058	ABCIXIMAB	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
MTNR1A	hgnc:7463	MTNR1A	ChEMBL	33	agonist	7.501095891	RAMELTEON	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.2692701089009974	METHOXAMINE HYDROCHLORIDE	rxcui:203187	METHOXAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.6563458904461812	NEPAFENAC	rxcui:298665	NEPAFENAC	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1158257453728555	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.057912873	DICLOFENAC SODIUM	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1158257453728555	NAPROXEN SODIUM	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.4039051633514962	NITRIC OXIDE	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.3500511415712967	NITRIC OXIDE	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.5834185692854945	NITRIC OXIDE	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.092443083	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	1.795134059339982	ISOCARBOXAZID	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.305277158	DILTIAZEM MALATE	rxcui:81999	DILTIAZEM MALATE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.07631929	DILTIAZEM HYDROCHLORIDE	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	ChEMBL	33	inhibitor	0.7955707762984014	TRIMETHAPHAN CAMSYLATE	rxcui:38680	TRIMETHAPHAN CAMSYLATE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.078136416	BOCEPREVIR	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.3860858179095183	RIVASTIGMINE TARTRATE	rxcui:994808	RIVASTIGMINE TARTRATE	TRUE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	ChEMBL	33	inhibitor	2.187819634820604	TRIMETHAPHAN CAMSYLATE	rxcui:38680	TRIMETHAPHAN CAMSYLATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.035982643	ENZALUTAMIDE	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	2.386712328895204	INAMRINONE LACTATE	rxcui:91236	INAMRINONE LACTATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.1356787370431382	TIMOLOL MALEATE	rxcui:42933	TIMOLOL MALEATE	TRUE	FALSE	FALSE
MTTP	hgnc:7467	MTTP	ChEMBL	33	inhibitor	5.250767123569449	LOMITAPIDE MESYLATE	rxcui:1364478	LOMITAPIDE MESYLATE	TRUE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	ChEMBL	33	inhibitor	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB11	hgnc:31963	PSMB11	ChEMBL	33	inhibitor	0.4375639269641209	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD12	hgnc:9557	PSMD12	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
CNR1	hgnc:2159	CNR1	ChEMBL	33	agonist	3.500511415712966	NABILONE	rxcui:31447	NABILONE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.6250913242344582	METOCURINE IODIDE	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.3409589041278864	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.6250913242344582	ATRACURIUM BESYLATE	rxcui:1219	ATRACURIUM BESYLATE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.3947945205691315	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.4605936073306534	METOCURINE IODIDE	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.3750547945406749	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.4605936073306534	ATRACURIUM BESYLATE	rxcui:1219	ATRACURIUM BESYLATE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.5357925636295356	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.081030357	METHAMPHETAMINE HYDROCHLORIDE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.1785975212098452	ETRETINATE	rxcui:4182	ETRETINATE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
KCNC1	hgnc:6233	KCNC1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.003648646	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNC2	hgnc:6234	KCNC2	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNA3	hgnc:6221	KCNA3	ChEMBL	33	blocker	0.1829535583125243	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNG3	hgnc:18306	KCNG3	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH7	hgnc:18863	KCNH7	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH4	hgnc:6253	KCNH4	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNB1	hgnc:6231	KCNB1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH6	hgnc:18862	KCNH6	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH3	hgnc:6252	KCNH3	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	3.889457128569962	OBINUTUZUMAB	rxcui:974779	OBINUTUZUMAB	TRUE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	positive modulator	1.615620653405984	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
PDE1A	hgnc:8774	PDE1A	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE6B	hgnc:8786	PDE6B	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.025390557	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE8A	hgnc:8793	PDE8A	ChEMBL	33	inhibitor	0.1241316104862754	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.057912873	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.031032903	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.008866544	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE6H	hgnc:8790	PDE6H	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.2041114528112516	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	1.093909817410302	PEGINTERFERON BETA-1A	rxcui:1546168	PEGINTERFERON BETA-1A	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	0.7095631248066824	NETUPITANT	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.1325951293830669	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.1290114772375786	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.017059022	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
PTGIR	hgnc:9602	PTGIR	ChEMBL	33	agonist	5.625821918110125	SELEXIPAG	rxcui:1729002	SELEXIPAG	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.029090123	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
SRMS	hgnc:11298	SRMS	ChEMBL	33	inhibitor	0.3454452054979901	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.019461702	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.046840028	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	ChEMBL	33	inhibitor	0.076765601	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.045304289	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.058471794	HE3235	chembl:CHEMBL3545237	HE3235	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.058471794	GSK2849466	chembl:CHEMBL3545046	GSK2849466	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.020268015	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.081030357	4SC-203	drugbank:DB12669	4SC-203	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.010777437	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.006375385	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RORC	hgnc:10260	RORC	ChEMBL	33	inhibitor	0.5707355569097228	JTE-151	chembl:CHEMBL3545357	JTE-151	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.010777437	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CDK12	hgnc:24224	CDK12	ChEMBL	33	inhibitor	0.1458546423213736	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
PIM2	hgnc:8987	PIM2	ChEMBL	33	inhibitor	2.187819634820604	AZD-1208	chembl:CHEMBL3545423	AZD-1208	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	ChEMBL	33	inhibitor	0.1342907192728759	AZD-1080	chembl:CHEMBL1969664	AZD-1080	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1848861663228679	BMS-817378	chembl:CHEMBL3545050	BMS-817378	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.596678082	BALAMAPIMOD	ncit:C76769	BALAMAPIMOD	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.2025758921130189	SERABELISIB	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.2612321952024601	MK-6592	chembl:CHEMBL3545378	MK-6592	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	ChEMBL	33	inhibitor	1.093909817410302	MK-8033	chembl:CHEMBL2323775	MK-8033	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.093763699	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	1.250182648468916	RG7893	chembl:CHEMBL3707353	RG7893	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.089298761	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.108711535	AZD8108	chembl:CHEMBL3707355	AZD8108	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.1136529680426287	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.057700738	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.04464938	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	modulator	0.2004109589148645	DAGROCORAT	ncit:C174807	DAGROCORAT	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.42006137	EFATUTAZONE HYDROCHLORIDE	chembl:CHEMBL3545279	EFATUTAZONE HYDROCHLORIDE	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	ChEMBL	33	inhibitor	0.08607815	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
PRKD1	hgnc:9407	PRKD1	ChEMBL	33	inhibitor	0.08607815	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	CP-778875	chembl:CHEMBL3545276	CP-778875	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	ChEMBL	33	inhibitor	0.035865896	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.071341945	PEFICITINIB	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.5000730593875666	AMG-337	drugbank:DB15639	AMG-337	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.2112984757975633	AFURESERTIB	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.2381300282797936	DUVELISIB	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.073954467	UPROSERTIB	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.1154014752432845	DUVELISIB	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.49187514	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.4518732464345482	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1852122442176172	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.2500365296937833	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.5707355569097228	R-333	chembl:CHEMBL3545159	R-333	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.2500365296937833	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.2711239478607289	PEXIDARTINIB	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	SAR-407899	iuphar.ligand:8910	SAR407899	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.2869271652223742	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	1.419126249613364	DNK333	chembl:CHEMBL105060	DNK333	FALSE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.3182283105193606	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	PF-03654764	drugbank:DB12360	PF-03654764	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.8514757497680189	VIPADENANT	ncit:C152892	VIPADENANT	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	JNJ-17216498	drugbank:DB17087	JNJ-17216498	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	inhibitor	1.750255707856483	AZD2207	chembl:CHEMBL3545289	AZD2207	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.5357925636295356	N6-PHENYLADENOSINE	chembl:CHEMBL262083	N6-PHENYLADENOSINE	FALSE	FALSE	FALSE
KCNMA1	hgnc:6284	KCNMA1	ChEMBL	33	activator	2.917092846427472	ANDOLAST	ncit:C74213	ANDOLAST	FALSE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	modulator	0.096167896	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	modulator	0.096167896	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	modulator	0.1442518440541058	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	modulator	0.2243917574174979	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.050246575	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
MAP3K10	hgnc:6849	MAP3K10	ChEMBL	33	inhibitor	0.9723642821424908	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	0.2386712328895204	IUPHAR.LIGAND:2294	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	ChEMBL	33	inhibitor	0.036463661	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PRKCE	hgnc:9401	PRKCE	ChEMBL	33	inhibitor	0.072927321	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	modulator	0.2243917574174979	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	modulator	0.048083948	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	modulator	0.1187956362798518	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
KCNC4	hgnc:6236	KCNC4	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	1.093909817410302	CARDAMOMIN	chembl:CHEMBL378104	CARDAMOMIN	FALSE	FALSE	FALSE
KCNA7	hgnc:6226	KCNA7	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
F9	hgnc:3551	F9	ChEMBL	33	inhibitor	2.763561643983921	PEGNIVACOGIN	ncit:C174625	PEGNIVACOGIN	FALSE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	1.544343271638073	CILANSETRON	ncit:C76106	CILANSETRON	FALSE	FALSE	FALSE
UNIPROT:P00390	hgnc:4623	GSR	TdgClinicalTrial	Jan-14	NULL	0.6509215442441467	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
CETP	hgnc:1869	CETP	ChEMBL	33	inhibitor	2.692701089009974	DALCETRAPIB	ncit:C81529	DALCETRAPIB	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.303074581	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
FAU	hgnc:3597	FAU	ChEMBL	33	inhibitor	0.065634589	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL10A	hgnc:10299	RPL10A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
KCNS1	hgnc:6300	KCNS1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	agonist	0.1798207919030633	CENEGERMIN	rxcui:2104331	CENEGERMIN-BKBJ	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.4089382494991783	ERDAFITINIB	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.035287413	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.03070624	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	2.187819634820604	NIRAPARIB TOSYLATE	rxcui:2637447	NIRAPARIB TOSYLATE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1894216134043813	COPANLISIB	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.3017682254924971	NERATINIB MALEATE	rxcui:1940642	NERATINIB MALEATE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	positive modulator	5.966780822238011	ELEXACAFTOR	rxcui:2256951	ELEXACAFTOR	TRUE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.7501095890813501	RAMOSETRON HYDROCHLORIDE	ncit:C88299	RAMOSETRON HYDROCHLORIDE	FALSE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.6177373086552295	RAMOSETRON HYDROCHLORIDE	ncit:C88299	RAMOSETRON HYDROCHLORIDE	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	0.7955707762984014	OPIGOLIX	ncit:C174927	OPIGOLIX	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.3182283105193605	DARUNAVIR	rxcui:460132	DARUNAVIR	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.1630673019742065	DELGOCITINIB	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
GP	hgnc:18280	RNF130	ChEMBL	33	inhibitor	7.501095891	MAFTIVIMAB	rxcui:2461339	MAFTIVIMAB	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.009972967	TRAZODONE HYDROCHLORIDE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
RPS3A	hgnc:10421	RPS3A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1296485709523321	HARMINE HYDROCHLORIDE	chembl:CHEMBL1593867	HARMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
RPS4Y1	hgnc:10425	RPS4Y1	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPS14	hgnc:10387	RPS14	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPS4X	hgnc:10424	RPS4X	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS25	hgnc:10413	RPS25	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	HEXYLRESORCINOL	rxcui:5321	HEXYLRESORCINOL	TRUE	FALSE	FALSE
RPL23A	hgnc:10317	RPL23A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL14	hgnc:10305	RPL14	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL24	hgnc:10325	RPL24	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL10A	hgnc:10299	RPL10A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL35	hgnc:10344	RPL35	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL37	hgnc:10347	RPL37	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	1.250182648468916	MONTEPLASE	ncit:C166422	MONTEPLASE	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	BALSTILIMAB	ncit:C136465	BALSTILIMAB	FALSE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.3500511415712967	ISOSORBIDE MONONITRATE	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
CMA1	hgnc:2097	CMA1	ChEMBL	33	inhibitor	10.50153424713889	FULACIMSTAT	ncit:C170012	FULACIMSTAT	FALSE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	ChEMBL	33	inhibitor	3.088686543276147	ABT-384	drugbank:DB12501	ABT-384	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	1.117184494376478	OSI-7904	chembl:CHEMBL169896	OSI-7904	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	modulator	0.133607306	AZD-5423	drugbank:DB12280	AZD-5423	FALSE	FALSE	FALSE
NPY5R	hgnc:7958	NPY5R	ChEMBL	33	inhibitor	7.501095891	MK-0557	drugbank:DB12168	MK-0557	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	1.193356164447602	ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
MAGEA3	hgnc:6801	MAGEA3	ChEMBL	33	vaccine	17.50255707856483	BIROPEPIMUT-S	ncit:C166968	BIROPEPIMUT-S	FALSE	FALSE	FALSE
GART	hgnc:4163	GART	ChEMBL	33	inhibitor	2.561349816375341	PELITREXOL	ncit:C2633	PELITREXOL	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	modulator	2.917092846427472	T-62	drugbank:DB12919	T-62	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	negative modulator	1.141471113819445	BNC-210	chembl:CHEMBL4650452	BNC-210	FALSE	FALSE	FALSE
ELANE	hgnc:3309	ELANE	ChEMBL	33	inhibitor	3.804903712731485	SIVELESTAT	ncit:C66539	SIVELESTAT	FALSE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	1.458546423213736	ONZIGOLIDE	ncit:C88345	ONZIGOLIDE	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.042174836	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.035719504	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	4.039051633514961	ONGERICIMAB	ncit:C174940	ONGERICIMAB	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	binder	0.021590325	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
CRTC1	hgnc:16062	CRTC1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.458546423213736	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.7143900848393808	BAY 869766	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1143957978991165	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.068037151	NVP-BEZ238	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.068037151	NVP-BEZ242	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.034018575	NVP-BEZ236	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00908123	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.088695391	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.061919424	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.1250182648468916	CUCURBITACIN B	iuphar.ligand:12432	CUCURBITACIN B	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:6316	rxcui:1546030	SAXAGLIPTIN ANHYDROUS	TRUE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.084689792	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	PT-103	chembl:CHEMBL398765	CHEMBL:CHEMBL398765	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1325951293830669	TCMDC-125606	chembl:CHEMBL536166	CHEMBL:CHEMBL536166	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.007282617	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	QUINOCIDE	ncit:C73004	QUINOCIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	KHELLIN	rxcui:6147	KHELLIN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.040328473	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.050488145	CHIR-265	iuphar.ligand:5674	CHIR-265	FALSE	FALSE	TRUE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:11220	iuphar.ligand:11220	SUPRASTAT	FALSE	FALSE	FALSE
PLD2	hgnc:9068	PLD2	DTC	9/2/20	NULL	8.751278539282415	HALOPEMIDE	ncit:C65840	HALOPEMIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.1495945049449986	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	chembl:CHEMBL1336287	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.021301287	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	0.031488858	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.012971263	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	SE-(METHYL)SELENOCYSTEINE HCL	chembl:CHEMBL1256174	CHEMBL:CHEMBL1256174	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	DTC	9/2/20	NULL	3.182283105193606	2'H,4H-[2,6'-BICHROMEN]-4-ONE	chembl:CHEMBL2347759	CHEMBL:CHEMBL2347759	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	BUNAMIDINE	ncit:C81513	BUNAMIDINE	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.2344092465879218	FUSARIC ACID	chembl:CHEMBL24510	FUSARIC ACID	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.004719791	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.1319288222002374	LY-367385	iuphar.ligand:1379	LY367385	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.1117184494376478	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GLA	hgnc:4296	GLA	DTC	9/2/20	NULL	0.4487835148349957	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.055155117	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	1.312691780892362	PYRIDABEN	chembl:CHEMBL225963	PYRIDABEN	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	1.500219178	TCMDC-124482	chembl:CHEMBL529939	CHEMBL:CHEMBL529939	FALSE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	DTC	9/2/20	NULL	0.5000730593875666	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.082950507	DNDI1417149	chembl:CHEMBL1622802	CHEMBL:CHEMBL1622802	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	L-732138	iuphar.ligand:9461	L-732,138	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CEFONICID SODIUM	ncit:C65300	CEFONICID SODIUM	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	SJ000147993	chembl:CHEMBL601618	CHEMBL:CHEMBL601618	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GR-55562	iuphar.ligand:113	GR-55562	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.059030547	TICRYNAFEN	ncit:C152613	TICRYNAFEN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	DIMETHENAMID	chembl:CHEMBL1565335	DIMETHENAMID	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011810092	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	CID 838877	chembl:CHEMBL405317	CHEMBL:CHEMBL405317	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	CYCLOBENZAPRINE HYDROCHLORIDE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DINOSEB	chembl:CHEMBL1892987	DINOSEB	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.01875274	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.020226376	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000434533	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.067839369	SJ000018300	chembl:CHEMBL590927	CHEMBL:CHEMBL590927	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.089298761	MIBEFRADIL DIHYDROCHLORIDE	rxcui:83214	MIBEFRADIL DIHYDROCHLORIDE	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1810609352954983	GNF-PF-3352	chembl:CHEMBL600306	CHEMBL:CHEMBL600306	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	SB-408124	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	LOPERAMIDE HYDROCHLORIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BUPIRIMATE	chembl:CHEMBL3183902	BUPIRIMATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	ISOBUTYLMETHYLXANTHINE	drugbank:DB07954	3-ISOBUTYL-1-METHYL-7H-XANTHINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.025298806	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	SB-408124	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
SRMS	hgnc:11298	SRMS	DTC	9/2/20	NULL	0.1491695205559502	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124062	chembl:CHEMBL537087	CHEMBL:CHEMBL537087	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.006551175	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	NSC-24047	chembl:CHEMBL1288013	CHEMBL:CHEMBL1288013	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.042863405	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.026253836	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.006847636	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	GNF-PF-3925	chembl:CHEMBL584248	CHEMBL:CHEMBL584248	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.059163573	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.012466209	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
PABPC1	hgnc:8554	PABPC1	DTC	9/2/20	NULL	2.625383561784725	SJ000040829	chembl:CHEMBL589711	CHEMBL:CHEMBL589711	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00517674	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.5834185692854944	DIFFRACTAIC ACID	chembl:CHEMBL367741	DIFFRACTAIC ACID	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	MOFEBUTAZONE	rxcui:30202	MOFEBUTAZONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	TDR77593	chembl:CHEMBL1510164	CHEMBL:CHEMBL1510164	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	NSC-24047	chembl:CHEMBL1288013	CHEMBL:CHEMBL1288013	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	FOSFONET	drugbank:DB02823	PHOSPHONOACETIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	SKF-83565 HYDROBROMIDE	chembl:CHEMBL541585	CHEMBL:CHEMBL541585	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.1852122442176172	PLX3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
HCP5	hgnc:21659	HCP5	PharmGKB	4/5/24	NULL	0.3977853881492008	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	R-N-PROPYLNORAPOMORPHINE	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.056826484	HOE-33342	chembl:CHEMBL343002	CHEMBL:CHEMBL343002	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.032252869	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BROTIZOLAM	rxcui:19790	BROTIZOLAM	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006265084	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.1183271464466354	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.1367387271762877	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1902451856365742	2,4-HEXADIENAL	chembl:CHEMBL1576086	2,4-HEXADIENAL	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	MMV006389	chembl:CHEMBL586000	CHEMBL:CHEMBL586000	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.01275077	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:3380	iuphar.ligand:3380	BGC201531	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.016491103	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.2263261691193728	(R)-PIA	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1591141552596802	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.033148782	TRANILAST	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.3977853881492008	NS-398	drugbank:DB14060	NS-398	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.023151531	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
POLA1	hgnc:9173	POLA1	DTC	9/2/20	NULL	6.563458904461812	DIGALLIC ACID	chembl:CHEMBL366356	DIGALLIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.004409445	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	METHYL AMINOLEVULINATE HYDROCHLORIDE	rxcui:1300479	METHYL AMINOLEVULINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	SJ000071821	chembl:CHEMBL589924	CHEMBL:CHEMBL589924	FALSE	FALSE	FALSE
UNIPROT:P68133	hgnc:129	ACTA1	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	THYMOSIN BETA-4	drugbank:DB12003	THYMOSIN BETA-4	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.091796628	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	R-N-PROPYLNORAPOMORPHINE	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	1.500219178	ETOCARLIDE	ncit:C65584	ETOCARLIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.031822831	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.010588359	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002737341	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.016206071	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	DTC	9/2/20	NULL	0.4546118721705151	ALPHA-NAPHTHOFLAVONE	drugbank:DB07453	ALPHA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	ARISTOLACTONE	chembl:CHEMBL2333547	ARISTOLACTONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.2536602475154323	SJ000191886	chembl:CHEMBL601616	CHEMBL:CHEMBL601616	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	NSC-402538	chembl:CHEMBL121556	CHEMBL:CHEMBL121556	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001424864	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010488109	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	TCMDC-138263	chembl:CHEMBL535307	CHEMBL:CHEMBL535307	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	1.750255707856483	HU-310	iuphar.ligand:5545	2-ARACHIDONYL GLYCERYL ETHER	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.729273212	GNF-PF-1260	chembl:CHEMBL584849	CHEMBL:CHEMBL584849	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TETRADIFON	chembl:CHEMBL437926	TETRADIFON	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004340912	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.074797252	NELFINAVIR	rxcui:134527	NELFINAVIR	TRUE	FALSE	TRUE
LPAR3	hgnc:14298	LPAR3	DTC	9/2/20	NULL	52.50767123569449	NSC-255523	chembl:CHEMBL519155	CHEMBL:CHEMBL519155	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	METHOCARBAMOL	rxcui:6845	METHOCARBAMOL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	LINOLEIC ACID	rxcui:6400	LINOLEIC ACID	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	BENZYL SALICYLATE	rxcui:1362907	BENZYL SALICYLATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	2,4-DIHYDROXYBENZOPHENONE	chembl:CHEMBL1392	2,4-DIHYDROXYBENZOPHENONE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.020591244	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	TCMDC-125814	chembl:CHEMBL533082	CHEMBL:CHEMBL533082	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001210747	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	NSC-158389	chembl:CHEMBL192626	CHEMBL:CHEMBL192626	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PYRIDABEN	chembl:CHEMBL225963	PYRIDABEN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DIETHYLCARBAMAZINE CITRATE	rxcui:203175	DIETHYLCARBAMAZINE CITRATE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.013788779	DICLOFENAC SODIUM	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.030814361	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
DDR2	hgnc:2731	DDR2	DTC	9/2/20	NULL	1.312691780892362	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-3925	chembl:CHEMBL584248	CHEMBL:CHEMBL584248	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.08334551	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.1392776425349986	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.4688184931758437	DIHYDROXANTHOHUMOL	chembl:CHEMBL510279	DIHYDROXANTHOHUMOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	BUFOGENIN	ncit:C77829	BUFOGENIN	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:6276	iuphar.ligand:6276	TCS 5861528	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.003861994	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	LOPINAVIR	rxcui:195088	LOPINAVIR	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	RAC-GONIOTHALAMIN	chembl:CHEMBL1170485	CHEMBL:CHEMBL1170485	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CARBOSULFAN	ncit:C163638	CARBOSULFAN	FALSE	FALSE	FALSE
STS	hgnc:11425	STS	DTC	9/2/20	NULL	7.001022831425932	17ALPHA-3'-TRIFLUOROMETHYLBENZYLESTRADIOL	chembl:CHEMBL1823787	CHEMBL:CHEMBL1823787	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.1131630845596864	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	MIBEFRADIL DIHYDROCHLORIDE	rxcui:83214	MIBEFRADIL DIHYDROCHLORIDE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.2067231151011594	ERUCIC ACID	chembl:CHEMBL1173380	ERUCIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.000769411	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1544343271638073	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003981473	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	DTC	9/2/20	NULL	3.182283105193606	3-(DIMETHYLAMINO)BUTYL 4-CYANOPHENYL(METHYL)CARBAMATE	chembl:CHEMBL466398	CHEMBL:CHEMBL466398	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.01192814	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-4279	chembl:CHEMBL601320	CHEMBL:CHEMBL601320	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	NSC-48300	chembl:CHEMBL1091971	CHEMBL:CHEMBL1091971	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.1000146118775133	NCG-C00093820-01	chembl:CHEMBL544115	CHEMBL:CHEMBL544115	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.09972967	SOTALOL HYDROCHLORIDE	rxcui:7008	SOTALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.034544521	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.029845209	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-2905	chembl:CHEMBL582694	CHEMBL:CHEMBL582694	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NSC-28081	chembl:CHEMBL512832	CHEMBL:CHEMBL512832	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.2573905452730122	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	VINBURNINE	rxcui:57954	VINBURNINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-312948A	chembl:CHEMBL480382	GSK-312948A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	PYRILAMINE	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	0.4054646427466756	L-733060	chembl:CHEMBL1256740	CHEMBL:CHEMBL1256740	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.006068848	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.1111273465305703	YUANHUADINE	chembl:CHEMBL1911631	YUANHUADINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BETAMETHASONE VALERATE	rxcui:227897	BETAMETHASONE VALERATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	EPIRUBICIN HYDROCHLORIDE	rxcui:203213	EPIRUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.086551106	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.046466966	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009630901	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.022315202	CIANIDANOL	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	(R)-PIA	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	CHARTREUSIN	chembl:CHEMBL1554674	CHARTREUSIN	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.5000730593875666	CUCURBITACIN B	iuphar.ligand:12432	CUCURBITACIN B	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.3500511415712966	DIHYDROSPINGOSINE	iuphar.ligand:2453	DIHYDROSPHINGOSINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002744064	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.1223955040459079	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	TEBUCONAZOLE	chembl:CHEMBL487186	TEBUCONAZOLE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	DIPHENYLPYRALINE	rxcui:23386	DIPHENYLPYRALINE	TRUE	FALSE	FALSE
NCBIGENE:701	hgnc:1149	BUB1B	GuideToPharmacology	2024.1	blocker	8.751278539282415	IUPHAR.LIGAND:4104	iuphar.ligand:4104	3-PHENYL-CPP	FALSE	FALSE	FALSE
HRH4	hgnc:17383	HRH4	DTC	9/2/20	NULL	14.32027397337122	PF-03893787	ncit:C169765	ADRIFORANT	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.026412309	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.008693323	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003720782	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.4234489615781814	PROPAZINE	chembl:CHEMBL1333189	PROPAZINE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.02091106	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.013186256	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	5,7,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL242385	CHEMBL:CHEMBL242385	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TRIFLUMIZOLE	chembl:CHEMBL463781	TRIFLUMIZOLE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	NS-398	drugbank:DB14060	NS-398	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.088996053	NCG-C00093820-01	chembl:CHEMBL544115	CHEMBL:CHEMBL544115	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	NS-398	drugbank:DB14060	NS-398	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.010171963	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.011355465	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.1615620653405984	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	chembl:CHEMBL1336287	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1400204566285186	DIBUTYLDICHLOROSTANNANE	chembl:CHEMBL1088184	DIBUTYLDICHLOROSTANNANE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.1259176768242074	ANDALUSOL	chembl:CHEMBL2180484	ANDALUSOL	FALSE	FALSE	FALSE
NCBIGENE:236	hgnc:425	AKR1B1P2	GuideToPharmacology	2024.1	modulator	0.5357925636295356	IUPHAR.LIGAND:5339	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	CINACALCET HYDROCHLORIDE	rxcui:384379	CINACALCET HYDROCHLORIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004952619	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007946076	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.013560866	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.577007376	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	EMETINE HYDROCHLORIDE	rxcui:82015	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.017386646	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	RAC-GONIOTHALAMIN	chembl:CHEMBL1170485	CHEMBL:CHEMBL1170485	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.002896496	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	TICLOPIDINE HYDROCHLORIDE	rxcui:97	TICLOPIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	ACACETIN DIACETATE	chembl:CHEMBL1566650	ACACETIN DIACETATE	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.042073455	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.068191781	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.042073455	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	TCMDC-125195	chembl:CHEMBL531709	CHEMBL:CHEMBL531709	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.2885036881082115	NSC-663284	drugbank:DB17038	NSC-663284	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	(R)-NITRENDIPINE	chembl:CHEMBL268609	(R)-NITRENDIPINE	FALSE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	0.6863747873946994	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
SPECC1L-ADORA2A	hgnc:49185	SPECC1L-ADORA2A	DTC	9/2/20	NULL	15.00219178162699	CGS-21680	iuphar.ligand:375	CGS 21680	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.010975684	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	TORSEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.085239726	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	CUMINGIANOSIDE A	chembl:CHEMBL451574	CUMINGIANOSIDE A	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.000994897	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	GYKI-52466	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-4837	chembl:CHEMBL600769	CHEMBL:CHEMBL600769	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001976425	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.036162308	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	LAURYL ISOQUINOLINIUM	chembl:CHEMBL1398631	LAURYL ISOQUINOLINIUM	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.057197899	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	BENZENE-1,2-DIAMINE	chembl:CHEMBL70582	CHEMBL:CHEMBL70582	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00402481	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.009098539	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011188509	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.075768645	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.037398626	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	DTC	9/2/20	NULL	0.7095631248066824	XYLOMETAZOLINE HYDROCHLORIDE	rxcui:54220	XYLOMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	GERONTOXANTHONE H	chembl:CHEMBL514057	GERONTOXANTHONE H	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.105015342	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.044198376	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	SULFOBROMOPHTHALEIN	rxcui:10212	SULFOBROMOPHTHALEIN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.022305723	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.028882107	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.029987248	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.018488617	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.056826484	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	DTC	9/2/20	NULL	2.187819634820604	SALERMIDE	chembl:CHEMBL597845	SALERMIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	METHYL PARATHIONE	chembl:CHEMBL346516	METHYL PARATHIONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	MECAMYLAMINE	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	AC-55649	iuphar.ligand:4055	AC55649	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.1539814405738841	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	2.282942227638891	IRISOLIDONE	chembl:CHEMBL265945	IRISOLIDONE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1400204566285186	TRIPHENYLSTANNANOL	chembl:CHEMBL506538	TRIPHENYLSTANNANOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	HYDROXYZINE	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.034727296	GLAFENINE	ncit:C72119	GLAFENINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	PIRENZEPINE HYDROCHLORIDE	rxcui:235775	PIRENZEPINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TRICHLORFON	rxcui:1000581	TRICHLORFON	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	PIPERACETAZINE	rxcui:8338	PIPERACETAZINE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.045461187	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	ASCORBYL PALMITATE	ncit:C81556	ASCORBYL PALMITATE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011810092	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	GNF-PF-4463	chembl:CHEMBL584520	CHEMBL:CHEMBL584520	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-125602	chembl:CHEMBL580183	CHEMBL:CHEMBL580183	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	AG-370	chembl:CHEMBL59150	CHEMBL:CHEMBL59150	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123826	chembl:CHEMBL598369	CHEMBL:CHEMBL598369	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.04907259	TRIPHENYLSTANNANOL	chembl:CHEMBL506538	TRIPHENYLSTANNANOL	FALSE	FALSE	FALSE
S1PR3	hgnc:3167	S1PR3	DTC	9/2/20	NULL	3.281729452230906	SJ000189154	chembl:CHEMBL604664	CHEMBL:CHEMBL604664	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.032492371	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	METHOXYCHLOR	rxcui:2598123	METHOXYCHLOR	FALSE	FALSE	FALSE
TRPM8	hgnc:17961	TRPM8	DTC	9/2/20	NULL	2.763561643983921	5-BENZYLOXYTRYPTAMINE	iuphar.ligand:265	5-BENZYLOXYTRYPTAMINE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	DNDI1417995	chembl:CHEMBL1439833	CHEMBL:CHEMBL1439833	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.042140988	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	DNDI1417099	chembl:CHEMBL1565444	CHEMBL:CHEMBL1565444	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	CID 893238	chembl:CHEMBL473735	CHEMBL:CHEMBL473735	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.005747966	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	L-690330	iuphar.ligand:5208	L690330	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.074163377	METHIOTHEPIN MESYLATE	chembl:CHEMBL1256737	METHIOTHEPIN MESYLATE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	DNDI1417099	chembl:CHEMBL1565444	CHEMBL:CHEMBL1565444	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	ETHACRIDINE	rxcui:4106	ETHACRIDINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005294179	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	MIBEFRADIL DIHYDROCHLORIDE	rxcui:83214	MIBEFRADIL DIHYDROCHLORIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.022249013	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.056826484	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV396794	chembl:CHEMBL2028063	CHEMBL:CHEMBL2028063	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004191225	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	CLIOXANIDE	ncit:C65338	CLIOXANIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.025739055	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000112483	chembl:CHEMBL603024	CHEMBL:CHEMBL603024	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.002011788	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.008585296	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009922085	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	5,7,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL242385	CHEMBL:CHEMBL242385	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.018206543	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.041214813	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.007899454	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
PTBP1	hgnc:9583	PTBP1	DTC	9/2/20	NULL	0.6731752722524936	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.039331589	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	CHELIDONINE (+)	chembl:CHEMBL436279	CHELIDONINE (+)	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	BUPIRIMATE	chembl:CHEMBL3183902	BUPIRIMATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	CLOROPHENE	rxcui:21290	CLOROPHENE	FALSE	FALSE	FALSE
GRM4	hgnc:4596	GRM4	DTC	9/2/20	NULL	7.501095891	N-(3-(DIFLUOROMETHOXY)PHENYL)PICOLINAMIDE	chembl:CHEMBL541754	CHEMBL:CHEMBL541754	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DEBRISOQUIN SULFATE	ncit:C77302	DEBRISOQUIN SULFATE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	PECTOLINARIGENIN	chembl:CHEMBL78010	PECTOLINARIGENIN	FALSE	FALSE	FALSE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	0.4102161815288632	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.2885036881082116	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	TCMDC-124440	chembl:CHEMBL547407	CHEMBL:CHEMBL547407	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	DIHYDROCAPSAICIN	rxcui:2166037	DIHYDROCAPSAICIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001750547	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.001635753	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.028977744	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-2588	chembl:CHEMBL578636	CHEMBL:CHEMBL578636	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.00256824	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.022099188	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009579944	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	GNF-PF-1813	chembl:CHEMBL577662	CHEMBL:CHEMBL577662	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	FDA	10-Apr-24	NULL	0.091732479	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.080781033	Chloroprocaine	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	FDA	10-Apr-24	NULL	0.051731696	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SERPINC1	hgnc:775	SERPINC1	FDA	10-Apr-24	NULL	0.031032903	Estradiol	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.3962843112127887	OK-432	ncit:C745	PICIBANIL	FALSE	FALSE	FALSE
FCGR1C	hgnc:3615	FCGR1CP	NCI	14-Sep-17	NULL	2.692701089009974	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.026418954	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.070765056	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.2892984641085096	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.099071078	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.6364566210387212	OK-432	ncit:C745	PICIBANIL	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.018521224	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
FH	hgnc:3700	FH	NCI	14-Sep-17	NULL	3.750547945406749	DIETHYLDITHIOCARBAMATE	rxcui:1427193	DIETHYLDITHIOCARBAMATE	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.5676505	NEOVASTAT	drugbank:DB05387	NEOVASTAT	FALSE	FALSE	TRUE
FOSL1	hgnc:13718	FOSL1	NCI	14-Sep-17	NULL	5.250767124	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.030868707	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.252440727	DXM	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.3106962795011509	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
GALC	hgnc:4115	GALC	NCI	14-Sep-17	NULL	8.290684931951763	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
GCLM	hgnc:4312	GCLM	NCI	14-Sep-17	NULL	0.3106962795011509	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.2778183663264259	MNU	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
H2AFX	hgnc:4739	H2AX	NCI	14-Sep-17	NULL	0.7501095890813501	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.035719504	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
HBEGF	hgnc:3059	HBEGF	NCI	14-Sep-17	NULL	0.096788334	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
GUCA2A	hgnc:4682	GUCA2A	NCI	14-Sep-17	NULL	1.250182648468916	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:9592	iuphar.ligand:9592	TISLELIZUMAB	FALSE	FALSE	FALSE
HOXA9	hgnc:5109	HOXA9	NCI	14-Sep-17	NULL	9.546849315580818	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.2960958904268487	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.2960958904268487	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
HMOX1	hgnc:5013	HMOX1	NCI	14-Sep-17	NULL	0.8975670296699916	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
HOXB1	hgnc:5111	HOXB1	NCI	14-Sep-17	NULL	7.001022831425932	HEXAMETHYLENEBISACETAMIDE	chembl:CHEMBL291481	HEXAMETHYLENEBISACETAMIDE	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.1535312024435511	MNU	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1162960603226899	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.087222045	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.2472888755213241	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.1795134059339982	HERCEPTIN	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
HTT	hgnc:4851	HTT	NCI	14-Sep-17	NULL	0.2318219480604613	BRAIN-DERIVED NEUROTROPHIC FACTOR	rxcui:47324	BRAIN-DERIVED NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
IFI27	hgnc:5397	IFI27	NCI	14-Sep-17	NULL	2.019525816757481	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	HARMAN-3-CARBOXYLIC ACID	chembl:CHEMBL504850	HARMAN-3-CARBOXYLIC ACID	FALSE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	0.7343730242754476	ALPHA-METHYL-P-TYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
IFNGR1	hgnc:5439	IFNGR1	NCI	14-Sep-17	NULL	8.751278539282415	INDOLE-3-CARBINOL	rxcui:2598119	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.4688184931758437	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
IHH	hgnc:5956	IHH	NCI	14-Sep-17	NULL	5.000730593875666	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	PharmGKB	4/5/24	NULL	0.02357776	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.8751278539282416	ACYCLOVIR	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
IGFBP6	hgnc:5475	IGFBP6	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1470803115845784	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.013792401	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.3571950424196904	SERM	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
IL7	hgnc:6023	IL7	NCI	14-Sep-17	NULL	4.375639269641208	ALUM	rxcui:221456	ALUM, POTASSIUM	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.5357925636295356	HMG-COA REDUCTASE INHIBITOR	ncit:C1655	HMG-COA REDUCTASE INHIBITOR	FALSE	FALSE	FALSE
ILF3	hgnc:6038	ILF3	NCI	14-Sep-17	NULL	1.750255707856483	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.09972967	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	1.346350544504987	SPD-557	chembl:CHEMBL3545035	REVEXEPRIDE	FALSE	FALSE	FALSE
IL9R	hgnc:6030	IL9R	NCI	14-Sep-17	NULL	35.00511415712966	IL-9	iuphar.ligand:5000	IL-9	FALSE	FALSE	FALSE
LIPC	hgnc:6619	LIPC	NCI	14-Sep-17	NULL	8.751278539282415	HEMOCLAR	chembl:CHEMBL1201516	PENTOSAN POLYSULFATE SODIUM	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.325124899	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4332	iuphar.ligand:4332	UBP141	FALSE	FALSE	FALSE
MAGEA3	hgnc:6801	MAGEA3	NCI	14-Sep-17	NULL	3.500511415712967	DNA VACCINE	ncit:C39619	DNA VACCINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.050007306	URACIL	rxcui:10995	URACIL	TRUE	FALSE	TRUE
MARK2	hgnc:3332	MARK2	NCI	14-Sep-17	NULL	0.096167896	APAP	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	NCI	14-Sep-17	NULL	0.305277158	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.3697723326457359	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.1250182648468916	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.2500365296937833	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	BIZELESIN	ncit:C1472	BIZELESIN	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.071439008	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.001259177	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.054020238	TAXOL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.026892533	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.1325951293830669	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.1944728564284981	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.2580229544751573	ECG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1232574442152452	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	3.281729452230906	BASIC FIBROBLAST GROWTH FACTOR	drugbank:DB14131	BASIC FIBROBLAST GROWTH FACTOR	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	NCI	14-Sep-17	NULL	0.025584378	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.1553481397505754	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.2375912725597036	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.2125816649218401	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	NCI	14-Sep-17	NULL	0.062620956	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	NCI	14-Sep-17	NULL	0.052090944	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	NCI	14-Sep-17	NULL	0.014585464	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.010569177	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.008103036	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.020836377	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.1041818873724097	UROKINASE-TYPE PLASMINOGEN ACTIVATOR	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.032055965	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.2692701089009974	BRAIN-DERIVED NEUROTROPHIC FACTOR	rxcui:47324	BRAIN-DERIVED NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.079798892	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.096167896	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
PRF1	hgnc:9360	PRF1	NCI	14-Sep-17	NULL	1.166837138570988	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	0.1262203635473425	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	ChEMBL	33	binder	1.591141552596803	PRASINEZUMAB	ncit:C174831	PRASINEZUMAB	FALSE	FALSE	FALSE
PREP	hgnc:9358	PREP	NCI	14-Sep-17	NULL	0.760980743	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.4861821410712453	ESTRONE-SULFATE	ncit:C1091	ESTRONE SULFATE	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1215455352678113	FCA	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
PTGER4	hgnc:9596	PTGER4	NCI	14-Sep-17	NULL	0.1342907192728759	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	NCI	14-Sep-17	NULL	0.2651902587661338	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
PTGES3	hgnc:16049	PTGES3	NCI	14-Sep-17	NULL	0.6035364509849942	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	blocker	0.2273059360852575	IUPHAR.LIGAND:2294	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.070860555	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.02726255	sacituzumab govitecan-hziy	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	PharmGKB	4/5/24	NULL	0.3079628811477683	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	0.546954909	sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
LHFPL3	hgnc:6589	LHFPL3	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
NCBIGENE:416	hgnc:721	ARSF	GuideToPharmacology	2024.1	blocker	0.4565884455277782	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	PharmGKB	4/5/24	NULL	0.1286952726365061	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	0.8334550989792776	letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	0.192335792	didanosine	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
CHRNA5	hgnc:1959	CHRNA5	PharmGKB	4/5/24	NULL	0.9723642821424908	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
RHOA	hgnc:667	RHOA	PharmGKB	4/5/24	NULL	0.300043836	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CHRNA6	hgnc:15963	CHRNA6	PharmGKB	4/5/24	NULL	0.9723642821424908	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
MAML3	hgnc:16272	MAML3	PharmGKB	4/5/24	NULL	4.039051633514962	perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
STX4	hgnc:11439	STX4	PharmGKB	4/5/24	NULL	1.060761035064535	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.002465612	topiramate	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.1172046232939609	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.1767935058440892	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
LTA	hgnc:6709	LTA	PharmGKB	4/5/24	NULL	2.386712328895204	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
LTB	hgnc:6711	LTB	PharmGKB	4/5/24	NULL	4.773424657790409	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
FNTB	hgnc:3785	FNTB	PharmGKB	4/5/24	NULL	0.1944728564284981	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	fosamprenavir	rxcui:358262	FOSAMPRENAVIR	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.010451368	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00903591	cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.016780975	cisapride	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	desloratadine	rxcui:275635	DESLORATADINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.01305187	saquinavir	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.016780975	sulfamethoxazole	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004195244	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
KIR2DS2	hgnc:6334	KIR2DS2	PharmGKB	4/5/24	NULL	1.640864726115453	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	0.040798501	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
MIR6076	hgnc:50232	MIR6076	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	0.040798501	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP27A1	hgnc:2605	CYP27A1	NCI	14-Sep-17	NULL	13.12691780892362	PHYTOSTEROLS	rxcui:8310	PHYTOSTEROLS	TRUE	FALSE	FALSE
SULF2	hgnc:20392	SULF2	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ENG	hgnc:3349	ENG	PharmGKB	4/5/24	NULL	0.1562728310586145	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.007325289	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
BAHD1	hgnc:29153	BAHD1	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
FGFR1OP2	hgnc:23098	FGFR1OP2	PharmGKB	4/5/24	NULL	7.501095890813499	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
CARBONIC ANHYDRASE VI	hgnc:1380	CA6	TTD	2020.06.01	NULL	1.500219178	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.218327115	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.05913026	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
DRD1	hgnc:3020	DRD1	PharmGKB	4/5/24	NULL	0.182318303	drotrecogin alfa	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
SOCS3	hgnc:19391	SOCS3	PharmGKB	4/5/24	NULL	0.8204323630577265	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.047734247	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
SCNN1B	hgnc:10600	SCNN1B	PharmGKB	4/5/24	NULL	1.544343271638073	amiloride	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	PharmGKB	4/5/24	NULL	0.074797252	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
CYB5R4	hgnc:20147	CYB5R4	PharmGKB	4/5/24	NULL	0.9546849315580819	primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.5073204950308647	rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	PharmGKB	4/5/24	NULL	0.037398626	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.5147810905460245	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH2	hgnc:404	ALDH2	PharmGKB	4/5/24	NULL	0.1342907192728759	naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
CPS1	hgnc:2323	CPS1	PharmGKB	4/5/24	NULL	1.250182648468916	glycerol phenylbutyrate	rxcui:1368451	GLYCEROL PHENYLBUTYRATE	TRUE	FALSE	FALSE
UNIPROT:P53779	hgnc:6872	MAPK10	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	AM-111	iuphar.ligand:9101	BRIMAPITIDE	FALSE	FALSE	FALSE
BDNF-AS	hgnc:20608	BDNF-AS	PharmGKB	4/5/24	NULL	6.563458904461812	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
VKORC1L1	hgnc:21492	VKORC1L1	PharmGKB	4/5/24	NULL	3.182283105193606	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	TALC	12-May-16	inhibitor	0.1852122442176172	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	TALC	12-May-16	inhibitor	0.064824285	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.075442056	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.1769126389342806	FK-228	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.1769126389342806	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.4518732464345482	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.067897851	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.089501712	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
NAIP	hgnc:7634	NAIP	TALC	12-May-16	inhibitor	3.750547945406749	LCL161	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	TALC	12-May-16	inhibitor	1.921012362281506	OBLIMERSEN	ncit:C1870	OBLIMERSEN	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.1875273972703374	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.099220845	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:9915	ncit:C90996	PAMAPIMOD	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.3968833804663227	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
RICTOR	hgnc:28611	RICTOR	TALC	12-May-16	inhibitor	1.154014752432846	AZD 8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
SRC	hgnc:11283	SRC	TALC	12-May-16	inhibitor	0.097236428	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
TNFRSF11A	hgnc:11908	TNFRSF11A	TALC	12-May-16	antibody	2.500365296937833	DENOSUMAB	rxcui:993449	DENOSUMAB	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	OncoKB	23-Jul-20	NULL	0.088333021	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	TALC	12-May-16	inhibitor	1.413668071730236	AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
ABL1	hgnc:76	ABL1	TALC	12-May-16	inhibitor	0.8008364246019593	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
BIRC2	hgnc:590	BIRC2	TALC	12-May-16	inhibitor	0.3750547945406749	LCL161	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
CHEK2	hgnc:16627	CHEK2	TALC	12-May-16	inhibitor	0.6177373086552295	AZD7762	iuphar.ligand:7713	AZD7762	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.092606122	AV 203	ncit:C102535	ANTI-ERBB3 MONOCLONAL ANTIBODY AV-203	FALSE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.034727296	ARRY 380	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
CTSK	hgnc:2536	CTSK	TALC	12-May-16	inhibitor	23.33674277141977	ODANACATIB	ncit:C66981	ODANACATIB	FALSE	FALSE	TRUE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.007907782	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P20648	hgnc:819	ATP4A	TdgClinicalTrial	Jan-14	NULL	0.2243917574174979	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.1448487482363986	ACAMPROSATE	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	L-745870	iuphar.ligand:3303	L745870	FALSE	FALSE	FALSE
UNIPROT:P14780	hgnc:7176	MMP9	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	AE-941	ncit:C1798	SHARK CARTILAGE EXTRACT AE-941	FALSE	FALSE	FALSE
UNIPROT:Q14416	hgnc:4594	GRM2	TdgClinicalTrial	Jan-14	NULL	3.750547945	ADX-71149	iuphar.ligand:8946	JNJ-40411813	FALSE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	AE-941	ncit:C1798	SHARK CARTILAGE EXTRACT AE-941	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.4167275494896388	MECAMYLAMINE	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.0701037	LEVONORGESTREL	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.4449802647092754	BENAZEPRIL	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
UNIPROT:P31639	hgnc:11037	SLC5A2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	BI-10773	rxcui:1545653	EMPAGLIFLOZIN	TRUE	FALSE	FALSE
UNIPROT:P17252	hgnc:9393	PRKCA	TdgClinicalTrial	Jan-14	NULL	0.546954909	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	OGLEMILAST	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	NXN-188	drugbank:DB06096	NXN-188	FALSE	FALSE	FALSE
UNIPROT:P43235	hgnc:2536	CTSK	TdgClinicalTrial	Jan-14	NULL	23.33674277141977	ODANACATIB	ncit:C66981	ODANACATIB	FALSE	FALSE	TRUE
UNIPROT:P42338	hgnc:8976	PIK3CB	TdgClinicalTrial	Jan-14	NULL	0.052090944	RIGOSERTIB	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
UNIPROT:Q8IUQ4	hgnc:10857	SIAH1	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	OMIGAPIL	ncit:C97362	OMIGAPIL	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.005297384	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:P04406	hgnc:4141	GAPDH	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	OMIGAPIL	ncit:C97362	OMIGAPIL	FALSE	FALSE	FALSE
UNIPROT:P53350	hgnc:9077	PLK1	TdgClinicalTrial	Jan-14	NULL	0.072927321	RIGOSERTIB	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	1.117184494376478	OSI-7904L	drugbank:DB05457	OSI-7904L	FALSE	FALSE	FALSE
UNIPROT:P49721	hgnc:9539	PSMB2	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.027538988	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UNIPROT:P00740	hgnc:3551	F9	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	PEGNIVACOGIN	ncit:C174625	PEGNIVACOGIN	FALSE	FALSE	FALSE
UNIPROT:P20701	hgnc:6148	ITGAL	TdgClinicalTrial	Jan-14	NULL	2.414145803939977	EFALIZUMAB	rxcui:356988	EFALIZUMAB	TRUE	TRUE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.008821853	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
UNIPROT:P01112	hgnc:5173	HRAS	TdgClinicalTrial	Jan-14	NULL	0.2302968036653267	REOLYSIN	chembl:CHEMBL3545069	PELAREOREP	FALSE	FALSE	TRUE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	0.8975670296699915	ELETRIPTAN	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
UNIPROT:Q9H3N8	hgnc:17383	HRH4	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	REV131	drugbank:DB05032	REV131	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	ROCURONIUM	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
UNIPROT:P21453	hgnc:3165	S1PR1	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	RPC1063	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
UNIPROT:P05771	hgnc:9395	PRKCB	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	RUBOXISTAURIN	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
UNIPROT:P15509	hgnc:2435	CSF2RA	TdgClinicalTrial	Jan-14	NULL	11.66837138570988	SARGRAMOSTIM	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
GASTRIN-RELEASING PEPTIDE RECEPTOR	hgnc:4609	GRPR	TTD	2020.06.01	NULL	26.25383561784724	RC-3095	iuphar.ligand:6183	[D-TPI6, LEU13 &PSI;(CH2NH)-LEU14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.2536602475154323	SB1518	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.051655358	DEXTROAMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	1.500219178	SGX523	ncit:C74062	MET TYROSINE KINASE INHIBITOR SGX523	FALSE	FALSE	TRUE
UNIPROT:P30519	hgnc:5014	HMOX2	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	STANNSOPORFIN	ncit:C152424	STANNSOPORFIN	FALSE	FALSE	FALSE
UNIPROT:P00451	hgnc:3546	F8	TdgClinicalTrial	Jan-14	NULL	9.26605963	TB-402	drugbank:DB06050	TB-402	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	TC-5214	chembl:CHEMBL2103881	DEXMECAMYLAMINE	FALSE	FALSE	FALSE
UNIPROT:P49354	hgnc:3782	FNTA	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	TIPIFARNIB	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
UNIPROT:Q16099	hgnc:4582	GRIK4	TdgClinicalTrial	Jan-14	NULL	0.8334550989792778	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P49841	hgnc:4617	GSK3B	TdgClinicalTrial	Jan-14	NULL	0.760980743	TIDEGLUSIB	ncit:C97364	TIDEGLUSIB	FALSE	FALSE	FALSE
UNIPROT:P51857	hgnc:388	AKR1D1	TdgClinicalTrial	Jan-14	NULL	1.875273972703374	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
UNIPROT:P31213	hgnc:11285	SRD5A2	TdgClinicalTrial	Jan-14	NULL	3.750547945	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012112496	ACETYLCYSTEINE	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
UNIPROT:O95838	hgnc:4325	GLP2R	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	ZP1848	iuphar.ligand:10885	GLEPAGLUTIDE	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.079197091	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.07182992	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.099446347	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1367387271762877	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P10253	hgnc:4065	GAA	TEND	1-Aug-11	NULL	0.364636606	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.5933070196123671	CANDOXATRIL	ncit:C171870	CANDOXATRIL	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.063761592	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.07160137	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.076840494	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.079758488	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.075010959	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.150021918	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.055271233	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.065125794	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.029260335	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.112036283	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	DOXYLAMINE	rxcui:3642	DOXYLAMINE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.116943588	DROMOSTANOLONE	rxcui:23678	DROMOSTANOLONE	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1383601350084176	DROPERIDOL	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TEND	1-Aug-11	NULL	0.9907107780319716	MECASERMIN	rxcui:274403	MECASERMIN	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	1.093909817410302	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.021846337	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TEND	1-Aug-11	NULL	0.4243044140258141	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
UNIPROT:P17181	hgnc:5432	IFNAR1	TEND	1-Aug-11	NULL	1.458546423213736	INTERFERON ALFA-N1	rxcui:202912	INTERFERON ALFA-N1	FALSE	TRUE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TEND	1-Aug-11	NULL	0.072851434	INFLIXIMAB	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.4070362111294147	LEVOBUNOLOL	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TEND	1-Aug-11	NULL	0.8751278539282416	BECAPLERMIN	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.1363835616511545	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.093763699	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.1295419520617463	MEPIVACAINE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.2282942227638891	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P49721	hgnc:9539	PSMB2	TEND	1-Aug-11	NULL	0.4579157375205915	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.027538988	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1442518440541058	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.1426838892274307	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P00813	hgnc:186	ADA	TEND	1-Aug-11	NULL	3.043922970185188	PENTOSTATIN	rxcui:8011	PENTOSTATIN	TRUE	FALSE	TRUE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1025540453822158	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TEND	1-Aug-11	NULL	2.734774543525755	PRALATREXATE	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
UNIPROT:P05546	hgnc:4838	SERPIND1	TEND	1-Aug-11	NULL	7.501095890813499	ARDEPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.087318744	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.085239726	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1223955040459079	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
LYSYL OXIDASE HOMOLOG 2	hgnc:6666	LOXL2	TTD	2020.06.01	NULL	52.50767123569449	GS-6624	ncit:C91735	SIMTUZUMAB	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.1363835616511545	SCATTER FACTOR	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
TANKYRASE	hgnc:11941	TNKS	TTD	2020.06.01	NULL	3.750547945406749	BGB-290	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
SODIUM/HYDROGEN EXCHANGER 3	hgnc:11073	SLC9A3	TTD	2020.06.01	NULL	13.12691780892362	RDX-5791	iuphar.ligand:8449	TENAPANOR	FALSE	FALSE	FALSE
E-SELECTIN	hgnc:10718	SELE	TTD	2020.06.01	NULL	4.773424657790408	GMI-1271	ncit:C119743	UPROLESELAN	FALSE	FALSE	FALSE
INTERLEUKIN-8	hgnc:6025	CXCL8	TTD	2020.06.01	NULL	0.6482428547616604	MDX-018	drugbank:DB05484	MDX-018	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	2.838252499226729	Orvepitant	ncit:C90613	ORVEPITANT	FALSE	FALSE	FALSE
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	10.50153424713889	IR502	drugbank:DB06463	IR502	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	0.1290114772375786	Selegiline	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
INTERLEUKIN 4 RECEPTOR ALPHA	hgnc:6015	IL4R	TTD	2020.06.01	NULL	2.917092846427472	SAR-156597	chembl:CHEMBL4298097	ROMILKIMAB	FALSE	FALSE	FALSE
HAPTOGLOBIN	hgnc:5141	HP	TTD	2020.06.01	NULL	2.500365296937833	AT1001	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.079197091	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 1	hgnc:6877	MAPK3	TTD	2020.06.01	NULL	0.7925686224255775	GDC-0994	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	MEDI0680	drugbank:DB15768	MEDI0680	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.6908904109959803	PF-01247324	iuphar.ligand:8521	PF-01247324	FALSE	FALSE	FALSE
QUINONE REDUCTASE 2	hgnc:7856	NQO2	TTD	2020.06.01	NULL	0.1065064325267636	Melatonin	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.9334697108567911	Simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
SQUALENE MONOOXYGENASE	hgnc:11279	SQLE	TTD	2020.06.01	NULL	0.7721716358190368	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	0.082429625	Tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.7955707762984013	Icosapent	rxcui:90	EICOSAPENTAENOIC ACID	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	0.1121958787087489	TRYPTAMINE	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.048260727	Tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.3454452054979901	Rilpivirine	rxcui:1102270	RILPIVIRINE	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	1.944728564284981	Bimakalim	ncit:C166767	BIMAKALIM	FALSE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	1.014640990061729	Desmopressin	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.3697723326457359	Fadolmidine	ncit:C75054	FADOLMIDINE	FALSE	FALSE	FALSE
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	0.6250913242344582	UK-356202	iuphar.ligand:6543	UK-356202	FALSE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	0.3125456621172291	Alteplase	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	4.039051633514961	LIDORESTAT	ncit:C72815	LIDORESTAT	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	0.074797252	Ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	1.334940794127826	Spirapril	rxcui:36908	SPIRAPRIL	TRUE	FALSE	FALSE
CHOLECYSTOKININ RECEPTOR TYPE A	hgnc:1570	CCKAR	TTD	2020.06.01	NULL	1.312691780892362	PD-170292	chembl:CHEMBL14153	PD-170292	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.5048814541893701	NM-3	drugbank:DB12818	NM-3	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.061992528	Ro 31-7453	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	4.565884455277782	DX-890	ncit:C87386	DEPELESTAT	FALSE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	0.00598378	HP-184	ncit:C80997	NERISPIRDINE	FALSE	FALSE	FALSE
TRANSCRIPTION FACTOR SP1	hgnc:11205	SP1	TTD	2020.06.01	NULL	52.50767123569449	Terameprocol	ncit:C61441	TERAMEPROCOL	FALSE	FALSE	FALSE
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	3.182283105193605	Monobenzone	rxcui:17145	MONOBENZONE	TRUE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	0.8975670296699915	Eletriptan	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.1160818081850283	Hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.1658136986390352	Lorazepam	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.064347636	Pergolide	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.061041236	Pergolide	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.1884246575443582	Temazepam	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.061055432	Talbutal	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.046303061	Vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NCBIGENE:64	hgnc:137	ACTBP4	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:3656	iuphar.ligand:3656	[125I]CCL21 (HUMAN)	FALSE	FALSE	FALSE
THYROTROPIN RECEPTOR	hgnc:12373	TSHR	TTD	2020.06.01	NULL	0.2234368988752957	Thyrotropin	rxcui:10579	THYROTROPIN	TRUE	FALSE	FALSE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	0.1172046232939609	Trimethoprim	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.3281729452230906	BAY1125976	iuphar.ligand:10908	BAY1125976	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.1545479653736408	CGM097	ncit:C104280	P53/HDM2 INTERACTION INHIBITOR CGM097	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	1.458546423213736	G1T28-1	chembl:CHEMBL3894860	TRILACICLIB	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.546954909	Iruplinalkib	ncit:C154279	IRUPLINALKIB	FALSE	FALSE	FALSE
APOPTOSIS MEDIATING SURFACE ANTIGEN FAS	hgnc:11920	FAS	TTD	2020.06.01	NULL	0.9053046764774912	VB-111	ncit:C71539	OFRANERGENE OBADENOVEC	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	1.381780822	TEN010	drugbank:DB15151	RO-6870810	FALSE	FALSE	FALSE
INTERLEUKIN-13	hgnc:5973	IL13	TTD	2020.06.01	NULL	1.458546423213736	SAR-156597	chembl:CHEMBL4298097	ROMILKIMAB	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.2822993077187876	COVA322	iuphar.ligand:10469	COVA322	FALSE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	0.1875273972703375	Dinoprostone	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.4189441853911795	Benztropine	rxcui:1424	BENZTROPINE	TRUE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:1057	iuphar.ligand:1057	GW1100	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.1470803115845784	Bethanechol	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1226814748497534	Cyclofenil	rxcui:2983	CYCLOFENIL	TRUE	FALSE	FALSE
B2 BRADYKININ RECEPTOR	hgnc:1030	BDKRB2	TTD	2020.06.01	NULL	2.187819634820604	Icatibant	rxcui:1148138	ICATIBANT	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	5-METHOXY DMT OXALATE	chembl:CHEMBL1256920	CHEMBL:CHEMBL1256920	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	1.050153425	Gliclazide	rxcui:4816	GLICLAZIDE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Fosfestrol	rxcui:25284	FOSFESTROL	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR	hgnc:2438	CSF3	TTD	2020.06.01	NULL	4.375639269641208	Interleukin-3	rxcui:1311225	INTERLEUKIN-3	FALSE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	2.333674277141977	Minodronate	drugbank:DB06548	MINODRONIC ACID	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.9907107780319716	Mecasermin	rxcui:274403	MECASERMIN	TRUE	FALSE	FALSE
CLEC4C	hgnc:13258	CLEC4C	ChEMBL	33	inhibitor	52.50767123569449	LITIFILIMAB	ncit:C186413	LITIFILIMAB	FALSE	FALSE	FALSE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	6.563458904461812	MCB-3837	ncit:C173413	QUINOLONYL-OXAZOLIDINONE ANTIBIOTIC DNV3837	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.077217164	Mirtazapine	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
ADENOSINE DEAMINASE	hgnc:186	ADA	TTD	2020.06.01	NULL	3.043922970185188	Pentostatin	rxcui:8011	PENTOSTATIN	TRUE	FALSE	TRUE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1221108633388244	Secobarbital	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	0.6731752722524935	Tranylcypromine	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
INTERLEUKIN-12 ALPHA	hgnc:5969	IL12A	TTD	2020.06.01	NULL	1.050153425	Ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	1.887530665335423	Zileuton	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	3.500511415712966	VX-148	drugbank:DB06103	VX-148	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1835932560688619	Vortioxetine	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	AST-1306	ncit:C179280	ALLITINIB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007937668	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE ATR	hgnc:882	ATR	TTD	2020.06.01	NULL	0.8751278539282416	AZD6738	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	4.039051633514961	LY-2334737	drugbank:DB12906	LY-2334737	FALSE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.8334550989792777	GS-9901	chembl:CHEMBL3928407	GS-9901	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	3.000438356	KUC-7483	chembl:CHEMBL2107773	RITOBEGRON	FALSE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	1.078924751	LOXO-101	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
SERUM AMYLOID P-COMPONENT	hgnc:584	APCS	TTD	2020.06.01	NULL	6.563458904461812	GSK2398852	ncit:C153210	DEZAMIZUMAB	FALSE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	0.2853677784548614	SAR408701	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	0.9460841664089098	GW274150	iuphar.ligand:9849	GW274150	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	GS-4059	ncit:C102876	TIRABRUTINIB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	3.000438356	GS-9876	ncit:C174607	LANRAPLENIB	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR B	hgnc:8800	PDGFB	TTD	2020.06.01	NULL	1.458546423213736	E-10030	chembl:CHEMBL3301576	PEGPLERANIB SODIUM	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.2778183663264259	SNDX-275	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	7.001022831425932	Telcagepant	ncit:C152545	TELCAGEPANT	FALSE	FALSE	FALSE
NCBIGENE:1878	ncbigene:1878	E11S	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:12060	iuphar.ligand:12060	BT7480	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005864158	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.033583416	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NCBIGENE:1446	hgnc:2445	CSN1S1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:10210	iuphar.ligand:10210	I3MT-3	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.037721028	IUPHAR.LIGAND:2	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.06466462	IUPHAR.LIGAND:3	iuphar.ligand:3	1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:44	iuphar.ligand:44	NAFADOTRIDE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:6	iuphar.ligand:6	7-METHOXY-1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:5620	iuphar.ligand:5620	PSB-11	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:474	iuphar.ligand:474	MRS1523	FALSE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TdgClinicalTrial	Jan-14	NULL	1.123158743009508	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:404	iuphar.ligand:404	XANTHINE AMINE CONGENER	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:373	iuphar.ligand:373	2-HEXYNYL-NECA	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.072125922	IUPHAR.LIGAND:422	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:390	iuphar.ligand:390	MRE 2029F20	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:449	iuphar.ligand:449	MRS1754	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:439	iuphar.ligand:439	AS74	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.09741683	IUPHAR.LIGAND:403	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:454	iuphar.ligand:450	OSIP339391	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:3289	iuphar.ligand:3289	BAY 60-6583	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.077330885	IUPHAR.LIGAND:422	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:11277	iuphar.ligand:11277	AZD1390	FALSE	FALSE	FALSE
VITAMIN K EPOXIDE REDUCTASE COMPLEX 1	hgnc:23663	VKORC1	TTD	2020.06.01	NULL	7.001022831425932	Phenindione	rxcui:8130	PHENINDIONE	TRUE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:8061	iuphar.ligand:8061	MK-5108	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:8354	iuphar.ligand:8354	HESPERADIN	FALSE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:8768	iuphar.ligand:8768	COMPOUND 38 [PMID: 20817473]	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.1367387271762877	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	1.591141552596802	IUPHAR.LIGAND:3416	iuphar.ligand:3391	5-OXO-ETE	FALSE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	NULL	2.625383561784724	IUPHAR.LIGAND:11726	iuphar.ligand:11726	COMPOUND 20 [PMID: 34432979]	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:635	iuphar.ligand:635	D-NAL-CYS-TYR-D-TRP-LYS-VAL-CYS-NAL-NH2	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:626	iuphar.ligand:626	PD 176252	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:6178	iuphar.ligand:6178	NEUROMEDIN C	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:627	iuphar.ligand:627	[(3-PH-PR6), HIS7,D-ALA11,D-PRO13,&PSI;13-14),PHE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10520	iuphar.ligand:10520	AM-6494	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:9963	iuphar.ligand:9963	ATABECESTAT	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:549	rxcui:1520	BETAXOLOL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:549	rxcui:1520	BETAXOLOL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:7297	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.5645986154375752	IUPHAR.LIGAND:562	iuphar.ligand:562	[125I]ICYP	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:11544	iuphar.ligand:11544	BELVARAFENIB	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:3697	iuphar.ligand:3697	R-SPONDIN-1	FALSE	FALSE	FALSE
NCBIGENE:1587	hgnc:209	ADAM3A	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8627	iuphar.ligand:8627	COMPOUND 1B [PMID: 18078750]	FALSE	FALSE	FALSE
NCBIGENE:2598	hgnc:1372	CA14	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:3310	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:6829	rxcui:6845	METHOCARBAMOL	TRUE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:7046	iuphar.ligand:7046	INDISULAM	FALSE	FALSE	FALSE
NCBIGENE:1998	hgnc:3317	ELF2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12692	iuphar.ligand:12692	SR-4133	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	0.252440727	IUPHAR.LIGAND:717	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
NCBIGENE:2346	hgnc:3788	FOLH1	GuideToPharmacology	2024.1	inhibitor	0.6482428547616604	IUPHAR.LIGAND:8674	iuphar.ligand:8674	GRASSYSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2346	hgnc:3788	FOLH1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:6566	iuphar.ligand:6566	COMPOUND 2 [PMID: 8410973]	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2088	iuphar.ligand:2088	KASSININ	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.1436598392221464	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:734	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:747	iuphar.ligand:747	JWH-133	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:6666	iuphar.ligand:6666	[125I]DTYR-GLY-[(NLE28,31)CCK-26-33	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.023598953	IUPHAR.LIGAND:7671	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.038131933	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.029498692	IUPHAR.LIGAND:7625	iuphar.ligand:7625	BP 897	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.1179947668217853	IUPHAR.LIGAND:6675	iuphar.ligand:6675	PG01037	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:980	ncit:C73294	SONEPIPRAZOLE	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:3302	iuphar.ligand:3302	L741742	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.095122593	IUPHAR.LIGAND:2	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.1000146118775133	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:1232	hgnc:1604	CCR3	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:11758	iuphar.ligand:11758	MUPADOLIMAB	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.4688184931758437	CEFOXITIN	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2012	hgnc:3333	EMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8128	iuphar.ligand:8128	COMPOUND 1A [PMID: 24900749]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:7647	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:7879	iuphar.ligand:7879	BMS-690514	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.2333674277141978	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:12750	iuphar.ligand:12750	EC5026	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.097236428	IUPHAR.LIGAND:1916	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1917	iuphar.ligand:1917	CICAPROST	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1928	iuphar.ligand:1928	AH13205	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.2160809515872201	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	0.6482428547616604	IUPHAR.LIGAND:10603	iuphar.ligand:10603	TG11-77	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:1967	ncit:C76896	BERAPROST	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:5822	iuphar.ligand:5822	DG-041	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	NULL	0.9053046764774912	IUPHAR.LIGAND:5031	iuphar.ligand:5031	NEUREGULIN-4	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.031822831	IUPHAR.LIGAND:2820	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.031822831	IUPHAR.LIGAND:2820	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:2823	ncit:C545	HEXESTROL	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:8908	iuphar.ligand:8908	GSK5182	FALSE	FALSE	FALSE
NCBIGENE:622	hgnc:1027	BDH1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:2833	drugbank:DB06833	1-CYCLOHEXYL-N-{[1-(4-METHYLPHENYL)-1H-INDOL-3-YL]METHYL}METHANAMINE	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.2323348284765243	demeclocycline	rxcui:3154	DEMECLOCYCLINE	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:995	iuphar.ligand:995	SARAFOTOXIN S6B	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.087512785	IUPHAR.LIGAND:2820	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2651	hgnc:4204	GCNT2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7017	iuphar.ligand:7017	UNC0642	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	ChEMBL	33	inhibitor	0.1553481397505754	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
NCBIGENE:2652	hgnc:4206	OPN1MW	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7375	iuphar.ligand:7375	BRD9539	FALSE	FALSE	FALSE
NCBIGENE:2652	hgnc:4206	OPN1MW	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7017	iuphar.ligand:7017	UNC0642	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:1382	iuphar.ligand:1382	CPCCOET	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:12109	iuphar.ligand:12109	BMS-986339	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3151	iuphar.ligand:3151	DIPHOSPHORIC ACID	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	1.193356164447602	IUPHAR.LIGAND:9798	iuphar.ligand:9798	DARIGABAT	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.1988926940746003	IUPHAR.LIGAND:4321	iuphar.ligand:4321	TETRAHYDRODEOXYCORTICOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.4605936073306534	IUPHAR.LIGAND:4296	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.1151484018326633	IUPHAR.LIGAND:4367	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:4197	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.055271233	IUPHAR.LIGAND:6963	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.2134458180312784	IUPHAR.LIGAND:4296	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4095	iuphar.ligand:4095	&ALPHA;5IA	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4257	iuphar.ligand:4257	MRK016	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	inhibitor	0.1829535583125243	IUPHAR.LIGAND:2312	iuphar.ligand:2312	BICUCULLINE	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:4067	iuphar.ligand:4067	(&PLUSMN;)-CIS-2-CAMP	FALSE	FALSE	FALSE
NCBIGENE:240	hgnc:435	ALOX5	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:1066	iuphar.ligand:1066	CGP 47656	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.4145342465975881	MGAH22	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:3900	iuphar.ligand:3900	M871	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:5871	iuphar.ligand:5871	ABBOTT 14C	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:1101	iuphar.ligand:1101	BIM 28163	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:9734	iuphar.ligand:9734	LIVER ENRICHED ANTIMICROBIAL PEPTIDE 2	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4245	ncit:C80379	TEZAMPANEL ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:250	hgnc:439	ALPP	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:1143	iuphar.ligand:1143	GLUCAGON-LIKE PEPTIDE 2-(3-33)	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:12583	iuphar.ligand:12583	NVP-DKY709	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:1138	ncit:C133230	AVEXITIDE	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.1389091831632129	IUPHAR.LIGAND:4167	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11309	iuphar.ligand:11309	4‐BCCA	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.2917092846427472	IUPHAR.LIGAND:4133	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.6563458904461812	IUPHAR.LIGAND:4219	iuphar.ligand:4219	IDRA-21	FALSE	FALSE	FALSE
NCBIGENE:666	hgnc:1087	BOK	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:12431	rxcui:15842	5-METHOXYPSORALEN	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:4141	iuphar.ligand:4141	ATPO	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.305277158	IUPHAR.LIGAND:7079	rxcui:4491	FLUOROMETHOLONE	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	modulator	0.1187956362798518	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.1221108633388244	IUPHAR.LIGAND:7061	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:3445	iuphar.ligand:3445	RU28362	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	0.3947945205691315	IUPHAR.LIGAND:4075	iuphar.ligand:4075	[3H]SYM2081	FALSE	FALSE	FALSE
NCBIGENE:2798	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	modulator	0.3977853881492007	IUPHAR.LIGAND:12124	ncit:C169919	DORZAGLIATIN	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	blocker	0.1521961485092594	IUPHAR.LIGAND:4128	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.108711535	IUPHAR.LIGAND:2361	drugbank:DB01931	5,7-DICHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	modulator	0.093596562	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	modulator	0.2375912725597036	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	CALPEPTIN	iuphar.ligand:11643	CALPEPTIN	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:9810	iuphar.ligand:9810	COMPOUND 2F [JIANG ET AL., 2018]	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.1271372184883643	IUPHAR.LIGAND:8114	drugbank:DB07149	(7S)-2-(2-AMINOPYRIMIDIN-4-YL)-7-(2-FLUOROETHYL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4490	iuphar.ligand:4490	[3H]GSK931145	FALSE	FALSE	FALSE
NCBIGENE:403	hgnc:694	ARL3	GuideToPharmacology	2024.1	blocker	0.9376369863516875	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	0.030246354	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:11118	drugbank:DB14979	MARTINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:10490	iuphar.ligand:10490	SS-208	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:9702	iuphar.ligand:9702	TUBASTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:7008	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.1835932560688619	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:1254	iuphar.ligand:1254	METHIMEPIP	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:9879	iuphar.ligand:9879	H4 ANTAGONIST 48	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:3319	iuphar.ligand:3319	PSN632408	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:3623	iuphar.ligand:3623	OLEOYL-LYSOPHOSPHATIDYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	1.591141552596802	IUPHAR.LIGAND:3354	iuphar.ligand:3354	LTC4	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:5525	iuphar.ligand:5525	O-1602	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5524	iuphar.ligand:5524	ASN06917370	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:3635	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:123	hgnc:248	PLIN2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:7798	iuphar.ligand:7798	COMPOUND 2 [PMID: 24793972]	FALSE	FALSE	FALSE
NCBIGENE:147	hgnc:278	ADRA1B	GuideToPharmacology	2024.1	agonist	0.2536602475154323	IUPHAR.LIGAND:3700	iuphar.ligand:3700	R-SPONDIN-4	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.2885036881082115	IUPHAR.LIGAND:1635	iuphar.ligand:1635	CTAP	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:1640	iuphar.ligand:1640	NALTRIBEN	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.028444026	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.1773907812016706	IUPHAR.LIGAND:7118	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.074690855	IUPHAR.LIGAND:2147	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:7545	iuphar.ligand:7545	N-DESALKYLQUETIAPINE	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.054581779	IUPHAR.LIGAND:202	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:3112	hgnc:4937	HLA-DOB	GuideToPharmacology	2024.1	NULL	13.12691780892362	IUPHAR.LIGAND:12060	iuphar.ligand:12060	BT7480	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.1646008502686348	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	modulator	1.346350544504987	IUPHAR.LIGAND:12170	iuphar.ligand:12170	UCM-1306	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.088695391	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:8909	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:11198	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8071	iuphar.ligand:8071	GNF-5837	FALSE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:9537	iuphar.ligand:9537	ATRACURIUM	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:9537	iuphar.ligand:9537	ATRACURIUM	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:3994	ncit:C66518	RIVANICLINE	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	0.4412409347537352	IUPHAR.LIGAND:2906	iuphar.ligand:2906	LPA	FALSE	FALSE	FALSE
NCBIGENE:2117	hgnc:3492	ETV3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8149	iuphar.ligand:8149	COMPOUND 2 [PMID: 21627121]	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.094608417	IUPHAR.LIGAND:7266	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2113	iuphar.ligand:2113	[PHE(ME)7]NEUROKININ B	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:2111	ncit:C152301	SAREDUTANT	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:3522	iuphar.ligand:3522	RP67580	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:7927	iuphar.ligand:7927	COMPOUND 6B [PMID: 24999562]	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:7928	iuphar.ligand:7928	PEG40-NMU	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1690	iuphar.ligand:1690	[F/G]N/OFQ-(1-13)-NH2	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	CIViC	10-Apr-24	NULL	0.1752202599633854	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:11235	iuphar.ligand:11235	COMPOUND 46 [PMID: 25268943]	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:4037	iuphar.ligand:4037	EMPA	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9306	iuphar.ligand:9306	MK-1064	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:9308	iuphar.ligand:9308	SELTOREXANT	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:4037	iuphar.ligand:4037	EMPA	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9303	iuphar.ligand:9303	ACT-462206	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:1704	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	modulator	1.640864726115453	IUPHAR.LIGAND:6496	iuphar.ligand:6496	MRS 2219	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:5909	iuphar.ligand:5909	MRS2802	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.087952548	IUPHAR.LIGAND:1732	iuphar.ligand:1732	AP4A	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:6148	iuphar.ligand:6148	COMPOUND 4 [PMID: 23083103]	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	CID 5310655	chembl:CHEMBL408563	CHEMBL:CHEMBL408563	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:1771	iuphar.ligand:1771	R-138727	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.1319288222002374	IUPHAR.LIGAND:1764	iuphar.ligand:1764	2MESAMP	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:1732	iuphar.ligand:1732	AP4A	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:5903	iuphar.ligand:5903	MRS2957	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8333	iuphar.ligand:8333	CYCLIC INSL3 B-CHAIN ANALOGUE 6	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:1989	iuphar.ligand:1989	RELAXIN	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:11916	iuphar.ligand:11916	&DELTA;R3/I5	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.2286255641612242	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:10309	iuphar.ligand:10309	RP-001	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1356787370431382	IUPHAR.LIGAND:7285	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:2199	hgnc:3601	FBLN2	GuideToPharmacology	2024.1	inhibitor	0.4565884455277782	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:11672	ncit:C167205	SUNVOZERTINIB	FALSE	FALSE	FALSE
NCBIGENE:2969	hgnc:4659	GTF2I	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:6149	iuphar.ligand:6149	IL-37	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:11586	ncit:C171846	BLARCAMESINE	FALSE	FALSE	FALSE
NCBIGENE:960	hgnc:1681	CD44	GuideToPharmacology	2024.1	NULL	1.381780822	IUPHAR.LIGAND:4546	iuphar.ligand:4546	[3H]TAUROCHOLIC ACID	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:4754	rxcui:1545653	EMPAGLIFLOZIN	TRUE	FALSE	FALSE
NCBIGENE:960	hgnc:1681	CD44	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:6530	iuphar.ligand:6530	SC-435	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10000	iuphar.ligand:10000	GUSACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10219	iuphar.ligand:10219	MP-A08	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6041	iuphar.ligand:6041	SKI II	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:6623	iuphar.ligand:6623	PF-543	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.9907107780319716	LINSITINIB	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
NCBIGENE:1418	hgnc:2408	CRYGA	GuideToPharmacology	2024.1	inhibitor	7.501095890813499	IUPHAR.LIGAND:8787	iuphar.ligand:8787	COMPOUND 12E [PMID: 18605714]	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:8172	iuphar.ligand:8172	COMPOUND 7 [PMID: 22464456]	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:6623	iuphar.ligand:6623	PF-543	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:8183	iuphar.ligand:8183	PD166285	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:10598	iuphar.ligand:10598	COMPOUND 41 [PMID: 31855425]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2051	ncit:C152317	SEGLITIDE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:2027	iuphar.ligand:2027	BIM 23627	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:2029	iuphar.ligand:2029	[L-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:9632	iuphar.ligand:9632	CIS-1,2-CYCLOPROPANEDICARBOXYLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:9348	iuphar.ligand:9348	COMPOUND 5 [PMID: 17618114]	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	inhibitor	0.2548916079402645	IUPHAR.LIGAND:2633	iuphar.ligand:2633	NH-3	FALSE	FALSE	FALSE
NCBIGENE:392	hgnc:673	ARHGAP1	GuideToPharmacology	2024.1	blocker	1.458546423213736	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:1911	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8246	iuphar.ligand:8246	SD-208	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:9718	iuphar.ligand:9718	GSK2256294	FALSE	FALSE	FALSE
NCBIGENE:2421	hgnc:3931	FRA8C	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:6432	ncit:C73213	CAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.025942525	IUPHAR.LIGAND:2585	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:10285	iuphar.ligand:10285	CLEMIZOLE	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.1426838892274307	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	activator	1.141471113819445	IUPHAR.LIGAND:10278	iuphar.ligand:10278	GSK1702934A	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.172722603	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.1363835616511545	IUPHAR.LIGAND:2489	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:4213	iuphar.ligand:4213	HC067047	FALSE	FALSE	FALSE
NCBIGENE:255	hgnc:12373	TSHR	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:3806	iuphar.ligand:3806	[125I]TSH (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2245	hgnc:3663	FGD1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9929	iuphar.ligand:9929	XILIERTINIB	FALSE	FALSE	FALSE
PSMA2	hgnc:9531	PSMA2	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:2246	hgnc:3665	FGF1	GuideToPharmacology	2024.1	inhibitor	0.2536602475154323	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	NULL	0.2117244807890907	IUPHAR.LIGAND:12310	iuphar.ligand:12310	SJ988497	FALSE	FALSE	FALSE
NCBIGENE:3209	hgnc:5102	HOXA13	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12224	iuphar.ligand:12224	COMPOUND 61 [PMID: 36221183]	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:2790	rxcui:11516	DOXERCALCIFEROL	TRUE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:2777	ncit:C26669	SEOCALCITOL	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.053579256	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2268	iuphar.ligand:2268	PG 97-269	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2778183663264258	IUPHAR.LIGAND:2180	iuphar.ligand:2180	[VAL4]AVP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2192	iuphar.ligand:2192	LS-192629	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.019490598	IUPHAR.LIGAND:2185	iuphar.ligand:2185	D[D-PHE2]AVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.014617949	IUPHAR.LIGAND:2169	ncit:C87380	ARGIPRESTOCIN	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:2206	iuphar.ligand:2206	[125I]3-N3-PHPA-LVA	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.058471794	IUPHAR.LIGAND:2191	iuphar.ligand:2191	D[LEU4]LVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:2185	iuphar.ligand:2185	D[D-PHE2]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:2216	iuphar.ligand:2216	D(CH2)5[D-TYR(ET)2,VAL4,TYR-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	NULL	0.8751278539282416	IUPHAR.LIGAND:3817	iuphar.ligand:3817	[3H]DESGLY-NH2[D-ILE2,ILE4]VP	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1545	iuphar.ligand:1545	[LEU31,PRO34]NPY	FALSE	FALSE	FALSE
PRPS1	hgnc:9462	PRPS1	CIViC	10-Apr-24	NULL	0.5303805175322677	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.099446347	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NT5C2	hgnc:8022	NT5C2	CIViC	10-Apr-24	NULL	0.2651902587661338	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	CIViC	10-Apr-24	NULL	0.091732479	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
SLFN11	hgnc:26633	SLFN11	CIViC	10-Apr-24	NULL	0.6482428547616604	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
PPY	hgnc:9327	PPY	NCI	14-Sep-17	NULL	1.842374429322614	ONDANSETRON	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
AKT2	hgnc:392	AKT2	CIViC	10-Apr-24	NULL	0.04321619	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.1848861663228679	RAPALINK-1	iuphar.ligand:9212	RAPALINK-1	FALSE	FALSE	TRUE
NCBIGENE:1381	hgnc:2338	CRABP1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11392	iuphar.ligand:11392	TFC007	FALSE	FALSE	FALSE
GNAQ	hgnc:4390	GNAQ	CIViC	10-Apr-24	NULL	0.8204323630577265	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
IGF2	hgnc:5466	IGF2	CIViC	10-Apr-24	NULL	0.035145697	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.005847179	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
IGF2	hgnc:5466	IGF2	CIViC	10-Apr-24	NULL	0.1325951293830669	CABAZITAXEL	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.097236428	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	CIViC	10-Apr-24	NULL	0.006794471	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NCBIGENE:607	hgnc:1008	BCL9	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:2757	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
SGK1	hgnc:10810	SGK1	CIViC	10-Apr-24	NULL	0.5000730593875666	ALPELISIB	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.02302968	ZOLEDRONIC ACID	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	CIViC	10-Apr-24	NULL	0.039778539	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CDK4	hgnc:1773	CDK4	CIViC	10-Apr-24	NULL	0.029074015	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
AKT3	hgnc:393	AKT3	CIViC	10-Apr-24	NULL	1.640864726115453	PAN-AKT KINASE INHIBITOR GSK690693	ncit:C71711	PAN-AKT KINASE INHIBITOR GSK690693	FALSE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.092606122	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.3241214273808302	TYRPHOSTIN AG 1295	ncit:C2031	TYRPHOSTIN AG 1295	FALSE	FALSE	TRUE
RAC1	hgnc:9801	RAC1	CIViC	10-Apr-24	NULL	0.2160809515872201	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1245241215075758	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.006297772	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.088396753	Niclosamide	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.093596562	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	1.438566335224506	ART0380	ncit:C179292	ATR INHIBITOR ART0380	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.1438566335224507	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.1598407039138341	AZD6482	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.068727318	Ganetespib	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.043636393	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1694	iuphar.ligand:1694	UFP-101	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6373	rxcui:1546400	PERINDOPRILAT	TRUE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.072424374	IUPHAR.LIGAND:1059	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:2323	iuphar.ligand:2323	CYPPA	FALSE	FALSE	FALSE
R-SPONDIN-3	hgnc:20866	RSPO3	TTD	2020.06.01	NULL	52.50767123569449	Rosmantuzumab	ncit:C122921	ROSMANTUZUMAB	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.5114383561918295	REFAMETINIB	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.145450613	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1339481409073839	ERGOTAMINE TARTRATE	rxcui:42676	ERGOTAMINE TARTRATE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.297915865	AMLODIPINE BESYLATE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.064824285	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.003632492	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.013259513	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	DIMETHYLPHENYLPIPERAZINIUM	iuphar.ligand:3967	DMPP	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1861974157294131	CHRYSIN DIMETHYL ETHER	chembl:CHEMBL275391	CHRYSIN DIMETHYL ETHER	FALSE	FALSE	FALSE
PRKAB1	hgnc:9378	PRKAB1	NCI	14-Sep-17	NULL	0.6563458904461813	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.045579576	MRS-1523	iuphar.ligand:474	MRS1523	FALSE	FALSE	FALSE
REACTIVE OXYGEN SPECIES	hgnc:10261	ROS1	TTD	2020.06.01	NULL	0.546954909	Tafenoquine	rxcui:2054023	TAFENOQUINE	TRUE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.053253216	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:1358	iuphar.ligand:1358	4P-PDOT	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.009211872	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.007435241	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005903055	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.1223955040459079	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
KLK3	hgnc:6364	KLK3	ChEMBL	33	binder	0.4375639269641208	CAPROMAB	ncit:C174682	CAPROMAB	TRUE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.2206204673768676	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	(+)-THALIPORPHINE	chembl:CHEMBL1397308	CHEMBL:CHEMBL1397308	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	JNJ-68284528	ncit:C148498	CILTACABTAGENE AUTOLEUCEL	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.062509132	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	1.009762908	LXH254	chembl:CHEMBL4583691	LXH254	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.020391329	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.013113804	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.172722603	PELITINIB	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.305277158	Fadolmidine	ncit:C75054	FADOLMIDINE	FALSE	FALSE	FALSE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	0.03070624	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:400	hgnc:692	ARL1	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:11060	iuphar.ligand:11060	PF-956980	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	modulator	0.1835932560688619	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:2673	hgnc:4241	GFPT1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8230	iuphar.ligand:8230	IOX1	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9306	iuphar.ligand:9306	MK-1064	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	activator	0.3088686543276147	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.072927321	IUPHAR.LIGAND:6044	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1682938180631233	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	DTC	9/2/20	NULL	0.9546849315580818	HU-308	ncit:C184881	ONTERNABEZ	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	PharmGKB	4/5/24	NULL	0.1555782851427985	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	PharmGKB	4/5/24	NULL	0.1196983386831941	niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:12718	ncit:C146660	MEZIGDOMIDE	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.064268875	IUPHAR.LIGAND:7080	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.087222045	ERGOTAMINE TARTRATE	rxcui:42676	ERGOTAMINE TARTRATE	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.031555091	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.038837035	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	TCMDC-125195	chembl:CHEMBL531709	CHEMBL:CHEMBL531709	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.049723174	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	CHLORTHALIDONE	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
GADD45A	hgnc:4095	GADD45A	NCI	14-Sep-17	NULL	0.1551950873961413	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.6908904109959803	HEXYLCAINE	rxcui:26879	HEXYLCAINE	TRUE	FALSE	FALSE
RPL9	hgnc:10369	RPL9	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1286952726365061	MK-212	drugbank:DB12111	MK-212	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.004428785	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.094535416	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.5125748858722557	IUPHAR.LIGAND:6495	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	2.625383561784724	BASIC FIBROBLAST GROWTH FACTOR	drugbank:DB14131	BASIC FIBROBLAST GROWTH FACTOR	FALSE	FALSE	FALSE
F3	hgnc:3541	F3	ChEMBL	33	binder	0.2187819634820604	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.04321619	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
PSMC6	hgnc:9553	PSMC6	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	THEONELLASTEROL B	chembl:CHEMBL1782598	THEONELLASTEROL B	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.034184682	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	1.419126249613364	PBF509	iuphar.ligand:10193	PBF-509	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.026885648	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1842374429322613	U0126	iuphar.ligand:5282	U0126	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	RG-7160	chembl:CHEMBL2109393	RG-7160	FALSE	FALSE	FALSE
OPRL1	hgnc:8155	OPRL1	ChEMBL	33	inhibitor	6.563458904461812	LY-2940094	iuphar.ligand:9462	LY2940094	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
SMAD7	hgnc:6773	SMAD7	PharmGKB	4/5/24	NULL	2.187819634820604	tegafur	rxcui:10995	URACIL	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.5585922471882393	CYCLOPENTOLATE	rxcui:3001	CYCLOPENTOLATE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.069824031	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:8698	iuphar.ligand:8698	COMPOUND 16 [PMID: 23412139]	FALSE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.577007376	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	U0126	iuphar.ligand:5282	U0126	FALSE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.055504938	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:470	iuphar.ligand:470	MRS1191	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.09741683	IUPHAR.LIGAND:3283	iuphar.ligand:3283	SCH442416	FALSE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	blocker	0.3431873936973497	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.019665794	IUPHAR.LIGAND:129	iuphar.ligand:129	S33084	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:5701	iuphar.ligand:5701	PI-103	FALSE	FALSE	FALSE
CA12	hgnc:1371	CA12	ChEMBL	33	inhibitor	0.9376369863516875	ACETAZOLAMIDE SODIUM	rxcui:91406	ACETAZOLAMIDE SODIUM	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.008599357	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.020737627	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5556367326528519	ICOTINIB	ncit:C138996	ICOTINIB	FALSE	FALSE	TRUE
UNIPROT:P35228	hgnc:7873	NOS2	TdgClinicalTrial	Jan-14	NULL	0.6081969641200136	TILARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.1060761035064535	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
KCNH4	hgnc:6253	KCNH4	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.075768645	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	PharmGKB	4/5/24	NULL	0.034727296	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
E3 UBIQUITIN-PROTEIN LIGASE COP1	hgnc:17440	COP1	TTD	2020.06.01	NULL	1.050153425	Flecainide	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.09699693	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.2375912725597036	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	0.7955707762984013	Desmopressin	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:373	iuphar.ligand:373	2-HEXYNYL-NECA	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.035098711	IUPHAR.LIGAND:7933	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:8383	iuphar.ligand:8383	BIMIRALISIB	FALSE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	0.5048814541893701	ACETAZOLAMIDE SODIUM	rxcui:91406	ACETAZOLAMIDE SODIUM	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1400204566285186	PYRACLOSTROBIN	chembl:CHEMBL519873	PYRACLOSTROBIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	THIOTHIXENE	rxcui:10510	THIOTHIXENE	TRUE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.1209854175937661	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	inhibitor	1.009762908	DACLIZUMAB	rxcui:190353	DACLIZUMAB	TRUE	TRUE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.055504938	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:8369	iuphar.ligand:8369	MLS1547	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.6250913242344582	DSP-2230	chembl:CHEMBL5095026	DSP-2230	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.8751278539282416	arformoterol	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
NCBIGENE:1888	hgnc:3143	EBVS1	GuideToPharmacology	2024.1	NULL	2.187819634820604	IUPHAR.LIGAND:4872	iuphar.ligand:4872	BDNF	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.021742307	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.014369915	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
PADI4	hgnc:18368	PADI4	DTC	9/2/20	NULL	4.375639269641208	O-F-AMIDINE	iuphar.ligand:8625	O-F-AMIDINE	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:10461	iuphar.ligand:10461	FADRACICLIB	FALSE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	ChEMBL	33	positive modulator	0.1591141552596803	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.055271233	AZD-4547	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	7.501095891	BUSERELIN ACETATE	rxcui:42569	BUSERELIN ACETATE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.058406753	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:2220	hgnc:3624	FCN2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
LRRC15	hgnc:20818	LRRC15	PharmGKB	4/5/24	NULL	2.692701089009974	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1041818873724097	PKI-592	ncit:C84837	PI3K/MTOR KINASE INHIBITOR PF-04691502	FALSE	FALSE	TRUE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:12721	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
NCBIGENE:2951	hgnc:4640	GSTP1P1	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:9686	rxcui:2602286	TAPINAROF	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.069454592	sacituzumab govitecan-hziy	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
VASOPRESSIN V1B RECEPTOR	hgnc:896	AVPR1B	TTD	2020.06.01	NULL	1.666910197958555	Desmopressin	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ATRANORIN	chembl:CHEMBL173395	ATRANORIN	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.2117244807890907	Mepyramine maleate	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:541	iuphar.ligand:541	CGP 20712A	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.035122188	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.058799184	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.082559232	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.0191914	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1207072901969988	NSC-117271	chembl:CHEMBL287689	CHEMBL:CHEMBL287689	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:607	iuphar.ligand:607	ALX40-4C	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.059330702	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:7597	rxcui:1546365	PRALIDOXIME CATION	TRUE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:12074	iuphar.ligand:12074	ASNUCICLIB	FALSE	FALSE	FALSE
INHBA	hgnc:6066	INHBA	ChEMBL	33	inhibitor	26.25383561784724	GARETOSMAB	ncit:C170022	GARETOSMAB	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.1988926940746004	TRANILAST	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6140	iuphar.ligand:6140	GALANIN(1-10)	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.067231333	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
KCNH7	hgnc:18863	KCNH7	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011762471	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.4375639269641208	levamisole	rxcui:6371	LEVAMISOLE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	FENCAMFAMINE	ncit:C87695	FENCAMFAMIN	TRUE	FALSE	FALSE
NCBIGENE:434	hgnc:745	ASIP	GuideToPharmacology	2024.1	activator	10.50153424713889	IUPHAR.LIGAND:10260	iuphar.ligand:10260	VU0810464	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:3392	iuphar.ligand:3392	5-OXO-C20:3	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	2.282942227638891	PALBINONE	chembl:CHEMBL575924	PALBINONE	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.085009721	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1241316104862754	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:8868	iuphar.ligand:8868	SCH221510	FALSE	FALSE	FALSE
NCBIGENE:2239	hgnc:4452	GPC4	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8119	iuphar.ligand:8119	COMPOUND 35 [PMID: 22902653]	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.077217164	Surufatinib	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.2318219480604613	p28	iuphar.ligand:6152	IL-27 SUBUNIT &ALPHA;	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CGI	2/1/22	NULL	0.6721614540713904	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	blocker	0.078136416	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	EPITINIB	iuphar.ligand:11608	EPITINIB	FALSE	FALSE	FALSE
RPS23	hgnc:10410	RPS23	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.025244073	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.096521454	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.2631963470460877	PROSTAGLANDIN D2	drugbank:DB02056	PROSTAGLANDIN D2	FALSE	FALSE	FALSE
GRM2	hgnc:4594	GRM2	NCI	14-Sep-17	NULL	1.250182648468916	OPIATE	ncit:C1657	OPIATE	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.5676505	BENZODIAZEPINE	ncit:C1012	BENZODIAZEPINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SKF-62604	chembl:CHEMBL346551	CHEMBL:CHEMBL346551	FALSE	FALSE	FALSE
NCBIGENE:1816	hgnc:3026	DRD5	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	LINSIDOMINE	ncit:C72628	LINSIDOMINE	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.067883221	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:10717	iuphar.ligand:10717	PSB-1584	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.037948209	perhexiline	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.7721716358190367	IUPHAR.LIGAND:10284	iuphar.ligand:10284	GSK2833503A	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.009787078	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	GERONTOXANTHONE H	chembl:CHEMBL514057	GERONTOXANTHONE H	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	CKD-516	ncit:C101264	VALECOBULIN	FALSE	FALSE	FALSE
HYOU1	hgnc:16931	HYOU1	DTC	9/2/20	NULL	11.66837138570989	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CancerCommons	25-Jul-13	inhibitor	0.5498185469706229	PLX3603	ncit:C92591	BRAF(V600E) KINASE INHIBITOR RO5212054	FALSE	FALSE	TRUE
UNIPROT:P16234	hgnc:8803	PDGFRA	TEND	1-Aug-11	NULL	0.8607814956671229	BECAPLERMIN	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.020351811	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.102191151	alendronate	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.2154897588332195	yohimbine	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.073954467	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.012291122	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.6250913242344582	HT-0712	drugbank:DB11650	HT-0712	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.2386712328895204	NSC-353263	chembl:CHEMBL1383812	CHEMBL:CHEMBL1383812	FALSE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.081030357	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	AZD5153	ncit:C151943	BIVALENT BRD4 INHIBITOR AZD5153	FALSE	FALSE	FALSE
NCBIGENE:1567	hgnc:29499	ERAP2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8666	iuphar.ligand:8666	COMPOUND 17 [PMID: 23916253]	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.6604738520213144	ISTIRATUMAB	ncit:C103863	ISTIRATUMAB	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	1.521961485092594	ALVESPIMYCIN	ncit:C38142	ALVESPIMYCIN	FALSE	FALSE	TRUE
UNIPROT:Q96KS0	hgnc:14660	EGLN2	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	FG-4592	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:2077	hgnc:3444	ERF	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:3887	iuphar.ligand:3887	IRL 2500	FALSE	FALSE	FALSE
GSC1	hgnc:4612	GSC	ChEMBL	33	inhibitor	10.50153424713889	IBREXAFUNGERP	rxcui:2560213	IBREXAFUNGERP	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:2609	iuphar.ligand:2609	APETX-1	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1093909817410302	GW9662	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	DTC	9/2/20	NULL	3.938075342677087	TAK-220	iuphar.ligand:800	TAK-220	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.030814361	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.053854022	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P23415	hgnc:4326	GLRA1	TdgClinicalTrial	Jan-14	NULL	0.1539814405738841	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UGT1A	hgnc:12529	UGT1A	PharmGKB	4/5/24	NULL	0.4167275494896388	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:Q07820	hgnc:32041	ADAMTSL4-AS1	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	AT-101	ncit:C187300	ANTI-CD19 CAR T CELLS AT101	FALSE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.7160136986685613	LEVOBUNOLOL	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
NCBIGENE:596	hgnc:990	BCL2	GuideToPharmacology	2024.1	agonist	0.2134458180312784	IUPHAR.LIGAND:8901	iuphar.ligand:8901	SR9009	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:6118	iuphar.ligand:6118	GALNON	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:4854	iuphar.ligand:4854	E. COLI HEAT-STABLE ENTEROTOXIN (STA)	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:2066	iuphar.ligand:2066	PRL-2915	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.5000730593875667	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.065145994	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	LERCANIDIPINE HYDROCHLORIDE	rxcui:153679	LERCANIDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	1.514644363	ALMOTRIPTAN	rxcui:279645	ALMOTRIPTAN	TRUE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.032694689	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	1.357957014716237	INNO-206	ncit:C68921	ALDOXORUBICIN	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.024275391	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	TCMDC-123528	chembl:CHEMBL529138	CHEMBL:CHEMBL529138	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.3621218705909966	DEXRAZOXANE	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.6783936852156912	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.025421288	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	0.3860858179095184	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	7.501095891	s-adenosylmethionine	rxcui:9504	S-ADENOSYLMETHIONINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-11437	chembl:CHEMBL1814509	CHEMBL:CHEMBL1814509	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-668	chembl:CHEMBL604528	CHEMBL:CHEMBL604528	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	1.514644363	RO5520985	ncit:C118578	VANUCIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:9382	iuphar.ligand:9382	NVP-TAE 226	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.017724108	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	2.308029504865692	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.078136416	ERGOTAMINE TARTRATE	rxcui:42676	ERGOTAMINE TARTRATE	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2220197515251353	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
UNIPROT:Q9P0X4	hgnc:1396	CACNA1I	TdgClinicalTrial	Jan-14	NULL	0.4546118721705151	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	1.458546423213736	imidapril	rxcui:60245	IMIDAPRIL	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.058602312	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.3571950424196904	TRILACICLIB	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	1.250182648468916	ERTEBEREL	ncit:C166610	ERTEBEREL	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.3125456621172291	GNF-PF-3955	chembl:CHEMBL605747	CHEMBL:CHEMBL605747	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.2375912725597036	IUPHAR.LIGAND:8204	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.038382801	IUPHAR.LIGAND:2055	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.047734247	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
VALOSIN-CONTAINING PROTEIN P97	hgnc:12666	VCP	TTD	2020.06.01	NULL	35.00511415712966	CB-5083	drugbank:DB16874	CB-5083	FALSE	FALSE	FALSE
NATRIURETIC PEPTIDE RECEPTOR	hgnc:7945	NPR3	TTD	2020.06.01	NULL	26.25383561784724	ANX-042	chembl:CHEMBL4594397	ANX-042	FALSE	FALSE	FALSE
NCBIGENE:3014	hgnc:4739	H2AX	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:10036	rxcui:2178390	SELINEXOR	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
SCNN1G	hgnc:10602	SCNN1G	ChEMBL	33	blocker	1.458546423213736	AMILORIDE HYDROCHLORIDE	rxcui:142424	AMILORIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.172722603	PELITINIB	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	4-METHYLDAPHNETIN	chembl:CHEMBL276618	4-METHYLDAPHNETIN	FALSE	FALSE	FALSE
UNIPROT:P43357	hgnc:6801	MAGEA3	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	MAGE-A3	ncit:C78478	ASTUPROTIMUT-R	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
UNIPROT:Q9H3N8	hgnc:17383	HRH4	TEND	1-Aug-11	NULL	0.098421127	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
LIPE	hgnc:6621	LIPE	NCI	14-Sep-17	NULL	1.381780822	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	positive modulator	0.2734774543525755	MEVIDALEN	ncit:C175136	MEVIDALEN	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.003615484	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.039688338	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	ORYZALIN	chembl:CHEMBL295960	ORYZALIN	FALSE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.150667636	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.3723948314588262	Dexefaroxan	ncit:C77943	DEXEFAROXAN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.2917092846427472	BISPECIFIC ANTIBODY	ncit:C1454	BISPECIFIC ANTIBODY	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.004987431	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.021003068	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.2051080907644316	IUPHAR.LIGAND:410	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	TALC	12-May-16	antibody	4.286340509036285	ALD518	ncit:C82359	CLAZAKIZUMAB	FALSE	FALSE	TRUE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.019534104	nifedipine	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1861974157294131	IUPHAR.LIGAND:12	iuphar.ligand:12	EMDT	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:1671	iuphar.ligand:1671	PL017	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001914661	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.2243917574174978	METOCHALCONE	chembl:CHEMBL36584	METOCHALCONE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1400204566285186	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	CID 3241312	chembl:CHEMBL265715	CHEMBL:CHEMBL265715	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.043592919	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.014790893	PAROXETINE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:294	rxcui:194	ACETYLCHOLINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.002506094	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PDE2A	hgnc:8777	PDE2A	ChEMBL	33	inhibitor	0.093098708	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.01214331	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.004923825	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.01823183	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2094720926955897	SCOPOLAMINE	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	NALIDIXIC ACID	rxcui:7240	NALIDIXIC ACID	TRUE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:1761	iuphar.ligand:1761	NF157	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.067059606	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	SJ000019194	chembl:CHEMBL592106	CHEMBL:CHEMBL592106	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.020391329	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.2333674277141977	ABAMECTIN	ncit:C95196	ABAMECTIN	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.03357268	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
ATF2	hgnc:784	ATF2	NCI	14-Sep-17	NULL	0.8334550989792776	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.056601873	Thiethylperazine	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	GNF-PF-2347	chembl:CHEMBL579045	CHEMBL:CHEMBL579045	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	4SC-205	ncit:C90557	EG5 KINESIN-RELATED MOTOR PROTEIN INHIBITOR 4SC-205	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.053038052	Amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.3070624048871023	IUPHAR.LIGAND:4150	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	DTC	9/2/20	NULL	0.5933070196123671	TECADENOSON	ncit:C77980	TECADENOSON	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	DTC	9/2/20	NULL	0.3088686543276147	CID 100335	chembl:CHEMBL1520346	CHEMBL:CHEMBL1520346	FALSE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Aceprometazine	rxcui:161203	ACEPROMETAZINE	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	Descartes-08	ncit:C156706	AUTOLOGOUS ANTI-BCMA-CAR-MRNA-TRANSFECTED CD8+ T-LYMPHOCYTES	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:5555	iuphar.ligand:5555	RVD1-ME	FALSE	FALSE	FALSE
NCBIGENE:661	hgnc:1080	POLR3D	GuideToPharmacology	2024.1	agonist	0.7501095890813498	IUPHAR.LIGAND:6510	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:2209	hgnc:3613	FCGR1A	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	modulator	0.042968634	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:5796	iuphar.ligand:5796	2-HYDROXYOCTANOIC ACID	FALSE	FALSE	FALSE
TRM3	hgnc:11568	TARBP1	ChEMBL	33	inhibitor	26.25383561784724	LETERMOVIR	rxcui:1988648	LETERMOVIR	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	1-NAPHTHOL	rxcui:1740233	1-NAPHTHOL	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.038467158	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.064824285	C-1311	chembl:CHEMBL338604	C-1311	FALSE	FALSE	FALSE
NCBIGENE:768	hgnc:1383	CA9	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:11741	ncit:C71621	BIRICODAR	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.3394892536790592	donepezil	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9162	iuphar.ligand:9162	COMPOUND C10 [PMID: 24297249]	FALSE	FALSE	FALSE
UNIPROT:P54219	hgnc:10934	SLC18A1	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.192335792	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:3289	iuphar.ligand:3289	BAY 60-6583	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	P-PHENYLENEDIAMINE	rxcui:1362740	4-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
EPO	hgnc:3415	EPO	NCI	14-Sep-17	NULL	2.500365296937833	ALPHA INTERFERON	ncit:C225	RECOMBINANT INTERFERON ALFA	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.032899543	IUPHAR.LIGAND:2868	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.01186614	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.1058622403945453	AZELASTINE HYDROCHLORIDE	rxcui:235824	AZELASTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	blocker	0.1312691780892362	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
NCBIGENE:1486	hgnc:2496	CTBS	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:5290	iuphar.ligand:5290	Y27632	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	GNF-PF-3276	chembl:CHEMBL582081	CHEMBL:CHEMBL582081	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	IPA-3	iuphar.ligand:8940	IPA-3	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.024861587	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:744	hgnc:1180	MPPED2	GuideToPharmacology	2024.1	activator	5.250767123569449	IUPHAR.LIGAND:4124	iuphar.ligand:4124	ADENOPHOSTIN A	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	DoCM	10-Apr-24	NULL	0.546954909	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.041672755	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	TICARCILLIN	rxcui:10591	TICARCILLIN	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	3.150460274	KU-0058948	drugbank:DB08058	4-[3-(1,4-DIAZEPAN-1-YLCARBONYL)-4-FLUOROBENZYL]PHTHALAZIN-1(2H)-ONE	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.038523603	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	PIPOBROMAN	rxcui:8347	PIPOBROMAN	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	OPC-34712	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.2344092465879218	IUPHAR.LIGAND:240	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006324701	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.1174668260306364	DIRLOTAPIDE	rxcui:1592684	DIRLOTAPIDE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.024309107	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.008621949	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.05853698	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.789589041	C5A	iuphar.ligand:3576	C5A	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	SAPPANONE A 7-METHYL ETHER	chembl:CHEMBL1603788	SAPPANONE A 7-METHYL ETHER	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003185179	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2158	iuphar.ligand:2158	[125I]U-II (HUMAN)	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.192335792	PHENELZINE SULFATE	rxcui:8124	PHENELZINE SULFATE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	NCI	14-Sep-17	NULL	0.024908762	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.050007306	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.054020238	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
UNIPROT:P63316	hgnc:11943	TNNC1	TEND	1-Aug-11	NULL	1.750255707856483	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.004572246	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	0.3409589041278863	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:72	ncit:C74143	ROBALZOTAN	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:11665	iuphar.ligand:11665	XMD-12	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10750	iuphar.ligand:10750	MLN-3897	FALSE	FALSE	FALSE
NCBIGENE:544	hgnc:881	ALDH7A1P4	GuideToPharmacology	2024.1	blocker	0.5250767123569451	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.048483538	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:6778	rxcui:712566	OFATUMUMAB	TRUE	TRUE	TRUE
PSMD4	hgnc:9561	PSMD4	CIViC	10-Apr-24	NULL	0.2778183663264259	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.022290572	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.2983390411119005	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:76	iuphar.ligand:76	SB 649915	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.008103036	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	BROMFENAC SODIUM	rxcui:47364	BROMFENAC SODIUM	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
NCBIGENE:2591	hgnc:4125	GALNT3	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6697	iuphar.ligand:6697	GSK-264220A	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.1500219178162699	IUPHAR.LIGAND:2054	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.1553481397505754	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.076765601	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.027276712	SAHA	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P04746	hgnc:477	AMY2A	TEND	1-Aug-11	NULL	1.312691780892362	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	6.177373086552294	Eloctate	rxcui:1543095	EFMOROCTOCOG ALFA	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	1.009762908	NARATRIPTAN HYDROCHLORIDE	rxcui:236690	NARATRIPTAN HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	MEN1611	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.011316308	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	modulator	0.1262203635473425	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.048618214	SACITUZUMAB GOVITECAN	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2917092846427472	LOTAMILAST	ncit:C170131	LOTAMILAST	FALSE	FALSE	FALSE
UNIPROT:P07327	hgnc:249	ADH1A	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
UNIPROT:P32927	hgnc:2436	CSF2RB	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	SARGRAMOSTIM	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.09963505	Levobupivacaine	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:51	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
NCBIGENE:685	hgnc:1121	BTC	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	5.250767123569449	IUPHAR.LIGAND:12585	iuphar.ligand:12585	6-PRENYLNARINGENIN	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.1411496538593938	Cyproheptadine	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:3980	iuphar.ligand:3980	[3H]METHYLLYCACONITINE	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:11343	iuphar.ligand:11343	EST64454	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.025366025	Rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.0701037	medroxyprogesterone	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	PharmGKB	4/5/24	NULL	0.073885091	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	0.6775183385250904	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1211715490054488	quinine	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:9371	iuphar.ligand:9371	PF-670462	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	CID 838877	chembl:CHEMBL405317	CHEMBL:CHEMBL405317	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	DIALLYLDISULFIDE	chembl:CHEMBL366603	DIALLYLDISULFIDE	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:5964	iuphar.ligand:5964	EGFR/ERBB-2 INHIBITOR	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	U-50488	iuphar.ligand:1652	U50488	FALSE	FALSE	FALSE
HLA-G	hgnc:4964	HLA-G	PharmGKB	4/5/24	NULL	1.050153425	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	PIRIBEDIL	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	1.193356164447602	BAY1834845	iuphar.ligand:11415	ZABEDOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.035098711	IUPHAR.LIGAND:7111	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.073437302	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.093098708	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
NCBIGENE:1933	hgnc:3208	EEF1B2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12095	iuphar.ligand:12095	EXARAFENIB	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	0.3337351985319565	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:7903	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	agonist	0.037693949	IUPHAR.LIGAND:1712	iuphar.ligand:1712	ADP	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	PharmGKB	4/5/24	NULL	0.019949723	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PURINE NUCLEOSIDE PHOSPHORYLASE	hgnc:7892	PNP	TTD	2020.06.01	NULL	8.751278539282415	Peldesine	ncit:C1650	PELDESINE	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.4688184931758437	BAY-57-9352	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	TRIPHENYLSTANNANOL	chembl:CHEMBL506538	TRIPHENYLSTANNANOL	FALSE	FALSE	FALSE
NCBIGENE:2010	hgnc:3331	EMD	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9268	iuphar.ligand:9268	AZ191	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:1265	iuphar.ligand:1265	CIPROXIFAN	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:8095	iuphar.ligand:8095	AC710	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011311433	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.2561349816375342	HESPERIDIN	rxcui:5281	HESPERIDIN	TRUE	FALSE	FALSE
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	0.3571950424196904	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.030386384	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
RPL26	hgnc:10327	RPL26	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	NORSTICTIC ACID	chembl:CHEMBL228281	NORSTICTIC ACID	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	inhibitor	0.6403374540938354	OBEXELIMAB	ncit:C170236	OBEXELIMAB	FALSE	FALSE	FALSE
NCBIGENE:315	hgnc:1611	ACKR4	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:817	iuphar.ligand:817	CCL25	FALSE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	NEDOCROMIL	rxcui:31563	NEDOCROMIL	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.018118589	IUPHAR.LIGAND:197	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.03574382	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.1548898856510162	AMG-232	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
ATP7A	hgnc:869	ATP7A	PharmGKB	4/5/24	NULL	0.3153613888029699	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-125252	chembl:CHEMBL1408031	CHEMBL:CHEMBL1408031	FALSE	FALSE	FALSE
CKM	hgnc:1994	CKM	NCI	14-Sep-17	NULL	1.875273972703374	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	1.250182648468916	GONADOTROPIN-RELEASING HORMONE ANALOG	ncit:C1910	GONADOTROPIN-RELEASING HORMONE ANALOG	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	METAPHIT METHANESULFONATE	chembl:CHEMBL1256971	METAPHIT METHANESULFONATE	FALSE	FALSE	FALSE
NCBIGENE:2592	hgnc:4135	GALT	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6701	iuphar.ligand:6701	GR148672X	FALSE	FALSE	FALSE
CALR	hgnc:1455	CALR	NCI	14-Sep-17	NULL	13.12691780892362	VACCINIA VACCINE	ncit:C2313	VACCINIA VACCINE	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.5303805175322677	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.272767123	KETOPROFEN	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.044763573	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:8164	iuphar.ligand:8164	COMPOUND 7K [PMID: 23521020]	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1565523888959287	IUPHAR.LIGAND:4362	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:7399	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	1.944728564284981	IUPHAR.LIGAND:2500	iuphar.ligand:2500	4&ALPHA;-PDD	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.007330914	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:8193	iuphar.ligand:8193	COMPOUND 30 [PMID: 17280833]	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.4167275494896388	PD98059	iuphar.ligand:5241	PD98059	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	TCMDC-125784	chembl:CHEMBL581574	CHEMBL:CHEMBL581574	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TEND	1-Aug-11	NULL	0.2263261691193728	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	BRILLIANT GREEN OXALATE	chembl:CHEMBL1789985	BRILLIANT GREEN OXALATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.042073455	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.021850883	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	TCMDC-125578	chembl:CHEMBL195350	CHEMBL:CHEMBL195350	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	0.4730420832044549	FR139317	iuphar.ligand:998	FR139317	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	LANSOPRAZOLE SULFIDE	chembl:CHEMBL899	LANSOPRAZOLE SULFIDE	FALSE	FALSE	FALSE
RCSD1	hgnc:28310	RCSD1	CIViC	10-Apr-24	NULL	0.7001022831425933	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CD63	hgnc:1692	CD63	NCI	14-Sep-17	NULL	3.088686543276147	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	1.381780822	MK-1029	chembl:CHEMBL3545031	MK-1029	FALSE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.1356787370431382	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.106290832	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.097236428	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:477	iuphar.ligand:459	MRE 3008F20	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.05565201	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	NCI	14-Sep-17	NULL	0.2375912725597036	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1383601350084176	MOLINDONE	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	SJ000157363	chembl:CHEMBL590947	CHEMBL:CHEMBL590947	FALSE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	ChEMBL	33	agonist	1.093909817410302	PASIREOTIDE PAMOATE	rxcui:1597818	PASIREOTIDE PAMOATE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.042898424	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.041672755	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TdgClinicalTrial	Jan-14	NULL	0.05593857	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P23921	hgnc:10451	RRM1	TdgClinicalTrial	Jan-14	NULL	0.487687349	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
NCBIGENE:90	hgnc:171	ACVR1	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:9573	iuphar.ligand:9573	ADROPIN	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1471	iuphar.ligand:1471	NEUROMEDIN U-25	FALSE	FALSE	FALSE
NCBIGENE:2397	hgnc:3908	FRA5D	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:6432	ncit:C73213	CAMOSTAT	FALSE	FALSE	FALSE
B7 HOMOLOG 3	hgnc:19137	CD276	TTD	2020.06.01	NULL	31.50460274141669	MGA271	ncit:C97510	ENOBLITUZUMAB	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.024461995	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	PharmGKB	4/5/24	NULL	0.3309307010653015	niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
UNIPROT:P23415	hgnc:4326	GLRA1	TEND	1-Aug-11	NULL	0.1539814405738841	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
ISOCITRATE DEHYDROGENASE	hgnc:5382	IDH1	TTD	2020.06.01	NULL	0.064190307	ENASIDENIB MESYLATE	rxcui:1940331	ENASIDENIB MESYLATE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.5834185692854944	HYDROXYCAMPTOTHECIN	chembl:CHEMBL273862	HYDROXYCAMPTOTHECIN	FALSE	FALSE	FALSE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547592	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.2548916079402645	SJ000112483	chembl:CHEMBL603024	CHEMBL:CHEMBL603024	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.050879526	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
ASS1	hgnc:758	ASS1	PharmGKB	4/5/24	NULL	0.1875273972703375	sodium phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004540615	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	PENBUTOLOL SULFATE	rxcui:82070	PENBUTOLOL SULFATE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	2.059124362184098	RILZABRUTINIB	ncit:C174769	RILZABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:591	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004786261	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:4612	iuphar.ligand:4612	CI-966	FALSE	FALSE	FALSE
NCBIGENE:1219	hgnc:10956	SLCO1A2	GuideToPharmacology	2024.1	NULL	0.729273212	IUPHAR.LIGAND:4748	ncit:C47521	ESTROPIPATE	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8724	iuphar.ligand:8724	CCG-63802	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	ACETOMENAPHTHONE	ncit:C80886	ACETOMENAPHTHONE	FALSE	FALSE	FALSE
INTERLEUKIN 6 RECEPTOR	hgnc:6019	IL6R	TTD	2020.06.01	NULL	5.385402178019948	SA-237	rxcui:2391541	SATRALIZUMAB	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	PIRIBEDIL	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
GABA TRANSPORTER GAT-1	hgnc:11042	SLC6A1	TTD	2020.06.01	NULL	10.50153424713889	Metadoxine	drugbank:DB16554	METADOXINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	PHENAZINE-1-CARBOXYLIC ACID	chembl:CHEMBL463686	PHENAZINE-1-CARBOXYLIC ACID	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.1219690388750162	GDC-0199	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.1591141552596803	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.5048814541893701	ABT-165	ncit:C116750	DILPACIMAB	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.054020238	BROXURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.2822993077187876	AMARANTH	chembl:CHEMBL1408927	AMARANTH	FALSE	FALSE	FALSE
UNIPROT:P00797	hgnc:9958	REN	TEND	1-Aug-11	NULL	5.250767123569449	ALISKIREN	rxcui:325646	ALISKIREN	TRUE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7521	iuphar.ligand:7521	COMPOUND 36 [PMID: 24000170]	FALSE	FALSE	FALSE
NCBIGENE:2677	hgnc:4247	GGCX	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8230	iuphar.ligand:8230	IOX1	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	(5Z)-7-OXOZEAENOL	iuphar.ligand:8077	5Z-7-OXOZEAENOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	DSM-97	chembl:CHEMBL492528	CHEMBL:CHEMBL492528	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.1000146118775133	LY2801653	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	1.193356164447602	[19F]-HALOPERIDOL	chembl:CHEMBL2234294	[19F]-HALOPERIDOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	GANGALEOIDIN	chembl:CHEMBL1491099	GANGALEOIDIN	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	5.250767123569449	Dihydroartemisinin	ncit:C87432	ARTENIMOL	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.016480751	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	blocker	0.192335792	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.2706580991530644	IUPHAR.LIGAND:416	iuphar.ligand:416	AB-MECA	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1305078821102597	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:P04629	hgnc:8031	NTRK1	TdgClinicalTrial	Jan-14	NULL	0.1798207919030633	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:2641	iuphar.ligand:2641	BMS493	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.3977853881492006	ENSIFENTRINE	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
HSP90AA2	hgnc:5256	HSP90AA2P	MyCancerGenome	20-Jun-17	other/unknown	1.312691780892362	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
SPP1	hgnc:11255	SPP1	PharmGKB	4/5/24	NULL	0.4667348554283955	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.097870776	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
NCBIGENE:2360	hgnc:3868	FRA1A	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12133	iuphar.ligand:12133	FXIA INHIBITOR 3F	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.2692701089009974	DOXAZOSIN MESYLATE	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	0.4412409347537352	ETRETINATE	rxcui:4182	ETRETINATE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.4070362111294147	Zaleplon	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
NCBIGENE:2278	ncbigene:2278	FIM1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:11731	iuphar.ligand:11731	AZENOSERTIB	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	PharmGKB	4/5/24	NULL	0.4055851016423223	ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.053253216	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1250182648468916	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
IL22	hgnc:14900	IL22	ChEMBL	33	inhibitor	78.76150685354175	FEZAKINUMAB	ncit:C87764	FEZAKINUMAB	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9885	iuphar.ligand:9885	CORTISTATIN A	FALSE	FALSE	FALSE
CCNE1	hgnc:1589	CCNE1	CIViC	10-Apr-24	NULL	0.2187819634820604	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.003780794	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
ERAP1	hgnc:18173	ERAP1	DTC	9/2/20	NULL	2.917092846427472	TCMDC-124377	chembl:CHEMBL531269	CHEMBL:CHEMBL531269	FALSE	FALSE	FALSE
CTSG	hgnc:2532	CTSG	NCI	14-Sep-17	NULL	1.458546423213736	VITAMIN K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
INTERLEUKIN-18	hgnc:5986	IL18	TTD	2020.06.01	NULL	8.290684931951763	GSK-1070806	chembl:CHEMBL2109606	GSK-1070806	FALSE	FALSE	FALSE
POLR2A	hgnc:9187	POLR2A	DTC	9/2/20	NULL	35.00511415712966	3'-DCTP	chembl:CHEMBL480328	CHEMBL:CHEMBL480328	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	2,3,4-TRIHYDROXYBENZOPHENONE	chembl:CHEMBL1527	CHEMBL:CHEMBL1527	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	chembl:CHEMBL1336287	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3319450480417468	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.01097339	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	0.7895890411382631	MBX-8025	chembl:CHEMBL3545019	MBX-8025	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.9479406894984094	PD 0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.025280535	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UNIPROT:Q96RJ0	hgnc:17734	TAAR1	TdgClinicalTrial	Jan-14	NULL	0.075442056	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:509	rxcui:66887	RACEPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:1874	hgnc:3118	E2F4	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:5077	iuphar.ligand:5077	CD40 LIGAND	FALSE	FALSE	FALSE
NCBIGENE:1628	hgnc:2697	DBP	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:6482	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	SJ000032149	chembl:CHEMBL600778	CHEMBL:CHEMBL600778	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	NSC-44661	chembl:CHEMBL571228	CHEMBL:CHEMBL571228	FALSE	FALSE	FALSE
EIF4E	hgnc:3287	EIF4E	NCI	14-Sep-17	NULL	0.061376588	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.5834185692854944	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	HYDROXYZINE	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
KCNV1	hgnc:18861	KCNV1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.729273212	ILAPRAZOLE	ncit:C65887	ILAPRAZOLE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006434764	DEFEROXAMINE MESYLATE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003190792	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	MECLIZINE HYDROCHLORIDE	rxcui:82041	MECLIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001771873	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.5645986154375752	AME-527	drugbank:DB05879	AME-527	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6130	iuphar.ligand:6130	GALANIN(2-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5784	iuphar.ligand:5784	MK 0354	FALSE	FALSE	FALSE
NCBIGENE:1222	hgnc:13819	SLCO1C1	GuideToPharmacology	2024.1	NULL	1.093909817410302	IUPHAR.LIGAND:4748	ncit:C47521	ESTROPIPATE	FALSE	FALSE	FALSE
CDA	hgnc:1712	CDA	ChEMBL	33	inhibitor	0.300043836	CEDAZURIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NCBIGENE:1795	hgnc:2989	DOCK3	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:5062	iuphar.ligand:5062	TGF&BETA;3	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.1305078821102597	yohimbine	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	1.842374429322613	HEXAMETHYLENEBISACETAMIDE	chembl:CHEMBL291481	HEXAMETHYLENEBISACETAMIDE	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	0.31919557	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
AMY2A	hgnc:477	AMY2A	ChEMBL	33	inhibitor	1.312691780892362	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.03729238	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	BENZENE-1,2-DIAMINE	chembl:CHEMBL70582	CHEMBL:CHEMBL70582	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
POLA2	hgnc:30073	POLA2	ChEMBL	33	inhibitor	0.080656945	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.098884503	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	8.751278539282415	TAK-441	iuphar.ligand:8200	TAK-441	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.037398626	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:108	hgnc:233	ADCY2	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:8840	iuphar.ligand:8840	COMPOUND 7A [PMID: 24884590]	FALSE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.088248187	BROMOCRIPTINE MESYLATE	rxcui:142426	BROMOCRIPTINE MESYLATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.182318303	4-hydroxycyclophosphamide	rxcui:2675983	4-HYDROXYCYCLOPHOSPHAMIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1875273972703375	sulfamethoxazole	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.023388718	PERICIAZINE	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.050488145	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007244436	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	L-733060	chembl:CHEMBL1256740	CHEMBL:CHEMBL1256740	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	SJ000147993	chembl:CHEMBL601618	CHEMBL:CHEMBL601618	FALSE	FALSE	FALSE
SRP19	hgnc:11300	SRP19	PharmGKB	4/5/24	NULL	0.9376369863516874	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	PharmGKB	4/5/24	NULL	0.060156088	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	1.419126249613364	ISOCARBOXAZID	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.069089041	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
GCLM	hgnc:4312	GCLM	NCI	14-Sep-17	NULL	0.2785552850699973	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	2.386712328895204	ADEFOVIR	rxcui:16521	ADEFOVIR	TRUE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.5556367326528517	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.081597003	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	5.834185692854944	BENDROFLUMETHIAZIDE	rxcui:1369	BENDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
PTCH1	hgnc:9585	PTCH1	CIViC	10-Apr-24	NULL	19.69037671338543	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	SNX-5422	drugbank:DB06070	SNX-5422	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.063415062	PEXMETINIB	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	ChEMBL	33	inhibitor	0.021036727	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	GLESATINIB	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:9717	iuphar.ligand:9717	BI-1935	FALSE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.2500365296937833	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.078958904	IUPHAR.LIGAND:302	iuphar.ligand:302	OXOTREMORINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.029090123	IUPHAR.LIGAND:305	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:323	iuphar.ligand:323	HEXOCYCLIUM	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2465148884304905	METHYLTESTOSTERONE	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
FGA	hgnc:3661	FGA	ChEMBL	33	cleavage	1.591141552596802	PLASMINOGEN	rxcui:2557200	PLASMINOGEN	TRUE	FALSE	FALSE
PLD1	hgnc:9067	PLD1	DTC	9/2/20	NULL	4.375639269641208	HALOPEMIDE	ncit:C65840	HALOPEMIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.008288504	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	(R)-FELODIPINE	chembl:CHEMBL254609	(R)-FELODIPINE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
UNIPROT:P06213	hgnc:6091	INSR	TdgClinicalTrial	Jan-14	NULL	1.500219178	INSULIN DETEMIR	rxcui:139825	INSULIN DETEMIR	TRUE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:1892	iuphar.ligand:1892	BUTAPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	MUROMONAB	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	VINDESINE	rxcui:11204	VINDESINE	FALSE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1127984344483232	CIGLITAZONE	ncit:C72726	CIGLITAZONE	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1326	iuphar.ligand:1326	[125I]NDP-MSH	FALSE	FALSE	FALSE
MT-CYB	hgnc:7427	MT-CYB	ChEMBL	33	inhibitor	26.25383561784724	ATOVAQUONE	rxcui:60212	ATOVAQUONE	TRUE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	inhibitor	1.093909817410302	PG-102	chembl:CHEMBL2109475	PG-102	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.027577558	IUPHAR.LIGAND:189	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:7351	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.06714536	IUPHAR.LIGAND:5663	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:11288	iuphar.ligand:11288	R-VK4-40	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.010058941	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	1.193356164447602	Albumin Human	rxcui:2054166	ALBUMIN HUMAN-KJDA	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE	chembl:CHEMBL513116	N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	ANIRACETAM	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	1.029562181092048	16,16-dimethyl-PGE2	iuphar.ligand:1926	16,16-DIMETHYL-PGE2	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1642918374083057	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.055622533	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	activator	0.1209854175937661	IUPHAR.LIGAND:2505	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
NCBIGENE:433	hgnc:743	ASGR2	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:361	iuphar.ligand:361	TRIPITRAMINE	FALSE	FALSE	FALSE
NCBIGENE:1433	hgnc:9067	PLD1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8781	iuphar.ligand:8781	FIPI	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:2479	iuphar.ligand:2479	HCL	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
GPBAR1	hgnc:19680	GPBAR1	DTC	9/2/20	NULL	26.25383561784724	TAUROLITHOCHOLIC ACID	iuphar.ligand:4548	TAUROLITHOCHOLIC ACID-3-SULPHATE	FALSE	FALSE	FALSE
RAC1	hgnc:9801	RAC1	DTC	9/2/20	NULL	5.834185692854944	TCMDC-124310	chembl:CHEMBL579882	CHEMBL:CHEMBL579882	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	GNF-PF-3352	chembl:CHEMBL600306	CHEMBL:CHEMBL600306	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	CIViC	10-Apr-24	NULL	0.4735986033023426	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.022136455	disopyramide	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
ENPP2	hgnc:3357	ENPP2	DTC	9/2/20	NULL	17.50255707856483	NSC-1741	chembl:CHEMBL483302	CHEMBL:CHEMBL483302	FALSE	FALSE	FALSE
KCNK2	hgnc:6277	KCNK2	ChEMBL	33	potentiator	0.2083637747448194	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:2766	hgnc:4376	GMPR	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:10609	iuphar.ligand:10609	MEZAGITAMAB	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1918	ncit:C169951	ENPROSTIL	FALSE	FALSE	FALSE
NCBIGENE:833	hgnc:1493	CARS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:6782	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.011171845	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	MyCancerGenome	20-Jun-17	other/unknown	0.729273212	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	NCI	14-Sep-17	NULL	0.5527123287967842	THYMIDINE	rxcui:1372538	THYMIDINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	TCMDC-125580	chembl:CHEMBL528807	CHEMBL:CHEMBL528807	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.6886251965336985	NORGESTIMATE	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.035418328	Fesoterodine	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.012561644	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.093596562	Ro 31-7453	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	BUTEIN	ncit:C1028	BUTEIN	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.1110098757625676	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1193356164447602	DEXKETOPROFEN	rxcui:237162	DEXKETOPROFEN	TRUE	FALSE	FALSE
HSPA1L	hgnc:5234	HSPA1L	PharmGKB	4/5/24	NULL	2.143170254518142	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	DIACYLGLYCEROL KINASE INHIBITOR II	iuphar.ligand:5957	DIACYLGLYCEROL KINASE INHIBITOR II	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.078136416	MISOPROSTOL	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	PIMARIC ACID	chembl:CHEMBL1410398	PIMARIC ACID	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.091159151	DOBUTAMINE	rxcui:3616	DOBUTAMINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003772103	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	CLIOXANIDE	ncit:C65338	CLIOXANIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.001933984	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6210	iuphar.ligand:6210	COMPOUND 27 [PMID: 20346665]	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.017620024	quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
ANGIOPOIETIN 1 RECEPTOR	hgnc:11724	TEK	TTD	2020.06.01	NULL	0.3125456621172291	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.019461702	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	SKIMMIANINE	chembl:CHEMBL21396	SKIMMIANINE	FALSE	FALSE	FALSE
SLC5A1	hgnc:11036	SLC5A1	ChEMBL	33	inhibitor	6.300920548283339	SOTAGLIFLOZIN	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	inhibitor	3.088686543276147	NOLASIBAN	ncit:C166647	NOLASIBAN	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	inhibitor	0.045226246	IUPHAR.LIGAND:4197	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:9600	iuphar.ligand:9600	MIVAVOTINIB	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	0.3500511415712967	IUPHAR.LIGAND:1324	rxcui:2262250	AFAMELANOTIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	NSC-601359	chembl:CHEMBL1306524	CHEMBL:CHEMBL1306524	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.093763699	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.1103102336884338	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.078958904	FRENTIZOLE	ncit:C167023	FRENTIZOLE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.005593658	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	PHENYL BIGUANIDE	iuphar.ligand:2284	1-PHENYLBIGUANIDE	FALSE	FALSE	FALSE
GRIK1	hgnc:4579	GRIK1	ChEMBL	33	inhibitor	1.432027397337122	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	0.6000876712650799	MUROMONAB	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
NCBIGENE:1886	hgnc:17755	TNFRSF13C	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:10656	iuphar.ligand:10656	IANALUMAB	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	inhibitor	0.1495945049449985	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2748	iuphar.ligand:2748	DESMOSTEROL	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	ALATROFLOXACIN MESYLATE	rxcui:221054	ALATROFLOXACIN MESYLATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DoCM	10-Apr-24	NULL	0.6241137025199848	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	AMG-548	chembl:CHEMBL585902	AMG-548	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.6731752722524935	DE-104	chembl:CHEMBL3545153	DE-104	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	ChEMBL	33	modulator	1.193356164447602	PLOVAMER ACETATE	ncit:C96530	PLOVAMER ACETATE	FALSE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	1.193356164447602	K-134	drugbank:DB12685	K-134	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:11473	iuphar.ligand:11473	JNJ-67869386	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.01083079	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.3500511415712966	MESOTRIONE	chembl:CHEMBL1873440	MESOTRIONE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	TAXIFOLIN	drugbank:DB02224	TAXIFOLIN	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M4	hgnc:1953	CHRM4	TTD	2020.06.01	NULL	0.2778183663264258	Diphenidol	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1367387271762877	EMETINE HYDROCHLORIDE	rxcui:82015	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.055859225	TIOTROPIUM	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9840	iuphar.ligand:9840	SR7826	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.1574442915613028	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.084281976	IUPHAR.LIGAND:5701	iuphar.ligand:5701	PI-103	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.1562728310586145	NSC-367089	chembl:CHEMBL1543865	CHEMBL:CHEMBL1543865	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.040515178	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	ACETOCHLOR	chembl:CHEMBL1517425	ACETOCHLOR	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.019339842	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1500219178162699	Glipizide	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.041214813	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
KCNS3	hgnc:6302	KCNS3	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1376949420516464	Fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
RPL8	hgnc:10368	RPL8	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	0.9723642821424906	CARBETAPENTANE CITRATE	rxcui:283547	CARBETAPENTANE CITRATE	TRUE	FALSE	FALSE
ADIPOQ	hgnc:13633	ADIPOQ	NCI	14-Sep-17	NULL	1.193356164447602	NEVIRAPINE	rxcui:53654	NEVIRAPINE	TRUE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.1223955040459079	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	0.3750547945406749	Interferon Alfa-2b	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
KCNE1	hgnc:6240	KCNE1	PharmGKB	4/5/24	NULL	1.250182648468916	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.8468979231563628	DEOXYCYTIDINE	rxcui:2642208	DEOXYCYTIDINE	FALSE	FALSE	FALSE
CD70	hgnc:11937	CD70	ChEMBL	33	inhibitor	4.039051633514961	CUSATUZUMAB	ncit:C106116	CUSATUZUMAB	FALSE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TEND	1-Aug-11	NULL	0.3725599732909588	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P32241	hgnc:12694	VIPR1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	VASOACTIVE INTESTINAL PEPTIDE	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
UNIPROT:P01112	hgnc:5173	HRAS	TdgClinicalTrial	Jan-14	NULL	0.6908904109959803	ISIS-2503	chembl:CHEMBL4594562	ISIS-2503	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:1918	ncit:C169951	ENPROSTIL	FALSE	FALSE	FALSE
ARRB2	hgnc:712	ARRB2	PharmGKB	4/5/24	NULL	0.1207072901969988	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.005448974	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.2263261691193728	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.061055432	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	CancerCommons	25-Jul-13	inhibitor	0.6141248097742047	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	CGI	2/1/22	NULL	0.028413242	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.01798824	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2035181055647073	PRONETALOL	ncit:C82257	PRONETALOL	TRUE	FALSE	FALSE
AKT3	hgnc:393	AKT3	CGI	2/1/22	NULL	0.4922594178346359	GSK2141795	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	CGI	2/1/22	NULL	0.3509871071904712	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.2363572458670459	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.2778183663264259	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.6945459158160648	Nimotuzumab	ncit:C2733	NIMOTUZUMAB	FALSE	TRUE	TRUE
NRG1	hgnc:7997	NRG1	CGI	2/1/22	NULL	0.1151484018326633	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.021878196	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1635752997996713	CENTANAFADINE	ncit:C171666	CENTANAFADINE	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.1058622403945453	DIPHENHYDRAMINE HYDROCHLORIDE	rxcui:1362	DIPHENHYDRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	1.640864726115453	VARDENAFIL HYDROCHLORIDE	rxcui:1309396	VARDENAFIL HYDROCHLORIDE TRIHYDRATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.051885051	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.3236220106976548	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	1.009762908	IUPHAR.LIGAND:10696	iuphar.ligand:10696	AXT914	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	inhibitor	1.141471113819445	CONIVAPTAN HYDROCHLORIDE	rxcui:1294548	CONIVAPTAN HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.3059887601147698	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
NCBIGENE:2943	hgnc:1682	CD47	GuideToPharmacology	2024.1	antibody	6.563458904461812	IUPHAR.LIGAND:12652	iuphar.ligand:12652	MAGROLIMAB	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN PURIFIED BEEF	chembl:CHEMBL1201629	INSULIN PURIFIED BEEF	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.111481255	ERGOCALCIFEROL	rxcui:4018	ERGOCALCIFEROL	TRUE	FALSE	FALSE
TYR	hgnc:12442	TYR	ChEMBL	33	inhibitor	4.773424657790408	MEQUINOL	rxcui:15080	MEQUINOL	TRUE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	ChEMBL	33	agonist	3.281729452230906	CORTICOTROPIN ZINC HYDROXIDE	ncit:C169866	CORTICOTROPIN-ZINC HYDROXIDE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.042073455	QUETIAPINE FUMARATE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:5993	iuphar.ligand:5993	JAK3 INHIBITOR II	FALSE	FALSE	TRUE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.026626608	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	3.750547945	CARBOPROST TROMETHAMINE	rxcui:20259	CARBOPROST TROMETHAMINE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	ChEMBL	33	inhibitor	0.1909369863116163	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:8104	iuphar.ligand:8104	LY2874455	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.3125456621172291	ESTRAMUSTINE PHOSPHATE SODIUM	rxcui:4090	ESTRAMUSTINE PHOSPHATE SODIUM	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	ECHOTHIOPHATE IODIDE	rxcui:3740	ECHOTHIOPHATE IODIDE	TRUE	FALSE	FALSE
FSHR	hgnc:3969	FSHR	ChEMBL	33	agonist	18.37768493249307	UROFOLLITROPIN	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.038173516	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:4368	iuphar.ligand:4368	[18F]FLUOROETHYLFLUMAZENIL	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	FLUOCINONIDE	rxcui:4462	FLUOCINONIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	MEPREDNISONE	rxcui:29523	MEPREDNISONE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	ABACAVIR SULFATE	rxcui:221052	ABACAVIR SULFATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1115286134997759	ESTRONE	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.736088849	GUANADREL SULFATE	rxcui:91239	GUANADREL SULFATE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	0.729273212	ROSUVASTATIN CALCIUM	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.1442518440541057	TOREMIFENE CITRATE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	negative modulator	0.6035364509849942	MEMANTINE HYDROCHLORIDE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.2486158675932504	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.3561566847382379	BRIMONIDINE TARTRATE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.2344092465879218	BRIMONIDINE TARTRATE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.100976291	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.1367387271762877	DOXAZOSIN MESYLATE	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
GRIK3	hgnc:4581	GRIK3	ChEMBL	33	inhibitor	0.1704794520639432	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.2536602475154323	METHOXAMINE HYDROCHLORIDE	rxcui:203187	METHOXAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.039778539	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.3088686543276147	NITRIC OXIDE	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.9723642821424906	OCTREOTIDE ACETATE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
SSTR3	hgnc:11332	SSTR3	ChEMBL	33	agonist	0.3241214273808303	OCTREOTIDE ACETATE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.5834185692854945	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2442217266776488	AMLODIPINE BESYLATE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.2476776945079929	DILTIAZEM MALATE	rxcui:81999	DILTIAZEM MALATE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.074478966	VERAPAMIL HYDROCHLORIDE	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.1848861663228679	BUPRENORPHINE HYDROCHLORIDE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	0.050978322	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	LEVALBUTEROL TARTRATE	rxcui:487066	LEVALBUTEROL TARTRATE	TRUE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	0.5357925636295356	APIXABAN	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	ChEMBL	33	inhibitor	0.729273212	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC5	hgnc:9552	PSMC5	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC3	hgnc:9549	PSMC3	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC4	hgnc:9551	PSMC4	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1909369863116163	LOPINAVIR	rxcui:195088	LOPINAVIR	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.4167275494896388	ATRACURIUM BESYLATE	rxcui:1219	ATRACURIUM BESYLATE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.251232877	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
GLRB	hgnc:4329	GLRB	ChEMBL	33	positive modulator	0.1750255707856483	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	ChEMBL	33	positive modulator	0.044198376	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	0.4412409347537352	ETRETINATE	rxcui:4182	ETRETINATE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.091796628	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.085239726	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.091796628	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.081365193	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.020351811	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.020836377	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.021344582	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.019889269	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.020836377	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.096050618	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.030527716	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.076840494	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.085147575	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.07160137	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.1017590527823536	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.054886067	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.018462613	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.011306561	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.016206071	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.016027983	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.4526523382387456	NORFLOXACIN	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.6035364509849942	SPARFLOXACIN	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.096521454	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	KANAMYCIN SULFATE	rxcui:203183	KANAMYCIN SULFATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.03043923	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	agonist	0.1715936968486748	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
CSF2RB	hgnc:2436	CSF2RB	ChEMBL	33	agonist	13.12691780892362	SARGRAMOSTIM	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.6250913242344583	INTERFERON ALFA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.023440925	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.050488145	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.05593857	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.05293112	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.029766254	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.039688338	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.1754935535952356	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNK2	hgnc:6277	KCNK2	ChEMBL	33	potentiator	0.2500365296937833	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
KCNK3	hgnc:6278	KCNK3	ChEMBL	33	potentiator	0.2500365296937833	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1000146118775133	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	blocker	0.128067491	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNV2	hgnc:19698	KCNV2	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH5	hgnc:6254	KCNH5	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNC4	hgnc:6236	KCNC4	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.4055851016423223	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
PDE6D	hgnc:8788	PDE6D	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE7B	hgnc:8792	PDE7B	ChEMBL	33	inhibitor	0.093098708	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE8B	hgnc:8794	PDE8B	ChEMBL	33	inhibitor	0.1241316104862754	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE10A	hgnc:21160	LINC00473	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.9723642821424906	PEGINTERFERON BETA-1A	rxcui:1546168	PEGINTERFERON BETA-1A	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	2.019525817	SECUKINUMAB	rxcui:1599788	SECUKINUMAB	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.025827679	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	ChEMBL	33	inhibitor	0.09869863	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.051177067	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.058471794	AZD3514	chembl:CHEMBL2346976	AZD3514	FALSE	FALSE	FALSE
FGR	hgnc:3697	FGR	ChEMBL	33	inhibitor	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
FYN	hgnc:4037	FYN	ChEMBL	33	inhibitor	0.025147352	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
HCK	hgnc:4840	HCK	ChEMBL	33	inhibitor	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
FRK	hgnc:3955	FRK	ChEMBL	33	inhibitor	0.03233231	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.8334550989792777	AMG-319	drugbank:DB16879	AMG-319	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.033207482	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.04525223	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.2749092734853114	ARQ-736	chembl:CHEMBL3545296	ARQ-736	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.042898424	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK11B	hgnc:1729	CDK11B	ChEMBL	33	inhibitor	0.1286952726365061	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK5	hgnc:1774	CDK5	ChEMBL	33	inhibitor	0.049723174	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK19	hgnc:19338	CDK19	ChEMBL	33	inhibitor	0.1458546423213736	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK3	hgnc:1772	CDK3	ChEMBL	33	inhibitor	0.364636606	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	1.237091730683901	LIFIRAFENIB	ncit:C124995	LIFIRAFENIB	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	ChEMBL	33	inhibitor	0.315361389	MSC-2363318A	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	1.109316997937207	PF-00337210	chembl:CHEMBL3545136	PF-00337210	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1215455352678113	PWT-33579	chembl:CHEMBL3545323	PWT-33579	FALSE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	ChEMBL	33	inhibitor	0.2500365296937833	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	3.000438356	MIVAVOTINIB CITRATE	ncit:C188286	MIVAVOTINIB CITRATE	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1223955040459079	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.063568609	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.3125456621172291	LY2245461	chembl:CHEMBL3545389	LY2245461	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.2885036881082115	AZD8108	chembl:CHEMBL3707355	AZD8108	FALSE	FALSE	FALSE
PRKCI	hgnc:9404	PRKCI	ChEMBL	33	inhibitor	0.1721562991334246	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	6.177373086552294	PALOVAROTENE	rxcui:2663954	PALOVAROTENE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.111481255	INECALCITOL	ncit:C83818	INECALCITOL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.061628722	AEE-788	drugbank:DB12558	AEE-788	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.7876150685354174	BAFETINIB	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.1944728564284981	UPROSERTIB	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	0.750109589	R-333	chembl:CHEMBL3545159	R-333	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.3918482928036902	DANUSERTIB	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.2187819634820604	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.045898314	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1767935058440892	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	inhibitor	9.845188356692718	ELINOGREL	ncit:C96896	ELINOGREL	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	agonist	0.1286952726365061	VABICASERIN HYDROCHLORIDE	ncit:C142993	VABICASERIN HYDROCHLORIDE	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.1052961321571413	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
CXCR2	hgnc:6027	CXCR2	ChEMBL	33	inhibitor	2.917092846427472	ELUBRIXIN	ncit:C174724	ELUBRIXIN	FALSE	FALSE	FALSE
GRM2	hgnc:4594	GRM2	ChEMBL	33	modulator	1.875273972703375	DECOGLURANT	ncit:C166865	DECOGLURANT	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	ChEMBL	33	inhibitor	1.750255707856483	LY2590443	chembl:CHEMBL3545220	LY2590443	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	1.312691780892362	AZD5672	iuphar.ligand:7686	AZD5672	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	inhibitor	5.250767123569449	PF-06291874	drugbank:DB15065	PF-06291874	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	2.019525817	GW842166X	drugbank:DB11903	GW842166	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	7.001022831425932	OLCEGEPANT	ncit:C170245	OLCEGEPANT	FALSE	FALSE	FALSE
OPRL1	hgnc:8155	OPRL1	ChEMBL	33	inhibitor	6.563458904461812	LY2940094	iuphar.ligand:9462	LY2940094	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	modulator	0.063110182	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	modulator	0.1553481397505754	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	modulator	0.1262203635473425	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	modulator	0.1262203635473425	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	1.591141552596803	K-877	chembl:CHEMBL3545412	K-877	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.1400204566285186	IMIGLITAZAR	ncit:C83791	IMIGLITAZAR	FALSE	FALSE	FALSE
MAP3K12	hgnc:6851	MAP3K12	ChEMBL	33	inhibitor	5.834185692854945	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	modulator	0.2019525816757481	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.1256164383629055	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	blocker	0.093763699	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	ChEMBL	33	blocker	0.059667808	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNA3	hgnc:6221	KCNA3	ChEMBL	33	blocker	0.1875273972703375	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.005795549	Azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
SV2A	hgnc:20566	SV2A	ChEMBL	33	modulator	10.50153424713889	BRIVARACETAM	rxcui:1739745	BRIVARACETAM	TRUE	FALSE	FALSE
KCNG4	hgnc:19697	KCNG4	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	agonist	0.3125456621172291	TELBERMIN	ncit:C152544	TELBERMIN	FALSE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.2800409132570373	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	1.750255707856483	CILANSETRON	ncit:C76106	CILANSETRON	FALSE	FALSE	FALSE
CETP	hgnc:1869	CETP	ChEMBL	33	inhibitor	4.039051633514961	EVACETRAPIB	ncit:C166804	EVACETRAPIB	FALSE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.7721716358190367	TEZACITABINE	ncit:C1539	TEZACITABINE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.3571950424196904	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.1030370314672184	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	1.312691780892362	TEZACITABINE	ncit:C1539	TEZACITABINE	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	3.281729452230906	VOSAROXIN	ncit:C95148	VOSAROXIN	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	ChEMBL	33	negative modulator	0.6035364509849942	EFAPROXIRAL	ncit:C1435	EFAPROXIRAL	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.091159151	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
FDFT1	hgnc:3629	FDFT1	ChEMBL	33	inhibitor	26.25383561784724	LAPAQUISTAT ACETATE	ncit:C81535	LAPAQUISTAT ACETATE	FALSE	FALSE	FALSE
EGLN3	hgnc:14661	EGLN3	ChEMBL	33	inhibitor	3.500511415712966	ROXADUSTAT	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
EGLN2	hgnc:14660	EGLN2	ChEMBL	33	inhibitor	3.500511415712966	ROXADUSTAT	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	HYDROCORTISONE SODIUM SUCCINATE	rxcui:235483	HYDROCORTISONE SODIUM SUCCINATE	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.33338204	CRISABOROLE	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.5114383561918295	CRISABOROLE	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.2586584789935689	CRISABOROLE	rxcui:1865953	CRISABOROLE	TRUE	FALSE	FALSE
ITGB7	hgnc:6162	ITGB7	ChEMBL	33	inhibitor	2.917092846427472	FIRATEGRAST	ncit:C76692	FIRATEGRAST	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.312691780892362	SOTAGLIFLOZIN	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.02271093	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CRBN	hgnc:30185	CRBN	ChEMBL	33	inhibitor	0.8975670296699916	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.6250913242344582	ARZOXIFENE	ncit:C1805	ARZOXIFENE	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.4773424657790409	PARECOXIB	rxcui:279950	PARECOXIB	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.525076712	SJ000279525	chembl:CHEMBL600841	CHEMBL:CHEMBL600841	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	1.117184494376478	RALTITREXED	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
SOST	hgnc:13771	SOST	ChEMBL	33	inhibitor	6.563458904461812	BLOSOZUMAB	ncit:C171830	BLOSOZUMAB	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.5645986154375752	ONERCEPT	ncit:C96757	ONERCEPT	FALSE	FALSE	FALSE
NCAM1	hgnc:7656	NCAM1	ChEMBL	33	binder	13.12691780892362	ONCOLYSIN S	chembl:CHEMBL2109634	ONCOLYSIN S	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.021189536	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	0.596678082	ZONAMPANEL	ncit:C152963	ZONAMPANEL	FALSE	FALSE	FALSE
TYRP1	hgnc:12450	TYRP1	ChEMBL	33	other/unknown	105.0153424713889	FLANVOTUMAB	ncit:C91384	FLANVOTUMAB	FALSE	FALSE	FALSE
TNC	hgnc:5318	TNC	ChEMBL	33	other/unknown	6.563458904461812	TENATUMOMAB	ncit:C88600	TENATUMOMAB	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	1.129197231	OZORALIZUMAB	ncit:C175183	OZORALIZUMAB	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.267214612	DESONIDE	rxcui:3254	DESONIDE	TRUE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	inhibitor	0.546954909	FORALUMAB	ncit:C95785	FORALUMAB	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	ChEMBL	33	inhibitor	1.346350544504987	BENDAZAC	ncit:C80537	BENDAZAC	TRUE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	3.281729452230906	EBROTIDINE	ncit:C77440	EBROTIDINE	TRUE	FALSE	FALSE
CD38	hgnc:1667	CD38	ChEMBL	33	inhibitor	23.33674277141977	ISATUXIMAB	rxcui:2282018	ISATUXIMAB	TRUE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	0.252440727	BENZBROMARONE	rxcui:1385	BENZBROMARONE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.041739007	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
DDC	hgnc:2719	DDC	ChEMBL	33	inhibitor	3.000438356325399	BENSERAZIDE	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.029833904	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
TRPV4	hgnc:18083	TRPV4	ChEMBL	33	inhibitor	0.9723642821424906	BUTAMBEN PICRATE	rxcui:221067	BUTAMBEN PICRATE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	agonist	0.062065805	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	5.250767123569449	VALBENAZINE TOSYLATE	rxcui:1923002	VALBENAZINE TOSYLATE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	GLECAPREVIR	rxcui:1940635	GLECAPREVIR	TRUE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.1067229090156392	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	ChEMBL	33	inhibitor	4.039051633514961	MEDI-8968	chembl:CHEMBL2109607	MEDI-8968	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	2.917092846427472	MONO-DGA-RFB4	chembl:CHEMBL2109354	MONO-DGA-RFB4	FALSE	FALSE	FALSE
IFNA13	hgnc:5419	IFNA13	ChEMBL	33	inhibitor	1.166837138570988	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:1915	rxcui:8814	EPOPROSTENOL	TRUE	FALSE	FALSE
CSF1	hgnc:2432	CSF1	ChEMBL	33	inhibitor	3.750547945	MCS-110	chembl:CHEMBL2109512	MCS-110	FALSE	FALSE	FALSE
CD70	hgnc:11937	CD70	ChEMBL	33	modulator	12.11715490054488	MDX-1411	chembl:CHEMBL2109492	MDX-1411	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M2	hgnc:1951	CHRM2	TTD	2020.06.01	NULL	0.1535312024435511	Methacholine Chloride	rxcui:40165	METHACHOLINE CHLORIDE	TRUE	FALSE	FALSE
NOTCH3	hgnc:7883	NOTCH3	ChEMBL	33	inhibitor	21.00306849427779	TAREXTUMAB	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
RPS7	hgnc:10440	RPS7	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS15	hgnc:10388	RPS15	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS4X	hgnc:10424	RPS4X	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS29	hgnc:10419	RPS29	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL7	hgnc:10363	RPL7	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	LIPIDYL PSEUDOPTERANE A	chembl:CHEMBL508425	LIPIDYL PSEUDOPTERANE A	FALSE	FALSE	FALSE
RPL28	hgnc:10330	RPL28	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	4.375639269641208	GLASDEGIB MALEATE	rxcui:2105844	GLASDEGIB MALEATE	TRUE	FALSE	FALSE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	3.000438356	FOSTAMATINIB DISODIUM	rxcui:2055929	FOSTAMATINIB DISODIUM	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.033295923	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.06466462	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	(5Z,9Z)-5,9-HEXADECADIENOIC ACID	chembl:CHEMBL464637	CHEMBL:CHEMBL464637	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	ChEMBL	33	inhibitor	0.577007376	APABETALONE	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
ACLY	hgnc:115	ACLY	ChEMBL	33	inhibitor	39.38075342677087	BEMPEDOIC ACID	rxcui:2282403	BEMPEDOIC ACID	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.007024908	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.7501095890813501	RAMOSETRON HYDROCHLORIDE	ncit:C88299	RAMOSETRON HYDROCHLORIDE	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	1.346350544504987	MOCLOBEMIDE	rxcui:30121	MOCLOBEMIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.08334551	BLONANSERIN	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.081533651	DELGOCITINIB	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	ChEMBL	33	inhibitor	4.039051633514961	LINERIXIBAT	rxcui:2665338	LINERIXIBAT	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
RPS19	hgnc:10402	RPS19	ChEMBL	33	inhibitor	0.042516333	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPS10	hgnc:10383	RPS10	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TNNI2	hgnc:11946	TNNI2	ChEMBL	33	activator	8.751278539282415	TIRASEMTIV	ncit:C152657	TIRASEMTIV	FALSE	FALSE	FALSE
RPL31	hgnc:10334	RPL31	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL11	hgnc:10301	RPL11	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPLP1	hgnc:10372	RPLP1	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPLP0	hgnc:10371	RPLP0	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	PF-06459988	drugbank:DB14768	PF-06459988	FALSE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	6.058577450272442	VERINURAD	ncit:C152863	VERINURAD	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	1.250182648468916	PAMITEPLASE	ncit:C96708	PAMITEPLASE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.3182283105193605	DANUGLIPRON	ncit:C177080	DANUGLIPRON	FALSE	FALSE	FALSE
LTB4R	hgnc:6713	LTB4R	ChEMBL	33	inhibitor	1.093909817410302	NOMACOPAN	ncit:C167012	NOMACOPAN	FALSE	FALSE	FALSE
IL1RAP	hgnc:5995	IL1RAP	ChEMBL	33	inhibitor	8.751278539282415	IMSIDOLIMAB	ncit:C177088	IMSIDOLIMAB	FALSE	FALSE	FALSE
C3	hgnc:1318	C3	ChEMBL	33	inhibitor	5.834185692854944	AL-78898A	iuphar.ligand:9219	AL-78898A	FALSE	FALSE	FALSE
F7	hgnc:3544	F7	ChEMBL	33	inhibitor	0.3125456621172291	PCI-27483	drugbank:DB13000	PCI-27483	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	JNJ-39220675	drugbank:DB12929	JNJ-39220675	FALSE	FALSE	FALSE
RPL29	hgnc:10331	RPL29	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
LAG3	hgnc:6476	LAG3	ChEMBL	33	inhibitor	6.563458904461812	FIANLIMAB	ncit:C132339	FIANLIMAB	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	2.019525817	PEGTEOGRASTIM	ncit:C128891	PEGTEOGRASTIM	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	inhibitor	0.8975670296699914	PIBOSEROD	ncit:C74393	PIBOSEROD	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	2.019525817	ABICIPAR PEGOL	ncit:C174693	ABICIPAR PEGOL	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:6282	iuphar.ligand:6282	ML221	FALSE	FALSE	FALSE
E2F8	hgnc:24727	E2F8	ChEMBL	33	inhibitor	3.281729452230906	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	VECABRUTINIB	ncit:C136416	VECABRUTINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.081030357	SKLB1028	iuphar.ligand:12089	RUSERONTINIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.6848826682916673	Iruplinalkib	ncit:C154279	IRUPLINALKIB	FALSE	FALSE	FALSE
ARAF	hgnc:646	ARAF	ChEMBL	33	inhibitor	0.2386712328895204	BELVARAFENIB	ncit:C121646	BELVARAFENIB	FALSE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.3125456621172291	ESTETROL	rxcui:2539031	ESTETROL	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	GC1118	chembl:CHEMBL4650290	GC1118	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.4167275494896388	TRILACICLIB DIHYDROCHLORIDE	rxcui:2479691	TRILACICLIB DIHYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
GHR	hgnc:4263	GHR	ChEMBL	33	agonist	5.250767123569449	LONAPEGSOMATROPIN	rxcui:2569562	LONAPEGSOMATROPIN	TRUE	FALSE	FALSE
RB1	hgnc:9884	RB1	DTC	9/2/20	NULL	0.2586584789935689	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.3088686543276147	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	ChEMBL	33	inhibitor	1.875273972703375	CFI-400945	chembl:CHEMBL3408947	CFI-400945	FALSE	FALSE	FALSE
MYL3	hgnc:7584	MYL3	ChEMBL	33	activator	2.500365296937833	DANICAMTIV	ncit:C167013	DANICAMTIV	FALSE	FALSE	FALSE
MYH6	hgnc:7576	MYH6	ChEMBL	33	activator	2.500365296937833	DANICAMTIV	ncit:C167013	DANICAMTIV	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	1.009762908	PEGAPTANIB OCTASODIUM	chembl:CHEMBL2108752	PEGAPTANIB OCTASODIUM	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	negative modulator	0.038894571	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	negative modulator	0.035719504	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	4.773424657790408	VALTORCITABINE	ncit:C95912	VALTORCITABINE	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.021951368	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
IL33	hgnc:16028	IL33	ChEMBL	33	inhibitor	13.12691780892362	TORUDOKIMAB	ncit:C179128	TORUDOKIMAB	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	QUINUPRISTIN/DALFOPRISTIN	chembl:CHEMBL3137691	QUINUPRISTIN/DALFOPRISTIN	TRUE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	MOSUNETUZUMAB	rxcui:2625122	MOSUNETUZUMAB	TRUE	FALSE	FALSE
TIGIT	hgnc:26838	TIGIT	ChEMBL	33	inhibitor	6.563458904461812	ASP-8374	chembl:CHEMBL4297894	ASP-8374	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.03219848	PRIMAQUINE	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.4773424657790409	GW-406381	drugbank:DB12009	GW-406381	FALSE	FALSE	FALSE
TNFRSF4	hgnc:11918	TNFRSF4	ChEMBL	33	agonist	7.001022831425932	IVUXOLIMAB	ncit:C121927	IVUXOLIMAB	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.067839369	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	0.9723642821424906	MOSUNETUZUMAB	rxcui:2625122	MOSUNETUZUMAB	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1988926940746003	NS-2359	drugbank:DB05805	NS-2359	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	ChEMBL	33	inhibitor	0.2678962818147678	NIROGACESTAT	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.1411496538593938	OXATOMIDE	rxcui:54236	OXATOMIDE	TRUE	FALSE	FALSE
CCKAR	hgnc:1570	CCKAR	ChEMBL	33	agonist	2.625383561784724	SINCALIDE	rxcui:9800	SINCALIDE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	modulator	0.2243917574174979	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.041672755	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.042174836	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1435420208739598	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.041214813	NVP-BEZ237	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	COSMIC	4-Sep-20	NULL	0.1124502911321247	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1112450661773188	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	chembl:CHEMBL1256180	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123502	chembl:CHEMBL529640	CHEMBL:CHEMBL529640	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	RANOLAZINE HYDROCHLORIDE	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.005469549	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	1.050153425	CID 5310801	chembl:CHEMBL260451	CHEMBL:CHEMBL260451	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.079197091	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.009972967	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.00854617	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.009905239	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-725317	chembl:CHEMBL260417	CHEMBL:CHEMBL260417	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.040989595	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1988926940746003	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	DTC	9/2/20	NULL	0.1562728310586145	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1025540453822158	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005795549	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.2400350685060319	CIGLITAZONE	ncit:C72726	CIGLITAZONE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.080905503	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.1296485709523321	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006356861	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.1988926940746004	LAS38096	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.042073455	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.035358701	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002542252	TRIAMCINOLONE ACETONIDE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.030386384	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	GNF-PF-2243	chembl:CHEMBL600908	CHEMBL:CHEMBL600908	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	1-(4-HYDROXYPHENYL)MALEIMIDE	chembl:CHEMBL565893	CHEMBL:CHEMBL565893	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002356506	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	SJ000019194	chembl:CHEMBL592106	CHEMBL:CHEMBL592106	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.1017590527823536	PHENYLEPHRINE HYDROCHLORIDE	rxcui:8164	PHENYLEPHRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV006558	chembl:CHEMBL585243	CHEMBL:CHEMBL585243	FALSE	FALSE	FALSE
NLRP1	hgnc:14374	NLRP1	DTC	9/2/20	NULL	2.386712328895204	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.095122593	RAC-GONIOTHALAMIN	chembl:CHEMBL1170485	CHEMBL:CHEMBL1170485	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BROMOCHLOROACETIC ACID	chembl:CHEMBL504842	BROMOCHLOROACETIC ACID	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.008357102	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.052090944	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.005650847	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	H89	drugbank:DB07995	H-89	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.041085815	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.1262203635473425	AG-014361	iuphar.ligand:8094	AG14361	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005107253	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	PROGLUMETACIN	rxcui:34769	PROGLUMETACIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.010650643	DICLOFENAC SODIUM	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PALMATINE CHLORIDE HYDRATE	chembl:CHEMBL2163795	PALMATINE CHLORIDE HYDRATE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.012932924	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1025540453822158	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.06714536	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1312691780892362	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.043109746	HOE-33342	chembl:CHEMBL343002	CHEMBL:CHEMBL343002	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	PROSTAGLANDIN A2	iuphar.ligand:6279	PROSTAGLANDIN A2	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.042863405	TCMDC-125784	chembl:CHEMBL581574	CHEMBL:CHEMBL581574	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	MMV666022	chembl:CHEMBL599100	CHEMBL:CHEMBL599100	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016780975	GLAFENINE	ncit:C72119	GLAFENINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-1307	chembl:CHEMBL585030	CHEMBL:CHEMBL585030	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.3962843112127887	YUANHUADINE	chembl:CHEMBL1911631	YUANHUADINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.120017534	YUANHUADINE	chembl:CHEMBL1911631	YUANHUADINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	SCH-58261	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.018699313	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.01097339	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BENAZEPRIL HYDROCHLORIDE	rxcui:235758	BENAZEPRIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	PHENACYL CHLORIDE	iuphar.ligand:6285	OMEGA-CHLOROACETOPHENONE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015088411	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.001353012	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1172046232939609	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.023264365	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.012123683	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	4-HYDROXYDERRICIN	chembl:CHEMBL458094	CHEMBL:CHEMBL458094	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.040235763	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
DHX36	hgnc:14410	DHX36	DTC	9/2/20	NULL	52.50767123569449	MANOALIDE	chembl:CHEMBL463914	MANOALIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00282664	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
PABPC1	hgnc:8554	PABPC1	DTC	9/2/20	NULL	4.375639269641208	SJ000027778	chembl:CHEMBL592588	CHEMBL:CHEMBL592588	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	PROPOXYCAINE	ncit:C66492	PROPOXYCAINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.015002192	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	L-655240	chembl:CHEMBL362223	CHEMBL:CHEMBL362223	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.1508841127462485	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	MERSALYL	rxcui:6774	MERSALYL	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.305277158	RX-821002	iuphar.ligand:526	RX821002	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.012738397	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	REL-CISAPRIDE	chembl:CHEMBL74656	REL-CISAPRIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	2-ANILINOPYRIDINE	chembl:CHEMBL555260	CHEMBL:CHEMBL555260	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
GLO1	hgnc:4323	GLO1	DTC	9/2/20	NULL	17.50255707856483	2-(4-METHOXYBENZAMIDO)BENZOIC ACID	chembl:CHEMBL1701911	CHEMBL:CHEMBL1701911	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.054355767	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.011355465	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.4861821410712453	GNF-PF-1307	chembl:CHEMBL585030	CHEMBL:CHEMBL585030	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.6731752722524935	2,4-DIHYDROXYBENZOPHENONE	chembl:CHEMBL1392	2,4-DIHYDROXYBENZOPHENONE	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.013330203	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01823183	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	CLOROPHENE	rxcui:21290	CLOROPHENE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	1-PHYTEN-3-OL	chembl:CHEMBL453797	CHEMBL:CHEMBL453797	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00149902	HYDROCORTISONE BUTYRATE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
CDC25A	hgnc:1725	CDC25A	DTC	9/2/20	NULL	35.00511415712966	3-(3-STIBONOPHENYL)PROPANOIC ACID	iuphar.ligand:8877	P6949	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.017064567	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	CID 893238	chembl:CHEMBL473735	CHEMBL:CHEMBL473735	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001851731	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	TAXIFOLIN	drugbank:DB02224	TAXIFOLIN	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.024593757	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	NICOTINE BITARTRATE	rxcui:1306107	NICOTINE BITARTRATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.013120358	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	2.663432598912039	OBETICHOLIC ACID	rxcui:1798288	OBETICHOLIC ACID	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	SJ000191886	chembl:CHEMBL601616	CHEMBL:CHEMBL601616	FALSE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	1.166837138570989	TCMDC-125528	chembl:CHEMBL375673	CHEMBL:CHEMBL375673	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FOLPET	chembl:CHEMBL1883819	FOLPET	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.4861821410712453	BUFOTENINE	drugbank:DB01445	BUFOTENINE	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	DTC	9/2/20	NULL	2.234368988752957	DEOXYURIDINE MONOPHOSPHATE	drugbank:DB03800	DEOXYURIDINE MONOPHOSPHATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	KAVAIN	chembl:CHEMBL578607	KAVAIN	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.011585982	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.1084869240406911	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	TCMDC-123828	chembl:CHEMBL588804	CHEMBL:CHEMBL588804	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.001699277	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	HARMOL	chembl:CHEMBL486817	HARMOL	FALSE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	DTC	9/2/20	NULL	6.563458904461812	CL-075	iuphar.ligand:9270	3M-002	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.020117882	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.029041854	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.008640393	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.038837035	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	AMITRIPTYLINOXIDE	ncit:C72698	AMITRIPTYLINOXIDE	FALSE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.057764215	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-2243	chembl:CHEMBL600908	CHEMBL:CHEMBL600908	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.043902735	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	GNF-PF-308	chembl:CHEMBL600334	CHEMBL:CHEMBL600334	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	LASSBIO-294	chembl:CHEMBL233194	CHEMBL:CHEMBL233194	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1274458039701322	METHYL PARATHIONE	chembl:CHEMBL346516	METHYL PARATHIONE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.021240967	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.1842374429322613	ARTESUNATE	rxcui:18346	ARTESUNATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002767057	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.2983390411119005	SJ000180366	chembl:CHEMBL609036	CHEMBL:CHEMBL609036	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	METHYL ROBUSTONE	chembl:CHEMBL1403041	METHYL ROBUSTONE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.276356164	JL-18	chembl:CHEMBL63329	CHEMBL:CHEMBL63329	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	ISOPROPAMIDE	rxcui:89784	ISOPROPAMIDE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.750109589	GNF-PF-910	chembl:CHEMBL585408	CHEMBL:CHEMBL585408	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	DNDI1417411	chembl:CHEMBL1445650	CHEMBL:CHEMBL1445650	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.033086119	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.085239726	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	SHINPTEROCARPIN	chembl:CHEMBL591773	SHINPTEROCARPIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01823183	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.028413242	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	VANITIOLIDE	ncit:C74234	VANITIOLIDE	FALSE	FALSE	FALSE
KISS1R	hgnc:4510	KISS1R	DTC	9/2/20	NULL	6.563458904461812	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
RPS6KA5	hgnc:10434	RPS6KA5	DTC	9/2/20	NULL	0.074268276	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004264756	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005953251	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.003371279	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	NSC-119236	chembl:CHEMBL458765	CHEMBL:CHEMBL458765	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	2.282942227638891	HOLACANTHONE	chembl:CHEMBL519243	HOLACANTHONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	BRILLIANT GREEN OXALATE	chembl:CHEMBL1789985	BRILLIANT GREEN OXALATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	GNF-PF-4668	chembl:CHEMBL584860	CHEMBL:CHEMBL584860	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2365210416022274	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.1548898856510162	SJ000244629	chembl:CHEMBL592115	CHEMBL:CHEMBL592115	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.095122593	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.009430257	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003147942	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	FLUNARIZINE HYDROCHLORIDE	rxcui:82019	FLUNARIZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.130291988	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003401858	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.020737627	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	SJ000032149	chembl:CHEMBL600778	CHEMBL:CHEMBL600778	FALSE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	4.039051633514961	DNDI1417874	chembl:CHEMBL1865517	CHEMBL:CHEMBL1865517	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	HYDROFLUMETHIAZIDE	rxcui:5495	HYDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	WHILE OLIVETOL	chembl:CHEMBL154533	WHILE OLIVETOL	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.050764748	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CHLORBROMURON	chembl:CHEMBL1275654	CHLORBROMURON	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002663877	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	GNF-PF-1307	chembl:CHEMBL585030	CHEMBL:CHEMBL585030	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	N-HISTIDYL-2-AMINONAPHTHALENE (BETANA)	chembl:CHEMBL1489988	N-HISTIDYL-2-AMINONAPHTHALENE (BETANA)	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ETHOFUMESATE	chembl:CHEMBL2133153	ETHOFUMESATE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	GIPARMEN	ncit:C74115	GIPARMEN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	METHYLBENZETHONIUM	rxcui:29829	METHYLBENZETHONIUM	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.005881236	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	S-(+)-FLUOXETINE HCL	chembl:CHEMBL1257031	CHEMBL:CHEMBL1257031	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013825085	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	GR-103545	iuphar.ligand:1649	GR 89696	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.2117244807890907	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1981421556063943	DNDI1417809	chembl:CHEMBL1442783	CHEMBL:CHEMBL1442783	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	MMV006513	chembl:CHEMBL585622	CHEMBL:CHEMBL585622	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	KALOPANAX-SAPONIN F METHYL ESTER	chembl:CHEMBL1834951	CHEMBL:CHEMBL1834951	FALSE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.078252863	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.033148782	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
CDK5R1	hgnc:1775	CDK5R1	DTC	9/2/20	NULL	0.2083637747448194	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	TCMDC-125738	chembl:CHEMBL527585	CHEMBL:CHEMBL527585	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	GNF-PF-4057	chembl:CHEMBL598903	CHEMBL:CHEMBL598903	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.008245551	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.007952093	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	THIOTEPA	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	2-ANILINOPYRIDINE	chembl:CHEMBL555260	CHEMBL:CHEMBL555260	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.035005114	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2220197515251353	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2075402025126264	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.1591141552596803	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2128689374420047	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.1221108633388244	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	THIABENDAZOLE	rxcui:10450	THIABENDAZOLE	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2128689374420047	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.026372512	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.027440643	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	L-655240	chembl:CHEMBL362223	CHEMBL:CHEMBL362223	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	3,4-DIHYDROXYPHENYLACETIC ACID	chembl:CHEMBL1284	3,4-DIHYDROXYPHENYLACETIC ACID	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2430910705356226	GNF-PF-4242	chembl:CHEMBL584514	CHEMBL:CHEMBL584514	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	CLOFOCTOL	rxcui:21264	CLOFOCTOL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	DIHYDROXANTHOHUMOL	chembl:CHEMBL510279	DIHYDROXANTHOHUMOL	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	UNGEREMINE	chembl:CHEMBL479291	UNGEREMINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	CAPENSIN	chembl:CHEMBL1327256	CAPENSIN	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	TCMDC-124327	chembl:CHEMBL581929	CHEMBL:CHEMBL581929	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	METHOPRENE	chembl:CHEMBL1875086	METHOPRENE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	PYRANTEL PAMOATE	rxcui:8985	PYRANTEL PAMOATE	TRUE	FALSE	FALSE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8954	iuphar.ligand:8954	GSK591	FALSE	FALSE	FALSE
SETD7	hgnc:30412	SETD7	DTC	9/2/20	NULL	52.50767123569449	SINEFUNGIN	ncit:C73041	SINEFUNGIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.051478109	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008279355	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.2365210416022274	PECTOLINARIGENIN	chembl:CHEMBL78010	PECTOLINARIGENIN	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.04464938	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CHRM1	hgnc:1950	CHRM1	DTC	9/2/20	NULL	0.1117184494376478	PIPERTRAMINE	chembl:CHEMBL127273	PIPERTRAMINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	TCMDC-124032	chembl:CHEMBL536375	CHEMBL:CHEMBL536375	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.025280535	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	FENDILINE HYDROCHLORIDE	rxcui:236767	FENDILINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	TORSEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	NISOXETINE HYDROCHLORIDE	chembl:CHEMBL1256695	NISOXETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.2853677784548614	SU-11274	iuphar.ligand:5057	SU11274	FALSE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.009181268	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	NSC-24047	chembl:CHEMBL1288013	CHEMBL:CHEMBL1288013	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	ROEMERINE	chembl:CHEMBL36654	ROEMERINE	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	RAC-ARISTOYUNNOLIN D	chembl:CHEMBL2333543	CHEMBL:CHEMBL2333543	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010678802	PHENOXYBENZAMINE	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	DTC	9/2/20	NULL	5.834185692854944	ALAPROCLATE HYDROCHLORIDE	chembl:CHEMBL1256359	ALAPROCLATE HYDROCHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.010588359	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.013045384	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.042863405	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.8078103267029924	GNF-PF-4227	chembl:CHEMBL585654	CHEMBL:CHEMBL585654	FALSE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.7001022831425934	rasburicase	rxcui:283821	RASBURICASE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DEBRISOQUIN SULFATE	ncit:C77302	DEBRISOQUIN SULFATE	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.5303805175322676	DIFLUFENICAN	chembl:CHEMBL1425995	DIFLUFENICAN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1029562181092048	SJ000082806	chembl:CHEMBL494668	CHEMBL:CHEMBL494668	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	BW-723C86	iuphar.ligand:161	BW723C86	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.026899422	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	GNF-PF-3537	chembl:CHEMBL601110	CHEMBL:CHEMBL601110	FALSE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	DTC	9/2/20	NULL	0.4922594178346359	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.012268147	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.036977233	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
CDK5R1	hgnc:1775	CDK5R1	DTC	9/2/20	NULL	0.375054795	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE	chembl:CHEMBL513116	N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006356861	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.032412143	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.016807833	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009579944	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2713574740862764	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007374673	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	METHAZOLAMIDE	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002861765	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
RPS27A	hgnc:10417	RPS27A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	PANTOPRAZOLE SODIUM	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	AMARANTH	chembl:CHEMBL1408927	AMARANTH	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001771873	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.040989595	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	N-METHYLDOPAMINE HCL	chembl:CHEMBL1256484	CHEMBL:CHEMBL1256484	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	DIMENHYDRINATE	rxcui:3444	DIMENHYDRINATE	TRUE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	0.1154014752432846	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.062065805	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	NSC-677438	chembl:CHEMBL118678	CHEMBL:CHEMBL118678	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.045898314	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-2954	chembl:CHEMBL582722	CHEMBL:CHEMBL582722	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.004139351	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	THIOTEPA	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	ASARININ	chembl:CHEMBL43469	ASARININ	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001276441	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.02091106	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.014046996	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	ASARININ	chembl:CHEMBL43469	ASARININ	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	METHIOTHEPIN MESYLATE	chembl:CHEMBL1256737	METHIOTHEPIN MESYLATE	FALSE	FALSE	FALSE
PIM2	hgnc:8987	PIM2	DTC	9/2/20	NULL	0.064984742	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.073954467	TIVOZANIB HYDROCHLORIDE	rxcui:2534245	TIVOZANIB HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.1056492378987816	TCMDC-125543	chembl:CHEMBL546170	CHEMBL:CHEMBL546170	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009144492	MONTELUKAST SODIUM	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	MECYSTEINE HYDROCHLORIDE	rxcui:235828	MECYSTEINE HYDROCHLORIDE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	DNDI1417085	chembl:CHEMBL1522984	CHEMBL:CHEMBL1522984	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	TIOTIDINE	ncit:C152643	TIOTIDINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.011419676	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	CINTAZONE	ncit:C73084	CINTAZONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	ARCTIGENIN	drugbank:DB16880	ARCTIGENIN	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.013777925	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.076765601	2',4'-DIHYDROXYCHALCONE	chembl:CHEMBL105310	2',4'-DIHYDROXYCHALCONE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	TACRINE	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	CP-339818	iuphar.ligand:2558	CP-339818	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.03849536	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.03223307	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.002443467	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
SOD1	hgnc:11179	SOD1	DTC	9/2/20	NULL	0.4565884455277782	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	FLUACIZINE	ncit:C65702	FLUACIZINE	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.029498692	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.04464938	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
ATP7B	hgnc:870	ATP7B	NCI	14-Sep-17	NULL	0.1207072901969988	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	PHYSOSTIGMINE	rxcui:8299	PHYSOSTIGMINE	TRUE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.015525627	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	PIPERIDINE-2,3-DICARBOXYLIC ACID	chembl:CHEMBL124460	CHEMBL:CHEMBL124460	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	TRIPHENYLSTANNYL ACETATE	chembl:CHEMBL474376	TRIPHENYLSTANNYL ACETATE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	ORYZALIN	chembl:CHEMBL295960	ORYZALIN	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.045898314	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-4674	chembl:CHEMBL584452	CHEMBL:CHEMBL584452	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	PAPAVEROLINE	ncit:C66306	PAPAVEROLINE	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.3281729452230906	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.013415348	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	NSC-48300	chembl:CHEMBL1091971	CHEMBL:CHEMBL1091971	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CROMOLYN SODIUM	rxcui:3538	CROMOLYN SODIUM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	PF-03715455	drugbank:DB12138	PF-03715455	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.05664258	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.025865848	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	HYMECROMONE	rxcui:5556	HYMECROMONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TCMDC-125606	chembl:CHEMBL536166	CHEMBL:CHEMBL536166	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.1627303860610366	icotinib	ncit:C138996	ICOTINIB	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	TCMDC-125321	chembl:CHEMBL587449	CHEMBL:CHEMBL587449	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.1944728564284981	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.031612084	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004919212	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008345148	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.091796628	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	DTC	9/2/20	NULL	1.666910197958555	GNF-2	iuphar.ligand:5935	BCR-ABL INHIBITOR GNF-2	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.059667808	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.045579576	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TRENBOLONE ACETATE	rxcui:1484277	TRENBOLONE ACETATE	TRUE	FALSE	FALSE
NTSR1	hgnc:8039	NTSR1	DTC	9/2/20	NULL	0.3804903712731485	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.056888051	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	DTC	9/2/20	NULL	7.501095891	OXACILLIN	rxcui:7773	OXACILLIN	TRUE	FALSE	FALSE
BMP2	hgnc:1069	BMP2	DTC	9/2/20	NULL	26.25383561784724	ISOPROPYL 4-AMINOBENZOATE	chembl:CHEMBL1467165	CHEMBL:CHEMBL1467165	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.3017682254924971	2,3,4,4'-TETRAMETHOXYBIPHENYL	chembl:CHEMBL28250	2,3,4,4'-TETRAMETHOXYBIPHENYL	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.035502144	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	BENZALKONIUM CHLORIDE	rxcui:1379	BENZALKONIUM CHLORIDE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.019339842	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	ENNIATIN B	chembl:CHEMBL469036	ENNIATIN B	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BUPROFEZIN	chembl:CHEMBL1891512	BUPROFEZIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.3241214273808302	CENTANAFADINE	ncit:C171666	CENTANAFADINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010058941	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.172722603	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.030176823	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	LINSIDOMINE	ncit:C72628	LINSIDOMINE	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.021661581	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.037398626	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.010685322	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.030004384	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
UNIPROT:Q9GZP0	hgnc:30620	PDGFD	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	CR002	drugbank:DB05139	CR002	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.016491103	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.003353837	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
FPR1	hgnc:3826	FPR1	DTC	9/2/20	NULL	1.166837138570988	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00988845	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.042344896	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.002998382	PARAPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	1.500219178	BAS-8770957	chembl:CHEMBL500812	CHEMBL:CHEMBL500812	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ALFATRADIOL	rxcui:1926478	ALFATRADIOL	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.016491103	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.4375639269641208	CGP-60474	chembl:CHEMBL300389	CHEMBL:CHEMBL300389	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.173866461	GNF-PF-3268	chembl:CHEMBL582073	CHEMBL:CHEMBL582073	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.028850369	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003616231	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	CHLORQUINALDOL	rxcui:2407	CHLORQUINALDOL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.006858369	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:5719	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.010975684	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.004883526	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.021240967	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	5-BENZYLOXYTRYPTAMINE	iuphar.ligand:265	5-BENZYLOXYTRYPTAMINE	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.060008767	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1232574442152452	TCMDC-125580	chembl:CHEMBL528807	CHEMBL:CHEMBL528807	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	NSC-111847	chembl:CHEMBL1984884	CHEMBL:CHEMBL1984884	FALSE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.063722902	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1591141552596803	5-(N-ETHYL-N-ISOPROPYL)AMILORIDE	iuphar.ligand:4186	ETHYLISOPROPYLAMILORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	HOE-33342	chembl:CHEMBL343002	CHEMBL:CHEMBL343002	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	5-METHOXYISATIN	chembl:CHEMBL222660	5-METHOXYISATIN	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.018786287	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.1682938180631234	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.02926849	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.138178082	(R)-NITRENDIPINE	chembl:CHEMBL268609	(R)-NITRENDIPINE	FALSE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	0.4150804050252529	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.028645756	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.008821853	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	DTC	9/2/20	NULL	1.029562181092048	DESMOPRESSIN	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1207072901969988	OXETHAZAINE	ncit:C81409	OXETHAZAINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004252322	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.005101299	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	ISOXSUPRINE	rxcui:6066	ISOXSUPRINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	GLYASPERIN D	chembl:CHEMBL1563332	GLYASPERIN D	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	PENICILLIN V BENZATHINE	rxcui:18926	PENICILLIN V BENZATHINE	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.046881849	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.00825852	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.021240967	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004427291	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	XCT790	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	1.981421556063943	PYROCATECHOL VIOLET	chembl:CHEMBL210574	PYROCATECHOL VIOLET	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001657439	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.01274458	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	PHENAZINE-1-CARBOXYLIC ACID	chembl:CHEMBL463686	PHENAZINE-1-CARBOXYLIC ACID	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	SJ000262868	chembl:CHEMBL589444	CHEMBL:CHEMBL589444	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.045461187	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.017811286	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-124009	chembl:CHEMBL1366623	CHEMBL:CHEMBL1366623	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.1363835616511545	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.056826484	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	(S)-ALAPROCLATE	chembl:CHEMBL251941	(S)-ALAPROCLATE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.020117882	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	CIViC	10-Apr-24	NULL	0.08334551	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.021070494	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	MMV006389	chembl:CHEMBL586000	CHEMBL:CHEMBL586000	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.069454592	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.009430257	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.1278595890479573	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	TRANILAST	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.034318739	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.081281225	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1023541349623674	TCMDC-124536	chembl:CHEMBL580851	CHEMBL:CHEMBL580851	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	QUINOXYFEN	chembl:CHEMBL1869863	QUINOXYFEN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	GNF-PF-910	chembl:CHEMBL585408	CHEMBL:CHEMBL585408	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007378818	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.013411921	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.071439008	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 4	hgnc:3691	FGFR4	TTD	2020.06.01	NULL	1.117184494376478	ISIS-FGFR4Rx	drugbank:DB16198	IONIS-FGFR4RX	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	LINOLEIC ACID	rxcui:6400	LINOLEIC ACID	TRUE	FALSE	FALSE
CAMK2A	hgnc:1460	CAMK2A	DTC	9/2/20	NULL	0.072826174	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	GNF-PF-5242	chembl:CHEMBL600107	CHEMBL:CHEMBL600107	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.018106094	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.019724895	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	IMIDACLOPRID	rxcui:1251576	IMIDACLOPRID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.001990737	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1861974157294131	(S)-VERAPAMIL	chembl:CHEMBL36148	(S)-VERAPAMIL	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.007264481	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	LACTIC ACID	rxcui:1314409	DL-LACTIC ACID	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006978691	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.005158431	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.002998382	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.019483366	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
CA1	hgnc:1368	CA1	DTC	9/2/20	NULL	0.2386712328895204	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ALPHA-ENDOSULFAN	chembl:CHEMBL1890408	ALPHA-ENDOSULFAN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	CHLORACYZINE	ncit:C80874	CHLORACYZINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	METHOCARBAMOL	rxcui:6845	METHOCARBAMOL	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.009409977	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	KAVAIN	chembl:CHEMBL578607	KAVAIN	FALSE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.1539814405738841	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	3.424413341458336	JANEX-1	chembl:CHEMBL405130	WHI-P131	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.4667348554283955	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.4102161815288632	NSC-50654	chembl:CHEMBL1372046	CHEMBL:CHEMBL1372046	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE	chembl:CHEMBL457504	CHEMBL:CHEMBL457504	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005899738	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.3201687270469177	NSC-50654	chembl:CHEMBL1372046	CHEMBL:CHEMBL1372046	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	FIDUXOSIN HYDROCHLORIDE	ncit:C81371	FIDUXOSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
PSMA8	hgnc:22985	PSMA8	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.01917038	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.017679351	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.008385128	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DITHIODIMORPHOLINE	chembl:CHEMBL582932	DITHIODIMORPHOLINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.043902735	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003720782	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
DUSP3	hgnc:3069	DUSP3	DTC	9/2/20	NULL	0.258658479	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.013206155	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.016116535	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.038382801	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	1R,9S-HYDRASTINE	chembl:CHEMBL475536	1R,9S-HYDRASTINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	GNF-PF-2968	chembl:CHEMBL582473	CHEMBL:CHEMBL582473	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.6250913242344582	CEP-5214	chembl:CHEMBL150894	CEP-5214	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.3697723326457359	HL010183	chembl:CHEMBL2348411	CHEMBL:CHEMBL2348411	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007596596	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	N-METHYLDOPAMINE HCL	chembl:CHEMBL1256484	CHEMBL:CHEMBL1256484	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	CHLORHEXIDINE HYDROCHLORIDE	rxcui:2361	CHLORHEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	CID 926663	chembl:CHEMBL265686	CHEMBL:CHEMBL265686	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.003259524	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.364636606	NSC-158389	chembl:CHEMBL192626	CHEMBL:CHEMBL192626	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.039155609	TICRYNAFEN	ncit:C152613	TICRYNAFEN	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.212581665	MMV000634	chembl:CHEMBL602946	CHEMBL:CHEMBL602946	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002450766	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.024141458	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	HYDRAMETHYLNON	chembl:CHEMBL464812	HYDRAMETHYLNON	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	NORGESTIMATE	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIBEKACIN	rxcui:3328	DIBEKACIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	GNF-PF-3352	chembl:CHEMBL600306	CHEMBL:CHEMBL600306	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	CHARTREUSIN	chembl:CHEMBL1554674	CHARTREUSIN	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	COSMIC	4-Sep-20	NULL	0.384671584	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
AKR1C3	hgnc:386	AKR1C3	DTC	9/2/20	NULL	7.001022831425932	3-((4-(TRIFLUOROMETHYL)PHENYL)AMINO)BENZOIC ACID	chembl:CHEMBL1682202	CHEMBL:CHEMBL1682202	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.018567069	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	(R)-NITRENDIPINE	chembl:CHEMBL268609	(R)-NITRENDIPINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004585022	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,7-BIS[3-(PYRROLIDINO)PROPIONAMIDO]ANTHRAQUINONE	chembl:CHEMBL144757	CHEMBL:CHEMBL144757	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.025739055	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	TRANSPLATIN	chembl:CHEMBL1386	TRANSPLATIN	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.054638576	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	HYDROXYZINE	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1526385791735305	CCG-63808	iuphar.ligand:8725	CCG-63808	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.5556367326528519	TETRAHYDROAPLYSULPHURIN-1	chembl:CHEMBL1077773	CHEMBL:CHEMBL1077773	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.024354207	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
IL4R	hgnc:6015	IL4R	ChEMBL	33	binder	5.834185692854944	CINTREDEKIN BESUDOTOX	ncit:C2599	CINTREDEKIN BESUDOTOX	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.068907705	ARACHIDONOYL DOPAMINE	iuphar.ligand:4261	NADA	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	METHYCLOTHIAZIDE	rxcui:6860	METHYCLOTHIAZIDE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.8607814956671229	TIOPRONIN	rxcui:6765	TIOPRONIN	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.012020987	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CDK5R1	hgnc:1775	CDK5R1	DTC	9/2/20	NULL	1.250182648468916	CGP-60474	chembl:CHEMBL300389	CHEMBL:CHEMBL300389	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.1988926940746003	CGP-60474	chembl:CHEMBL300389	CHEMBL:CHEMBL300389	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	NSC-61836	chembl:CHEMBL521171	CHEMBL:CHEMBL521171	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.036413087	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	FUSARIC ACID	chembl:CHEMBL24510	FUSARIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	ARACHIDONOYL DOPAMINE	iuphar.ligand:4261	NADA	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.004776899	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.046425881	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.02646556	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	NALED	chembl:CHEMBL1887067	NALED	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.014749346	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.1643432589536604	TALAROFLAVONE	chembl:CHEMBL408995	TALAROFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5612	ncit:C152892	VIPADENANT	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.011217191	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	2,4,6-TRIHYDROXYACETOPHENONE	chembl:CHEMBL452477	2,4,6-TRIHYDROXYACETOPHENONE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.7242437411819931	ARGENTEOSIDE A	chembl:CHEMBL2332352	ARGENTEOSIDE A	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	PROPIONYLPROMAZINE HYDROCHLORIDE	chembl:CHEMBL1256661	PROPIONYLPROMAZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	1.166837138570988	BAS-0338868	chembl:CHEMBL378903	CHEMBL:CHEMBL378903	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.2059124362184097	IUPHAR.LIGAND:8210	iuphar.ligand:8210	COMPOUND 27 [PMID: 21123062]	FALSE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.4375639269641208	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003307362	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.061628722	NSC-61836	chembl:CHEMBL521171	CHEMBL:CHEMBL521171	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.546954909	CYTARABINE HYDROCHLORIDE	ncit:C71603	CYTARABINE HYDROCHLORIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005483257	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	KHELLIN	rxcui:6147	KHELLIN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.006806802	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	TEROXIRONE	ncit:C2320	TEROXIRONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.078545507	ZM336372	iuphar.ligand:9130	ZM336372	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	FASUDIL HYDROCHLORIDE	chembl:CHEMBL541388	FASUDIL HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	CROMOLYN	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.002734775	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1112450661773188	A-77636 HCL	chembl:CHEMBL1256876	CHEMBL:CHEMBL1256876	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.8751278539282416	Arformoterol	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
MMP12	hgnc:7158	MMP12	DTC	9/2/20	NULL	0.8334550989792776	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.023620185	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	2.019525817	NSC-640558	chembl:CHEMBL1288281	CHEMBL:CHEMBL1288281	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.009065551	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.072927321	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.056826484	FRENTIZOLE	ncit:C167023	FRENTIZOLE	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.3182283105193606	MMV666022	chembl:CHEMBL599100	CHEMBL:CHEMBL599100	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.015516451	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	SAQUINAVIR	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	ACACETIN DIACETATE	chembl:CHEMBL1566650	ACACETIN DIACETATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.016856395	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	SCH-53020	chembl:CHEMBL66279	CHEMBL:CHEMBL66279	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	MK-212	drugbank:DB12111	MK-212	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.056826484	DNDI1417031	chembl:CHEMBL1333049	CHEMBL:CHEMBL1333049	FALSE	FALSE	FALSE
CHAT	hgnc:1912	CHAT	NCI	14-Sep-17	NULL	0.1356787370431382	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PBK	hgnc:18282	PBK	DTC	9/2/20	NULL	0.1179947668217854	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.035502144	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	PENTAMIDINE DIISETHIONATE	chembl:CHEMBL361506	PENTAMIDINE ISETHIONATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002088278	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.008334551	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.026045472	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
PRKG1	hgnc:9414	PRKG1	DTC	9/2/20	NULL	0.078252863	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.1319288222002374	ASCORBYL PALMITATE	ncit:C81556	ASCORBYL PALMITATE	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.020696756	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.027476542	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	1.363835616511545	LEUCETTAMINE B	chembl:CHEMBL485053	LEUCETTAMINE B	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	CID 5310801	chembl:CHEMBL260451	CHEMBL:CHEMBL260451	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.2143170254518142	DOMIPHEN BROMIDE	rxcui:49255	DOMIPHEN BROMIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.010724606	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	NORDEFRIN	ncit:C81340	NORDEFRIN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.4907258993990139	4-(1,1-DIETHYLPROPYL)PHENOL	chembl:CHEMBL2313444	CHEMBL:CHEMBL2313444	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.016927038	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.044955198	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	DTC	9/2/20	NULL	0.06714536	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	SJ000082806	chembl:CHEMBL494668	CHEMBL:CHEMBL494668	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	CID 893238	chembl:CHEMBL473735	CHEMBL:CHEMBL473735	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.056459862	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.014537008	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
RPS6KA5	hgnc:10434	RPS6KA5	DTC	9/2/20	NULL	0.1704794520639432	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	DTC	9/2/20	NULL	8.751278539282415	3-(2-AZIDOETHYL)THIOPHENE	chembl:CHEMBL589270	CHEMBL:CHEMBL589270	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.024275391	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	CHRYSIN DIMETHYL ETHER	chembl:CHEMBL275391	CHRYSIN DIMETHYL ETHER	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	THAPSIGARGIN	ncit:C128634	THAPSIGARGIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007937668	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.037398626	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011205222	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	PAPAVEROLINE	ncit:C66306	PAPAVEROLINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	BOPINDOLOL	rxcui:19605	BOPINDOLOL	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.4375639269641209	DNQX	chembl:CHEMBL155265	DNQX	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	TCMDC-125738	chembl:CHEMBL527585	CHEMBL:CHEMBL527585	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.003207947	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.108040476	1-O-ACETYLGEOPYXIN A	chembl:CHEMBL1902074	CHEMBL:CHEMBL1902074	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ARTHONIOIC ACID	chembl:CHEMBL1332204	ARTHONIOIC ACID	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	PECTOLINARIGENIN	chembl:CHEMBL78010	PECTOLINARIGENIN	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	CONICASTEROL E	chembl:CHEMBL1950810	CONICASTEROL E	FALSE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.030581055	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SLC22A1	hgnc:10963	SLC22A1	DTC	9/2/20	NULL	0.8204323630577265	ELTROMBOPAG	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.023514407	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	NSC-108783	chembl:CHEMBL1489812	CHEMBL:CHEMBL1489812	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.021357605	SILDENAFIL	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.015930725	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.151537291	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.1875273972703374	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.021951368	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	2.625383561784724	LISSOCLINIDINE B	chembl:CHEMBL461462	LISSOCLINIDINE B	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.048083948	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1810609352954982	DIACYLGLYCEROL KINASE INHIBITOR II	iuphar.ligand:5957	DIACYLGLYCEROL KINASE INHIBITOR II	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	TCMDC-138263	chembl:CHEMBL535307	CHEMBL:CHEMBL535307	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	SALAGEN	chembl:CHEMBL611494	SALAGEN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005953251	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	3,3',4'-TRIHYDROXYFLAVONE	chembl:CHEMBL122701	CHEMBL:CHEMBL122701	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	1,4-BIS(2,6-DIFLUOROPHENYLSULFONYL)PIPERAZINE	chembl:CHEMBL1093369	CHEMBL:CHEMBL1093369	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.084689792	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SJ000071821	chembl:CHEMBL589924	CHEMBL:CHEMBL589924	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.036463661	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	PURGIN II	chembl:CHEMBL2336636	PURGIN II	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	2.019525817	BERKELEYAMIDE C	chembl:CHEMBL468641	BERKELEYAMIDE C	FALSE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.4039051633514962	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.052090944	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	AMINACRINE	rxcui:645	AMINACRINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.0053937	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	DIMETHENAMID	chembl:CHEMBL1565335	DIMETHENAMID	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	NSC-367089	chembl:CHEMBL1543865	CHEMBL:CHEMBL1543865	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.2958178661165888	NORBINALTORPHIMINE	iuphar.ligand:1642	NOR-BINALTORPHIMINE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	3,4-DIHYDROXYPHENYLACETIC ACID	chembl:CHEMBL1284	3,4-DIHYDROXYPHENYLACETIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	ORYZALIN	chembl:CHEMBL295960	ORYZALIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.014832675	IDAZOXAN	ncit:C170049	IDAZOXAN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	GSK0660	iuphar.ligand:3441	GSK0660	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	2,4-DIHYDROXYBENZOPHENONE	chembl:CHEMBL1392	2,4-DIHYDROXYBENZOPHENONE	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	FDA	10-Apr-24	NULL	0.7059854956059763	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.009862448	Doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.007378818	Codeine	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	FDA	10-Apr-24	NULL	0.760980743	Elagolix	rxcui:2049846	ELAGOLIX	TRUE	FALSE	FALSE
PROC	hgnc:9451	PROC	FDA	10-Apr-24	NULL	0.1117184494376478	Estradiol	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.1229687850953032	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	FDA	10-Apr-24	NULL	0.4735986033023426	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.048618214	Ospemifene	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.5666295457089334	Omacetaxine	rxcui:1546446	OMACETAXINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.6168664383892681	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.013622434	Perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.056622219	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.018782447	Trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1500219178162699	Tolazamide	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.1132444383228493	Toremifene	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.078958904	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.16256245	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	MyCancerGenome	20-Jun-17	inhibitor	0.5834185692854944	NMS-1286937	chembl:CHEMBL1094408	NMS-1286937	FALSE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	MyCancerGenome	20-Jun-17	inhibitor	1.346350544504987	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PRKCA	hgnc:9393	PRKCA	MyCancerGenome	20-Jun-17	inhibitor	0.1215455352678113	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	antibody	3.962843112127886	FIGITUMUMAB	ncit:C52187	FIGITUMUMAB	FALSE	TRUE	TRUE
IL6R	hgnc:6019	IL6R	MyCancerGenome	20-Jun-17	immunotherapy	4.039051633514961	TOCILIZUMAB	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	MyCancerGenome	20-Jun-17	other/unknown	0.2263261691193728	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
NOTCH4	hgnc:7884	NOTCH4	MyCancerGenome	20-Jun-17	other/unknown	1.750255707856483	RO4929097	iuphar.ligand:7338	RO4929097	FALSE	FALSE	TRUE
NOTCH2	hgnc:7882	NOTCH2	MyCancerGenome	20-Jun-17	other/unknown	1.500219178	RO4929097	iuphar.ligand:7338	RO4929097	FALSE	FALSE	TRUE
PARP1	hgnc:270	PARP1	MyCancerGenome	20-Jun-17	other/unknown	1.225178995499538	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
PSMD4	hgnc:9561	PSMD4	MyCancerGenome	20-Jun-17	other/unknown	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC4	hgnc:9551	PSMC4	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC5	hgnc:9552	PSMC5	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD10P2	hgnc:30151	PSMD10P2	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC1P1	hgnc:30147	PSMC1P1	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA2	hgnc:9531	PSMA2	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC3	hgnc:9549	PSMC3	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1190650141398968	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
FOLR1	hgnc:3791	FOLR1	NCI	14-Sep-17	NULL	0.067839369	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PSME2	hgnc:9569	PSME2	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1099061668983662	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.082429625	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.052824619	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
DDR2	hgnc:2731	DDR2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.6364566210387212	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.074975256	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.094535416	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
ABCB4	hgnc:45	ABCB4	NCI	14-Sep-17	NULL	0.2414145803939976	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.1495945049449985	QUINONE	rxcui:319868	1,4-BENZOQUINONE	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	1.721562991334245	MS-209	ncit:C2231	DOFEQUIDAR FUMARATE	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.032817295	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.08607815	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.091159151	DEHYDROEPIANDROSTERONE	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
ABCC6	hgnc:57	ABCC6	NCI	14-Sep-17	NULL	0.062509132	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.073062622	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	NCI	14-Sep-17	NULL	2.187819634820604	SULFONATES	ncit:C222	ALKYLSULFONATE COMPOUND	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.01127621	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
ACE	hgnc:2707	ACE	NCI	14-Sep-17	NULL	0.052350619	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
ACP5	hgnc:124	ACP5	NCI	14-Sep-17	NULL	0.08780547	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	1.544343271638073	MAGNESIUM CHLORIDE	rxcui:1311539	MAGNESIUM CHLORIDE ANHYDROUS	TRUE	FALSE	FALSE
ACP5	hgnc:124	ACP5	NCI	14-Sep-17	NULL	0.3671865121377238	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	0.046798281	6-THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ACLY	hgnc:115	ACLY	NCI	14-Sep-17	NULL	2.386712328895204	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
ADCYAP1	hgnc:241	ADCYAP1	NCI	14-Sep-17	NULL	0.5707355569097228	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	MEPANIPYRIM	chembl:CHEMBL2269513	MEPANIPYRIM	FALSE	FALSE	FALSE
ADCYAP1R1	hgnc:242	ADCYAP1R1	NCI	14-Sep-17	NULL	0.2941606231691568	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.02339914	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ALPP	hgnc:439	ALPP	NCI	14-Sep-17	NULL	0.7778914257139926	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	NCI	14-Sep-17	NULL	0.090843722	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
ATF2	hgnc:784	ATF2	NCI	14-Sep-17	NULL	0.6731752722524936	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.050007306	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	3,6-DIMETHOXYFLAVONE	chembl:CHEMBL1331521	3,6-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
BCAR3	hgnc:973	BCAR3	NCI	14-Sep-17	NULL	7.001022831425933	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.065675636	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.027840759	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.008537833	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.04685396	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
NCBIGENE:2764	hgnc:4373	GMFB	GuideToPharmacology	2024.1	antibody	4.375639269641208	IUPHAR.LIGAND:11131	rxcui:2387211	TAFASITAMAB	TRUE	FALSE	FALSE
CCND2	hgnc:1583	CCND2	NCI	14-Sep-17	NULL	0.84012274	5-AZA-2-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	0.3365876361262468	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
CCR6	hgnc:1607	CCR6	NCI	14-Sep-17	NULL	2.333674277141977	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	NCI	14-Sep-17	NULL	0.760980743	OPIATE	ncit:C1657	OPIATE	FALSE	FALSE	FALSE
CD38	hgnc:1667	CD38	NCI	14-Sep-17	NULL	0.4861821410712453	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.201952582	PHENYLEPHRINE HYDROCHLORIDE	rxcui:8164	PHENYLEPHRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CD63	hgnc:1692	CD63	NCI	14-Sep-17	NULL	3.088686543276147	NONSTEROIDAL ANTI-INFLAMMATORY DRUGS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	1.750255707856483	DNA VACCINE	ncit:C39619	DNA VACCINE	FALSE	FALSE	FALSE
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	1.500219178162699	INTERLEUKINS	ncit:C593	RECOMBINANT INTERLEUKIN	FALSE	FALSE	FALSE
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	0.300043836	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.040112812	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.151537291	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.064944553	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
CORT	hgnc:2257	CORT	NCI	14-Sep-17	NULL	2.386712328895204	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
COL1A2	hgnc:2198	COL1A2	NCI	14-Sep-17	NULL	0.2991890098899971	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.031822831	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.037843367	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
CST3	hgnc:2475	CST3	NCI	14-Sep-17	NULL	1.029562181092049	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	1.750255707856483	NEUROTROPHIC FACTOR	ncit:C2259	RECOMBINANT NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	0.252440727	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.014683353	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.030430409	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
EPHA8	hgnc:3391	EPHA8	NCI	14-Sep-17	NULL	0.1392776425349986	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.3947945205691315	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.032899543	9-CIS-RETINOIC ACID	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
ERCC6	hgnc:3438	ERCC6	NCI	14-Sep-17	NULL	0.6563458904461812	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.1835932560688619	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.036013492	TAXOL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.021215221	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	2.100306849	INTERLEUKIN-1-BETA	ncit:C585	RECOMBINANT INTERLEUKIN-1-BETA	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.037398626	TYROSINE KINASE INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.028382525	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.2258394461750301	RETINOIC ACIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	1.050153425	CO-TRIMOXAZOLE	chembl:CHEMBL195591	CO-TRIMOXAZOLE	FALSE	FALSE	FALSE
FXN	hgnc:3951	FXN	NCI	14-Sep-17	NULL	0.6177373086552295	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.1553481397505754	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	OSM-S-31	chembl:CHEMBL1588237	CHEMBL:CHEMBL1588237	FALSE	FALSE	FALSE
GC	hgnc:4187	GC	NCI	14-Sep-17	NULL	0.6731752722524936	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.043109746	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	2.500365296937833	LUTEINIZING HORMONE	rxcui:6383	LUTEINIZING HORMONE	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.4861821410712453	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	CGI	2/1/22	NULL	1.831662950082366	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
HDC	hgnc:4855	HDC	NCI	14-Sep-17	NULL	0.7095631248066824	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	NCI	14-Sep-17	NULL	0.1103102336884338	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
HIST4H4	hgnc:20510	H4C16	NCI	14-Sep-17	NULL	2.625383561784725	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.2592971419046642	RHGH	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.6908904109959803	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
HMOX2	hgnc:5014	HMOX2	NCI	14-Sep-17	NULL	0.4773424657790409	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.030038714	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.030038714	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.1121958787087489	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
HYAL2	hgnc:5321	HYAL2	NCI	14-Sep-17	NULL	0.7955707762984016	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	0.4773424657790409	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
HYAL2	hgnc:5321	HYAL2	NCI	14-Sep-17	NULL	0.8751278539282418	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.2634164108814105	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.3889457128569963	SOMATOTROPIN	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.1495945049449985	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	1.312691780892362	MACROLIDE ANTIBIOTIC	ncit:C261	MACROLIDE ANTIBIOTIC	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.036013492	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.5357925636295356	ECHINACEA	rxcui:228041	ECHINACEA PREPARATION	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	1.29648571	RU 41740	ncit:C1018	KLEBSIELLA PNEUMONIAE GLYCOPROTEIN	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.2210849315187136	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.4688184931758437	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
MAGEA1	hgnc:6796	MAGEA1	NCI	14-Sep-17	NULL	6.300920548	5-AZA-2-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
MAGEA1	hgnc:6796	MAGEA1	NCI	14-Sep-17	NULL	6.300920548	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
MAGEA1	hgnc:6796	MAGEA1	NCI	14-Sep-17	NULL	0.6482428547616604	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:9448	iuphar.ligand:9448	CMF-019	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.384671584	GONADOTROPINS	ncit:C527	THERAPEUTIC GONADOTROPIN	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.1630673019742065	C5A	iuphar.ligand:3576	C5A	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.02926849	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.013299815	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.4773424657790409	TEMOZOLOMIDE	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.2273059360852575	IFOSFAMIDE	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	1.193356164447602	CCNU	rxcui:6466	LOMUSTINE	TRUE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.089756703	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	1.166837138570988	ANTICOAGULANT	ncit:C263	ANTICOAGULANT AGENT	FALSE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.086219493	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
MT2A	hgnc:7406	MT2A	NCI	14-Sep-17	NULL	1.009762908	PARACETAMOL	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
MT1H	hgnc:7400	MT1H	NCI	14-Sep-17	NULL	0.4412409347537353	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.5000730593875666	QUINAPRIL	rxcui:35208	QUINAPRIL	TRUE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:5961	iuphar.ligand:5961	DNA-PK INHIBITOR V	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.004061861	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.011110383	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.1902451856365742	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.1259176768242074	CYTOPROTECTIVE AGENT	ncit:C2080	CYTOPROTECTIVE AGENT	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.9460841664089098	DNCB	ncit:C439	DINITROCHLOROBENZENE	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	0.7955707762984013	COMPLETE FREUNDS ADJUVANT	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.2983390411119005	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	NCI	14-Sep-17	NULL	0.02357776	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.2375912725597036	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
OPLAH	hgnc:8149	OPLAH	NCI	14-Sep-17	NULL	5.000730593875666	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	0.2778183663264258	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.031273181	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
PHEX	hgnc:8918	PHEX	NCI	14-Sep-17	NULL	2.333674277141977	RHGH	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
PHEX	hgnc:8918	PHEX	NCI	14-Sep-17	NULL	4.039051633514961	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.009922085	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
PHEX	hgnc:8918	PHEX	NCI	14-Sep-17	NULL	2.917092846427472	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.039688338	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.027781837	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.073540156	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.053854022	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1154014752432845	IL-4	iuphar.ligand:4996	IL-4	FALSE	FALSE	FALSE
PLAT	hgnc:9051	PLAT	NCI	14-Sep-17	NULL	0.4546118721705151	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.037318885	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	NCI	14-Sep-17	NULL	0.014356164	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:9619	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
PRKD1	hgnc:9407	PRKD1	NCI	14-Sep-17	NULL	0.4039051633514962	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	ECHINACEA	rxcui:228041	ECHINACEA PREPARATION	TRUE	FALSE	FALSE
RIPK1	hgnc:10019	RIPK1	NCI	14-Sep-17	NULL	1.071585127259071	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
S100A2	hgnc:10492	S100A2	NCI	14-Sep-17	NULL	1.500219178	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.081281225	AZA	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.2397610558707511	Berzosertib	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
SCD	hgnc:10571	SCD	NCI	14-Sep-17	NULL	0.9376369863516875	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
SLC11A1	hgnc:10907	SLC11A1	NCI	14-Sep-17	NULL	9.546849315580818	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
SLC16A3	hgnc:10924	SLC16A3	NCI	14-Sep-17	NULL	2.282942227638891	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	NCI	14-Sep-17	NULL	0.021974334	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	MyCancerGenome	20-Jun-17	inhibitor	0.6000876712650799	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
SILV	hgnc:10880	PMEL	NCI	14-Sep-17	NULL	0.4487835148349957	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
SLC28A1	hgnc:11001	SLC28A1	NCI	14-Sep-17	NULL	4.200613698855561	THYMIDINE	rxcui:1372538	THYMIDINE	TRUE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	NCI	14-Sep-17	NULL	2.100306849	THYMIDINE	rxcui:1372538	THYMIDINE	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1905904582057876	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	PharmGKB	4/5/24	NULL	0.005445442	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1065064325267637	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1724389859957126	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
TAGLN	hgnc:11553	TAGLN	NCI	14-Sep-17	NULL	2.500365296937833	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
TERC	hgnc:11727	TERC	NCI	14-Sep-17	NULL	0.9723642821424907	AZIDOTHYMIDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.1004931506903244	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	NCI	14-Sep-17	NULL	0.600087671	HOMOHARRINGTONINE	rxcui:27100	OMACETAXINE MEPESUCCINATE	TRUE	FALSE	FALSE
TFAP2A	hgnc:11742	TFAP2A	NCI	14-Sep-17	NULL	0.3977853881492008	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.4234489615781814	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.1579178082276526	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.2991890098899971	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.1121958787087489	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
THY1	hgnc:11801	THY1	NCI	14-Sep-17	NULL	2.917092846427472	FCA	ncit:C2347	FREUND'S ADJUVANT	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.5770073762164232	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
TLR3	hgnc:11849	TLR3	NCI	14-Sep-17	NULL	1.500219178162699	IL-4	iuphar.ligand:4996	IL-4	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.051885051	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
THBS4	hgnc:11788	THBS4	NCI	14-Sep-17	NULL	4.039051633514962	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.5645986154375752	SODIUM CROMOGLYCATE	rxcui:3538	CROMOLYN SODIUM	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.112919723	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	1.129197231	IMMUNOSTIMULANT	ncit:C2139	IMMUNOSTIMULANT	FALSE	FALSE	FALSE
TNFRSF10A	hgnc:11904	TNFRSF10A	NCI	14-Sep-17	NULL	0.8078103267029924	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.406619897	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.025757994	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.057955487	TIRAPAZAMINE	ncit:C1464	TIRAPAZAMINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.012878997	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	0.2625383561784725	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
TYMP	hgnc:3148	TYMP	NCI	14-Sep-17	NULL	3.281729452230906	5-DEOXY-5-FLUOROURIDINE	ncit:C978	DOXIFLURIDINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	NCI	14-Sep-17	NULL	0.031919557	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.3271505995993426	Amitifadine	ncit:C169780	AMITIFADINE	FALSE	FALSE	FALSE
TSPO	hgnc:1158	TSPO	NCI	14-Sep-17	NULL	0.064268875	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
TYMP	hgnc:3148	TYMP	NCI	14-Sep-17	NULL	13.12691780892362	S-1	ncit:C1833	TEGAFUR-GIMERACIL-OTERACIL POTASSIUM	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.006370357	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.060028368	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.102191151	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.128537751	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	0.3547815624033412	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.2302968036653267	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
CHST3	hgnc:1971	CHST3	PharmGKB	4/5/24	NULL	1.419126249613364	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.2083637747448194	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	PharmGKB	4/5/24	NULL	3.938075342677087	imiquimod	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.030386384	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.095468493	ceftriaxone	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.081030357	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.060772768	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.3182283105193606	ceftriaxone	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
CDKL5	hgnc:11411	CDKL5	PharmGKB	4/5/24	NULL	2.917092846427472	ganaxolone	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.058733413	(S)-methadone	chembl:CHEMBL350719	ESMETHADONE	FALSE	FALSE	FALSE
TPH2	hgnc:20692	TPH2	PharmGKB	4/5/24	NULL	0.2035181055647073	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
SULT1A1	hgnc:11453	SULT1A1	PharmGKB	4/5/24	NULL	2.917092846427472	minoxidil	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
OTC	hgnc:8512	OTC	PharmGKB	4/5/24	NULL	2.917092846427472	glycerol phenylbutyrate	rxcui:1368451	GLYCEROL PHENYLBUTYRATE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.1973972602845657	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	1.166837138570989	rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.058083707	forskolin	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.008297672	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.024456298	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.011063563	hydrocortisone	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.010560674	topiramate	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.007148764	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.074797252	mefloquine	rxcui:6694	MEFLOQUINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.041508041	Analgesics	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.2500365296937833	Analgesics	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
ZDHHC3	hgnc:18470	ZDHHC3	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
TCF7L2	hgnc:11641	TCF7L2	PharmGKB	4/5/24	NULL	0.4828291607879953	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
DSE	hgnc:21144	DSE	PharmGKB	4/5/24	NULL	1.875273972703374	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.024416494	naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
RAPGEF5	hgnc:16862	RAPGEF5	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.1108536338543867	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.4487835148349957	atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	CancerCommons	25-Jul-13	inhibitor	0.1320947704042629	SB939	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
CYCSP5	hgnc:24416	CYCSP5	PharmGKB	4/5/24	NULL	0.7143900848393808	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.138178082	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.2403097081725148	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.086933231	zanubrutinib	rxcui:2262435	ZANUBRUTINIB	TRUE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	0.2763561643983921	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
CPS1	hgnc:2323	CPS1	PharmGKB	4/5/24	NULL	0.7501095890813501	sodium phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
CXCR2	hgnc:6027	CXCR2	PharmGKB	4/5/24	NULL	0.1458546423213736	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	0.2273059360852576	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.2625383561784725	3-aminopyridine-2-carboxaldehyde thiosemicarbazone	ncit:C2242	TRIAPINE	FALSE	FALSE	TRUE
PRKAG1	hgnc:9385	PRKAG1	PharmGKB	4/5/24	NULL	1.795134059339982	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	PharmGKB	4/5/24	NULL	0.025244073	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	PharmGKB	4/5/24	NULL	0.7955707762984013	odevixibat	rxcui:2563966	ODEVIXIBAT	TRUE	FALSE	FALSE
ACOT7	hgnc:24157	ACOT7	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ABCC9	hgnc:60	ABCC9	ChEMBL	33	potentiator	1.193356164447602	SARAKALIM	ncit:C72978	SARAKALIM	FALSE	FALSE	FALSE
LHX2	hgnc:6594	LHX2	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	PharmGKB	4/5/24	NULL	0.069225671	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ZNF613	hgnc:25827	ZNF613	PharmGKB	4/5/24	NULL	1.944728564284981	letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	0.4145342465975881	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.008854582	quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	4.449802647092754	cilazapril	rxcui:21102	CILAZAPRIL	TRUE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.1268301237577161	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	PharmGKB	4/5/24	NULL	0.2778183663264259	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
GRIK1	hgnc:4579	GRIK1	PharmGKB	4/5/24	NULL	1.432027397337122	topiramate	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.008345148	fosphenytoin	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
FSHR	hgnc:3969	FSHR	PharmGKB	4/5/24	NULL	18.37768493249307	urofollitropin	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.013622434	perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
SKOR2	hgnc:32695	SKOR2	PharmGKB	4/5/24	NULL	4.039051633514962	perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	2.333674277141977	voxilaprevir	rxcui:1939323	VOXILAPREVIR	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.031851787	medroxyprogesterone	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.5250767123569451	mirtazapine	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
SULT2A1	hgnc:11458	SULT2A1	PharmGKB	4/5/24	NULL	0.4039051633514962	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.023493365	dorzolamide	rxcui:60207	DORZOLAMIDE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.201952582	TG100-115	drugbank:DB05552	TG100-115	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	indinavir	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.01305187	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.014683353	dolasetron	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.0017798	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.1944728564284981	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.3500511415712967	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
NUP50	hgnc:8065	NUP50	PharmGKB	4/5/24	NULL	5.834185692854945	teniposide	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.092606122	ramucirumab	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
TOMM40	hgnc:18001	TOMM40	PharmGKB	4/5/24	NULL	3.889457128569963	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1429428436543407	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.290901226	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1973972602845657	methimazole	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1151484018326633	sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
DMD	hgnc:2928	DMD	PharmGKB	4/5/24	NULL	15.00219178	eteplirsen	rxcui:1810569	ETEPLIRSEN	TRUE	FALSE	FALSE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.1296485709523321	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	PharmGKB	4/5/24	NULL	0.007905401	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ARG1	hgnc:663	ARG1	PharmGKB	4/5/24	NULL	0.4167275494896388	glycerol phenylbutyrate	rxcui:1368451	GLYCEROL PHENYLBUTYRATE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.1495945049449985	probucol	rxcui:8699	PROBUCOL	TRUE	FALSE	FALSE
SCNN1A	hgnc:10599	SCNN1A	PharmGKB	4/5/24	NULL	2.470949234620918	amiloride	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.015892152	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
FOLH1	hgnc:3788	FOLH1	PharmGKB	4/5/24	NULL	0.069454592	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
FGG	hgnc:3694	FGG	PharmGKB	4/5/24	NULL	2.187819634820604	abciximab	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1995646288518794	1372540-25-4	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	PharmGKB	4/5/24	NULL	0.041085815	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
SPIDR	hgnc:28971	SPIDR	PharmGKB	4/5/24	NULL	0.9723642821424908	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
FGG	hgnc:3694	FGG	PharmGKB	4/5/24	NULL	2.625383561784725	tirofiban	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
MDM4	hgnc:6974	MDM4	PharmGKB	4/5/24	NULL	0.4861821410712454	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	1.179947668217853	drotrecogin alfa	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.326134604	sulfinpyrazone	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
ALDH2	hgnc:404	ALDH2	PharmGKB	4/5/24	NULL	0.2634164108814105	nitroglycerin	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
CES2	hgnc:1864	CES2	PharmGKB	4/5/24	NULL	0.2083637747448194	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
OAS1	hgnc:8086	OAS1	PharmGKB	4/5/24	NULL	1.207072901969988	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
PDGFRA	hgnc:8803	PDGFRA	PharmGKB	4/5/24	NULL	0.2869271652223742	mepolizumab	rxcui:1720597	MEPOLIZUMAB	TRUE	FALSE	FALSE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	0.300043836	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
PTGDR	hgnc:9591	PTGDR	PharmGKB	4/5/24	NULL	0.061055432	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	PharmGKB	4/5/24	NULL	0.065675636	interferons	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
CDH13	hgnc:1753	CDH13	PharmGKB	4/5/24	NULL	0.4251633298436801	amphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
SCAP	hgnc:30634	SCAP	PharmGKB	4/5/24	NULL	1.050153425	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.069180068	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
FCGR2A	hgnc:3616	FCGR2A	PharmGKB	4/5/24	NULL	0.1620607136904151	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.054243462	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	16.70698630226643	losigamone	ncit:C90707	LOSIGAMONE	FALSE	FALSE	FALSE
MVK	hgnc:7530	MVK	PharmGKB	4/5/24	NULL	8.751278539282415	alendronate	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.09741683	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SLC22A3	hgnc:10967	SLC22A3	PharmGKB	4/5/24	NULL	1.346350544504987	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.1293292394967845	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.065634589	sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
GC	hgnc:4187	GC	PharmGKB	4/5/24	NULL	0.2187819634820604	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
KLRK1	hgnc:18788	KLRK1	PharmGKB	4/5/24	NULL	0.8204323630577265	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
LPA	hgnc:6667	LPA	PharmGKB	4/5/24	NULL	2.187819634820604	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
PRDM16	hgnc:14000	PRDM16	PharmGKB	4/5/24	NULL	1.050153425	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
AGXT	hgnc:341	AGXT	PharmGKB	4/5/24	NULL	26.25383561784724	nedosiran	rxcui:2675287	NEDOSIRAN	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.082559232	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
TIGD1	hgnc:14523	TIGD1	PharmGKB	4/5/24	NULL	0.4861821410712453	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	0.4375639269641208	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	PharmGKB	4/5/24	NULL	0.729273212	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
UNIPROT:P00441	hgnc:11179	SOD1	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	ISIS-SOD1RX	chembl:CHEMBL3833346	TOFERSEN	FALSE	FALSE	FALSE
FOXA3	hgnc:5023	FOXA3	PharmGKB	4/5/24	NULL	0.729273212	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	1.875273972703375	l-arginine	rxcui:1091	ARGININE	TRUE	FALSE	FALSE
NPIPB8	hgnc:37490	NPIPB8	PharmGKB	4/5/24	NULL	1.009762908	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	0.1835932560688619	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.1187956362798518	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.024041974	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.3512218811752141	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	0.3739862623624964	cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
CHL1	hgnc:1939	CHL1	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.058341857	ethinyl estradiol	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.055622533	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.030292887	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.1172046232939609	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
OASL	hgnc:8090	OASL	PharmGKB	4/5/24	NULL	1.640864726115453	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
LIG3	hgnc:6600	LIG3	PharmGKB	4/5/24	NULL	0.4861821410712453	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.020164236	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	0.3818739726232327	primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
GAL	hgnc:4114	GAL	PharmGKB	4/5/24	NULL	1.640864726115453	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
GLCCI1	hgnc:18713	GLCCI1	PharmGKB	4/5/24	NULL	10.50153424713889	nedocromil	rxcui:31563	NEDOCROMIL	TRUE	FALSE	FALSE
DTYMK	hgnc:3061	DTYMK	PharmGKB	4/5/24	NULL	0.4861821410712453	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	2.100306849	sofosbuvir / velpatasvir / voxilaprevir	wikidata:Q48564241	SOFOSBUVIR / VELPATASVIR / VOXILAPREVIR	FALSE	FALSE	FALSE
PDZRN3	hgnc:17704	PDZRN3	PharmGKB	4/5/24	NULL	1.666910197958555	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.017525925	capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.039068208	MELEVODOPA	ncit:C83927	MELEVODOPA	TRUE	FALSE	FALSE
MIR23B	hgnc:31606	MIR23B	PharmGKB	4/5/24	NULL	26.25383561784724	acetaminophen / tramadol	wikidata:Q48564239	ACETAMINOPHEN/TRAMADOL	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.066676408	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.088665436	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.036237178	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.2206204673768676	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	PharmGKB	4/5/24	NULL	0.1660584163051692	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.3454452054979901	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.036770078	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	TALC	12-May-16	inhibitor	0.4526523382387456	PELITINIB	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	TALC	12-May-16	inhibitor	0.061340737	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	TALC	12-May-16	inhibitor	0.1124502911321247	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.1785975212098452	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.1785975212098452	FK-228	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.033207482	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ITGB5	hgnc:6160	ITGB5	TALC	12-May-16	NULL	7.876150685354174	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	0.9907107780319716	OSI906	hemonc:75494	LINSITINIB	FALSE	FALSE	TRUE
MAGEA3	hgnc:6801	MAGEA3	TALC	12-May-16	vaccine	35.00511415712966	ASTUPROTIMUT-R	ncit:C78478	ASTUPROTIMUT-R	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.5125748858722557	GSK1120212	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	TALC	12-May-16	inhibitor	0.1075976869583903	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.1312691780892362	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.094535416	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
RICTOR	hgnc:28611	RICTOR	TALC	12-May-16	inhibitor	0.1530835896084387	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIGF	hgnc:8962	PIGF	TALC	12-May-16	inhibitor	21.00306849	AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
RPS6	hgnc:10429	RPS6	TALC	12-May-16	inhibitor	0.4861821410712454	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
SGPP1	hgnc:17720	SGPP1	TALC	12-May-16	antibody	26.25383561784724	SONEPCIZUMAB	ncit:C78195	SONEPCIZUMAB	FALSE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	TALC	12-May-16	inhibitor	0.5527123287967842	AZD7762	iuphar.ligand:7713	AZD7762	FALSE	FALSE	TRUE
BIRC3	hgnc:591	BIRC3	TALC	12-May-16	inhibitor	0.3571950424196904	LCL161	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.49187514	LEVONORGESTREL	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TdgClinicalTrial	Jan-14	NULL	7.876150685354174	AZD-8848	drugbank:DB14868	AZD-8848	FALSE	FALSE	FALSE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	AVOSENTAN	ncit:C79485	AVOSENTAN	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	ChEMBL	33	inhibitor	0.089756703	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
UNIPROT:P33681	hgnc:1700	CD80	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	BELATACEPT	rxcui:1112973	BELATACEPT	TRUE	FALSE	FALSE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.8514757497680189	BINODENOSON	ncit:C174671	BINODENOSON	FALSE	FALSE	FALSE
UNIPROT:P17252	hgnc:9393	PRKCA	TdgClinicalTrial	Jan-14	NULL	0.1562728310586145	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:Q15139	hgnc:9407	PRKD1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:Q04759	hgnc:9410	PRKCQ	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:P05771	hgnc:9395	PRKCB	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	3.750547945	BRIAKINUMAB	ncit:C95321	BRIAKINUMAB	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.032899543	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	0.577007376	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
UNIPROT:Q14957	hgnc:4587	GRIN2C	TdgClinicalTrial	Jan-14	NULL	0.2419708351875322	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
UNIPROT:P68400	hgnc:2457	CSNK2A1	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	CX-4945	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.1013661606866689	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.2180551131050435	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.3271505995993426	DOV 21947	chembl:CHEMBL1818442	AMITIFADINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.1088116604009326	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:P00451	hgnc:3546	F8	TdgClinicalTrial	Jan-14	NULL	4.118248724368195	DROTRECOGIN ALFA	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P00790	hgnc:8885	PGA3	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	ECABET	ncit:C65504	ECABET	FALSE	FALSE	FALSE
UNIPROT:P11926	hgnc:8109	ODC1	TdgClinicalTrial	Jan-14	NULL	2.864054794674245	EFLORNITHINE	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TdgClinicalTrial	Jan-14	NULL	0.6035364509849942	DP-VPA	drugbank:DB05821	DP-VPA	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.2044691247495891	VENLAFAXINE	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1491695205559502	VENLAFAXINE	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
UNIPROT:P18405	hgnc:11284	SRD5A1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
UNIPROT:P12259	hgnc:3542	F5	TdgClinicalTrial	Jan-14	NULL	1.179947668217853	DROTRECOGIN ALFA	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.2430910705356227	TAMSULOSIN	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P20142	hgnc:8890	PGC	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	ECABET	ncit:C65504	ECABET	FALSE	FALSE	FALSE
UNIPROT:Q9P0X4	hgnc:1396	CACNA1I	TdgClinicalTrial	Jan-14	NULL	0.1000146118775133	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q15858	hgnc:10597	SCN9A	TdgClinicalTrial	Jan-14	NULL	0.050007306	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.047734247	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q9NY72	hgnc:20665	SCN3B	TdgClinicalTrial	Jan-14	NULL	2.100306849	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:P35499	hgnc:10591	SCN4A	TdgClinicalTrial	Jan-14	NULL	0.064624826	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	1.381780822	EP217609	drugbank:DB18393	EP-217609	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.1151484018326633	GGF-2	chembl:CHEMBL3039542	CIMAGLERMIN ALFA	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.05309168	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	0.729273212	GLPG0187	ncit:C96223	INTEGRIN RECEPTOR ANTAGONIST GLPG0187	FALSE	FALSE	FALSE
UNIPROT:P06756	hgnc:6150	ITGAV	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	GLPG0187	ncit:C96223	INTEGRIN RECEPTOR ANTAGONIST GLPG0187	FALSE	FALSE	FALSE
UNIPROT:P37088	hgnc:10599	SCNN1A	TdgClinicalTrial	Jan-14	NULL	2.470949234620918	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.064505739	Succinylcholine	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.068436196	ADALIMUMAB	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.3081436105381133	IMC-1121B	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
UNIPROT:P06213	hgnc:6091	INSR	TdgClinicalTrial	Jan-14	NULL	1.500219178	INSULIN GLARGINE	rxcui:2563969	INSULIN GLARGINE-YFGN	TRUE	FALSE	FALSE
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TdgClinicalTrial	Jan-14	NULL	3.938075342677087	IMIQUIMOD	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	1.357957014716237	INNO-206	ncit:C68921	ALDOXORUBICIN	FALSE	FALSE	FALSE
UNIPROT:Q6UUV9	hgnc:16062	CRTC1	TdgClinicalTrial	Jan-14	NULL	0.5966780822238011	INK128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
OSGEP	hgnc:18028	OSGEP	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.111481255	INECALCITOL	ncit:C83818	INECALCITOL	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.42006137	AMG-131	drugbank:DB05490	AMG-131	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.1535312024435511	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
UNIPROT:P18031	hgnc:9642	PTPN1	TdgClinicalTrial	Jan-14	NULL	2.100306849	ISIS 113715	drugbank:DB05506	ISIS 113715	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	FDA	10-Apr-24	NULL	0.6250913242344582	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
UNIPROT:P01589	hgnc:6008	IL2RA	TdgClinicalTrial	Jan-14	NULL	0.1715936968486748	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.1495945049449985	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.157680694	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.2163777660811586	ITI-007	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	LESOGABERAN	ncit:C166751	LESOGABERAN	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.030814361	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.1052961321571413	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
GUANYLATE CYCLASE	hgnc:4187	GC	TTD	2020.06.01	NULL	0.3977853881492008	Isosorbide Dinitrate	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
UNIPROT:Q96LZ3	hgnc:9318	PPP3R2	TdgClinicalTrial	Jan-14	NULL	1.207072901969988	CYCLOSPORINE A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.1767935058440892	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
UNIPROT:P31639	hgnc:11037	SLC5A2	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	LX4211	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.088945801	OPC-34712	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:O00329	hgnc:8977	PIK3CD	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	RIGOSERTIB	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.8607814956671229	PROGESTOGEN	wikidata:Q45071	PROGESTOGEN	TRUE	FALSE	FALSE
UNIPROT:P40763	hgnc:11364	STAT3	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	OPB-51602	ncit:C95889	STAT3 INHIBITOR OPB-51602	FALSE	FALSE	FALSE
UNIPROT:Q15858	hgnc:10597	SCN9A	TdgClinicalTrial	Jan-14	NULL	0.078136416	RANOLAZINE	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
UNIPROT:P15121	hgnc:381	AKR1B1	TdgClinicalTrial	Jan-14	NULL	8.078103267029922	RANIRESTAT	ncit:C96307	RANIRESTAT	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1666910197958555	ROPINIROL	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1640864726115453	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
UNIPROT:P00451	hgnc:3546	F8	TdgClinicalTrial	Jan-14	NULL	3.088686543276147	RECOMBINANT FACTOR VIIA	wikidata:Q5940878	RECOMBINANT FACTOR VIIA	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.3431873936973497	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	0.3025133322221082	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:Q06124	hgnc:9644	PTPN11	TdgClinicalTrial	Jan-14	NULL	7.501095891	STIBOGLUCONATE	chembl:CHEMBL2068504	STIBOGLUCONATE	FALSE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.9546849315580818	TASPOGLUTIDE	ncit:C152518	TASPOGLUTIDE	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.2536602475154323	TAMSULOSIN	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	ISOEUGENITOL	chembl:CHEMBL1371435	ISOEUGENITOL	FALSE	FALSE	FALSE
UNIPROT:P48039	hgnc:7463	MTNR1A	TdgClinicalTrial	Jan-14	NULL	5.625821918110125	TASIMELTEON	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.016501468	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.3319450480417468	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
UNIPROT:P49763	hgnc:8893	PGF	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	TB-403	chembl:CHEMBL2109545	TB-403	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	0.5834185692854944	ABITUZUMAB	ncit:C82422	ABITUZUMAB	FALSE	FALSE	FALSE
UNIPROT:P49286	hgnc:7464	MTNR1B	TdgClinicalTrial	Jan-14	NULL	7.876150685354174	TASIMELTEON	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
UNIPROT:P49840	hgnc:4616	GSK3A	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	TIDEGLUSIB	ncit:C97364	TIDEGLUSIB	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.092118721	TIOTROPIUM	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
UNIPROT:Q16478	hgnc:4583	GRIK5	TdgClinicalTrial	Jan-14	NULL	1.166837138570989	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	ChEMBL	33	inhibitor	1.166837138570988	ELIMUSERTIB	ncit:C146807	ELIMUSERTIB	FALSE	FALSE	TRUE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.077217164	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P16410	hgnc:2505	CTLA4	TdgClinicalTrial	Jan-14	NULL	0.9723642821424907	TREMELIMUMAB	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.1419126249613365	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	TRANEXAMIC ACID	rxcui:10691	TRANEXAMIC ACID	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.073540156	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	ACEPROMETAZINE	rxcui:161203	ACEPROMETAZINE	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.080225625	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.07182992	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1583941817064691	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.070197421	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.1228249619548409	AMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
CCND2	hgnc:1583	CCND2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.5834185692854945	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:O14920	hgnc:5960	IKBKB	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	AURANOFIN	rxcui:1227	AURANOFIN	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.6105543166941221	APRACLONIDINE	rxcui:14845	APRACLONIDINE	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.2344092465879218	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TdgClinicalTrial	Jan-14	NULL	1.514644363	BRINZOLAMIDE	rxcui:194881	BRINZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TdgClinicalTrial	Jan-14	NULL	3.750547945	CARBOPROST TROMETHAMINE	rxcui:20259	CARBOPROST TROMETHAMINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.4817217544559128	DIPHENOXYLATE	rxcui:3500	DIPHENOXYLATE	TRUE	FALSE	FALSE
NOTCH4	hgnc:7884	NOTCH4	MyCancerGenome	20-Jun-17	other/unknown	1.750255707856483	REGN421	ncit:C82367	ENOTICUMAB	FALSE	FALSE	TRUE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.406619897	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.024416494	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
UNIPROT:Q16647	hgnc:9603	PTGIS	TdgClinicalTrial	Jan-14	NULL	7.501095890813499	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	RHODOMYRTOXIN B	chembl:CHEMBL1552997	RHODOMYRTOXIN B	FALSE	FALSE	FALSE
UNIPROT:Q8TCC7	hgnc:10972	SLC22A8	TdgClinicalTrial	Jan-14	NULL	2.045753424767318	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.3182283105193605	SALICYLIC ACID	rxcui:9525	SALICYLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	2.669881588255652	SAPRISARTAN	ncit:C152297	SAPRISARTAN	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.1603287671318916	RIMEXOLONE	rxcui:55681	RIMEXOLONE	TRUE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.036718651	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	SALSALATE	rxcui:36108	SALSALATE	TRUE	FALSE	FALSE
UNIPROT:P00797	hgnc:9958	REN	TdgClinicalTrial	Jan-14	NULL	15.75230137070834	REMIKIREN	ncit:C73099	REMIKIREN	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2094720926955897	SCOPOLAMINE	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	1.154014752432846	RIZATRIPTAN	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
SIRT3	hgnc:14931	SIRT3	DTC	9/2/20	NULL	26.25383561784724	4-METHYLNICOTINAMIDE	chembl:CHEMBL1501622	CHEMBL:CHEMBL1501622	FALSE	FALSE	FALSE
UNIPROT:P03886	hgnc:7455	MT-ND1	TdgClinicalTrial	Jan-14	NULL	0.2838252499226729	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.093763699	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.4565884455277783	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.096050618	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.081281225	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TEND	1-Aug-11	NULL	1.312691780892362	DEMECARIUM BROMIDE	rxcui:22482	DEMECARIUM BROMIDE	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	2.128689374420047	ORG-13011	rxcui:2672253	GEPIRONE	TRUE	FALSE	FALSE
UNIPROT:P10696	hgnc:441	ALPG	TEND	1-Aug-11	NULL	0.6177373086552295	AMIFOSTINE	rxcui:1545987	AMIFOSTINE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P07327	hgnc:249	ADH1A	TEND	1-Aug-11	NULL	3.281729452230906	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
UNIPROT:O95180	hgnc:1395	CACNA1H	TEND	1-Aug-11	NULL	0.4440395030502706	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
NCBIGENE:85	ncbigene:85	ACTL5	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:12665	iuphar.ligand:12665	EXAMPLE 494 [WO2014028479] PARENT MOLECULE	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.052648066	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q9P0X4	hgnc:1396	CACNA1I	TEND	1-Aug-11	NULL	0.4546118721705151	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.056500364	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.050912416	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1187956362798518	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.031929262	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:9469	iuphar.ligand:9469	MRS4162-BODIPY CONJUGATE	FALSE	FALSE	FALSE
UNIPROT:P13688	hgnc:1814	CEACAM1	TEND	1-Aug-11	NULL	8.751278539282415	ARCITUMOMAB	ncit:C1494	ARCITUMOMAB	TRUE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5292	iuphar.ligand:5292	YM976	FALSE	FALSE	FALSE
UNIPROT:P02458	hgnc:2200	COL2A1	TEND	1-Aug-11	NULL	1.875273972703375	COLLAGENASE	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
NCBIGENE:1584	hgnc:2591	CYP11B1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8554	iuphar.ligand:8554	COMPOUND 35 [PMID: 24157366]	FALSE	FALSE	FALSE
UNIPROT:O14646	hgnc:1915	CHD1	TEND	1-Aug-11	NULL	2.917092846427472	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1642918374083057	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P62158	hgnc:1442	CALM1	TEND	1-Aug-11	NULL	0.729273212	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2094720926955897	BIPERIDEN	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.6250913242344582	BIPERIDEN	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TEND	1-Aug-11	NULL	1.514644363	BRINZOLAMIDE	rxcui:194881	BRINZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.055155117	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	1.848379561100067	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.077789143	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.011940798	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.008458066	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	AZINPHOS-ETHYL	ncit:C163587	AZINPHOS-ETHYL	FALSE	FALSE	FALSE
UNIPROT:P00492	hgnc:5157	HPRT1	TEND	1-Aug-11	NULL	0.5834185692854944	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.1840222122746302	DESVENLAFAXINE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1226814748497534	DESOGESTREL	rxcui:22656	DESOGESTREL	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.079718124	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TEND	1-Aug-11	NULL	0.6250913242344583	INTERFERON ALFA-2B, RECOMBINANT	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.2812910959055062	KETOPROFEN	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.089501712	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	1.050153425	METHAZOLAMIDE	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.096050618	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.104285345	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	3.750547945	METHYCLOTHIAZIDE	rxcui:6860	METHYCLOTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.072125922	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	0.2734774543525755	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
UNIPROT:P07949	hgnc:9967	RET	TEND	1-Aug-11	NULL	0.034572952	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P20648	hgnc:819	ATP4A	TEND	1-Aug-11	NULL	0.4375639269641208	PANTOPRAZOLE	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.092988792	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.546954909	PHENYLPROPANOLAMINE	rxcui:8175	PHENYLPROPANOLAMINE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	DELAVIRDINE MESYLATE	rxcui:142152	DELAVIRDINE MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.2470949234620917	PRAMIPEXOLE	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1245241215075758	PRAMIPEXOLE	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.024416494	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	0.4412409347537352	RIVASTIGMINE	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.3182283105193605	SALICYLIC ACID	rxcui:9525	SALICYLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.101562227	SUCCINYLCHOLINE	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TEND	1-Aug-11	NULL	3.938075342677087	IMIQUIMOD	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:5290	iuphar.ligand:5290	Y27632	FALSE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TEND	1-Aug-11	NULL	1.060761035064535	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	0.3236220106976548	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
UNIPROT:P00439	hgnc:8582	PAH	TEND	1-Aug-11	NULL	3.500511415712967	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.023612219	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
UNIPROT:P17752	hgnc:12008	TPH1	TEND	1-Aug-11	NULL	2.625383561784725	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:P30531	hgnc:11042	SLC6A1	TEND	1-Aug-11	NULL	14.00204566285186	TIAGABINE	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	4-METHYLDAPHNETIN	chembl:CHEMBL276618	4-METHYLDAPHNETIN	FALSE	FALSE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TEND	1-Aug-11	NULL	0.4023576339899961	TIAGABINE	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.016156207	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
UNIPROT:P37088	hgnc:10599	SCNN1A	TEND	1-Aug-11	NULL	2.917092846427472	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
UNIPROT:P51172	hgnc:10601	SCNN1D	TEND	1-Aug-11	NULL	1.944728564284981	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
TEK	hgnc:11724	TEK	DTC	9/2/20	NULL	1.312691780892362	GW559768X	chembl:CHEMBL237347	GW559768X	FALSE	FALSE	FALSE
UNIPROT:Q16881	hgnc:12437	TXNRD1	TEND	1-Aug-11	NULL	1.009762908	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	1.875273972703375	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:Q16739	hgnc:12524	UGCG	TEND	1-Aug-11	NULL	7.001022831425932	MIGLUSTAT	rxcui:402316	MIGLUSTAT	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.2154897588332195	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TEND	1-Aug-11	NULL	0.1305078821102597	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:8983	iuphar.ligand:8983	ST-1006	FALSE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TEND	1-Aug-11	NULL	0.3512218811752141	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TEND	1-Aug-11	NULL	0.6035364509849942	VIGABATRIN	rxcui:14851	VIGABATRIN	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TEND	1-Aug-11	NULL	0.3671865121377238	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2222	iuphar.ligand:2222	D(CH2)5[TYR(ME)2,THR4]OVT	FALSE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TEND	1-Aug-11	NULL	0.6364566210387212	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
PLACENTA GROWTH FACTOR	hgnc:8893	PGF	TTD	2020.06.01	NULL	52.50767123569449	RO-5323441	chembl:CHEMBL2109545	TB-403	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.2187819634820604	CRLX101	ncit:C62600	DAVAMOTECAN PEGADEXAMER	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.2470949234620917	M7824	ncit:C124229	BINTRAFUSP ALFA	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	2.059124362184098	CDX-3379	chembl:CHEMBL4650292	CDX-3379	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005294179	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.6177373086552294	FAZ053	ncit:C131537	ANTI-PD-L1 MONOCLONAL ANTIBODY FAZ053	FALSE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	5.250767123569449	JNJ-63709178	ncit:C128486	ANTI-CD123/CD3 BISPECIFIC ANTIBODY JNJ-63709178	FALSE	FALSE	FALSE
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	2.386712328895204	VX-15	chembl:CHEMBL4297884	PEPINEMAB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.5048814541893701	Navicixizumab	ncit:C119620	NAVICIXIZUMAB	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.9723642821424906	RG7828	rxcui:2625122	MOSUNETUZUMAB	TRUE	FALSE	FALSE
TANK	hgnc:11562	TANK	PharmGKB	4/5/24	NULL	3.182283105193606	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
PHOSPHODIESTERASE I BETA	hgnc:3358	ENPP3	TTD	2020.06.01	NULL	3.281729452230906	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1852122442176172	MM-151	iuphar.ligand:9125	MM-151	FALSE	TRUE	TRUE
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	17.50255707856483	JNJ-54175446	drugbank:DB15358	JNJ-54175446	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.092443083	PF-04449913	rxcui:2105845	GLASDEGIB	TRUE	FALSE	TRUE
RETINOIC ACID-INDUCIBLE GENE-1	hgnc:19102	RIGI	TTD	2020.06.01	NULL	26.25383561784724	SB-9200	chembl:CHEMBL1076930	INARIGIVIR SOPROXIL	FALSE	FALSE	FALSE
UGT2B17	hgnc:12547	UGT2B17	PharmGKB	4/5/24	NULL	2.625383561784725	belzutifan	rxcui:2567226	BELZUTIFAN	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.175415383	APC-100	chembl:CHEMBL37676	APC-100	FALSE	FALSE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	0.3750547945406749	Interferon alpha-2b	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	0.2885036881082116	Fenretinide	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
BETA-MICROSEMINOPROTEIN	hgnc:7372	MSMB	TTD	2020.06.01	NULL	52.50767123569449	Tigapotide	ncit:C78474	TIGAPOTIDE	FALSE	FALSE	FALSE
OPIOID RECEPTOR ZETA	hgnc:15768	OGFR	TTD	2020.06.01	NULL	52.50767123569449	INNO-105	chembl:CHEMBL2108291	METENKEFALIN	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.056581542	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	2.917092846427472	EC0489	ncit:C81935	FOLATE RECEPTOR-TARGETED VINCA ALKALOID EC0489	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	0.2749092734853114	ARQ 736	chembl:CHEMBL3545296	ARQ-736	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.2430910705356226	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
DNA-BINDING FACTOR KBF1	hgnc:14372	SCYL1	TTD	2020.06.01	NULL	26.25383561784724	CAT 1004	chembl:CHEMBL3786673	EDASALONEXENT	FALSE	FALSE	FALSE
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	0.8078103267029924	Rontalizumab	ncit:C95794	RONTALIZUMAB	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	13.12691780892362	Dabelotine	ncit:C74103	DABELOTINE	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.041739007	Treximet	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	1.009762908	BLZ-945	drugbank:DB16838	BLZ-945	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	NCI	14-Sep-17	NULL	0.005332352	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.5834185692854944	HT-0712	drugbank:DB11650	HT-0712	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	0.5000730593875667	RM-493	iuphar.ligand:9272	SETMELANOTIDE	FALSE	FALSE	FALSE
THYROTROPIN-RELEASING HORMONE	hgnc:12298	TRH	TTD	2020.06.01	NULL	10.50153424713889	KPS-0373	chembl:CHEMBL4297622	ROVATIRELIN	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	2.917092846427472	AZD-5122	chembl:CHEMBL5095219	AZD-5122	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	LY-255283	chembl:CHEMBL15766	LY-255283	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.087222045	LY2874455	iuphar.ligand:8104	LY2874455	FALSE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	1.458546423213736	PF-05190457	iuphar.ligand:9060	PF-05190457	FALSE	FALSE	FALSE
PALMITOYL-PROTEIN THIOESTERASE 1	hgnc:9325	PPT1	TTD	2020.06.01	NULL	26.25383561784724	Plitidepsin	ncit:C1689	PLITIDEPSIN	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:5655	iuphar.ligand:5655	A-674563	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	1.514644363	RG7221	ncit:C118578	VANUCIZUMAB	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.010923169	Olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
AROMATIC-L-AMINO-ACID DECARBOXYLASE	hgnc:2719	DDC	TTD	2020.06.01	NULL	3.000438356325399	Benserazide	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.5357925636295356	SR-123781A	drugbank:DB05361	SR-123781A	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 EPSILON	hgnc:1674	CD3E	TTD	2020.06.01	NULL	0.8334550989792776	Muromonab	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
B2 BRADYKININ RECEPTOR	hgnc:1030	BDKRB2	TTD	2020.06.01	NULL	1.093909817410302	DELTIBANT	ncit:C166885	DELTIBANT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.010417155	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.009745299	Prasterone	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	1.029562181092048	Desmopressin	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 1	hgnc:6026	CXCR1	TTD	2020.06.01	NULL	0.192335792	Ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	0.5000730593875667	CYTISINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
FATTY ACID SYNTHASE	hgnc:3594	FASN	TTD	2020.06.01	NULL	0.1143957978991165	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.028536778	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.071585127259071	BIBT986	chembl:CHEMBL1270156	TANOGITRAN	FALSE	FALSE	FALSE
PURINE NUCLEOSIDE PHOSPHORYLASE	hgnc:7892	PNP	TTD	2020.06.01	NULL	8.751278539282415	Guanosine	rxcui:1591890	GUANOSINE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.6250913242344582	ARZOXIFENE	ncit:C1805	ARZOXIFENE	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.8514757497680189	Binodenoson	ncit:C174671	BINODENOSON	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 29 MEMBER 1	hgnc:11003	SLC29A1	TTD	2020.06.01	NULL	0.1779921058837101	LIDOFLAZINE	rxcui:6390	LIDOFLAZINE	FALSE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	1.250182648468916	Tranexamic Acid	rxcui:10691	TRANEXAMIC ACID	TRUE	FALSE	FALSE
VITAMIN K EPOXIDE REDUCTASE COMPLEX 1	hgnc:23663	VKORC1	TTD	2020.06.01	NULL	0.6364566210387212	Warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	0.364636606	Meprobamate	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	0.5147810905460244	Naratriptan	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
FOLLICLE-STIMULATING HORMONE RECEPTOR	hgnc:3969	FSHR	TTD	2020.06.01	NULL	18.37768493249307	Follitropin beta	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	0.6863747873946993	Rilonacept	rxcui:763450	RILONACEPT	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.018867291	Phenoxybenzamine	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.033207482	R763	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.04525223	R763	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	10.50153424713889	RGI-2001	ncit:C163753	LIPOSOMAL ALPHA GALACTOSYLCERAMIDE	FALSE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	3.281729452230906	ATF-936	chembl:CHEMBL597800	ATF-936	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	2.561349816375341	XEN-D0501	drugbank:DB18673	XEN-D0501	FALSE	FALSE	FALSE
MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN	hgnc:7467	MTTP	TTD	2020.06.01	NULL	13.12691780892362	SLx-4090	drugbank:DB05678	SLX-4090	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	1.193356164447602	RX-3117	ncit:C113444	RODUCITABINE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	Terbutaline	rxcui:10368	TERBUTALINE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.3977853881492006	GSK-356278	drugbank:DB12542	GSK-356278	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.3025133322221082	PF-05280586	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	10.74020548002842	VX-661	rxcui:1999382	TEZACAFTOR	TRUE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	3.500511415712966	OPB-51602	ncit:C95889	STAT3 INHIBITOR OPB-51602	FALSE	FALSE	FALSE
PROTEIN KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	2.187819634820604	RV-568	chembl:CHEMBL3695568	JNJ-49095397	FALSE	FALSE	FALSE
CERAMIDE GLUCOSYLTRANSFERASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	10.50153424713889	Eliglustat tartrate	rxcui:1547219	ELIGLUSTAT TARTRATE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	0.750109589	GS-9973	ncit:C105402	ENTOSPLETINIB	FALSE	FALSE	FALSE
FREE FATTY ACID RECEPTOR 1	hgnc:4498	FFAR1	TTD	2020.06.01	NULL	3.750547945	TAK-875	ncit:C132780	FASIGLIFAM	FALSE	FALSE	FALSE
SCLEROSTIN	hgnc:13771	SOST	TTD	2020.06.01	NULL	13.12691780892362	Romosozumab	rxcui:2123126	ROMOSOZUMAB	TRUE	FALSE	FALSE
TISSUE FACTOR	hgnc:3541	F3	TTD	2020.06.01	NULL	3.500511415712966	ALT-836	ncit:C96430	ANTI-TF MONOCLONAL ANTIBODY ALT-836	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	7.001022831425932	PF-04937319	drugbank:DB15009	PF-04937319	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	1.237091730683901	BGB-283	ncit:C124995	LIFIRAFENIB	FALSE	FALSE	FALSE
EUKARYOTIC ELONGATION FACTOR 2 KINASE	hgnc:24615	EEF2K	TTD	2020.06.01	NULL	1.693795846312725	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	2.763561643983921	ONO-2952	drugbank:DB14802	ONO-2952	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.083016081	Cariprazine	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	1.193356164447602	ABBV-2222	chembl:CHEMBL4101487	GALICAFTOR	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.042073455	TRYPTAMINE	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.1131630845596864	Pefloxacin	rxcui:7960	PEFLOXACIN	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.8468979231563628	Phenindamine	rxcui:33283	PHENINDAMINE	TRUE	FALSE	FALSE
ILEAL SODIUM/BILE ACID COTRANSPORTER	hgnc:10906	SLC10A2	TTD	2020.06.01	NULL	2.019525817	Taurocholic Acid	drugbank:DB04348	TAUROCHOLIC ACID	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP3	hgnc:9595	PTGER3	TTD	2020.06.01	NULL	1.944728564284981	16,16-dimethyl-PGE2	iuphar.ligand:1926	16,16-DIMETHYL-PGE2	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.2456499239096818	Ondansetron	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.252440727	Squalamine	ncit:C143004	SQUALAMINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.013631275	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
CILIARY NEUROTROPHIC FACTOR RECEPTOR ALPHA	hgnc:2170	CNTFR	TTD	2020.06.01	NULL	10.50153424713889	NT-501	drugbank:DB05344	CILIARY NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
DUFFY ANTIGEN CHEMOKINE RECEPTOR	hgnc:4035	ACKR1	TTD	2020.06.01	NULL	26.25383561784724	AQ-13	drugbank:DB17749	AQ-13	FALSE	FALSE	FALSE
GASTRIC H(+)/K(+) ATPASE ALPHA	hgnc:819	ATP4A	TTD	2020.06.01	NULL	0.201178817	Dexlansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE	hgnc:1530	MICU1	TTD	2020.06.01	NULL	6.563458904461812	PF-4427429	rxcui:2056691	FREMANEZUMAB	TRUE	FALSE	FALSE
NOCICEPTIN RECEPTOR	hgnc:8155	OPRL1	TTD	2020.06.01	NULL	6.563458904461812	SER-100	drugbank:DB16013	SER-100	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	CART-BCMA	ncit:C156272	AUTOLOGOUS ANTI-BCMA-CAR-TCRZ/4-1BB-EXPRESSING T-LYMPHOCYTES CART-BCMA	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.062645859	Estradiol Valerate	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.038173516	Hydrocortisone	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.4039051633514962	ISOSORBIDE MONONITRATE	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	4.375639269641208	Insulin Susp Protamine Zinc Beef/Pork	chembl:CHEMBL1201628	INSULIN SUSP PROTAMINE ZINC BEEF/PORK	TRUE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	0.2715914029432474	Glibenclamide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA 1	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	0.3814116554650932	Pirfenidone	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.05593857	Nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	0.1810609352954982	Peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	1.381780822	XL844	drugbank:DB05149	XL844	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	ICARITIN	drugbank:DB12672	ICARITIN	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	2.072671233	AMG 853	ncit:C152874	VIDUPIPRANT	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	Sarizotan	ncit:C77567	SARIZOTAN	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	2.838252499226729	LY-2584702	drugbank:DB12690	LY-2584702	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	1.050153425	MGD007	ncit:C118442	ANTI-GPA33/CD3 MONOCLONAL ANTIBODY MGD007	FALSE	FALSE	FALSE
CELL SURFACE A33 ANTIGEN	hgnc:4445	GPA33	TTD	2020.06.01	NULL	6.563458904461812	MGD007	ncit:C118442	ANTI-GPA33/CD3 MONOCLONAL ANTIBODY MGD007	FALSE	FALSE	FALSE
COLLAGEN	hgnc:633	AQP1	TTD	2020.06.01	NULL	0.049349315	Collagenase	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.2419708351875322	Cetirizine	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.1411496538593938	Hydroxyzine	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1221108633388244	Hexobarbital	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
THYROID HORMONE RECEPTOR ALPHA	hgnc:11796	THRA	TTD	2020.06.01	NULL	0.9092237443410304	Liothyronine	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.081281225	Methysergide	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1A	hgnc:7463	MTNR1A	TTD	2020.06.01	NULL	1.034633915974276	Melatonin	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.02726255	Mitotane	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	10.50153424713889	Pegvisomant	rxcui:278739	PEGVISOMANT	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.068115956	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	0.6035364509849942	Vigabatrin	rxcui:14851	VIGABATRIN	TRUE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	AMG 330	ncit:C123332	ELUVIXTAMAB	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.092606122	Sym013	ncit:C131175	ANTI-EGFR/HER2/HER3 MONOCLONAL ANTIBODY MIXTURE SYM013	FALSE	FALSE	FALSE
NICOTINIC ACID RECEPTOR	hgnc:24827	HCAR2	TTD	2020.06.01	NULL	4.375639269641208	GSK-256073	iuphar.ligand:8470	GSK256073	FALSE	FALSE	FALSE
CYTIDINE DEAMINASE	hgnc:1712	CDA	TTD	2020.06.01	NULL	11.25164383622025	Tetrahydrouridine	ncit:C868	TETRAHYDROURIDINE	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3319450480417468	Tanespimycin	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	4.039051633514961	TD-5108	ncit:C84238	VELUSETRAG	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	4.565884455277782	Resatorvid	ncit:C87682	RESATORVID	FALSE	FALSE	FALSE
NCBIGENE:1388	hgnc:2349	ATF6B	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11390	iuphar.ligand:11390	PD-146176	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.9907107780319716	M-carboxycinnamic acid bishydroxamide	ncit:C1797	CARBOXYCINNAMIC ACID BISHYDROXAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1519	hgnc:2542	CTSO	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:8007	iuphar.ligand:8007	BX-912	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:3924	iuphar.ligand:3924	NLX-101	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.075442056	IUPHAR.LIGAND:12	iuphar.ligand:12	EMDT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:8	iuphar.ligand:8	BMY-14802	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:68	iuphar.ligand:68	P-MPPI	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:66	iuphar.ligand:66	(S)-FLUROCARAZOLOL	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:76	iuphar.ligand:76	SB 649915	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.079077818	IUPHAR.LIGAND:109	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.078136416	IUPHAR.LIGAND:109	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:10446	ncit:C79719	AVITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:28	iuphar.ligand:28	SB 216641	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.034727296	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:129	iuphar.ligand:129	S33084	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:147	iuphar.ligand:147	DOI	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:210	ncit:C73158	SARPOGRELATE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:129	iuphar.ligand:129	S33084	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.021933029	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.016027983	IUPHAR.LIGAND:209	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:195	iuphar.ligand:195	SDZ SER-082	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:163	ncit:C80757	BROLAMFETAMINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.039479452	IUPHAR.LIGAND:189	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:175	iuphar.ligand:175	SPIRAMIDE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.029090123	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.042898424	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:163	ncit:C80757	BROLAMFETAMINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.276356164	IUPHAR.LIGAND:232	iuphar.ligand:232	[3H]MESULERGINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:166	iuphar.ligand:166	RO 60-0175	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.032173818	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.064347636	IUPHAR.LIGAND:168	iuphar.ligand:168	VER-3323	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.014849455	IUPHAR.LIGAND:202	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.077217164	IUPHAR.LIGAND:190	iuphar.ligand:190	SB 215505	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:242	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:276	iuphar.ligand:276	SB 271046	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.068458502	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:6693	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:6599	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.031479419	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9810	iuphar.ligand:9810	COMPOUND 2F [JIANG ET AL., 2018]	FALSE	FALSE	FALSE
NCBIGENE:1673	hgnc:2767	DEFB4A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8679	iuphar.ligand:8679	INCB3619	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.052142673	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.030959712	IUPHAR.LIGAND:2404	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:486	iuphar.ligand:486	(+)-CYCLAZOSIN	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.082559232	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:373	iuphar.ligand:373	2-HEXYNYL-NECA	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.201178817	IUPHAR.LIGAND:369	iuphar.ligand:369	(R,S)-PHPNECA	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:3289	iuphar.ligand:3289	BAY 60-6583	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.063110182	IUPHAR.LIGAND:414	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:5618	iuphar.ligand:5618	KF26777	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:404	iuphar.ligand:404	XANTHINE AMINE CONGENER	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:5613	iuphar.ligand:5613	ST-1535	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:474	iuphar.ligand:474	MRS1523	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.5413161983061289	IUPHAR.LIGAND:5600	iuphar.ligand:5600	2-PHENYLETHYLYL-ADENOSINE DERIVATIVE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:5618	iuphar.ligand:5618	KF26777	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:449	iuphar.ligand:449	MRS1754	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5613	iuphar.ligand:5613	ST-1535	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:5728	iuphar.ligand:3284	PSB603	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1136529680426287	IUPHAR.LIGAND:404	iuphar.ligand:404	XANTHINE AMINE CONGENER	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.077330885	IUPHAR.LIGAND:375	iuphar.ligand:375	CGS 21680	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:6894	iuphar.ligand:6894	ANGIOTENSIN A	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.050294704	IUPHAR.LIGAND:5696	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:8008	iuphar.ligand:8008	GSK2334470	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.081281225	IUPHAR.LIGAND:8353	iuphar.ligand:8353	ZM447439	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:8061	iuphar.ligand:8061	MK-5108	FALSE	FALSE	FALSE
NCBIGENE:2901	hgnc:4583	GRIK5	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11590	iuphar.ligand:11590	BIO-32546	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10478	ncit:C121854	BEMCENTINIB	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.064347636	IUPHAR.LIGAND:6044	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.053253216	IUPHAR.LIGAND:5696	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:6172	iuphar.ligand:6172	D-NAL,CYS,TYR,D-TRP,ORN,VAL,CYS,NAL-NH2	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:623	iuphar.ligand:623	[125I][TYR4]BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:613	iuphar.ligand:613	NEUROMEDIN B	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:6183	iuphar.ligand:6183	[D-TPI6, LEU13 &PSI;(CH2NH)-LEU14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:6172	iuphar.ligand:6172	D-NAL,CYS,TYR,D-TRP,ORN,VAL,CYS,NAL-NH2	FALSE	FALSE	FALSE
NCBIGENE:2845	hgnc:4477	GPR22	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11086	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:8699	ncit:C152868	VERUBECESTAT	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:9963	iuphar.ligand:9963	ATABECESTAT	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:7789	iuphar.ligand:7789	LANABECESTAT	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.085239726	IUPHAR.LIGAND:2561	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:559	rxcui:36117	SALMETEROL	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.05293112	IUPHAR.LIGAND:536	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:6828	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.091796628	IUPHAR.LIGAND:6849	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:6828	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	1.009762908	IUPHAR.LIGAND:9042	ncit:C153105	EVOCALCET	FALSE	FALSE	FALSE
NCBIGENE:2343	ncbigene:2343	FNTBL1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:6534	iuphar.ligand:6534	Z-ARG-LEU-VAL-AGLY-ILE-VAL-OME	FALSE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	0.3088686543276147	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.00757031	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NCBIGENE:389	hgnc:669	RHOC	GuideToPharmacology	2024.1	blocker	0.5147810905460245	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
NCBIGENE:2352	hgnc:3795	FOLR3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11377	iuphar.ligand:11377	CITRUSININE II	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:12752	drugbank:DB05048	CANNABINOR	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:902	iuphar.ligand:902	LY-288513	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3725	iuphar.ligand:3725	DESULFATED CHOLECYSTOKININ-8	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	0.4039051633514962	IUPHAR.LIGAND:758	iuphar.ligand:758	CCL5	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	2.763561643983921	ALPIDEM	ncit:C80669	ALPIDEM	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:771	iuphar.ligand:771	CCL2	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:791	iuphar.ligand:791	RO320-2947/001	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:758	iuphar.ligand:758	CCL5	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	0.08334551	IUPHAR.LIGAND:6780	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.1773907812016706	DMSO	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
NCBIGENE:3010	hgnc:4720	H1-6	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:9951	iuphar.ligand:9951	OTLERTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2601	hgnc:4153	GAPDHP60	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:7983	iuphar.ligand:7983	LINTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1993	hgnc:3313	ELAVL2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10081	iuphar.ligand:10081	KINASE INHIBITOR 2 [PMID: 30199702]	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:7960	ncit:C81937	RABUSERTIB	FALSE	FALSE	TRUE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:5991	iuphar.ligand:5991	ISOGRANULATIMIDE	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	NULL	8.353493151133215	IUPHAR.LIGAND:7481	rxcui:1655922	LUMACAFTOR	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.027010119	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
NCBIGENE:703	hgnc:2022	CLCN4	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:6469	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.02804897	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
NCBIGENE:2607	hgnc:3546	F8	GuideToPharmacology	2024.1	inhibitor	4.118248724368195	IUPHAR.LIGAND:6788	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11364	iuphar.ligand:11364	JTV-803	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.017059022	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
NCBIGENE:3195	hgnc:5056	TLX1	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:11763	iuphar.ligand:11763	SOTEVTAMAB	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:7711	iuphar.ligand:7711	AZD6495	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	antibody	0.9907107780319716	IUPHAR.LIGAND:9106	iuphar.ligand:9106	AMG820	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.012383885	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	NULL	0.061919424	IUPHAR.LIGAND:4942	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	NULL	0.090064616	IUPHAR.LIGAND:4934	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:10448	iuphar.ligand:10448	COMPOUND 9 [KUMAR ET AL., 2019]	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:685	rxcui:235481	HUMAN CALCITONIN	TRUE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:922	iuphar.ligand:922	UROTENSIN 1 (FISH)	FALSE	FALSE	FALSE
PSMA3	hgnc:9532	PSMA3	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:3215	hgnc:5116	HOXB5	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12314	iuphar.ligand:12314	COMPOUND 27 [PMID: 36449304]	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:829	iuphar.ligand:829	CXCL5	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:8497	iuphar.ligand:8497	NAVARIXIN	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	0.5000730593875666	IUPHAR.LIGAND:4358	iuphar.ligand:4358	CXCL12&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:11587	ncit:C91094	BALIXAFORTIDE	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:8051	iuphar.ligand:8051	BMS-265246	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	CEFDITORIN PIVOXIL	chembl:CHEMBL1514735	CEFDITORIN PIVOXIL	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:11064	iuphar.ligand:11064	(S)-CR8	FALSE	FALSE	FALSE
NCBIGENE:1353	hgnc:2261	COX11	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9866	ncit:C66288	OZAGREL	FALSE	FALSE	FALSE
UNIPROT:P19838	hgnc:7794	NFKB1	TdgClinicalTrial	Jan-14	NULL	0.276356164	HMPL-004	chembl:CHEMBL186141	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
NCBIGENE:1353	hgnc:2261	COX11	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11379	ncit:C73157	PICOTAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1338	hgnc:2278	COX6A1P1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8804	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:10420	iuphar.ligand:10420	CHMFL-KIT-64	FALSE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9893	iuphar.ligand:9893	COMPOUND 9 [PMID: 20718420]	FALSE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:9892	ncit:C48264	TALABOSTAT	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.053433858	Celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
NCBIGENE:2637	hgnc:4186	GBX2	GuideToPharmacology	2024.1	inhibitor	0.3977853881492008	IUPHAR.LIGAND:7242	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:1886	iuphar.ligand:1886	RS 93520	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:1878	iuphar.ligand:1878	BW 245C	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	0.2333674277141978	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.070860555	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.043756393	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.009076521	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.007374673	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:12197	iuphar.ligand:12197	TTK21	FALSE	FALSE	FALSE
NCBIGENE:2012	hgnc:3333	EMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8127	iuphar.ligand:8127	COMPOUND 3B [PMID: 23454515]	FALSE	FALSE	FALSE
NCBIGENE:1232	hgnc:1604	CCR3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:10706	iuphar.ligand:10706	COMPOUND 15 [PMID: 32045236]	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:6999	iuphar.ligand:6999	ANACARDIC ACID	FALSE	FALSE	FALSE
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	5.527123287967842	Oleclumab	ncit:C123914	OLECLUMAB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.062509132	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.031254566	IUPHAR.LIGAND:5916	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.105015342	IUPHAR.LIGAND:1916	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:1918	ncit:C169951	ENPROSTIL	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1967	ncit:C76896	BERAPROST	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:1923	iuphar.ligand:1923	SC-51089	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:1916	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:7879	iuphar.ligand:7879	BMS-690514	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:10603	iuphar.ligand:10603	TG11-77	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	antibody	0.8204323630577265	IUPHAR.LIGAND:8931	iuphar.ligand:8931	MM-111	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.2344092465879218	IUPHAR.LIGAND:7643	iuphar.ligand:7643	AEE788	FALSE	FALSE	TRUE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:5029	iuphar.ligand:5029	NEUREGULIN-2	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	antibody	2.917092846427472	IUPHAR.LIGAND:8931	iuphar.ligand:8931	MM-111	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:12387	iuphar.ligand:12387	ZONGERTINIB	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009974862	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:12145	iuphar.ligand:12145	LSZ102	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:991	iuphar.ligand:991	[125I]ET-1 (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:623	hgnc:1029	BDKRB1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:2834	iuphar.ligand:2834	DY131	FALSE	FALSE	FALSE
NCBIGENE:622	hgnc:1027	BDH1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:2832	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:993	iuphar.ligand:993	[125I]SARAFOTOXIN S6B	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:3461	iuphar.ligand:3461	PHTPP	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:991	iuphar.ligand:991	[125I]ET-1 (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3859	iuphar.ligand:3859	BQ 3020	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	NSC-402083	chembl:CHEMBL1546228	CHEMBL:CHEMBL1546228	FALSE	FALSE	FALSE
NCBIGENE:868	hgnc:1542	CBLB	GuideToPharmacology	2024.1	NULL	1.500219178162699	IUPHAR.LIGAND:4075	iuphar.ligand:4075	[3H]SYM2081	FALSE	FALSE	FALSE
NCBIGENE:1875	hgnc:3119	E2F5	GuideToPharmacology	2024.1	NULL	1.458546423213736	IUPHAR.LIGAND:5078	iuphar.ligand:5078	FAS LIGAND	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:3177	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9077	iuphar.ligand:9077	EXAMPLE 13 [WO2009109743]	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	0.4375639269641209	IUPHAR.LIGAND:3176	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.041150213	IUPHAR.LIGAND:3364	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.047734247	IUPHAR.LIGAND:6963	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.036162308	IUPHAR.LIGAND:7313	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2386712328895204	IUPHAR.LIGAND:7712	iuphar.ligand:7712	AZD7325	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	GNF-PF-5061	chembl:CHEMBL601385	CHEMBL:CHEMBL601385	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4095	iuphar.ligand:4095	&ALPHA;5IA	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:2312	iuphar.ligand:2312	BICUCULLINE	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.4605936073306534	IUPHAR.LIGAND:4321	iuphar.ligand:4321	TETRAHYDRODEOXYCORTICOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.057574201	IUPHAR.LIGAND:4367	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.106290832	IUPHAR.LIGAND:4348	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:2312	iuphar.ligand:2312	BICUCULLINE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:2312	iuphar.ligand:2312	BICUCULLINE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.047647615	IUPHAR.LIGAND:3364	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.058212496	IUPHAR.LIGAND:4193	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:4197	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.4688184931758437	COLFORSIN	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.1422972120208523	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.3017682254924971	IUPHAR.LIGAND:4296	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	1.810609352954982	IUPHAR.LIGAND:12405	iuphar.ligand:12405	LAU463	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6086	iuphar.ligand:6086	GALANIN(1-15)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6115	iuphar.ligand:6115	GAL-B2-C18	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6114	iuphar.ligand:6114	GAL-B2-C14	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:3876	iuphar.ligand:3876	GALANIN(2-29) (RAT/MOUSE)	FALSE	FALSE	FALSE
CA4	hgnc:1375	CA4	ChEMBL	33	inhibitor	0.364636606	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6092	iuphar.ligand:6092	GALANIN(3-29) (RAT/MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3198	iuphar.ligand:3198	BPH-252	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:3730	iuphar.ligand:3730	EXENDIN-3	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:7387	rxcui:1440051	LIXISENATIDE	TRUE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:1102	iuphar.ligand:1102	[D-ARG1,D-PHE5,D-TRP7,9,LEU11]SUBSTANCE P	FALSE	FALSE	FALSE
NCBIGENE:250	hgnc:439	ALPP	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:9896	iuphar.ligand:9896	GLP-2 ANALOGUE 10	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.1935172158563679	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.2778183663264259	IUPHAR.LIGAND:4167	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.2083637747448194	IUPHAR.LIGAND:4133	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:4219	iuphar.ligand:4219	IDRA-21	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:4304	iuphar.ligand:4304	S18986	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:4245	ncit:C80379	TEZAMPANEL ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:4304	iuphar.ligand:4304	S18986	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:4245	ncit:C80379	TEZAMPANEL ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:4102	iuphar.ligand:4102	2,4-EPI-NEODYSIHERBAINE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.088945801	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
NCBIGENE:3110	hgnc:4979	MNX1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10719	iuphar.ligand:10719	C1-27	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:279	ncit:C73316	FLUPERLAPINE	FALSE	FALSE	FALSE
NCBIGENE:2613	hgnc:4149	GAPDHP71	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6835	rxcui:25953	GLUTATHIONE DISULFIDE	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.030598876	IUPHAR.LIGAND:2367	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:2361	drugbank:DB01931	5,7-DICHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:4290	iuphar.ligand:4290	PREGNENOLONE SULPHATE	FALSE	FALSE	FALSE
NCBIGENE:2029	hgnc:3360	ENSA	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8016	iuphar.ligand:8016	CHIR-98014	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:2368	iuphar.ligand:2368	CYANOTRIPHENYLBORATE	FALSE	FALSE	FALSE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:4201	iuphar.ligand:4201	GINKGOLIDE X	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:7819	iuphar.ligand:7819	AZD1080	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:5991	iuphar.ligand:5991	ISOGRANULATIMIDE	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:6706	iuphar.ligand:6706	LSP4-2022	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10065	iuphar.ligand:10065	GLYT1 INHIBITOR 51B	FALSE	FALSE	FALSE
NCBIGENE:311	hgnc:535	ANXA11	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:8467	iuphar.ligand:8467	COMPOUND 2 [PMID: 24486398]	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:1596	rxcui:16817	ACIPIMOX	TRUE	FALSE	FALSE
NCBIGENE:403	hgnc:694	ARL3	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:2355	ncit:C81347	CILOBRADINE	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:5799	iuphar.ligand:5799	D-KYNURENINE	FALSE	FALSE	FALSE
NCBIGENE:400	hgnc:692	ARL1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:2357	rxcui:1649480	IVABRADINE	TRUE	FALSE	FALSE
NCBIGENE:1887	ncbigene:1887	EBVM1	GuideToPharmacology	2024.1	NULL	5.834185692854944	IUPHAR.LIGAND:5064	iuphar.ligand:5064	LYMPHOTOXIN-&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:2615	hgnc:4161	LRRC32	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:11120	iuphar.ligand:11120	ACY-738	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:1237	iuphar.ligand:1236	(R)-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1276	iuphar.ligand:1276	IMPROGAN	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5727	iuphar.ligand:5727	JNJ-38431055	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5741	iuphar.ligand:5741	COMPOUND 29A [PMID: 21444206]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5735	iuphar.ligand:5735	COMPOUND 42 [PMID: 22545772]	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4350	iuphar.ligand:4350	7&ALPHA;,25-DIHYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:99	hgnc:4487	GPR32	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:4356	iuphar.ligand:4356	[3H]RESOLVIN D1	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:2752	iuphar.ligand:2752	27-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:9871	iuphar.ligand:9871	PSB-17365	FALSE	FALSE	FALSE
NCBIGENE:114	hgnc:239	ADCY8	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:10572	iuphar.ligand:10572	POMC (141-162)	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:5540	iuphar.ligand:5540	R-SPONDIN-2	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:5539	iuphar.ligand:5539	R-SPONDIN-1	FALSE	FALSE	FALSE
NCBIGENE:149	hgnc:19719	LGR6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:3700	iuphar.ligand:3700	R-SPONDIN-4	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8221	ncit:C92582	EPACADOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1463	hgnc:2465	NCAN	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:5212	rxcui:42351	LITHIUM CARBONATE	TRUE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:7952	iuphar.ligand:7952	BMS-754807	FALSE	FALSE	FALSE
NCBIGENE:2451	hgnc:3848	FRA12D	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:7533	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
NCBIGENE:2446	hgnc:3843	FRA11H	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:8407	iuphar.ligand:8407	ETROLIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2451	hgnc:3848	FRA12D	GuideToPharmacology	2024.1	antibody	5.250767123569449	IUPHAR.LIGAND:9598	iuphar.ligand:9598	ROVELIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1630	hgnc:2701	DCC	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:2443	hgnc:3841	FRA11F	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11487	ncit:C152814	VALATEGRAST	FALSE	FALSE	FALSE
NCBIGENE:2456	hgnc:3853	FRA13D	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:9598	iuphar.ligand:9598	ROVELIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:5683	iuphar.ligand:5683	GSK-1838705A	FALSE	FALSE	FALSE
NCBIGENE:1710	hgnc:18969	IL31RA	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:8720	iuphar.ligand:8720	NEMOLIZUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	MK-8353	iuphar.ligand:9974	MK-8353	FALSE	FALSE	FALSE
NCBIGENE:2041	hgnc:3385	EPHA1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8116	iuphar.ligand:8116	COMPOUND 22 [PMID: 21823616]	FALSE	FALSE	FALSE
ERCC2	hgnc:3434	ERCC2	NCI	14-Sep-17	NULL	0.1646008502686348	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:7552	rxcui:1729002	SELEXIPAG	TRUE	FALSE	FALSE
NCBIGENE:2884	hgnc:4561	GPX1P2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:12340	iuphar.ligand:12340	LY3410738	FALSE	FALSE	FALSE
NCBIGENE:671	hgnc:1095	BPI	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:6412	iuphar.ligand:6412	VANILLIN	FALSE	FALSE	FALSE
NCBIGENE:659	hgnc:1078	BMPR2	GuideToPharmacology	2024.1	agonist	2.625383561784725	IUPHAR.LIGAND:12424	iuphar.ligand:12424	L-TRP-TRP-TRP	FALSE	FALSE	FALSE
NCBIGENE:671	hgnc:1095	BPI	GuideToPharmacology	2024.1	agonist	0.3977853881492008	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
NCBIGENE:661	hgnc:1080	POLR3D	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:12424	iuphar.ligand:12424	L-TRP-TRP-TRP	FALSE	FALSE	FALSE
NCBIGENE:661	hgnc:1080	POLR3D	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:2367	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:663	hgnc:1083	BNIP2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:12436	iuphar.ligand:12436	GRANDININ	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	7.001022831425932	LY-2608204	drugbank:DB12284	LY-2608204	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	NULL	0.2187819634820604	IUPHAR.LIGAND:12310	iuphar.ligand:12310	SJ988497	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:12171	iuphar.ligand:12171	COMPOUND 8L [PMID: 36053746]	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:9177	iuphar.ligand:9177	AC430	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:8123	iuphar.ligand:8123	COMPOUND 1D [PMID: 21493067]	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:8315	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.09869863	IUPHAR.LIGAND:5716	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:10527	iuphar.ligand:10527	LASW1393	FALSE	FALSE	FALSE
NCBIGENE:2375	hgnc:3887	FRA2C	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8483	iuphar.ligand:8483	COMPOUND 4D [PMID: 25489658]	FALSE	FALSE	FALSE
NCBIGENE:2376	hgnc:3888	FRA2D	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:10576	iuphar.ligand:10576	COMPOUND 32 [PMID: 31675166]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.1151484018326633	IUPHAR.LIGAND:9002	iuphar.ligand:9002	BW373U86	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:9189	iuphar.ligand:9189	HS665	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.057574201	IUPHAR.LIGAND:1670	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:1631	iuphar.ligand:1631	&BETA;-FNA	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0296486	IUPHAR.LIGAND:10033	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.041508041	IUPHAR.LIGAND:11743	drugbank:DB08577	3-[(3-(2-CARBOXYETHYL)-4-METHYLPYRROL-2-YL)METHYLENE]-2-INDOLINONE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.042689164	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
LIPID PEROXIDATION	hgnc:6678	LPO	TTD	2020.06.01	NULL	5.250767123569449	T-817MA	chembl:CHEMBL4297438	T-817 MALEATE	FALSE	FALSE	FALSE
NCBIGENE:523	hgnc:851	ATP6V1A	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:517	hgnc:842	ATP5MC2	GuideToPharmacology	2024.1	activator	0.7292732116068681	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	0.3750547945406749	IUPHAR.LIGAND:2312	iuphar.ligand:2312	BICUCULLINE	FALSE	FALSE	FALSE
NCBIGENE:387	hgnc:667	RHOA	GuideToPharmacology	2024.1	activator	2.500365296937833	IUPHAR.LIGAND:4271	iuphar.ligand:4271	NS004	FALSE	FALSE	FALSE
NCBIGENE:576	hgnc:944	ADGRB2	GuideToPharmacology	2024.1	blocker	6.563458904461812	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.3977853881492008	IUPHAR.LIGAND:2561	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:12993	iuphar.ligand:12993	TPT-004	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.364636606	CRIDANIMOD	ncit:C77948	CRIDANIMOD	FALSE	FALSE	FALSE
NCBIGENE:2685	ncbigene:2685	GGTL2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8230	iuphar.ligand:8230	IOX1	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.596678082	DAPOXETINE	ncit:C75168	DAPOXETINE	TRUE	FALSE	FALSE
NCBIGENE:3097	hgnc:4921	HIVEP2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10485	iuphar.ligand:10485	CCT365623	FALSE	FALSE	FALSE
NCBIGENE:1816	hgnc:3026	DRD5	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:2680	hgnc:9886	KDM5A	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:7027	iuphar.ligand:7027	GSK-J1	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:3633	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.051478109	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:8292	iuphar.ligand:8292	AM7	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:8178	iuphar.ligand:8178	COMPOUND 16 [PMID: 18945615]	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:1368	iuphar.ligand:1368	L-CCG-I	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1000146118775133	IUPHAR.LIGAND:7672	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6257	iuphar.ligand:6257	CYPPTS	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1368	iuphar.ligand:1368	L-CCG-I	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6408	iuphar.ligand:6408	[3H]CTEP	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:4059	iuphar.ligand:4059	VU-1545	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	1.029562181092049	SERIBANTUMAB	ncit:C78859	SERIBANTUMAB	FALSE	FALSE	TRUE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1368	iuphar.ligand:1368	L-CCG-I	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:1439	iuphar.ligand:1439	MCCG	FALSE	FALSE	FALSE
NCBIGENE:1051	hgnc:1834	CEBPB	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12853	iuphar.ligand:12853	CTPI-2	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	0.4318065068724876	IUPHAR.LIGAND:2875	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
NCBIGENE:1051	hgnc:1834	CEBPB	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:4701	iuphar.ligand:4701	1,2,3-BENZENETRICARBOXYLIC ACID	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.305277158	FPA144	chembl:CHEMBL4650291	FPA144	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2871	rxcui:3256	DESOXYCORTICOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:12122	iuphar.ligand:12122	COMPOUND 4E [PMID: 35546685]	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10429	iuphar.ligand:10429	J30-8	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:5998	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:7818	iuphar.ligand:7818	PH-797804	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:12706	drugbank:DB15498	BOS172722	FALSE	FALSE	FALSE
NCBIGENE:1494	hgnc:6877	MAPK3	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:5966	drugbank:DB07794	5-(2-PHENYLPYRAZOLO[1,5-A]PYRIDIN-3-YL)-1H-PYRAZOLO[3,4-C]PYRIDAZIN-3-AMINE	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.089046362	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:2090	hgnc:3462	ESA4	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8176	iuphar.ligand:8176	BS-194	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8058	iuphar.ligand:8058	JNK-IN-8	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:12334	iuphar.ligand:12334	COMPOUND 25C [PMID: 36649216]	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:8836	iuphar.ligand:8836	PP1	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.4167275494896389	IUPHAR.LIGAND:5998	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
NCBIGENE:2084	hgnc:6861	MAP3K9	GuideToPharmacology	2024.1	inhibitor	0.7292732116068681	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
NCBIGENE:2084	hgnc:6861	MAP3K9	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8070	iuphar.ligand:8070	P505-15	FALSE	FALSE	FALSE
NCBIGENE:2089	ncbigene:2089	ERVT1	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
UNIPROT:P14780	hgnc:7176	MMP9	TdgClinicalTrial	Jan-14	NULL	1.050153425	COL-3	ncit:C2454	INCYCLINIDE	FALSE	FALSE	FALSE
NCBIGENE:2083	ncbigene:2083	ERPL2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:6051	iuphar.ligand:6051	TPL2 KINASE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:8629	iuphar.ligand:8629	SL422	FALSE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:6514	iuphar.ligand:6514	COMPOUND 1A [PMID: 15055993]	FALSE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:8629	iuphar.ligand:8629	SL422	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1463	iuphar.ligand:1463	MOTILIN-(1-19) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.1262203635473425	IUPHAR.LIGAND:348	iuphar.ligand:348	THIOCHROME	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	NIGULDIPINE	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:12304	iuphar.ligand:12304	T440	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.1262203635473425	IUPHAR.LIGAND:7632	iuphar.ligand:7632	VU0119498	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:293	iuphar.ligand:293	NNC 11-1607	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:292	iuphar.ligand:292	NNC 11-1585	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:303	iuphar.ligand:303	OXOTREMORINE-M	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:10470	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:361	iuphar.ligand:361	TRIPITRAMINE	FALSE	FALSE	FALSE
KDM4D	hgnc:25498	KDM4D	DTC	9/2/20	NULL	17.50255707856483	N-METHOXYCARBONYLMETHYL-OXALAMIC ACID METHYL ESTER	chembl:CHEMBL92309	CHEMBL:CHEMBL92309	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1344	iuphar.ligand:1344	2-[125I]MELATONIN	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1353	iuphar.ligand:1353	S24014	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:12955	iuphar.ligand:12955	ISOTONITAZENE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:9150	rxcui:1876597	NALDEMEDINE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.096167896	IUPHAR.LIGAND:1628	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.157680694	IUPHAR.LIGAND:2586	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:8123	iuphar.ligand:8123	COMPOUND 1D [PMID: 21493067]	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:11198	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:12389	ncit:C179627	ZURLETRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.2678962818147678	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:6506	ncit:C73039	DAGLUTRIL	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	agonist	0.034590034	IUPHAR.LIGAND:2585	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
NCBIGENE:2118	hgnc:3493	ETV4	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:2115	iuphar.ligand:2115	GR 159897	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:9280	ncit:C81499	SERLOPITANT	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:3795	iuphar.ligand:3795	[125I]NKA (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:2861	hgnc:4494	GPR37	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11362	iuphar.ligand:11362	IMR-1	FALSE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:1496	iuphar.ligand:1496	NEUROPEPTIDE W-30	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1478	iuphar.ligand:1478	EFWSLAAPQRF-NH2	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:11073	iuphar.ligand:11073	S‐Y048	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9303	iuphar.ligand:9303	ACT-462206	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:11527	iuphar.ligand:11527	[3H]-TCS 1102	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:11527	iuphar.ligand:11527	[3H]-TCS 1102	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	NULL	0.5834185692854944	IUPHAR.LIGAND:3798	iuphar.ligand:3798	[125I]OREXIN A (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4266	iuphar.ligand:4266	NF023	FALSE	FALSE	FALSE
NCBIGENE:2137	hgnc:3518	EXTL3	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8937	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
NCBIGENE:479	hgnc:13816	ATP12A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9539	iuphar.ligand:9539	PSB-10211	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11969	ncit:C175513	ELIAPIXANT	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	0.4412409347537352	IUPHAR.LIGAND:1712	iuphar.ligand:1712	ADP	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4122	iuphar.ligand:4122	A839977	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4119	iuphar.ligand:4119	A740003	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11826	iuphar.ligand:11826	ITH15004	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	agonist	0.3750547945406749	IUPHAR.LIGAND:1712	iuphar.ligand:1712	ADP	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1732	iuphar.ligand:1732	AP4A	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:1737	ncit:C78118	DENUFOSOL	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:1709	drugbank:DB02189	2',3'-DIDEOXYADENOSINE TRIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2261	iuphar.ligand:2261	[125I]PACAP-27	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2257	iuphar.ligand:2257	PACAP-27	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:3851	iuphar.ligand:3851	2-FUROYL-LIGRLO-AMIDE	FALSE	FALSE	FALSE
NCBIGENE:3100	hgnc:9360	PRF1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10501	iuphar.ligand:10501	COMPOUND 16 [PMID: 31525966]	FALSE	FALSE	FALSE
NCBIGENE:2877	hgnc:4554	GPX2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8685	iuphar.ligand:8685	CL-AMIDINE	FALSE	FALSE	FALSE
NCBIGENE:3171	hgnc:5023	FOXA3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11398	iuphar.ligand:11398	AG-122018	FALSE	FALSE	FALSE
NCBIGENE:2877	hgnc:4554	GPX2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8684	iuphar.ligand:8684	COMPOUND 14B [PMID: 25742366]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:10162	iuphar.ligand:10162	RV1729	FALSE	FALSE	FALSE
NCBIGENE:2149	hgnc:3537	F2R	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.096521454	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9330	iuphar.ligand:9330	CDP840	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9852	iuphar.ligand:9852	MK-0359	FALSE	FALSE	FALSE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:7399	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:5225	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9368	iuphar.ligand:9368	CX-6258	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:7698	iuphar.ligand:7698	AZD1208	FALSE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.2536602475154323	IUPHAR.LIGAND:8482	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:8095	iuphar.ligand:8095	AC710	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:5656	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.087512785	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.070010228	IUPHAR.LIGAND:7882	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
NCBIGENE:1434	hgnc:2431	CSE1L	GuideToPharmacology	2024.1	activator	1.093909817410302	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
NCBIGENE:1434	hgnc:2431	CSE1L	GuideToPharmacology	2024.1	activator	0.7955707762984016	IUPHAR.LIGAND:1054	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:9402	iuphar.ligand:9402	MLN0905	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	0.546954909	IUPHAR.LIGAND:12990	ncit:C132992	SINTILIMAB	FALSE	FALSE	FALSE
NCBIGENE:2387	hgnc:3899	FRA3D	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:8668	iuphar.ligand:8668	FURIN INHIBITOR PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1476	hgnc:2482	CSTB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:5983	drugbank:DB07995	H-89	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8010	iuphar.ligand:8010	NU-7441	FALSE	FALSE	TRUE
NCBIGENE:2173	hgnc:3562	FABP7	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9370	iuphar.ligand:9370	BPKDI	FALSE	FALSE	FALSE
NCBIGENE:2174	hgnc:9408	PRKD3	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:8048	iuphar.ligand:8048	CRT 0066101	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:8805	iuphar.ligand:8805	COMPOUND 82 [PMID: 21332118]	FALSE	FALSE	FALSE
NCBIGENE:2181	hgnc:3570	ACSL3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9763	iuphar.ligand:9763	CONTELTINIB	FALSE	FALSE	FALSE
NCBIGENE:3203	hgnc:5107	HOXA6	GuideToPharmacology	2024.1	modulator	17.50255707856483	IUPHAR.LIGAND:12970	iuphar.ligand:12970	MIGOPROTAFIB	FALSE	FALSE	FALSE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11562	iuphar.ligand:11562	COMPOUND V [PMID: 29351497]	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.1666910197958555	IUPHAR.LIGAND:2645	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:8729	iuphar.ligand:8729	(5Z)-5-[(5-BROMOTHIOPHEN-2-YL)METHYLIDENE]-1-METHYL-2-SULFANYLIDENE-1,3-DIAZINANE-4,6-DIONE	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.3182283105193606	IUPHAR.LIGAND:6952	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:2651	iuphar.ligand:2651	BMS641	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:2640	iuphar.ligand:2640	AGN193109	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:2648	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:10186	iuphar.ligand:10186	COMPOUND 28 [HEITEL ET AL., 2019]	FALSE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:8904	iuphar.ligand:8904	FLUOROBEXAROTENE	FALSE	FALSE	FALSE
NCBIGENE:597	hgnc:991	BCL2A1	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:8900	iuphar.ligand:8900	SR9011	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:11678	iuphar.ligand:11678	VEPAFESTINIB	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8342	iuphar.ligand:8342	EUROPIUM-LABELLED R3(B1-22R)	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:11465	iuphar.ligand:11465	NANOLUC R3/I5 CHIMERA	FALSE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	activator	0.280789686	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:8336	iuphar.ligand:8336	MINIMISED RELAXIN-3 ANALOGUE 2	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.046965717	IUPHAR.LIGAND:202	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2199	hgnc:3601	FBLN2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5678	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12268	iuphar.ligand:12268	TTI-101	FALSE	FALSE	FALSE
NCBIGENE:2712	hgnc:4291	GK2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8816	iuphar.ligand:8816	AKK(THIOAC)LM21	FALSE	FALSE	FALSE
NCBIGENE:1170	hgnc:13448	SLC38A2	GuideToPharmacology	2024.1	NULL	10.50153425	IUPHAR.LIGAND:4543	rxcui:426	ALANINE	TRUE	FALSE	FALSE
NCBIGENE:960	hgnc:1681	CD44	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:11194	rxcui:2563966	ODEVIXIBAT	TRUE	FALSE	FALSE
NCBIGENE:1419	hgnc:2409	CRYGB	GuideToPharmacology	2024.1	inhibitor	7.501095890813499	IUPHAR.LIGAND:8787	iuphar.ligand:8787	COMPOUND 12E [PMID: 18605714]	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:6624	iuphar.ligand:6624	OPAGANIB	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:6041	iuphar.ligand:6041	SKI II	FALSE	FALSE	FALSE
NCBIGENE:1417	hgnc:2400	CRYBB3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8787	iuphar.ligand:8787	COMPOUND 12E [PMID: 18605714]	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2008	iuphar.ligand:2008	CST-17	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:2029	iuphar.ligand:2029	[L-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2064	iuphar.ligand:2064	[111IN]DOTA-NOC-ATE	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:10113	iuphar.ligand:10113	DOTA-JR11	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:10115	iuphar.ligand:10115	J-2156	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2064	iuphar.ligand:2064	[111IN]DOTA-NOC-ATE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2051	ncit:C152317	SEGLITIDE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2008	iuphar.ligand:2008	CST-17	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	0.2234368988752957	IUPHAR.LIGAND:2027	iuphar.ligand:2027	BIM 23627	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	0.2234368988752957	IUPHAR.LIGAND:2029	iuphar.ligand:2029	[L-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10673	iuphar.ligand:10673	RK-287107	FALSE	FALSE	FALSE
NCBIGENE:2414	hgnc:3925	FRA7G	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8780	iuphar.ligand:8780	COMPOUND 8E [PMID: 23044371]	FALSE	FALSE	FALSE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11600	iuphar.ligand:11600	COMPOUND 21 [PMID: 34141085]	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:10454	iuphar.ligand:10454	ULOTARONT	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5510	iuphar.ligand:5510	2-PHENYL-PROPYLAMINE	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:2633	iuphar.ligand:2633	NH-3	FALSE	FALSE	FALSE
NCBIGENE:615	hgnc:7973	NR2E1	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:11832	iuphar.ligand:11832	COMPOUND 10 [PMID: 34989568]	FALSE	FALSE	FALSE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11858	iuphar.ligand:11858	UM-9	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1986	ncit:C169873	DALTROBAN	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:1974	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	activator	1.312691780892362	IUPHAR.LIGAND:2794	iuphar.ligand:2794	PHOSPHATIDYL (3,5) INOSITOL BISPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2244	hgnc:3662	FGB	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:11833	iuphar.ligand:11833	COMPOUND 21K [PMID: 34985886]	FALSE	FALSE	FALSE
NCBIGENE:3196	hgnc:5057	TLX2	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:11773	iuphar.ligand:11773	LEPUNAFUSP ALFA	FALSE	FALSE	FALSE
NCBIGENE:486	hgnc:4026	FXYD2	GuideToPharmacology	2024.1	blocker	0.2734774543525755	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:8372	iuphar.ligand:8372	(-)-ENGLERIN A	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	0.3454452054979901	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.3860858179095183	IUPHAR.LIGAND:10285	iuphar.ligand:10285	CLEMIZOLE	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	activator	0.2344092465879218	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	1.875273972703375	IUPHAR.LIGAND:10038	iuphar.ligand:10038	COMPOUND 5 [PMID: 29579323]	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10038	iuphar.ligand:10038	COMPOUND 5 [PMID: 29579323]	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.056097939	IUPHAR.LIGAND:2693	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:2455	rxcui:309	ADENOSINE MONOPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	0.2917092846427472	IUPHAR.LIGAND:4290	iuphar.ligand:4290	PREGNENOLONE SULPHATE	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	0.1103102336884338	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.2143170254518142	IUPHAR.LIGAND:11576	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	1.093909817410302	IUPHAR.LIGAND:6386	iuphar.ligand:6386	ML SA1	FALSE	FALSE	FALSE
NCBIGENE:502	hgnc:13357	MCOLN2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11861	iuphar.ligand:11861	PRU-10	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	activator	0.8751278539282418	IUPHAR.LIGAND:2478	rxcui:21183	CITRIC ACID	TRUE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	0.6563458904461813	IUPHAR.LIGAND:2794	iuphar.ligand:2794	PHOSPHATIDYL (3,5) INOSITOL BISPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	blocker	0.4375639269641208	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	activator	0.3281729452230906	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	1.117184494376478	IUPHAR.LIGAND:9169	iuphar.ligand:9169	COMPOUND 34H [PMID: 27055065]	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:11425	iuphar.ligand:11425	TYK2 INHIBITOR 14L	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:11060	iuphar.ligand:11060	PF-956980	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2261	iuphar.ligand:2261	[125I]PACAP-27	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:2180	iuphar.ligand:2180	[VAL4]AVP	FALSE	FALSE	FALSE
NCBIGENE:2280	hgnc:3711	FKBP1A	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:8836	iuphar.ligand:8836	PP1	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:7432	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2234	iuphar.ligand:2234	[3H]SR 121463A	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:2202	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:1485	iuphar.ligand:1485	BIBP3226	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1524	iuphar.ligand:1524	[LEU31,PRO34]NPY (PIG)	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1540	iuphar.ligand:1540	NPY-(26-36) (PIG)	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.2363572458670459	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.096167896	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.6168664383892681	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
HLA-C	hgnc:4933	HLA-C	CIViC	10-Apr-24	NULL	1.458546423213736	THERAPEUTIC TUMOR INFILTRATING LYMPHOCYTES	ncit:C28699	THERAPEUTIC TUMOR INFILTRATING LYMPHOCYTES	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.2044691247495891	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.5556367326528519	GRACILIN J	chembl:CHEMBL1077759	GRACILIN J	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	1.029066006546944	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CD44	hgnc:1681	CD44	CIViC	10-Apr-24	NULL	0.033295923	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.040230625	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	ICRF-193	chembl:CHEMBL275665	ICRF-193	FALSE	FALSE	FALSE
SUFU	hgnc:16466	SUFU	CIViC	10-Apr-24	NULL	8.751278539282415	SONIDEGIB	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.1931849567170511	RG7112	drugbank:DB14793	RO-5045337	FALSE	FALSE	TRUE
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	0.7292732116068681	hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
GAS6	hgnc:4168	GAS6	CIViC	10-Apr-24	NULL	0.2108741816694558	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.5147810905460244	QUARFLOXIN	ncit:C71726	QUARFLOXIN	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	CIViC	10-Apr-24	NULL	0.043180651	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.004501686	CAPECITABINE	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.8178764989983567	PEMIGATINIB	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
PALB2	hgnc:26144	PALB2	CIViC	10-Apr-24	NULL	0.4861821410712453	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	CIViC	10-Apr-24	NULL	0.07458476	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:12991	iuphar.ligand:12991	PROLGOLIMAB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.001193302	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	CIViC	10-Apr-24	NULL	0.012466209	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1591141552596803	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1446492320542548	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.078545507	BI2536	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	Pimasertib	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.028937818	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:2632	hgnc:4180	GBE1	GuideToPharmacology	2024.1	activator	3.500511415712966	IUPHAR.LIGAND:6819	rxcui:321208	FONDAPARINUX	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.7059854956059763	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.016472995	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.091317689	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.6543011991986852	E7090	ncit:C118672	TASURGRATINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.4070362111294147	HMPL-453	chembl:CHEMBL4650297	HMPL-453	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.276356164	Derazantinib	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.051177067	Foretinib	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.010685322	Tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	ERAS-601	ncit:C176881	SHP2 INHIBITOR ERAS-601	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	AGL2043	iuphar.ligand:5918	AGL 2043	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.8899605294185507	NERVIANO	chembl:CHEMBL1172241	NERVIANO	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.108040476	Abivertinib	ncit:C147125	ABIVERTINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.108040476	PRT062607	iuphar.ligand:8070	P505-15	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.1973972602845657	Pralsetinib	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.2302968036653267	SCH772984	iuphar.ligand:8056	SCH772984	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.010270449	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.006669123	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	1.016277507787635	Upadacitinib	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.5135224570728067	IDH305	chembl:CHEMBL4167360	IDH305	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.8561033353645842	AZ960	iuphar.ligand:8476	AZ960	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2282942227638891	Luminespib	ncit:C71467	LUMINESPIB	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.043902735	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	1.712206670729168	BMS-911543	drugbank:DB12591	BMS-911543	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.091159151	Pimasertib	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.027010119	AZD6482	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.5339763176511304	RESCINNAMINE	rxcui:9259	RESCINNAMINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.027010119	Ado-trastuzumab emtansine	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	GSK1059615	iuphar.ligand:9826	GSK1059615	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.1448487482363986	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	1.346350544504987	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.3977853881492008	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.064824285	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.2586584789935689	Capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	Prodigiosin	chembl:CHEMBL275787	PRODIGIOSIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.012878997	Rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.086933231	Zanubrutinib	rxcui:2262435	ZANUBRUTINIB	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.028977744	Pegylated liposomal doxorubicin	rxcui:214525	DOXORUBICIN LIPOSOME	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.017386646	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.028977744	Ganetespib	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	4.039051633514961	TA-8995	ncit:C175167	OBICETRAPIB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.077273983	Alvespimycin	ncit:C38142	ALVESPIMYCIN	FALSE	FALSE	TRUE
KCNA4	hgnc:6222	KCNA4	ChEMBL	33	blocker	0.1875273972703375	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	inhibitor	2.059124362184098	INOLIMOMAB	ncit:C170069	INOLIMOMAB	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:5677	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
GUCY2C	hgnc:4688	GUCY2C	ChEMBL	33	agonist	13.12691780892362	DOLCANATIDE	ncit:C153478	DOLCANATIDE	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.085691834	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2580229544751573	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.033148782	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.017386646	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.043692674	ARIPIPRAZOLE LAUROXIL	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.048708415	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	NSC-309895	chembl:CHEMBL552439	CHEMBL:CHEMBL552439	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	LASSBIO-294	chembl:CHEMBL233194	CHEMBL:CHEMBL233194	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ETHAVERINE HYDROCHLORIDE	rxcui:235229	ETHAVERINE HYDROCHLORIDE	FALSE	FALSE	FALSE
AANAT	hgnc:19	AANAT	NCI	14-Sep-17	NULL	0.042619863	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	ChEMBL	33	inhibitor	1.093909817410302	ICATIBANT ACETATE	rxcui:1294605	ICATIBANT ACETATE	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.9512259281828714	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.2263261691193728	IRBESARTAN	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.069043618	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	0.7001022831425934	ANTICONVULSANT DRUGS	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.046059361	IUPHAR.LIGAND:2	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NCBIGENE:451	hgnc:769	ASS1P6	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:4231	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2826	hgnc:4474	CCR10	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6531	iuphar.ligand:6531	FTI 276	FALSE	FALSE	FALSE
NCBIGENE:115	hgnc:240	ADCY9	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:758	iuphar.ligand:758	CCL5	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00292359	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.00637229	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	0.4102161815288632	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1988926940746003	LIAFENSINE	ncit:C170121	LIAFENSINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	AMG-232	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.212581665	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.1682938180631233	ANTHRACYCLINE	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
CXCL10	hgnc:10637	CXCL10	PharmGKB	4/5/24	NULL	0.2130128650535273	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	GW642444	rxcui:1424884	VILANTEROL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	LY-310762	chembl:CHEMBL1256663	CHEMBL:CHEMBL1256663	FALSE	FALSE	FALSE
RBX1	hgnc:9928	RBX1	ChEMBL	33	inhibitor	0.5770073762164232	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CancerCommons	25-Jul-13	inhibitor	1.346350544504987	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PTH1R	hgnc:9608	PTH1R	DTC	9/2/20	NULL	0.3409589041278864	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.2365210416022274	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.022949157	PAN-90806	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:3724	iuphar.ligand:3724	CHIPS	FALSE	FALSE	FALSE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.3889457128569963	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	QUINOCIDE	ncit:C73004	QUINOCIDE	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6576	ncit:C152419	SPIRAPRILAT	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.062509132	IUPHAR.LIGAND:6044	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.065799087	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.1470803115845784	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
UCP1	hgnc:12517	UCP1	NCI	14-Sep-17	NULL	2.692701089009974	ALPHA-METHYL-P-TYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.043502627	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.2853677784548614	PACRITINIB CITRATE	rxcui:2595242	PACRITINIB CITRATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
TMPRSS15	hgnc:9490	TMPRSS15	DTC	9/2/20	NULL	0.5250767123569451	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.2019525816757481	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.048327355	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.096344351	Analgesics	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
UNIPROT:P07333	hgnc:2433	CSF1R	TdgClinicalTrial	Jan-14	NULL	0.035800685	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:1272	iuphar.ligand:1272	CCL16	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:4071	drugbank:DB02818	IODO-WILLARDIINE	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.7721716358190367	ZT-1	ncit:C99560	MIMOPEZIL	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9509	iuphar.ligand:9509	SB-3CT	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	DNDI1417063	chembl:CHEMBL2094422	CHEMBL:CHEMBL2094422	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9885	iuphar.ligand:9885	CORTISTATIN A	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1519	iuphar.ligand:1519	[125I]PYY	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.4254093734373397	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	AC-3579	chembl:CHEMBL1569213	CHEMBL:CHEMBL1569213	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.2465148884304905	KP201	chembl:CHEMBL3137310	BENZHYDROCODONE HYDROCHLORIDE	FALSE	FALSE	FALSE
PSMB3	hgnc:9540	PSMB3	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.2917092846427472	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1154014752432845	C5A	iuphar.ligand:3576	C5A	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.035216413	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:6918	iuphar.ligand:6918	COMPOUND 21 [PMID: 22802221]	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.014385663	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1907	iuphar.ligand:1907	L-888,607	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.043039075	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	MECYSTEINE HYDROCHLORIDE	rxcui:235828	MECYSTEINE HYDROCHLORIDE	FALSE	FALSE	FALSE
S1PR2	hgnc:3169	S1PR2	ChEMBL	33	agonist	1.500219178	FINGOLIMOD HYDROCHLORIDE	rxcui:1012891	FINGOLIMOD HYDROCHLORIDE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	ChEMBL	33	inhibitor	0.013286354	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1944728564284981	GNF-PF-4242	chembl:CHEMBL584514	CHEMBL:CHEMBL584514	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00292359	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.4773424657790409	TOLMETIN	rxcui:10636	TOLMETIN	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.058931169	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
SLC28A3	hgnc:16484	SLC28A3	DTC	9/2/20	NULL	1.875273972703375	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	CancerCommons	25-Jul-13	inhibitor	1.944728564284981	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.043866058	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.029301156	IUPHAR.LIGAND:536	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
UGCG	hgnc:12524	UGCG	ChEMBL	33	inhibitor	10.50153424713889	ELIGLUSTAT TARTRATE	rxcui:1547219	ELIGLUSTAT TARTRATE	TRUE	FALSE	FALSE
NCBIGENE:3208	hgnc:5144	HPCA	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12224	iuphar.ligand:12224	COMPOUND 61 [PMID: 36221183]	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016780975	TACRINE	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	PharmGKB	4/5/24	NULL	0.059397818	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	CancerCommons	25-Jul-13	inhibitor	0.2273059360852575	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
FGFR1OP	hgnc:17012	CEP43	PharmGKB	4/5/24	NULL	7.501095890813499	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	DIXANTHOGEN	drugbank:DB13712	DIXANTHOGEN	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	COUMARIN-3-CARBOXYLIC ACID	chembl:CHEMBL83294	COUMARIN-3-CARBOXYLIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.095295229	Diazepam	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	0.760980743	LJN452	ncit:C152764	TROPIFEXOR	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:12578	iuphar.ligand:12578	CIMATEROL	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.013025967	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:2606	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	1.179947668217853	IUPHAR.LIGAND:6788	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2656	iuphar.ligand:2656	GW409544	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW837331X	chembl:CHEMBL520037	GW837331X	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.003796101	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.0037759	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
FXYD2	hgnc:4026	FXYD2	ChEMBL	33	inhibitor	0.1286952726365061	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TRITIOZINE	ncit:C90780	TRITIOZINE	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.070197421	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
AKR1C4	hgnc:387	AKR1C4	PharmGKB	4/5/24	NULL	3.088686543276147	naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
ZFP91-CNTF	hgnc:33441	ZFP91-CNTF	PharmGKB	4/5/24	NULL	5.000730593875666	iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.046221542	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:1241	iuphar.ligand:1241	N-[3H]METHYLHISTAMINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.006954658	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.052090944	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2917092846427472	YANGONIN	chembl:CHEMBL1098658	YANGONIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.004931224	Clobazam	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	NCI	14-Sep-17	NULL	0.021715331	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.1555782851427985	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	TRAZODONE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.4773424657790409	MCS-110	chembl:CHEMBL2109512	MCS-110	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.4922594178346359	UPROSERTIB	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	DIHYDROSPINGOSINE	iuphar.ligand:2453	DIHYDROSPHINGOSINE	FALSE	FALSE	FALSE
THBD	hgnc:11784	THBD	NCI	14-Sep-17	NULL	1.250182648468916	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	2.625383561784724	DSP-0509	ncit:C153314	GURETOLIMOD	FALSE	FALSE	FALSE
UNIPROT:P01111	hgnc:7989	NRAS	TdgClinicalTrial	Jan-14	NULL	0.1411496538593938	REOLYSIN	chembl:CHEMBL3545069	PELAREOREP	FALSE	FALSE	TRUE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.022632617	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	VE800	ncit:C167393	COMMENSAL BACTERIAL STRAIN FORMULATION VE800	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.04427291	donepezil	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
UNIPROT:P21860	hgnc:3431	ERBB3	TdgClinicalTrial	Jan-14	NULL	0.3431873936973496	GGF-2	chembl:CHEMBL3039542	CIMAGLERMIN ALFA	FALSE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	DEMECARIUM BROMIDE	rxcui:22482	DEMECARIUM BROMIDE	TRUE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TEND	1-Aug-11	NULL	0.8334550989792776	MUROMONAB	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.1457197166578015	NICOTINE POLACRILEX	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	Docarpamine	ncit:C65453	DOCARPAMINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	PRIDINOL	rxcui:34479	PRIDINOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ALDRIN	chembl:CHEMBL195953	ALDRIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BUTACHLOR	chembl:CHEMBL1399036	BUTACHLOR	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	XANTHURENATE	chembl:CHEMBL312535	XANTHURENATE	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.08334551	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1400204566285186	DIFENOCONAZOLE	chembl:CHEMBL466426	DIFENOCONAZOLE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.034819411	IUPHAR.LIGAND:7351	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	Namitecan	ncit:C95910	NAMITECAN	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.09741683	IUPHAR.LIGAND:422	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12353	iuphar.ligand:12353	SKLB-03220	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.1438566335224507	ALTIRATINIB	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:5943	iuphar.ligand:5943	CDK/CRK INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:348	iuphar.ligand:348	THIOCHROME	FALSE	FALSE	FALSE
NA	hgnc:12811	XK	ChEMBL	33	inhibitor	1.693795846312725	LANINAMIVIR OCTANOATE	drugbank:DB11888	LANINAMIVIR OCTANOATE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.011603905	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.3081436105381133	RAMUCIRUMAB	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.019490598	STANOZOLOL	rxcui:10032	STANOZOLOL	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	AXOMADOL	ncit:C72138	AXOMADOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	LAUROCAPRAM	rxcui:1603852	LAUROCAPRAM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	REL-CISAPRIDE	chembl:CHEMBL74656	REL-CISAPRIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008503267	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.192335792	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.1221108633388244	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.1376949420516464	cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.054886067	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:Q9H6Z9	hgnc:14661	EGLN3	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	FG-4592	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.2778183663264259	IUPHAR.LIGAND:4133	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.028093992	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.09741683	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.375054795	INSULIN SUSP PROTAMINE ZINC BEEF/PORK	chembl:CHEMBL1201628	INSULIN SUSP PROTAMINE ZINC BEEF/PORK	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.089222891	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	THIOTEPA	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	ALPHA-CYPERMETHRIN	chembl:CHEMBL373204	ALPHA-CYPERMETHRIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.018641225	amphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	15.00219178	dihydrostreptomycin	rxcui:1549540	DIHYDROSTREPTOMYCIN	FALSE	FALSE	FALSE
UNIPROT:Q9Y233	hgnc:21160	LINC00473	TdgClinicalTrial	Jan-14	NULL	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	1.640864726115453	Taprenepag	ncit:C152512	TAPRENEPAG	FALSE	FALSE	FALSE
HEPARANASE	hgnc:5164	HPSE	TTD	2020.06.01	NULL	0.076765601	Suramin	rxcui:10256	SURAMIN	FALSE	FALSE	FALSE
NCBIGENE:1847	hgnc:3071	DUSP5	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8123	iuphar.ligand:8123	COMPOUND 1D [PMID: 21493067]	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.00809554	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.2302968036653267	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:4766	iuphar.ligand:4766	[3H]TBZOH	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	CGI	2/1/22	NULL	0.030202859	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.093763699	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
PDGFA	hgnc:8799	PDGFA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5357925636295356	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013887244	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	OncoKB	23-Jul-20	NULL	0.3509871071904712	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.015930725	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	H3B-6545	ncit:C142980	SELECTIVE ESTROGEN RECEPTOR COVALENT ANTAGONIST H3B-6545	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1283	iuphar.ligand:1283	KISSPEPTIN-10	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005046873	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.054020238	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.064824285	eszopiclone	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1037701012563132	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.1117184494376478	AZD-4547	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	HAPLAMINE	chembl:CHEMBL1488010	HAPLAMINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.015123177	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:10136	ncit:C148147	LAZERTINIB	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:3860	rxcui:1825	BUSERELIN	TRUE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:7959	ncit:C143046	RALIMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:6045	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
NCBIGENE:1330	hgnc:2270	COX5BP1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11354	iuphar.ligand:11354	12-IMIDAZOLYL-1-DODECANOL	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1446	iuphar.ligand:1446	KOS1326	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	HYDRASTININE	chembl:CHEMBL1314044	HYDRASTININE	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2580229544751573	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	N-HISTIDYL-2-AMINONAPHTHALENE (BETANA)	chembl:CHEMBL1489988	N-HISTIDYL-2-AMINONAPHTHALENE (BETANA)	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	8-(P-SULFOPHENYL)THIOPHYLLINE	chembl:CHEMBL8488	CHEMBL:CHEMBL8488	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	GNF-PF-3889	chembl:CHEMBL598270	CHEMBL:CHEMBL598270	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.010526799	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	NAFRONYL OXALATE	ncit:C87286	NAFRONYL OXALATE	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.3763990769583835	R115777	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
NCBIGENE:611	hgnc:1012	OPN1SW	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:10186	iuphar.ligand:10186	COMPOUND 28 [HEITEL ET AL., 2019]	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MAP3K11	hgnc:6850	MAP3K11	ChEMBL	33	inhibitor	17.50255707856483	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	CIViC	10-Apr-24	NULL	0.1112450661773188	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4141	iuphar.ligand:4141	ATPO	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.069638821	IUPHAR.LIGAND:7791	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.3860858179095183	IUPHAR.LIGAND:6223	iuphar.ligand:6223	COMPOUND 3 [PMID: 21105727]	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6462	rxcui:39990	ZOFENOPRIL	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.5585922471882393	TEBANICLINE TOSYLATE	ncit:C75076	TEBANICLINE TOSYLATE	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	1.117184494376478	FGF401	chembl:CHEMBL3545293	FGF401	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:7516	iuphar.ligand:7516	COMPOUND 4D [PMID: 21851057]	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:4201	iuphar.ligand:4201	GINKGOLIDE X	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:4498	iuphar.ligand:4498	LYS[Z(NO2)]-PRO	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.019881738	Foretinib	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.044124093	LEVOMEPROMAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:P28908	hgnc:11923	TNFRSF8	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	MDX-1401	ncit:C77886	ANTI-CD30 MONOCLONAL ANTIBODY MDX-1401	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1752592497853621	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:5802	iuphar.ligand:5802	PPTN	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	CGI	2/1/22	NULL	0.3923362732430473	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
EIF2B1	hgnc:3257	EIF2B1	NCI	14-Sep-17	NULL	1.193356164447602	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.04427291	ECHINACEA	rxcui:228041	ECHINACEA PREPARATION	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.025390557	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.018385039	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.006819178	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.6250913242344582	2-(3,4-DICHLOROBENZYLIDENE)HYDRAZINECARBOXIMIDAMIDE	chembl:CHEMBL572531	CHEMBL:CHEMBL572531	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.023829213	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.038467158	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.1319288222002374	ISOSPAGLUMIC ACID	rxcui:236303	ISOSPAGLUMIC ACID	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.017578732	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	CGI	2/1/22	NULL	0.3704244884352345	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
GC	hgnc:4187	GC	NCI	14-Sep-17	NULL	0.062065805	ASA	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	3.750547945	LY-2979165	chembl:CHEMBL4303379	LY2979165	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4353	iuphar.ligand:4353	7&ALPHA;,27-DIHYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:521	hgnc:846	ATP5ME	GuideToPharmacology	2024.1	activator	3.750547945	IUPHAR.LIGAND:10337	iuphar.ligand:10337	GI‐530159	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.1446492320542548	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FLUSILAZOLE	chembl:CHEMBL1900522	FLUSILAZOLE	FALSE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	CGI	2/1/22	NULL	0.9723642821424906	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
ACP3	hgnc:125	ACP3	ChEMBL	33	binder	5.250767123569449	SIPULEUCEL-T	rxcui:997261	SIPULEUCEL-T	TRUE	FALSE	FALSE
CCNE1	hgnc:1589	CCNE1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.6563458904461812	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6482428547616604	AFURESERTIB HYDROCHLORIDE	ncit:C142902	AFURESERTIB HYDROCHLORIDE	FALSE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1041818873724097	TRICLABENDAZOLE	rxcui:2118525	TRICLABENDAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.08854582	Valbenazine	rxcui:1918219	VALBENAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.012945678	colchicine	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:9790	iuphar.ligand:9790	PIM447	FALSE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	CGI	2/1/22	NULL	3.125456621172291	Abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.2282942227638891	PH-797804	drugbank:DB07941	PH-797804	FALSE	FALSE	FALSE
RPL27A	hgnc:10329	RPL27A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01495945	FLECAINIDE ACETATE	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	1.29648571	FOSCARNET	rxcui:33562	FOSCARNET	TRUE	FALSE	FALSE
GSTA1	hgnc:4626	GSTA1	PharmGKB	4/5/24	NULL	0.1944728564284981	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.2778183663264259	HM61713	ncit:C101791	OLMUTINIB	FALSE	FALSE	TRUE
TANC2	hgnc:30212	TANC2	PharmGKB	4/5/24	NULL	11.66837138570989	calcium channel blockers	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:9174	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2160809515872201	AGI-5198	iuphar.ligand:9240	AGI-5198	FALSE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.072424374	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.1426838892274307	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1905904582057876	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.1286952726365061	Umeclidinium	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	SJ000032081	chembl:CHEMBL590184	CHEMBL:CHEMBL590184	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.008481291	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	1.750255707856483	RO5520985	ncit:C118578	VANUCIZUMAB	FALSE	FALSE	FALSE
STAT4	hgnc:11365	STAT4	NCI	14-Sep-17	NULL	17.50255707856483	INTERLEUKIN-12	rxcui:1309680	INTERLEUKIN-12	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	CGI	2/1/22	NULL	0.024896952	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	4.039051633514961	SOPHORAFLAVANONE G	chembl:CHEMBL243148	SOPHORAFLAVANONE G	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	S-(2,4-DICHLOROBENZYL)ISOTHIOUREA HYDROBROMIDE	chembl:CHEMBL1224483	CHEMBL:CHEMBL1224483	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	PharmGKB	4/5/24	NULL	0.054271495	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.1056492378987816	ERGOTAMINE TARTRATE	rxcui:42676	ERGOTAMINE TARTRATE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
UNIPROT:P48443	hgnc:10479	RXRG	TEND	1-Aug-11	NULL	0.1049104320393496	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	CGI	2/1/22	NULL	0.5173169579871378	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
KCNK2	hgnc:6277	KCNK2	DTC	9/2/20	NULL	15.00219178	AG-30	chembl:CHEMBL73820	CHEMBL:CHEMBL73820	FALSE	FALSE	FALSE
FOLLICLE-STIMULATING HORMONE RECEPTOR	hgnc:3969	FSHR	TTD	2020.06.01	NULL	18.37768493249307	Menotropins	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	SALAGEN	chembl:CHEMBL611494	SALAGEN	FALSE	FALSE	FALSE
UNIPROT:P05230	hgnc:3665	FGF1	TdgClinicalTrial	Jan-14	NULL	2.333674277141978	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.9723642821424906	NAV5001	chembl:CHEMBL4297407	ALTROPANE I-123	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	CGI	2/1/22	NULL	0.012486961	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	ChEMBL	33	inhibitor	1.400204566285186	LENZILUMAB	ncit:C125081	LENZILUMAB	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.1750255707856483	TRYPTANTHRIN	iuphar.ligand:8224	TRYPTANTHRIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	TRICLOCARBAN	rxcui:38609	TRICLOCARBAN	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.008275441	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.2536602475154323	Tipifarnib	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
CCND1	hgnc:1582	CCND1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.02232469	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.2363572458670459	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
PRKG2	hgnc:9416	PRKG2	DTC	9/2/20	NULL	0.5966780822238011	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.1411496538593938	CYPROHEPTADINE HYDROCHLORIDE	rxcui:104592	CYPROHEPTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE CHK2	hgnc:16627	CHEK2	TTD	2020.06.01	NULL	1.544343271638073	XL844	drugbank:DB05149	XL844	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.3	hgnc:10590	SCN3A	TTD	2020.06.01	NULL	0.1750255707856483	LIDOFLAZINE	rxcui:6390	LIDOFLAZINE	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	2.500365296937833	META-IODOBENZYLGUANIDINE	rxcui:14448	3-IODOBENZYLGUANIDINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	AROMOLINE	chembl:CHEMBL509999	AROMOLINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.1132444383228493	TOREMIFENE CITRATE	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1400204566285186	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.025489161	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.069180068	THIOTHIXENE	rxcui:10510	THIOTHIXENE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	GNF-PF-2243	chembl:CHEMBL600908	CHEMBL:CHEMBL600908	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.031612084	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.049349315	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.012591768	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.066297565	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.007012242	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665850	chembl:CHEMBL580159	CHEMBL:CHEMBL580159	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	4.922594178346359	AVANAFIL	rxcui:1291301	AVANAFIL	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.052824619	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:12337	iuphar.ligand:12337	COMPOUND 16D [PMID: 36573286]	FALSE	FALSE	FALSE
NCBIGENE:2757	hgnc:23177	KEAP1	GuideToPharmacology	2024.1	NULL	2.100306849	IUPHAR.LIGAND:9710	iuphar.ligand:9710	CPUY192018	FALSE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	1.312691780892362	BENZPHETAMINE HYDROCHLORIDE	rxcui:142425	BENZPHETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.033658764	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	PharmGKB	4/5/24	NULL	0.045421861	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.081872668	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.1486416737033106	Paricalcitol	rxcui:73710	PARICALCITOL	TRUE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	0.5966780822238011	SILDENAFIL CITRATE	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	ChEMBL	33	inhibitor	0.5000730593875666	LGH-447	drugbank:DB14943	LGH-447	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1861974157294131	OXYPHENONIUM BROMIDE	rxcui:42833	OXYPHENONIUM BROMIDE	TRUE	FALSE	FALSE
STS	hgnc:11425	STS	ChEMBL	33	inhibitor	7.001022831425932	IROSUSTAT	ncit:C79827	IROSUSTAT	FALSE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.7001022831425934	PENTAERYTHRITOL TETRANITRATE	rxcui:7992	PENTAERYTHRITOL TETRANITRATE	TRUE	FALSE	FALSE
F7	hgnc:3544	F7	ChEMBL	33	positive modulator	0.6250913242344582	EPTACOG ALFA (ACTIVATED)	chembl:CHEMBL2108334	EPTACOG ALFA (ACTIVATED)	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.010346339	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.067751834	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1562728310586145	HYDROXYPROGESTERONE CAPROATE	rxcui:12488	HYDROXYPROGESTERONE CAPROATE (USP)	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	3-PHENYLUMBELLIFERONE	chembl:CHEMBL153505	CHEMBL:CHEMBL153505	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.04726163	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	TCMDC-125578	chembl:CHEMBL195350	CHEMBL:CHEMBL195350	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1278595890479573	FLUOXETINE HYDROCHLORIDE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ANKS1B	hgnc:24600	ANKS1B	PharmGKB	4/5/24	NULL	3.281729452230906	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:12421	drugbank:DB18303	DEUCRICTIBANT	FALSE	FALSE	FALSE
NCBIGENE:1213	hgnc:2092	CLTC	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:4840	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.2734774543525755	DUAL IGF-1R/INSR INHIBITOR BMS-754807	ncit:C74043	DUAL IGF-1R/INSR INHIBITOR BMS-754807	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.006643177	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.138178082	CANERTINIB DIHYDROCHLORIDE	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	ChEMBL	33	inhibitor	3.500511415712966	PHENPROCOUMON	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	DTC	9/2/20	NULL	10.50153424713889	(+)-NEO-OLIVIL	chembl:CHEMBL464631	CHEMBL:CHEMBL464631	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.019490598	IUPHAR.LIGAND:2180	iuphar.ligand:2180	[VAL4]AVP	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.089501712	IMIPRAMINE HYDROCHLORIDE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:8107	iuphar.ligand:8107	VACTOSERTIB	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.1666910197958555	GRT-6005	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	0.046940525	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
TMSB4X	hgnc:11881	TMSB4X	PharmGKB	4/5/24	NULL	52.50767123569449	timbetasin	ncit:C166566	TIMBETASIN	FALSE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.5357925636295356	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.8334550989792777	GSK-2269557	chembl:CHEMBL3545250	GSK-2269557	FALSE	FALSE	FALSE
REN	hgnc:9958	REN	ChEMBL	33	inhibitor	2.625383561784724	SPH-3127	iuphar.ligand:12196	SITOKIREN	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.073954467	CHIR-265	iuphar.ligand:5674	CHIR-265	FALSE	FALSE	TRUE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	1.166837138570988	OGLEMILAST	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.021814571	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.021814571	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:2599	hgnc:1375	CA4	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:6828	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	agonist	0.364636606	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	2.500365296937833	IUPHAR.LIGAND:10554	iuphar.ligand:10554	SKA-111	FALSE	FALSE	FALSE
ATRIAL NATRIURETIC PEPTIDE RECEPTOR B	hgnc:7944	NPR2	TTD	2020.06.01	NULL	4.375639269641208	Chimeric natriuretic peptide	ncit:C171663	CENDERITIDE	FALSE	FALSE	FALSE
UNIPROT:P23416	hgnc:4327	GLRA2	TEND	1-Aug-11	NULL	0.8204323630577265	PICROTOXIN	rxcui:2539172	PICROTOXIN	FALSE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	ChEMBL	33	inhibitor	5.527123287967842	TERIFLUNOMIDE	rxcui:1310520	TERIFLUNOMIDE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	TTC-352	chembl:CHEMBL3763743	TTC-352	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009974862	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TAF1	hgnc:11535	TAF1	NCI	14-Sep-17	NULL	0.7001022831425933	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.074163377	FIDUXOSIN HYDROCHLORIDE	ncit:C81371	FIDUXOSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.013749063	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	0.1930429089547592	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	inhibitor	0.1930429089547592	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	0.6250913242344582	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
MOCOS	hgnc:18234	MOCOS	PharmGKB	4/5/24	NULL	5.527123287967842	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.1842374429322614	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
PSMD4	hgnc:9561	PSMD4	ChEMBL	33	inhibitor	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.014849455	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.546954909	SILODOSIN	rxcui:720825	SILODOSIN	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.1442518440541057	toremifene	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
CDK19	hgnc:19338	CDK19	DTC	9/2/20	NULL	0.067317527	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
XRCC5	hgnc:12833	XRCC5	PharmGKB	4/5/24	NULL	0.7501095890813501	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.064347636	LOXAPINE SUCCINATE	rxcui:6476	LOXAPINE SUCCINATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	OncoKB	23-Jul-20	NULL	0.2044691247495891	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	1.093909817410302	emtricitabine	rxcui:276237	EMTRICITABINE	TRUE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.095122593	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
UNIPROT:Q9UI33	hgnc:10583	SCN11A	TdgClinicalTrial	Jan-14	NULL	0.067751834	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
PTGIR	hgnc:9602	PTGIR	ChEMBL	33	agonist	3.750547945	EPOPROSTENOL SODIUM	rxcui:104463	EPOPROSTENOL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.2243917574174978	IUPHAR.LIGAND:6077	iuphar.ligand:6077	A68930	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:1896	iuphar.ligand:1896	AH6809	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.1105424657593568	IUPHAR.LIGAND:332	iuphar.ligand:332	N-BENZYL BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1853	iuphar.ligand:1853	SCH 37370	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	0.2678962818147678	IUPHAR.LIGAND:7219	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
NCBIGENE:1841	hgnc:3061	DTYMK	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8213	iuphar.ligand:8213	COMPOUND R-16 [PMID: 21967808]	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.010468037	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.096521454	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
RPS12	hgnc:10385	RPS12	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.013282993	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	TCMDC-125738	chembl:CHEMBL527585	CHEMBL:CHEMBL527585	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	NCI	14-Sep-17	NULL	0.078722146	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.049164486	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001392186	HYDROCORTISONE BUTYRATE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.7001022831425934	mesoridazine	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.014206621	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	LINCOMYCIN HYDROCHLORIDE	rxcui:82036	LINCOMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	agonist	0.8751278539282416	SAD448	chembl:CHEMBL2397751	SAD448	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.5556367326528519	ICOTINIB	ncit:C138996	ICOTINIB	FALSE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
UNIPROT:P19793	hgnc:10477	RXRA	TdgClinicalTrial	Jan-14	NULL	0.4667348554283955	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8504	iuphar.ligand:8504	COMPOUND 22E [PMID: 20167483]	FALSE	FALSE	FALSE
NCBIGENE:64	hgnc:137	ACTBP4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:811	iuphar.ligand:811	CCL21	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.013957382	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.2201579506737715	MNU	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
CELLULAR INHIBITOR OF APOPTOSIS 2	hgnc:591	BIRC3	TTD	2020.06.01	NULL	1.071585127259071	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	DNDI1417809	chembl:CHEMBL1442783	CHEMBL:CHEMBL1442783	FALSE	FALSE	FALSE
COMPLEMENT FACTOR D	hgnc:2771	CFD	TTD	2020.06.01	NULL	17.50255707856483	ACH-4471	ncit:C148181	DANICOPAN	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.4167275494896388	DEXTRAN SULFATE	rxcui:40068	DEXTRAN SULFATE	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	0.4375639269641209	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	TCMDC-125814	chembl:CHEMBL533082	CHEMBL:CHEMBL533082	FALSE	FALSE	FALSE
UNIPROT:P19793	hgnc:10477	RXRA	TEND	1-Aug-11	NULL	0.4667348554283955	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
F13A1	hgnc:3531	F13A1	PharmGKB	4/5/24	NULL	1.000146118775133	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.049723174	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
SLCO1A2	hgnc:10956	SLCO1A2	NCI	14-Sep-17	NULL	0.1988926940746004	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
CDX2	hgnc:1806	CDX2	PharmGKB	4/5/24	NULL	2.917092846427472	tegafur	rxcui:10995	URACIL	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123523	chembl:CHEMBL526981	CHEMBL:CHEMBL526981	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.020296742	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.076263865	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.061055432	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:792	iuphar.ligand:792	RO330-0802/001	FALSE	FALSE	FALSE
NCBIGENE:2096	hgnc:3463	ESAT	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8178	iuphar.ligand:8178	COMPOUND 16 [PMID: 18945615]	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.015290527	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003622218	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	SALICYLANILIDE	ncit:C84142	SALICYLANILIDE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	NCI	14-Sep-17	NULL	0.059667808	PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
NCBIGENE:756	hgnc:29	ABCA1	GuideToPharmacology	2024.1	NULL	0.5048814541893701	IUPHAR.LIGAND:9183	iuphar.ligand:9183	BIHELICAL APOA-I MIMETIC PEPTIDE 5A	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.091796628	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.028645756	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TEND	1-Aug-11	NULL	0.096264064	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	PROROXAN HYDROCHLORIDE	ncit:C84120	PROROXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
TNFRSF11B	hgnc:11909	TNFRSF11B	NCI	14-Sep-17	NULL	1.500219178	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	DNDI1417784	chembl:CHEMBL1504762	CHEMBL:CHEMBL1504762	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.072927321	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.001804015	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SE-(METHYL)SELENOCYSTEINE HCL	chembl:CHEMBL1256174	CHEMBL:CHEMBL1256174	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.1232574442152452	DNDI1318925	chembl:CHEMBL1390716	CHEMBL:CHEMBL1390716	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	CHLOROPHACINONE	chembl:CHEMBL1874081	CHLOROPHACINONE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	2.386712328895204	Amtolmetin guacil	ncit:C72142	AMTOLMETIN GUACIL	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	EP-217609	drugbank:DB18393	EP-217609	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3169	iuphar.ligand:3169	COMPOUND 5E [PMID: 17975902]	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1989	iuphar.ligand:1989	RELAXIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DIBUTYLDICHLOROSTANNANE	chembl:CHEMBL1088184	DIBUTYLDICHLOROSTANNANE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.017715139	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.1988926940746004	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.100976291	IUPHAR.LIGAND:332	iuphar.ligand:332	N-BENZYL BRUCINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	ONC201	iuphar.ligand:9978	ONC201	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.015475294	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.2059124362184098	Nisoldipine	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	2.323348284765243	RIFAXIMIN	rxcui:35619	RIFAXIMIN	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.5357925636295356	levetiracetam	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	GNF-PF-4803	chembl:CHEMBL585240	CHEMBL:CHEMBL585240	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	TCMDC-123579	chembl:CHEMBL533954	CHEMBL:CHEMBL533954	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	PharmGKB	4/5/24	NULL	0.6963882126749933	diazoxide	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.058733413	posaconazole	rxcui:282446	POSACONAZOLE	TRUE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.3088686543276147	IUPHAR.LIGAND:12424	iuphar.ligand:12424	L-TRP-TRP-TRP	FALSE	FALSE	FALSE
PLA2G10	hgnc:9029	PLA2G10	ChEMBL	33	inhibitor	5.834185692854944	VARESPLADIB METHYL	ncit:C152833	VARESPLADIB METHYL	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.035145697	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.305277158	GLUTAMINE	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004919212	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.020056406	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.6105543166941221	Apraclonidine	rxcui:14845	APRACLONIDINE	TRUE	FALSE	FALSE
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	1.531473744374423	AMG 232	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.053145416	IUPHAR.LIGAND:2367	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	0.3750547945406749	IUPHAR.LIGAND:1712	iuphar.ligand:1712	ADP	FALSE	FALSE	FALSE
NCBIGENE:2235	hgnc:3647	FECH	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:8114	drugbank:DB07149	(7S)-2-(2-AMINOPYRIMIDIN-4-YL)-7-(2-FLUOROETHYL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.065634589	Sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
EIF4H	hgnc:12741	EIF4H	DTC	9/2/20	NULL	26.25383561784724	GNF-PF-4618	chembl:CHEMBL585964	CHEMBL:CHEMBL585964	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.4118248724368196	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	L-694247	iuphar.ligand:15	L-694,247	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.2300445618212245	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.066297565	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	ISOETHARINE HYDROCHLORIDE	rxcui:102397	ISOETHARINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.017787152	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
UNIPROT:Q02750	hgnc:6840	MAP2K1	TdgClinicalTrial	Jan-14	NULL	0.2083637747448194	ARRY-300	chembl:CHEMBL3545359	ARRY-300	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.089222891	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.2734774543525755	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.009678833	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	SJ000027778	chembl:CHEMBL592588	CHEMBL:CHEMBL592588	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	SECURININE	ncit:C81359	SECURININE	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9999	iuphar.ligand:9999	MRS4478	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	FDA	10-Apr-24	NULL	0.071471422	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TEND	1-Aug-11	NULL	0.9723642821424906	FLUVASTATIN	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
UNIPROT:P14410	hgnc:10856	SI	TEND	1-Aug-11	NULL	2.187819634820604	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
NUBPL	hgnc:20278	NUBPL	PharmGKB	4/5/24	NULL	5.000730593875666	iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.025489161	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	ARTEANNUIN B	chembl:CHEMBL515516	ARTEANNUIN B	FALSE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	0.051177067	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.009008007	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.002768954	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.084146909	levomilnacipran	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	1.280674908	SAF312	chembl:CHEMBL3544953	SAF312	FALSE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	ChEMBL	33	inhibitor	5.250767123569449	KAI-1678	drugbank:DB16211	KAI-1678	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.033701971	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	DEXFENFLURAMINE	rxcui:3268	DEXFENFLURAMINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.082559232	IUPHAR.LIGAND:7170	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DINITRAMINE	chembl:CHEMBL1223066	DINITRAMINE	FALSE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.100976291	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
COAGULATION FACTOR VA	hgnc:3542	F5	TTD	2020.06.01	NULL	1.179947668217853	Drotrecogin alfa	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
RPE65	hgnc:10294	RPE65	ChEMBL	33	positive modulator	15.00219178	VORETIGENE NEPARVOVEC	rxcui:1995537	VORETIGENE NEPARVOVEC	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.062509132	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
UNIPROT:P10826	hgnc:9865	RARB	TdgClinicalTrial	Jan-14	NULL	0.1187956362798518	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
UNIPROT:P10599	hgnc:12435	TXN	TdgClinicalTrial	Jan-14	NULL	39.38075342677087	PX-12	drugbank:DB05448	PX-12	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	1.250182648468916	TESTOSTERONE ENANTHATE	rxcui:37859	TESTOSTERONE ENANTHATE	TRUE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TEND	1-Aug-11	NULL	1.029066006546944	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	L-165041	drugbank:DB08078	{4-[3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPOXY]PHENOXY}ACETIC ACID	FALSE	FALSE	FALSE
RPS18	hgnc:10401	RPS18	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.04636439	AZD7648	iuphar.ligand:10601	AZD7648	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	4.286340509036285	Clazakizumab	ncit:C82359	CLAZAKIZUMAB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	5-BENZYLOXYTRYPTAMINE	iuphar.ligand:265	5-BENZYLOXYTRYPTAMINE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	0.04525223	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.009869863	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.079557078	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
KCNA7	hgnc:6226	KCNA7	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	JI-101	chembl:CHEMBL3545155	JI-101	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.8255923150266431	GANITUMAB	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
RPS9	hgnc:10442	RPS9	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1132444383228493	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8627	iuphar.ligand:8627	COMPOUND 1B [PMID: 18078750]	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.061992528	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PRKG1	hgnc:9414	PRKG1	DTC	9/2/20	NULL	0.1084869240406911	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TEND	1-Aug-11	NULL	0.063072278	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	10.50153424713889	PF-04457845	drugbank:DB12012	PF-04457845	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	TDR78834	chembl:CHEMBL1507526	CHEMBL:CHEMBL1507526	FALSE	FALSE	FALSE
LMO2	hgnc:6642	LMO2	NCI	14-Sep-17	NULL	2.500365296937833	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.2812910959055062	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	CIViC	10-Apr-24	NULL	0.1909369863116163	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	1.419126249613364	BXT-51072	chembl:CHEMBL4297259	ALT-2074	FALSE	FALSE	FALSE
RPS3	hgnc:10420	RPS3	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:7887	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:2603	hgnc:2861	DHFR	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:7162	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:10456	iuphar.ligand:10456	ZORIFERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1274	hgnc:4855	HDC	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:5134	iuphar.ligand:5134	AMA	FALSE	FALSE	FALSE
NCBIGENE:2884	hgnc:4561	GPX1P2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9240	iuphar.ligand:9240	AGI-5198	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	R-N-PROPYLNORAPOMORPHINE	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	OTILONIUM	rxcui:32311	OCTYLONIUM	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:4050	iuphar.ligand:4050	2-FUROYL-LIGRL[N-(ALEXA FLUOR 594)-O]-NH2	FALSE	FALSE	FALSE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:6824	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	0.4167275494896388	GERONTOXANTHONE H	chembl:CHEMBL514057	GERONTOXANTHONE H	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1458546423213736	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.068637479	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	NCI	14-Sep-17	NULL	0.3409589041278864	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.3409589041278864	ABACAVIR	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.9460841664089098	QUERCETAGETIN	chembl:CHEMBL413552	QUERCETAGETIN	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.3314878234576672	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	LXH 254	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	DIPYRITHIONE	rxcui:1362743	DIPYRITHIONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.1319288222002374	DEXPROPRANOLOL HYDROCHLORIDE	ncit:C77945	DEXPROPRANOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.037042449	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CYTOTOXIC T-LYMPHOCYTE PROTEIN 4	hgnc:2505	CTLA4	TTD	2020.06.01	NULL	1.750255707856483	AGEN1884	ncit:C126113	ZALIFRELIMAB	FALSE	FALSE	FALSE
HNMT	hgnc:5028	HNMT	DTC	9/2/20	NULL	1.666910197958555	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.2792961235941196	GNF-PF-4097	chembl:CHEMBL597246	CHEMBL:CHEMBL597246	FALSE	FALSE	FALSE
NA	hgnc:12811	XK	ChEMBL	33	inhibitor	0.8468979231563628	OSELTAMIVIR PHOSPHATE	rxcui:259275	OSELTAMIVIR PHOSPHATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1103102336884338	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.042174836	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.038159645	IUPHAR.LIGAND:2404	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
KCNS2	hgnc:6301	KCNS2	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
UNIPROT:Q9UM47	hgnc:7883	NOTCH3	TdgClinicalTrial	Jan-14	NULL	21.00306849427779	OMP-59R5	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
NCBIGENE:82	hgnc:154	ACTG1P9	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:3422	iuphar.ligand:3422	CHEMERIN C-TERMINAL PEPTIDE	FALSE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	0.2625383561784725	(-)-Phenserine	drugbank:DB04892	PHENSERINE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	XCT790	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	2.917092846427472	RHTPO	ncit:C878	RECOMBINANT HUMAN THROMBOPOIETIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.034453853	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
SERINE PROTEASE UNSPECIFIC	hgnc:11756	TFF2	TTD	2020.06.01	NULL	4.375639269641208	Sivelestat sodium hydrate	chembl:CHEMBL3182314	SIVELESTAT SODIUM	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	DOMOIC ACID	drugbank:DB02852	DOMOIC ACID	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.42006137	MMF	rxcui:1546433	MONOMETHYL FUMARATE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	CGI	2/1/22	NULL	0.1219690388750162	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CD69	hgnc:1694	CD69	CGI	2/1/22	NULL	2.917092846427472	Bendamustine	rxcui:134547	BENDAMUSTINE	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	CGI	2/1/22	NULL	0.4735986033023426	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
ERBB3	hgnc:3431	ERBB3	CGI	2/1/22	NULL	0.1660584163051692	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.2044691247495891	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	CGI	2/1/22	NULL	0.095295229	Afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CGI	2/1/22	NULL	0.042793538	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	CGI	2/1/22	NULL	0.053145416	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1773907812016706	CLIDINIUM BROMIDE	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	1.514644363	BRINZOLAMIDE	rxcui:194881	BRINZOLAMIDE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	1.848379561100067	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	ChEMBL	33	inhibitor	2.625383561784724	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	3.938075342677087	MARAVIROC	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.079718124	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	1.500219178	INSULIN DETEMIR	rxcui:139825	INSULIN DETEMIR	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.100976291	LOXAPINE HYDROCHLORIDE	rxcui:91138	LOXAPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN SUSP ISOPHANE PURIFIED BEEF	chembl:CHEMBL1201655	INSULIN SUSP ISOPHANE PURIFIED BEEF	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.8078103267029922	LEVOBUPIVACAINE HYDROCHLORIDE	rxcui:259454	LEVOBUPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.4907258993990139	BETHANIDINE SULFATE	rxcui:81966	BETHANIDINE SULFATE	TRUE	FALSE	FALSE
CLCN2	hgnc:2020	CLCN2	ChEMBL	33	potentiator	35.00511415712966	LUBIPROSTONE	rxcui:623033	LUBIPROSTONE	TRUE	FALSE	FALSE
NPR1	hgnc:7943	NPR1	ChEMBL	33	agonist	4.039051633514961	NESIRITIDE	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	ChEMBL	33	inhibitor	0.6563458904461812	DOXYCYCLINE CALCIUM	rxcui:82012	DOXYCYCLINE CALCIUM	TRUE	FALSE	FALSE
MMP7	hgnc:7174	MMP7	ChEMBL	33	inhibitor	1.875273972703375	DOXYCYCLINE CALCIUM	rxcui:82012	DOXYCYCLINE CALCIUM	TRUE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	ChEMBL	33	inhibitor	3.500511415712966	RISEDRONATE SODIUM	rxcui:1926958	RISEDRONATE SODIUM ANHYDROUS	TRUE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	2.250328767244049	AMBRISENTAN	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	ChEMBL	33	inhibitor	2.045753424767318	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.03849536	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.035574303	BRENTUXIMAB VEDOTIN	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.007531221	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.021087418	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	negative modulator	0.3571950424196904	MEMANTINE HYDROCHLORIDE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	negative modulator	0.4227670791923872	MEMANTINE HYDROCHLORIDE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.085239726	GUANFACINE HYDROCHLORIDE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.055504938	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.067231333	GUANFACINE HYDROCHLORIDE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.2812910959055062	KETOPROFEN	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.068369364	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2035181055647073	METIPRANOLOL HYDROCHLORIDE	rxcui:314731	METIPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
PSMA2	hgnc:9531	PSMA2	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB3	hgnc:9540	PSMB3	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.4167275494896388	METOCURINE IODIDE	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.4605936073306534	ROCURONIUM BROMIDE	rxcui:32521	ROCURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.5000730593875667	TUBOCURARINE CHLORIDE	rxcui:82115	TUBOCURARINE CHLORIDE	TRUE	FALSE	FALSE
ATP1A1	hgnc:799	ATP1A1	ChEMBL	33	inhibitor	0.3088686543276147	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
ATP1A2	hgnc:800	ATP1A2	ChEMBL	33	inhibitor	0.2206204673768676	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
ATP1B3	hgnc:806	ATP1B3	ChEMBL	33	inhibitor	0.8751278539282418	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.055504938	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.083257407	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.080781033	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.079758488	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.017444409	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.020273232	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.017363648	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.015498132	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.027752469	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.014553124	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.015299438	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	OXYTETRACYCLINE CALCIUM	rxcui:82065	OXYTETRACYCLINE CALCIUM	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.096167896	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	blocker	0.2243917574174979	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNK10	hgnc:6273	KCNK10	ChEMBL	33	potentiator	0.2917092846427472	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.038049037	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.036237178	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.043180651	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.018359326	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.043180651	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.019889269	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.071439008	BROMOCRIPTINE MESYLATE	rxcui:142426	BROMOCRIPTINE MESYLATE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inverse agonist	0.008128122	HALOPERIDOL DECANOATE	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.1071585127259071	LEVOMEPROMAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inverse agonist	0.008128122	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.021301287	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	ChEMBL	33	blocker	0.072927321	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNG3	hgnc:18306	KCNG3	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNC2	hgnc:6234	KCNC2	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNG4	hgnc:19697	KCNG4	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNA4	hgnc:6222	KCNA4	ChEMBL	33	blocker	0.1562728310586145	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	blocker	0.060772768	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	blocker	0.1093909817410302	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNV2	hgnc:19698	KCNV2	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNH8	hgnc:18864	KCNH8	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNH1	hgnc:6250	KCNH1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.1037701012563132	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	agonist	0.1469979597863787	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.088945801	BREXPIPRAZOLE	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	3.281729452230906	DAPAGLIFLOZIN PROPYLENE GLYCOL	chembl:CHEMBL2103802	DAPAGLIFLOZIN PROPYLENE GLYCOL	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.3125456621172291	COBIMETINIB FUMARATE	rxcui:1722380	COBIMETINIB FUMARATE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.092443083	CM-082	chembl:CHEMBL3545427	CM-082	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.079376676	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.2273059360852575	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.1829535583125243	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1346350544504987	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.080781033	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.018488617	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.3241214273808302	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	1.367387271762877	LAROTRECTINIB	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
PIM2	hgnc:8987	PIM2	ChEMBL	33	inhibitor	4.375639269641208	LGH-447	drugbank:DB14943	LGH-447	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	ChEMBL	33	inhibitor	2.838252499226729	LY-2584702	drugbank:DB12690	LY-2584702	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.084146909	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.5498185469706229	RG-7256	chembl:CHEMBL3545080	RG-7256	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.075768645	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1363835616511545	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	ChEMBL	33	inhibitor	2.500365296937833	TOLCAPONE	rxcui:72937	TOLCAPONE	TRUE	FALSE	FALSE
FGR	hgnc:3697	FGR	ChEMBL	33	inhibitor	0.2083637747448194	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	ChEMBL	33	inhibitor	0.2083637747448194	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1875273972703375	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	8.751278539282415	TAK-441	iuphar.ligand:8200	TAK-441	FALSE	FALSE	FALSE
SRMS	hgnc:11298	SRMS	ChEMBL	33	inhibitor	0.546954909	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	ChEMBL	33	inhibitor	0.1041818873724097	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.06970816	TRIAMCINOLONE ACETONIDE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
GRM3	hgnc:4595	GRM3	ChEMBL	33	agonist	2.625383561784724	LY2969822	chembl:CHEMBL3545270	LY2969822	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.2917092846427472	AZD6280	chembl:CHEMBL1783256	AZD6280	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.6908904109959803	DSP-2230	chembl:CHEMBL5095026	DSP-2230	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.082429625	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1099061668983662	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.041214813	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.750109589	BMS-777607	drugbank:DB12064	BMS-777607	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1008469998124734	CABOZANTINIB S-MALATE	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.040703621	LUCITANIB	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.08334551	LUCITANIB	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	2.561349816375341	NGD-8243	chembl:CHEMBL3545227	NGD-8243	FALSE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	2.917092846427472	LESOGABERAN	ncit:C166751	LESOGABERAN	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	2.625383561784724	INCB-9471	drugbank:DB12960	INCB-9471	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	2.072671233	VIDUPIPRANT	ncit:C152874	VIDUPIPRANT	FALSE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	ChEMBL	33	inhibitor	1.810609352954982	RUPLIZUMAB	ncit:C152273	RUPLIZUMAB	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.06970816	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.034544521	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	BETAMETHASONE VALERATE	rxcui:227897	BETAMETHASONE VALERATE	TRUE	FALSE	FALSE
MAP3K13	hgnc:6852	MAP3K13	ChEMBL	33	inhibitor	5.834185692854945	CEP-1347	drugbank:DB05403	CEP-1347	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.6168664383892681	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.025827679	TAMOXIFEN CITRATE	rxcui:40137	TAMOXIFEN CITRATE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.020542907	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PRKD1	hgnc:9407	PRKD1	ChEMBL	33	inhibitor	0.1458546423213736	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PRKCA	hgnc:9393	PRKCA	ChEMBL	33	inhibitor	0.1215455352678113	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	2.917092846427472	ANAMORELIN HYDROCHLORIDE	ncit:C72701	ANAMORELIN HYDROCHLORIDE	FALSE	FALSE	FALSE
TACR2	hgnc:11527	TACR2	ChEMBL	33	inhibitor	10.50153424713889	IBODUTANT	ncit:C166502	IBODUTANT	FALSE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	1.500219178	RITOBEGRON	ncit:C87677	RITOBEGRON	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.4773424657790409	RILPIVIRINE HYDROCHLORIDE	rxcui:1102270	RILPIVIRINE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.2386712328895204	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.2300445618212245	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.2263261691193728	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	modulator	1.250182648468916	MIROGABALIN BESYLATE	ncit:C175142	MIROGABALIN BESYLATE	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.3409589041278864	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.1193356164447602	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	binder	2.423430980108977	BAPINEUZUMAB	ncit:C79569	BAPINEUZUMAB	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	agonist	0.05309168	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
PAGA	hgnc:9352	PRDX1	ChEMBL	33	binder	8.751278539282415	OBILTOXAXIMAB	rxcui:1746906	OBILTOXAXIMAB	TRUE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	ChEMBL	33	blocker	0.087512785	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNC1	hgnc:6233	KCNC1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	0.4167275494896388	DEFIBROTIDE SODIUM	rxcui:1311089	DEFIBROTIDE	TRUE	FALSE	FALSE
KCNC2	hgnc:6234	KCNC2	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.1562728310586145	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNG2	hgnc:6249	KCNG2	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN PEGLISPRO	ncit:C166970	INSULIN PEGLISPRO	FALSE	FALSE	FALSE
KCNH6	hgnc:18862	KCNH6	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.1084869240406911	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.729273212	ESOMEPRAZOLE MAGNESIUM	rxcui:283562	ESOMEPRAZOLE MAGNESIUM	TRUE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	0.1367387271762877	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	ChEMBL	33	inhibitor	9.723642821424907	FICLATUZUMAB	ncit:C78844	FICLATUZUMAB	FALSE	TRUE	TRUE
NCAM1	hgnc:7656	NCAM1	ChEMBL	33	binder	1.640864726115453	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	binder	2.423430980108977	PONEZUMAB	ncit:C97941	PONEZUMAB	FALSE	FALSE	FALSE
DLL4	hgnc:2910	DLL4	ChEMBL	33	inhibitor	31.50460274141669	DEMCIZUMAB	ncit:C80041	DEMCIZUMAB	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	inhibitor	0.3889457128569962	NALMEFENE HYDROCHLORIDE	rxcui:236069	NALMEFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	ChEMBL	33	agonist	0.3500511415712966	CARBETAPENTANE CITRATE	rxcui:283547	CARBETAPENTANE CITRATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	CLOMETACIN	ncit:C77348	CLOMETACIN	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.027752469	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.030996264	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.087318744	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.1081888830405793	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.029465584	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.4861821410712453	PYROVALERONE HYDROCHLORIDE	ncit:C73830	PYROVALERONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.4773424657790409	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	DULIGOTUZUMAB	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	2.561349816375341	DENINTUZUMAB MAFODOTIN	ncit:C105150	DENINTUZUMAB MAFODOTIN	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	ALOXIPRIN	rxcui:17393	ALOXIPRIN	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.029170928	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
DRD5	hgnc:3026	DRD5	ChEMBL	33	inhibitor	0.077217164	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
IFNA17	hgnc:5422	IFNA17	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
IFNA21	hgnc:5424	IFNA21	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
IFNA7	hgnc:5428	IFNA7	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
IL6R	hgnc:6019	IL6R	ChEMBL	33	inhibitor	4.039051633514961	VOBARILIZUMAB	ncit:C152901	VOBARILIZUMAB	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.080781033	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPS27	hgnc:10416	RPS27	ChEMBL	33	inhibitor	0.093763699	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS12	hgnc:10385	RPS12	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL3	hgnc:10332	RPL3	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL21	hgnc:10313	RPL21	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL14	hgnc:10305	RPL14	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.091159151	TERAZOSIN HYDROCHLORIDE	rxcui:235224	TERAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPL19	hgnc:10312	RPL19	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	ChEMBL	33	inhibitor	0.2983390411119005	APOLIZUMAB	ncit:C2228	APOLIZUMAB	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.063110182	CARVEDILOL PHOSPHATE	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
RPLP1	hgnc:10372	RPLP1	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
KCNA7	hgnc:6226	KCNA7	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.003561774	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	blocker	0.1250182648468916	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.02926849	CARVEDILOL PHOSPHATE	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
KCNB2	hgnc:6232	KCNB2	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNS3	hgnc:6302	KCNS3	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNV1	hgnc:18861	KCNV1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNA3	hgnc:6221	KCNA3	ChEMBL	33	blocker	0.1785975212098452	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	ChEMBL	33	blocker	0.08334551	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.2333674277141978	RAMOSETRON HYDROCHLORIDE	ncit:C88299	RAMOSETRON HYDROCHLORIDE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPS7	hgnc:10440	RPS7	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.1346350544504987	TERAZOSIN HYDROCHLORIDE	rxcui:235224	TERAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPL10	hgnc:10298	RPL10	ChEMBL	33	inhibitor	0.092118721	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL19	hgnc:10312	RPL19	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL22	hgnc:10315	RPL22	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS29	hgnc:10419	RPS29	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL4	hgnc:10353	RPL4	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
FAU	hgnc:3597	FAU	ChEMBL	33	inhibitor	0.055271233	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.048958202	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
PDE7A	hgnc:8791	PDE7A	ChEMBL	33	inhibitor	1.312691780892362	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.1646008502686348	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
GP	hgnc:18280	RNF130	ChEMBL	33	binder	7.501095891	ANSUVIMAB	rxcui:2472151	ANSUVIMAB-ZYKL	TRUE	FALSE	FALSE
PA	hgnc:8549	BLOC1S6	ChEMBL	33	inhibitor	8.751278539282415	FAVIPIRAVIR	ncit:C81605	FAVIPIRAVIR	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.073540156	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.2075402025126264	SUMANIROLE	ncit:C76651	SUMANIROLE	FALSE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	1.458546423213736	SODIUM OXYBATE	rxcui:9899	SODIUM OXYBATE	TRUE	FALSE	FALSE
EPHX2	hgnc:3402	EPHX2	ChEMBL	33	inhibitor	1.500219178	GSK2256294	iuphar.ligand:9718	GSK2256294	FALSE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	ChEMBL	33	inhibitor	4.565884455277782	RESATORVID	ncit:C87682	RESATORVID	FALSE	FALSE	FALSE
LGALS3	hgnc:6563	LGALS3	ChEMBL	33	inhibitor	13.12691780892362	OLITIGALTIN	ncit:C174126	OLITIGALTIN	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	ChEMBL	33	inhibitor	1.250182648468916	NEBICAPONE	ncit:C83923	NEBICAPONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.058471794	ETHYLESTRENOL	rxcui:4162	ETHYLESTRENOL	TRUE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	ChEMBL	33	inhibitor	1.810609352954982	RAVAGALIMAB	ncit:C170363	RAVAGALIMAB	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	DOVRAMILAST	ncit:C189964	DOVRAMILAST	FALSE	FALSE	FALSE
ICOS	hgnc:5351	ICOS	ChEMBL	33	agonist	17.50255707856483	FELADILIMAB	ncit:C126804	FELADILIMAB	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2917092846427472	DOVRAMILAST	ncit:C189964	DOVRAMILAST	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.3125456621172291	LOTAMILAST	ncit:C170131	LOTAMILAST	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2983390411119005	TRANIMILAST	ncit:C171863	TRANIMILAST	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.116943588	OXANDROLONE	rxcui:7779	OXANDROLONE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	ChEMBL	33	inhibitor	1.029562181092049	LUTIKIZUMAB	ncit:C166465	LUTIKIZUMAB	FALSE	FALSE	FALSE
RPS6	hgnc:10429	RPS6	ChEMBL	33	modulator	0.1067229090156392	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS17	hgnc:10397	RPS17	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS13	hgnc:10386	RPS13	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	2.386712328895204	MILRINONE LACTATE	rxcui:155120	MILRINONE LACTATE	TRUE	FALSE	FALSE
RPL11	hgnc:10301	RPL11	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL13A	hgnc:10304	RPL13A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL18	hgnc:10310	RPL18	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
FAU	hgnc:3597	FAU	ChEMBL	33	modulator	0.064033745	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL18A	hgnc:10311	RPL18A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL23A	hgnc:10317	RPL23A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS28	hgnc:10418	RPS28	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL15	hgnc:10306	RPL15	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL37	hgnc:10347	RPL37	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL39	hgnc:10350	RPL39	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
CD86	hgnc:1705	CD86	ChEMBL	33	inhibitor	2.333674277141978	BELATACEPT	rxcui:1112973	BELATACEPT	TRUE	FALSE	FALSE
RPL36	hgnc:13631	RPL36	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL37A	hgnc:10348	RPL37A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.078136416	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.3684748858645228	FESOTERODINE FUMARATE	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	agonist	7.876150685354174	AZD-8848	drugbank:DB14868	AZD-8848	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.3241214273808302	BICIFADINE	ncit:C79930	BICIFADINE	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	4.861821410712453	TOSITUMOMAB	rxcui:263010	TOSITUMOMAB	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.3387591692625452	GUSACITINIB	ncit:C166736	GUSACITINIB	FALSE	FALSE	FALSE
UGCG	hgnc:12524	UGCG	ChEMBL	33	inhibitor	5.250767123569449	LUCERASTAT	ncit:C170135	LUCERASTAT	FALSE	FALSE	FALSE
P2RX7	hgnc:8537	P2RX7	ChEMBL	33	inhibitor	17.50255707856483	JNJ-54175446	drugbank:DB15358	JNJ-54175446	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.8899605294185507	FIMASARTAN	ncit:C81417	FIMASARTAN	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	2.763561643983921	BI-671800	drugbank:DB12524	BI-671800	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	3.500511415712966	OLENDALIZUMAB	ncit:C118441	OLENDALIZUMAB	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	TISLELIZUMAB	rxcui:2677426	TISLELIZUMAB	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	ChEMBL	33	inhibitor	1.250182648468916	TILARGININE ACETATE	ncit:C90899	TILARGININE ACETATE	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.101562227	FUTIBATINIB	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	negative modulator	0.039538909	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	negative modulator	0.040021091	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
ENPP3	hgnc:3358	ENPP3	ChEMBL	33	binder	3.281729452230906	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	negative modulator	0.033487035	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	agonist	0.8751278539282416	EFINOPEGDUTIDE	ncit:C169932	EFINOPEGDUTIDE	FALSE	FALSE	FALSE
E2F4	hgnc:3118	E2F4	ChEMBL	33	inhibitor	1.640864726115453	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
SLC6A9	hgnc:11056	SLC6A9	ChEMBL	33	inhibitor	11.66837138570988	ORG-25935	drugbank:DB12220	ORG-25935	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.4123639102279672	BELVARAFENIB	ncit:C121646	BELVARAFENIB	FALSE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.078958904	CHIGLITAZAR	iuphar.ligand:12287	CHIGLITAZAR	FALSE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.7501095890813501	PIPECURONIUM BROMIDE	rxcui:66983	PIPECURONIUM BROMIDE	TRUE	FALSE	FALSE
ENPP2	hgnc:3357	ENPP2	ChEMBL	33	inhibitor	4.375639269641208	ZIRITAXESTAT	ncit:C170396	ZIRITAXESTAT	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.8468979231563628	TALAMPANEL	ncit:C38139	TALAMPANEL	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.082171629	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	ChEMBL	33	positive modulator	1.381780822	FIDANACOGENE ELAPARVOVEC	ncit:C171800	FIDANACOGENE ELAPARVOVEC	FALSE	FALSE	FALSE
IL21	hgnc:6005	IL21	ChEMBL	33	binder	17.50255707856483	NNC0114-0006	drugbank:DB18361	NNC0114-0006	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1259176768242074	UMBRALISIB TOSYLATE	rxcui:2478438	UMBRALISIB TOSYLATE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	REPROTEROL	rxcui:35373	REPROTEROL	TRUE	FALSE	FALSE
MYL7	hgnc:21719	MYL7	ChEMBL	33	inhibitor	1.944728564284981	MAVACAMTEN	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
MYH6	hgnc:7576	MYH6	ChEMBL	33	inhibitor	1.944728564284981	MAVACAMTEN	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	ChEMBL	33	inhibitor	0.8204323630577265	PEMETREXED TROMETHAMINE	ncit:C170306	PEMETREXED TROMETHAMINE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.007276562	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.019261802	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2332563532602643	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1196983386831941	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3309307010653015	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
ATR	hgnc:882	ATR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1250182648468916	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.060772768	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
CCNE1	hgnc:1589	CCNE1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1875273972703374	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.072125922	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
MYC	hgnc:7553	MYC	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.016669102	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.095500063	PF-05212384	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
NF1	hgnc:7765	NF1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2536602475154323	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
AKT3	hgnc:393	AKT3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.546954909	AFURESERTIB HYDROCHLORIDE	ncit:C142902	AFURESERTIB HYDROCHLORIDE	FALSE	FALSE	TRUE
ACVRL1	hgnc:175	ACVRL1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	2.917092846427472	DALANTERCEPT	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.192335792	PF-05212384	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6141248097742047	CS1229	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.5000730593875667	PIPECURONIUM BROMIDE	rxcui:66983	PIPECURONIUM BROMIDE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4167275494896388	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.09699693	PAZOPANI	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4296082192011368	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.375054795	MEK164	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1620607136904151	SIBUTRAMINE HYDROCHLORIDE	rxcui:1294535	SIBUTRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.073437302	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
VEGFC	hgnc:12682	VEGFC	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4375639269641208	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
MET	hgnc:7029	MET	COSMIC	4-Sep-20	NULL	1.500219178	Capmatinib	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002542252	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
PDE8B	hgnc:8794	PDE8B	ChEMBL	33	inhibitor	2.187819634820604	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007232462	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.2000292237550266	PHA-665752	iuphar.ligand:5700	PHA-665752	FALSE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	3.281729452230906	TETRADECANOYL PHORBOL ACETATE	chembl:CHEMBL502495	TETRADECANOYL PHORBOL ACETATE	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.2625383561784725	TCMDC-125000	chembl:CHEMBL579742	CHEMBL:CHEMBL579742	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.011394894	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	ERGONOVINE	rxcui:4021	ERGONOVINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	QUINELORANE	ncit:C152121	QUINELORANE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	(S)-ALAPROCLATE	chembl:CHEMBL251941	(S)-ALAPROCLATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	IPRONIAZID	rxcui:5981	IPRONIAZID	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.006614723	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	MALATHION	rxcui:6606	MALATHION	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	3',4' DICHLOROBENZAMIL	iuphar.ligand:4597	3,4-DICHLOROBENZAMIL	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2117244807890907	BISMUTH SUBSALICYLATE	rxcui:19478	BISMUTH SUBSALICYLATE	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.014565235	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.2143170254518142	CLIOXANIDE	ncit:C65338	CLIOXANIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.010819631	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW784684X	chembl:CHEMBL475761	GW784684X	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.082300425	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	5-AMINOISOQUINOLINE	drugbank:DB04605	5-AMINOISOQUINOLINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	DIAZIRINE	chembl:CHEMBL592862	DIAZIRINE	FALSE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	ChEMBL	33	agonist	0.9376369863516875	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	2.500365296937833	SC-514	chembl:CHEMBL193093	CHEMBL:CHEMBL193093	FALSE	FALSE	FALSE
TXN	hgnc:12435	TXN	DTC	9/2/20	NULL	13.12691780892362	BIOTINYLATED GAMBOGIC ACID	chembl:CHEMBL2205161	BIOTINYLATED GAMBOGIC ACID	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.013336975	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	CYCLOHETERPHYLLIN	chembl:CHEMBL461820	CYCLOHETERPHYLLIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.008789366	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FURAZABOL	ncit:C65782	FURAZABOL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	TCMDC-125543	chembl:CHEMBL546170	CHEMBL:CHEMBL546170	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	6-CHLOROFLAVONE	ncit:C63698	6-CHLOROFLAVONE	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	0.048083948	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
S100A4	hgnc:10494	S100A4	DTC	9/2/20	NULL	1.591141552596803	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE	chembl:CHEMBL457504	CHEMBL:CHEMBL457504	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.00822231	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	PORFIROMYCIN	ncit:C763	PORFIROMYCIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-711237	chembl:CHEMBL408732	CHEMBL:CHEMBL408732	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.097236428	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	TDR78834	chembl:CHEMBL1507526	CHEMBL:CHEMBL1507526	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.010205573	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	DTC	9/2/20	NULL	0.2117244807890907	PYRILAMINE	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.021484317	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.036770078	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	DTC	9/2/20	NULL	0.364636606	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	THIOTEPA	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.016460085	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.020296742	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.026319635	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.025942525	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006439499	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.06714536	BUPROPION HYDROCHLORIDE	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-279835	chembl:CHEMBL2003658	CHEMBL:CHEMBL2003658	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	TRICLOCARBAN	rxcui:38609	TRICLOCARBAN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.008421439	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
HEXA	hgnc:4878	HEXA	DTC	9/2/20	NULL	5.250767123569449	N-ACETYLGLUCOSAMINE THIAZOLINE	chembl:CHEMBL257158	CHEMBL:CHEMBL257158	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	HETEROCODEINE	chembl:CHEMBL358043	HETEROCODEINE	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	2.763561643983921	C-1027	chembl:CHEMBL506048	CHEMBL:CHEMBL506048	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.010620484	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.034318739	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.015498132	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.028078969	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001670623	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	KRESOXIM-METHYL	chembl:CHEMBL203191	KRESOXIM-METHYL	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.009579944	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	chembl:CHEMBL1256180	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.044198376	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.4150804050252529	5-OH-DPAT	iuphar.ligand:128	5-OH-DPAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003053304	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	NSC-172033	chembl:CHEMBL238624	CHEMBL:CHEMBL238624	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.063645662	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	SULFOBROMOPHTHALEIN	rxcui:10212	SULFOBROMOPHTHALEIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.014765937	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.037884323	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.031051254	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	NSC-126757	chembl:CHEMBL228132	CHEMBL:CHEMBL228132	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00517674	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.023171964	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	TRYPTANTHRIN	iuphar.ligand:8224	TRYPTANTHRIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.023420014	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.2500365296937833	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	CARNOSIC ACID	chembl:CHEMBL484853	CARNOSIC ACID	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.012442576	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1750255707856483	TRIBUTYLCHLOROSTANNANE	chembl:CHEMBL1088186	TRIBUTYLCHLOROSTANNANE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TECTOQUINONE	chembl:CHEMBL21745	TECTOQUINONE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.010346339	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	DTC	9/2/20	NULL	0.4321619031744402	RO-4882224	chembl:CHEMBL1077391	CHEMBL:CHEMBL1077391	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.035098711	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	2-BFI	chembl:CHEMBL404505	CHEMBL:CHEMBL404505	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	DTC	9/2/20	NULL	0.031198854	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005483257	PROCHLORPERAZINE MALEATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PROPICONAZOLE	ncit:C97997	PROPICONAZOLE	FALSE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	0.1973972602845657	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.1640864726115453	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.093596562	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	DTC	9/2/20	NULL	0.192335792	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	MEPHOBARBITAL	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.5000730593875666	SJ000170251	chembl:CHEMBL603154	CHEMBL:CHEMBL603154	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.053145416	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
DHRS9	hgnc:16888	DHRS9	DTC	9/2/20	NULL	15.00219178	SESQUITERPENE O-BENZOQUINONE	chembl:CHEMBL517425	CHEMBL:CHEMBL517425	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.018874073	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SJ000240587	chembl:CHEMBL592834	CHEMBL:CHEMBL592834	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-4364	chembl:CHEMBL528647	CHEMBL:CHEMBL528647	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.020296742	CIANIDANOL	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.085239726	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.058931169	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.011464557	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	AG-99	chembl:CHEMBL296407	CHEMBL:CHEMBL296407	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-3107	chembl:CHEMBL602383	CHEMBL:CHEMBL602383	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	2,3,4-TRIHYDROXYBENZOPHENONE	chembl:CHEMBL1527	CHEMBL:CHEMBL1527	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.167488584	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1216662358986632	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	INDIGOTINDISULFONATE	rxcui:1426889	INDIGO	TRUE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	0.5770073762164232	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	1.029562181092049	PROTUBOXEPIN A	chembl:CHEMBL1802135	PROTUBOXEPIN A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	2.386712328895204	N-TRIFLUOROACETYLHOMOCYSTEINE THIOLACTONE	chembl:CHEMBL1945287	CHEMBL:CHEMBL1945287	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.000833098	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	KHELLIN	rxcui:6147	KHELLIN	FALSE	FALSE	FALSE
CCBL1	hgnc:1564	KYAT1	DTC	9/2/20	NULL	35.00511415712966	INDOLE-3-ACETIC ACID	chembl:CHEMBL82411	INDOLE-3-ACETIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.2476776945079929	METAPHIT METHANESULFONATE	chembl:CHEMBL1256971	METAPHIT METHANESULFONATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.035418328	ZOXAZOLAMINE	ncit:C152966	ZOXAZOLAMINE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.009995749	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.008780547	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.021951368	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.023336743	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	NAFTOPIDIL DIHYDROCHLORIDE	chembl:CHEMBL1257069	NAFTOPIDIL DIHYDROCHLORIDE	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.017047945	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.013957382	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	FIDUXOSIN HYDROCHLORIDE	ncit:C81371	FIDUXOSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.364636606	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.036212187	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	NSC-749235	chembl:CHEMBL2336666	CHEMBL:CHEMBL2336666	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.011365297	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	ORTHO-PHTHALALDEHYDE	chembl:CHEMBL160145	ORTHO-PHTHALALDEHYDE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.364636606	GNF-PF-2718	chembl:CHEMBL579143	CHEMBL:CHEMBL579143	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.015344147	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BENZOPHENONE	rxcui:18997	BENZOPHENONE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	GNF-PF-3416	chembl:CHEMBL579550	CHEMBL:CHEMBL579550	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.025651036	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	MMV006319	chembl:CHEMBL579105	CHEMBL:CHEMBL579105	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.025390557	PHENOXYBENZAMINE	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016780975	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	TCMDC-125814	chembl:CHEMBL533082	CHEMBL:CHEMBL533082	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.2917092846427472	TEROXIRONE	ncit:C2320	TEROXIRONE	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.3043922970185188	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.3977853881492007	TCMDC-123884	chembl:CHEMBL580955	CHEMBL:CHEMBL580955	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	VANITIOLIDE	ncit:C74234	VANITIOLIDE	FALSE	FALSE	FALSE
MATK	hgnc:6906	MATK	DTC	9/2/20	NULL	0.084281976	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.064984742	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.042619863	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.031880796	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	2,3,4,6-TETRACHLORO-PHENOL	chembl:CHEMBL320361	CHEMBL:CHEMBL320361	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	THIABENDAZOLE	rxcui:10450	THIABENDAZOLE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00445925	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	2,4-HEXADIENAL	chembl:CHEMBL1576086	2,4-HEXADIENAL	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.2586584789935689	PROROXAN HYDROCHLORIDE	ncit:C84120	PROROXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.004698253	PARAPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	OXETHAZAINE	ncit:C81409	OXETHAZAINE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	NSC-93401	chembl:CHEMBL452954	CHEMBL:CHEMBL452954	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.070574827	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	GNF-PF-1549	chembl:CHEMBL227959	CHEMBL:CHEMBL227959	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	TAXIFOLIN	drugbank:DB02224	TAXIFOLIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010058941	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.084553416	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
TMPRSS15	hgnc:9490	TMPRSS15	DTC	9/2/20	NULL	1.166837138570989	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.01207443	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	DNDI1417185	chembl:CHEMBL1549738	CHEMBL:CHEMBL1549738	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	TEROXIRONE	ncit:C2320	TEROXIRONE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	CHLORPROPHAM	chembl:CHEMBL104560	CHLORPROPHAM	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.014369915	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	2-AMINOANTHRACENE	chembl:CHEMBL83154	2-AMINOANTHRACENE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.008529511	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.057073556	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	ANIRACETAM	rxcui:17939	ANIRACETAM	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	BENZYDAMINE	rxcui:1425	BENZYDAMINE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.03070624	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002592587	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	SPERMINE	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SE-METHYLSELENOCYSTEINE	ncit:C63678	METHYLSELENOCYSTEINE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	TCMDC-125625	chembl:CHEMBL549208	CHEMBL:CHEMBL549208	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.008245551	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GNF-PF-2243	chembl:CHEMBL600908	CHEMBL:CHEMBL600908	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.015945239	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.040112812	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.108711535	O-DEMETHYLATED ADAPALENE	iuphar.ligand:3431	AHPN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.027276712	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.03409589	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.010526799	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	DTC	9/2/20	NULL	1.458546423213736	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005795549	HYDRALAZINE HYDROCHLORIDE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	GNF-PF-4057	chembl:CHEMBL598903	CHEMBL:CHEMBL598903	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.059397818	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.090634645	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.5000730593875666	CIGLITAZONE	ncit:C72726	CIGLITAZONE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1325951293830669	LINOLEIC ACID	rxcui:6400	LINOLEIC ACID	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	PORFIROMYCIN	ncit:C763	PORFIROMYCIN	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.062509132	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	NSC-111847	chembl:CHEMBL1984884	CHEMBL:CHEMBL1984884	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.032412143	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	VINCLOZOLIN	chembl:CHEMBL513221	VINCLOZOLIN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.065145994	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.03233231	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.1121958787087489	2',4'-DIHYDROXYCHALCONE	chembl:CHEMBL105310	2',4'-DIHYDROXYCHALCONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	GNF-PF-1307	chembl:CHEMBL585030	CHEMBL:CHEMBL585030	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	METAPHIT METHANESULFONATE	chembl:CHEMBL1256971	METAPHIT METHANESULFONATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	THIABENDAZOLE	rxcui:10450	THIABENDAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003106871	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.04726163	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.021440454	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
YWHAG	hgnc:12852	YWHAG	DTC	9/2/20	NULL	0.1750255707856483	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	4-METHYLESCULETIN	chembl:CHEMBL313244	4-METHYLESCULETIN	FALSE	FALSE	FALSE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	2.625383561784724	IRINOTECAN HYDROCHLORIDE HYDRATE	chembl:CHEMBL1200512	IRINOTECAN HYDROCHLORIDE HYDRATE	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	DNDI1417185	chembl:CHEMBL1549738	CHEMBL:CHEMBL1549738	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	NSC-93401	chembl:CHEMBL452954	CHEMBL:CHEMBL452954	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.182318303	CID 667285	chembl:CHEMBL267160	CHEMBL:CHEMBL267160	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.014206621	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.014832675	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.068907705	DIPYRITHIONE	rxcui:1362743	DIPYRITHIONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.039155609	OKADAIC ACID	iuphar.ligand:5349	OKADAIC ACID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	3',4' DICHLOROBENZAMIL	iuphar.ligand:4597	3,4-DICHLOROBENZAMIL	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.006512983	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
FOLR2	hgnc:3793	FOLR2	DTC	9/2/20	NULL	1.750255707856483	LOMETREXOL	ncit:C979	LOMETREXOL	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	DTC	9/2/20	NULL	1.151484018326633	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.1491695205559502	LAS38096	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	CIANIDANOL	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	P-TOLUENESULFONAMIDE	drugbank:DB17299	P-TOLUENESULFONAMIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	KRESOXIM-METHYL	chembl:CHEMBL203191	KRESOXIM-METHYL	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.033002936	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE	chembl:CHEMBL457504	CHEMBL:CHEMBL457504	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.02302968	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.041672755	PROROXAN HYDROCHLORIDE	ncit:C84120	PROROXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01323278	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.022869195	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002035536	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PROPICONAZOLE	ncit:C97997	PROPICONAZOLE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.020117882	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	LASSBIO-294	chembl:CHEMBL233194	CHEMBL:CHEMBL233194	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.028093992	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	AMBAZONE	ncit:C72627	AMBAZONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	DNDI1417099	chembl:CHEMBL1565444	CHEMBL:CHEMBL1565444	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.042073455	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.061628722	PENTAMIDINE DIISETHIONATE	chembl:CHEMBL361506	PENTAMIDINE ISETHIONATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.02804897	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	METHYL ROBUSTONE	chembl:CHEMBL1403041	METHYL ROBUSTONE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.051478109	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.023943307	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	KINETIN	rxcui:16054	KINETIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001464159	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.006938117	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.045226246	NSC-139257	chembl:CHEMBL1256364	CHEMBL:CHEMBL1256364	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.042481935	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.058341857	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.03591496	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	NSC-24047	chembl:CHEMBL1288013	CHEMBL:CHEMBL1288013	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	ANISINDIONE	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.061412481	EHNA	iuphar.ligand:5179	EHNA	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010093747	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.055622533	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.030386384	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.012561644	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.1029562181092049	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	DTC	9/2/20	NULL	0.1773907812016706	CCG-50014	iuphar.ligand:7784	CCG-50014	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000713071	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CETRIMIDE	rxcui:288088	CETRIMIDE	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.015930725	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PABPC1	hgnc:8554	PABPC1	DTC	9/2/20	NULL	6.563458904461812	GNF-PF-4618	chembl:CHEMBL585964	CHEMBL:CHEMBL585964	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.036212187	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	METHYLTHIOURACIL	ncit:C81590	METHYLTHIOURACIL	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.100976291	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.097236428	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005524797	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	R-N-PROPYLNORAPOMORPHINE	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
PRKCI	hgnc:9404	PRKCI	DTC	9/2/20	NULL	0.1721562991334246	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.014849455	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	LANSOPRAZOLE SULFIDE	chembl:CHEMBL899	LANSOPRAZOLE SULFIDE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.027929612	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	CID 667285	chembl:CHEMBL267160	CHEMBL:CHEMBL267160	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.020795117	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.108711535	CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE	chembl:CHEMBL457504	CHEMBL:CHEMBL457504	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.042276708	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SPICLOMAZINE	ncit:C66557	SPICLOMAZINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	QUINESTROL	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1562728310586145	DIFLUPREDNATE	rxcui:23043	DIFLUPREDNATE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	SJ000071821	chembl:CHEMBL589924	CHEMBL:CHEMBL589924	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2853677784548614	DIPHENHYDRAMINE HYDROCHLORIDE	rxcui:1362	DIPHENHYDRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.00192618	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	binder	1.346350544504987	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00655895	ZIDOVUDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.033148782	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013964806	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	DNDI1417031	chembl:CHEMBL1333049	CHEMBL:CHEMBL1333049	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.010875657	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005412046	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
MAP3K10	hgnc:6849	MAP3K10	DTC	9/2/20	NULL	0.086646322	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.022249013	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.014732792	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	CHOLESTEROL	rxcui:2438	CHOLESTEROL	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.024861587	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	DNDI1417809	chembl:CHEMBL1442783	CHEMBL:CHEMBL1442783	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.025244073	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
IFNGR1	hgnc:5439	IFNGR1	ChEMBL	33	agonist	39.38075342677087	INTERFERON GAMMA-1B	rxcui:5882	INTERFERON GAMMA-1B	TRUE	TRUE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIB	chembl:CHEMBL1095015	AESCULIOSIDE IIB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	WOGONIN	rxcui:2001619	WOGONIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	PENTETIC ACID	rxcui:3690	PENTETIC ACID	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DIPYRIDYL	chembl:CHEMBL39879	DIPYRIDYL	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.6604738520213144	SPIRUCHOSTATIN C	chembl:CHEMBL1835659	SPIRUCHOSTATIN C	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014160645	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
YWHAG	hgnc:12852	YWHAG	DTC	9/2/20	NULL	0.7955707762984016	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.00275284	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	BMY-7378	iuphar.ligand:9	BMY-7378	FALSE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	DTC	9/2/20	NULL	2.386712328895204	HYDROXYPROGESTERONE CAPROATE	rxcui:12488	HYDROXYPROGESTERONE CAPROATE (USP)	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1312691780892362	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.1508841127462485	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.096521454	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	FLAVIN ADENINE DINUCLEOTIDE	ncit:C80888	FLAVIN ADENINE DINUCLEOTIDE	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.084689792	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.039068208	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002107049	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	0.6731752722524935	BERGAMOTTIN	chembl:CHEMBL1078442	BERGAMOTTIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	SPHAEROPSIDIN A	chembl:CHEMBL1834675	SPHAEROPSIDIN A	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.078136416	2',3'-DIDEOXYADENOSINE	ncit:C429	DIDEOXYADENOSINE	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.070574827	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PADI3	hgnc:18337	PADI3	DTC	9/2/20	NULL	8.751278539282415	O-F-AMIDINE	iuphar.ligand:8625	O-F-AMIDINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.080781033	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.019949723	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.021240967	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.002480521	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1810609352954983	CID 100335	chembl:CHEMBL1520346	CHEMBL:CHEMBL1520346	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	3,4-DIHYDROXYPHENYLACETIC ACID	chembl:CHEMBL1284	3,4-DIHYDROXYPHENYLACETIC ACID	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.057574201	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1591141552596803	THIOGUANOSINE	chembl:CHEMBL283078	THIOGUANOSINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.013695272	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-125840	chembl:CHEMBL475813	CHEMBL:CHEMBL475813	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	DTC	9/2/20	NULL	0.044198376	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	TOMELUKAST	ncit:C74135	TOMELUKAST	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.014287802	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.01644462	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	PYRIDINE-2,4-DICARBOXYLIC ACID	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.03140411	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	GNF-PF-4227	chembl:CHEMBL585654	CHEMBL:CHEMBL585654	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	DIHYDROCAPSAICIN	rxcui:2166037	DIHYDROCAPSAICIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.021357605	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.157680694	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	ANTIAROL	chembl:CHEMBL1319047	ANTIAROL	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	GNF-PF-2954	chembl:CHEMBL582722	CHEMBL:CHEMBL582722	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.2900976311364336	DIGALLIC ACID	chembl:CHEMBL366356	DIGALLIC ACID	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.7778914257139926	MILTIRONE	chembl:CHEMBL45830	MILTIRONE	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.7778914257139926	MILTIRONE	chembl:CHEMBL45830	MILTIRONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	BUTYLPARABEN	rxcui:1306937	BUTYLPARABEN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002518354	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	GEOPYXIN A	chembl:CHEMBL1899565	GEOPYXIN A	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.032899543	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.2282942227638891	MILTIRONE	chembl:CHEMBL45830	MILTIRONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	MMV666022	chembl:CHEMBL599100	CHEMBL:CHEMBL599100	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TILIQUINOL	ncit:C72867	TILIQUINOL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	DAPHNETIN	chembl:CHEMBL244948	DAPHNETIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	TCMDC-125625	chembl:CHEMBL549208	CHEMBL:CHEMBL549208	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002035536	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	U-50488	iuphar.ligand:1652	U50488	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	N-(3,4-DIMETHOXYPHENYL)PICOLINAMIDE	chembl:CHEMBL572346	CHEMBL:CHEMBL572346	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-4782	chembl:CHEMBL584619	CHEMBL:CHEMBL584619	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTK6	hgnc:9617	PTK6	DTC	9/2/20	NULL	0.063722902	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	LEOIDIN	chembl:CHEMBL1328088	LEOIDIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.037505479	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.092443083	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.003740129	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.025567767	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.1508841127462485	DIBROMOACETIC ACID	chembl:CHEMBL449362	DIBROMOACETIC ACID	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.042242696	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	DROPERIDOL	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.086219493	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE	chembl:CHEMBL457504	CHEMBL:CHEMBL457504	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.030176823	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.006347639	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
ADK	hgnc:257	ADK	DTC	9/2/20	NULL	1.166837138570989	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	METHYL PARATHIONE	chembl:CHEMBL346516	METHYL PARATHIONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PAMICOGREL	ncit:C66300	PAMICOGREL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	2,4-DINITROTOLUENE	chembl:CHEMBL259865	CHEMBL:CHEMBL259865	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-3702	chembl:CHEMBL598268	CHEMBL:CHEMBL598268	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	3,5-DINITROCATECHOL (OR-486)	chembl:CHEMBL168276	3,5-DINITROCATECHOL (OR-486)	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	ZINC 03877300	chembl:CHEMBL1738937	CHEMBL:CHEMBL1738937	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.01083079	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRMT1	hgnc:5187	PRMT1	DTC	9/2/20	NULL	6.563458904461812	NSC-45174	iuphar.ligand:7028	AMI-1	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	RP-67580	drugbank:DB16742	RP-67580	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01495945	SPIROXATRINE	ncit:C74108	SPIROXATRINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	BETA-CCM	chembl:CHEMBL453066	BETA-CCM	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	LINOLEIC ACID	rxcui:6400	LINOLEIC ACID	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	GLYCINE	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	CID 926663	chembl:CHEMBL265686	CHEMBL:CHEMBL265686	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.019233579	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.054695491	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	PYRACLOSTROBIN	chembl:CHEMBL519873	PYRACLOSTROBIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	ORTHO-PHTHALALDEHYDE	chembl:CHEMBL160145	ORTHO-PHTHALALDEHYDE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005677733	ISOPROTERENOL HYDROCHLORIDE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.020575106	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	(E)-DIBENZYLIDENEACETONE	chembl:CHEMBL17201	CHEMBL:CHEMBL17201	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-3543	chembl:CHEMBL598679	CHEMBL:CHEMBL598679	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.094099769	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
CDK5R1	hgnc:1775	CDK5R1	DTC	9/2/20	NULL	1.875273972703375	GW8510	chembl:CHEMBL1276446	CHEMBL:CHEMBL1276446	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.2983390411119005	GW8510	chembl:CHEMBL1276446	CHEMBL:CHEMBL1276446	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DODINE	chembl:CHEMBL450348	DODINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NSC-154983	chembl:CHEMBL227298	CHEMBL:CHEMBL227298	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	2-MERCAPTOBENZIMIDAZOLE	chembl:CHEMBL70141	2-MERCAPTOBENZIMIDAZOLE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.021370644	L-733060	chembl:CHEMBL1256740	CHEMBL:CHEMBL1256740	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013887244	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.1389091831632129	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FLUACIZINE	ncit:C65702	FLUACIZINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	MIZORIBINE	ncit:C66172	MIZORIBINE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.010759769	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	HYDROXYCAMPTOTHECIN	chembl:CHEMBL273862	HYDROXYCAMPTOTHECIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.035418328	ZOXAZOLAMINE	ncit:C152966	ZOXAZOLAMINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	E-64C	chembl:CHEMBL418661	E-64C	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.031707531	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.021933029	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.3889457128569963	DNQX	chembl:CHEMBL155265	DNQX	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.015193192	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	PYRACLOSTROBIN	chembl:CHEMBL519873	PYRACLOSTROBIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	CITRIC ACID	rxcui:21183	CITRIC ACID	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.06697407	DNDI1417031	chembl:CHEMBL1333049	CHEMBL:CHEMBL1333049	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	CLADRIN	chembl:CHEMBL454746	CLADRIN	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDO1	hgnc:6059	IDO1	DTC	9/2/20	NULL	7.501095891	ZINC 00387478	chembl:CHEMBL1668301	CHEMBL:CHEMBL1668301	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	DIBUTYLDICHLOROSTANNANE	chembl:CHEMBL1088184	DIBUTYLDICHLOROSTANNANE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.007157534	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.020795117	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	GNF-PF-4668	chembl:CHEMBL584860	CHEMBL:CHEMBL584860	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW785804X	chembl:CHEMBL361237	GW785804X	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.051177067	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	DTC	9/2/20	NULL	3.750547945	BERKELEYTRIONE	chembl:CHEMBL252716	BERKELEYTRIONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.042863405	O-DEMETHYLATED ADAPALENE	iuphar.ligand:3431	AHPN	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.012573676	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.018131102	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.1521961485092594	DIFENOCONAZOLE	chembl:CHEMBL466426	DIFENOCONAZOLE	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.040452751	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003147942	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.019607047	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.03729238	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.2051080907644316	GNF-PF-1235	chembl:CHEMBL585769	CHEMBL:CHEMBL585769	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1215455352678113	ISOQUERCETIN	ncit:C117288	ISOQUERCETIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006356861	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	DIFLUFENICAN	chembl:CHEMBL1425995	DIFLUFENICAN	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.036718651	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	TCMDC-123641	chembl:CHEMBL532849	CHEMBL:CHEMBL532849	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.022099188	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.020470827	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	CANTHARIDIN	rxcui:1984	CANTHARIDIN	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.3977853881492007	IRINOTECAN HYDROCHLORIDE HYDRATE	chembl:CHEMBL1200512	IRINOTECAN HYDROCHLORIDE HYDRATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	SJ000032150	chembl:CHEMBL607140	CHEMBL:CHEMBL607140	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005677733	ISOPRENALINE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.1000146118775133	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	SJ000018300	chembl:CHEMBL590927	CHEMBL:CHEMBL590927	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.020591244	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.2154897588332195	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.048083948	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002170994	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.5303805175322676	SJ000029700	chembl:CHEMBL591864	CHEMBL:CHEMBL591864	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	ARACHIDONOYL DOPAMINE	iuphar.ligand:4261	NADA	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BROMAMINIC ACID	chembl:CHEMBL270415	BROMAMINIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.015268296	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
FGG	hgnc:3694	FGG	ChEMBL	33	inhibitor	1.640864726115453	FIBRINOLYSIN, HUMAN	rxcui:4388	PLASMIN	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	LASSBIO-294	chembl:CHEMBL233194	CHEMBL:CHEMBL233194	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2282942227638891	NAFRONYL OXALATE	ncit:C87286	NAFRONYL OXALATE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IID	chembl:CHEMBL1095016	AESCULIOSIDE IID	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.021011473	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.050781113	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011850072	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011143394	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003740928	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.750109589	CASTANOSPERMINE	drugbank:DB01816	CASTANOSPERMINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.002913047	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002447226	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	DTC	9/2/20	NULL	2.625383561784724	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
FGA	hgnc:3661	FGA	ChEMBL	33	inhibitor	1.193356164447602	FIBRINOLYSIN, HUMAN	rxcui:4388	PLASMIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	ORTHO-PHTHALALDEHYDE	chembl:CHEMBL160145	ORTHO-PHTHALALDEHYDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.005770074	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.026816992	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.1250182648468916	APREMILAST	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.012268147	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.021733308	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	QUINIZARIN	chembl:CHEMBL17594	QUINIZARIN	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2333674277141978	APREMILAST	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	0.2243917574174978	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007374673	ANANDAMIDE	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.4907258993990139	4-TRIETHYLGERMYLPHENOL	chembl:CHEMBL2313446	4-TRIETHYLGERMYLPHENOL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	GNF-PF-4242	chembl:CHEMBL584514	CHEMBL:CHEMBL584514	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	DNDI1417827	chembl:CHEMBL1363249	CHEMBL:CHEMBL1363249	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.029987248	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.3580068493342807	APREMILAST	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.039361073	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	NIFEKALANT	ncit:C75132	NIFEKALANT	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	SJ000189154	chembl:CHEMBL604664	CHEMBL:CHEMBL604664	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.015071088	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.002499413	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.006061842	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	AZELASTINE HYDROCHLORIDE	rxcui:235824	AZELASTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.9546849315580818	ALBIGLUTIDE	rxcui:1534763	ALBIGLUTIDE	TRUE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.025489161	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.026830696	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.025147352	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006077277	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	CID 5310801	chembl:CHEMBL260451	CHEMBL:CHEMBL260451	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.018860514	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00202529	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
NA	hgnc:12811	XK	ChEMBL	33	inhibitor	1.693795846312725	PERAMIVIR	rxcui:1598096	PERAMIVIR ANHYDROUS	TRUE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	modulator	0.5122699632750684	BLINATUMOMAB	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
HMBS	hgnc:4982	HMBS	FDA	10-Apr-24	NULL	5.834185692854944	Givosiran	rxcui:2265712	GIVOSIRAN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.050597611	Meclizine	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	MyCancerGenome	20-Jun-17	inhibitor	0.4526523382387456	PELITINIB	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	0.046965717	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
PTK2	hgnc:9611	PTK2	MyCancerGenome	20-Jun-17	inhibitor	0.1143957978991165	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.2363572458670459	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	MyCancerGenome	20-Jun-17	inhibitor	0.7876150685354174	BAFETINIB	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	1.029066006546944	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	1.500219178	INCB028060	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.6667640791834221	PF-04217903	drugbank:DB12848	PF-04217903	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.375054795	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.028444026	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.2386712328895204	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.2651902587661338	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1403948428761885	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.1491695205559502	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1235474617310458	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1816874437221263	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547592	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.1764963739014941	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
MLST8	hgnc:24825	MLST8	MyCancerGenome	20-Jun-17	inhibitor	1.458546423213736	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
RICTOR	hgnc:28611	RICTOR	MyCancerGenome	20-Jun-17	inhibitor	0.8334550989792778	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
AKT1S1	hgnc:28426	AKT1S1	MyCancerGenome	20-Jun-17	inhibitor	1.458546423213736	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.092443083	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.3409589041278864	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.6945459158160648	NIMOTUZUMAB	ncit:C2733	NIMOTUZUMAB	FALSE	TRUE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.020542907	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.225178995499538	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2363572458670459	BIBW 2992	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.095500063	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.192335792	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.7501095890813498	PD 0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2363572458670459	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1124502911321247	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.045421861	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NOS2	hgnc:7873	NOS2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.061701141	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.0081597	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.4487835148349957	BRYOSTATIN 1	ncit:C1026	BRYOSTATIN 1	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.2243917574174978	ANTIPARASITIC	ncit:C276	ANTIPARASITIC AGENT	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02639903	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02639903	DESFERRIOXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.049864835	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.040798501	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	1.779921058837101	ANTISENSE C-FOS	ncit:C2457	C-FOS ANTISENSE	FALSE	FALSE	FALSE
ALPP	hgnc:439	ALPP	NCI	14-Sep-17	NULL	1.944728564284981	DDA	ncit:C429	DIDEOXYADENOSINE	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.3088686543276147	BETULINIC ACID	ncit:C38126	BETULINIC ACID	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.077217164	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.9131768910555565	PROTEIN PHOSPHATASE INHIBITOR	ncit:C2159	PROTEIN PHOSPHATASE INHIBITOR	FALSE	FALSE	FALSE
APRT	hgnc:626	APRT	NCI	14-Sep-17	NULL	0.1875273972703375	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
APRT	hgnc:626	APRT	NCI	14-Sep-17	NULL	0.1875273972703375	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
ATF2	hgnc:784	ATF2	NCI	14-Sep-17	NULL	0.3804903712731485	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
AQP1	hgnc:633	AQP1	NCI	14-Sep-17	NULL	0.081281225	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.3201687270469177	DDTC	ncit:C432	DITIOCARB	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.050222545	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	NCI	14-Sep-17	NULL	0.078136416	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1219690388750162	GONADOTROPINS	ncit:C527	THERAPEUTIC GONADOTROPIN	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1422972120208522	OPIATE	ncit:C1657	OPIATE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1707566544250227	K-252A	drugbank:DB02152	K-252A	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.03049226	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.050222545	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.4268916360625568	INTERLEUKIN-1 RECEPTOR ANTAGONIST	ncit:C2486	RECOMBINANT INTERLEUKIN-1 RECEPTOR ANTAGONIST	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.032837818	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.1182605208011137	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.8537832721251137	VERTEPORFIN	rxcui:118886	VERTEPORFIN	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.218327115	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.099446347	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.020575106	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.085239726	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
CA2	hgnc:1373	CA2	NCI	14-Sep-17	NULL	0.3671865121377238	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
CASR	hgnc:1514	CASR	NCI	14-Sep-17	NULL	0.5048814541893702	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	NCI	14-Sep-17	NULL	0.090452491	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CDKN2D	hgnc:1790	CDKN2D	NCI	14-Sep-17	NULL	5.625821918110125	IL-4	iuphar.ligand:4996	IL-4	FALSE	FALSE	FALSE
CSF1	hgnc:2432	CSF1	NCI	14-Sep-17	NULL	1.714536203614514	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.2333674277141977	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.1785975212098452	ADENOVIRAL VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.043109746	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.3500511415712967	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.3977853881492007	FADROZOLE	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.086361301	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	ChEMBL	33	modulator	1.250182648468916	BMS-852927	chembl:CHEMBL3545047	BMS-852927	FALSE	FALSE	FALSE
CYP24A1	hgnc:2602	CYP24A1	NCI	14-Sep-17	NULL	0.8975670296699916	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.014757637	VORICONAZOLE	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.00607587	MAO INHIBITORS	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.8140724222588294	QUINONE	rxcui:319868	1,4-BENZOQUINONE	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1221108633388244	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.8140724222588294	TOPOISOMERASE INHIBITORS	ncit:C1748	TOPOISOMERASE INHIBITOR	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.6105543166941221	RO-31-8220	ncit:C1310	RO 31-8220	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.01732069	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	0.7160136986685613	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.1136529680426287	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
NR1H2	hgnc:7965	NR1H2	ChEMBL	33	agonist	2.019525817	CS-8080	chembl:CHEMBL3545238	CS-8080	FALSE	FALSE	FALSE
DFFB	hgnc:2773	DFFB	NCI	14-Sep-17	NULL	0.5303805175322677	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
DNTT	hgnc:2983	DNTT	NCI	14-Sep-17	NULL	6.563458904461812	ADA INHIBITOR	ncit:C2157	ADENOSINE DEAMINASE INHIBITOR	FALSE	FALSE	FALSE
DOCK10	hgnc:23479	DOCK10	NCI	14-Sep-17	NULL	21.00306849	INTERLEUKIN-4	rxcui:1426682	BINETRAKIN	FALSE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.8334550989792776	LANREOTIDE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.1187956362798518	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
F11	hgnc:3529	F11	NCI	14-Sep-17	NULL	0.2302968036653267	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.089298761	SU-014813	chembl:CHEMBL1721885	SU-014813	FALSE	FALSE	FALSE
F8	hgnc:3546	F8	NCI	14-Sep-17	NULL	0.8824818695074704	C5A	iuphar.ligand:3576	C5A	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.4605936073306534	DEXTRAN SULFATE	rxcui:40068	DEXTRAN SULFATE	FALSE	FALSE	FALSE
F8	hgnc:3546	F8	NCI	14-Sep-17	NULL	2.059124362184097	SORBITOL	rxcui:9945	SORBITOL	TRUE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.043109746	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
FABP1	hgnc:3555	FABP1	NCI	14-Sep-17	NULL	0.3860858179095183	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.046303061	SU-014813	chembl:CHEMBL1721885	SU-014813	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.015215205	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.03292017	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	NCI	14-Sep-17	NULL	0.2187819634820604	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	1.346350544504987	ALPHA-ADRENERGIC ANTAGONIST	ncit:C29713	ALPHA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
GDF15	hgnc:30142	GDF15	NCI	14-Sep-17	NULL	2.500365296937833	INDOLE-3-CARBINOL	rxcui:2598119	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.260583976	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
GDF15	hgnc:30142	GDF15	NCI	14-Sep-17	NULL	0.8824818695074707	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.017733087	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
GDF15	hgnc:30142	GDF15	NCI	14-Sep-17	NULL	1.250182648468916	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.2991890098899972	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	1.381780822	PF-03882845	drugbank:DB11814	PF-03882845	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	NCI	14-Sep-17	NULL	0.065799087	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.789589041	DIETHYLDITHIOCARBAMATE	rxcui:1427193	DIETHYLDITHIOCARBAMATE	FALSE	FALSE	FALSE
GRM1	hgnc:4593	GRM1	NCI	14-Sep-17	NULL	9.024755993634992	DHPG	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.9546849315580819	AMIFOSTINE	rxcui:1545987	AMIFOSTINE ANHYDROUS	TRUE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	0.6863747873946994	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	2.917092846427472	ATROPINE SULFATE	rxcui:153971	ATROPINE SULFATE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.1061833594250647	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.175610941	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.138178082	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.026519026	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.049026771	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	0.6213925590023018	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.042022946	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	RTGF-BETA	ncit:C898	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.4102161815288632	MACROLIDE ANTIBIOTIC	ncit:C261	MACROLIDE ANTIBIOTIC	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.046798281	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.3431873936973496	DEXTRAN SULFATE	rxcui:40068	DEXTRAN SULFATE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.2059124362184098	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1715936968486748	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.035040154	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1810609352954983	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.061376588	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
IRF2	hgnc:6117	IRF2	NCI	14-Sep-17	NULL	2.019525816757481	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
IRS2	hgnc:6126	IRS2	NCI	14-Sep-17	NULL	0.1861974157294131	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.1591141552596803	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1508841127462485	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
MAPKAPK2	hgnc:6887	MAPKAPK2	ChEMBL	33	inhibitor	2.917092846427472	AT-13148	chembl:CHEMBL3544960	AT-13148	FALSE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	NCI	14-Sep-17	NULL	0.1591141552596803	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
KIR2DL3	hgnc:6331	KIR2DL3	NCI	14-Sep-17	NULL	0.6731752722524935	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.2917092846427472	ISOLATED SOY PROTEIN	ncit:C1803	SOY PROTEIN ISOLATE	FALSE	FALSE	FALSE
LCAT	hgnc:6522	LCAT	NCI	14-Sep-17	NULL	0.4565884455277782	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	1.458546423213736	ANTICOAGULANT	ncit:C263	ANTICOAGULANT AGENT	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.1411496538593938	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	2.692701089009974	BLEOMYCIN A5	ncit:C1279	PINGYANGMYCIN	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	NCI	14-Sep-17	NULL	0.192335792	TYROSINE KINASE INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.1417211099478934	CHLORHEXIDINE	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.1544343271638073	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.2447910080918158	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.048394167	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	NCI	14-Sep-17	NULL	0.075442056	INTERFERON ALPHA-2A	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.3281729452230906	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.00299804	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1682938180631233	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.2143170254518142	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	0.3079628811477683	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.7573221812840553	DICOUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.1553481397505754	TYROSINE KINASE INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.084146909	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.325124899	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.1988926940746004	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.182318303	ANTHRACYCLINE	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.027010119	CYTOSINE ARABINOSIDE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
PC	hgnc:8636	PC	NCI	14-Sep-17	NULL	1.250182648468916	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
PAX2	hgnc:8616	PAX2	NCI	14-Sep-17	NULL	1.346350544504987	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.017951341	HERCEPTIN	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1888765152363111	AZD-0424	drugbank:DB13088	AZD-0424	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.040390516	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.040390516	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
PIP	hgnc:8993	PIP	NCI	14-Sep-17	NULL	1.193356164447602	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
PLAT	hgnc:9051	PLAT	NCI	14-Sep-17	NULL	0.280789686	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2273059360852575	G-CSF	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
PLAUR	hgnc:9053	PLAUR	NCI	14-Sep-17	NULL	0.8751278539282417	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
PPIB	hgnc:9255	PPIB	NCI	14-Sep-17	NULL	0.6035364509849942	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
PPP1R1B	hgnc:9287	PPP1R1B	NCI	14-Sep-17	NULL	1.875273972703374	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRKD1	hgnc:9407	PRKD1	NCI	14-Sep-17	NULL	0.2143170254518142	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
PZP	hgnc:9750	PZP	NCI	14-Sep-17	NULL	0.3723948314588262	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.052090944	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.016669102	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RNASEH2A	hgnc:18518	RNASEH2A	NCI	14-Sep-17	NULL	1.250182648468916	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
RNASEH2A	hgnc:18518	RNASEH2A	NCI	14-Sep-17	NULL	1.544343271638073	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
SDHB	hgnc:10681	SDHB	NCI	14-Sep-17	NULL	1.141471113819445	GENTAMYCIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
SI	hgnc:10856	SI	NCI	14-Sep-17	NULL	0.2853677784548614	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.3281729452230906	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	1.750255707856483	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.047518255	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.100976291	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	1.050153425	THYMIDINE	rxcui:1372538	THYMIDINE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.080781033	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
SLC2A5	hgnc:11010	SLC2A5	NCI	14-Sep-17	NULL	1.141471113819445	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1077080435603989	RHGH	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
SLC9A3	hgnc:11073	SLC9A3	NCI	14-Sep-17	NULL	0.7721716358190368	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.1099637093941246	CEP-32496	iuphar.ligand:7880	AGERAFENIB	FALSE	FALSE	FALSE
SOCS1	hgnc:19383	SOCS1	NCI	14-Sep-17	NULL	1.750255707856483	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	NCI	14-Sep-17	NULL	0.045858228	LEUPROLIDE ACETATE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	1.400204566285186	PROTEIN PHOSPHATASE INHIBITOR	ncit:C2159	PROTEIN PHOSPHATASE INHIBITOR	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.2692701089009974	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	NCI	14-Sep-17	NULL	0.1902451856365742	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	4.039051633514961	VALINOMYCIN	ncit:C924	VALINOMYCIN	FALSE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	1.050153425	ALUM	rxcui:221456	ALUM, POTASSIUM	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.3292017005372696	EQUINE GONADOTROPIN	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
TFPI2	hgnc:11761	TFPI2	NCI	14-Sep-17	NULL	2.625383561784725	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.030688294	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.5608295993131588	ROGARATINIB	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.6775183385250904	POLYETHYLENE GLYCOL	rxcui:1310594	POLYETHYLENE GLYCOL 4000	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.3814116554650932	PIRFENIDONE	rxcui:1592254	PIRFENIDONE	TRUE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	2.500365296937833	MIBG	rxcui:14448	3-IODOBENZYLGUANIDINE	TRUE	FALSE	FALSE
XRCC5	hgnc:12833	XRCC5	NCI	14-Sep-17	NULL	0.7501095890813501	PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.028252715	VP-16	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.9723642821424906	BAY-1125976	chembl:CHEMBL4751394	BAY-1125976	FALSE	FALSE	FALSE
ZAP70	hgnc:12858	ZAP70	NCI	14-Sep-17	NULL	2.019525816757481	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.020579138	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	OncoKB	23-Jul-20	NULL	0.546954909	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	0.4948366922735607	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	OncoKB	23-Jul-20	NULL	0.2287915957982331	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	OncoKB	23-Jul-20	NULL	0.6168664383892681	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	OncoKB	23-Jul-20	NULL	0.2007335520076852	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.6250913242344582	CEP-5214	chembl:CHEMBL150894	CEP-5214	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	OncoKB	23-Jul-20	NULL	0.5125748858722557	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	OncoKB	23-Jul-20	NULL	0.033903258	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
SRSF2	hgnc:10783	SRSF2	OncoKB	23-Jul-20	NULL	6.563458904461812	H3B-8800	drugbank:DB14017	H3B-8800	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	OncoKB	23-Jul-20	NULL	0.054695491	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.4839416703750644	Glucarpidase	rxcui:1242127	GLUCARPIDASE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.5427149481725528	ritodrine	rxcui:9392	RITODRINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.016397374	theophylline	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ERCC1	hgnc:3433	ERCC1	PharmGKB	4/5/24	NULL	0.2365210416022274	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
ADRA1D	hgnc:280	ADRA1D	PharmGKB	4/5/24	NULL	0.1346350544504987	methoxamine	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1032599237673441	memantine	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
APOC3	hgnc:610	APOC3	PharmGKB	4/5/24	NULL	0.2083637747448194	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
PPCDC	hgnc:28107	PPCDC	PharmGKB	4/5/24	NULL	1.750255707856483	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.3070624048871023	oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
SLC28A3	hgnc:16484	SLC28A3	PharmGKB	4/5/24	NULL	0.4167275494896389	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.106290832	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.7001022831425934	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
ZNF423	hgnc:16762	ZNF423	PharmGKB	4/5/24	NULL	0.8078103267029924	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.1595977849109255	ROGARATINIB	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.081030357	siponimod	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
NCOA1	hgnc:7668	NCOA1	PharmGKB	4/5/24	NULL	0.4039051633514962	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
HNF4A	hgnc:5024	HNF4A	PharmGKB	4/5/24	NULL	0.2734774543525755	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.088695391	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.021036727	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.045579576	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.060772768	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.4070362111294147	methacholine	rxcui:155080	METHACHOLINE	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	6.563458904461812	cycloguanil	ncit:C81015	CYCLOGUANIL	FALSE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.1442518440541057	nifedipine	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.021846337	amphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
NUP153	hgnc:8062	NUP153	PharmGKB	4/5/24	NULL	11.66837138570989	ticagrelor	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	PharmGKB	4/5/24	NULL	0.06697407	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
SORCS2	hgnc:16698	SORCS2	PharmGKB	4/5/24	NULL	17.50255707856483	atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	PharmGKB	4/5/24	NULL	0.040328473	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.032055965	nefazodone	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.4102161815288632	ethambutol	rxcui:142435	ETHAMBUTOL HYDROCHLORIDE	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	PharmGKB	4/5/24	NULL	0.1905904582057876	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.1118771404169627	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.037398626	paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.037398626	aldosterone	rxcui:1312358	ALDOSTERONE	FALSE	FALSE	FALSE
CDH15	hgnc:1754	CDH15	PharmGKB	4/5/24	NULL	0.5000730593875666	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.069638821	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
TTK	hgnc:12401	TTK	ChEMBL	33	inhibitor	17.50255707856483	BAY-1161909	chembl:CHEMBL4303241	BAY-1161909	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	PharmGKB	4/5/24	NULL	0.036770078	iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.074128477	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
RGS17	hgnc:14088	RGS17	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.038382801	sacituzumab govitecan-hziy	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	7.292732116	letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
SYNE3	hgnc:19861	SYNE3	PharmGKB	4/5/24	NULL	0.8334550989792777	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.059030547	tolperisone	rxcui:10639	TOLPERISONE	FALSE	FALSE	FALSE
AGAP3	hgnc:16923	AGAP3	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	PharmGKB	4/5/24	NULL	0.092606122	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.3125456621172291	hydrocortisone	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
LST1	hgnc:14189	LST1	PharmGKB	4/5/24	NULL	9.546849315580818	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	2.512328767	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	PharmGKB	4/5/24	NULL	0.6731752722524936	amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.3947945205691315	ROGARATINIB	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.095468493	prilocaine	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.028413242	ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.2778183663264259	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.2125816649218401	stavudine	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.025439763	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.3889457128569962	apixaban	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.760980743	apixaban	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
RGS5	hgnc:10001	RGS5	PharmGKB	4/5/24	NULL	0.5556367326528519	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.024461995	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.1440539677248134	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.1296485709523321	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NCF4	hgnc:7662	NCF4	PharmGKB	4/5/24	NULL	0.2592971419046642	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.01609924	3,4-methylenedioxymethamphetamine	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.006811217	colchicine	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.014757637	sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.009081623	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.018782447	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
SSTR4	hgnc:11333	SSTR4	PharmGKB	4/5/24	NULL	3.500511415712967	lutetium (177Lu) oxodotreotide	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
IMPDH2	hgnc:6053	IMPDH2	PharmGKB	4/5/24	NULL	0.2763561643983921	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.2465148884304905	bucindolol	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
CASP9	hgnc:1511	CASP9	PharmGKB	4/5/24	NULL	0.3454452054979901	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
IMPDH1	hgnc:6052	IMPDH1	PharmGKB	4/5/24	NULL	0.1842374429322614	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.3125456621172291	hydrocortisone	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	PharmGKB	4/5/24	NULL	0.043003826	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.1136529680426288	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	2.386712328895204	Influenza vaccines	wikidata:Q383260	INFLUENZA VACCINE	FALSE	FALSE	FALSE
CTNNA3	hgnc:2511	CTNNA3	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	PharmGKB	4/5/24	NULL	0.020383413	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
HLA-E	hgnc:4962	HLA-E	PharmGKB	4/5/24	NULL	0.1562728310586145	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.047821194	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
RALBP1	hgnc:9841	RALBP1	PharmGKB	4/5/24	NULL	0.2381300282797936	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
HLA-DPB1	hgnc:4940	HLA-DPB1	PharmGKB	4/5/24	NULL	1.381780822	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
PTPN22	hgnc:9652	PTPN22	PharmGKB	4/5/24	NULL	0.5527123287967842	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
SACM1L	hgnc:17059	SACM1L	PharmGKB	4/5/24	NULL	6.177373086552294	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.4605936073306534	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
HLA-DRB3	hgnc:4951	HLA-DRB3	PharmGKB	4/5/24	NULL	0.8204323630577265	heparin	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.074797252	bisoprolol	rxcui:19484	BISOPROLOL	TRUE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1495945049449985	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
BCHE	hgnc:983	BCHE	PharmGKB	4/5/24	NULL	0.2917092846427472	memantine	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.2333674277141978	edoxaban	rxcui:1599538	EDOXABAN	TRUE	FALSE	FALSE
ATIC	hgnc:794	ATIC	PharmGKB	4/5/24	NULL	0.2414145803939976	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
FASTKD3	hgnc:28758	FASTKD3	PharmGKB	4/5/24	NULL	0.9460841664089098	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
SHMT1	hgnc:10850	SHMT1	PharmGKB	4/5/24	NULL	0.9460841664089098	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.1132444383228493	toremifene	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.3182283105193605	rofecoxib	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	PharmGKB	4/5/24	NULL	0.1773907812016706	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	PharmGKB	4/5/24	NULL	0.035478156	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
FGB	hgnc:3662	FGB	PharmGKB	4/5/24	NULL	1.400204566285186	tirofiban	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
JAG1	hgnc:6188	JAG1	PharmGKB	4/5/24	NULL	2.917092846427472	odevixibat	rxcui:2563966	ODEVIXIBAT	TRUE	FALSE	FALSE
CDH13	hgnc:1753	CDH13	PharmGKB	4/5/24	NULL	0.2308029504865692	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CES1P1	hgnc:18546	CES1P1	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.028850369	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.095468493	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
LTA	hgnc:6709	LTA	PharmGKB	4/5/24	NULL	0.5357925636295356	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.2019525816757481	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	2.100306849	pegloticase	rxcui:1011650	PEGLOTICASE	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.1881995384791917	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.1117184494376478	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
CAPN10	hgnc:1477	CAPN10	PharmGKB	4/5/24	NULL	1.346350544504987	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.004216468	bromazepam	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
APOA5	hgnc:17288	APOA5	PharmGKB	4/5/24	NULL	0.8078103267029924	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	1.334940794127826	PF-03814735	drugbank:DB13059	PF-03814735	FALSE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.017679351	triazolam	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1296485709523321	cyclobenzaprine	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	PharmGKB	4/5/24	NULL	0.3281729452230906	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.015940398	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
INSRR	hgnc:6093	INSRR	PharmGKB	4/5/24	NULL	7.501095890813499	Glucarpidase	rxcui:1242127	GLUCARPIDASE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.018636263	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.091317689	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
P2RY12	hgnc:18124	P2RY12	PharmGKB	4/5/24	NULL	2.187819634820604	ticagrelor	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.1666910197958555	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SSTR3	hgnc:11332	SSTR3	PharmGKB	4/5/24	NULL	1.166837138570989	lutetium (177Lu) oxodotreotide	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	PharmGKB	4/5/24	NULL	1.367387271762877	larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.3365876361262467	inclisiran	rxcui:2588243	INCLISIRAN	TRUE	FALSE	FALSE
SLC22A7	hgnc:10971	SLC22A7	PharmGKB	4/5/24	NULL	0.6482428547616604	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.093098708	sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	0.067317527	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.5666295457089334	omacetaxine	rxcui:1546446	OMACETAXINE	TRUE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	PharmGKB	4/5/24	NULL	1.009762908	deferasirox	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.1250182648468916	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
FGA	hgnc:3661	FGA	PharmGKB	4/5/24	NULL	1.591141552596802	abciximab	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	PharmGKB	4/5/24	NULL	0.2785552850699973	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.3431873936973497	oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	PharmGKB	4/5/24	NULL	0.2393966773663883	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.1293292394967845	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
VEGFC	hgnc:12682	VEGFC	PharmGKB	4/5/24	NULL	0.4375639269641208	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.1209854175937661	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
RHBDF2	hgnc:20788	RHBDF2	PharmGKB	4/5/24	NULL	1.166837138570988	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
EPB41	hgnc:3377	EPB41	PharmGKB	4/5/24	NULL	2.059124362184098	bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.1704794520639431	cisapride	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.4773424657790409	mirtazapine	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	TALC	12-May-16	inhibitor	0.2311077079035849	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.061197752	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
CRP	hgnc:2367	CRP	PharmGKB	4/5/24	NULL	0.3977853881492008	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	TALC	12-May-16	inhibitor	0.6035364509849942	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.1426838892274307	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
ITGB3	hgnc:6156	ITGB3	TALC	12-May-16	NULL	3.500511415712966	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	TALC	12-May-16	inhibitor	0.3319450480417468	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
CDK16	hgnc:8749	CDK16	ChEMBL	33	inhibitor	0.5000730593875666	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
UNIPROT:Q92633	hgnc:3166	LPAR1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	AM-152	iuphar.ligand:9498	BMS-986020	FALSE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	0.2885036881082115	AM-101	chembl:CHEMBL2364609	ESKETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.031929262	APD421	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
UNIPROT:Q16881	hgnc:12437	TXNRD1	TdgClinicalTrial	Jan-14	NULL	1.009762908	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
UNIPROT:O14920	hgnc:5960	IKBKB	TdgClinicalTrial	Jan-14	NULL	0.192335792	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
UNIPROT:P24941	hgnc:1771	CDK2	TdgClinicalTrial	Jan-14	NULL	1.363835616511545	AT7519	ncit:C64761	CDK INHIBITOR AT7519	FALSE	FALSE	FALSE
UNIPROT:P14210	hgnc:4893	HGF	TdgClinicalTrial	Jan-14	NULL	9.723642821424907	FICLATUZUMAB	ncit:C78844	FICLATUZUMAB	FALSE	TRUE	TRUE
UNIPROT:Q15139	hgnc:9407	PRKD1	TdgClinicalTrial	Jan-14	NULL	0.3750547945406749	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:P20594	hgnc:7944	NPR2	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	CD-NP	ncit:C171663	CENDERITIDE	FALSE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.060761035064535	CETRORELIX	rxcui:68147	CETRORELIX	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.1002054794574322	CLOBETASOL	rxcui:2590	CLOBETASOL	TRUE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	0.3061671792168775	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.03070624	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	1.790034246671403	CONIVAPTAN	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
UNIPROT:P06746	hgnc:9174	POLB	TdgClinicalTrial	Jan-14	NULL	0.007162904	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	1.109316997937207	CR845	rxcui:2569089	DIFELIKEFALIN	TRUE	FALSE	FALSE
UNIPROT:Q15116	hgnc:8760	PDCD1	TdgClinicalTrial	Jan-14	NULL	2.561349816375341	CT-011	drugbank:DB05916	CT-011	FALSE	TRUE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.09814518	ETONOGESTREL	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.025244073	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TdgClinicalTrial	Jan-14	NULL	0.1187956362798518	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	3.962843112127886	FIGITUMUMAB	ncit:C52187	FIGITUMUMAB	FALSE	TRUE	TRUE
UNIPROT:P48549	hgnc:6264	KCNJ3	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
UNIPROT:Q15303	hgnc:3432	ERBB4	TdgClinicalTrial	Jan-14	NULL	0.3017682254924971	GGF-2	chembl:CHEMBL3039542	CIMAGLERMIN ALFA	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.02926849	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:Q02156	hgnc:9401	PRKCE	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	KAI-1678	drugbank:DB16211	KAI-1678	FALSE	FALSE	FALSE
UNIPROT:Q16620	hgnc:8032	NTRK2	TdgClinicalTrial	Jan-14	NULL	0.182318303	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
UNIPROT:P06734	hgnc:3612	FCER2	TdgClinicalTrial	Jan-14	NULL	31.50460274141669	LUMILIXIMAB	ncit:C26448	GOMILIXIMAB	FALSE	FALSE	FALSE
UNIPROT:P13866	hgnc:11036	SLC5A1	TdgClinicalTrial	Jan-14	NULL	6.300920548283339	LX4211	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.1389091831632129	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
UNIPROT:P08631	hgnc:4840	HCK	TdgClinicalTrial	Jan-14	NULL	0.1470803115845784	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.3977853881492007	LY-674	iuphar.ligand:2658	LY-518674	FALSE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.4227670791923872	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.596678082	MEM 1414	drugbank:DB05888	MEM 1414	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.6035364509849942	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O94829	hgnc:16853	IPO13	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
UNIPROT:P33402	hgnc:4684	GUCY1A2	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	NCX 4016	ncit:C61499	NITRIC OXIDE-RELEASING ACETYLSALICYLIC ACID DERIVATIVE	FALSE	FALSE	FALSE
CDK10	hgnc:1770	CDK10	ChEMBL	33	inhibitor	0.5000730593875666	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.2465148884304905	NALMEFENE	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.080286959	NALMEFENE	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.018031481	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.051885051	PALIPERIDONE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.5000730593875666	SGX-523	drugbank:DB06314	SGX-523	FALSE	FALSE	FALSE
UNIPROT:P08620	hgnc:3682	FGF4	TdgClinicalTrial	Jan-14	NULL	6.300920548283339	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.1902451856365742	RWJ-67657	chembl:CHEMBL190333	RWJ-67657	FALSE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	PEG-INTERFERON ALFACON-1	drugbank:DB05860	PEGINTERFERON ALFACON-1	FALSE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	PEG-INTERFERON ALFACON-1	drugbank:DB05860	PEGINTERFERON ALFACON-1	FALSE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	PH-797804	drugbank:DB07941	PH-797804	FALSE	FALSE	FALSE
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.3889457128569963	PH-797804	drugbank:DB07941	PH-797804	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	1.721562991334245	TELAPRISTONE	ncit:C104057	TELAPRISTONE	FALSE	FALSE	FALSE
UNIPROT:P40238	hgnc:7217	MPL	TdgClinicalTrial	Jan-14	NULL	2.983390411119005	ELTROMBOPAG	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	1.567393171214761	TAK-901	drugbank:DB12756	TAK-901	FALSE	FALSE	FALSE
UNIPROT:P12931	hgnc:11283	SRC	TdgClinicalTrial	Jan-14	NULL	0.038894571	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1840222122746302	DESVENLAFAXINE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.059085902	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.1154014752432845	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P51681	hgnc:1606	CCR5	TdgClinicalTrial	Jan-14	NULL	3.938075342677087	MARAVIROC	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.078136416	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.108711535	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	2.561349816375341	PAC-14028	drugbank:DB12428	PAC-14028	FALSE	FALSE	FALSE
UNIPROT:Q09428	hgnc:59	ABCC8	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.1124502911321247	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.089298761	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.3535870116881784	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	0.8975670296699914	TEGASEROD	rxcui:139778	TEGASEROD	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.027752469	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P39086	hgnc:4579	GRIK1	TdgClinicalTrial	Jan-14	NULL	1.432027397337122	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	0.157680694	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	0.2243917574174978	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	positive modulator	0.3125456621172291	CX1739	chembl:CHEMBL3707399	CX1739	FALSE	FALSE	FALSE
UNIPROT:P13612	hgnc:6140	ITGA4	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	VEDOLIZUMAB	rxcui:1538097	VEDOLIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	1.848379561100067	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1583941817064691	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.047886613	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.057700738	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.2453629496995069	GTX-758	drugbank:DB14969	GTX-758	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.064033745	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.061055432	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.062509132	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.3739862623624964	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1204304386139782	CODEINE	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1137761023525341	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.1376949420516464	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.1744440904840348	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	DIETHYLPROPION	rxcui:3389	DIETHYLPROPION	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.217423069	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.6250913242344582	RG6029	chembl:CHEMBL3707380	RG6029	FALSE	FALSE	FALSE
UNIPROT:O14646	hgnc:1915	CHD1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.054953083	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	AVE8134	chembl:CHEMBL3545334	AVE8134	FALSE	FALSE	FALSE
UNIPROT:O95180	hgnc:1395	CACNA1H	TdgClinicalTrial	Jan-14	NULL	0.4440395030502706	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.056826484	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	inhibitor	0.8607814956671229	LONAPRISAN	ncit:C71532	LONAPRISAN	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.087318744	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.059532507	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.8950171233357017	HEXYLCAINE	rxcui:26879	HEXYLCAINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1241316104862754	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.9546849315580818	LIRAGLUTIDE RECOMBINANT	rxcui:475968	LIRAGLUTIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1017590527823536	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.089501712	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.42006137	OMS405	chembl:CHEMBL5095027	OMS405	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.096050618	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	3.750547945	METHYCLOTHIAZIDE	rxcui:6860	METHYCLOTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.2853677784548614	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.064347636	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
UNIPROT:P20963	hgnc:1677	CD247	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	MUROMONAB	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	TERBUTALINE	rxcui:10368	TERBUTALINE	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TdgClinicalTrial	Jan-14	NULL	0.6364566210387212	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	1.250182648468916	NRX195183	chembl:CHEMBL107430	NRX195183	FALSE	FALSE	FALSE
UNIPROT:P01019	hgnc:333	AGT	TEND	1-Aug-11	NULL	0.9723642821424906	CILAZAPRIL	rxcui:21102	CILAZAPRIL	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1077080435603989	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.1744440904840348	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.217423069	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TEND	1-Aug-11	NULL	9.845188356692718	BETAZOLE	drugbank:DB00272	BETAZOLE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.2187819634820604	DAPIPRAZOLE	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TEND	1-Aug-11	NULL	0.3088686543276147	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.076098074	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.11707396	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.07963752	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.093763699	ANLOTINIB	ncit:C138997	ANLOTINIB	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.088945801	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.075261832	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.081533651	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.087318744	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	0.3017682254924971	GLIBENCLAMIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
UNIPROT:P48039	hgnc:7463	MTNR1A	TEND	1-Aug-11	NULL	1.034633915974276	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
UNIPROT:P51787	hgnc:6294	KCNQ1	TEND	1-Aug-11	NULL	1.432027397337122	INDAPAMIDE	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
UNIPROT:P00439	hgnc:8582	PAH	TEND	1-Aug-11	NULL	3.500511415712967	SAPROPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TEND	1-Aug-11	NULL	0.201178817	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
CDK11B	hgnc:1729	CDK11B	ChEMBL	33	inhibitor	0.1470803115845784	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.272767123	KETOPROFEN	rxcui:6142	KETOPROFEN	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.1691068316769549	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P27815	hgnc:8780	PDE4A	TEND	1-Aug-11	NULL	0.3977853881492006	MILRINONE	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.8950171233357017	MORICIZINE	rxcui:40169	MORICIZINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.085009721	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
CDK18	hgnc:8751	CDK18	ChEMBL	33	inhibitor	0.5000730593875666	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TEND	1-Aug-11	NULL	4.773424657790408	NEDOCROMIL	rxcui:31563	NEDOCROMIL	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.4303907478335614	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TEND	1-Aug-11	NULL	0.1182605208011137	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.08178765	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P49788	hgnc:9867	RARRES1	TEND	1-Aug-11	NULL	0.5770073762164231	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.073885091	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.078682824	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.1470803115845784	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.070448575	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.078682824	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.083257407	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.064505739	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.050781113	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.6563458904461812	SALSALATE	rxcui:36108	SALSALATE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.4565884455277783	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
CDK16	hgnc:8749	CDK16	ChEMBL	33	inhibitor	0.5000730593875666	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
ATP-DEPENDENT RNA HELICASE DDX5	hgnc:2746	DDX5	TTD	2020.06.01	NULL	52.50767123569449	RX-5902	ncit:C113293	P-P68 INHIBITOR RX-5902	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	TrasGEX	ncit:C97917	GLYCOOPTIMIZED TRASTUZUMAB-GEX	FALSE	FALSE	FALSE
TRYPTOPHAN 5-HYDROXYLASE 1	hgnc:12008	TPH1	TTD	2020.06.01	NULL	13.12691780892362	KAR5585	ncit:C171781	RODATRISTAT ETHYL	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.09741683	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
APELIN RECEPTOR	hgnc:339	APLNR	TTD	2020.06.01	NULL	13.12691780892362	AMG 986	iuphar.ligand:10061	AZELAPRAG	FALSE	FALSE	FALSE
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	0.9376369863516875	AMG 176	ncit:C127817	TAPOTOCLAX	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.7095631248066824	AZD4635	ncit:C148039	IMARADENANT	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.1346350544504987	GDC-0077	ncit:C132166	INAVOLISIB	FALSE	FALSE	TRUE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	1.544343271638073	DV281	ncit:C143006	CPG OLIGODEOXYNUCLEOTIDE TLR9 AGONIST DV281	FALSE	FALSE	FALSE
CDK17	hgnc:8750	CDK17	ChEMBL	33	inhibitor	0.6250913242344582	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
NOTCH-1 RECEPTOR	hgnc:7881	NOTCH1	TTD	2020.06.01	NULL	2.187819634820604	LY3039478	ncit:C171871	CRENIGACESTAT	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 BETA	hgnc:5258	HSP90AB1	TTD	2020.06.01	NULL	1.141471113819445	TAS-116	drugbank:DB14876	TAS-116	FALSE	FALSE	FALSE
CASEIN KINASE II ALPHA	hgnc:2457	CSNK2A1	TTD	2020.06.01	NULL	1.875273972703375	CX-4945	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	ChEMBL	33	inhibitor	0.042619863	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.2592971419046642	CEP-32496	iuphar.ligand:7880	AGERAFENIB	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	PEN-866	drugbank:DB16186	PEN-866	FALSE	FALSE	FALSE
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	2.625383561784724	Cibinetide	ncit:C171683	CIBINETIDE	FALSE	FALSE	FALSE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	2.019525817	SHR-1314	iuphar.ligand:9296	VUNAKIZUMAB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	2.019525817	Abicipar pegol	ncit:C174693	ABICIPAR PEGOL	FALSE	FALSE	FALSE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	0.5527123287967842	AZD7762	iuphar.ligand:7713	AZD7762	FALSE	FALSE	TRUE
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	1.367387271762877	LOXO-101	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
EPHRIN TYPE-A RECEPTOR 2	hgnc:3386	EPHA2	TTD	2020.06.01	NULL	2.917092846427472	MEDI-547	drugbank:DB18360	MEDI-547	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	1.050153425	Methazolamide	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	ChEMBL	33	inhibitor	0.1666910197958555	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
LIVER CARBOXYLESTERASE	hgnc:1863	CES1	TTD	2020.06.01	NULL	1.141471113819445	GR148672X	iuphar.ligand:6701	GR148672X	FALSE	FALSE	FALSE
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	10.50153424713889	Camicinal	ncit:C166668	CAMICINAL	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.08178765	Androgen restored contraceptive	wikidata:Q85759692	ETHINYLESTRADIOL/DROSPIRENONE/PRASTERONE	FALSE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.8607814956671229	Virexxa	ncit:C114298	CRIDANIMOD SODIUM	FALSE	FALSE	FALSE
ENDOPLASMIC RETICULUM CHAPERONE BIP	hgnc:5238	HSPA5	TTD	2020.06.01	NULL	3.281729452230906	IT-139	drugbank:DB17145	IT-139	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.034544521	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	CC-8490	ncit:C38711	SELECTIVE ESTROGEN RECEPTOR MODULATOR CC-8490	FALSE	FALSE	FALSE
LYMPHOCYTE IGE RECEPTOR	hgnc:3612	FCER2	TTD	2020.06.01	NULL	31.50460274141669	Lumiliximab	ncit:C26448	GOMILIXIMAB	FALSE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	15.75230137070834	Remikiren	ncit:C73099	REMIKIREN	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.1426838892274307	RALIMETINIB	ncit:C143046	RALIMETINIB	FALSE	FALSE	FALSE
STERYL-SULFATASE	hgnc:11425	STS	TTD	2020.06.01	NULL	7.001022831425932	STX 64	ncit:C79827	IROSUSTAT	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR BETA-2	hgnc:1962	CHRNB2	TTD	2020.06.01	NULL	1.166837138570989	CYTISINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.078252863	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	0.3571950424196904	PMX-53	iuphar.ligand:579	PMX53	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.2983390411119005	Ketorolac	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
IODOTHYRONINE DEIODINASE TYPE I	hgnc:2883	DIO1	TTD	2020.06.01	NULL	5.250767124	Propylthiouracil	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.029465584	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.3271505995993426	DOV 21947	chembl:CHEMBL1818442	AMITIFADINE HYDROCHLORIDE	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	0.5834185692854945	Artemisinin	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
LACTOYLGLUTATHIONE LYASE	hgnc:4323	GLO1	TTD	2020.06.01	NULL	1.250182648468916	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	2.983390411119005	Eltrombopag	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.059667808	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	1.419126249613364	Pimagedine HCl	rxcui:1311669	PIMAGEDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.1278595890479573	Sotalol	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.1881995384791917	Ortataxel	ncit:C1867	ORTATAXEL	FALSE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	1.334940794127826	Moexipril	rxcui:30131	MOEXIPRIL	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.052824619	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	3.889457128569962	Veltuzumab	ncit:C48406	VELTUZUMAB	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1115286134997759	Estrone	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.035098711	Bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1132444383228493	Toremifene	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.2044691247495891	Venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	4.118248724368195	Drotrecogin alfa	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1491695205559502	Venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.2917092846427472	DAP-81	chembl:CHEMBL1242101	CHEMBL:CHEMBL1242101	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.1151484018326633	TESEVATINIB	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.5000730593875666	P276-00	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.300043836	Alvimopan	rxcui:1516803	ALVIMOPAN ANHYDROUS	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.1470803115845784	R-roscovitine	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.096167896	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
UROTENSIN II RECEPTOR	hgnc:4468	UTS2R	TTD	2020.06.01	NULL	1.810609352954982	SB-436811	iuphar.ligand:2164	SB-436811	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.6105543166941221	Org-25435	drugbank:DB12312	ORG-25435	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.033615667	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
CYTOCHROME P450 1B1	hgnc:2597	CYP1B1	TTD	2020.06.01	NULL	0.2273059360852575	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	1.312691780892362	THAPSIGARGIN	ncit:C128634	THAPSIGARGIN	FALSE	FALSE	FALSE
ALPHA-GLUCOSIDASE	hgnc:4296	GLA	TTD	2020.06.01	NULL	2.019525817	Maltose	rxcui:1311261	MALTOSE	TRUE	FALSE	FALSE
EPHB4	hgnc:3395	EPHB4	ChEMBL	33	inhibitor	5.469549087051511	TESEVATINIB	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	4.039051633514961	BAY-38-1315	chembl:CHEMBL1086624	CHEMBL:CHEMBL1086624	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-3	hgnc:4077	GABRA3	TTD	2020.06.01	NULL	0.072927321	Adipiplon	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.9723642821424906	AME-133v	chembl:CHEMBL2109346	AME-133V	FALSE	FALSE	FALSE
C-X-C MOTIF CHEMOKINE 10	hgnc:10637	CXCL10	TTD	2020.06.01	NULL	6.177373086552294	MDX-1100	iuphar.ligand:9047	ELDELUMAB	FALSE	FALSE	FALSE
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	17.50255707856483	CE-224535	drugbank:DB12113	CE-224535	FALSE	FALSE	FALSE
VITAMIN K-DEPENDENT PROTEIN C	hgnc:9451	PROC	TTD	2020.06.01	NULL	5.250767123569449	3K3A-APC	wikidata:Q123598631	3K3A-ACTIVATED PROTEIN C	FALSE	FALSE	FALSE
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	0.6250913242344582	Vatreptacog alfa (activated)	chembl:CHEMBL2108322	VATREPTACOG ALFA (ACTIVATED)	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1071585127259071	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	2.917092846427472	INO-8875	chembl:CHEMBL3545407	TRABODENOSON	FALSE	FALSE	FALSE
VITAMIN K EPOXIDE REDUCTASE COMPLEX 1	hgnc:23663	VKORC1	TTD	2020.06.01	NULL	2.625383561784724	Dicumarol	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	1.981421556063943	BIIB 022	chembl:CHEMBL2109356	BIIB-022	FALSE	FALSE	FALSE
SUBSTANCE-K RECEPTOR	hgnc:11527	TACR2	TTD	2020.06.01	NULL	10.50153424713889	Ibodutant	ncit:C166502	IBODUTANT	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inverse agonist	0.7721716358190367	MK-0249	drugbank:DB11910	MK-0249	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	2.561349816375341	Axicabtagene ciloleucel	rxcui:1987398	AXICABTAGENE CILOLEUCEL	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.051885051	Ergonovine	rxcui:4021	ERGONOVINE	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.591141552596803	Elagolix sodium	rxcui:2049847	ELAGOLIX SODIUM	TRUE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.3889457128569962	BIMU-1	iuphar.ligand:233	BIMU 1	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	0.1640864726115453	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.8950171233357017	Moricizine	rxcui:40169	MORICIZINE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	2.838252499226729	VESTIPITANT MESYLATE	ncit:C95195	VESTIPITANT MESYLATE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR	hgnc:3229	EGF	TTD	2020.06.01	NULL	8.751278539282415	Epidermal growth factor	rxcui:1427158	EPIDERMAL GROWTH FACTOR	FALSE	FALSE	FALSE
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	1.750255707856483	RG7221	ncit:C118578	VANUCIZUMAB	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.3070624048871023	BATEFENTEROL	ncit:C166503	BATEFENTEROL	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.2051080907644316	Indibulin	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
INTERLEUKIN-1 ALPHA	hgnc:5991	IL1A	TTD	2020.06.01	NULL	5.250767123569449	Xilonix	chembl:CHEMBL2109653	BERMEKIMAB	FALSE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	3.750547945	Tafluprost	rxcui:1244607	TAFLUPROST	TRUE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	ZATOSETRON MALEATE	ncit:C95281	ZATOSETRON MALEATE	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.1052961321571413	Tedatioxetine	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE	hgnc:1530	MICU1	TTD	2020.06.01	NULL	26.25383561784724	ALD-403	iuphar.ligand:10694	EPTINEZUMAB	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	2.917092846427472	GSK1325756	ncit:C169874	DANIRIXIN	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE LYN	hgnc:6735	LYN	TTD	2020.06.01	NULL	0.7876150685354174	Bafetinib	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.3977853881492007	MURAGLITAZAR	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	1.225178995499538	ABT-888	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	7.001022831425932	Olcegepant	ncit:C170245	OLCEGEPANT	FALSE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	2.386712328895204	Celgosivir	ncit:C79567	CELGOSIVIR	FALSE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR ALPHA	hgnc:6008	IL2RA	TTD	2020.06.01	NULL	2.059124362184098	Inolimomab	ncit:C170069	INOLIMOMAB	FALSE	FALSE	FALSE
INTERLEUKIN-12 BETA	hgnc:5970	IL12B	TTD	2020.06.01	NULL	3.750547945	ABT-874	ncit:C95321	BRIAKINUMAB	FALSE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	1.458546423213736	Combotox	ncit:C67061	DEGLYCOSYLATED RICIN A CHAIN-CONJUGATED ANTI-CD19/ANTI-CD22 IMMUNOTOXINS	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-1	hgnc:1955	CHRNA1	TTD	2020.06.01	NULL	0.8334550989792776	Decamethonium	ncit:C77363	DECAMETHONIUM	TRUE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.1022212937748757	AZD-1152-HQPA	iuphar.ligand:5663	BARASERTIB-HQPA	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	NLX-101	iuphar.ligand:3924	NLX-101	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.04362008	Amitriptyline	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.4070362111294147	Barbital	rxcui:1325	BARBITAL	TRUE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	1.923357921	Cisapride	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	1.750255707856483	Ethosuximide	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	0.9723642821424906	TECADENOSON	ncit:C77980	TECADENOSON	FALSE	FALSE	FALSE
ACETYL-COA CARBOXYLASE 2	hgnc:85	ACACB	TTD	2020.06.01	NULL	0.043430663	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.1457197166578015	Nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 22 MEMBER 8	hgnc:10972	SLC22A8	TTD	2020.06.01	NULL	2.045753424767318	Probenecid	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.024416494	Pimozide	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	1.009762908	Temanogrel	ncit:C96894	TEMANOGREL	FALSE	FALSE	FALSE
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	2.625383561784724	ARA 290	ncit:C171683	CIBINETIDE	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE ENDOTHELIAL	hgnc:7876	NOS3	TTD	2020.06.01	NULL	1.875273972703375	L-NAME	iuphar.ligand:5213	L-NAME	FALSE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	11.66837138570988	ORG-25935	drugbank:DB12220	ORG-25935	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.7095631248066824	AZD8683	chembl:CHEMBL3545222	AZD8683	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.5585922471882393	Xanomeline tartrate	ncit:C152927	XANOMELINE TARTRATE	FALSE	FALSE	FALSE
FREE FATTY ACID RECEPTOR 1	hgnc:4498	FFAR1	TTD	2020.06.01	NULL	3.750547945	Fasiglifam hemihydrate	ncit:C132780	FASIGLIFAM	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.3163112725041837	IUPHAR.LIGAND:66	iuphar.ligand:66	(S)-FLUROCARAZOLOL	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.3163112725041837	IUPHAR.LIGAND:118	iuphar.ligand:118	[3H]ELETRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.089756703	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	agonist	2.763561643983921	NAMODENOSON	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:218	iuphar.ligand:218	2-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1396480617970598	IUPHAR.LIGAND:142	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.020094784	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.027781837	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.070860555	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.034727296	IUPHAR.LIGAND:2	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.052090944	IUPHAR.LIGAND:109	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.016027983	IUPHAR.LIGAND:202	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:184	iuphar.ligand:184	LY86057	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1037701012563132	SB-773812	drugbank:DB16042	SB-773812	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.025123288	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:129	iuphar.ligand:129	S33084	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.046059361	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.081281225	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:256	iuphar.ligand:256	SB 204070	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.057574201	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.091159151	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.068458502	IUPHAR.LIGAND:7351	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	2.386712328895204	SB-649868	drugbank:DB14822	SB-649868	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:3248	iuphar.ligand:3248	[3H]5-HT	FALSE	FALSE	FALSE
NCBIGENE:1784	ncbigene:1784	DNCM	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:8120	iuphar.ligand:8120	COMPOUND 13D [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1787	hgnc:2977	TRDMT1	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:8120	iuphar.ligand:8120	COMPOUND 13D [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:2611	hgnc:4147	GAPDHP69	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10200	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	inhibitor	6.300920548	BURIXAFOR	ncit:C88323	BURIXAFOR	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:7706	iuphar.ligand:7706	AZD3463	FALSE	FALSE	TRUE
NCBIGENE:2919	hgnc:4602	CXCL1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:5289	iuphar.ligand:5289	WWL70	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:503	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.054243462	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.029057925	IUPHAR.LIGAND:516	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.034341185	IUPHAR.LIGAND:522	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.034341185	IUPHAR.LIGAND:521	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.053964719	IUPHAR.LIGAND:12574	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:7310	rxcui:10634	TOLAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:12576	rxcui:18475	ATIPAMEZOLE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:9868	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:9868	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:9043	rxcui:1999574	APALUTAMIDE	TRUE	FALSE	TRUE
GRM5	hgnc:4597	GRM5	ChEMBL	33	modulator	2.917092846427472	RASEGLURANT	ncit:C152157	RASEGLURANT	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:2864	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:10439	rxcui:2180325	DAROLUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:6945	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
NCBIGENE:2767	hgnc:4379	GNA11	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9754	ncit:C83968	MOFEGILINE	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:3556	iuphar.ligand:3556	APELIN-17	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:406	iuphar.ligand:406	[3H]DPCPX	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:470	iuphar.ligand:470	MRS1191	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.077330885	IUPHAR.LIGAND:3283	iuphar.ligand:3283	SCH442416	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.077330885	IUPHAR.LIGAND:403	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
NCBIGENE:2719	hgnc:4451	GPC3	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:10445	iuphar.ligand:10445	COMPOUND 23 [PMID: 31398032]	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8768	iuphar.ligand:8768	COMPOUND 38 [PMID: 20817473]	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	blocker	0.5173169579871378	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:7432	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:10131	iuphar.ligand:10131	UNC4203	FALSE	FALSE	FALSE
NCBIGENE:2957	hgnc:4646	GTF2A1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9672	iuphar.ligand:9672	FX1	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	1.250182648468916	MF101	drugbank:DB05052	MF101	FALSE	FALSE	FALSE
NCBIGENE:1467	hgnc:2471	CSRP2P1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8437	iuphar.ligand:8437	COMPOUND 101 [PMID: 21596927]	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:541	iuphar.ligand:541	CGP 20712A	FALSE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:3415	iuphar.ligand:3415	[3H]CGS23131	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	agonist	0.042619863	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:10402	iuphar.ligand:10402	ZAK INHIBITOR 6P	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:2487	iuphar.ligand:2487	LTB4	FALSE	FALSE	FALSE
NCBIGENE:1786	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:8120	iuphar.ligand:8120	COMPOUND 13D [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.074797252	IUPHAR.LIGAND:6494	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.061197752	IUPHAR.LIGAND:5891	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	agonist	0.039068208	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:7521	iuphar.ligand:7521	COMPOUND 36 [PMID: 24000170]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:7522	iuphar.ligand:7522	COMPOUND 38 [PMID: 24000170]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7527	iuphar.ligand:7527	ISOXAZOLE AZEPINE COMPOUND 3	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:642	iuphar.ligand:642	[LEU9,DES-ARG10]KALLIDIN	FALSE	FALSE	FALSE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:574	iuphar.ligand:574	C5A DES-ARG	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:3853	iuphar.ligand:3853	ACPHE-ORN-PRO-D-CHA-TRP-ARG	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5761	iuphar.ligand:5761	FLPLAR	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	1.019566431761058	EPROTIROME	ncit:C81533	EPROTIROME	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8380	iuphar.ligand:8380	AC-RHYPLWR	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:3774	iuphar.ligand:3774	[125I]C5A (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8381	iuphar.ligand:8381	COMPOUND 21 [PMID: 25259874]	FALSE	FALSE	FALSE
NCBIGENE:1953	hgnc:3232	MEGF6	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:4314	iuphar.ligand:4314	SITS	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.1582152052299645	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
NCBIGENE:1627	hgnc:2695	DBN1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8674	iuphar.ligand:8674	GRASSYSTATIN A	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.6019397937072561	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:1549	hgnc:2611	CYP2A7	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8140	iuphar.ligand:8140	COMPOUND 2C [PMID: 22115617]	FALSE	FALSE	FALSE
NCBIGENE:528	hgnc:856	ATP6V1C1	GuideToPharmacology	2024.1	activator	5.250767123569449	IUPHAR.LIGAND:4318	iuphar.ligand:4318	SZ(+)-(S)-202-791	FALSE	FALSE	FALSE
NCBIGENE:533	hgnc:861	ATP6V0B	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:7766	iuphar.ligand:7766	TROX-1	FALSE	FALSE	FALSE
NCBIGENE:528	hgnc:856	ATP6V1C1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2733	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	inhibitor	0.3431873936973497	IUPHAR.LIGAND:2524	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.042174836	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
NCBIGENE:2345	ncbigene:2345	FNZ	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8674	iuphar.ligand:8674	GRASSYSTATIN A	FALSE	FALSE	FALSE
NCBIGENE:388	hgnc:668	RHOB	GuideToPharmacology	2024.1	blocker	1.458546423213736	IUPHAR.LIGAND:4269	iuphar.ligand:4269	NNC55-0396	FALSE	FALSE	FALSE
NCBIGENE:388	hgnc:668	RHOB	GuideToPharmacology	2024.1	blocker	0.3431873936973497	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8613	iuphar.ligand:8613	COMPOUND 1B [PMID: 16290936]	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10029	iuphar.ligand:10029	AM6545	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:4382	iuphar.ligand:4382	CCL18	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.041672755	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:758	iuphar.ligand:758	CCL5	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.5000730593875666	IUPHAR.LIGAND:771	iuphar.ligand:771	CCL2	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:3910	iuphar.ligand:3910	R5-HIV-1 GP120	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:799	iuphar.ligand:799	[125I]CCL4 (HUMAN)	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	1.346350544504987	PRUCALOPRIDE	rxcui:2107310	PRUCALOPRIDE	TRUE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:9620	iuphar.ligand:9620	LORECIVIVINT	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:4153	iuphar.ligand:4153	CFTRINH-172	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:4198	iuphar.ligand:4198	GATX1	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.028536778	IUPHAR.LIGAND:1909	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:9551	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:11689	iuphar.ligand:11689	COMPOUND 10 [PMID: 34279934]	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.4280516676822921	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3729	iuphar.ligand:3729	CYTOKINE DOMAIN OF TYROSYL TRNA SYNTHETASE	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:839	iuphar.ligand:839	NBI-74330	FALSE	FALSE	FALSE
NCBIGENE:74	hgnc:147	ACTG1P2	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10390	iuphar.ligand:10390	JMS-17-2	FALSE	FALSE	FALSE
PARP3	hgnc:273	PARP3	ChEMBL	33	inhibitor	0.3977853881492008	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NCBIGENE:3165	ncbigene:3165	HMS1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11324	iuphar.ligand:11324	PF‐06928215	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:10547	iuphar.ligand:10547	THAL-SNS-032	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.2333674277141978	IUPHAR.LIGAND:7934	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:8176	iuphar.ligand:8176	BS-194	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:5923	iuphar.ligand:5923	ALOISINE	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:5952	iuphar.ligand:5952	CDK4 INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:7934	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:10530	iuphar.ligand:10530	BSJ-03-204	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:10532	iuphar.ligand:10532	BSJ-03-123	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:8176	iuphar.ligand:8176	BS-194	FALSE	FALSE	FALSE
NCBIGENE:1359	hgnc:2298	CPA3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8310	rxcui:2286252	OSILODROSTAT	TRUE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	0.280789686	IUPHAR.LIGAND:7073	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
NCBIGENE:1365	hgnc:2045	CLDN3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8819	iuphar.ligand:8819	CTA091	FALSE	FALSE	FALSE
NCBIGENE:1324	hgnc:2615	CYP2B6	GuideToPharmacology	2024.1	inhibitor	0.2461297089173179	IUPHAR.LIGAND:7622	rxcui:10473	THIOTEPA	TRUE	FALSE	FALSE
NCBIGENE:1369	hgnc:2312	CPN1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8819	iuphar.ligand:8819	CTA091	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:7118	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:4639	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
NCBIGENE:3002	hgnc:4709	GZMB	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9932	iuphar.ligand:9932	SETANAXIB	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:3354	iuphar.ligand:3354	LTC4	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1161674142382621	IUPHAR.LIGAND:10652	ncit:C170277	OXYCODEGOL	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10342	rxcui:2121751	SOLRIAMFETOL	TRUE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:4605	iuphar.ligand:4605	[3H]WIN35428	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1548898856510162	IUPHAR.LIGAND:1631	iuphar.ligand:1631	&BETA;-FNA	FALSE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	ChEMBL	33	modulator	0.3125456621172291	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.010101514	IUPHAR.LIGAND:1627	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.2323348284765243	IUPHAR.LIGAND:9838	iuphar.ligand:9838	UFP-505	FALSE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:9893	iuphar.ligand:9893	COMPOUND 9 [PMID: 20718420]	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.004214099	IUPHAR.LIGAND:7279	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.1179947668217853	IUPHAR.LIGAND:6674	iuphar.ligand:6674	NGB 2904	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.060077427	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9620	iuphar.ligand:9620	LORECIVIVINT	FALSE	FALSE	FALSE
CASP5	hgnc:1506	CASP5	ChEMBL	33	inhibitor	4.039051633514962	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
NCBIGENE:1566	ncbigene:1566	CYP2D7BP	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8666	iuphar.ligand:8666	COMPOUND 17 [PMID: 23916253]	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:12352	iuphar.ligand:12352	COMPOUND 15A [PMID: 36642961]	FALSE	FALSE	FALSE
NCBIGENE:1831	hgnc:3051	TSC22D3	GuideToPharmacology	2024.1	inhibitor	0.6731752722524936	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.3271505995993426	ESREBOXETINE	rxcui:60842	REBOXETINE	TRUE	FALSE	FALSE
NCBIGENE:1824	hgnc:3036	DSC2	GuideToPharmacology	2024.1	inhibitor	4.773424657790409	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:1827	hgnc:3040	RCAN1	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3160	iuphar.ligand:3160	NE11808	FALSE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	ChEMBL	33	modulator	0.364636606	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	0.3977853881492008	IUPHAR.LIGAND:1054	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
NCBIGENE:227	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	modulator	6.563458904461812	IUPHAR.LIGAND:12859	iuphar.ligand:12859	FHQC	FALSE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:8418	iuphar.ligand:8418	COMPOUND A [PMID 24997608]	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:9769	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
SELP	hgnc:10721	SELP	ChEMBL	33	inhibitor	5.250767123569449	BIMOSIAMOSE	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:8183	iuphar.ligand:8183	PD166285	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8862	iuphar.ligand:8862	BLU-9931	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12874	iuphar.ligand:12874	RESIGRATINIB	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.092606122	IUPHAR.LIGAND:7877	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.108040476	IUPHAR.LIGAND:7877	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
NCBIGENE:3175	hgnc:8138	ONECUT1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11482	iuphar.ligand:11482	SAFIT2	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.030386384	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.4773424657790409	POLMACOXIB	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12869	iuphar.ligand:12869	IRPAGRATINIB	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	NULL	0.2734774543525755	IUPHAR.LIGAND:5086	iuphar.ligand:5086	VEGFB	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:9905	iuphar.ligand:9905	COMPOUND 8I [PMID: 22765894]	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.006250913	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.058602312	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.010255405	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NQO1	hgnc:2874	NQO1	ChEMBL	33	modulator	2.019525817	VATIQUINONE	ncit:C152840	VATIQUINONE	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6245	iuphar.ligand:6245	T21/DP107	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6267	iuphar.ligand:6267	PSM&ALPHA;3	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1907	iuphar.ligand:1907	L-888,607	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1040	iuphar.ligand:1040	WRWWWW	FALSE	FALSE	FALSE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:1040	iuphar.ligand:1040	WRWWWW	FALSE	FALSE	FALSE
NCBIGENE:229	hgnc:417	ALDOB	GuideToPharmacology	2024.1	antibody	10.50153425	IUPHAR.LIGAND:10197	iuphar.ligand:10197	VANTICTUMAB	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	ChEMBL	33	inhibitor	0.729273212	LIFITEGRAST	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.045226246	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:230	hgnc:418	ALDOC	GuideToPharmacology	2024.1	antibody	10.50153425	IUPHAR.LIGAND:10197	iuphar.ligand:10197	VANTICTUMAB	FALSE	FALSE	FALSE
NCBIGENE:234	hgnc:4044	FZD6	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:3549	iuphar.ligand:3549	WNT-3A	FALSE	FALSE	FALSE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:8836	iuphar.ligand:8836	PP1	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4257	iuphar.ligand:4257	MRK016	FALSE	FALSE	FALSE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	2.625383561784724	POLMACOXIB	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.056142926	IUPHAR.LIGAND:3364	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:3898	iuphar.ligand:3898	M35	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6121	iuphar.ligand:6121	GALP(1-32) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6093	iuphar.ligand:6093	GALANIN(10-29) (RAT/MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:11419	iuphar.ligand:11419	QU-SPX	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:3898	iuphar.ligand:3898	M35	FALSE	FALSE	FALSE
SELL	hgnc:10720	SELL	ChEMBL	33	inhibitor	23.33674277141977	RIVIPANSEL	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:3897	iuphar.ligand:3897	M32	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3898	iuphar.ligand:3898	M35	FALSE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:4583	iuphar.ligand:4583	(R/S) EF-1500	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:4141	iuphar.ligand:4141	ATPO	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.4688184931758437	IUPHAR.LIGAND:4304	iuphar.ligand:4304	S18986	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:3505	iuphar.ligand:3505	L-168,049	FALSE	FALSE	FALSE
NCBIGENE:451	hgnc:769	ASS1P6	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:4102	iuphar.ligand:4102	2,4-EPI-NEODYSIHERBAINE	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.066297565	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
NCBIGENE:453	hgnc:771	ASS1P8	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:4231	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:4066	iuphar.ligand:4066	(+)-HA966	FALSE	FALSE	FALSE
NCBIGENE:454	hgnc:772	ASS1P9	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:4185	iuphar.ligand:4185	DYSIHERBAINE	FALSE	FALSE	FALSE
NCBIGENE:454	hgnc:772	ASS1P9	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:4075	iuphar.ligand:4075	[3H]SYM2081	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8886	iuphar.ligand:8886	COMPOUND 8 [PMID: 17562362}	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1209854175937661	IUPHAR.LIGAND:2361	drugbank:DB01931	5,7-DICHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.036013492	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:9057	iuphar.ligand:9057	PF-03463275	FALSE	FALSE	FALSE
NCBIGENE:1707	hgnc:2435	CSF2RA	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:4942	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
RBX1	hgnc:9928	RBX1	ChEMBL	33	inhibitor	0.2027323213733378	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:4853	iuphar.ligand:4853	[SER11](N-CNP,C-ANP)PBNP2-15	FALSE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:725	rxcui:314709	ORNITHINE, (L)-ISOMER	TRUE	FALSE	FALSE
NCBIGENE:1719	hgnc:2861	DHFR	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:6969	rxcui:2048018	PEGFILGRASTIM-JMDB	TRUE	FALSE	FALSE
NCBIGENE:1719	hgnc:2861	DHFR	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:4934	rxcui:70167	LENOGRASTIM	TRUE	FALSE	FALSE
NCBIGENE:1720	hgnc:52354	DHFRP3	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:4944	iuphar.ligand:4944	GROWTH HORMONE 2	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5793	iuphar.ligand:5793	COMPOUND 8F [PMID: 20615702]	FALSE	FALSE	FALSE
NCBIGENE:400	hgnc:692	ARL1	GuideToPharmacology	2024.1	blocker	2.100306849	IUPHAR.LIGAND:2355	ncit:C81347	CILOBRADINE	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:8367	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:11120	iuphar.ligand:11120	ACY-738	FALSE	FALSE	FALSE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:8365	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
GFRA1	hgnc:4243	GFRA1	ChEMBL	33	agonist	13.12691780892362	LIATERMIN	ncit:C1459	LIATERMIN	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:7916	iuphar.ligand:7916	SANTACRUZAMATE A	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.1058622403945453	IUPHAR.LIGAND:7008	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.1164249916534246	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:7490	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1202	iuphar.ligand:1202	UR-PG55B	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.046425881	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.086219493	IUPHAR.LIGAND:1222	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.2573905452730122	IUPHAR.LIGAND:1237	iuphar.ligand:1236	(R)-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.035574303	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
NCBIGENE:638	hgnc:1051	BIK	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:3040	iuphar.ligand:3040	(S)-3-HYDROXY-3-METHYLGLUTARYL-COA	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3003	iuphar.ligand:3003	COMPOUND 2D [PMID: 2153213]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:7993	iuphar.ligand:7993	COMPOUND 3 [DREYER ET AL., 1991]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:2951	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.034727296	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
NCBIGENE:3094	hgnc:4912	HINT1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:10438	iuphar.ligand:10438	COMPOUND 24 [PMID: 31343176]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5650	iuphar.ligand:5650	1-PALMITOYL-LYSOPHOSPHATIDYLCHOLINE	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.071148606	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:10541	iuphar.ligand:10541	MSMB (91-114)	FALSE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	0.6081969641200136	IUPHAR.LIGAND:11467	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8222	iuphar.ligand:8222	BETA-CARBOLINE	FALSE	FALSE	FALSE
PDK3	hgnc:8811	PDK3	ChEMBL	33	inhibitor	4.375639269641208	SODIUM DICHLOROACETATE	rxcui:1366930	SODIUM DICHLOROACETATE	TRUE	FALSE	FALSE
NCBIGENE:2885	hgnc:4566	GRB2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12340	iuphar.ligand:12340	LY3410738	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:12428	iuphar.ligand:12428	PARTHENOLIDE	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:5716	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:12350	iuphar.ligand:12350	CEE321	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:10458	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:10157	iuphar.ligand:10157	JAK3 INHIBITOR 34	FALSE	FALSE	FALSE
PRIM1	hgnc:9369	PRIM1	ChEMBL	33	inhibitor	0.6250913242344582	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:1624	ncit:C65596	ETONITAZENE	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1600	iuphar.ligand:1600	&ALPHA;-NEOENDORPHIN	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9759	iuphar.ligand:9759	MP1104	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.041508041	IUPHAR.LIGAND:8007	iuphar.ligand:8007	BX-912	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.1037701012563132	IUPHAR.LIGAND:12865	iuphar.ligand:12865	CANLITINIB	FALSE	FALSE	FALSE
ITGB6	hgnc:6161	ITGB6	ChEMBL	33	inhibitor	6.563458904461812	STX-100	drugbank:DB16334	STX-100	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.02075402	IUPHAR.LIGAND:9133	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1651184630053286	IUPHAR.LIGAND:10420	iuphar.ligand:10420	CHMFL-KIT-64	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:5055	iuphar.ligand:5055	STEM CELL FACTOR	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.070765056	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:525	hgnc:853	ATP6V1B1	GuideToPharmacology	2024.1	blocker	0.5250767123569451	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:2321	iuphar.ligand:2321	UCL1848	FALSE	FALSE	FALSE
NCBIGENE:434	hgnc:745	ASIP	GuideToPharmacology	2024.1	blocker	1.050153425	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:437	hgnc:6266	KCNJ5	GuideToPharmacology	2024.1	activator	0.729273212	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
NCBIGENE:443	hgnc:756	ASPA	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:7662	iuphar.ligand:7662	VU0405601	FALSE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.2187819634820604	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	4.039051633514961	IUPHAR.LIGAND:7669	iuphar.ligand:7669	QO-58	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	0.252440727	IUPHAR.LIGAND:2598	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6714	iuphar.ligand:6714	COMPOUND 6 [PMID: 22533316]	FALSE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:5702	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.577007376	IUPHAR.LIGAND:8937	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
NCBIGENE:2886	hgnc:4567	GRB7	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9007	iuphar.ligand:9007	GSK180	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.1154014752432846	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.088248187	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:8068	iuphar.ligand:8068	WH-4-023	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:8836	iuphar.ligand:8836	PP1	FALSE	FALSE	FALSE
NCBIGENE:1570	hgnc:6656	LNPEP	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8666	iuphar.ligand:8666	COMPOUND 17 [PMID: 23916253]	FALSE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:254	hgnc:6585	LHCGR	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:3775	iuphar.ligand:3775	[125I]CHORIONIC GONADOTROPIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.2778183663264259	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:2752	iuphar.ligand:2752	27-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:2055	hgnc:2079	CLN8	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:10402	iuphar.ligand:10402	ZAK INHIBITOR 6P	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:9499	iuphar.ligand:9499	ONO-7300243	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:6987	iuphar.ligand:6987	ANTI-BRP-LPA	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	0.8078103267029924	IUPHAR.LIGAND:2910	drugbank:DB07780	FARNESYL DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2684	ncbigene:2684	GGTL1	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:7027	iuphar.ligand:7027	GSK-J1	FALSE	FALSE	FALSE
NCBIGENE:2681	hgnc:4253	GGTA1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7027	iuphar.ligand:7027	GSK-J1	FALSE	FALSE	FALSE
NCBIGENE:2094	ncbigene:2094	ERVT4	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:8163	iuphar.ligand:8163	COMPOUND 33 [PMID: 19364658]	FALSE	FALSE	FALSE
NCBIGENE:1217	hgnc:26439	SLC47A2	GuideToPharmacology	2024.1	NULL	0.9723642821424908	IUPHAR.LIGAND:4575	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1323	iuphar.ligand:1323	MT-II	FALSE	FALSE	FALSE
NCBIGENE:2847	hgnc:4479	MCHR1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:11086	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:10460	iuphar.ligand:10460	PAMUFETINIB	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6337	iuphar.ligand:6337	VU0469650	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6329	iuphar.ligand:6328	[3H]2,2,2-TEMPS	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	modulator	0.375054795	IUPHAR.LIGAND:7921	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:2065	hgnc:3431	ERBB3	GuideToPharmacology	2024.1	inhibitor	0.3431873936973496	IUPHAR.LIGAND:6006	iuphar.ligand:6006	MEK INHIBITOR I	FALSE	FALSE	FALSE
NCBIGENE:2064	hgnc:3430	ERBB2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:6006	iuphar.ligand:6006	MEK INHIBITOR I	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	0.5303805175322677	IUPHAR.LIGAND:5998	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	modulator	0.3281729452230906	IUPHAR.LIGAND:7921	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.072125922	IUPHAR.LIGAND:302	iuphar.ligand:302	OXOTREMORINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.1262203635473425	IUPHAR.LIGAND:341	iuphar.ligand:341	ALCURONIUM	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:10712	iuphar.ligand:10712	MK-7622	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:300	iuphar.ligand:300	METHYLFURMETHIDE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.5527123287967841	IUPHAR.LIGAND:7634	iuphar.ligand:7634	C7/3-PHTH	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:10129	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:293	iuphar.ligand:293	NNC 11-1607	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:335	iuphar.ligand:335	G&OUML; 7874	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:10470	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:332	iuphar.ligand:332	N-BENZYL BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:8586	iuphar.ligand:8586	AE9C90CB	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:349	rxcui:11201	VINCAMINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:302	iuphar.ligand:302	OXOTREMORINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.049723174	IUPHAR.LIGAND:325	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:310	iuphar.ligand:310	HEXAHYDROSILADIFENIDOL	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:293	iuphar.ligand:293	NNC 11-1607	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:330	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.099446347	IUPHAR.LIGAND:294	rxcui:194	ACETYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:10470	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.03140411	IUPHAR.LIGAND:305	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.079557078	IUPHAR.LIGAND:298	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:12486	iuphar.ligand:12486	[3H]IPEROXO	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.041872146	IUPHAR.LIGAND:305	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:10129	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:307	iuphar.ligand:307	4-DAMP	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.7955707762984014	IUPHAR.LIGAND:8687	iuphar.ligand:8687	ML380	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.1591141552596803	IUPHAR.LIGAND:344	iuphar.ligand:344	N-CHLOROMETHYL-BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:7779	iuphar.ligand:7779	[125I]S70254	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1622	iuphar.ligand:1622	DYNORPHIN B	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.048083948	IUPHAR.LIGAND:1673	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:1216	hgnc:25588	SLC47A1	GuideToPharmacology	2024.1	NULL	0.5834185692854945	IUPHAR.LIGAND:4575	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
NCBIGENE:970	hgnc:11937	CD70	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:4167	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:3001	hgnc:4708	GZMA	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9932	iuphar.ligand:9932	SETANAXIB	FALSE	FALSE	FALSE
NCBIGENE:750	hgnc:1197	GAS8-AS1	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:2614	iuphar.ligand:2614	ATX-II	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:2625	iuphar.ligand:2625	SAXITOXIN	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:2614	iuphar.ligand:2614	ATX-II	FALSE	FALSE	FALSE
NCBIGENE:981	hgnc:23089	SLC13A5	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12850	iuphar.ligand:12850	PF-06761281	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:9980	iuphar.ligand:9980	PF‐06526290	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:4637	ncit:C75172	NISOXETINE	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.157680694	IUPHAR.LIGAND:7285	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	modulator	0.9053046764774912	IUPHAR.LIGAND:10693	iuphar.ligand:10693	BNC375	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2092	iuphar.ligand:2092	NEUROPEPTIDE-&GAMMA;	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:5771	iuphar.ligand:5771	ZM 253270	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:5778	iuphar.ligand:5778	ZM-274773	FALSE	FALSE	FALSE
NCBIGENE:1219	hgnc:10956	SLCO1A2	GuideToPharmacology	2024.1	NULL	2.187819634820604	IUPHAR.LIGAND:3819	iuphar.ligand:3819	[3H]DPDPE	FALSE	FALSE	FALSE
NCBIGENE:630	hgnc:7981	NR4A2	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:12651	iuphar.ligand:12651	COMPOUND 29 [VIETOR, ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:1219	hgnc:10956	SLCO1A2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4738	iuphar.ligand:4738	NARINGIN	FALSE	FALSE	FALSE
NCBIGENE:1019	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.064111931	IUPHAR.LIGAND:516	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1722	iuphar.ligand:1722	MRS2298	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	0.2419708351875322	IUPHAR.LIGAND:1712	iuphar.ligand:1712	ADP	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11451	iuphar.ligand:11451	PSB-16133	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:5910	iuphar.ligand:5910	RP-5-OME-UDP&ALPHA;B	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1860	ncit:C77989	APAFANT	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1850	iuphar.ligand:1850	ABT-491	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3305	iuphar.ligand:3305	M65	FALSE	FALSE	FALSE
NCBIGENE:347	hgnc:612	APOD	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4048	ncit:C169794	ATOPAXAR	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:3741	iuphar.ligand:3741	SLIGRL-NH2	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:10268	iuphar.ligand:10268	I-191	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:4599	iuphar.ligand:4599	[14C]GLYSAR	FALSE	FALSE	FALSE
NCBIGENE:3171	hgnc:5023	FOXA3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11400	iuphar.ligand:11400	AG-17724	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:2689	iuphar.ligand:2689	L-796449	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.084281976	IUPHAR.LIGAND:10096	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:8805	iuphar.ligand:8805	COMPOUND 82 [PMID: 21332118]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.065552648	IUPHAR.LIGAND:8059	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:8383	iuphar.ligand:8383	BIMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.073746729	IUPHAR.LIGAND:8527	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.053633985	IUPHAR.LIGAND:7951	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.049164486	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.026816992	IUPHAR.LIGAND:7933	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:8383	iuphar.ligand:8383	BIMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.075768645	IUPHAR.LIGAND:7951	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:11732	iuphar.ligand:11732	BAY-8400	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:8382	iuphar.ligand:8382	VS-5584	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:9692	iuphar.ligand:9692	STK16-IN-1	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:7795	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
NCBIGENE:2151	hgnc:3539	F2RL2	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:5701	iuphar.ligand:5701	PI-103	FALSE	FALSE	FALSE
NCBIGENE:1296	hgnc:2216	COL8A2	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:5285	rxcui:24506	VINPOCETINE	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:7399	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
NCBIGENE:1302	hgnc:2187	COL11A2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9852	iuphar.ligand:9852	MK-0359	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:8468	iuphar.ligand:8468	ME0328	FALSE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7337	iuphar.ligand:7337	ELND006	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.2134458180312784	IUPHAR.LIGAND:7460	rxcui:1005920	ULIPRISTAL ACETATE	TRUE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.2134458180312784	IUPHAR.LIGAND:7460	rxcui:1005920	ULIPRISTAL ACETATE	TRUE	FALSE	FALSE
NCBIGENE:2181	hgnc:3570	ACSL3	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:9382	iuphar.ligand:9382	NVP-TAE 226	FALSE	FALSE	FALSE
NCBIGENE:1213	hgnc:2092	CLTC	GuideToPharmacology	2024.1	NULL	0.06697407	IUPHAR.LIGAND:4674	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1807	iuphar.ligand:1807	[PHE23]PTH-(1-34) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3803	iuphar.ligand:3803	[125I]QRFP43 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:598	hgnc:992	BCL2L1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:10143	iuphar.ligand:10143	SR1001	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:10089	iuphar.ligand:10089	PN10	FALSE	FALSE	FALSE
NCBIGENE:2630	hgnc:4178	GBA1LP	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:6822	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
NCBIGENE:2630	hgnc:4178	GBA1LP	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:6802	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
NCBIGENE:1527	hgnc:2563	TEX28	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:5683	iuphar.ligand:5683	GSK-1838705A	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.4039051633514961	IUPHAR.LIGAND:8346	iuphar.ligand:8346	A(4-24)(B7-24)H2	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.4039051633514961	IUPHAR.LIGAND:1994	iuphar.ligand:1994	RELAXIN	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:12502	iuphar.ligand:12502	LY3540378	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.4039051633514961	IUPHAR.LIGAND:1988	iuphar.ligand:1988	RELAXIN-1	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:11495	iuphar.ligand:11495	BMS-986104 DERIVATIVE 24	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:9492	iuphar.ligand:9492	COMPOUND 43 [PMID: 26751273]	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:9492	iuphar.ligand:9492	COMPOUND 43 [PMID: 26751273]	FALSE	FALSE	FALSE
NCBIGENE:2198	ncbigene:2198	FAUNA@	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5678	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ITGB8	hgnc:6163	ITGB8	ChEMBL	33	inhibitor	8.751278539282415	ABITUZUMAB	ncit:C82422	ABITUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2291	hgnc:28646	NIM1K	GuideToPharmacology	2024.1	inhibitor	7.501095890813499	IUPHAR.LIGAND:8114	drugbank:DB07149	(7S)-2-(2-AMINOPYRIMIDIN-4-YL)-7-(2-FLUOROETHYL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE	FALSE	FALSE	FALSE
NCBIGENE:2211	hgnc:11388	STK10	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:1534	hgnc:2571	CYB561	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10739	iuphar.ligand:10739	PO-322	FALSE	FALSE	FALSE
NCBIGENE:952	hgnc:1667	CD38	GuideToPharmacology	2024.1	inhibitor	0.3431873936973497	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.076098074	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3111	iuphar.ligand:3111	COMPOUND 3F [PMID: 12238936]	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:6047	iuphar.ligand:6047	SYK INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3124	iuphar.ligand:3124	COMPOUND 19 [PMID: 19191557]	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	3.962843112127886	DALOTUZUMAB	rxcui:1432293	DALOTUZUMAB	FALSE	TRUE	TRUE
NCBIGENE:2290	hgnc:3811	FOXG1	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:8213	iuphar.ligand:8213	COMPOUND R-16 [PMID: 21967808]	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	0.251232877	IUPHAR.LIGAND:2147	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	7.876150685354174	LERONLIMAB	ncit:C137824	LERONLIMAB	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2637	rxcui:13982	TIRATRICOL	FALSE	FALSE	FALSE
NCBIGENE:392	hgnc:673	ARHGAP1	GuideToPharmacology	2024.1	activator	3.500511415712967	IUPHAR.LIGAND:2794	iuphar.ligand:2794	PHOSPHATIDYL (3,5) INOSITOL BISPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6297	iuphar.ligand:6297	O3	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6302	iuphar.ligand:6302	ARTEPILLIN C	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.099446347	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:6386	iuphar.ligand:6386	ML SA1	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.093763699	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:12757	iuphar.ligand:12757	A-1165442	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4228	iuphar.ligand:4228	JNJ17203212	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	2.386712328895204	IUPHAR.LIGAND:11377	iuphar.ligand:11377	CITRUSININE II	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.2234368988752957	IUPHAR.LIGAND:9403	iuphar.ligand:9403	RO3280	FALSE	FALSE	FALSE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:6798	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
NCBIGENE:1836	hgnc:10994	SLC26A2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10131	iuphar.ligand:10131	UNC4203	FALSE	FALSE	FALSE
TNC	hgnc:5318	TNC	ChEMBL	33	binder	6.563458904461812	81C6 131I	chembl:CHEMBL2109582	81C6 131I	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:10527	iuphar.ligand:10527	LASW1393	FALSE	FALSE	FALSE
NCBIGENE:3223	hgnc:5128	HOXC6	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12479	iuphar.ligand:12479	BAY-805	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2258	iuphar.ligand:2258	PACAP-38	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2275	iuphar.ligand:2275	PHV	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:2173	iuphar.ligand:2173	OPC-51803	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2184	iuphar.ligand:2184	D[D-PAL2]AVP	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2268	iuphar.ligand:2268	PG 97-269	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	DEFLAZACORT	rxcui:22396	DEFLAZACORT	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	CIViC	10-Apr-24	NULL	1.367387271762877	LAROTRECTINIB	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.1151484018326633	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
FN1	hgnc:3778	FN1	CIViC	10-Apr-24	NULL	0.2692701089009974	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.055441823	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
RXRA	hgnc:10477	RXRA	ChEMBL	33	inhibitor	0.1750255707856483	DANTHRON	rxcui:22293	DANTHRON	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	2.080014029626545	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
WT1	hgnc:12796	WT1	CIViC	10-Apr-24	NULL	0.044385183	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	1.111273465305703	MOBOCERTINIB	rxcui:2570736	MOBOCERTINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.1944728564284981	TIRBANIBULIN	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	1.029562181092049	AMG-888	chembl:CHEMBL2109396	AMG-888	FALSE	FALSE	FALSE
DLL3	hgnc:2909	DLL3	CIViC	10-Apr-24	NULL	78.76150685354175	ROVALPITUZUMAB TESIRINE	ncit:C107678	ROVALPITUZUMAB TESIRINE	FALSE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	CIViC	10-Apr-24	NULL	0.095295229	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
NF2	hgnc:7773	NF2	CIViC	10-Apr-24	NULL	0.3365876361262468	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	CIViC	10-Apr-24	NULL	0.1495945049449986	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	0.2282942227638891	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CIViC	10-Apr-24	NULL	0.084553416	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
KDM6A	hgnc:12637	KDM6A	CIViC	10-Apr-24	NULL	5.250767123569449	BET INHIBITOR	ncit:C128462	BET INHIBITOR	FALSE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inverse agonist	0.2117244807890907	BILASTINE	ncit:C73045	BILASTINE	TRUE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	CIViC	10-Apr-24	NULL	0.290901226	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.2287915957982331	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	0.1620607136904151	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.011049594	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	BEZAFIBRATE	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
GNA11	hgnc:4379	GNA11	CIViC	10-Apr-24	NULL	0.3281729452230906	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.020257589	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
PML	hgnc:9113	PML	CIViC	10-Apr-24	NULL	1.346350544504987	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
CD3D	hgnc:1673	CD3D	ChEMBL	33	modulator	0.6563458904461813	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	CIViC	10-Apr-24	NULL	0.051731696	ALPELISIB	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.1725162436059257	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
ERCC1	hgnc:3433	ERCC1	CIViC	10-Apr-24	NULL	0.546954909	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	0.375054795	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.4948366922735607	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.045658845	Alvocidib	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1826353782111113	GSK1838705A	iuphar.ligand:5683	GSK-1838705A	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2199274187882492	Ravoxertinib	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1718182959283197	LXH 254	ncit:C125003	NAPORAFENIB	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	modulator	0.8401227397711121	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.026604123	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.3665456979804153	SCH772984	iuphar.ligand:8056	SCH772984	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.021992742	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	Tubastatin A	iuphar.ligand:9702	TUBASTATIN A	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	CGM097	ncit:C104280	P53/HDM2 INTERACTION INHIBITOR CGM097	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.032342267	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
TPH2	hgnc:20692	TPH2	ChEMBL	33	inhibitor	2.187819634820604	TELOTRISTAT ETIPRATE	rxcui:1872448	TELOTRISTAT ETIPRATE	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.4150804050252529	Repotrectinib	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	3.320643240202023	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	2.763561643983921	REC-2282	ncit:C116850	HDAC INHIBITOR REC-2282	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.075496292	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.3680444245492605	Derazantinib	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.036633259	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1088116604009326	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.1017590527823536	ISOXSUPRINE HYDROCHLORIDE	rxcui:82033	ISOXSUPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.084012274	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	1.029066006546944	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.05751114	Copanlisib	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.5125748858722557	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.2500365296937833	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.058602312	Romidepsin	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	2.625383561784724	BI 907828	ncit:C156709	BRIGIMADLIN	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.062509132	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	2.917092846427472	YTTRIUM Y 90 EPRATUZUMAB	chembl:CHEMBL2108817	YTTRIUM Y 90 EPRATUZUMAB	FALSE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	1.875273972703374	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	1.325951293830669	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	Tubastatin A	iuphar.ligand:9702	TUBASTATIN A	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	CC-90003	ncit:C119747	ERK INHIBITOR CC-90003	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	MRTX-1133	ncit:C200319	KRAS G12D INHIBITOR MRTX1133	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1337207247088994	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.6351734423672721	GI-4000	drugbank:DB05698	GI-4000	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.097236428	BAY1125976	iuphar.ligand:10908	BAY1125976	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.008529511	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	1.071585127259071	MEDI-5117	chembl:CHEMBL2109614	MEDI-5117	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	CCT128930	chembl:CHEMBL263664	CHEMBL:CHEMBL263664	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.364636606	Torin 1	iuphar.ligand:8004	TORIN 1	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.037398626	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.097236428	NVP-AEW541	iuphar.ligand:8067	NVP-AEW541	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.054581779	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1182605208011137	Rigosertib Sodium	ncit:C71355	RIGOSERTIB SODIUM	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.053217234	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	1.419126249613364	FOSNETUPITANT CHLORIDE HYDROCHLORIDE	rxcui:2044416	FOSNETUPITANT CHLORIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CancerCommons	25-Jul-13	inhibitor	0.030386384	SAR260301	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CancerCommons	25-Jul-13	inhibitor	0.5125748858722557	MEKINIST	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.077789143	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CYP19A1	hgnc:2594	CYP19A1	ChEMBL	33	inhibitor	1.250182648468916	TESTOLACTONE	rxcui:10378	TESTOLACTONE	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.1643432589536604	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1041818873724097	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	1.346350544504987	PRUCALOPRIDE SUCCINATE	rxcui:2107309	PRUCALOPRIDE SUCCINATE	TRUE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.031822831	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	TCMDC-124495	chembl:CHEMBL532452	CHEMBL:CHEMBL532452	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.013025967	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.1715936968486748	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	0.7778914257139926	P276-00	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	0.3889457128569963	Adenosine	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:7483	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9378	iuphar.ligand:9378	VPS34-IN-1	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
NCBIGENE:1420	hgnc:2410	CRYGC	GuideToPharmacology	2024.1	inhibitor	7.501095890813499	IUPHAR.LIGAND:8787	iuphar.ligand:8787	COMPOUND 12E [PMID: 18605714]	FALSE	FALSE	FALSE
NCBIGENE:504	hgnc:828	ATP5F1AP2	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	BETULIN	rxcui:2467840	BETULIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.082950507	CHARTREUSIN	chembl:CHEMBL1554674	CHARTREUSIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	LANSOPRAZOLE SULFIDE	chembl:CHEMBL899	LANSOPRAZOLE SULFIDE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.5000730593875666	LY377604	chembl:CHEMBL2012520	LY377604	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.138178082	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:1323	iuphar.ligand:1323	MT-II	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9910	drugbank:DB12933	RO-4987655	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.088333021	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
UNIPROT:P41587	hgnc:12695	VIPR2	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	VASOACTIVE INTESTINAL PEPTIDE	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2064	iuphar.ligand:2064	[111IN]DOTA-NOC-ATE	FALSE	FALSE	FALSE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	activator	6.563458904461812	IUPHAR.LIGAND:11849	iuphar.ligand:11849	TPC2-A1-P	FALSE	FALSE	FALSE
HTR1F	hgnc:5292	HTR1F	ChEMBL	33	agonist	4.773424657790408	LASMIDITAN SUCCINATE	ncit:C170094	LASMIDITAN SUCCINATE	TRUE	FALSE	FALSE
TRM1	hgnc:12318	TRX-CAT1-2	ChEMBL	33	inhibitor	26.25383561784724	LETERMOVIR	rxcui:1988648	LETERMOVIR	TRUE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	ChEMBL	33	inhibitor	2.059124362184097	AZD-4017	drugbank:DB14875	AZD-4017	FALSE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.7721716358190367	VERICIGUAT	rxcui:2475830	VERICIGUAT	TRUE	FALSE	FALSE
SELP	hgnc:10721	SELP	ChEMBL	33	blocker	13.12691780892362	CRIZANLIZUMAB	rxcui:2262279	CRIZANLIZUMAB	TRUE	FALSE	FALSE
F13A1	hgnc:3531	F13A1	ChEMBL	33	positive modulator	17.50255707856483	CATRIDECACOG	rxcui:1091605	FACTOR XIII, HUMAN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TEND	1-Aug-11	NULL	1.400204566285186	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TEND	1-Aug-11	NULL	0.2639729920045843	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.2027323213733378	IPRONIAZID	rxcui:5981	IPRONIAZID	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	0.1099637093941246	CEP-32496	iuphar.ligand:7880	AGERAFENIB	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:7943	iuphar.ligand:7943	MK-8776	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.019636377	Romidepsin	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.049349315	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
ELAVL1	hgnc:3312	ELAVL1	DTC	9/2/20	NULL	21.00306849427779	DEHYDROMUTACTIN	chembl:CHEMBL1242196	DEHYDROMUTACTIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009875432	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
NCBIGENE:2011	hgnc:3332	MARK2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8127	iuphar.ligand:8127	COMPOUND 3B [PMID: 23454515]	FALSE	FALSE	FALSE
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TdgClinicalTrial	Jan-14	NULL	0.1235474617310458	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.014881721	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:986	hgnc:18068	SLC15A3	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:4623	iuphar.ligand:4623	[14C]HISTIDINE	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:12966	iuphar.ligand:12966	CADONILIMAB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.025757994	AZD6482	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	ChEMBL	33	inhibitor	0.31115657	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004207345	DULOXETINE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00449706	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	DIHYDROCAPSAICIN	rxcui:2166037	DIHYDROCAPSAICIN	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.063415062	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2243917574174978	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.036847489	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.2243917574174978	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TEND	1-Aug-11	NULL	0.3409589041278864	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
PI3-KINASE BETA	hgnc:8976	PIK3CB	TTD	2020.06.01	NULL	0.2083637747448194	INK-1117	chembl:CHEMBL3545055	INK-1117	FALSE	FALSE	TRUE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11861	iuphar.ligand:11861	PRU-10	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	agonist	0.051885051	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003844181	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	1.500219178	TETRAETHYLAMMONIUM CHLORIDE	chembl:CHEMBL434435	TETRAETHYLAMMONIUM CHLORIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	SPERMINE	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.037884323	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	5-AMINOISOQUINOLINE	drugbank:DB04605	5-AMINOISOQUINOLINE	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:11732	iuphar.ligand:11732	BAY-8400	FALSE	FALSE	FALSE
UNIPROT:Q9UD71	hgnc:9287	PPP1R1B	TdgClinicalTrial	Jan-14	NULL	3.750547945406749	ITI-007	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
NCBIGENE:3103	hgnc:10721	SELP	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9049	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.03849536	Copanlisib	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.4861821410712453	LAM-002A	ncit:C126661	APILIMOD DIMESYLATE CAPSULE	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.1785975212098452	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2083637747448194	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	1.129197231	HEXAMETHYLENEBISACETAMIDE	chembl:CHEMBL291481	HEXAMETHYLENEBISACETAMIDE	FALSE	FALSE	FALSE
RPL34	hgnc:10340	RPL34	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00195341	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	PharmGKB	4/5/24	NULL	0.1110098757625676	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:1841	hgnc:3061	DTYMK	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3977853881492008	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
UBA1	hgnc:12469	UBA1	DTC	9/2/20	NULL	52.50767123569449	HYRTIOERECTINE B	chembl:CHEMBL526126	HYRTIOERECTINE B	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	0.2019525816757481	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.1207072901969988	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.003574869	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	AGN-211745	chembl:CHEMBL4650436	AGN-211745	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.059532507	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:10750	iuphar.ligand:10750	MLN-3897	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1737	ncit:C78118	DENUFOSOL	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.1356787370431382	ramipril	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
MC1R	hgnc:6929	MC1R	ChEMBL	33	agonist	7.501095891	DERSIMELAGON	ncit:C166490	DERSIMELAGON	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.07631929	CID 667285	chembl:CHEMBL267160	CHEMBL:CHEMBL267160	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	NORDEFRIN	ncit:C81340	NORDEFRIN	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:3897	iuphar.ligand:3897	M32	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1430	iuphar.ligand:1430	PTEB	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	NETILMICIN SULFATE	rxcui:203193	NETILMICIN SULFATE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.2778183663264258	UMBRALISIB TOSYLATE	rxcui:2478438	UMBRALISIB TOSYLATE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.3043922970185188	ANTICONVULSANT	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.012558639	clotrimazole	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.023780648	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	3.088686543276147	BMS-816336	chembl:CHEMBL4086816	BMS-816336	FALSE	FALSE	FALSE
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.4773424657790409	AMG 820	ncit:C98295	ANTI-C-FMS MONOCLONAL ANTIBODY AMG 820	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.1084869240406911	IUPHAR.LIGAND:522	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	activator	0.1682938180631233	IUPHAR.LIGAND:3310	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	3.088686543276147	IUPHAR.LIGAND:12598	iuphar.ligand:12598	GLYCYL-[13C3]-SARCOSINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	SB-408124	iuphar.ligand:1704	SB-408124	FALSE	FALSE	FALSE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.046343929	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.4189441853911795	Trihexyphenidyl	rxcui:10811	TRIHEXYPHENIDYL	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.025814981	tetracycline	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	13.12691780892362	FP-1201	ncit:C201077	LYOPHILIZED HUMAN RECOMBINANT INTERFERON-BETA 1A FP-1201	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	MMV665817	chembl:CHEMBL590919	CHEMBL:CHEMBL590919	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.2273059360852575	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.092226589	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
RPS2	hgnc:10404	RPS2	ChEMBL	33	modulator	0.1067229090156392	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	NSC-309895	chembl:CHEMBL552439	CHEMBL:CHEMBL552439	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1458546423213736	ANANDRON	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
SRR	hgnc:14398	SRR	PharmGKB	4/5/24	NULL	2.692701089009974	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.019799273	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	CLIOXANIDE	ncit:C65338	CLIOXANIDE	FALSE	FALSE	FALSE
DTNBP1	hgnc:17328	DTNBP1	PharmGKB	4/5/24	NULL	0.5122699632750682	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002623285	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	MyCancerGenome	20-Jun-17	inhibitor	0.2983390411119005	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	0.2763561643983921	DEXTROAMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:1251	hgnc:7872	NOS1	GuideToPharmacology	2024.1	inhibitor	0.7395446652914718	IUPHAR.LIGAND:9147	iuphar.ligand:9147	COMPOUND 14J [PMID: 27050842]	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	inhibitor	0.040515178	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
RPS14	hgnc:10387	RPS14	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:10651	rxcui:2559612	SAMIDORPHAN	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.076208521	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	TCMDC-125602	chembl:CHEMBL580183	CHEMBL:CHEMBL580183	FALSE	FALSE	FALSE
IFIT1	hgnc:5407	IFIT1	PharmGKB	4/5/24	NULL	1.640864726115453	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.6250913242344582	AZD-8330	drugbank:DB06061	AZD-8330	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.2465148884304905	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	modulator	0.046965717	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
NCBIGENE:84	ncbigene:84	ACTL4	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10207	iuphar.ligand:10207	GPR4 ANTAGONIST 3B	FALSE	FALSE	FALSE
NCBIGENE:74	hgnc:147	ACTG1P2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:3664	iuphar.ligand:3664	[125I]CX3CL1 (HUMAN)	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.038049037	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.3580068493342807	APREMILAST	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	2,3,4,6-TETRACHLORO-PHENOL	chembl:CHEMBL320361	CHEMBL:CHEMBL320361	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	inhibitor	0.1547594520630995	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
UNIPROT:P35498	hgnc:10585	SCN1A	TdgClinicalTrial	Jan-14	NULL	0.098451884	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
PTCH1	hgnc:9585	PTCH1	CIViC	10-Apr-24	NULL	4.375639269641208	SONIDEGIB	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.003244419	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
HMOX1	hgnc:5013	HMOX1	NCI	14-Sep-17	NULL	0.082754407	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
FRAGILE HISTIDINE TRIAD PROTEIN	hgnc:3701	FHIT	TTD	2020.06.01	NULL	4.375639269641208	Fructose	rxcui:4570	FRUCTOSE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.4000584475100533	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.017218453	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MYD88	hgnc:7562	MYD88	PharmGKB	4/5/24	NULL	1.166837138570988	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	inhibitor	0.039068208	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.012736852	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
PROTEIN KINASE C EPSILON	hgnc:9401	PRKCE	TTD	2020.06.01	NULL	0.2917092846427472	Meprobamate	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.693795846312725	Olopatadine	rxcui:135391	OLOPATADINE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	DTC	9/2/20	NULL	0.4167275494896388	RO-4882224	chembl:CHEMBL1077391	CHEMBL:CHEMBL1077391	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.8751278539282418	SJ000014858	chembl:CHEMBL591628	CHEMBL:CHEMBL591628	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.078682824	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	2.625383561784724	SOM3355	chembl:CHEMBL2106060	BEVANTOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4907258993990139	Amfepramone	rxcui:3389	DIETHYLPROPION	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:246	iuphar.ligand:246	DAU 6285	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.3547815624033412	CEVIMELINE HYDROCHLORIDE	rxcui:260036	CEVIMELINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2418	hgnc:3929	FRA8A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10733	iuphar.ligand:10733	I-432	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.1400204566285186	DIMETHENAMID	chembl:CHEMBL1565335	DIMETHENAMID	FALSE	FALSE	FALSE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:10546	iuphar.ligand:10546	DBRD9-A	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:11313	iuphar.ligand:11313	CPX	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:10136	ncit:C148147	LAZERTINIB	FALSE	FALSE	FALSE
NCBIGENE:2289	hgnc:3721	FKBP5	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:10402	iuphar.ligand:10402	ZAK INHIBITOR 6P	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.059667808	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	(S)-ALAPROCLATE	chembl:CHEMBL251941	(S)-ALAPROCLATE	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Cyclizine	rxcui:2977	CYCLIZINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.1259176768242074	SUFORAPHANE ISOSELENOCYANATE	chembl:CHEMBL1089972	SUFORAPHANE ISOSELENOCYANATE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	NSC-402538	chembl:CHEMBL121556	CHEMBL:CHEMBL121556	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.00822231	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	CARNOSIC ACID	chembl:CHEMBL484853	CARNOSIC ACID	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.023482858	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
DES	hgnc:2770	DES	NCI	14-Sep-17	NULL	1.458546423213736	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
RRAS2	hgnc:17271	RRAS2	PharmGKB	4/5/24	NULL	1.615620653405984	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	1.346350544504987	LC-350189	chembl:CHEMBL3652780	TIGULIXOSTAT	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	0.3000438356325399	IUPHAR.LIGAND:1911	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
RPS19	hgnc:10402	RPS19	ChEMBL	33	modulator	0.049256727	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:1299	hgnc:2219	COL9A3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5225	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	2.187819634820604	AZ20	iuphar.ligand:8477	AZ20	FALSE	FALSE	TRUE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.057260274	Mifepristone	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.046673486	IUPHAR.LIGAND:968	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.061484393	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
ADM	hgnc:259	ADM	NCI	14-Sep-17	NULL	0.6563458904461813	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	EVOGLIPTIN	ncit:C171769	EVOGLIPTIN	FALSE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	ChEMBL	33	inhibitor	0.7501095890813501	COBICISTAT	rxcui:1306284	COBICISTAT	TRUE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.1930429089547592	Soblidotin	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	3.088686543276147	ONO-4578	ncit:C150376	EP4 ANTAGONIST ONO-4578	FALSE	FALSE	FALSE
AMP-ACTIVATED PROTEIN KINASE	hgnc:9377	PRKAA2	TTD	2020.06.01	NULL	1.363835616511545	Acadesine	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.7395446652914718	BFH-772	chembl:CHEMBL4080062	BFH-772	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.02646556	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P51170	hgnc:10602	SCNN1G	TEND	1-Aug-11	NULL	1.620607136904151	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.8950171233357017	Penbutolol	rxcui:7973	PENBUTOLOL	TRUE	FALSE	FALSE
UNIPROT:P51172	hgnc:10601	SCNN1D	TdgClinicalTrial	Jan-14	NULL	2.059124362184098	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.2430910705356226	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
VAV1	hgnc:12657	VAV1	NCI	14-Sep-17	NULL	2.333674277141977	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.03357268	ERYTHROMYCIN ETHYLSUCCINATE	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	0.31115657	Mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:332	iuphar.ligand:332	N-BENZYL BRUCINE	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.046303061	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.0055883	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
NCBIGENE:1169	hgnc:13447	SLC38A1	GuideToPharmacology	2024.1	NULL	10.50153425	IUPHAR.LIGAND:4543	rxcui:426	ALANINE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1346350544504987	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.000146118775133	JNJ-38877605	drugbank:DB13113	JNJ-38877605	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3968	iuphar.ligand:3968	PSAB-OFP	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.062808219	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.06714536	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	PENTAMIDINE DIISETHIONATE	chembl:CHEMBL361506	PENTAMIDINE ISETHIONATE	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.4189441853911795	TRIHEXYPHENIDYL	rxcui:10811	TRIHEXYPHENIDYL	TRUE	FALSE	FALSE
TISSUE FACTOR PATHWAY INHIBITOR	hgnc:11760	TFPI	TTD	2020.06.01	NULL	2.763561643983921	Tifacogin	ncit:C152614	TIFACOGIN	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	0.6908904109959803	SR-123781A	drugbank:DB05361	SR-123781A	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	L-165041	drugbank:DB08078	{4-[3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPOXY]PHENOXY}ACETIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	DNDI1417346	chembl:CHEMBL1490332	CHEMBL:CHEMBL1490332	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.083478015	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1628144844517658	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	0.2500365296937833	Cerdulatinib	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.070956312	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.043692674	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.003198567	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.077789143	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00224853	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.1458546423213736	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NU-1025	chembl:CHEMBL123904	CHEMBL:CHEMBL123904	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.08780547	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
PSMC1	hgnc:9547	PSMC1	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
LEP	hgnc:6553	LEP	PharmGKB	4/5/24	NULL	0.050294704	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	8-OH-DPAT	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	NCI	14-Sep-17	NULL	0.032858367	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2264	iuphar.ligand:2264	MAXADILAN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.1233298208706858	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1516	iuphar.ligand:1516	PYY-(13-36) (MOUSE, RAT, PIG)	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.081030357	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	HARMOL	chembl:CHEMBL486817	HARMOL	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	1.312691780892362	OSM-S-85	chembl:CHEMBL1494650	CHEMBL:CHEMBL1494650	FALSE	FALSE	FALSE
UNIPROT:P62942	hgnc:3711	FKBP1A	TEND	1-Aug-11	NULL	2.917092846427472	PIMECROLIMUS	rxcui:321952	PIMECROLIMUS	TRUE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	3.500511415712966	Viramidine	chembl:CHEMBL2107375	TARIBAVIRIN HYDROCHLORIDE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.5585922471882393	NGX-267	chembl:CHEMBL4297408	NGX-267	FALSE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE	hgnc:1189	AHSA1	TTD	2020.06.01	NULL	4.375639269641208	AZD7624	iuphar.ligand:11714	AZD7624	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	1.693795846312725	NW-3509	chembl:CHEMBL3678076	EVENAMIDE	FALSE	FALSE	FALSE
CFD	hgnc:2771	CFD	ChEMBL	33	inhibitor	17.50255707856483	LAMPALIZUMAB	ncit:C123730	LAMPALIZUMAB	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	binder	2.282942227638891	T84.66	chembl:CHEMBL2109370	T84.66	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2234368988752957	LERCANIDIPINE HYDROCHLORIDE	rxcui:153679	LERCANIDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FIPRONIL	rxcui:1433761	FIPRONIL	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	PROROXAN HYDROCHLORIDE	ncit:C84120	PROROXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	VANILLIN	rxcui:1368176	VANILLIN	TRUE	FALSE	FALSE
GLA	hgnc:4296	GLA	DTC	9/2/20	NULL	0.1442518440541057	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
IRF3	hgnc:6118	IRF3	NCI	14-Sep-17	NULL	2.692701089009974	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.2263261691193728	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.019490598	Androgen restored contraceptive	wikidata:Q85759692	ETHINYLESTRADIOL/DROSPIRENONE/PRASTERONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.015193192	nabumetone	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TEND	1-Aug-11	NULL	0.5625821918110125	RIVASTIGMINE	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
ANGIOPOIETIN-1	hgnc:484	ANGPT1	TTD	2020.06.01	NULL	2.625383561784724	AMG 780	ncit:C116627	ANTI-ANGIOPOIETIN MONOCLONAL ANTIBODY AMG 780	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1154649175056503	Bupropion	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.3088686543276147	(-)-Phenserine	drugbank:DB04892	PHENSERINE	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10661	iuphar.ligand:10661	JNJ-42226314	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	2.072671233	RABUSERTIB	ncit:C81937	RABUSERTIB	FALSE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.3205596534535683	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	3-HYDROXYFLAVONOL	chembl:CHEMBL242172	CHEMBL:CHEMBL242172	FALSE	FALSE	FALSE
TPP1	hgnc:2073	TPP1	FDA	10-Apr-24	NULL	157.5230137070835	Cerliponase Alfa	rxcui:1922436	CERLIPONASE ALFA	TRUE	FALSE	FALSE
ERCC6	hgnc:3438	ERCC6	NCI	14-Sep-17	NULL	0.4039051633514962	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	NCX 4016	ncit:C61499	NITRIC OXIDE-RELEASING ACETYLSALICYLIC ACID DERIVATIVE	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	2.100306849	Balixafortide	ncit:C91094	BALIXAFORTIDE	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	BROMFENAC	rxcui:19737	BROMFENAC	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.1415301111474245	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:12788	drugbank:DB14946	PCO-371	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	PharmGKB	4/5/24	NULL	0.06286838	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
TLR7	hgnc:15631	TLR7	ChEMBL	33	activator	2.625383561784724	VESATOLIMOD	ncit:C152870	VESATOLIMOD	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	2.763561643983921	trichloroethylene	rxcui:2534464	TRICHLOROETHYLENE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	0.078761507	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	0.525076712	ELTROMBOPAG	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.106290832	IUPHAR.LIGAND:7434	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	1.842374429322613	Setipiprant	ncit:C152348	SETIPIPRANT	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.033412454	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	modulator	0.4646696569530486	IUPHAR.LIGAND:9748	iuphar.ligand:9748	BMS-986187	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.1141471113819445	Alvocidib	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	SULFENTRAZONE	chembl:CHEMBL1884669	SULFENTRAZONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	DOMPERIDONE	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.267214612	HALOBETASOL PROPIONATE	rxcui:41208	HALOBETASOL	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.305277158	AMLODIPINE BENZOATE	rxcui:2184116	AMLODIPINE BENZOATE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2859	ncit:C72100	MIBOLERONE	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:10081	iuphar.ligand:10081	KINASE INHIBITOR 2 [PMID: 30199702]	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.077444943	IUPHAR.LIGAND:10651	rxcui:2559612	SAMIDORPHAN	TRUE	FALSE	FALSE
CARD16	hgnc:33701	CARD16	PharmGKB	4/5/24	NULL	1.640864726115453	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.020795117	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	inhibitor	0.038159645	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
CUX1	hgnc:2557	CUX1	PharmGKB	4/5/24	NULL	0.5048814541893702	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.1428780169678761	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1591141552596803	TCMDC-138263	chembl:CHEMBL535307	CHEMBL:CHEMBL535307	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CORTODOXONE	ncit:C80813	CORTODOXONE	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	inhibitor	0.042073455	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002493952	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.039068208	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.07182992	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	inhibitor	0.044347695	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.06714536	IUPHAR.LIGAND:5230	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.048663273	IUPHAR.LIGAND:7351	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:6412	iuphar.ligand:6412	VANILLIN	FALSE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	ChEMBL	33	agonist	13.12691780892362	MOTOLIMOD	ncit:C80521	MOTOLIMOD	FALSE	FALSE	TRUE
NCBIGENE:1430	hgnc:2421	CRYZP1	GuideToPharmacology	2024.1	inhibitor	7.501095890813499	IUPHAR.LIGAND:8787	iuphar.ligand:8787	COMPOUND 12E [PMID: 18605714]	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.07699072	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	EPIRUBICIN HYDROCHLORIDE	rxcui:203213	EPIRUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:882	iuphar.ligand:882	PD-135158	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.058277105	IUPHAR.LIGAND:5656	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
KCNH7	hgnc:18863	KCNH7	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	DIMIRACETAM	ncit:C79121	DIMIRACETAM	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.175415383	GLPG0492	chembl:CHEMBL3545417	GLPG0492	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:8383	iuphar.ligand:8383	BIMIRALISIB	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	inhibitor	0.03729238	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11561	iuphar.ligand:11561	COMPOUND IV [PMID: 29351497]	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	BI-3406	iuphar.ligand:12061	BI-3406	FALSE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	PharmGKB	4/5/24	NULL	1.121958787087489	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	1.500219178	CIRSIMARITIN	chembl:CHEMBL348436	CIRSIMARITIN	FALSE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	DTC	9/2/20	NULL	1.790034246671403	PYRIDINE-2,4-DICARBOXYLIC ACID	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-1030062A	chembl:CHEMBL482326	GSK-1030062A	FALSE	FALSE	FALSE
KCNJ3	hgnc:6264	KCNJ3	ChEMBL	33	blocker	2.187819634820604	VERNAKALANT HYDROCHLORIDE	ncit:C152865	VERNAKALANT HYDROCHLORIDE	FALSE	FALSE	FALSE
ENOSF1	hgnc:30365	ENOSF1	NCI	14-Sep-17	NULL	2.333674277141978	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00292359	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1000146118775133	DEMECLOCYCLINE HYDROCHLORIDE	rxcui:81993	DEMECLOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.024932417	VERNAKALANT HYDROCHLORIDE	ncit:C152865	VERNAKALANT HYDROCHLORIDE	FALSE	FALSE	FALSE
LTB	hgnc:6711	LTB	ChEMBL	33	inhibitor	13.12691780892362	BAMINERCEPT	ncit:C96762	BAMINERCEPT ALFA	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.068637479	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
NCBIGENE:2679	hgnc:4252	GGT3P	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8744	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:8383	iuphar.ligand:8383	BIMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.03140411	IUPHAR.LIGAND:305	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.072927321	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	2.838252499226729	GW-328267	chembl:CHEMBL186113	GW-328267	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.056157937	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003720782	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4907258993990139	Iobenguane I-123	rxcui:1426748	IOBENGUANE I-123	TRUE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.050488145	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
SMAD2	hgnc:6768	SMAD2	DTC	9/2/20	NULL	0.1988926940746004	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.1861974157294131	AZELNIDIPINE	ncit:C73023	AZELNIDIPINE	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	FDA	10-Apr-24	NULL	0.9883796938483671	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
EZH2	hgnc:3527	EZH2	CIViC	10-Apr-24	NULL	0.108040476	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
DDHD1	hgnc:19714	DDHD1	PharmGKB	4/5/24	NULL	3.182283105193606	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.04907259	ENCLOMIPHENE	ncit:C28211	ENCLOMIPHENE	FALSE	FALSE	FALSE
NCBIGENE:1971	hgnc:8751	CDK18	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8217	iuphar.ligand:8217	COMPOUND 77 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:11425	iuphar.ligand:11425	TYK2 INHIBITOR 14L	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	ChEMBL	33	positive modulator	1.810609352954982	BETIBEGLOGENE AUTOTEMCEL	rxcui:2610349	BETIBEGLOGENE AUTOTEMCEL	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.2263261691193728	TARLOXOTINIB	drugbank:DB14944	TARLOXOTINIB	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	MK-212	drugbank:DB12111	MK-212	FALSE	FALSE	FALSE
RPL38	hgnc:10349	RPL38	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.008500513	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.018206543	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	INDIGOTINDISULFONATE	rxcui:1426889	INDIGO	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.3431873936973496	Homatropine Methylbromide	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:626	iuphar.ligand:626	PD 176252	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	RO6839921	ncit:C114980	MDM2 ANTAGONIST RO6839921	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	1.944728564284981	PRALSETINIB	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.678633990910949	INCB018424	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.4906052389860809	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CancerCommons	25-Jul-13	inhibitor	0.1099637093941246	CHIR-265	iuphar.ligand:5674	CHIR-265	FALSE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	TETRACYCLINE HYDROCHLORIDE	rxcui:142446	TETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:666	iuphar.ligand:666	COMPOUND 12 [PMID: 12723943]	FALSE	FALSE	FALSE
NCBIGENE:2004	hgnc:3325	ELK3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9422	iuphar.ligand:9422	DAPK INHIBITOR 13	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.09869863	IUPHAR.LIGAND:5671	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6130	iuphar.ligand:6130	GALANIN(2-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:453	hgnc:771	ASS1P8	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:4185	iuphar.ligand:4185	DYSIHERBAINE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:363	hgnc:639	AQP6	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:2137	iuphar.ligand:2137	METRH	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	Miransertib	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.039258072	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
IDO1	hgnc:6059	IDO1	DTC	9/2/20	NULL	7.501095891	2-HYDRAZINYLBENZO[D]THIAZOLE	chembl:CHEMBL1933308	CHEMBL:CHEMBL1933308	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	PharmGKB	4/5/24	NULL	0.4526523382387456	luspatercept	rxcui:2262543	LUSPATERCEPT-AAMT	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
CANCER STEMNESS KINASE	hgnc:2444	CSK	TTD	2020.06.01	NULL	17.50255707856483	BBI503	ncit:C104745	AMCASERTIB	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	DNDI1417085	chembl:CHEMBL1522984	CHEMBL:CHEMBL1522984	FALSE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	agonist	3.281729452230906	BETAZOLE HYDROCHLORIDE	chembl:CHEMBL1200949	BETAZOLE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12942	iuphar.ligand:12942	COMPOUND 42 [PMID: 37721854]	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	blocker	0.7955707762984014	IUPHAR.LIGAND:2368	iuphar.ligand:2368	CYANOTRIPHENYLBORATE	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:3982	iuphar.ligand:3982	&ALPHA;-CONOTOXIN PNIA	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:4054	iuphar.ligand:4054	AC261066	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.1930429089547591	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	PYRACLOSTROBIN	chembl:CHEMBL519873	PYRACLOSTROBIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.015930725	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.042619863	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.068369364	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.089756703	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.060984519	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:12095	iuphar.ligand:12095	EXARAFENIB	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.006948216	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.034704343	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
EEF2	hgnc:3214	EEF2	DTC	9/2/20	NULL	5.834185692854944	LACTIMIDOMYCIN	chembl:CHEMBL1221911	LACTIMIDOMYCIN	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-2	hgnc:4087	GABRG2	TTD	2020.06.01	NULL	0.1562728310586145	THIOCOLCHICOSIDE	rxcui:38085	THIOCOLCHICOSIDE	FALSE	FALSE	FALSE
KCND3	hgnc:6239	KCND3	ChEMBL	33	blocker	0.1640864726115453	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2625	iuphar.ligand:2625	SAXITOXIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.016023092	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1544343271638073	BERBERRUBINE	chembl:CHEMBL203135	BERBERRUBINE	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.2822993077187876	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Acolbifene	ncit:C64183	ACOLBIFENE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.030386384	dipyrone	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.3697723326457359	ONATASERTIB	ncit:C92575	ONATASERTIB	FALSE	FALSE	TRUE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.081365193	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.9053046764774912	PRULIFLOXACIN	ncit:C72637	PRULIFLOXACIN	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	SOTORASIB	rxcui:2550714	SOTORASIB	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.3684748858645228	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
DHRS9	hgnc:16888	DHRS9	DTC	9/2/20	NULL	15.00219178	(+/-)-SPONGIAQUINONE	chembl:CHEMBL514876	CHEMBL:CHEMBL514876	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.045265234	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	DNDI1417905	chembl:CHEMBL1449731	CHEMBL:CHEMBL1449731	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1372749574789398	ANTICONVULSANT	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	CGI	2/1/22	NULL	0.5303805175322677	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.095468493	PAROXETINE MESYLATE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1562728310586145	4SC-203	drugbank:DB12669	4SC-203	FALSE	FALSE	FALSE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.046303061	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	LEVOCABASTINE	rxcui:28627	LEVOCABASTINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.2108741816694558	IUPHAR.LIGAND:75	iuphar.ligand:75	SB 272183	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1325951293830669	IUPHAR.LIGAND:294	rxcui:194	ACETYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9558	iuphar.ligand:9558	BELUMOSUDIL	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10219	iuphar.ligand:10219	MP-A08	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.8649519486500064	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
PSMB4	hgnc:9541	PSMB4	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.2518353536484148	GNF-2	iuphar.ligand:5935	BCR-ABL INHIBITOR GNF-2	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	SCH-58261	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.024041974	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	3.750547945	Ifetroban sodium	ncit:C81569	IFETROBAN SODIUM	FALSE	FALSE	FALSE
FOXP3	hgnc:6106	FOXP3	PharmGKB	4/5/24	NULL	0.4688184931758437	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	0.384671584	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
MDH2	hgnc:6971	MDH2	NCI	14-Sep-17	NULL	3.750547945406749	GONADOTROPINS	ncit:C527	THERAPEUTIC GONADOTROPIN	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.1704794520639431	DNDI1417346	chembl:CHEMBL1490332	CHEMBL:CHEMBL1490332	FALSE	FALSE	FALSE
PSMD13	hgnc:9558	PSMD13	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.085796848	NS-398	drugbank:DB14060	NS-398	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	NSC-67436	chembl:CHEMBL1331995	CHEMBL:CHEMBL1331995	FALSE	FALSE	FALSE
SULT1A4	hgnc:30004	SULT1A4	PharmGKB	4/5/24	NULL	1.514644363	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.1785975212098452	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	0.108040476	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.039214094	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
PSMB4	hgnc:9541	PSMB4	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC6	hgnc:9553	PSMC6	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
RPL28	hgnc:10330	RPL28	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:8999	iuphar.ligand:8999	(S)-ARN2508	FALSE	FALSE	FALSE
NCBIGENE:1370	hgnc:2313	CPN2	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8819	iuphar.ligand:8819	CTA091	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:10129	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3962	iuphar.ligand:3962	4BP-TQS	FALSE	FALSE	FALSE
ADRM1	hgnc:15759	ADRM1	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:4582	rxcui:1373458	CANAGLIFLOZIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FLUROCHLORIDONE	chembl:CHEMBL2272973	FLUROCHLORIDONE	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.1801292323694494	WEDELOLACTONE	iuphar.ligand:5551	WEDELOLACTONE	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	1.628144844517658	PEMIGATINIB	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	LECANORIC ACID	chembl:CHEMBL1451874	LECANORIC ACID	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.4070362111294147	Amobarbital	rxcui:719	AMOBARBITAL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.021554873	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.5672124979164529	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:8095	iuphar.ligand:8095	AC710	FALSE	FALSE	FALSE
PSMD7	hgnc:9565	PSMD7	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.041872146	IUPHAR.LIGAND:7313	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2278	iuphar.ligand:2278	[ALA11,22,28]VIP	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.01992701	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1000146118775133	RHGH	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	BISMUTH SUBSALICYLATE	rxcui:19478	BISMUTH SUBSALICYLATE	TRUE	FALSE	FALSE
PSMA7	hgnc:9536	PSMA7	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.003398555	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9885	iuphar.ligand:9885	CORTISTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.091796628	IUPHAR.LIGAND:7503	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.4730420832044549	IUPHAR.LIGAND:4792	rxcui:7500	NOMIFENSINE	FALSE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:4582	rxcui:1373458	CANAGLIFLOZIN	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-1030058A	chembl:CHEMBL473420	GSK-1030058A	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.035430277	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	0.252440727	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1363835616511545	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8218	iuphar.ligand:8218	COMPOUND 1 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	inhibitor	0.2011788169949981	IUPHAR.LIGAND:4197	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	0.3431873936973497	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
NCBIGENE:103	hgnc:225	ADAR	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:6067	iuphar.ligand:6067	PROSAPTIDE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:7483	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.07661359	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.003616231	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.7343730242754476	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	SARCOLYSIN	ncit:C61936	SARCOLYSIN	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.098513454	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.033232703	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
RPL22	hgnc:10315	RPL22	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.4167275494896388	LENIOLISIB	rxcui:2633005	LENIOLISIB	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.009430257	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.017092341	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.075442056	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	NSC-402538	chembl:CHEMBL121556	CHEMBL:CHEMBL121556	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	ChEMBL	33	inhibitor	0.1093909817410302	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1562728310586145	IBCASERTIB	ncit:C115970	IBCASERTIB	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1077080435603989	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
RPL22	hgnc:10315	RPL22	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
PSMD11	hgnc:9556	PSMD11	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PTGER4	hgnc:9596	PTGER4	ChEMBL	33	inhibitor	3.088686543276147	CR-6086	chembl:CHEMBL3920982	CR-6086	FALSE	FALSE	FALSE
NCBIGENE:1297	hgnc:2217	COL9A1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5225	rxcui:52769	MILRINONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.019799273	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.2375912725597036	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	1.381780822	ICHORCUMAB	chembl:CHEMBL4298002	ICHORCUMAB	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1468061637531067	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	inhibitor	1.193356164447602	CONIVAPTAN HYDROCHLORIDE	rxcui:1294548	CONIVAPTAN HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.058602312	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.06286838	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10527	iuphar.ligand:10527	LASW1393	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.076765601	IUPHAR.LIGAND:7793	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
NCBIGENE:1502	hgnc:6875	MAPK13	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:12122	iuphar.ligand:12122	COMPOUND 4E [PMID: 35546685]	FALSE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	ChEMBL	33	inhibitor	0.7955707762984013	RG-4733	drugbank:DB11870	RG-4733	FALSE	FALSE	FALSE
TBXT	hgnc:11515	TBXT	PharmGKB	4/5/24	NULL	4.773424657790409	flunisolide	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.5048814541893701	TCMDC-123789	chembl:CHEMBL588859	CHEMBL:CHEMBL588859	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:2645	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
MC1R	hgnc:6929	MC1R	ChEMBL	33	agonist	4.500657534488099	AFAMELANOTIDE	rxcui:2262250	AFAMELANOTIDE	TRUE	FALSE	FALSE
RPL10A	hgnc:10299	RPL10A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.02385628	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.032016873	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q99460	hgnc:9554	PSMD1	TdgClinicalTrial	Jan-14	NULL	0.5385402178019948	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
RPL19	hgnc:10312	RPL19	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:865	iuphar.ligand:865	GW-5823	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:7399	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8172	iuphar.ligand:8172	COMPOUND 7 [PMID: 22464456]	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	MRX-2843	chembl:CHEMBL4650408	MRX-2843	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.080781033	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	CIViC	10-Apr-24	NULL	0.3241214273808303	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
RPL13A	hgnc:10304	RPL13A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	5.250767123569449	Lobeline	rxcui:6464	LOBELINE	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.2125816649218401	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	FASUDIL HYDROCHLORIDE	chembl:CHEMBL541388	FASUDIL HYDROCHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	N-METHYLANTHRANILIC ACID	chembl:CHEMBL1528955	N-METHYLANTHRANILIC ACID	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	1.628144844517658	INDIPLON	ncit:C74385	INDIPLON	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.175610941	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	2.100306849	POL-6326	ncit:C91094	BALIXAFORTIDE	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	3.424413341458336	GTS-21	drugbank:DB05708	GTS-21	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:8208	iuphar.ligand:8208	COMPOUND 5N [PMID: 20483621]	FALSE	FALSE	FALSE
RPL7	hgnc:10363	RPL7	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:12873	iuphar.ligand:12873	PIMICOTINIB	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.046343929	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:4561	iuphar.ligand:4561	[3H]PAROXETINE	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	ChEMBL	33	inhibitor	2.100306849	DIMETHYL FUMARATE	rxcui:1373478	DIMETHYL FUMARATE	TRUE	FALSE	FALSE
KCNB1	hgnc:6231	KCNB1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
RPL9P8	hgnc:30334	RPL9P8	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:2928	iuphar.ligand:2928	CYM5442	FALSE	FALSE	FALSE
CD44	hgnc:1681	CD44	ChEMBL	33	binder	0.172722603	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
RPL6	hgnc:10362	RPL6	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:5991	iuphar.ligand:5991	ISOGRANULATIMIDE	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	modulator	0.2500365296937833	CARIPRAZINE HYDROCHLORIDE	rxcui:1721073	CARIPRAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH5	hgnc:6254	KCNH5	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.8325740682192574	FUTIBATINIB	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9001	iuphar.ligand:9001	BIA 10-2474	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1026	iuphar.ligand:1026	SPINORPHIN	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.049723174	IUPHAR.LIGAND:325	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.7369497717290455	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.007479725	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
RPL9	hgnc:10369	RPL9	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
PDYN	hgnc:8820	PDYN	NCI	14-Sep-17	NULL	2.250328767	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
CST4	hgnc:2476	CST4	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
RPL9P9	hgnc:30334	RPL9P8	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.6250913242344582	Estrogen	chembl:CHEMBL592868	ESTROGEN	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.064505739	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
PLA2G4A	hgnc:9035	PLA2G4A	ChEMBL	33	inhibitor	4.375639269641208	GIRIPLADIB	ncit:C166518	GIRIPLADIB	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2273059360852575	DIFFERENTIATION INDUCER	ncit:C1934	DIFFERENTIATION INDUCER	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.084689792	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
RPL26	hgnc:10327	RPL26	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.028977744	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1278595890479573	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.034184682	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1525	hgnc:2559	CXADR	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10437	iuphar.ligand:10437	COMPOUND E22 [PMID: 31298542]	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.095468493	PAROXETINE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	LAVENDUSTIN B	ncit:C1616	LAVENDUSTIN B	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV000839	chembl:CHEMBL600374	CHEMBL:CHEMBL600374	FALSE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	inhibitor	2.187819634820604	BLESELUMAB	ncit:C171700	BLESELUMAB	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.005218413	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004557958	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
CPB2	hgnc:2300	CPB2	NCI	14-Sep-17	NULL	2.143170254518142	C5A	iuphar.ligand:3576	C5A	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.037003292	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:3313	rxcui:8156	PHENYLALANINE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW809897X	chembl:CHEMBL189353	GW809897X	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.022632617	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	PharmGKB	4/5/24	NULL	0.088770366	cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	DINOSEB	chembl:CHEMBL1892987	DINOSEB	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	binder	3.500511415712966	TESIDOLUMAB	ncit:C129315	TESIDOLUMAB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009922085	BROXURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-1232	chembl:CHEMBL601822	CHEMBL:CHEMBL601822	FALSE	FALSE	FALSE
PON1	hgnc:9204	PON1	PharmGKB	4/5/24	NULL	2.100306849	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NCBIGENE:470	ncbigene:470	ATHS	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:3980	iuphar.ligand:3980	[3H]METHYLLYCACONITINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.005357926	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.055271233	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	CLOROTEPINE	ncit:C77572	CLOROTEPINE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
TSC2	hgnc:12363	TSC2	OncoKB	23-Jul-20	NULL	2.250328767	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	GNF-PF-2976	chembl:CHEMBL579956	CHEMBL:CHEMBL579956	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:3283	iuphar.ligand:3283	SCH442416	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:9600	iuphar.ligand:9600	MIVAVOTINIB	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.07182992	IUPHAR.LIGAND:7936	iuphar.ligand:7936	PF-04691502	FALSE	FALSE	TRUE
POLD2	hgnc:9176	POLD2	ChEMBL	33	inhibitor	0.7955707762984016	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	1.193356164447602	Pelubiprofen	ncit:C66333	PELUBIPROFEN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.009270422	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.056826484	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4907258993990139	BLI-1005	ncit:C171390	RADIX POLYGALAE EXTRACT PDC-1421	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	0.6863747873946993	ISTIRATUMAB	ncit:C103863	ISTIRATUMAB	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.066803653	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.012841201	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.2083637747448194	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.045304289	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	1.944728564284981	ETRUMADENANT	ncit:C159564	ETRUMADENANT	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.061055432	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1988926940746003	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.029416062	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.3621218705909965	AMFONELIC ACID	ncit:C90833	AMFONELIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.004782119	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.010417155	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
POLE	hgnc:9177	POLE	ChEMBL	33	inhibitor	0.4773424657790409	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
GLUCOSE-6-PHOSPHATE DEHYDROGENASE	hgnc:4057	G6PD	TTD	2020.06.01	NULL	0.2625383561784725	EPIANDROSTERONE	ncit:C61747	EPIANDROSTERONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00133485	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.3677319929494733	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	CYCLOBENZAPRINE HYDROCHLORIDE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	2.059124362184098	LENTINAN	ncit:C28168	LENTINAN	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	ChEMBL	33	inhibitor	0.2263261691193728	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	TALC	12-May-16	inhibitor	0.7395446652914718	RIDAFOROLIMUS	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	0.6000876712650799	R-roscovitine	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
FATTY ACID SYNTHASE	hgnc:3594	FASN	TTD	2020.06.01	NULL	1.944728564284981	Cerulenin	drugbank:DB01034	CERULENIN	FALSE	FALSE	FALSE
SLC10A1	hgnc:10905	SLC10A1	PharmGKB	4/5/24	NULL	0.729273212	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
MAD1L1	hgnc:6762	MAD1L1	PharmGKB	4/5/24	NULL	0.4861821410712453	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	2.763561643983921	QAV-680	drugbank:DB11658	QAV-680	FALSE	FALSE	FALSE
NCBIGENE:2278	ncbigene:2278	FIM1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8183	iuphar.ligand:8183	PD166285	FALSE	FALSE	FALSE
MMP12	hgnc:7158	MMP12	ChEMBL	33	inhibitor	2.917092846427472	AZD-1236	drugbank:DB11961	AZD-1236	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	positive modulator	1.071585127259071	COAGULATION FACTOR X HUMAN	ncit:C82272	COAGULATION FACTOR X HUMAN	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.05293112	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1136529680426287	DNDI1417099	chembl:CHEMBL1565444	CHEMBL:CHEMBL1565444	FALSE	FALSE	FALSE
MYB	hgnc:7545	MYB	NCI	14-Sep-17	NULL	0.1470803115845784	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
SGK1	hgnc:10810	SGK1	NCI	14-Sep-17	NULL	1.250182648468916	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.067231333	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.020025809	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	NALBUPHINE HYDROCHLORIDE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.1223955040459079	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
UNIPROT:O95180	hgnc:1395	CACNA1H	TdgClinicalTrial	Jan-14	NULL	0.048844345	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.014369915	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2051	ncit:C152317	SEGLITIDE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014160645	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.034544521	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
CBL	hgnc:1541	CBL	CIViC	10-Apr-24	NULL	0.6563458904461812	SU11274	iuphar.ligand:5057	SU11274	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SJ000029700	chembl:CHEMBL591864	CHEMBL:CHEMBL591864	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.011993529	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	PharmGKB	4/5/24	NULL	1.831662950082366	larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.2027323213733378	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
GPNMB	hgnc:4462	GPNMB	ChEMBL	33	binder	1.640864726115453	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
CFB	hgnc:1037	CFB	ChEMBL	33	inhibitor	26.25383561784724	IPTACOPAN	rxcui:2671061	IPTACOPAN	TRUE	FALSE	FALSE
NCBIGENE:1324	hgnc:2615	CYP2B6	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:2586	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	NULL	0.6908904109959803	IUPHAR.LIGAND:3798	iuphar.ligand:3798	[125I]OREXIN A (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.039287446	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	DTC	9/2/20	NULL	0.6403374540938354	PROTUBOXEPIN A	chembl:CHEMBL1802135	PROTUBOXEPIN A	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.036013492	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inverse agonist	0.006579909	HALOPERIDOL DECANOATE	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.067317527	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6381	ncit:C77996	XIMELAGATRAN	TRUE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:7643	iuphar.ligand:7643	AEE788	FALSE	FALSE	TRUE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:7542	ncit:C80679	LASOFOXIFENE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	NSC-677438	chembl:CHEMBL118678	CHEMBL:CHEMBL118678	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.008345148	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	NSC-117271	chembl:CHEMBL287689	CHEMBL:CHEMBL287689	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	OncoKB	23-Jul-20	NULL	1.678633990910949	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-270822A	chembl:CHEMBL441702	GSK-270822A	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	PHANQUONE	ncit:C90620	PHANQUONE	FALSE	FALSE	FALSE
FGB	hgnc:3662	FGB	PharmGKB	4/5/24	NULL	1.166837138570988	abciximab	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	A-77636 HCL	chembl:CHEMBL1256876	CHEMBL:CHEMBL1256876	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.019739726	HYDRALAZINE HYDROCHLORIDE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
BAD	hgnc:936	BAD	DTC	9/2/20	NULL	0.4102161815288632	RUBOXISTAURIN	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.043768551	VP-16	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.049442252	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:9509	iuphar.ligand:9509	SB-3CT	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	XANTHOANGELOL	chembl:CHEMBL494083	XANTHOANGELOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	DNDI1417519	chembl:CHEMBL1402376	CHEMBL:CHEMBL1402376	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.033086119	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
SMARCA4	hgnc:11100	SMARCA4	CIViC	10-Apr-24	NULL	0.9376369863516874	TAZEMETOSTAT	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
ALOX12	hgnc:429	ALOX12	ChEMBL	33	inhibitor	1.693795846312725	BENOXAPROFEN	ncit:C76796	BENOXAPROFEN	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	NCI	14-Sep-17	NULL	0.1314334699266445	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	PharmGKB	4/5/24	NULL	0.2917092846427472	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.016807833	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.021501913	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	0.760980743	FR139317	iuphar.ligand:998	FR139317	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.2302968036653267	NERATINIB MALEATE	rxcui:1940642	NERATINIB MALEATE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	0.05913026	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P17342	hgnc:7945	NPR3	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	CARDIODILATIN	drugbank:DB15591	ATRIAL NATRIURETIC PEPTIDE	FALSE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	2.333674277141978	BETA-ADRENERGIC BLOCKING AGENT	ncit:C29576	BETA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.4861821410712453	PHENMETRAZINE HYDROCHLORIDE	rxcui:203198	PHENMETRAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	CancerCommons	25-Jul-13	inhibitor	0.010564924	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PTGER2	hgnc:9594	PTGER2	ChEMBL	33	agonist	3.281729452230906	SIMENEPAG ISOPROPYL	ncit:C152363	SIMENEPAG ISOPROPYL	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	CancerCommons	25-Jul-13	inhibitor	0.1582152052299645	MLN8237	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CancerCommons	25-Jul-13	inhibitor	0.1852122442176172	PLX3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	CGI	2/1/22	NULL	2.407466349146467	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	0.837888371	DOXIFLURIDINE	ncit:C978	DOXIFLURIDINE	FALSE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	CGI	2/1/22	NULL	0.5770073762164232	Enzalutamide	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.06714536	Vinblastine	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CGI	2/1/22	NULL	0.070574827	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	ChEMBL	33	inhibitor	0.1415301111474245	TEMUTERKIB	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	METHDILAZINE HYDROCHLORIDE	rxcui:91121	METHDILAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	1.693795846312725	OLOPATADINE HYDROCHLORIDE	rxcui:135391	OLOPATADINE	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.3725599732909588	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.8899605294185507	LOSARTAN POTASSIUM	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	0.7955707762984014	DEGARELIX ACETATE	rxcui:835863	DEGARELIX ACETATE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.7721716358190367	FROVATRIPTAN SUCCINATE	rxcui:322249	FROVATRIPTAN SUCCINATE	TRUE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	ChEMBL	33	inhibitor	7.001022831425932	PHENINDIONE	rxcui:8130	PHENINDIONE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.1223955040459079	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	1.458546423213736	FONDAPARINUX SODIUM	rxcui:321208	FONDAPARINUX	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.375054795	INSULIN SUSP ISOPHANE RECOMBINANT HUMAN	chembl:CHEMBL1201540	INSULIN SUSP ISOPHANE RECOMBINANT HUMAN	TRUE	FALSE	FALSE
MERTK	hgnc:7027	MERTK	ChEMBL	33	inhibitor	2.100306849	NINGETINIB	drugbank:DB16256	NINGETINIB	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	ChEMBL	33	inhibitor	0.9616789603607051	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.01152495	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.1158257453728555	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.063110182	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
GGCX	hgnc:4247	GGCX	ChEMBL	33	inhibitor	5.250767123569449	ANISINDIONE	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	4.039051633514961	PEGFILGRASTIM	rxcui:2048018	PEGFILGRASTIM-JMDB	TRUE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	agonist	1.670698630226643	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	1.381780822	DROSPIRENONE	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1204304386139782	BUPRENORPHINE HYDROCHLORIDE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.1603287671318916	CLOCORTOLONE PIVALATE	rxcui:21249	CLOCORTOLONE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.267214612	HALOBETASOL PROPIONATE	rxcui:41208	HALOBETASOL	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	CORTISONE ACETATE	rxcui:21655	CORTISONE ACETATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.047734247	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	ChEMBL	33	inhibitor	0.9907107780319716	ASN007	chembl:CHEMBL4650280	ASN007	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	0.9131768910555564	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1154649175056503	BUPROPION HYDROBROMIDE	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	ChEMBL	33	inhibitor	1.750255707856483	PAMIDRONATE DISODIUM	rxcui:105443	PAMIDRONATE DISODIUM	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	negative modulator	0.2243917574174978	MEMANTINE HYDROCHLORIDE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.3125456621172291	TIZANIDINE HYDROCHLORIDE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.182318303	METHOXAMINE HYDROCHLORIDE	rxcui:203187	METHOXAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.3170753093942904	DOXAZOSIN MESYLATE	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.095122593	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.4773424657790409	NEPAFENAC	rxcui:298665	NEPAFENAC	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1684738114514262	NAPROXEN SODIUM	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1684738114514262	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
SSTR4	hgnc:11333	SSTR4	ChEMBL	33	agonist	0.4861821410712454	OCTREOTIDE ACETATE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.7095631248066824	PARGYLINE HYDROCHLORIDE	rxcui:82069	PARGYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	ChEMBL	33	negative modulator	0.7955707762984014	MECAMYLAMINE HYDROCHLORIDE	rxcui:91240	MECAMYLAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2191733444543002	ALBUTEROL	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.1187188949127459	PROPRANOLOL HYDROCHLORIDE	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
GSC1	hgnc:4612	GSC	ChEMBL	33	inhibitor	5.250767123569449	CASPOFUNGIN ACETATE	rxcui:140108	CASPOFUNGIN	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	ChEMBL	33	inhibitor	0.1981421556063943	KO-947	iuphar.ligand:9976	KO-947	FALSE	FALSE	FALSE
CYP3A7	hgnc:2640	CYP3A7	ChEMBL	33	inhibitor	0.7501095890813501	COBICISTAT	rxcui:1306284	COBICISTAT	TRUE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	ChEMBL	33	inhibitor	0.9546849315580819	LOMITAPIDE MESYLATE	rxcui:1364478	LOMITAPIDE MESYLATE	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	ChEMBL	33	inhibitor	2.634164108814105	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PSMB2	hgnc:9539	PSMB2	ChEMBL	33	inhibitor	0.546954909	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA6	hgnc:9535	PSMA6	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB9	hgnc:9546	PSMB9	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
PSMA5	hgnc:9534	PSMA5	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA3	hgnc:9532	PSMA3	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA7	hgnc:9536	PSMA7	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC1	hgnc:9547	PSMC1	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD8	hgnc:9566	PSMD8	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
SEM1	hgnc:10845	SEM1	ChEMBL	33	inhibitor	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	0.326134604	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.7501095890813501	RAPACURONIUM BROMIDE	rxcui:228530	RAPACURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.3409589041278864	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.3571950424196904	DOXACURIUM CHLORIDE	rxcui:49275	DOXACURIUM CHLORIDE	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.6250913242344582	METOCURINE IODIDE	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.7501095890813501	RAPACURONIUM BROMIDE	rxcui:228530	RAPACURONIUM BROMIDE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.040893825	METHAMPHETAMINE HYDROCHLORIDE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	ChEMBL	33	agonist	0.1000146118775133	ETRETINATE	rxcui:4182	ETRETINATE	TRUE	FALSE	FALSE
RXRG	hgnc:10479	RXRG	ChEMBL	33	agonist	0.6819178082557726	ETRETINATE	rxcui:4182	ETRETINATE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.087318744	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.090634645	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.023652104	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.022730594	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.022439176	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.019233579	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.021344582	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.033658764	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
CA14	hgnc:1372	CA14	ChEMBL	33	inhibitor	0.546954909	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.070010228	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.077789143	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.081830137	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.069240885	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.017363648	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.016959842	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.018699313	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.087512785	CHLORAMPHENICOL	rxcui:2348	CHLORAMPHENICOL	TRUE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	4.375639269641208	INTERFERON ALFACON-1	rxcui:59744	INTERFERON ALFACON-1	TRUE	TRUE	TRUE
S1PR3	hgnc:3167	S1PR3	ChEMBL	33	agonist	2.625383561784725	FINGOLIMOD HYDROCHLORIDE	rxcui:1012891	FINGOLIMOD HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.1526385791735305	INFIGRATINIB PHOSPHATE	ncit:C175088	INFIGRATINIB PHOSPHATE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.025003653	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.019739726	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.051277023	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.042379073	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.041672755	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.054187483	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.1235474617310458	LOXAPINE HYDROCHLORIDE	rxcui:91138	LOXAPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.026779381	ZIPRASIDONE MESYLATE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
KCNK9	hgnc:6283	KCNK9	ChEMBL	33	potentiator	0.2430910705356227	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.026779381	ZIPRASIDONE HYDROCHLORIDE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
CA12	hgnc:1371	CA12	ChEMBL	33	inhibitor	0.3125456621172291	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1103102336884338	TROLEANDOMYCIN	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	ChEMBL	33	blocker	0.091476779	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	blocker	0.071148606	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNS1	hgnc:6300	KCNS1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNA4	hgnc:6222	KCNA4	ChEMBL	33	blocker	0.1829535583125243	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNS3	hgnc:6302	KCNS3	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	ChEMBL	33	blocker	0.1600843635234588	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNA10	hgnc:6219	KCNA10	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH4	hgnc:6253	KCNH4	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	positive modulator	1.400204566285186	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.2792961235941196	INFIGRATINIB PHOSPHATE	ncit:C175088	INFIGRATINIB PHOSPHATE	TRUE	FALSE	FALSE
PDE6C	hgnc:8787	PDE6C	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CA6	hgnc:1380	CA6	ChEMBL	33	inhibitor	0.6250913242344582	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
PDE6G	hgnc:8789	PDE6G	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE1C	hgnc:8776	PDE1C	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PDE1B	hgnc:8775	PDE1B	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1250182648468916	TIVOZANIB HYDROCHLORIDE	rxcui:2534245	TIVOZANIB HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.1164249916534246	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.090064616	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.2561349816375342	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.3040984820600068	BREXPIPRAZOLE	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	OSIMERTINIB MESYLATE	rxcui:1721559	OSIMERTINIB MESYLATE	TRUE	FALSE	FALSE
BLK	hgnc:1057	BLK	ChEMBL	33	inhibitor	0.065799087	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	ChEMBL	33	inhibitor	0.054187483	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.034544521	ENMD-981693	drugbank:DB16891	ENMD-981693	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.1226814748497534	CHF4227	chembl:CHEMBL3545355	CHF4227	FALSE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	1.250182648468916	EBDAROKIMAB	ncit:C179082	EBDAROKIMAB	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	ChEMBL	33	inhibitor	0.002176213	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1562728310586145	4SC-203	drugbank:DB12669	4SC-203	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.01484106	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
BLK	hgnc:1057	BLK	ChEMBL	33	inhibitor	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
LCK	hgnc:6524	LCK	ChEMBL	33	inhibitor	0.017751072	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	0.364636606	PEXMETINIB	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	1.009762908	ARQ-736	chembl:CHEMBL3545296	ARQ-736	FALSE	FALSE	FALSE
CDK13	hgnc:1733	CDK13	ChEMBL	33	inhibitor	0.4375639269641208	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.2853677784548614	AZD-6703	iuphar.ligand:7687	AZD6703	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	agonist	0.032134438	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.081030357	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK16	hgnc:8749	CDK16	ChEMBL	33	inhibitor	0.4375639269641208	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	AMIVANTAMAB	rxcui:2549198	AMIVANTAMAB-VMJW	TRUE	FALSE	TRUE
CDK17	hgnc:8750	CDK17	ChEMBL	33	inhibitor	0.546954909	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
CDK14	hgnc:8883	CDK14	ChEMBL	33	inhibitor	0.546954909	AZD-5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	agonist	0.032899543	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.092443083	CC-115	drugbank:DB12740	CC-115	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	SPEBRUTINIB BESYLATE	ncit:C141425	SPEBRUTINIB BESYLATE	FALSE	FALSE	FALSE
PRKDC	hgnc:9413	PRKDC	ChEMBL	33	inhibitor	3.281729452230906	CC-115	drugbank:DB12740	CC-115	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	agonist	0.034118045	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.596678082	AZD-8330	drugbank:DB06061	AZD-8330	FALSE	FALSE	FALSE
RPS6KB2	hgnc:10437	RPS6KB2	ChEMBL	33	inhibitor	1.458546423213736	MSC-2363318A	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.5000730593875666	MK-8033	chembl:CHEMBL2323775	MK-8033	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.1643432589536604	MSC-2363318A	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1875273972703375	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.023110771	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	0.3454452054979901	PF-00477736	chembl:CHEMBL3545137	PF-00477736	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.045579576	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.2749092734853114	PLX-8394	chembl:CHEMBL4303729	PLX-8394	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	agonist	0.033701971	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.067231333	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.2612321952024601	TTP-607	chembl:CHEMBL3545327	TTP-607	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1682938180631233	WX-037	chembl:CHEMBL3545385	WX-037	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.037884323	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	0.1704794520639431	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.060492709	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.065799087	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.04464938	IRAMPANEL	ncit:C65960	IRAMPANEL	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	inhibitor	0.736088849	BRILANESTRANT	ncit:C106235	BRILANESTRANT	FALSE	FALSE	TRUE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	TALQUETAMAB	rxcui:2644447	TALQUETAMAB	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.1226814748497534	LY2245461	chembl:CHEMBL3545389	LY2245461	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.096167896	AZD8108	chembl:CHEMBL3707355	AZD8108	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.087629625	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
PRKCZ	hgnc:9412	PRKCZ	ChEMBL	33	inhibitor	0.1434635826111871	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	ChEMBL	33	inhibitor	0.021519537	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	ChEMBL	33	inhibitor	0.043039075	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
PRKCH	hgnc:9403	PRKCH	ChEMBL	33	inhibitor	0.078252863	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	modulator	0.84012274	MBX-2044	chembl:CHEMBL3545020	MBX-2044	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.2117244807890907	PEFICITINIB	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1041818873724097	AEE-788	drugbank:DB12558	AEE-788	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.04907259	AZD-4547	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	ChEMBL	33	inhibitor	2.838252499226729	KD7040	drugbank:DB05214	KD7040	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.061055432	AZD-4547	drugbank:DB12247	AZD-4547	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.062509132	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2857560339357523	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.3337351985319565	DANUSERTIB	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.089756703	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1852122442176172	PEXIDARTINIB	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.2243917574174978	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.069454592	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	0.5000730593875666	R-406	iuphar.ligand:5706	TAMATINIB	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1041818873724097	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.1374546367426557	XL-281	chembl:CHEMBL3545027	XL-281	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.1356787370431382	LY377604	chembl:CHEMBL2012520	LY377604	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.2000292237550266	ETILEVODOPA	rxcui:1421444	ETILEVODOPA	FALSE	FALSE	FALSE
CLCN2	hgnc:2020	CLCN2	ChEMBL	33	activator	17.50255707856483	COBIPROSTONE	ncit:C78117	COBIPROSTONE	FALSE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.280789686	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	1.521961485092594	CENICRIVIROC	ncit:C166464	CENICRIVIROC	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	inhibitor	1.369765336583334	BALOVAPTAN	ncit:C169802	BALOVAPTAN	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	1.009762908	LY2828360	drugbank:DB16074	LY2828360	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	0.7095631248066824	UK432097	iuphar.ligand:8420	UK-432,097	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	AXOMADOL	ncit:C72138	AXOMADOL	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	modulator	0.046965717	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	modulator	0.038104261	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	modulator	0.2243917574174979	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.3704244884352345	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.9723642821424906	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.3968833804663227	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	modulator	0.2019525816757481	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	modulator	0.063110182	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	modulator	0.192335792	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	modulator	0.096167896	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
KCNH1	hgnc:6250	KCNH1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	blocker	0.072927321	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	ChEMBL	33	blocker	0.1640864726115453	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
KCNS2	hgnc:6301	KCNS2	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNF1	hgnc:6246	KCNF1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNH3	hgnc:6252	KCNH3	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
KCNG1	hgnc:6248	KCNG1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.4717670371580817	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
ITGB1	hgnc:6153	ITGB1	ChEMBL	33	inhibitor	2.917092846427472	FIRATEGRAST	ncit:C76692	FIRATEGRAST	FALSE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	0.3500511415712966	OMARIGLIPTIN	ncit:C174662	OMARIGLIPTIN	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.6563458904461812	NAPROXEN ETEMESIL	ncit:C166529	NAPROXEN ETEMESIL	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.6789785073581185	VOSAROXIN	ncit:C95148	VOSAROXIN	FALSE	FALSE	FALSE
P2RY2	hgnc:8541	P2RY2	ChEMBL	33	agonist	5.250767123569449	DENUFOSOL TETRASODIUM	ncit:C171672	DENUFOSOL TETRASODIUM	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.1458546423213736	BECATECARIN	ncit:C1620	BECATECARIN	FALSE	FALSE	FALSE
TNFSF13	hgnc:11928	TNFSF13	ChEMBL	33	inhibitor	39.38075342677087	ATACICEPT	ncit:C81166	ATACICEPT	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.3271505995993426	REBOXETINE	rxcui:60842	REBOXETINE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.3017682254924971	BECATECARIN	ncit:C1620	BECATECARIN	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	1.981421556063943	ROBATUMUMAB	ncit:C71527	ROBATUMUMAB	FALSE	FALSE	TRUE
CD3E	hgnc:1674	CD3E	ChEMBL	33	inhibitor	0.4861821410712453	FORALUMAB	ncit:C95785	FORALUMAB	FALSE	FALSE	FALSE
NGF	hgnc:7808	NGF	ChEMBL	33	inhibitor	15.00219178	FASINUMAB	ncit:C166446	FASINUMAB	FALSE	FALSE	FALSE
PTGDS	hgnc:9592	PTGDS	ChEMBL	33	inhibitor	26.25383561784724	ANTRAFENINE	ncit:C72107	ANTRAFENINE	TRUE	FALSE	FALSE
SOST	hgnc:13771	SOST	ChEMBL	33	inhibitor	6.563458904461812	ANTI-SCLEROSTIN	chembl:CHEMBL2109572	ANTI-SCLEROSTIN	FALSE	FALSE	FALSE
TACSTD2	hgnc:11530	TACSTD2	ChEMBL	33	binder	2.917092846427472	SACITUZUMAB GOVITECAN	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.082429625	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.031254566	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	ChEMBL	33	inhibitor	1.544343271638073	CARBENOXOLONE	rxcui:2017	CARBENOXOLONE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.031254566	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.8824818695074704	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.445925021	DIHYDROTACHYSTEROL	rxcui:3429	DIHYDROTACHYSTEROL	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	0.3070624048871023	ANTITHROMBIN ALFA	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
TRM2	hgnc:12318	TRX-CAT1-2	ChEMBL	33	inhibitor	26.25383561784724	LETERMOVIR	rxcui:1988648	LETERMOVIR	TRUE	FALSE	FALSE
IFNA5	hgnc:5426	IFNA5	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
IFNA2	hgnc:5423	IFNA2	ChEMBL	33	inhibitor	0.3500511415712967	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	4.039051633514961	RALPANCIZUMAB	ncit:C152149	RALPANCIZUMAB	FALSE	FALSE	FALSE
IFNA14	hgnc:5420	IFNA14	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	AMG-729	chembl:CHEMBL2109338	AMG-729	FALSE	FALSE	FALSE
CD44	hgnc:1681	CD44	ChEMBL	33	inhibitor	2.763561643983921	PF-03475952	chembl:CHEMBL2109479	PF-03475952	FALSE	FALSE	FALSE
NOTCH2	hgnc:7882	NOTCH2	ChEMBL	33	inhibitor	15.00219178	TAREXTUMAB	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
SDC1	hgnc:10658	SDC1	ChEMBL	33	binder	52.50767123569449	INDATUXIMAB RAVTANSINE	ncit:C78840	INDATUXIMAB RAVTANSINE	FALSE	FALSE	FALSE
RPS4Y1	hgnc:10425	RPS4Y1	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
COL4A4	hgnc:2206	COL4A4	ChEMBL	33	inhibitor	17.50255707856483	TRC-093	chembl:CHEMBL2109374	TRC-093	FALSE	FALSE	FALSE
RPL29	hgnc:10331	RPL29	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS25	hgnc:10413	RPS25	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL4	hgnc:10353	RPL4	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL17	hgnc:10307	RPL17	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS26	hgnc:10414	RPS26	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL23	hgnc:10316	RPL23	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL6	hgnc:10362	RPL6	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS19	hgnc:10402	RPS19	ChEMBL	33	inhibitor	0.050488145	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL7A	hgnc:10364	RPL7A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
KCNG4	hgnc:19697	KCNG4	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	agonist	0.2734774543525755	CENEGERMIN	rxcui:2104331	CENEGERMIN-BKBJ	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.8649519486500064	ERDAFITINIB	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.7369497717290455	ERDAFITINIB	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.032899543	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.033701971	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
EEF2	hgnc:3214	EEF2	ChEMBL	33	inhibitor	0.9723642821424906	MOXETUMOMAB PASUDOTOX	rxcui:2099295	MOXETUMOMAB PASUDOTOX	TRUE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	2.100306849	NIRAPARIB TOSYLATE	rxcui:2637447	NIRAPARIB TOSYLATE	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	ChEMBL	33	agonist	1.250182648468916	ABEQUOLIXRON	ncit:C131910	ABEQUOLIXRON	FALSE	FALSE	FALSE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	1.544343271638073	TRIFAROTENE	rxcui:2205637	TRIFAROTENE	TRUE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	ChEMBL	33	agonist	2.019525817	ABEQUOLIXRON	ncit:C131910	ABEQUOLIXRON	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	binder	0.3454452054979901	TRASTUZUMAB DERUXTECAN	rxcui:2267574	FAM-TRASTUZUMAB DERUXTECAN-NXKI	TRUE	FALSE	TRUE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inverse agonist	0.7721716358190367	PITOLISANT HYDROCHLORIDE	rxcui:2197879	PITOLISANT HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	3.281729452230906	IPRAGLIFLOZIN L-PROLINE	chembl:CHEMBL4297658	IPRAGLIFLOZIN L-PROLINE	FALSE	FALSE	FALSE
AKR1B1	hgnc:381	AKR1B1	ChEMBL	33	inhibitor	1.615620653405984	EPALRESTAT	ncit:C72762	EPALRESTAT	FALSE	FALSE	FALSE
PTAFR	hgnc:9582	PTAFR	ChEMBL	33	inhibitor	4.375639269641208	RUPATADINE	ncit:C73055	RUPATADINE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.069180068	BLONANSERIN	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1682938180631233	BLONANSERIN	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	RUPATADINE	ncit:C73055	RUPATADINE	FALSE	FALSE	FALSE
CETP	hgnc:1869	CETP	ChEMBL	33	inhibitor	4.039051633514961	OBICETRAPIB	ncit:C175167	OBICETRAPIB	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.2419708351875322	DELGOCITINIB	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	ChEMBL	33	inhibitor	2.100306849	DIROXIMEL FUMARATE	rxcui:2261783	DIROXIMEL FUMARATE	TRUE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.2419708351875322	DELGOCITINIB	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.5000730593875666	MOSAPRIDE	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
TPBG	hgnc:12004	TPBG	ChEMBL	33	binder	1.312691780892362	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	BREXUCABTAGENE AUTOLEUCEL	rxcui:2387277	BREXUCABTAGENE AUTOLEUCEL	TRUE	FALSE	FALSE
RPS15	hgnc:10388	RPS15	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	TISOTUMAB VEDOTIN	rxcui:2571093	TISOTUMAB VEDOTIN-TFTV	TRUE	FALSE	FALSE
RPS27	hgnc:10416	RPS27	ChEMBL	33	inhibitor	0.078958904	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS17	hgnc:10397	RPS17	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL41	hgnc:10354	RPL41	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL36	hgnc:13631	RPL36	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL37A	hgnc:10348	RPL37A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
MTTP	hgnc:7467	MTTP	ChEMBL	33	inhibitor	13.12691780892362	IMPLITAPIDE	ncit:C65901	IMPLITAPIDE	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	binder	1.853211925965688	SUGEMALIMAB	ncit:C154550	SUGEMALIMAB	FALSE	FALSE	FALSE
ATP1A3	hgnc:801	ATP1A3	ChEMBL	33	inhibitor	0.2187819634820604	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
GCK	hgnc:4195	GCK	ChEMBL	33	activator	3.500511415712966	AZD-1656	drugbank:DB14810	AZD-1656	FALSE	FALSE	FALSE
IL33	hgnc:16028	IL33	ChEMBL	33	binder	13.12691780892362	ETOKIMAB	ncit:C167049	ETOKIMAB	FALSE	FALSE	FALSE
RPLP0	hgnc:10371	RPLP0	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL24	hgnc:10325	RPL24	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	5.250767123569449	PF-232798	drugbank:DB14813	PF-232798	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	AMDOXOVIR	ncit:C76927	AMDOXOVIR	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	cleavage	0.1226814748497534	CAMIZESTRANT	ncit:C160603	CAMIZESTRANT	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.058212496	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	ChEMBL	33	inhibitor	0.5277152888009498	APX-3330	chembl:CHEMBL578390	APX-3330	FALSE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	inhibitor	0.375054795	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.2333674277141978	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	ChEMBL	33	inhibitor	1.346350544504987	BRIMAPITIDE	ncit:C166576	BRIMAPITIDE	FALSE	FALSE	FALSE
PTGER2	hgnc:9594	PTGER2	ChEMBL	33	agonist	3.281729452230906	EVATANEPAG	ncit:C83707	EVATANEPAG	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	ChEMBL	33	inhibitor	0.1545479653736408	IDASANUTLIN	ncit:C99131	IDASANUTLIN	FALSE	FALSE	FALSE
TIGIT	hgnc:26838	TIGIT	ChEMBL	33	inhibitor	6.563458904461812	OCIPERLIMAB	ncit:C170906	OCIPERLIMAB	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.064505739	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
MYH7B	hgnc:15906	MYH7B	ChEMBL	33	activator	2.500365296937833	DANICAMTIV	ncit:C167013	DANICAMTIV	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.3088686543276147	RIPASUDIL	ncit:C152226	RIPASUDIL	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	negative modulator	0.042689164	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	cleavage	0.2453629496995069	GIREDESTRANT	ncit:C147030	GIREDESTRANT	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
PTGER3	hgnc:9595	PTGER3	ChEMBL	33	agonist	3.889457128569962	SEPETAPROST	ncit:C152337	SEPETAPROST	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	ChEMBL	33	inhibitor	0.3500511415712966	REBIMASTAT	ncit:C1875	REBIMASTAT	FALSE	FALSE	FALSE
APH1B	hgnc:24080	APH1B	ChEMBL	33	inhibitor	0.2885036881082115	NIROGACESTAT	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
PSEN2	hgnc:9509	PSEN2	ChEMBL	33	inhibitor	0.3409589041278863	NIROGACESTAT	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.3182283105193605	NLY-01	chembl:CHEMBL4650495	NLY-01	FALSE	FALSE	FALSE
ACACB	hgnc:85	ACACB	ChEMBL	33	inhibitor	0.4234489615781814	CLESACOSTAT	ncit:C177068	CLESACOSTAT	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	2.128689374420047	GEPIRONE	rxcui:2672253	GEPIRONE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.042689164	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	2.763561643983921	ATECEGATRAN METOXIL	ncit:C166758	ATECEGATRAN METOXIL	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1888765152363111	ASCIMINIB HYDROCHLORIDE	rxcui:2584303	ASCIMINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	ChEMBL	33	positive modulator	2.763561643983921	VON WILLEBRAND FACTOR HUMAN	rxcui:1812589	VONICOG ALFA	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3337351985319565	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1093909817410302	SERALUTINIB	ncit:C175203	SERALUTINIB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2938862196027677	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.031659735	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.7395446652914718	DEFOROLIMUS	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1054370908347279	SERALUTINIB	ncit:C175203	SERALUTINIB	FALSE	FALSE	FALSE
GDF2	hgnc:4217	GDF2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.093909817410302	DALANTERCEPT	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1350505947420126	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.089046362	PAZOPANI	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	3.424413341458336	GTS-21	drugbank:DB05708	GTS-21	FALSE	FALSE	FALSE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.060772768	PKI-591	ncit:C84837	PI3K/MTOR KINASE INHIBITOR PF-04691502	FALSE	FALSE	TRUE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.088396753	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.075768645	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1470803115845784	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
WEE1	hgnc:12761	WEE1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	8.078103267029922	MK 1775	hemonc:32625	ADAVOSERTIB	FALSE	FALSE	TRUE
F8	hgnc:3546	F8	ChEMBL	33	positive modulator	3.088686543276147	OMFILOCTOCOG ALFA	ncit:C175177	OMFILOCTOCOG ALFA	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4688184931758437	DEHYDROEQUOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	COSMIC	4-Sep-20	NULL	0.6721614540713904	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.029665351	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	1.666910197958555	3-(3-STIBONOPHENYL)PROPANOIC ACID	iuphar.ligand:8877	P6949	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FLUORANTHENE	chembl:CHEMBL355014	FLUORANTHENE	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	0.729273212	NADROPARIN CALCIUM	ncit:C61320	NADROPARIN CALCIUM	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	BENSERAZIDE	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	MALATHION	rxcui:6606	MALATHION	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.012442576	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	NSC-117271	chembl:CHEMBL287689	CHEMBL:CHEMBL287689	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.009995749	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
FGG	hgnc:3694	FGG	ChEMBL	33	cleavage	2.187819634820604	PLASMINOGEN	rxcui:2557200	PLASMINOGEN	TRUE	FALSE	FALSE
CYBB	hgnc:2578	CYBB	DTC	9/2/20	NULL	0.8204323630577265	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
SMARCA2	hgnc:11098	SMARCA2	DTC	9/2/20	NULL	0.7292732116068681	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	AZELASTINE HYDROCHLORIDE	rxcui:235824	AZELASTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.3889457128569962	ENSIFENTRINE	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	MMV006389	chembl:CHEMBL586000	CHEMBL:CHEMBL586000	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	TIAPROFENIC ACID	rxcui:38253	TIAPROFENIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	DTC	9/2/20	NULL	2.100306849	URB597	iuphar.ligand:4339	URB597	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00359617	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	(E)-DIBENZYLIDENEACETONE	chembl:CHEMBL17201	CHEMBL:CHEMBL17201	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	TACRINE	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.033106981	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00399693	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	PHENAZINE-1-CARBOXYLIC ACID	chembl:CHEMBL463686	PHENAZINE-1-CARBOXYLIC ACID	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	1-AMINOCYCLOPROPANECARBOXYLIC ACID HCL	chembl:CHEMBL1255660	CHEMBL:CHEMBL1255660	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	GINSENOSIDE RH1	chembl:CHEMBL466844	GINSENOSIDE RH1	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.003068829	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	TRITIOZINE	ncit:C90780	TRITIOZINE	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1060761035064535	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.04593847	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
CRTC2	hgnc:27301	CRTC2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4688184931758437	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	GNF-PF-3416	chembl:CHEMBL579550	CHEMBL:CHEMBL579550	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	ALTISSIMACOUMARIN D	chembl:CHEMBL2071526	ALTISSIMACOUMARIN D	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.014114965	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	BENZENE-1,2-DIAMINE	chembl:CHEMBL70582	CHEMBL:CHEMBL70582	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.034590034	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	CUCURBITACIN B	iuphar.ligand:12432	CUCURBITACIN B	FALSE	FALSE	FALSE
TYR	hgnc:12442	TYR	DTC	9/2/20	NULL	0.1491695205559502	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	TIOTIDINE	ncit:C152643	TIOTIDINE	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.052090944	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	GNF-PF-1094	chembl:CHEMBL415914	CHEMBL:CHEMBL415914	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	2-AMINOANTHRACENE	chembl:CHEMBL83154	2-AMINOANTHRACENE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002552882	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	THIOPROPERAZINE MESYLATE	ncit:C80010	THIOPROPERAZINE MESYLATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	DITHIOLETHIONE	chembl:CHEMBL368700	DITHIOLETHIONE	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.028356978	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	CHRYSIN DIMETHYL ETHER	chembl:CHEMBL275391	CHRYSIN DIMETHYL ETHER	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.056581542	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012112496	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.064347636	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.049723174	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.033148782	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.018860514	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006811217	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010588359	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
CRTC1	hgnc:16062	CRTC1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4688184931758437	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
SLC15A1	hgnc:10920	SLC15A1	DTC	9/2/20	NULL	7.001022831425932	GLYCYLSARCOSINE	iuphar.ligand:4659	[3H]GLYSAR	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006439499	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.001325784	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.1539814405738841	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1426838892274307	ALDRIN	chembl:CHEMBL195953	ALDRIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00402481	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	NSC-88165	chembl:CHEMBL1709259	CHEMBL:CHEMBL1709259	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	DTC	9/2/20	NULL	0.2035181055647073	RO-229735	chembl:CHEMBL2170369	CHEMBL:CHEMBL2170369	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018006746	ZIDOVUDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.01715937	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.037003292	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GART	hgnc:4163	GART	DTC	9/2/20	NULL	0.5122699632750684	LOMETREXOL	ncit:C979	LOMETREXOL	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	PROSTAGLANDIN A2	iuphar.ligand:6279	PROSTAGLANDIN A2	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	PYRIDOSTIGMINE	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.9907107780319716	LINSITINIB	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.019142425	CIANIDANOL	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.010609754	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	MORNIFLUMATE	rxcui:30225	MORNIFLUMATE	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.006068848	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.072927321	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.039778539	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005677733	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.025390557	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	3,5-DINITROCATECHOL (OR-486)	chembl:CHEMBL168276	3,5-DINITROCATECHOL (OR-486)	FALSE	FALSE	FALSE
GLI1	hgnc:4317	GLI1	DTC	9/2/20	NULL	5.834185692854944	COLUBRINIC ACID	chembl:CHEMBL470503	COLUBRINIC ACID	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.6604738520213144	ANDROGRAPHOLIDE	ncit:C61637	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	COSMIC	4-Sep-20	NULL	0.6241137025199848	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	4.200613699	SILYCHRISTIN	chembl:CHEMBL130493	SILICRISTIN A	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.045898314	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.2983390411119005	AROMOLINE	chembl:CHEMBL509999	AROMOLINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	DNDI1417995	chembl:CHEMBL1439833	CHEMBL:CHEMBL1439833	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	SJ000200944	chembl:CHEMBL600173	CHEMBL:CHEMBL600173	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.2592971419046642	SPERMINE	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	2-TERT-BUTYLPHENOL	chembl:CHEMBL108851	CHEMBL:CHEMBL108851	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.4526523382387456	NSC-77833	chembl:CHEMBL1287981	CHEMBL:CHEMBL1287981	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.013286354	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.087077398	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.084012274	METHOXYCHLOR	rxcui:2598123	METHOXYCHLOR	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006555265	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-3276	chembl:CHEMBL582081	CHEMBL:CHEMBL582081	FALSE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	DTC	9/2/20	NULL	0.093763699	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	COSMIC	4-Sep-20	NULL	1.657092009619794	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	SODIUM AMINOSALICYLATE	chembl:CHEMBL1200966	SODIUM AMINOSALICYLATE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.015118823	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.020672312	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	DTC	9/2/20	NULL	1.750255707856483	PF-750	iuphar.ligand:5244	PF750	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	SJ000039423	chembl:CHEMBL589207	CHEMBL:CHEMBL589207	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.004154745	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1620607136904151	ALDRIN	chembl:CHEMBL195953	ALDRIN	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.075442056	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006054153	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00202529	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.017751072	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	BUCLADESINE	ncit:C83562	BUCLADESINE	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.053633985	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	BRILLIANT GREEN OXALATE	chembl:CHEMBL1789985	BRILLIANT GREEN OXALATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.004352426	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.013087655	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	MALTOL	rxcui:1362894	MALTOL	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2187819634820604	BENZENE-1,2-DIAMINE	chembl:CHEMBL70582	CHEMBL:CHEMBL70582	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV007181	chembl:CHEMBL577014	CHEMBL:CHEMBL577014	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	CIS-(Z)-FLUPENTHIXOL DIHYDROCHLORIDE	chembl:CHEMBL1256995	CHEMBL:CHEMBL1256995	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002861765	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.090530468	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.089756703	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	0.8751278539282416	METHACHOLINE CHLORIDE	rxcui:40165	METHACHOLINE CHLORIDE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	DTC	9/2/20	NULL	0.8751278539282417	ELUXADOLINE	rxcui:1653781	ELUXADOLINE	TRUE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	1.346350544504987	DNDI1417884	chembl:CHEMBL1346025	CHEMBL:CHEMBL1346025	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.073540156	BENSERAZIDE	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.010403739	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.034184682	R-N-PROPYLNORAPOMORPHINE	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	METHOCARBAMOL	rxcui:6845	METHOCARBAMOL	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.017751072	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.007110043	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	SPICLOMAZINE	ncit:C66557	SPICLOMAZINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	L-694247	iuphar.ligand:15	L-694,247	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	WHILE OLIVETOL	chembl:CHEMBL154533	WHILE OLIVETOL	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.017799211	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.2117244807890907	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.020446912	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	O-DEMETHYLATED ADAPALENE	iuphar.ligand:3431	AHPN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.016764901	EPIGALOCATECHIN GALLATE	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	PIPOBROMAN	rxcui:8347	PIPOBROMAN	TRUE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.5048814541893701	GW8510	chembl:CHEMBL1276446	CHEMBL:CHEMBL1276446	FALSE	FALSE	FALSE
INPP5D	hgnc:6079	INPP5D	DTC	9/2/20	NULL	52.50767123569449	TURNAGAINOLIDE B	chembl:CHEMBL1784528	TURNAGAINOLIDE B	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	DILAZEP	ncit:C65389	DILAZEP	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	METHYL ROBUSTONE	chembl:CHEMBL1403041	METHYL ROBUSTONE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.010193685	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	IRL-2500	iuphar.ligand:3887	IRL 2500	FALSE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	DTC	9/2/20	NULL	6.563458904461812	NSC-12352	chembl:CHEMBL392369	CHEMBL:CHEMBL392369	FALSE	FALSE	FALSE
CASP2	hgnc:1503	CASP2	DTC	9/2/20	NULL	2.917092846427472	SPERMINE	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	FLUORESCEIN DIPHOSPHATE	chembl:CHEMBL1818143	FLUORESCEIN DIPHOSPHATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	PYRIDOSTIGMINE	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.1902451856365742	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.1367387271762877	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	TCMDC-125321	chembl:CHEMBL587449	CHEMBL:CHEMBL587449	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.013229446	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
GCGR	hgnc:4192	GCGR	DTC	9/2/20	NULL	1.670698630226643	GLUCAGON	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.006068848	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.008428198	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	TCMDC-123579	chembl:CHEMBL533954	CHEMBL:CHEMBL533954	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-125281	chembl:CHEMBL525486	CHEMBL:CHEMBL525486	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.059364241	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1715936968486748	LINSIDOMINE	ncit:C72628	LINSIDOMINE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.1093909817410302	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.068191781	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	GANGALEOIDIN	chembl:CHEMBL1491099	GANGALEOIDIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.010191706	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.015290527	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.000901682	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.018619742	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002936671	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.2966535098061835	DNDI1417411	chembl:CHEMBL1445650	CHEMBL:CHEMBL1445650	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FURAZABOL	ncit:C65782	FURAZABOL	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	AMARANTH	chembl:CHEMBL1408927	AMARANTH	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-1631	chembl:CHEMBL577222	CHEMBL:CHEMBL577222	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.012378046	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.010195664	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.7001022831425933	2-PHENOXYETHANOL	rxcui:89552	PHENOXYETHANOL	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013299815	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.4930297768609811	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	CHLORHEXIDINE HYDROCHLORIDE	rxcui:2361	CHLORHEXIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	GNF-2	iuphar.ligand:5935	BCR-ABL INHIBITOR GNF-2	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.02321294	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.019665794	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	ARISTOLACTONE	chembl:CHEMBL2333547	ARISTOLACTONE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.070197421	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(+)-ELEUTHERIN	chembl:CHEMBL594153	CHEMBL:CHEMBL594153	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	NSC-172033	chembl:CHEMBL238624	CHEMBL:CHEMBL238624	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.006043701	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.018719312	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	ANTAZOLINE HYDROCHLORIDE	rxcui:81954	ANTAZOLINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.019995305	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	HALCINONIDE	rxcui:5084	HALCINONIDE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.01169957	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.051629962	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.077444943	GNF-PF-2954	chembl:CHEMBL582722	CHEMBL:CHEMBL582722	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.038722471	GNF-PF-3148	chembl:CHEMBL81782	CHEMBL:CHEMBL81782	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	4-HYDROXYDERRICIN	chembl:CHEMBL458094	CHEMBL:CHEMBL458094	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001886187	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.095122593	PHENACYL CHLORIDE	iuphar.ligand:6285	OMEGA-CHLOROACETOPHENONE	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.03729238	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00172405	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2651902587661338	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2328499833068492	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.00453826	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.01037701	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.212152207	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1801292323694494	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.8975670296699914	SPIRUCHOSTATIN C	chembl:CHEMBL1835659	SPIRUCHOSTATIN C	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2892984641085096	BUTYRYLHYDROXAMIC ACID	chembl:CHEMBL1672332	BUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.011316308	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.1921012362281506	PHENYLBUTANOIC ACID	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.015335184	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003096702	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BETAMETHASONE SODIUM PHOSPHATE	rxcui:203220	BETAMETHASONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	DIPHENADIONE	ncit:C75156	DIPHENADIONE	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.1161674142382621	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002663877	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.01555322	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.9907107780319716	NSC-7936	chembl:CHEMBL415711	CHEMBL:CHEMBL415711	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.010247399	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.251232877	CLOSANTEL	ncit:C79920	CLOSANTEL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	O-DEMETHYLATED ADAPALENE	iuphar.ligand:3431	AHPN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TECTOQUINONE	chembl:CHEMBL21745	TECTOQUINONE	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.8751278539282418	FENDILINE HYDROCHLORIDE	rxcui:236767	FENDILINE HYDROCHLORIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	NSC-61836	chembl:CHEMBL521171	CHEMBL:CHEMBL521171	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	3,3',4',5-TETRACHLOROSALICYLANILIDE	chembl:CHEMBL291338	3,3',4',5-TETRACHLOROSALICYLANILIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	CYSTEAMINE	rxcui:1426886	CYSTEAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	TCMDC-124536	chembl:CHEMBL580851	CHEMBL:CHEMBL580851	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	GNF-PF-3889	chembl:CHEMBL598270	CHEMBL:CHEMBL598270	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.026372512	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.055819636	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005795549	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	LIDAMIDINE HYDROCHLORIDE	ncit:C82241	LIDAMIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.006829822	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005412046	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.012020987	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	DNDI1417346	chembl:CHEMBL1490332	CHEMBL:CHEMBL1490332	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.019254738	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	SJ000260214	chembl:CHEMBL602740	CHEMBL:CHEMBL602740	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.089756703	LOPINAVIR	rxcui:195088	LOPINAVIR	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ALOE-EMODIN	chembl:CHEMBL40275	ALOE-EMODIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.020836377	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.018540844	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011738804	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.024536295	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DIMETHISTERONE	ncit:C65404	DIMETHISTERONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	YANGONIN	chembl:CHEMBL1098658	YANGONIN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.016086909	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TRIFLUMIZOLE	chembl:CHEMBL463781	TRIFLUMIZOLE	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	1.235474617310459	20(S)-PROTOPANAXADIOL	chembl:CHEMBL375563	CHEMBL:CHEMBL375563	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	DTC	9/2/20	NULL	0.1930429089547591	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	CAMBINOL	drugbank:DB15493	CAMBINOL	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.07458476	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.008143249	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.069454592	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.087512785	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIIA	chembl:CHEMBL1094690	AESCULIOSIDE IIIA	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.025298806	GLAFENINE	ncit:C72119	GLAFENINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.2143170254518142	TCMDC-125784	chembl:CHEMBL581574	CHEMBL:CHEMBL581574	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007479725	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	SJ000260153	chembl:CHEMBL589717	CHEMBL:CHEMBL589717	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-28620	chembl:CHEMBL1414990	CHEMBL:CHEMBL1414990	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	CAPTAN	rxcui:1368147	CAPTAN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002170994	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	DENATONIUM BENZOATE	rxcui:1313232	DENATONIUM BENZOATE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	SJ000039423	chembl:CHEMBL589207	CHEMBL:CHEMBL589207	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	FLUDIOXONIL	chembl:CHEMBL485833	FLUDIOXONIL	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.2083637747448194	DNDI1417031	chembl:CHEMBL1333049	CHEMBL:CHEMBL1333049	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.040782657	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	ANANDAMIDE	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	4.773424657790408	NCI-372939	chembl:CHEMBL84440	CHEMBL:CHEMBL84440	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	1.141471113819445	SANSALVAMIDE A-AMIDE	chembl:CHEMBL192264	CHEMBL:CHEMBL192264	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.012573676	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123661	chembl:CHEMBL581240	CHEMBL:CHEMBL581240	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.3409589041278864	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	SC-19220	iuphar.ligand:1922	SC-19220	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	CHINIOFON	ncit:C76415	CHINIOFON	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	DITHIOLETHIONE	chembl:CHEMBL368700	DITHIOLETHIONE	FALSE	FALSE	FALSE
POLL	hgnc:9184	POLL	DTC	9/2/20	NULL	8.751278539282415	TALAROFLAVONE	chembl:CHEMBL408995	TALAROFLAVONE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1411496538593938	ORTHO-PHTHALALDEHYDE	chembl:CHEMBL160145	ORTHO-PHTHALALDEHYDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006756874	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	DTC	9/2/20	NULL	0.305277158	RO-229735	chembl:CHEMBL2170369	CHEMBL:CHEMBL2170369	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	BENZALKONIUM CHLORIDE	rxcui:1379	BENZALKONIUM CHLORIDE	TRUE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.036212187	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
NPY1R	hgnc:7956	NPY1R	DTC	9/2/20	NULL	1.750255707856483	DNDI1417776	chembl:CHEMBL1585652	CHEMBL:CHEMBL1585652	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	DNDI1417383	chembl:CHEMBL2094665	CHEMBL:CHEMBL2094665	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	0.2447910080918158	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	DNDI1417827	chembl:CHEMBL1363249	CHEMBL:CHEMBL1363249	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.2333674277141977	FLUDIOXONIL	chembl:CHEMBL485833	FLUDIOXONIL	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.022439176	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.084963869	ORTHO-PHTHALALDEHYDE	chembl:CHEMBL160145	ORTHO-PHTHALALDEHYDE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.015344147	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	MMV020651	chembl:CHEMBL549216	CHEMBL:CHEMBL549216	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE	chembl:CHEMBL513116	N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	FOSFONET	drugbank:DB02823	PHOSPHONOACETIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.033985548	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	ISOQUERCETIN	ncit:C117288	ISOQUERCETIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007727398	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	MIANSERIN HYDROCHLORIDE	rxcui:203127	MIANSERIN HYDROCHLORIDE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW703087X	chembl:CHEMBL205798	GW703087X	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	chembl:CHEMBL224214	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	1.093909817410302	BAS-0338868	chembl:CHEMBL378903	CHEMBL:CHEMBL378903	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	BETA-HYDRASTINE	chembl:CHEMBL462731	CHEMBL:CHEMBL462731	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.210030685	TCMDC-125528	chembl:CHEMBL375673	CHEMBL:CHEMBL375673	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.043323161	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001124265	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007366396	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	LACTOFEN	chembl:CHEMBL1243178	LACTOFEN	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-75270	chembl:CHEMBL1333982	CHEMBL:CHEMBL1333982	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DESOXYCORTICOSTERONE PIVALATE	rxcui:22537	DESOXYCORTICOSTERONE PIVALATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.03292017	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-3265	chembl:CHEMBL581868	CHEMBL:CHEMBL581868	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007330402	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	CLOFENOXYDE	ncit:C78034	CLOFENOXYDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.00777661	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.023171964	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
HNRNPC	hgnc:5035	HNRNPC	DTC	9/2/20	NULL	5.834185692854945	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.034567262	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	QUINIZARIN	chembl:CHEMBL17594	QUINIZARIN	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.252440727	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	DIGITOXIGENIN	drugbank:DB04177	DIGITOXIGENIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	BETA-CCM	chembl:CHEMBL453066	BETA-CCM	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	NSC-93401	chembl:CHEMBL452954	CHEMBL:CHEMBL452954	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	NSC-48300	chembl:CHEMBL1091971	CHEMBL:CHEMBL1091971	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	DTC	9/2/20	NULL	1.312691780892362	BERBERRUBINE	chembl:CHEMBL203135	BERBERRUBINE	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	DTC	9/2/20	NULL	0.9053046764774912	BERBERRUBINE	chembl:CHEMBL203135	BERBERRUBINE	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	1.193356164447602	GNF-PF-231	chembl:CHEMBL601167	CHEMBL:CHEMBL601167	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	PF-03715455	drugbank:DB12138	PF-03715455	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.3500511415712966	ANTHRAQUINONE	chembl:CHEMBL55659	ANTHRAQUINONE	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.042140988	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008581087	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1041818873724097	TCMDC-125738	chembl:CHEMBL527585	CHEMBL:CHEMBL527585	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.015118823	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	MMV020651	chembl:CHEMBL549216	CHEMBL:CHEMBL549216	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	DIHYDROSPINGOSINE	iuphar.ligand:2453	DIHYDROSPHINGOSINE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.060492709	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	GNF-PF-4668	chembl:CHEMBL584860	CHEMBL:CHEMBL584860	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.729273212	NSC-77833	chembl:CHEMBL1287981	CHEMBL:CHEMBL1287981	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001976425	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	DNDI1417111	chembl:CHEMBL2094456	CHEMBL:CHEMBL2094456	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.007264481	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.008613463	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.015516451	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.011855424	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	PECTOLINARIGENIN	chembl:CHEMBL78010	PECTOLINARIGENIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	DNDI1417099	chembl:CHEMBL1565444	CHEMBL:CHEMBL1565444	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.026748686	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	EPIRUBICIN HYDROCHLORIDE	rxcui:203213	EPIRUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005574063	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	CID 649849	chembl:CHEMBL405914	CHEMBL:CHEMBL405914	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	TETRABROMOBENZOTRIAZOLE	iuphar.ligand:9372	TBBT	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.07631929	NSC-61836	chembl:CHEMBL521171	CHEMBL:CHEMBL521171	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	DOMIPHEN BROMIDE	rxcui:49255	DOMIPHEN BROMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	GNF-PF-5411	chembl:CHEMBL15134	CHEMBL:CHEMBL15134	FALSE	FALSE	FALSE
EPHX2	hgnc:3402	EPHX2	DTC	9/2/20	NULL	1.000146118775133	6BIO	chembl:CHEMBL409450	6BIO	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.2651902587661338	2,4-DIHYDROXYBENZOPHENONE	chembl:CHEMBL1392	2,4-DIHYDROXYBENZOPHENONE	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.065634589	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	MMV665817	chembl:CHEMBL590919	CHEMBL:CHEMBL590919	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.006233104	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.056399217	L-165041	drugbank:DB08078	{4-[3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPOXY]PHENOXY}ACETIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	CITRIC ACID	rxcui:21183	CITRIC ACID	TRUE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.3409589041278864	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	ATHRAQUINONES A	chembl:CHEMBL55814	ATHRAQUINONES A	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.021733308	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	4-AMINOBENZAMIDINE DIHYDROCHLORIDE	chembl:CHEMBL545184	CHEMBL:CHEMBL545184	FALSE	FALSE	FALSE
KLF5	hgnc:6349	KLF5	DTC	9/2/20	NULL	1.640864726115453	CID 926663	chembl:CHEMBL265686	CHEMBL:CHEMBL265686	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	PERHEXILINE MALEATE	rxcui:33169	PERHEXILINE MALEATE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.01708122	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.006912542	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	HYDROCOTARNINE	chembl:CHEMBL1606295	HYDROCOTARNINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	BUFOGENIN	ncit:C77829	BUFOGENIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	IDAZOXAN HYDROCHLORIDE	chembl:CHEMBL543467	IDAZOXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.005303805	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	DNDI1417157	chembl:CHEMBL1576659	CHEMBL:CHEMBL1576659	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	RISEDRONIC ACID	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	1.166837138570989	CITRIC ACID	rxcui:21183	CITRIC ACID	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	OXADIAZON	chembl:CHEMBL1080648	OXADIAZON	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.014993624	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	SC-560	iuphar.ligand:10240	SC-560	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	METHYLROSANILINE	chembl:CHEMBL592105	METHYLROSANILINE	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.003097798	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.1058622403945453	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.051478109	GUTHION	chembl:CHEMBL530115	GUTHION	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.007470148	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TCMDC-124064	chembl:CHEMBL537045	CHEMBL:CHEMBL537045	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.017649637	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.4070362111294147	SJ000019194	chembl:CHEMBL592106	CHEMBL:CHEMBL592106	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.009860596	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	INDIGOTINDISULFONATE	rxcui:1426889	INDIGO	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.093098708	CLOROTEPINE	ncit:C77572	CLOROTEPINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	TRANSPLATIN	chembl:CHEMBL1386	TRANSPLATIN	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.7001022831425933	TCMDC-124495	chembl:CHEMBL532452	CHEMBL:CHEMBL532452	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.035098711	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003772103	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	6-METHYLCOUMARIN	chembl:CHEMBL443436	CHEMBL:CHEMBL443436	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.4667348554283956	20(S)-PROTOPANAXADIOL	chembl:CHEMBL375563	CHEMBL:CHEMBL375563	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	TCMDC-125814	chembl:CHEMBL533082	CHEMBL:CHEMBL533082	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.009539911	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	3-HYDROXYFLAVONOL	chembl:CHEMBL242172	CHEMBL:CHEMBL242172	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.00314681	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.2792961235941196	E-64	chembl:CHEMBL374508	E-64	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	DNDI1417263	chembl:CHEMBL1431115	CHEMBL:CHEMBL1431115	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013964806	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	VIDARABINE	rxcui:11194	VIDARABINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005412046	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	GLAFENINE	ncit:C72119	GLAFENINE	TRUE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	0.4688184931758437	(R)-PIA	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.058083707	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.043109746	(E)-DIBENZYLIDENEACETONE	chembl:CHEMBL17201	CHEMBL:CHEMBL17201	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.07458476	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.1084869240406911	ZD-7155	iuphar.ligand:8324	ZD-7155	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	NSC-102029	chembl:CHEMBL74913	CHEMBL:CHEMBL74913	FALSE	FALSE	FALSE
PLCG1	hgnc:9065	PLCG1	DTC	9/2/20	NULL	0.7955707762984016	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	L-732138	iuphar.ligand:9461	L-732,138	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	NSC-111847	chembl:CHEMBL1984884	CHEMBL:CHEMBL1984884	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	TRANILAST	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1500219178162699	MMV006513	chembl:CHEMBL585622	CHEMBL:CHEMBL585622	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	DTC	9/2/20	NULL	0.4123639102279672	AZ628	iuphar.ligand:8475	AZ628	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	SJ000018309	chembl:CHEMBL591363	CHEMBL:CHEMBL591363	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.015945239	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CAMK1D	hgnc:19341	CAMK1D	DTC	9/2/20	NULL	0.063722902	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	NEROLIDOL	rxcui:2371699	NEROLIDOL	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.00854617	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PREDNISOLONE HEMISUCCINATE	drugbank:DB14633	PREDNISOLONE HEMISUCCINATE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.073954467	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001044139	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-358518	chembl:CHEMBL352222	CHEMBL:CHEMBL352222	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1458546423213736	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.060008767	TCMDC-125602	chembl:CHEMBL580183	CHEMBL:CHEMBL580183	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011810092	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	(S)-VERAPAMIL	chembl:CHEMBL36148	(S)-VERAPAMIL	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.050634206	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	NSC-663284	drugbank:DB17038	NSC-663284	FALSE	FALSE	FALSE
HSD17B3	hgnc:5212	HSD17B3	DTC	9/2/20	NULL	1.591141552596803	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	SJ000032081	chembl:CHEMBL590184	CHEMBL:CHEMBL590184	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	DTC	9/2/20	NULL	0.5515511684421691	TACRINE	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.016236138	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.031488858	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.019404165	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.01917038	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.018942161	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SJ000014858	chembl:CHEMBL591628	CHEMBL:CHEMBL591628	FALSE	FALSE	FALSE
CASP8	hgnc:1509	CASP8	DTC	9/2/20	NULL	4.200613698855561	20(S)-PROTOPANAXADIOL	chembl:CHEMBL375563	CHEMBL:CHEMBL375563	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.2169738480813822	LAS38096	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	GUAIAZULENE	rxcui:26290	GUAIAZULENE	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	4.200613699	SPERMINE BIS-1-NAPG	chembl:CHEMBL2347630	CHEMBL:CHEMBL2347630	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.067317527	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW828525X	chembl:CHEMBL185939	GW828525X	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	DIPHENADIONE	ncit:C75156	DIPHENADIONE	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.07767407	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	DNDI1417149	chembl:CHEMBL1622802	CHEMBL:CHEMBL1622802	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	3',4'-DIMETHOXYFLAVONE	chembl:CHEMBL91153	3',4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.007426828	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.01888086	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.016434326	CEFOTAXIME SODIUM	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.002000292	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.028692717	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.1290114772375786	LAS38096	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.6250913242344582	CEP-5214	chembl:CHEMBL150894	CEP-5214	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	FENDILINE HYDROCHLORIDE	rxcui:236767	FENDILINE HYDROCHLORIDE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.013716738	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.015892152	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.2625383561784725	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW280670X	chembl:CHEMBL270054	GW280670X	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.033412454	CYPROTERONE	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003844181	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.009539911	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	NSC-677438	chembl:CHEMBL118678	CHEMBL:CHEMBL118678	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1651184630053286	URSOLIC ACID	rxcui:1426931	URSOLIC ACID	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.013613604	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	O,O'-DIMETHYLCAFFEIC ACID	chembl:CHEMBL320295	O,O'-DIMETHYLCAFFEIC ACID	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.045579576	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002170994	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.023274677	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.050879526	PENTAMIDINE DIISETHIONATE	chembl:CHEMBL361506	PENTAMIDINE ISETHIONATE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.02832129	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.4102161815288632	DIPYRIDYL	chembl:CHEMBL39879	DIPYRIDYL	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.034318739	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	GLUTAMIC ACID HYDROCHLORIDE	rxcui:91269	GLUTAMIC ACID HYDROCHLORIDE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	DTC	9/2/20	NULL	0.1544343271638073	SKIMMIANINE	chembl:CHEMBL21396	SKIMMIANINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	MMV000704	chembl:CHEMBL582478	CHEMBL:CHEMBL582478	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.015184405	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	BILIRUBIN	iuphar.ligand:4577	BILIRUBIN	FALSE	FALSE	FALSE
PLK2	hgnc:19699	PLK2	DTC	9/2/20	NULL	1.875273972703374	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.047886613	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	NSC-31884	chembl:CHEMBL74644	CHEMBL:CHEMBL74644	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	GNF-PF-308	chembl:CHEMBL600334	CHEMBL:CHEMBL600334	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.081030357	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.020226376	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	NALED	chembl:CHEMBL1887067	NALED	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.095468493	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001223613	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.2763561643983921	VINCRISTINE SULFATE	rxcui:11203	VINCRISTINE SULFATE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	LASSBIO-294	chembl:CHEMBL233194	CHEMBL:CHEMBL233194	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.3804903712731485	QUINAPRIL HYDROCHLORIDE	rxcui:235759	QUINAPRIL HYDROCHLORIDE	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.729273212	TERAZOSIN HYDROCHLORIDE HYDRATE	chembl:CHEMBL1201091	TERAZOSIN HYDROCHLORIDE HYDRATE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.016574391	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.046798281	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.009318132	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PHENYL 2-PHENYLETHENESULFONATE	chembl:CHEMBL443343	CHEMBL:CHEMBL443343	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006574965	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.1770916399180253	3,4,5-TRIM-4'-MTS	chembl:CHEMBL74189	CHEMBL:CHEMBL74189	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.029698909	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	DEXPROPRANOLOL HYDROCHLORIDE	ncit:C77945	DEXPROPRANOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	2-STYRYL-QUINOLINE	chembl:CHEMBL127579	CHEMBL:CHEMBL127579	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	CID 893238	chembl:CHEMBL473735	CHEMBL:CHEMBL473735	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	H89	drugbank:DB07995	H-89	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DODECYL GALLATE	rxcui:1596928	DODECYL GALLATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	TRIOXSALEN	rxcui:10844	TRIOXSALEN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DNDI1417185	chembl:CHEMBL1549738	CHEMBL:CHEMBL1549738	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW513184X	chembl:CHEMBL1789961	GW513184X	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	BENZYDAMINE	rxcui:1425	BENZYDAMINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004176557	SOTALOL	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	1.750255707856483	N-[6-(4-CHLOROPHENYL)-7-(2,4-DICHLOROPHENYL)-2,2-DIMETHYL-3,4-DIHYDRO-2H-PYRANO[2,3-B]PYRIDINE-4-YL]-4,4,4-TRIFLUORO-3-HYDROXYBUTANAMIDE (DIASTEREOMERIC MIX)	chembl:CHEMBL1097456	N-[6-(4-CHLOROPHENYL)-7-(2,4-DICHLOROPHENYL)-2,2-DIMETHYL-3,4-DIHYDRO-2H-PYRANO[2,3-B]PYRIDINE-4-YL]-4,4,4-TRIFLUORO-3-HYDROXYBUTANAMIDE (DIASTEREOMERIC MIX)	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	PHTHALIC ACID	drugbank:DB02746	PHTHALIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	L-PHENYLALANINE	rxcui:8156	PHENYLALANINE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	CID 5310801	chembl:CHEMBL260451	CHEMBL:CHEMBL260451	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.033148782	BROXURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	ALTISSIMACOUMARIN C	chembl:CHEMBL2071525	ALTISSIMACOUMARIN C	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004287741	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	REL-CARINATIN D	chembl:CHEMBL2332128	CHEMBL:CHEMBL2332128	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1479089330582944	YUANHUADINE	chembl:CHEMBL1911631	YUANHUADINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010629083	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	PYRANTEL PAMOATE	rxcui:8985	PYRANTEL PAMOATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009875432	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	HOE-33342	chembl:CHEMBL343002	CHEMBL:CHEMBL343002	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.058602312	FRENTIZOLE	ncit:C167023	FRENTIZOLE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	PYRILAMINE	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	9-NITRO-ANTHRACENE	chembl:CHEMBL166112	CHEMBL:CHEMBL166112	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.012040282	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.7395446652914718	U-69593	iuphar.ligand:1655	U69593	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.031555091	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009630901	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	2-AMINOANTHRACENE	chembl:CHEMBL83154	2-AMINOANTHRACENE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	3',4'-DIMETHOXYFLAVONE	chembl:CHEMBL91153	3',4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.006233104	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	(R)-FLECAINIDE	chembl:CHEMBL398673	(R)-FLECAINIDE	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.217423069	SULFOBROMOPHTHALEIN	rxcui:10212	SULFOBROMOPHTHALEIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.019418517	MOMELOTINIB	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.039361073	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.050294704	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
GRM4	hgnc:4596	GRM4	DTC	9/2/20	NULL	7.501095891	N-(3-(TRIFLUOROMETHYL)PHENYL)PICOLINAMIDE	chembl:CHEMBL571453	CHEMBL:CHEMBL571453	FALSE	FALSE	FALSE
CCR1	hgnc:1602	CCR1	DTC	9/2/20	NULL	11.66837138570988	4'-CHLORO-[2,2'6',2']TERPYRIDINE	chembl:CHEMBL2205805	CHEMBL:CHEMBL2205805	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.010348378	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
PDK1	hgnc:8809	PDK1	DTC	9/2/20	NULL	3.750547945	N-ACETYLGLUCOSAMINE THIAZOLINE	chembl:CHEMBL257158	CHEMBL:CHEMBL257158	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	NALOXONE BENZOYLHYDRAZONE	iuphar.ligand:1664	NALOXONE BENZOYLHYDRAZONE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.026748686	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	STANOLONE	ncit:C72098	STANOLONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.3500511415712966	ISOQUERCETIN	ncit:C117288	ISOQUERCETIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	MMV666022	chembl:CHEMBL599100	CHEMBL:CHEMBL599100	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013825085	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.015744429	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	SJ000157363	chembl:CHEMBL590947	CHEMBL:CHEMBL590947	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665927	chembl:CHEMBL531611	CHEMBL:CHEMBL531611	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	1.050153425	SJ000174085	chembl:CHEMBL592842	CHEMBL:CHEMBL592842	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	SJ000147993	chembl:CHEMBL601618	CHEMBL:CHEMBL601618	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003622218	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.07699072	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.060492709	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
CAMK1D	hgnc:19341	CAMK1D	DTC	9/2/20	NULL	0.1075976869583903	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.017092341	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	SULFOBROMOPHTHALEIN	rxcui:10212	SULFOBROMOPHTHALEIN	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.022949157	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.033148782	LEFLUNOMIDE	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
AKT2	hgnc:392	AKT2	DTC	9/2/20	NULL	0.031880796	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.034773292	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.073437302	PARAROSANILINE	chembl:CHEMBL1368322	PARAROSANILINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	FRENTIZOLE	ncit:C167023	FRENTIZOLE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	DNDI1417973	chembl:CHEMBL1572415	CHEMBL:CHEMBL1572415	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	SB-228357	iuphar.ligand:192	SB 228357	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.2019525816757481	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	GUANFACINE HYDROCHLORIDE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	NSC-601359	chembl:CHEMBL1306524	CHEMBL:CHEMBL1306524	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011205222	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	METILDIGOXIN	ncit:C170170	METILDIGOXIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	AM-281	iuphar.ligand:741	AM281	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.00661639	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.020002922	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004972317	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005363398	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
HEXB	hgnc:4879	HEXB	DTC	9/2/20	NULL	2.625383561784724	N-ACETYLGLUCOSAMINE THIAZOLINE	chembl:CHEMBL257158	CHEMBL:CHEMBL257158	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.5834185692854944	R(+)-BUTYLINDAZONE	chembl:CHEMBL1256719	CHEMBL:CHEMBL1256719	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	LAWSONE	drugbank:DB04744	LAWSONE	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.029833904	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003806559	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	BUTACHLOR	chembl:CHEMBL1399036	BUTACHLOR	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.075010959	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.5073204950308646	SILYDIANIN	chembl:CHEMBL2397733	SILIDIANIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	SODIUM LAURYL SULFATE	rxcui:9871	SODIUM DODECYL SULFATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005899738	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1325951293830669	1-O-ACETYLGEOPYXIN A	chembl:CHEMBL1902074	CHEMBL:CHEMBL1902074	FALSE	FALSE	FALSE
SLC29A2	hgnc:11004	SLC29A2	DTC	9/2/20	NULL	7.001022831425932	TECADENOSON	ncit:C77980	TECADENOSON	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	TERCONAZOLE	rxcui:37806	TERCONAZOLE	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.008789366	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.9907107780319716	TCMDC-124676	chembl:CHEMBL588965	CHEMBL:CHEMBL588965	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
OPN1LW	hgnc:9936	OPN1LW	DTC	9/2/20	NULL	3.000438356325399	RETINAL	iuphar.ligand:2350	ALL-TRANS-RETINAL	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	MMV006513	chembl:CHEMBL585622	CHEMBL:CHEMBL585622	FALSE	FALSE	FALSE
MCOLN3	hgnc:13358	MCOLN3	DTC	9/2/20	NULL	3.281729452230906	GNF-PF-1025	chembl:CHEMBL584031	CHEMBL:CHEMBL584031	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	2-STYRYL-QUINOLINE	chembl:CHEMBL127579	CHEMBL:CHEMBL127579	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DIBROMOACETIC ACID	chembl:CHEMBL449362	DIBROMOACETIC ACID	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	TCMDC-125528	chembl:CHEMBL375673	CHEMBL:CHEMBL375673	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.027811267	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	PHENACYL CHLORIDE	iuphar.ligand:6285	OMEGA-CHLOROACETOPHENONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	CID 926663	chembl:CHEMBL265686	CHEMBL:CHEMBL265686	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	SB-228357	iuphar.ligand:192	SB 228357	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	5-METHOXYFLAVONE	chembl:CHEMBL16685	CHEMBL:CHEMBL16685	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	BISABOLOL	rxcui:19461	BISABOLOL	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.020257589	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	L-655240	chembl:CHEMBL362223	CHEMBL:CHEMBL362223	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.017751072	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	1.166837138570988	ZINC 06638999	chembl:CHEMBL608846	CHEMBL:CHEMBL608846	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.009320613	Aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	0.4734548598913698	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.04427291	Desvenlafaxine	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.8751278539282416	Dolutegravir	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.6019397937072561	Dacomitinib	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	1.050153425	Paritaprevir	rxcui:1597373	PARITAPREVIR	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.027121731	Drospirenone	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.022829422	Erythromycin	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	FDA	10-Apr-24	NULL	0.561579372	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.035418328	Formoterol	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
CPOX	hgnc:2321	CPOX	FDA	10-Apr-24	NULL	35.00511415712966	Givosiran	rxcui:2265712	GIVOSIRAN	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.015875335	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.1131630845596864	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.047734247	Primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.012054103	Ticagrelor	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	FDA	10-Apr-24	NULL	0.042516333	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
IL12B	hgnc:5970	IL12B	FDA	10-Apr-24	NULL	1.125164383622024	Ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	1.657092009619794	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	1.336059069138614	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.6241137025199848	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	2.341819737097098	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	MyCancerGenome	20-Jun-17	inhibitor	0.6482428547616604	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.2778183663264259	PELITINIB	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.1535312024435511	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1512704997187101	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
CD52	hgnc:1804	CD52	MyCancerGenome	20-Jun-17	antibody	70.01022831425932	ALEMTUZUMAB	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.0403388	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	immunotherapy	0.2561349816375342	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	antibody	0.2561349816375342	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	immunotherapy	0.1097721349875146	MK-3475	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	antibody	0.1097721349875146	MK-3475	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	antibody	3.962843112127886	DALOTUZUMAB	rxcui:1432293	DALOTUZUMAB	FALSE	TRUE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	MyCancerGenome	20-Jun-17	other/unknown	0.4280516676822921	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
PSMB6	hgnc:9543	PSMB6	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD8	hgnc:9566	PSMD8	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD1	hgnc:9554	PSMD1	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA8	hgnc:22985	PSMA8	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PIPSL	hgnc:23733	PIPSL	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA5	hgnc:9534	PSMA5	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA6	hgnc:9535	PSMA6	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB4	hgnc:9541	PSMB4	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB10	hgnc:9538	PSMB10	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB9	hgnc:9546	PSMB9	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1190650141398968	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PSME4	hgnc:20635	PSME4	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.678633990910949	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
MAPK11	hgnc:6873	MAPK11	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1446492320542548	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
ABL	hgnc:76	ABL1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.022894123	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	activator	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.067231333	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2243917574174978	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3241214273808303	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.069454592	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.089756703	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
TEK	hgnc:11724	TEK	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3977853881492008	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
EPHA2	hgnc:3386	EPHA2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1767935058440892	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
AKT2	hgnc:392	AKT2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.6482428547616604	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.043768551	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.4487835148349957	VINCA ALKALOIDS	ncit:C932	VINCA ALKALOID COMPOUND	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.059364241	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	0.3763990769583835	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1565057264849314	PROBENECID	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
ACTB	hgnc:132	ACTB	NCI	14-Sep-17	NULL	0.150021918	ETHINYLESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	NCI	14-Sep-17	NULL	0.068458502	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.018426977	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
ACP5	hgnc:124	ACP5	NCI	14-Sep-17	NULL	1.009762908	M-CSF	iuphar.ligand:4905	M-CSF	FALSE	FALSE	FALSE
ACTR2	hgnc:169	ACTR2	NCI	14-Sep-17	NULL	0.8899605294185507	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ADCYAP1	hgnc:241	ADCYAP1	NCI	14-Sep-17	NULL	2.187819634820604	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.4150804050252529	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.8078103267029924	POLYETHYLENE GLYCOL	rxcui:1310594	POLYETHYLENE GLYCOL 4000	TRUE	FALSE	FALSE
ASNS	hgnc:753	ASNS	NCI	14-Sep-17	NULL	14.58546423213736	L-ASPARAGINASE	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.2000292237550266	IL-4	iuphar.ligand:4996	IL-4	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.038894571	ERBITUX	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.023732281	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.053854022	VINORELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.2800409132570373	PROTEIN PHOSPHATASE INHIBITOR	ncit:C2159	PROTEIN PHOSPHATASE INHIBITOR	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.051226996	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1829535583125243	C5A	iuphar.ligand:3576	C5A	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1164249916534246	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.3201687270469177	LIPOSOMAL DOXORUBICIN	wikidata:Q29004943	CAELYX	FALSE	FALSE	TRUE
CCL11	hgnc:10610	CCL11	NCI	14-Sep-17	NULL	0.6731752722524936	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	13.12691780892362	CXC CHEMOKINES	ncit:C1592	RECOMBINANT ALPHA CHEMOKINE	FALSE	FALSE	FALSE
CCL7	hgnc:10634	CCL7	NCI	14-Sep-17	NULL	2.692701089009974	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.072125922	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
CCNA2	hgnc:1578	CCNA2	NCI	14-Sep-17	NULL	0.2263261691193728	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CD4	hgnc:1678	CD4	NCI	14-Sep-17	NULL	0.7292732116068681	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
CD163	hgnc:1631	CD163	NCI	14-Sep-17	NULL	1.544343271638073	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.06584034	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	0.1426838892274307	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CD52	hgnc:1804	CD52	NCI	14-Sep-17	NULL	70.01022831425932	CAMPATH	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
CD69	hgnc:1694	CD69	NCI	14-Sep-17	NULL	8.751278539282415	ANTITUMOR ANTIBIOTICS	ncit:C259	ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	2.442217266776488	INTERLEUKIN-16	ncit:C1147	RECOMBINANT INTERLEUKIN-16	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	NCI	14-Sep-17	NULL	0.192335792	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.2727671233023091	PROTEIN PHOSPHATASE INHIBITOR	ncit:C2159	PROTEIN PHOSPHATASE INHIBITOR	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	NCI	14-Sep-17	NULL	0.078722146	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.3535870116881784	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.053199262	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.3500511415712966	DDTC	ncit:C432	DITIOCARB	FALSE	FALSE	FALSE
CPD	hgnc:2301	CPD	NCI	14-Sep-17	NULL	0.272767123	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.2333674277141977	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.03043923	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.085937269	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	3.500511415712966	RETRO-INVERSO PEPTIDE	ncit:C1963	RETRO-INVERSO PEPTIDE	FALSE	FALSE	FALSE
CSPG4	hgnc:2466	CSPG4	NCI	14-Sep-17	NULL	1.050153425	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	0.4375639269641209	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.7501095890813501	BENZODIAZEPINE	ncit:C1012	BENZODIAZEPINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.00213576	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.003849818	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	0.069638821	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.057574201	URACIL	rxcui:10995	URACIL	TRUE	FALSE	TRUE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.84146909	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.175610941	PROSTAGLANDIN E1	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.1842374429322614	SOMATOTROPIN	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	NCI	14-Sep-17	NULL	0.2983390411119005	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.076263865	SU5416	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.1105424657593568	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
GADD45A	hgnc:4095	GADD45A	NCI	14-Sep-17	NULL	0.5770073762164232	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
GADD45A	hgnc:4095	GADD45A	NCI	14-Sep-17	NULL	0.258658479	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
GABPA	hgnc:4071	GABPA	NCI	14-Sep-17	NULL	0.1166837138570988	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.1166837138570989	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.055271233	BUSULFAN	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
GAL	hgnc:4114	GAL	NCI	14-Sep-17	NULL	0.3125456621172291	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
GALP	hgnc:24840	GALP	NCI	14-Sep-17	NULL	1.141471113819445	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	2.386712328895204	L-BUTHIONINE SULFOXIMINE	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.8334550989792776	SORBITOL	rxcui:9945	SORBITOL	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.047304208	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
GZMA	hgnc:4708	GZMA	NCI	14-Sep-17	NULL	1.666910197958555	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
GTF2B	hgnc:4648	GTF2B	NCI	14-Sep-17	NULL	3.029288725136221	VITAMIN D	rxcui:11253	VITAMIN D	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	NCI	14-Sep-17	NULL	0.3409589041278864	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	NCI	14-Sep-17	NULL	0.09876051	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.9546849315580819	ESTRAMUSTINE	rxcui:4089	ESTRAMUSTINE	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.079376676	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	1.093909817410302	ALPHA INTERFERON	ncit:C225	RECOMBINANT INTERFERON ALFA	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	NCI	14-Sep-17	NULL	0.1771513874348667	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
HMOX1	hgnc:5013	HMOX1	NCI	14-Sep-17	NULL	0.2651902587661338	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.040640612	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	MITOTANE	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	NCI	14-Sep-17	NULL	0.015123177	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.065799087	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.09869863	ADENOVIRAL VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.036451004	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1744440904840348	IFOSFAMIDE	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
HSPA8	hgnc:5241	HSPA8	NCI	14-Sep-17	NULL	0.075442056	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.1369170045259309	VP-16	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
HSPD1	hgnc:5261	HSPD1	NCI	14-Sep-17	NULL	0.6364566210387212	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.4688184931758437	DHPG	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1861974157294131	U-37883A	iuphar.ligand:13269	PNU-37883	FALSE	FALSE	FALSE
ICAM2	hgnc:5345	ICAM2	NCI	14-Sep-17	NULL	2.692701089009974	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	1.363835616511545	DIETHYLDITHIOCARBAMATE	rxcui:1427193	DIETHYLDITHIOCARBAMATE	FALSE	FALSE	FALSE
IBSP	hgnc:5341	IBSP	NCI	14-Sep-17	NULL	0.2414145803939976	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
IFIT2	hgnc:5409	IFIT2	NCI	14-Sep-17	NULL	2.692701089009974	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.2753898841032928	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.2083637747448194	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.087222045	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	NCI	14-Sep-17	NULL	0.1238388472539964	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.2206204673768676	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.106290832	AZA	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
AKR1C3	hgnc:386	AKR1C3	DTC	9/2/20	NULL	7.001022831425932	BACCHARIN	chembl:CHEMBL428354	BACCHARIN	FALSE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	NCI	14-Sep-17	NULL	3.750547945	ALUM	rxcui:221456	ALUM, POTASSIUM	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1029562181092049	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.2381300282797936	VITAMIN K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
LOH19CR1	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.092851762	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.117598368	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.2302968036653267	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.1256164383629055	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.2083637747448194	L-ASPARAGINASE	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.6250913242344582	DEXTRAN SULFATE	rxcui:40068	DEXTRAN SULFATE	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.067317527	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.027177884	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.2201579506737715	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.7071740233763569	METHYLNITROSOUREA	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.7071740233763569	MNU	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	3-(N-PHENETHYLSULFAMOYL)BENZOIC ACID	chembl:CHEMBL1871992	CHEMBL:CHEMBL1871992	FALSE	FALSE	FALSE
MSR1	hgnc:7376	MSR1	NCI	14-Sep-17	NULL	4.039051633514962	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
MTR	hgnc:7468	MTR	NCI	14-Sep-17	NULL	1.093909817410302	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
MUC5AC	hgnc:7515	MUC5AC	NCI	14-Sep-17	NULL	0.7721716358190368	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	1.458546423213736	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	GNF-PF-4576	chembl:CHEMBL527336	CHEMBL:CHEMBL527336	FALSE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.3125456621172291	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1000146118775133	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.062509132	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.9723642821424908	PTHRP	iuphar.ligand:3738	PTHRP	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.043756393	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCF1	hgnc:7660	NCF1	NCI	14-Sep-17	NULL	5.250767124	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2958178661165888	NEUROTROPHIC FACTOR	ncit:C2259	RECOMBINANT NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.060388351	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2105359712738352	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
NR6A1	hgnc:7985	NR6A1	NCI	14-Sep-17	NULL	4.500657534	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.1562728310586145	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	2.187819634820604	BRAIN-DERIVED NEUROTROPHIC FACTOR	rxcui:47324	BRAIN-DERIVED NEUROTROPHIC FACTOR	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.080471527	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.3671865121377238	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.026640117	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.2019525816757481	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	NCI	14-Sep-17	NULL	0.3125456621172291	DIETHYLDITHIOCARBAMATE	rxcui:1427193	DIETHYLDITHIOCARBAMATE	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.042310775	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.1389091831632129	INDOLE-3-CARBINOL	rxcui:2598119	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.092606122	SERM	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.023813003	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2083637747448194	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
PLAUR	hgnc:9053	PLAUR	NCI	14-Sep-17	NULL	0.9376369863516874	ADENOVIRAL VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.059532507	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.054355767	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	0.071341945	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.038382801	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1988926940746004	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.050294704	MONOAMINE OXIDASE INHIBITOR	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.025147352	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.069454592	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	NCI	14-Sep-17	NULL	1.500219178	INTERLEUKIN-4	rxcui:1426682	BINETRAKIN	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.1241316104862754	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
SCG5	hgnc:10816	SCG5	NCI	14-Sep-17	NULL	2.059124362184098	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.1930429089547591	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
S100B	hgnc:10500	S100B	NCI	14-Sep-17	NULL	1.141471113819445	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.16256245	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
SLAMF6	hgnc:21392	SLAMF6	NCI	14-Sep-17	NULL	21.00306849	INTERLEUKIN-4	rxcui:1426682	BINETRAKIN	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	NCI	14-Sep-17	NULL	0.045639002	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PYRIPROXYFEN	chembl:CHEMBL1883234	PYRIPROXYFEN	FALSE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.1135300999690691	FOLINIC ACID	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
TACR1	hgnc:11526	TACR1	NCI	14-Sep-17	NULL	0.1091635576625665	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
TBXA2R	hgnc:11608	TBXA2R	NCI	14-Sep-17	NULL	0.086219493	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
TDO2	hgnc:11708	TDO2	NCI	14-Sep-17	NULL	1.050153425	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.078781202	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.029665351	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.1077080435603989	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.025663573	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.024547766	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.056459862	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.1508841127462485	ANTHRACYCLINE	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
TNFSF13B	hgnc:11929	TNFSF13B	NCI	14-Sep-17	NULL	0.2224901323546377	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TNFRSF10A	hgnc:11904	TNFRSF10A	NCI	14-Sep-17	NULL	1.000146118775133	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
TNFRSF11B	hgnc:11909	TNFRSF11B	NCI	14-Sep-17	NULL	0.375054795	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.011591097	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.04636439	DNA VACCINE	ncit:C39619	DNA VACCINE	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	2.234368988752957	9-AC	ncit:C1488	AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.837888371	DOXIFLURIDINE	ncit:C978	DOXIFLURIDINE	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.049107011	DAUNOMYCIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.502465753	ORAL CONTRACEPTIVE	ncit:C389	ORAL CONTRACEPTIVE	FALSE	FALSE	FALSE
TSPYL2	hgnc:24358	TSPYL2	NCI	14-Sep-17	NULL	1.250182648468916	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.085937269	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
UCP1	hgnc:12517	UCP1	NCI	14-Sep-17	NULL	0.760980743	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	NCI	14-Sep-17	NULL	0.093680056	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
UGT1A5	hgnc:12537	UGT1A5	NCI	14-Sep-17	NULL	0.1842374429322614	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	LUZINDOLE	iuphar.ligand:1363	LUZINDOLE	FALSE	FALSE	FALSE
VCAM1	hgnc:12663	VCAM1	NCI	14-Sep-17	NULL	1.166837138570988	PHORBOL MYRISTATE ACETATE	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.022296251	CASODEX	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
VCAM1	hgnc:12663	VCAM1	NCI	14-Sep-17	NULL	0.6731752722524936	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.015201989	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.002752624	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
VIPR1	hgnc:12694	VIPR1	NCI	14-Sep-17	NULL	1.750255707856483	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	2.407466349146467	brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.03140411	ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
ST13	hgnc:11343	ST13	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	NORELGESTROMIN	rxcui:326374	NORELGESTROMIN	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.4145342465975881	margetuximab	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.024674658	capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.3677319929494733	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.091159151	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
B4GALT2	hgnc:925	B4GALT2	PharmGKB	4/5/24	NULL	3.000438356	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.086861325	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.100589408	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.03319069	cefaclor	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.01290749	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.008297672	nifedipine	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.018006746	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.7160136986685613	etodolac	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
EPHA5	hgnc:3389	EPHA5	PharmGKB	4/5/24	NULL	0.5834185692854945	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FGD4	hgnc:19125	FGD4	PharmGKB	4/5/24	NULL	0.9723642821424907	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
KCNE1	hgnc:6240	KCNE1	PharmGKB	4/5/24	NULL	1.125164383622024	quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.085378327	Analgesics	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	PharmGKB	4/5/24	NULL	0.016501468	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1693795846312726	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.1013661606866689	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
TSPYL1	hgnc:12382	TSPYL1	PharmGKB	4/5/24	NULL	1.875273972703374	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.077827576	cabergoline	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.3938075342677087	mafenide	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.022410444	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.3697723326457359	capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
ABCG1	hgnc:73	ABCG1	PharmGKB	4/5/24	NULL	0.8334550989792776	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	PharmGKB	4/5/24	NULL	0.5672124979164529	midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NPM1	hgnc:7910	NPM1	PharmGKB	4/5/24	NULL	0.4167275494896389	midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.039763477	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.019318496	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	2.500365296937833	nefazodone	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
CRH	hgnc:2355	CRH	PharmGKB	4/5/24	NULL	0.2524407270946851	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	HARMINE HYDROCHLORIDE	chembl:CHEMBL1593867	HARMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ANKK1	hgnc:21027	ANKK1	PharmGKB	4/5/24	NULL	7.501095891	nemonapride	ncit:C73036	NEMONAPRIDE	FALSE	FALSE	FALSE
ANKK1	hgnc:21027	ANKK1	PharmGKB	4/5/24	NULL	0.3488881809680698	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
STX1B	hgnc:18539	STX1B	PharmGKB	4/5/24	NULL	6.364566210387212	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	0.082300425	genistein	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	1.250182648468916	inotuzumab ozogamicin	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.014504882	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
PRPF31	hgnc:15446	PRPF31	PharmGKB	4/5/24	NULL	2.692701089009974	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
UMPS	hgnc:12563	UMPS	PharmGKB	4/5/24	NULL	1.419126249613364	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
GGH	hgnc:4248	GGH	PharmGKB	4/5/24	NULL	2.100306849	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	0.150021918	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.019079822	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.023110771	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.022225469	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
SULT1E1	hgnc:11377	SULT1E1	PharmGKB	4/5/24	NULL	3.029288725136221	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	PharmGKB	4/5/24	NULL	0.1715936968486748	sacituzumab govitecan-hziy	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.2500365296937833	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-4576	chembl:CHEMBL527336	CHEMBL:CHEMBL527336	FALSE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	0.1093909817410302	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	0.1715936968486748	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
DVL2	hgnc:3086	DVL2	PharmGKB	4/5/24	NULL	0.3860858179095184	gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
HMMR	hgnc:5012	HMMR	PharmGKB	4/5/24	NULL	0.7292732116068681	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.089501712	quinidine	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.5000730593875667	homoharringtonine	rxcui:27100	OMACETAXINE MEPESUCCINATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.1511012121890489	homoharringtonine	rxcui:27100	OMACETAXINE MEPESUCCINATE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	PharmGKB	4/5/24	NULL	0.03409589	topiramate	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UGT1A	hgnc:12529	UGT1A	PharmGKB	4/5/24	NULL	5.250767124	bilirubin	iuphar.ligand:4577	BILIRUBIN	FALSE	FALSE	FALSE
CD44	hgnc:1681	CD44	PharmGKB	4/5/24	NULL	0.106290832	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.1389091831632129	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.2169738480813822	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	PharmGKB	4/5/24	NULL	0.2019525816757481	perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.064268875	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
ASS1	hgnc:758	ASS1	PharmGKB	4/5/24	NULL	0.3125456621172291	glycerol phenylbutyrate	rxcui:1368451	GLYCEROL PHENYLBUTYRATE	TRUE	FALSE	FALSE
MCPH1	hgnc:6954	MCPH1	PharmGKB	4/5/24	NULL	4.039051633514962	perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.5527123287967842	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.8751278539282416	paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.9546849315580818	omega-3 polyunsaturated fatty acids	rxcui:4301	OMEGA-3 FATTY ACIDS	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.041805471	deferasirox	rxcui:614373	DEFERASIROX	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.005716987	interferons	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.002447226	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.2540693769469088	panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.018071819	toremifene	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.0017798	triazolam	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
MIR6076	hgnc:50232	MIR6076	PharmGKB	4/5/24	NULL	0.6482428547616604	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
FGF14	hgnc:3671	FGF14	PharmGKB	4/5/24	NULL	0.9376369863516874	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	DITHIAZANINE	ncit:C72743	DITHIAZANINE	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	PharmGKB	4/5/24	NULL	0.9616789603607051	metyrosine	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
ABCC10	hgnc:52	ABCC10	PharmGKB	4/5/24	NULL	0.108040476	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.4070362111294147	fenoterol	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.046303061	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	PharmGKB	4/5/24	NULL	0.076709527	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
SLC10A2	hgnc:10906	SLC10A2	PharmGKB	4/5/24	NULL	0.218327115	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
N6AMT1	hgnc:16021	N6AMT1	PharmGKB	4/5/24	NULL	4.500657534	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
C8ORF34	hgnc:30905	C8orf34	PharmGKB	4/5/24	NULL	1.666910197958555	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SOCS3	hgnc:19391	SOCS3	PharmGKB	4/5/24	NULL	0.9053046764774914	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1136529680426287	methimazole	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
CSPG4	hgnc:2466	CSPG4	PharmGKB	4/5/24	NULL	0.5250767123569451	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
FMO2	hgnc:3770	FMO2	PharmGKB	4/5/24	NULL	0.5303805175322677	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
PLCG1	hgnc:9065	PLCG1	PharmGKB	4/5/24	NULL	0.3365876361262468	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
FTCDNL1	hgnc:48661	FTCDNL1	PharmGKB	4/5/24	NULL	0.9376369863516874	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.083717588	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NFATC1	hgnc:7775	NFATC1	PharmGKB	4/5/24	NULL	0.2344092465879218	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
FOXO1	hgnc:3819	FOXO1	PharmGKB	4/5/24	NULL	0.5834185692854945	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.921187215	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.046089683	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.561579372	durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
C20ORF194	hgnc:17721	DNAAF9	PharmGKB	4/5/24	NULL	1.207072901969988	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.017599354	mibefradil	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	AG1295	iuphar.ligand:5914	AG 1295	FALSE	FALSE	TRUE
APC	hgnc:583	APC	PharmGKB	4/5/24	NULL	0.2557191780959147	nirogacestat	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
CXCL8	hgnc:6025	CXCL8	PharmGKB	4/5/24	NULL	0.048618214	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
WDR24	hgnc:20852	WDR24	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.015153729	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.002683207	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.01293611	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	0.2273059360852576	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	PharmGKB	4/5/24	NULL	0.1973972602845657	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	0.2273059360852576	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.056826484	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	PharmGKB	4/5/24	NULL	0.4167275494896388	leniolisib	rxcui:2633005	LENIOLISIB	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	PharmGKB	4/5/24	NULL	0.054695491	panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
ERBB4	hgnc:3432	ERBB4	PharmGKB	4/5/24	NULL	0.1508841127462485	paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
SLC22A2	hgnc:10966	SLC22A2	PharmGKB	4/5/24	NULL	3.281729452230906	l-tryptophan	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	PharmGKB	4/5/24	NULL	0.1752202599633854	lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
PRKAG2	hgnc:9386	PRKAG2	PharmGKB	4/5/24	NULL	1.346350544504987	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
IMPDH2	hgnc:6053	IMPDH2	PharmGKB	4/5/24	NULL	0.4224755156894959	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UMOD	hgnc:12559	UMOD	PharmGKB	4/5/24	NULL	0.4023576339899961	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1166837138570989	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
IL1RN	hgnc:6000	IL1RN	PharmGKB	4/5/24	NULL	0.8204323630577265	heparin	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.080471527	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CYP3A7	hgnc:2640	CYP3A7	PharmGKB	4/5/24	NULL	0.086219493	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.059364241	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
AADAC	hgnc:17	AADAC	PharmGKB	4/5/24	NULL	0.091796628	eslicarbazepine acetate	rxcui:1482501	ESLICARBAZEPINE ACETATE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW711782X	chembl:CHEMBL208437	GW711782X	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	PharmGKB	4/5/24	NULL	0.039479452	polatuzumab vedotin	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
APOA5	hgnc:17288	APOA5	PharmGKB	4/5/24	NULL	0.8751278539282416	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	PharmGKB	4/5/24	NULL	0.045461187	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
ASPH	hgnc:757	ASPH	PharmGKB	4/5/24	NULL	0.151537291	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	PharmGKB	4/5/24	NULL	0.058341857	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
CCT3	hgnc:1616	CCT3	PharmGKB	4/5/24	NULL	1.312691780892362	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	0.2885036881082116	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.2966535098061835	acetylcholine	rxcui:194	ACETYLCHOLINE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.4000584475100533	pramipexole	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.2972132334095915	desflurane	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.4375639269641208	dextropropoxyphene	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.03729238	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.2243917574174978	rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	0.1478048451391822	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
NOX3	hgnc:7890	NOX3	PharmGKB	4/5/24	NULL	1.666910197958555	methimazole	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
CPS1	hgnc:2323	CPS1	PharmGKB	4/5/24	NULL	1.000146118775133	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	PharmGKB	4/5/24	NULL	0.051782713	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
ALDH2	hgnc:404	ALDH2	PharmGKB	4/5/24	NULL	0.2853677784548614	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.5707355569097228	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
FGA	hgnc:3661	FGA	PharmGKB	4/5/24	NULL	1.909369863116163	tirofiban	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
FDPS	hgnc:3631	FDPS	TALC	12-May-16	NULL	1.633571993999384	ZOLEDRONATE	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.078136416	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	TALC	12-May-16	inhibitor	1.521961485092594	ASP3026	ncit:C116727	ALK INHIBITOR ASP3026	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.078136416	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	TALC	12-May-16	inhibitor	0.008240375	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	inhibitor	0.069089041	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.1458546423213736	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
KIF11	hgnc:6388	KIF11	TALC	12-May-16	inhibitor	6.563458904461812	ARQ-621	chembl:CHEMBL4303449	ARQ-621	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.2857560339357523	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.1205533268166455	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	TALC	12-May-16	inhibitor	0.089046362	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	TALC	12-May-16	inhibitor	0.2083637747448194	BI-2536	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.1350505947420126	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
BCR	hgnc:1014	BCR	TALC	12-May-16	inhibitor	0.4000584475100533	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
RRM2	hgnc:10452	RRM2	TALC	12-May-16	inhibitor	3.029288725136221	TRIAPINE	ncit:C2242	TRIAPINE	FALSE	FALSE	TRUE
XIAP	hgnc:592	XIAP	TALC	12-May-16	inhibitor	0.1190650141398968	LCL161	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	TALC	12-May-16	inhibitor	1.282909942931453	LGX818	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	TALC	12-May-16	inhibitor	0.012534655	AS703569	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	TALC	12-May-16	inhibitor	2.407466349146467	AP26113	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.2778183663264259	PELITINIB	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	A-007	ncit:C61305	SIVIFENE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.060772768	ON01910	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
UNIPROT:P41594	hgnc:4597	GRM5	TdgClinicalTrial	Jan-14	NULL	0.1166837138570988	ACAMPROSATE	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.041021618	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:Q8NER1	hgnc:12716	TRPV1	TdgClinicalTrial	Jan-14	NULL	0.301335273	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.048172175	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
UNIPROT:P08253	hgnc:7166	MMP2	TdgClinicalTrial	Jan-14	NULL	0.4487835148349957	AE-941	ncit:C1798	SHARK CARTILAGE EXTRACT AE-941	FALSE	FALSE	FALSE
UNIPROT:Q06643	hgnc:6711	LTB	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	BAMINERCEPT	ncit:C96762	BAMINERCEPT ALFA	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.066803653	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
UNIPROT:P29459	hgnc:5969	IL12A	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	BRIAKINUMAB	ncit:C95321	BRIAKINUMAB	FALSE	FALSE	FALSE
UNIPROT:P24723	hgnc:9403	PRKCH	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:P05771	hgnc:9395	PRKCB	TdgClinicalTrial	Jan-14	NULL	0.2344092465879218	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.1233298208706858	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.3256289689035318	FORMOTEROL	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P21730	hgnc:1338	C5AR1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	CCX168	iuphar.ligand:9450	AVACOPAN	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.033701971	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.192335792	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.5173169579871378	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	0.1030370314672184	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.032899543	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.1136529680426287	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	3.750547945	DESMOTEPLASE	ncit:C87246	DESMOTEPLASE	TRUE	FALSE	FALSE
UNIPROT:Q14957	hgnc:4587	GRIN2C	TdgClinicalTrial	Jan-14	NULL	0.1058622403945453	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
UNIPROT:Q8IWT1	hgnc:10592	SCN4B	TdgClinicalTrial	Jan-14	NULL	2.100306849	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.7778914257139925	RONOMILAST	ncit:C97274	RONOMILAST	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.053361455	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.028898003	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.054355767	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.02926849	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.05073205	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.051885051	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	DNDI1417006	chembl:CHEMBL1415258	CHEMBL:CHEMBL1415258	FALSE	FALSE	FALSE
UNIPROT:P08473	hgnc:7154	MME	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	ILEPATRIL	ncit:C87731	ILEPATRIL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001498507	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
UNIPROT:P15382	hgnc:6240	KCNE1	TdgClinicalTrial	Jan-14	NULL	0.1875273972703375	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
UNIPROT:Q53ET0	hgnc:27301	CRTC2	TdgClinicalTrial	Jan-14	NULL	0.5966780822238011	INK128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.059297201	ITI-007	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.1620607136904151	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P35228	hgnc:7873	NOS2	TdgClinicalTrial	Jan-14	NULL	2.838252499226729	KD7040	drugbank:DB05214	KD7040	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.3860858179095183	LORCASERIN	rxcui:1300701	LORCASERIN	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.040893825	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.2678962818147678	LOFEXIDINE	rxcui:28863	LOFEXIDINE	TRUE	FALSE	FALSE
UNIPROT:P08183	hgnc:40	ABCB1	TdgClinicalTrial	Jan-14	NULL	0.1121958787087489	LIM-0705	chembl:CHEMBL4297397	QUERCETIN-3'-O-PHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:P42336	hgnc:8975	PIK3CA	TdgClinicalTrial	Jan-14	NULL	0.060772768	RIGOSERTIB	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.089756703	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
UNIPROT:Q04721	hgnc:7882	NOTCH2	TdgClinicalTrial	Jan-14	NULL	15.00219178	OMP-59R5	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.1643432589536604	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
UNIPROT:P20618	hgnc:9537	PSMB1	TdgClinicalTrial	Jan-14	NULL	0.384671584	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.3040984820600068	OPC-34712	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q13200	hgnc:9559	PSMD2	TdgClinicalTrial	Jan-14	NULL	0.5385402178019948	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	0.9907107780319716	OSI-906	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.062733179	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.063110182	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.093098708	INDACATEROL	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.2237542808339254	RANOLAZINE	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	RECOMBINANT HUMAN CHORIONIC GONADOTROPIN	ncit:C528	RECOMBINANT HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.4145342465975881	ROPIVACAINE	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
UNIPROT:P50613	hgnc:1778	CDK7	TdgClinicalTrial	Jan-14	NULL	0.6000876712650799	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
UNIPROT:P16109	hgnc:10721	SELP	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	SELG1	rxcui:2262279	CRIZANLIZUMAB	TRUE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.052090944	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
UNIPROT:P63241	hgnc:3300	EIF5A	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	SNS01-T	drugbank:DB17302	SNS01-T	FALSE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	0.5097832158805291	SOBETIROME	ncit:C81539	SOBETIROME	FALSE	FALSE	FALSE
UNIPROT:P13639	hgnc:3214	EEF2	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	SS1(DSFV)-PE38	drugbank:DB17579	SS1(DSFV)-PE38	FALSE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.4906052389860809	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.1205533268166455	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1605739181519709	TAPENTADOL	rxcui:787390	TAPENTADOL	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	TAMSULOSIN	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.9512259281828714	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.1620607136904151	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.5073204950308647	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.2365210416022274	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
UNIPROT:P18031	hgnc:9642	PTPN1	TdgClinicalTrial	Jan-14	NULL	2.100306849	TRODUSQUEMINE	ncit:C123882	TRODUSQUEMINE	FALSE	FALSE	FALSE
UNIPROT:P29466	hgnc:1499	CASP1	TdgClinicalTrial	Jan-14	NULL	2.019525817	VX-765	drugbank:DB05507	VX-765	FALSE	FALSE	FALSE
UNIPROT:O14965	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.060956201	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	XL019	drugbank:DB05243	XL019	FALSE	FALSE	FALSE
UNIPROT:P01730	hgnc:1678	CD4	TdgClinicalTrial	Jan-14	NULL	9.845188356692718	ZANOLIMUMAB	ncit:C91701	ZANOLIMUMAB	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	YKP-1358	drugbank:DB06109	YKP-1358	FALSE	FALSE	FALSE
UNIPROT:P06454	hgnc:9623	PTMA	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	THYMALFASIN	rxcui:38221	THYMALFASIN	TRUE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TdgClinicalTrial	Jan-14	NULL	1.325951293830669	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
UNIPROT:P18405	hgnc:11284	SRD5A1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.2075402025126264	YKP-1358	drugbank:DB06109	YKP-1358	FALSE	FALSE	FALSE
UNIPROT:P52333	hgnc:6193	JAK3	TdgClinicalTrial	Jan-14	NULL	0.7134194461371536	ASP015K	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TdgClinicalTrial	Jan-14	NULL	1.633571993999384	ZOLEDRONATE	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.047886613	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.079197091	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.075333818	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	BENDROFLUMETHIAZIDE	rxcui:1369	BENDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:Q14432	hgnc:8778	PDE3A	TdgClinicalTrial	Jan-14	NULL	0.251232877	AMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.07939668	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.1526385791735305	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.070197421	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.073540156	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.075333818	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.068637479	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1962903597596056	CHLOROTRIANISENE	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.067883221	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	PHENPROCOUMON	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.736088849	PHENMETRAZINE	rxcui:8133	PHENMETRAZINE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.053579256	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.1304538415793652	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.063839114	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.050007306	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.051143836	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1875273972703375	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.2019525816757481	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.1154014752432846	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.100976291	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.091556532	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P04070	hgnc:9451	PROC	TdgClinicalTrial	Jan-14	NULL	15.75230137070834	SODIUM TETRADECYL SULFATE	rxcui:9913	SODIUM TETRADECYL SULFATE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TdgClinicalTrial	Jan-14	NULL	0.2027323213733378	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.1117184494376478	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.087512785	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TEND	1-Aug-11	NULL	0.2365210416022275	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
UNIPROT:P00326	hgnc:251	ADH1C	TEND	1-Aug-11	NULL	0.8751278539282417	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.059397818	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TEND	1-Aug-11	NULL	0.2941606231691568	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.058645947	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.2287915957982331	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.4189441853911795	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
UNIPROT:P31358	hgnc:1804	CD52	TEND	1-Aug-11	NULL	70.01022831425932	ALEMTUZUMAB	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.043692674	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.07939668	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.16256245	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.099446347	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.4375639269641208	BROMFENAC	rxcui:19737	BROMFENAC	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.1154649175056503	BUPROPION	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.056500364	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P38435	hgnc:4247	GGCX	TEND	1-Aug-11	NULL	5.250767123569449	ANISINDIONE	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.081830137	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.085147575	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1615620653405984	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O75311	hgnc:4328	GLRA3	TEND	1-Aug-11	NULL	13.12691780892362	PICROTOXIN	rxcui:2539172	PICROTOXIN	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.070010228	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.020494798	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
UNIPROT:Q8TDS4	hgnc:24827	HCAR2	TEND	1-Aug-11	NULL	2.917092846427472	MEPENZOLATE	rxcui:107770	MEPENZOLATE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TEND	1-Aug-11	NULL	3.214755381777214	COAGULATION FACTOR IX	wikidata:Q20801778	COAGULATION FACTOR IX	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.008730906	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TEND	1-Aug-11	NULL	0.445925021	DIHYDROTACHYSTEROL	rxcui:3429	DIHYDROTACHYSTEROL	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TEND	1-Aug-11	NULL	4.375639269641208	INTERFERON ALFACON-1	rxcui:59744	INTERFERON ALFACON-1	TRUE	TRUE	TRUE
UNIPROT:P01178	hgnc:8528	OXT	TEND	1-Aug-11	NULL	1.009762908	OXYTOCIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TEND	1-Aug-11	NULL	2.461297089173179	INTERFERON ALFA-N1	rxcui:202912	INTERFERON ALFA-N1	FALSE	TRUE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.1406455479527531	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.1141471113819445	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P20618	hgnc:9537	PSMB1	TEND	1-Aug-11	NULL	0.5233322714521046	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	LONIDAMINE	ncit:C1146	LONIDAMINE	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.092226589	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.5114383561918295	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TEND	1-Aug-11	NULL	4.039051633514961	NESIRITIDE	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
UNIPROT:P20594	hgnc:7944	NPR2	TEND	1-Aug-11	NULL	4.375639269641208	NESIRITIDE	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.063110182	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TEND	1-Aug-11	NULL	0.9546849315580819	PAMIDRONATE	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	1.790034246671403	BENZONATATE	rxcui:18993	BENZONATATE	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TEND	1-Aug-11	NULL	3.500511415712966	PHENPROCOUMON	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.6105543166941221	PHENYLPROPANOLAMINE	rxcui:8175	PHENYLPROPANOLAMINE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.9376369863516875	PICROTOXIN	rxcui:2539172	PICROTOXIN	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.090634645	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.4000584475100533	PRAMIPEXOLE	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	8.751278539282417	QUINETHAZONE	rxcui:59743	QUINETHAZONE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	28-THIOBETULINIC ACID	chembl:CHEMBL1080077	CHEMBL:CHEMBL1080077	FALSE	FALSE	FALSE
UNIPROT:P08185	hgnc:1540	SERPINA6	TEND	1-Aug-11	NULL	1.312691780892362	RIMEXOLONE	rxcui:55681	RIMEXOLONE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.1154014752432846	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TEND	1-Aug-11	NULL	0.5966780822238011	SILDENAFIL	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.4773424657790409	SALSALATE	rxcui:36108	SALSALATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1117184494376478	SOLIFENACIN	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1605739181519709	TAPENTADOL	rxcui:787390	TAPENTADOL	TRUE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TEND	1-Aug-11	NULL	1.123158743009508	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TEND	1-Aug-11	NULL	1.250182648468916	TESTOLACTONE	rxcui:10378	TESTOLACTONE	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.028626235	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TEND	1-Aug-11	NULL	0.1400204566285186	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P13631	hgnc:9866	RARG	TEND	1-Aug-11	NULL	0.1357664414626878	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
UNIPROT:P51168	hgnc:10600	SCNN1B	TEND	1-Aug-11	NULL	1.823183029	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.4189441853911795	TRIHEXYPHENIDYL	rxcui:10811	TRIHEXYPHENIDYL	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.6819178082557728	TUBOCURARINE	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TEND	1-Aug-11	NULL	0.2019525816757481	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.1654653505326507	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1565523888959287	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.088770366	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	1.250182648468916	Erteberel	ncit:C166610	ERTEBEREL	FALSE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV1.5	hgnc:6224	KCNA5	TTD	2020.06.01	NULL	3.500511415712966	BMS-919373	drugbank:DB15047	BMS-919373	FALSE	FALSE	FALSE
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	3.889457128569962	AMG-181	ncit:C139025	ABRILUMAB	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-2	hgnc:3676	FGF2	TTD	2020.06.01	NULL	0.7095631248066824	FPA144	chembl:CHEMBL4650291	FPA144	FALSE	FALSE	FALSE
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	10.50153424713889	BPX-701	ncit:C128029	PRAME-TARGETING T-CELL RECEPTOR/INDUCIBLE CASPASE 9 BPX-701	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	AMG 420	ncit:C159652	PACANALOTAMAB	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	1.009762908	AMG 820	ncit:C98295	ANTI-C-FMS MONOCLONAL ANTIBODY AMG 820	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	1.944728564284981	XmAb13676	ncit:C130050	PLAMOTAMAB	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR-I	hgnc:5464	IGF1	TTD	2020.06.01	NULL	13.12691780892362	Xentuzumab	ncit:C106118	XENTUZUMAB	FALSE	FALSE	FALSE
SCLEROSTIN	hgnc:13771	SOST	TTD	2020.06.01	NULL	6.563458904461812	BPS-804	iuphar.ligand:9202	BPS-804	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.028444026	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
FIBRONECTIN	hgnc:3778	FN1	TTD	2020.06.01	NULL	4.039051633514961	L19-TNF-alpha	ncit:C166939	ONFEKAFUSP ALFA	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.007250438	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.089756703	PA-799	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	0.6250913242344582	CB-813	chembl:CHEMBL4298072	MARZEPTACOG ALFA (ACTIVATED)	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.3125456621172291	EW-A-401	drugbank:DB05525	EW-A-401	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 1	hgnc:11036	SLC5A1	TTD	2020.06.01	NULL	10.50153424713889	GSK1614235	chembl:CHEMBL4297965	GSK-1614235	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.6019397937072561	Dacomitinib	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1389091831632129	Epidermal growth factor	rxcui:1427158	EPIDERMAL GROWTH FACTOR	FALSE	FALSE	FALSE
ENDOPLASMIN	hgnc:12028	HSP90B1	TTD	2020.06.01	NULL	26.25383561784724	HS-110	ncit:C61073	VIAGENPUMATUCEL-L	FALSE	FALSE	FALSE
NUCLEOLIN	hgnc:7667	NCL	TTD	2020.06.01	NULL	17.50255707856483	IPP-204106	ncit:C103297	NUCLEOLIN ANTAGONIST IPP-204106N	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.3889457128569963	Elpetrigine	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	NKTR-181	ncit:C170277	OXYCODEGOL	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	3.088686543276147	SD-101	ncit:C74084	TLR9 AGONIST SD-101	FALSE	FALSE	FALSE
FREE FATTY ACID RECEPTOR 1	hgnc:4498	FFAR1	TTD	2020.06.01	NULL	7.501095891	LY-2881835	drugbank:DB15046	LY-2881835	FALSE	FALSE	FALSE
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	2.917092846427472	Tabimorelin	ncit:C76887	TABIMORELIN	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	Lepirudin	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	Batabulin	ncit:C72716	BATABULIN	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.016829382	Beta-Lapachone	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.736088849	Phenmetrazine	rxcui:8133	PHENMETRAZINE	TRUE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 2	hgnc:6871	MAPK1	TTD	2020.06.01	NULL	0.020002922	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	2.019525817	Ethinamate	rxcui:24474	ETHINAMATE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4907258993990139	XEN-2174	drugbank:DB05012	XEN-2174	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Lucanthone	ncit:C83925	LUCANTHONE	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.7721716358190367	R-phenserine	chembl:CHEMBL4297417	BUNTANETAP	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	Odiparcil	ncit:C87248	ODIPARCIL	FALSE	FALSE	FALSE
BILE-SALT-ACTIVATED LIPASE	hgnc:1848	CEL	TTD	2020.06.01	NULL	3.750547945	Taurocholic Acid	drugbank:DB04348	TAUROCHOLIC ACID	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	YKP-1358	drugbank:DB06109	YKP-1358	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.5048814541893701	YKP-1358	drugbank:DB06109	YKP-1358	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.089298761	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.116943588	Oxandrolone	rxcui:7779	OXANDROLONE	TRUE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.4730420832044549	Dexefaroxan	ncit:C77943	DEXEFAROXAN	FALSE	FALSE	FALSE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	1.141471113819445	Sivelestat sodium hydrate	chembl:CHEMBL3182314	SIVELESTAT SODIUM	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	DN24-02	ncit:C2057	LAPULEUCEL-T	FALSE	FALSE	FALSE
NEUROPEPTIDE Y RECEPTOR TYPE 4	hgnc:9329	NPY4R	TTD	2020.06.01	NULL	52.50767123569449	TM30339	drugbank:DB05085	TM30339	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	1.312691780892362	E-913	iuphar.ligand:3500	E913	FALSE	FALSE	FALSE
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	0.9053046764774914	Divalproex sodium	rxcui:266856	DIVALPROEX SODIUM	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.090452491	Meprobamate	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.1539814405738841	Eslicarbazepine	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
RECEPTOR UNSPECIFIC	hgnc:16147	MCM8	TTD	2020.06.01	NULL	52.50767123569449	ATL-104	drugbank:DB05670	ATL-104	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.2442217266776488	Salmeterol	rxcui:36117	SALMETEROL	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	0.049864835	ISOQUINE	chembl:CHEMBL147587	ISOQUINE	FALSE	FALSE	FALSE
DEBRISOQUINE 4-HYDROXYLASE	hgnc:2625	CYP2D6	TTD	2020.06.01	NULL	0.029515273	ISOQUINE	chembl:CHEMBL147587	ISOQUINE	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.040328473	Phenytoin	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	0.079197091	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.1750255707856483	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.2103110997424346	Milnacipran	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	3.500511415712966	MK-3207	drugbank:DB12424	MK-3207	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.2500365296937833	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE XII	hgnc:1371	CA12	TTD	2020.06.01	NULL	0.9376369863516875	Sulfamylon	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.1312691780892362	Eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
ACYL-COA DESATURASE	hgnc:10571	SCD	TTD	2020.06.01	NULL	2.500365296937833	MK-8245	drugbank:DB13024	MK-8245	FALSE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	0.3500511415712966	FANG vaccine	ncit:C90552	GEMOGENOVATUCEL-T	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.1875273972703374	Famitinib	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
CATECHOL-O-METHYL-TRANSFERASE	hgnc:2228	COMT	TTD	2020.06.01	NULL	1.250182648468916	Opicapone	rxcui:2362167	OPICAPONE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1056492378987816	Famitinib	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
OVARIAN CARCINOMA ANTIGEN CA125	hgnc:15582	MUC16	TTD	2020.06.01	NULL	3.750547945	DMUC-5754A	chembl:CHEMBL3545372	SOFITUZUMAB VEDOTIN	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.3704244884352345	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	0.9723642821424906	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	1.019566431761058	MGL-3196	ncit:C170368	RESMETIROM	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.6482428547616604	BAF312	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
HYPERPOLARIZATION CYCLIC NUCLEOTIDE-GATED CHANNEL	hgnc:29665	MALAT1	TTD	2020.06.01	NULL	3.500511415712967	ZD-7288	iuphar.ligand:2359	ZD7288	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.4773424657790409	CG-100649	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	2.019525817	DRL-17822	iuphar.ligand:10721	DRL-17822	FALSE	FALSE	FALSE
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	1.831662950082366	LOXO-101	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.5122699632750684	Blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.3704244884352345	Idelalisib	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.3697723326457359	CC-223	ncit:C92575	ONATASERTIB	FALSE	FALSE	TRUE
PROTEIN KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	2.187819634820604	LX-7101	drugbank:DB16009	LX-7101	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.6403374540938354	JNJ 63723283	ncit:C129448	CETRELIMAB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.2561349816375342	M7824	ncit:C124229	BINTRAFUSP ALFA	FALSE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA3.1	hgnc:6293	KCNN4	TTD	2020.06.01	NULL	8.751278539282415	ASP-0819	iuphar.ligand:12646	ASP-0819	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.1539814405738841	Eslicarbazepine	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
GLUCOSE-6-PHOSPHATE DEHYDROGENASE	hgnc:4057	G6PD	TTD	2020.06.01	NULL	0.029170928	Prasterone	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
CHOLECYSTOKININ RECEPTOR TYPE A	hgnc:1570	CCKAR	TTD	2020.06.01	NULL	2.625383561784724	proglumide	rxcui:8730	PROGLUMIDE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1635752997996713	Protriptyline	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.034229251	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	1.790034246671403	Indecainide	ncit:C65910	INDECAINIDE	TRUE	FALSE	FALSE
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	1.250182648468916	Saruplase	ncit:C152306	SARUPLASE	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.2333674277141978	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	0.546954909	Besipirdine	ncit:C171657	BESIPIRDINE	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	1.093909817410302	16,16-dimethyl-PGE2	iuphar.ligand:1926	16,16-DIMETHYL-PGE2	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	1.591141552596802	Iralukast	ncit:C77981	IRALUKAST	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.007424727	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.016434326	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 19 MEMBER 1	hgnc:10937	SLC19A1	TTD	2020.06.01	NULL	0.364636606	Folic Acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.088695391	Methylscopolamine	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	1.029562181092048	NXN-188	drugbank:DB06096	NXN-188	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.1060761035064535	SAR425899	chembl:CHEMBL3545269	SAR425899	FALSE	FALSE	FALSE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	1.750255707856483	SAR425899	chembl:CHEMBL3545269	SAR425899	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	CARBIMAZOLE	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
P-SELECTIN	hgnc:10721	SELP	TTD	2020.06.01	NULL	13.12691780892362	SelG1	rxcui:2262279	CRIZANLIZUMAB	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.1154014752432846	Hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.6403374540938354	Anti-CD19 CAR T cells	ncit:C176018	ANTI-CD19 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.6403374540938354	Anti-CD19 CAR-T cells	ncit:C176018	ANTI-CD19 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.6403374540938354	Anti-CD20 CAR-T cells	ncit:C201174	ANTI-CD20 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.013673873	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.207267123	Clorazepate	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	0.5147810905460244	Eletriptan	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.007509678	Masoprocol	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.06970816	Triamcinolone	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.083744292	Triazolam	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.1286952726365061	Puerarin	drugbank:DB12290	PUERARIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	1.282909942931453	LGX818	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.7001022831425933	Pumosetrag	ncit:C84126	PUMOSETRAG	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.1508841127462485	Daniquidone	ncit:C66984	DANIQUIDONE	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	0.9053046764774912	MB-12066	drugbank:DB11948	LAPACHONE	FALSE	FALSE	FALSE
INTERLEUKIN-4	hgnc:6014	IL4	TTD	2020.06.01	NULL	3.500511415712966	SAR-156597	chembl:CHEMBL4298097	ROMILKIMAB	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.02232469	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	1.009762908	COVA322	iuphar.ligand:10469	COVA322	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.6105543166941221	Bentazepam	ncit:C74189	BENTAZEPAM	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.2817943000126717	Clonidine	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.7160136986685613	Etodolac	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	1.670698630226643	Glucagon recombinant	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	2.669881588255652	Forasartan	ncit:C65749	FORASARTAN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.3256289689035318	Formoterol	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.048958202	Ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003405608	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 2	hgnc:11331	SSTR2	TTD	2020.06.01	NULL	0.8334550989792776	Lanreotide acetate	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.09814518	Imipramine	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3677319929494733	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	1.628144844517658	Indiplon	ncit:C74385	INDIPLON	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.1684738114514262	Naproxen	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.2275522047050683	Temsirolimus	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
TUBULIN BETA-1 CHAIN	hgnc:16257	TUBB1	TTD	2020.06.01	NULL	0.2917092846427472	AI-850	drugbank:DB05842	AI-850	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.3201687270469177	AI-850	drugbank:DB05842	AI-850	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.1615620653405984	IPI-549	ncit:C125471	EGANELISIB	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.6403374540938354	AUTO3	drugbank:DB17364	AUTO3	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	0.6000876712650799	BGB-290	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	NSC-405662	chembl:CHEMBL118378	CHEMBL:CHEMBL118378	FALSE	FALSE	FALSE
CDC7-RELATED KINASE	hgnc:1745	CDC7	TTD	2020.06.01	NULL	12.11715490054488	BMS-863233	drugbank:DB12357	BMS-863233	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	2-HYDROXYESTRADIOL	ncit:C120474	2-HYDROXYESTRADIOL	FALSE	FALSE	FALSE
NEURAL CADHERIN	hgnc:1759	CDH2	TTD	2020.06.01	NULL	35.00511415712966	Exherin	ncit:C53399	ADH-1	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	2.838252499226729	VESTIPITANT MESYLATE	ncit:C95195	VESTIPITANT MESYLATE	FALSE	FALSE	FALSE
ADVANCED GLYCOSYLATION END PRODUCT RECEPTOR	hgnc:320	AGER	TTD	2020.06.01	NULL	10.50153424713889	Alagebrium chloride	ncit:C75185	ALAGEBRIUM CHLORIDE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	1.071585127259071	Bremelanotide	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
NCBIGENE:1519	hgnc:2542	CTSO	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8008	iuphar.ligand:8008	GSK2334470	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.06466462	IUPHAR.LIGAND:8182	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.037721028	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:20	iuphar.ligand:151	[3H]LY334370	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.06466462	IUPHAR.LIGAND:51	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:67	iuphar.ligand:67	9-OH-RISPERIDONE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.023823807	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003217973	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.3163112725041837	IUPHAR.LIGAND:10446	ncit:C79719	AVITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:3227	iuphar.ligand:3227	P-[18F]MPPF	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.090374649	IUPHAR.LIGAND:3	iuphar.ligand:3	1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:93	rxcui:8373	PIZOTYLINE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.1581556362520918	IUPHAR.LIGAND:218	iuphar.ligand:218	2-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.042174836	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:12	iuphar.ligand:12	EMDT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.039538909	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:142	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.1081888830405793	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:3248	iuphar.ligand:3248	[3H]5-HT	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1595977849109255	IUPHAR.LIGAND:51	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.2792961235941196	IUPHAR.LIGAND:218	iuphar.ligand:218	2-METHYL-5-HT	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	TCMDC-125142	chembl:CHEMBL528791	CHEMBL:CHEMBL528791	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.2792961235941196	IUPHAR.LIGAND:148	rxcui:4021	ERGONOVINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:187	iuphar.ligand:187	RS-102221	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.046059361	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:210	ncit:C73158	SARPOGRELATE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:195	iuphar.ligand:195	SDZ SER-082	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:187	iuphar.ligand:187	RS-102221	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.077217164	IUPHAR.LIGAND:147	iuphar.ligand:147	DOI	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DNDI1417420	chembl:CHEMBL1546223	CHEMBL:CHEMBL1546223	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.025739055	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.013313304	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.048260727	IUPHAR.LIGAND:193	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.097236428	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.021449212	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.01152495	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	LUZINDOLE	iuphar.ligand:1363	LUZINDOLE	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:12	iuphar.ligand:12	EMDT	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.049723174	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.049442252	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.040452751	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.1315981735230438	IUPHAR.LIGAND:3	iuphar.ligand:3	1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.070860555	IUPHAR.LIGAND:7351	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.041872146	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.02271093	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NCBIGENE:1385	hgnc:2345	CREB1	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:11610	iuphar.ligand:11610	HONOKIOL	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613069	IUPHAR.LIGAND:281	iuphar.ligand:281	SB 258719	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.6241137025199848	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.3777530304726222	IUPHAR.LIGAND:8065	iuphar.ligand:8065	GNF-5	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1888765152363111	IUPHAR.LIGAND:9173	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.053964719	IUPHAR.LIGAND:10402	iuphar.ligand:10402	ZAK INHIBITOR 6P	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	ALVERINE CITRATE	rxcui:71767	ALVERINE CITRATE	FALSE	FALSE	FALSE
NCBIGENE:1134	hgnc:1955	CHRNA1	GuideToPharmacology	2024.1	NULL	2.500365296937833	IUPHAR.LIGAND:4541	iuphar.ligand:4541	[14C]ACETYLCOA	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.006254636	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1656	hgnc:2747	DDX6	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8679	iuphar.ligand:8679	INCB3619	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.025489161	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
NCBIGENE:188	ncbigene:188	AGTRL2	GuideToPharmacology	2024.1	agonist	5.250767124	IUPHAR.LIGAND:5894	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:7902	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	modulator	1.166837138570988	IUPHAR.LIGAND:9429	iuphar.ligand:9429	MIRANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:9429	iuphar.ligand:9429	MIRANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:10437	iuphar.ligand:10437	COMPOUND E22 [PMID: 31298542]	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:7902	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	CRIDANIMOD	ncit:C77948	CRIDANIMOD	FALSE	FALSE	FALSE
NCBIGENE:1614	hgnc:13557	ACE2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11602	iuphar.ligand:11602	DX600	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:8523	iuphar.ligand:8523	MM07	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	activator	3.088686543276147	IUPHAR.LIGAND:4127	iuphar.ligand:4127	AGMATINE	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.075442056	IUPHAR.LIGAND:414	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:470	iuphar.ligand:470	MRS1191	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.056097939	IUPHAR.LIGAND:425	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.072125922	IUPHAR.LIGAND:375	iuphar.ligand:375	CGS 21680	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:416	iuphar.ligand:416	AB-MECA	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.056097939	IUPHAR.LIGAND:377	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:5620	iuphar.ligand:5620	PSB-11	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:445	iuphar.ligand:445	DEPX	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.075768645	IUPHAR.LIGAND:377	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:373	iuphar.ligand:373	2-HEXYNYL-NECA	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.09741683	IUPHAR.LIGAND:375	iuphar.ligand:375	CGS 21680	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:452	iuphar.ligand:452	[125I]ABOPX	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	CGP-12177	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:390	iuphar.ligand:390	MRE 2029F20	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:5599	iuphar.ligand:5599	HEMADO	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:470	iuphar.ligand:470	MRS1191	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.075768645	IUPHAR.LIGAND:448	iuphar.ligand:448	MRS1220	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:406	iuphar.ligand:406	[3H]DPCPX	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.2706580991530644	IUPHAR.LIGAND:462	iuphar.ligand:417	APNEA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.090219366	IUPHAR.LIGAND:404	iuphar.ligand:404	XANTHINE AMINE CONGENER	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11732	iuphar.ligand:11732	BAY-8400	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	CGS-12066B	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:8008	iuphar.ligand:8008	GSK2334470	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:12865	iuphar.ligand:12865	CANLITINIB	FALSE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8060	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.2638576444004749	CEPHALORIDINE	rxcui:2233	CEPHALORIDINE	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NCBIGENE:2957	hgnc:4646	GTF2A1	GuideToPharmacology	2024.1	NULL	10.50153424713889	IUPHAR.LIGAND:11338	iuphar.ligand:11338	BI-3802	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:11713	iuphar.ligand:11713	&BETA;-SECRETASE INHIBITOR IV	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.045461187	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9639	iuphar.ligand:9639	AMG-8718	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:8399	iuphar.ligand:8399	COMPOUND 13 [PMID: 23412139]	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:10455	ncit:C84132	RACTOPAMINE	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:10100	rxcui:2472254	VIBEGRON	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.3387591692625452	IUPHAR.LIGAND:3931	iuphar.ligand:3931	L 755507	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.2419708351875322	IUPHAR.LIGAND:509	rxcui:66887	RACEPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6158	iuphar.ligand:6158	RO5101576	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	FLAVANONE	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
NCBIGENE:2893	hgnc:4574	GRIA4	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:9084	iuphar.ligand:9084	COMPOUND 27 [PMID: 26938474]	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.056097939	IUPHAR.LIGAND:5893	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.053854022	IUPHAR.LIGAND:7047	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:5549	ncit:C63648	GALLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:10589	iuphar.ligand:10589	COMPOUND 18C [PMID:19143533]	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.1174668260306364	DIHYDROXYBERGAMOTTIN	chembl:CHEMBL513494	DIHYDROXYBERGAMOTTIN	FALSE	FALSE	FALSE
NCBIGENE:2345	ncbigene:2345	FNZ	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:10680	iuphar.ligand:10680	COMPOUND 33 [PMID: 32003991]	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.6105543166941221	IUPHAR.LIGAND:12565	ncit:C73026	EFONIDIPINE	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:7851	iuphar.ligand:7851	ORG27569	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.3029288725136221	IUPHAR.LIGAND:734	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.1187956362798518	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:749	iuphar.ligand:749	L-759,656	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:894	iuphar.ligand:894	A-71378	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:6666	iuphar.ligand:6666	[125I]DTYR-GLY-[(NLE28,31)CCK-26-33	FALSE	FALSE	FALSE
NCBIGENE:65	ncbigene:65	ACTBP5	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:816	iuphar.ligand:816	VMCC-I	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:10416	iuphar.ligand:10416	GSK2239633A	FALSE	FALSE	FALSE
NCBIGENE:1992	hgnc:3311	SERPINB1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12620	iuphar.ligand:12620	CIRTUVIVINT	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:9187	iuphar.ligand:9187	CCT245737	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:7943	iuphar.ligand:7943	MK-8776	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:8044	iuphar.ligand:8044	CCT241533	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.3431873936973497	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:2363	hgnc:3871	FRA1D	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:6552	iuphar.ligand:6552	COMPOUND 1 [PMID: 16650987]	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:10596	iuphar.ligand:10596	COMPOUND 29 [PMID: 31934767]	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:7882	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001719759	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:8999	iuphar.ligand:8999	(S)-ARN2508	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:914	iuphar.ligand:914	[125I]TYR0-CRF (HUMAN, RAT, MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:10684	ncit:C83650	DAVALINTIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	NSC-645827	chembl:CHEMBL95704	CHEMBL:CHEMBL95704	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.018699313	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:1994	hgnc:3312	ELAVL1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8836	iuphar.ligand:8836	PP1	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:3776	iuphar.ligand:3776	[125I]CT (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:818	iuphar.ligand:818	[125I]MINI-TYRRS	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:8532	iuphar.ligand:8532	CXCL12&EPSILON;	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:4358	iuphar.ligand:4358	CXCL12&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:850	iuphar.ligand:850	[125I]CXCL12&BETA; (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.072927321	IUPHAR.LIGAND:6045	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	0.043756393	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.07614901	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:1352	hgnc:2260	COX10	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11374	iuphar.ligand:11374	COMPOUND 7 [PMID: 32302132]	FALSE	FALSE	FALSE
NCBIGENE:1353	hgnc:2261	COX11	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:5157	ncit:C76006	CAMONAGREL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	N-OXALYLGLYCINE	chembl:CHEMBL90852	N-OXALYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	0.1256164383629055	IUPHAR.LIGAND:3340	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	agonist	0.9211872146613068	IUPHAR.LIGAND:3354	iuphar.ligand:3354	LTC4	FALSE	FALSE	FALSE
NCBIGENE:1353	hgnc:2261	COX11	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:8753	iuphar.ligand:8753	COMPOUND 10A [PMID: 1447738]	FALSE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12942	iuphar.ligand:12942	COMPOUND 42 [PMID: 37721854]	FALSE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:9892	ncit:C48264	TALABOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8164	iuphar.ligand:8164	COMPOUND 7K [PMID: 23521020]	FALSE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	GNF-PF-4576	chembl:CHEMBL527336	CHEMBL:CHEMBL527336	FALSE	FALSE	FALSE
NCBIGENE:2650	hgnc:4203	GCNT1	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7377	iuphar.ligand:7377	EPZ004777	FALSE	FALSE	TRUE
NCBIGENE:2637	hgnc:4186	GBX2	GuideToPharmacology	2024.1	inhibitor	0.2966535098061836	IUPHAR.LIGAND:6815	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1880	iuphar.ligand:1880	L-888,291	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:1887	iuphar.ligand:1887	SQ-27986	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:10169	ncit:C152874	VIDUPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.048083948	IUPHAR.LIGAND:7279	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:934	iuphar.ligand:934	N-PROPYLNORAPOMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.087512785	IUPHAR.LIGAND:969	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.058341857	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.009832897	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.039331589	IUPHAR.LIGAND:44	iuphar.ligand:44	NAFADOTRIDE	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.014749346	IUPHAR.LIGAND:969	iuphar.ligand:969	(-)-N-PORPHYNORAPOMORPHINE	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	SODIUM SELENITE	rxcui:56519	SODIUM SELENITE	TRUE	FALSE	FALSE
NCBIGENE:2325	hgnc:2895	EDAR	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:6144	iuphar.ligand:6144	ECTODYSPLASIN A1	FALSE	FALSE	FALSE
NCBIGENE:1822	hgnc:3033	ATN1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:5956	iuphar.ligand:5956	COMPOUND 56 [PMID: 8568816]	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-123947	chembl:CHEMBL525098	CHEMBL:CHEMBL525098	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.029416062	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12981	iuphar.ligand:12981	C34 [ZHU ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	antibody	0.013890918	IUPHAR.LIGAND:6882	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:10080	iuphar.ligand:10080	DIFLAPOLIN	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:1896	iuphar.ligand:1896	AH6809	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.023867123	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:1896	iuphar.ligand:1896	AH6809	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:1920	iuphar.ligand:1920	ONO-8711	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:5818	iuphar.ligand:5818	TG4-155	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:1918	ncit:C169951	ENPROSTIL	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.096521454	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:7647	iuphar.ligand:7647	BMS-599626	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:5858	rxcui:1862951	GRAPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:11676	ncit:C171059	TUXOBERTINIB	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:3459	iuphar.ligand:3459	METHYL-PIPERIDINO-PYRAZOLE	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:7542	ncit:C80679	LASOFOXIFENE	TRUE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:10565	iuphar.ligand:10565	ERD-308	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:1001	iuphar.ligand:1001	[125I]PD151242	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:3508	ncit:C75991	DARUSENTAN	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.020575106	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	CARBIMAZOLE	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011143394	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.014330696	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.3106962795011509	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.047561296	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.048260727	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:2834	iuphar.ligand:2834	DY131	FALSE	FALSE	FALSE
NCBIGENE:3014	hgnc:4739	H2AX	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:10037	ncit:C125193	ELTANEXOR	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	modulator	5.834185692854944	IUPHAR.LIGAND:12135	iuphar.ligand:12135	(R)-AS-1	FALSE	FALSE	FALSE
NCBIGENE:869	hgnc:1543	CBLN1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:4571	iuphar.ligand:4571	DIHYDROKAINATE	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.049723174	IUPHAR.LIGAND:4367	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.1970269089519493	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.091796628	IUPHAR.LIGAND:4348	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4257	iuphar.ligand:4257	MRK016	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.2302968036653267	IUPHAR.LIGAND:4296	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.2763561643983921	IUPHAR.LIGAND:7712	iuphar.ligand:7712	AZD7325	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.037666909	IUPHAR.LIGAND:7111	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.053361455	IUPHAR.LIGAND:4367	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.038808331	IUPHAR.LIGAND:7313	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2817943000126717	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.1065064325267637	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:4067	iuphar.ligand:4067	(&PLUSMN;)-CIS-2-CAMP	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	inhibitor	0.4167275494896389	IUPHAR.LIGAND:4287	iuphar.ligand:4287	PIPERIDINE-4-SULPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6076	iuphar.ligand:6076	J20 (GALANIN ANALOGUE)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6121	iuphar.ligand:6121	GALP(1-32) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3897	iuphar.ligand:3897	M32	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	MEPIVACAINE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:247	hgnc:434	ALOX15B	GuideToPharmacology	2024.1	agonist	0.3804903712731485	IUPHAR.LIGAND:6959	rxcui:1044584	TESAMORELIN	TRUE	FALSE	FALSE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8971	iuphar.ligand:8971	HUMAN GIP(3-30)NH2	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:1135	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:8544	iuphar.ligand:8544	WB4-24	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00449706	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:1099	ncit:C170105	LENOMORELIN	FALSE	FALSE	FALSE
NCBIGENE:247	hgnc:434	ALOX15B	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:6523	iuphar.ligand:6523	JI-38	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.2083637747448194	IUPHAR.LIGAND:4167	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:4245	ncit:C80379	TEZAMPANEL ANHYDROUS	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2071308530007672	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
NCBIGENE:877	hgnc:11007	SLC2A3	GuideToPharmacology	2024.1	NULL	2.625383561784724	IUPHAR.LIGAND:4643	iuphar.ligand:4643	[3H]2-DEOXYGLUCOSE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.218327115	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
NCBIGENE:2978	hgnc:4678	GUCA1A	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:10692	iuphar.ligand:10692	AMBROXOL	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1521961485092594	IUPHAR.LIGAND:4078	iuphar.ligand:4078	[3H]CGP39653	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	modulator	0.16256245	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	HARMAN	chembl:CHEMBL12014	HARMAN	FALSE	FALSE	FALSE
NCBIGENE:2029	hgnc:3360	ENSA	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:8015	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
NCBIGENE:2029	hgnc:3360	ENSA	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:7819	iuphar.ligand:7819	AZD1080	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7546	ncit:C174879	BITOPERTIN	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.2224901323546377	IUPHAR.LIGAND:8115	iuphar.ligand:8115	COMPOUND 2 [PMID: 22560567]	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:8171	iuphar.ligand:8171	COMPOUND 5B [PMID: 24900464]	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.1779921058837101	IUPHAR.LIGAND:8007	iuphar.ligand:8007	BX-912	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:8478	iuphar.ligand:8478	AZD2858	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:8016	iuphar.ligand:8016	CHIR-98014	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.022249013	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1170	iuphar.ligand:1170	[HIS5,D-TYR6]GNRH	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:5084	iuphar.ligand:5084	UROGUANYLIN	FALSE	FALSE	FALSE
NCBIGENE:403	hgnc:694	ARL3	GuideToPharmacology	2024.1	blocker	7.501095891	IUPHAR.LIGAND:6260	iuphar.ligand:6260	MEL57A	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:7008	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.2027323213733378	SB-242235	chembl:CHEMBL95692	SB-242235	FALSE	FALSE	FALSE
NCBIGENE:2615	hgnc:4161	LRRC32	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10490	iuphar.ligand:10490	SS-208	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	HYDRAMETHYLNON	chembl:CHEMBL464812	HYDRAMETHYLNON	FALSE	FALSE	FALSE
NCBIGENE:128	hgnc:253	ADH5	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:12945	iuphar.ligand:12945	NOX-6-7	FALSE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8774	iuphar.ligand:8774	LP-471756	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5517	iuphar.ligand:5517	ASN02563583	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	0.1842374429322614	IUPHAR.LIGAND:11209	iuphar.ligand:11209	EMBELIN	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	0.2375912725597036	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:123	hgnc:248	PLIN2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:12395	iuphar.ligand:12395	RTI-122	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	DNDI1417777	chembl:CHEMBL1412002	CHEMBL:CHEMBL1412002	FALSE	FALSE	FALSE
NCBIGENE:150	hgnc:281	ADRA2A	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7042	iuphar.ligand:7042	AR244555	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9940	iuphar.ligand:9940	LW106	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PAEONOL	drugbank:DB16830	PAEONOL	FALSE	FALSE	FALSE
NCBIGENE:2443	hgnc:3841	FRA11F	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10510	iuphar.ligand:10510	CAROTEGRAST METHYL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	5-(4-PHENYLBUTOXY)PSORALEN	iuphar.ligand:9583	PSORA-4	FALSE	FALSE	FALSE
NCBIGENE:1705	ncbigene:1705	DFNB13	GuideToPharmacology	2024.1	agonist	5.834185692854945	IUPHAR.LIGAND:4994	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1715936968486748	D-TRYPTOPHAN	drugbank:DB03225	D-TRYPTOPHAN	FALSE	FALSE	FALSE
NCBIGENE:1702	hgnc:5978	IL15RA	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:4981	iuphar.ligand:4981	IL-15	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.3017682254924971	8-AZAGUANINE	ncit:C28788	8-AZAGUANINE	FALSE	FALSE	FALSE
NCBIGENE:1706	ncbigene:1706	DFNB14	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:7674	rxcui:1989100	BENRALIZUMAB	TRUE	FALSE	FALSE
NCBIGENE:2044	hgnc:3389	EPHA5	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8213	iuphar.ligand:8213	COMPOUND R-16 [PMID: 21967808]	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	activator	2.917092846427472	IUPHAR.LIGAND:4124	iuphar.ligand:4124	ADENOPHOSTIN A	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:1967	ncit:C76896	BERAPROST	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12449	rxcui:155067	SILYBIN	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:12441	iuphar.ligand:12441	(&PLUSMN;)-EQUOL	FALSE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:2367	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10157	iuphar.ligand:10157	JAK3 INHIBITOR 34	FALSE	FALSE	FALSE
NCBIGENE:665	hgnc:1085	BNIP3L	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:10918	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:12350	iuphar.ligand:12350	CEE321	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:7793	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:8309	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:10632	iuphar.ligand:10632	ITACNOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:11060	iuphar.ligand:11060	PF-956980	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:10157	iuphar.ligand:10157	JAK3 INHIBITOR 34	FALSE	FALSE	FALSE
NCBIGENE:2378	hgnc:3890	FRA2F	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10576	iuphar.ligand:10576	COMPOUND 32 [PMID: 31675166]	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:9246	iuphar.ligand:9246	UPADACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2374	hgnc:3886	FRA2B	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10576	iuphar.ligand:10576	COMPOUND 32 [PMID: 31675166]	FALSE	FALSE	FALSE
NCBIGENE:2866	hgnc:4500	GPR42	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8483	iuphar.ligand:8483	COMPOUND 4D [PMID: 25489658]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.040640612	IUPHAR.LIGAND:1638	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.007686674	IUPHAR.LIGAND:7877	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:7879	iuphar.ligand:7879	BMS-690514	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.025942525	IUPHAR.LIGAND:10181	iuphar.ligand:10181	COMPOUND 19A [PMID: 30503936]	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.1037701012563132	IUPHAR.LIGAND:10472	ncit:C62791	PEGDINETANIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0148243	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.2075402025126264	IUPHAR.LIGAND:6055	iuphar.ligand:6055	VEGF RECEPTOR 2 KINASE INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.006289097	IUPHAR.LIGAND:5891	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1288	iuphar.ligand:1288	KISSPEPTIN-54	FALSE	FALSE	FALSE
NCBIGENE:525	hgnc:853	ATP6V1B1	GuideToPharmacology	2024.1	activator	0.3387591692625452	IUPHAR.LIGAND:2505	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
NCBIGENE:520	hgnc:844	ATP5MC2P1	GuideToPharmacology	2024.1	activator	0.364636606	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	activator	4.773424657790408	IUPHAR.LIGAND:11854	iuphar.ligand:11854	NS11021	FALSE	FALSE	FALSE
NCBIGENE:433	hgnc:743	ASGR2	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	0.375054795	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	0.4688184931758437	IUPHAR.LIGAND:2356	iuphar.ligand:2356	CS+	FALSE	FALSE	FALSE
NCBIGENE:441	hgnc:6269	KCNJ8	GuideToPharmacology	2024.1	activator	6.563458904461812	IUPHAR.LIGAND:2413	ncit:C79109	CROMAKALIM	FALSE	FALSE	FALSE
NCBIGENE:385	hgnc:18865	KCNT1	GuideToPharmacology	2024.1	blocker	0.5250767123569451	IUPHAR.LIGAND:2342	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:573	hgnc:937	BAG1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:2612	iuphar.ligand:2612	ERGTX-1	FALSE	FALSE	FALSE
NCBIGENE:545	hgnc:882	ATR	GuideToPharmacology	2024.1	blocker	0.1750255707856483	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:1242	hgnc:20692	TPH2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:12993	iuphar.ligand:12993	TPT-004	FALSE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10647	ncit:C171780	RODATRISTAT	FALSE	FALSE	FALSE
NCBIGENE:94	hgnc:175	ACVRL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:6991	iuphar.ligand:6991	[1-BROMO-(3S)-HYDROX-4-(PALMITOYLOXY)BUTYL]PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7003	iuphar.ligand:7003	PLUMBAGIN	FALSE	FALSE	FALSE
NCBIGENE:2682	hgnc:11114	KDM5C	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8229	iuphar.ligand:8229	IOX2	FALSE	FALSE	FALSE
NCBIGENE:2681	hgnc:4253	GGTA1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8576	iuphar.ligand:8576	KDOAM25	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1292	iuphar.ligand:1292	COMPOUND 2 [PMID: 11375253]	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:9692	iuphar.ligand:9692	STK16-IN-1	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:8004	iuphar.ligand:8004	TORIN 1	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:7884	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:8805	iuphar.ligand:8805	COMPOUND 82 [PMID: 21332118]	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:9174	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	antibody	0.3088686543276147	IUPHAR.LIGAND:7748	iuphar.ligand:7748	EMIBETUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:9841	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:3954	iuphar.ligand:3954	BIPHENYLINDANONE A	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.5357925636295356	IUPHAR.LIGAND:1424	iuphar.ligand:1424	3,3'-DIFLUOROBENZALDAZINE	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1423	iuphar.ligand:1423	CPPHA	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1420	iuphar.ligand:1420	ADX-47273	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:1438	iuphar.ligand:1438	PPG	FALSE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:5968	iuphar.ligand:5968	ERK INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.072725306	IUPHAR.LIGAND:7080	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:5966	drugbank:DB07794	5-(2-PHENYLPYRAZOLO[1,5-A]PYRIDIN-3-YL)-1H-PYRAZOLO[3,4-C]PYRIDAZIN-3-AMINE	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:9328	iuphar.ligand:9328	TAK-715	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:12846	iuphar.ligand:12846	NDPPC	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:7835	ncit:C96532	LOSMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.022099188	IUPHAR.LIGAND:4307	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
NCBIGENE:2093	ncbigene:2093	ERVT3	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11114	iuphar.ligand:11114	DCLK1-IN-1	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:7818	iuphar.ligand:7818	PH-797804	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9377	iuphar.ligand:9377	JNK INHIBITOR 9L	FALSE	FALSE	FALSE
NCBIGENE:2068	hgnc:3434	ERCC2	GuideToPharmacology	2024.1	modulator	0.2651902587661338	IUPHAR.LIGAND:7626	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:1635	hgnc:2710	DCTD	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8665	iuphar.ligand:8665	COMPOUND 10 [PMID: 18790648]	FALSE	FALSE	FALSE
NCBIGENE:1640	hgnc:7162	MMP16	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8629	iuphar.ligand:8629	SL422	FALSE	FALSE	FALSE
NCBIGENE:1639	hgnc:2711	DCTN1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8629	iuphar.ligand:8629	SL422	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7604	rxcui:11476	TILUDRONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8629	iuphar.ligand:8629	SL422	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	0.1339481409073839	IUPHAR.LIGAND:6510	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:989	hgnc:1717	SEPTIN7	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11735	iuphar.ligand:11735	COMPOUND 18N [PMID: 34382802]	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:11902	iuphar.ligand:11902	DS-3801B FREE BASE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:303	iuphar.ligand:303	OXOTREMORINE-M	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:293	iuphar.ligand:293	NNC 11-1607	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.100976291	IUPHAR.LIGAND:349	rxcui:11201	VINCAMINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.1105424657593568	IUPHAR.LIGAND:344	iuphar.ligand:344	N-CHLOROMETHYL-BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.138178082	IUPHAR.LIGAND:341	iuphar.ligand:341	ALCURONIUM	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:307	iuphar.ligand:307	4-DAMP	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:7483	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:298	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:7772	iuphar.ligand:7772	UCM 549	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:7772	iuphar.ligand:7772	UCM 549	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.048083948	IUPHAR.LIGAND:1670	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.4730420832044549	IUPHAR.LIGAND:4808	rxcui:60842	REBOXETINE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:10342	rxcui:2121751	SOLRIAMFETOL	TRUE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.1392776425349987	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:2998	hgnc:4707	GYS2	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:11335	iuphar.ligand:11335	EG00229	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:11198	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	agonist	0.081533651	IUPHAR.LIGAND:2585	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
NCBIGENE:467	hgnc:785	ATF3	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:3985	iuphar.ligand:3985	&ALPHA;-CONOTOXIN PIA	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	blocker	1.250182648468916	IUPHAR.LIGAND:3986	iuphar.ligand:3986	A-867744	FALSE	FALSE	FALSE
NCBIGENE:466	hgnc:783	ATF1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:3982	iuphar.ligand:3982	&ALPHA;-CONOTOXIN PNIA	FALSE	FALSE	FALSE
NCBIGENE:304	hgnc:539	ANXA2P2	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1496	iuphar.ligand:1496	NEUROPEPTIDE W-30	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1683	iuphar.ligand:1683	N/OFQ-NH2	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1696	iuphar.ligand:1696	PEPTIDE III-BTD	FALSE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3855	iuphar.ligand:3855	AVA3	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:11235	iuphar.ligand:11235	COMPOUND 46 [PMID: 25268943]	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:1485	iuphar.ligand:1485	BIBP3226	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:12603	ncit:C175783	FIRAZOREXTON	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	1.591141552596802	IUPHAR.LIGAND:3391	iuphar.ligand:3391	5-OXO-ETE	FALSE	FALSE	FALSE
NCBIGENE:162	hgnc:554	AP1B1	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:3636	rxcui:17511	ALPHA-KETOGLUTARIC ACID	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9136	iuphar.ligand:9136	SB-674042	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:8940	iuphar.ligand:8940	IPA-3	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:4038	iuphar.ligand:4038	TCS-OX2-29	FALSE	FALSE	FALSE
NCBIGENE:2138	hgnc:3519	EYA1	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:8937	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:4324	iuphar.ligand:4324	TNP-ATP	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9538	iuphar.ligand:9538	AF-906	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:4790	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	agonist	0.16256245	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	agonist	0.1544343271638073	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	2.187819634820604	IUPHAR.LIGAND:4142	iuphar.ligand:4142	AZ11645373	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	0.1816874437221263	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	2.187819634820604	IUPHAR.LIGAND:10338	rxcui:388	POLYMYXIN B SULFATE	TRUE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:1713	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1774	iuphar.ligand:1774	[33P]2MESADP	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5806	iuphar.ligand:5806	GLAXOSMITHKLINE COMPOUND 6I [PMID:18926700]	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:5453	iuphar.ligand:5453	AP5A	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:1735	iuphar.ligand:1735	UTP&GAMMA;S	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2266	iuphar.ligand:2266	N-STEARYL-[NLE17] NEUROTENSIN-(6-11)/VIP-(7-28)	FALSE	FALSE	FALSE
NCBIGENE:2590	hgnc:4124	GALNT2	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:5277	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:12490	iuphar.ligand:12490	AZ2429	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:9456	iuphar.ligand:9456	AC-55541	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:6659	iuphar.ligand:6659	P2PAL18S	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:10001	iuphar.ligand:10001	COMPOUND 52 [PMID: 28541707]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:8805	iuphar.ligand:8805	COMPOUND 82 [PMID: 21332118]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:10151	iuphar.ligand:10151	NEOLYMPHOSTIN A	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:9424	rxcui:2633005	LENIOLISIB	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:5701	iuphar.ligand:5701	PI-103	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:9692	iuphar.ligand:9692	STK16-IN-1	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9330	iuphar.ligand:9330	CDP840	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9852	iuphar.ligand:9852	MK-0359	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:7698	iuphar.ligand:7698	AZD1208	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:10195	iuphar.ligand:10195	COMPOUND 28 [PMID: 30624936]	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:10420	iuphar.ligand:10420	CHMFL-KIT-64	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:11747	iuphar.ligand:11747	BPR1R024	FALSE	FALSE	FALSE
NCBIGENE:1432	hgnc:6876	MAPK14	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:9797	iuphar.ligand:9797	COMPOUND 37 [PMID: 29193967]	FALSE	FALSE	FALSE
NCBIGENE:2394	hgnc:3906	FRA5B	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6570	rxcui:1056	APROTININ	TRUE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6064	iuphar.ligand:6064	TRIAZINE COMPOUND PC1	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:10420	iuphar.ligand:10420	CHMFL-KIT-64	FALSE	FALSE	FALSE
NCBIGENE:1434	hgnc:2431	CSE1L	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8781	iuphar.ligand:8781	FIPI	FALSE	FALSE	FALSE
NCBIGENE:2386	hgnc:3898	FRA3C	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:8668	iuphar.ligand:8668	FURIN INHIBITOR PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1252	hgnc:5187	PRMT1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8955	iuphar.ligand:8955	MS023	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	BROXYQUINOLINE	ncit:C73253	BROXYQUINOLINE	FALSE	FALSE	FALSE
NCBIGENE:1254	ncbigene:1254	CMTX3	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:8955	iuphar.ligand:8955	MS023	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5163	iuphar.ligand:5163	CGP53353	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:3263	hgnc:5171	HPX	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:5349	iuphar.ligand:5349	OKADAIC ACID	FALSE	FALSE	FALSE
NCBIGENE:3203	hgnc:5107	HOXA6	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12068	iuphar.ligand:12068	BATOPROTAFIB	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:10402	iuphar.ligand:10402	ZAK INHIBITOR 6P	FALSE	FALSE	FALSE
NCBIGENE:1014	hgnc:1755	CDH16	GuideToPharmacology	2024.1	NULL	0.1562728310586145	IUPHAR.LIGAND:4674	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	PAEONOL	drugbank:DB16830	PAEONOL	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:8728	iuphar.ligand:8728	(5E)-1-(4-FLUOROPHENYL)-5-[(5-METHYLTHIOPHEN-2-YL)METHYLIDENE]-2-SULFANYLIDENE-1,3-DIAZINANE-4,6-DIONE	FALSE	FALSE	FALSE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10386	iuphar.ligand:10386	CELASTROL	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:2648	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.2983390411119005	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:6952	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:2641	iuphar.ligand:2641	BMS493	FALSE	FALSE	FALSE
NCBIGENE:2911	hgnc:4593	GRM1	GuideToPharmacology	2024.1	antibody	6.563458904461812	IUPHAR.LIGAND:9290	iuphar.ligand:9290	ELEZANUMAB	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	inhibitor	0.1875273972703374	IUPHAR.LIGAND:2641	iuphar.ligand:2641	BMS493	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.012154554	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:8163	iuphar.ligand:8163	COMPOUND 33 [PMID: 19364658]	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.010012905	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.014268389	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:1997	iuphar.ligand:1997	RELAXIN-3 (B CHAIN)	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	XANTHOANGELOL B	chembl:CHEMBL494082	XANTHOANGELOL B	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12120	iuphar.ligand:12120	RLX-33	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:12505	iuphar.ligand:12505	DC591053	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2001	iuphar.ligand:2001	[125I]INSL5 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:11918	iuphar.ligand:11918	ANALOGUE 13: B7-24	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001655923	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:9492	iuphar.ligand:9492	COMPOUND 43 [PMID: 26751273]	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
NCBIGENE:2714	ncbigene:2714	GKP4	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8239	iuphar.ligand:8239	LLY-507	FALSE	FALSE	FALSE
NCBIGENE:2703	hgnc:4281	GJA8	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8235	iuphar.ligand:8235	(R)-PFI-2	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
NCBIGENE:1534	hgnc:2571	CYB561	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8040	iuphar.ligand:8040	GSK650394	FALSE	FALSE	FALSE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12915	iuphar.ligand:12915	SD-36	FALSE	FALSE	FALSE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10682	iuphar.ligand:10682	COMPOUND 8U [PMID: 31999451]	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	PINACIDIL	rxcui:33717	PINACIDIL	TRUE	FALSE	FALSE
NCBIGENE:1171	hgnc:14679	SLC38A4	GuideToPharmacology	2024.1	NULL	5.250767124	IUPHAR.LIGAND:4543	rxcui:426	ALANINE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.018719312	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NCBIGENE:959	hgnc:11935	CD40LG	GuideToPharmacology	2024.1	NULL	1.810609352954982	IUPHAR.LIGAND:12775	iuphar.ligand:12775	BULEVIRTIDE	FALSE	FALSE	FALSE
NCBIGENE:1173	hgnc:564	AP2M1	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:4623	iuphar.ligand:4623	[14C]HISTIDINE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015088411	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
NCBIGENE:1050	hgnc:1833	CEBPA	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11611	iuphar.ligand:11611	CGP-37157	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	DITHIAZANINE	ncit:C72743	DITHIAZANINE	FALSE	FALSE	FALSE
NCBIGENE:1422	hgnc:9029	PLA2G10	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8787	iuphar.ligand:8787	COMPOUND 12E [PMID: 18605714]	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11145	iuphar.ligand:11145	COMPOUND 55 [PMID: 30889352]	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.022730594	IUPHAR.LIGAND:5678	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8068	iuphar.ligand:8068	WH-4-023	FALSE	FALSE	FALSE
SLC22A6	hgnc:10970	SLC22A6	DTC	9/2/20	NULL	3.281729452230906	GS-9256	drugbank:DB12876	GS-9256	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2022	iuphar.ligand:2022	[125I]CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:2015	iuphar.ligand:2015	L-797,591	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.09869863	IUPHAR.LIGAND:2054	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.058341857	IUPHAR.LIGAND:2055	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2056	iuphar.ligand:2056	[111IN,90Y]DOTA-LAN	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:2066	iuphar.ligand:2066	PRL-2915	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2022	iuphar.ligand:2022	[125I]CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:2029	iuphar.ligand:2029	[L-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2022	iuphar.ligand:2022	[125I]CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:2739	hgnc:4323	GLO1	GuideToPharmacology	2024.1	NULL	4.375639269641208	IUPHAR.LIGAND:12842	iuphar.ligand:12842	SMD-3040	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:9631	iuphar.ligand:9631	CIS-EPOXYSUCCINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.2375912725597036	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:2235	hgnc:3647	FECH	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8218	iuphar.ligand:8218	COMPOUND 1 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10673	iuphar.ligand:10673	RK-287107	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:10105	iuphar.ligand:10105	DDR1/2 INHIBITOR 5N	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	NULL	4.773424657790408	IUPHAR.LIGAND:4867	iuphar.ligand:4867	ANGIOPOIETIN-1	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	GNF-PF-3756	chembl:CHEMBL597035	CHEMBL:CHEMBL597035	FALSE	FALSE	FALSE
NCBIGENE:2642	hgnc:4192	GCGR	GuideToPharmacology	2024.1	inhibitor	0.105015342	IUPHAR.LIGAND:6837	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
NCBIGENE:1759	hgnc:2972	DNM1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:9843	rxcui:2665622	AGATOLIMOD	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.169927739	IUPHAR.LIGAND:2637	rxcui:13982	TIRATRICOL	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1978	iuphar.ligand:1978	ONO-3708	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.2160809515872201	IUPHAR.LIGAND:8216	iuphar.ligand:8216	SB-431542	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.2465148884304905	MUCRONULATOL(+/-)	chembl:CHEMBL478971	MUCRONULATOL(+/-)	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6303	iuphar.ligand:6303	METHYLGLYOXAL	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:10288	iuphar.ligand:10288	M084	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:4211	iuphar.ligand:4211	HC030031	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	2.282942227638891	IUPHAR.LIGAND:10282	iuphar.ligand:10282	PYR10	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:4255	iuphar.ligand:4255	ML204	FALSE	FALSE	FALSE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	blocker	0.4102161815288632	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
STAT5A	hgnc:11366	STAT5A	DTC	9/2/20	NULL	5.625821918110125	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:12533	iuphar.ligand:12533	PYRAZOLO-PYRIMIDINE 14A [PMID: 29859875]	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.096521454	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:10297	iuphar.ligand:10297	CIM0216	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.1121958787087489	IUPHAR.LIGAND:2402	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	0.2573905452730122	IUPHAR.LIGAND:2421	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:255	hgnc:12373	TSHR	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:9113	iuphar.ligand:9113	COMPOUND 8B [PMID: 22408719]	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:12560	iuphar.ligand:12560	GSK3527497	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:8315	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:12350	iuphar.ligand:12350	CEE321	FALSE	FALSE	FALSE
BMP2	hgnc:1069	BMP2	DTC	9/2/20	NULL	26.25383561784724	METHYL 4-AMINOBENZOATE	chembl:CHEMBL1927048	CHEMBL:CHEMBL1927048	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.065145994	IUPHAR.LIGAND:7791	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:10157	iuphar.ligand:10157	JAK3 INHIBITOR 34	FALSE	FALSE	FALSE
NCBIGENE:2271	hgnc:3700	FH	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:8213	iuphar.ligand:8213	COMPOUND R-16 [PMID: 21967808]	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2156	iuphar.ligand:2156	UROTENSIN II-RELATED PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1010	hgnc:1751	CDH12	GuideToPharmacology	2024.1	inhibitor	4.773424657790409	IUPHAR.LIGAND:9605	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:2776	iuphar.ligand:2776	2MD	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2271	iuphar.ligand:2271	N-STEARYL-[NLE17]VIP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2175	iuphar.ligand:2175	[3H]AVP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.019490598	IUPHAR.LIGAND:2184	iuphar.ligand:2184	D[D-PAL2]AVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.014617949	IUPHAR.LIGAND:2202	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:2178	iuphar.ligand:2178	[PHE3]OT	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	10-DEACETOXYPACLITAXEL	chembl:CHEMBL306786	CHEMBL:CHEMBL306786	FALSE	FALSE	FALSE
NCBIGENE:2281	hgnc:3712	FKBP1B	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:8122	iuphar.ligand:8122	COMPOUND 25 [PMID: 17935989]	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.6482428547616604	IUPHAR.LIGAND:1545	iuphar.ligand:1545	[LEU31,PRO34]NPY	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.6482428547616604	IUPHAR.LIGAND:1527	iuphar.ligand:1527	[LEU31,PRO34]PYY (HUMAN)	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00402481	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
NCBIGENE:1579	hgnc:2642	CYP4A11	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8803	iuphar.ligand:8803	APSTATIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.061412481	U-73122	iuphar.ligand:5283	U73122	FALSE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:6044	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2285	hgnc:3717	FKBP1AP4	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6047	iuphar.ligand:6047	SYK INHIBITOR II	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.090821275	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PDGFB	hgnc:8800	PDGFB	CIViC	10-Apr-24	NULL	0.3500511415712966	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005574063	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	1.080404757936101	AGERAFENIB	ncit:C107245	AGERAFENIB	FALSE	FALSE	TRUE
IKZF1	hgnc:13176	IKZF1	CIViC	10-Apr-24	NULL	0.1154014752432846	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.5000730593875666	SAIT301	ncit:C119619	ANTI-C-MET MONOCLONAL ANTIBODY SAIT301	FALSE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.2573905452730122	PROPENTOFYLLINE	rxcui:34644	PROPENTOFYLLINE	FALSE	FALSE	FALSE
ZEB1	hgnc:11642	ZEB1	CIViC	10-Apr-24	NULL	17.50255707856483	SALINOMYCIN	rxcui:1311566	SALINOMYCIN	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	CIViC	10-Apr-24	NULL	0.103633562	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.007134194	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.010857666	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
DNMT3A	hgnc:2978	DNMT3A	CIViC	10-Apr-24	NULL	0.31115657	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.01823183	NIVOLUMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.07631929	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
DDX43	hgnc:18677	DDX43	CIViC	10-Apr-24	NULL	1.093909817410302	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	CLEMASTINE FUMARATE	rxcui:142430	CLEMASTINE FUMARATE	TRUE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	CIViC	10-Apr-24	NULL	0.1215455352678113	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	CIViC	10-Apr-24	NULL	0.04468738	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.017737081	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.029833904	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.014617949	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	TETRAZOLIUM RED	chembl:CHEMBL401540	TETRAZOLIUM RED	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
FOXO1	hgnc:3819	FOXO1	CIViC	10-Apr-24	NULL	5.250767123569449	BET INHIBITOR	ncit:C128462	BET INHIBITOR	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.3043922970185188	CGM097	ncit:C104280	P53/HDM2 INTERACTION INHIBITOR CGM097	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.2905562835176771	Repotrectinib	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	2.407466349146467	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.3043922970185188	TNO155	ncit:C139559	BATOPROTAFIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.038977062	Cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.032472277	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.095468493	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.061197752	Ibuprofen	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.1961681366215236	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.2615575154953649	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.034229251	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	1.060761035064535	MAK683	iuphar.ligand:10515	MAK683	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	1.438566335224506	PLX038	ncit:C167334	PEGYLATED SN-38 CONJUGATE PLX038	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	1.336059069138614	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.027490927	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	Pegylated liposomal doxorubicin	rxcui:214525	DOXORUBICIN LIPOSOME	TRUE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.1682938180631233	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.561579372	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Balstilimab	ncit:C136465	BALSTILIMAB	FALSE	FALSE	FALSE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	0.3182283105193606	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.3088686543276147	Pegylated liposomal doxorubicin	rxcui:214525	DOXORUBICIN LIPOSOME	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.019610708	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	IO102-IO103	ncit:C148154	PD-L1/IDO PEPTIDE VACCINE IO102-103	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.010614043	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.021215221	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	0.31115657	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.4565884455277783	Volasertib	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.089222891	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.07631929	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1547594520630995	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.007937668	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006555265	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	2',4'-DIHYDROXY FLAVONE	chembl:CHEMBL1374610	CHEMBL:CHEMBL1374610	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.00644424	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	IODOMELATONIN	drugbank:DB08190	N-[2-(2-IODO-5-METHOXY-1H-INDOL-3-YL)ETHYL]ACETAMIDE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.3684748858645227	PD98059	iuphar.ligand:5241	PD98059	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1296485709523321	Avapritinib	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.276356164	ASP5878	iuphar.ligand:11934	ASP5878	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.008643238	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.049864835	Momelotinib	rxcui:2665204	MOMELOTINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	Tuspetinib	ncit:C165254	TUSPETINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.038894571	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.058931169	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	VITAMIN B2	chembl:CHEMBL1397833	VITAMIN B2	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.076263865	Semaxanib	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.1243602739792764	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2282942227638891	AZD1208	iuphar.ligand:7698	AZD1208	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.029715717	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2038341274677581	Tofacitinib	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.5707355569097228	Ilginatinib	ncit:C98109	ILGINATINIB	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.05293112	Chloroquine	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	PKI-402	chembl:CHEMBL589258	CHEMBL:CHEMBL589258	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	KU-57788	iuphar.ligand:8010	NU-7441	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.073922431	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	1.944728564284981	Pralsetinib	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.729273212	TNO155	ncit:C139559	BATOPROTAFIB	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.2130128650535274	Exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.009272878	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	Pirtobrutinib	rxcui:2629338	PIRTOBRUTINIB	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.013589562	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.038636991	Hu5F9-G4	ncit:C117730	MAGROLIMAB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.008916229	Lenalidomide	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	GDC-0425	drugbank:DB14791	GDC-0425	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	GDC-0575	ncit:C116845	CHK1 INHIBITOR GDC-0575	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.009659248	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	PYRILAMINE	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.05664258	ERYTHROSINE	rxcui:4061	ERYTHROSINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004176557	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.1835932560688619	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	DTC	9/2/20	NULL	2.763561643983921	CF102	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	REL-CISAPRIDE	chembl:CHEMBL74656	REL-CISAPRIDE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.051177067	LINOLEIC ACID	rxcui:6400	LINOLEIC ACID	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.1562728310586145	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
UNIPROT:P21964	hgnc:2228	COMT	TdgClinicalTrial	Jan-14	NULL	1.500219178	ENTACAPONE	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.445925021	DIHYDROTACHYSTEROL	rxcui:3429	DIHYDROTACHYSTEROL	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:3232	iuphar.ligand:3232	SB258585	FALSE	FALSE	FALSE
NCBIGENE:2768	hgnc:4380	GNA12	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7404	rxcui:38386	TOLRESTAT	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:5613	iuphar.ligand:5613	ST-1535	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:8897	iuphar.ligand:8897	AC-186	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	NOSCAPINE	rxcui:7533	NOSCAPINE	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	ChEMBL	33	inhibitor	0.006311777	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2465148884304905	BRIMONIDINE TARTRATE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.075010959	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.4487835148349957	PREMARIN	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.2243917574174978	SONOLISIB	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007003824	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	NSC-108783	chembl:CHEMBL1489812	CHEMBL:CHEMBL1489812	FALSE	FALSE	FALSE
UNIPROT:O14788	hgnc:11926	TNFSF11	TdgClinicalTrial	Jan-14	NULL	2.019525816757481	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.068191781	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1997	hgnc:3316	ELF1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:9371	iuphar.ligand:9371	PF-670462	FALSE	FALSE	FALSE
NCBIGENE:389	hgnc:669	RHOC	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:4269	iuphar.ligand:4269	NNC55-0396	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.029498692	IUPHAR.LIGAND:9189	iuphar.ligand:9189	HS665	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.007354016	IUPHAR.LIGAND:4941	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.1105424657593568	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.085239726	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	HESPERIDIN	rxcui:5281	HESPERIDIN	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.093098708	ANTHRACYCLINE	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.063110182	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.034374908	OESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
TTN	hgnc:12403	TTN	NCI	14-Sep-17	NULL	5.250767124	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
PRKAB2	hgnc:9379	PRKAB2	PharmGKB	4/5/24	NULL	1.077080435603989	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.082043236	ethinyl estradiol	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.2117244807890907	RUPATADINE	ncit:C73055	RUPATADINE	FALSE	FALSE	FALSE
PSMB6	hgnc:9543	PSMB6	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001750547	CITALOPRAM	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	PROPIDIUM	drugbank:DB02166	PROPIDIUM	FALSE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.7501095890813501	TUBOCURARINE CHLORIDE	rxcui:82115	TUBOCURARINE CHLORIDE	TRUE	FALSE	FALSE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	1.750255707856483	TCMDC-137788	chembl:CHEMBL587564	CHEMBL:CHEMBL587564	FALSE	FALSE	FALSE
MIA	hgnc:7076	MIA	NCI	14-Sep-17	NULL	1.666910197958555	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001719759	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.085796848	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	AMARANTH	chembl:CHEMBL1408927	AMARANTH	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	(+)-CATECHIN HYDRATE	chembl:CHEMBL1256783	CHEMBL:CHEMBL1256783	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.012209667	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010629083	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
STIM1	hgnc:11386	STIM1	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002270307	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	3.088686543276147	IMO-2125	ncit:C125080	TILSOTOLIMOD SODIUM	FALSE	FALSE	FALSE
NCBIGENE:1662	hgnc:2735	DDX10	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:6482	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.1151484018326633	MP-412	chembl:CHEMBL5095024	MP-412	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	U-73122	iuphar.ligand:5283	U73122	FALSE	FALSE	FALSE
ASGR1	hgnc:742	ASGR1	ChEMBL	33	binder	3.750547945	VUPANORSEN	ncit:C174612	VUPANORSEN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	PYRIDINE-2,4-DICARBOXYLIC ACID	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003677523	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	THIOPROPERAZINE MESYLATE	ncit:C80010	THIOPROPERAZINE MESYLATE	FALSE	FALSE	FALSE
EPHA6	hgnc:19296	EPHA6	PharmGKB	4/5/24	NULL	0.3889457128569963	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:613	iuphar.ligand:613	NEUROMEDIN B	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8042	iuphar.ligand:8042	VE-821	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015088411	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
NFATC2	hgnc:7776	NFATC2	PharmGKB	4/5/24	NULL	0.1562728310586145	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-242718	chembl:CHEMBL275724	CHEMBL:CHEMBL275724	FALSE	FALSE	FALSE
PDE6A	hgnc:8785	PDE6A	ChEMBL	33	inhibitor	0.1861974157294131	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.033002936	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1017590527823536	THIOCOLCHICOSIDE	rxcui:38085	THIOCOLCHICOSIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	CINNAMALDEHYDE	rxcui:1368153	CINNAMIC ALDEHYDE	TRUE	FALSE	FALSE
RPS5	hgnc:10426	RPS5	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:344	iuphar.ligand:344	N-CHLOROMETHYL-BRUCINE	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.000146118775133	ABT-700	ncit:C106262	TELISOTUZUMAB	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
BHMT	hgnc:1047	BHMT	ChEMBL	33	other/unknown	8.751278539282415	BETAINE HYDROCHLORIDE	rxcui:81965	BETAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	1.009762908	DNDI1417722	chembl:CHEMBL1503190	CHEMBL:CHEMBL1503190	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.00854617	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.02339914	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
ERCC1	hgnc:3433	ERCC1	NCI	14-Sep-17	NULL	0.100589408	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.6584034010745392	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10582	iuphar.ligand:10582	COMPOUND 15B [PMID: 31811124]	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.2059124362184097	IUPHAR.LIGAND:11624	iuphar.ligand:11624	NINGETINIB	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1640864726115453	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.046940525	5-FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1320947704042629	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2734774543525755	SJ000029700	chembl:CHEMBL591864	CHEMBL:CHEMBL591864	FALSE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.1400204566285186	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
NCBIGENE:1840	hgnc:3060	DTX1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:11198	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.2243917574174978	IUPHAR.LIGAND:4066	iuphar.ligand:4066	(+)-HA966	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:4845	iuphar.ligand:4845	[125I]ANP (HUMAN)	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.004045275	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.02103111	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.022554842	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PSMA3	hgnc:9532	PSMA3	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
QUINONE REDUCTASE 2	hgnc:7856	NQO2	TTD	2020.06.01	NULL	3.088686543276147	Prolarix	ncit:C80048	CARICOTAMIDE/TRETAZICAR	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:1100	ncit:C76092	EXAMORELIN	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	inhibitor	0.017760078	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.050007306	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	MECLOCYCLINE SULFOSALICYLATE	rxcui:203162	MECLOCYCLINE SULFOSALICYLATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	DERRUBONE	chembl:CHEMBL412010	DERRUBONE	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.3182283105193606	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.019304291	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.078958904	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
SCG5	hgnc:10816	SCG5	NCI	14-Sep-17	NULL	1.666910197958555	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.2386712328895204	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.4688184931758437	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.1615620653405984	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	0.2573905452730122	TARLOXOTINIB	drugbank:DB14944	TARLOXOTINIB	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.7395446652914718	BTRX-335140	drugbank:DB16068	BTRX-335140	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	MUNDULONE	chembl:CHEMBL465339	MUNDULONE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	SIBUTRAMINE HYDROCHLORIDE	rxcui:1294535	SIBUTRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.065145994	APAP	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.4861821410712453	LISDEXAMFETAMINE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.035719504	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
UNIPROT:P30988	hgnc:1440	CALCR	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	CALCITONIN	rxcui:1311287	CALCITONIN	TRUE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:763	iuphar.ligand:763	[125I]CCL3 (HUMAN)	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006756874	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:12461	drugbank:DB03823	EPIGALLOCATECHIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.012430793	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013825085	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.1944728564284981	Rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	CYSTEAMINE HYDROCHLORIDE	rxcui:1426886	CYSTEAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	0.3804903712731485	CILOFEXOR	ncit:C169848	CILOFEXOR	FALSE	FALSE	FALSE
STAT1	hgnc:11362	STAT1	DTC	9/2/20	NULL	8.751278539282415	GUTTIFERONE K	chembl:CHEMBL388529	GUTTIFERONE K	FALSE	FALSE	FALSE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	1.250182648468916	ASCIMINIB HYDROCHLORIDE	rxcui:2584303	ASCIMINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.2169738480813822	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.093098708	THIABENDAZOLE	rxcui:10450	THIABENDAZOLE	TRUE	FALSE	FALSE
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	3.580068493342807	Suvorexant	rxcui:1547099	SUVOREXANT	TRUE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	1.875273972703375	ENRASENTAN	ncit:C87727	ENRASENTAN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	ETHYL ANTHRANILATE	rxcui:2396756	ETHYL ANTHRANILATE	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1442518440541057	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.729273212	DIC10	ncit:C29869	SN-1,2-DIDECANOYLGLYCEROL	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.6789785073581185	SNS-595	ncit:C95148	VOSAROXIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
RPS27A	hgnc:10417	RPS27A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.4907258993990139	BICIFADINE	ncit:C79930	BICIFADINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	GERALDOL	chembl:CHEMBL509256	GERALDOL	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.081533651	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1446492320542548	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
ERCC2	hgnc:3434	ERCC2	PharmGKB	4/5/24	NULL	0.1278595890479573	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.4375639269641208	indacaterol	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
NCBIGENE:2704	hgnc:29489	KMT5A	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:7022	iuphar.ligand:7022	NAHUOIC ACID A	FALSE	FALSE	FALSE
CDC42	hgnc:1736	CDC42	DTC	9/2/20	NULL	8.751278539282415	ZU-0073945	chembl:CHEMBL563777	CHEMBL:CHEMBL563777	FALSE	FALSE	FALSE
CERKL	hgnc:21699	CERKL	PharmGKB	4/5/24	NULL	5.000730593875666	iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	KETOTIFEN	rxcui:11404	KETOTIFEN FUMARATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	PHENMEDIPHAM	chembl:CHEMBL1079421	PHENMEDIPHAM	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	2.282942227638891	TPX-0131	chembl:CHEMBL4802183	TPX-0131	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	TELMISARTAN	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.092199598	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.6	hgnc:10596	SCN8A	TTD	2020.06.01	NULL	0.8899605294185507	XEN901	iuphar.ligand:11734	ZANDATRIGINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	CROMOLYN	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 2	hgnc:6871	MAPK1	TTD	2020.06.01	NULL	0.180026301	GDC-0994	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.145450613	IUPHAR.LIGAND:2147	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.1495945049449985	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.020025809	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.1232574442152452	AMINOQUINOL	ncit:C73273	AMINOQUINOL	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.004051518	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.1111273465305703	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.017352172	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:P49721	hgnc:9539	PSMB2	TdgClinicalTrial	Jan-14	NULL	0.546954909	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ONCOTROPHOBLAST GLYCOPROTEIN 5T4	hgnc:12004	TPBG	TTD	2020.06.01	NULL	1.312691780892362	PF-06263507	chembl:CHEMBL4297804	PF-06263507	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:190	iuphar.ligand:190	SB 215505	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.080781033	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.2907401508067248	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
E2F2	hgnc:3114	E2F2	ChEMBL	33	inhibitor	1.312691780892362	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1232574442152452	GNF-PF-308	chembl:CHEMBL600334	CHEMBL:CHEMBL600334	FALSE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1872	iuphar.ligand:1872	PRRP-20	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.034912015	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.03505185	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1040580087905162	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006909813	felodipine	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	DTC	9/2/20	NULL	1.029562181092048	6BIO	chembl:CHEMBL409450	6BIO	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.1159109740302306	ONYX-015	ncit:C2830	LONTUCIREV	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	NCI	14-Sep-17	NULL	0.1458546423213736	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.037721028	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	NCI	14-Sep-17	NULL	1.419126249613364	VITAMIN-B12	ncit:C939	COBALAMIN	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	positive modulator	0.3977853881492007	TAK-653	drugbank:DB16304	TAK-653	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001365893	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.015625733	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.002951527	fentanyl	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	0.3000438356325399	VILDAGLIPTIN	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	3.750547945	Hydroflumethiazide	rxcui:5495	HYDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	NSC-339578	chembl:CHEMBL353764	CHEMBL:CHEMBL353764	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	1.090323227845022	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	CONTEZOLID ACEFOSAMIL	ncit:C169864	CONTEZOLID ACEFOSAMIL	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.4102161815288632	GNF-PF-5007	chembl:CHEMBL1989853	CHEMBL:CHEMBL1989853	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.021215221	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.033615667	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:11713	iuphar.ligand:11713	&BETA;-SECRETASE INHIBITOR IV	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	LIDOCAINE HYDROCHLORIDE	rxcui:142440	LIDOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	1.141471113819445	PF-04634817	drugbank:DB14955	PF-04634817	FALSE	FALSE	FALSE
CUL4A	hgnc:2554	CUL4A	ChEMBL	33	inhibitor	1.009762908	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	inhibitor	0.1591141552596802	AVEXITIDE	ncit:C133230	AVEXITIDE	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1154649175056503	BUPROPION	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.105015342	NALED	chembl:CHEMBL1887067	NALED	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	CARNOSIC ACID	chembl:CHEMBL484853	CARNOSIC ACID	FALSE	FALSE	FALSE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	0.3182283105193606	6-THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.058406753	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
SMOX	hgnc:15862	SMOX	NCI	14-Sep-17	NULL	2.917092846427472	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.033487035	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	RACEPINEPHRINE HYDROCHLORIDE	rxcui:314610	RACEPINEPHRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TLK2	hgnc:11842	TLK2	CIViC	10-Apr-24	NULL	6.563458904461812	GF109203X	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.014488872	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.09741683	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
MICA	hgnc:7090	MICA	PharmGKB	4/5/24	NULL	1.071585127259071	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	PharmGKB	4/5/24	NULL	0.6563458904461812	donepezil	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	MADOLIN A	chembl:CHEMBL1224785	MADOLIN A	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.1356787370431382	INDACATEROL	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	1.944728564284981	DI-Leu16-IL2	chembl:CHEMBL4650391	DI-LEU16-IL2	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.1060761035064535	EFINOPEGDUTIDE	ncit:C169932	EFINOPEGDUTIDE	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.1223955040459079	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.013071365	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.081030357	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
PSME1	hgnc:9568	PSME1	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	activator	0.8751278539282418	IUPHAR.LIGAND:2794	iuphar.ligand:2794	PHOSPHATIDYL (3,5) INOSITOL BISPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2257	iuphar.ligand:2257	PACAP-27	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.064190307	Lomustine	rxcui:6466	LOMUSTINE	TRUE	FALSE	TRUE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	agonist	0.054355767	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	NSC-119915	chembl:CHEMBL1481974	CHEMBL:CHEMBL1481974	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	NSC-280795	chembl:CHEMBL84281	CHEMBL:CHEMBL84281	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.400821918	Betamethasone Valerate	rxcui:227897	BETAMETHASONE VALERATE	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	NCI	14-Sep-17	NULL	0.145450613	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	(E)-DIBENZYLIDENEACETONE	chembl:CHEMBL17201	CHEMBL:CHEMBL17201	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:12574	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:11411	iuphar.ligand:11411	EDAXETERKIB	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	NORDEFRIN	ncit:C81340	NORDEFRIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.2853677784548614	1-PHYTEN-3-OL	chembl:CHEMBL453797	CHEMBL:CHEMBL453797	FALSE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.9376369863516875	ILAPRAZOLE	ncit:C65887	ILAPRAZOLE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.029987248	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	EPALRESTAT	ncit:C72762	EPALRESTAT	FALSE	FALSE	FALSE
CD74	hgnc:1697	CD74	PharmGKB	4/5/24	NULL	1.312691780892362	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
UNIPROT:Q15116	hgnc:8760	PDCD1	TdgClinicalTrial	Jan-14	NULL	0.2561349816375342	MDX-1106	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.5097832158805291	IUPHAR.LIGAND:12768	drugbank:DB15137	VK-2809	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	ChEMBL	33	inhibitor	0.072927321	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.008500513	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11563	iuphar.ligand:11563	PSEUDOCHELERYTHRINE	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:10143	iuphar.ligand:10143	SR1001	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.1595977849109255	IUPHAR.LIGAND:2054	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.1428780169678761	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.023716202	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.056459862	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.06697407	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DILAZEP	ncit:C65389	DILAZEP	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	MECAMYLAMINE	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	DILTIAZEM MALATE	rxcui:81999	DILTIAZEM MALATE	TRUE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.9546849315580819	MILTIRONE	chembl:CHEMBL45830	MILTIRONE	FALSE	FALSE	FALSE
UNIPROT:Q14432	hgnc:8778	PDE3A	TdgClinicalTrial	Jan-14	NULL	0.596678082	NM-702	drugbank:DB05505	NM-702	FALSE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	modulator	0.2019525816757481	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
TNFRSF10A	hgnc:11904	TNFRSF10A	ChEMBL	33	agonist	42.00613698855559	MAPATUMUMAB	ncit:C61502	MAPATUMUMAB	FALSE	TRUE	TRUE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.044347695	IUPHAR.LIGAND:2404	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1682938180631233	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	0.2381300282797936	ANTITHROMBIN ALFA	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
KCND3	hgnc:6239	KCND3	ChEMBL	33	blocker	0.1562728310586145	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.06466462	DEHYDROEQUOL	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:7643	iuphar.ligand:7643	AEE788	FALSE	FALSE	TRUE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6092	iuphar.ligand:6092	GALANIN(3-29) (RAT/MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:2740	hgnc:4324	GLP1R	GuideToPharmacology	2024.1	NULL	0.1591141552596802	IUPHAR.LIGAND:12842	iuphar.ligand:12842	SMD-3040	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	NCI	14-Sep-17	NULL	0.1495945049449985	MOXIFLOXACIN	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
SMAD2	hgnc:6768	SMAD2	NCI	14-Sep-17	NULL	0.8204323630577265	BLM	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.2019525816757481	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.090219366	IUPHAR.LIGAND:474	iuphar.ligand:474	MRS1523	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	GO-Y034	chembl:CHEMBL595816	CHEMBL:CHEMBL595816	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.2333674277141977	TOBRAMYCIN	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	agonist	0.6482428547616604	SIPONIMOD	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
PDE10A	hgnc:21160	LINC00473	ChEMBL	33	inhibitor	4.375639269641208	MARDEPODECT	ncit:C170150	MARDEPODECT	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	TCMDC-124573	chembl:CHEMBL525826	CHEMBL:CHEMBL525826	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	GNF-PF-5251	chembl:CHEMBL576404	CHEMBL:CHEMBL576404	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	EHNA	iuphar.ligand:5179	EHNA	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.1519026168824334	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.1367387271762877	ZUCLOPENTHIXOL	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.042073455	IUPHAR.LIGAND:8473	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.072125922	IUPHAR.LIGAND:2693	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1250182648468916	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
TBX21	hgnc:11599	TBX21	NCI	14-Sep-17	NULL	2.187819634820604	DXM	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.1495945049449985	moxifloxacin	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	9.546849315580817	LGD-4665	ncit:C152703	TOTROMBOPAG	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.3125456621172291	DOVRAMILAST	ncit:C189964	DOVRAMILAST	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.4526523382387456	PEFLOXACIN	rxcui:7960	PEFLOXACIN	TRUE	FALSE	FALSE
CBR3	hgnc:1549	CBR3	PharmGKB	4/5/24	NULL	0.108040476	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.053038052	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:293	iuphar.ligand:293	NNC 11-1607	FALSE	FALSE	FALSE
UNIPROT:Q13003	hgnc:4581	GRIK3	TdgClinicalTrial	Jan-14	NULL	1.666910197958555	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TEND	1-Aug-11	NULL	2.763561643983921	BIVALIRUDIN	rxcui:60819	BIVALIRUDIN	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	DIPHENOXYLATE HYDROCHLORIDE	rxcui:82005	DIPHENOXYLATE HYDROCHLORIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.016491103	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
UNIPROT:Q13421	hgnc:7371	MSLN	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	SS1(DSFV)-PE38	drugbank:DB17579	SS1(DSFV)-PE38	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004961042	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.28382525	GOSSYPETIN	chembl:CHEMBL253570	GOSSYPETIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.034773292	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	XANTHURENATE	chembl:CHEMBL312535	XANTHURENATE	FALSE	FALSE	FALSE
UNIPROT:Q9P0X4	hgnc:1396	CACNA1I	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	PARAMETHADIONE	rxcui:32894	PARAMETHADIONE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.036847489	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.007906591	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.3125456621172291	DROTAVERINE	rxcui:23684	DROTAVERIN	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:2407	rxcui:1012892	FINGOLIMOD	TRUE	TRUE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	2,3,4,4'-TETRAMETHOXYBIPHENYL	chembl:CHEMBL28250	2,3,4,4'-TETRAMETHOXYBIPHENYL	FALSE	FALSE	FALSE
GTPASE KRAS	hgnc:6407	KRAS	TTD	2020.06.01	NULL	0.546954909	AZD4785	ncit:C147521	CET KRAS ANTISENSE OLIGONUCLEOTIDE AZD4785	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	RETINAL	iuphar.ligand:2350	ALL-TRANS-RETINAL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.002832129	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	SJ000032150	chembl:CHEMBL607140	CHEMBL:CHEMBL607140	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.3405902999072075	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.014732792	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	3-HYDROXYFLAVONOL	chembl:CHEMBL242172	CHEMBL:CHEMBL242172	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GROSSHEIMIN	iuphar.ligand:12468	GROSHEIMIN	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1280674908187671	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	JWH-015	iuphar.ligand:5558	JWH015	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Berubicin	ncit:C83552	BERUBICIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2035181055647073	FENOTEROL HBR	chembl:CHEMBL537445	FENOTEROL HBR	FALSE	FALSE	FALSE
KCNK3	hgnc:6278	KCNK3	ChEMBL	33	potentiator	0.2083637747448194	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	AZD-7624	chembl:CHEMBL9960	AZD-7624	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.7134194461371536	PEFICITINIB	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	1.372749574789398	DULIGOTUZUMAB	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:4324	iuphar.ligand:4324	TNP-ATP	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.042619863	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	PHENOXYBENZAMINE	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
CDH1	hgnc:1748	CDH1	NCI	14-Sep-17	NULL	0.750109589	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	3.500511415712966	BI-44370	chembl:CHEMBL3334624	BI-44370	FALSE	FALSE	FALSE
NCBIGENE:2843	hgnc:4475	GPR20	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8317	ncit:C174675	AZELIRAGON	FALSE	FALSE	FALSE
PB1	hgnc:30064	PBRM1	ChEMBL	33	inhibitor	1.381780822	FAVIPIRAVIR	ncit:C81605	FAVIPIRAVIR	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.3125456621172291	CHF4227	chembl:CHEMBL3545355	CHF4227	FALSE	FALSE	FALSE
RPL12	hgnc:10302	RPL12	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	3.281729452230906	HENAGLIFLOZIN	drugbank:DB11939	HENAGLIFLOZIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.1023541349623674	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	NXN-188	drugbank:DB06096	NXN-188	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	CGP-53353	iuphar.ligand:5163	CGP53353	FALSE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.4773424657790409	PROTEASE INHIBITOR	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	GNF-PF-4803	chembl:CHEMBL585240	CHEMBL:CHEMBL585240	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.022839352	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.03409589	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1544343271638073	CLINDAMYCIN PALMITATE HYDROCHLORIDE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.1479089330582944	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.1422972120208523	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.048260727	IUPHAR.LIGAND:142	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	antibody	1.544343271638073	IUPHAR.LIGAND:9614	iuphar.ligand:9614	CROTEDUMAB	FALSE	FALSE	FALSE
NCBIGENE:2136	hgnc:16059	PAK4	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8937	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.073746729	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
CTSL1	hgnc:2537	CTSL	NCI	14-Sep-17	NULL	0.5966780822238011	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.028199609	POLATUZUMAB VEDOTIN	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.074797252	MILTEFOSINE	rxcui:1494066	MILTEFOSINE	TRUE	FALSE	FALSE
SVEP1	hgnc:15985	SVEP1	PharmGKB	4/5/24	NULL	11.66837138570989	ticagrelor	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	CARDIODILATIN	drugbank:DB15591	ATRIAL NATRIURETIC PEPTIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
NCBIGENE:2788	hgnc:4410	GNG7	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:7708	iuphar.ligand:7708	AZD4877	FALSE	FALSE	TRUE
NCBIGENE:2200	hgnc:3603	FBN1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8249	iuphar.ligand:8249	RN486	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.008641816	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	MADOLIN A	chembl:CHEMBL1224785	MADOLIN A	FALSE	FALSE	FALSE
CYP51	hgnc:2649	CYP51A1	ChEMBL	33	inhibitor	17.50255707856483	ISAVUCONAZONIUM SULFATE	rxcui:1608321	ISAVUCONAZONIUM SULFATE	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.2333674277141978	APREMILAST	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	SOFALCONE	ncit:C81118	SOFALCONE	FALSE	FALSE	FALSE
NCBIGENE:522	hgnc:847	ATP5PF	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:1136	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:12115	iuphar.ligand:12115	COMPOUND 15 [PMID: 35034442]	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1325951293830669	NSC-695801	chembl:CHEMBL461193	CHEMBL:CHEMBL461193	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	0.3804903712731485	NIDUFEXOR	ncit:C174657	NIDUFEXOR	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.9512259281828714	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.052090944	QUINACRINE DIHYDROCHLORIDE	chembl:CHEMBL554190	QUINACRINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	NORFLOXACIN	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.089501712	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.040515178	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	ChEMBL	33	inhibitor	0.091159151	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	0.3281729452230906	IUPHAR.LIGAND:3633	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	GLIQUIDONE	rxcui:25793	GLIQUIDONE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	ChEMBL	33	inhibitor	0.4102161815288632	SNDX-5613	chembl:CHEMBL4650278	SNDX-5613	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.3182283105193606	CHIGLITAZAR	iuphar.ligand:12287	CHIGLITAZAR	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.017386646	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009579944	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-124280	chembl:CHEMBL528492	CHEMBL:CHEMBL528492	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.059667808	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.028444026	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.024920584	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	SJ000170251	chembl:CHEMBL603154	CHEMBL:CHEMBL603154	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.053579256	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003313623	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.014638325	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P17342	hgnc:7945	NPR3	TEND	1-Aug-11	NULL	6.563458904461812	NESIRITIDE	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TEND	1-Aug-11	NULL	0.069332312	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.024582243	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
NCBIGENE:2821	hgnc:4458	GPI	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7829	iuphar.ligand:7829	PF-04620110	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.056826484	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:11946	iuphar.ligand:11946	AZD9574	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	Tunlametinib	ncit:C173437	TUNLAMETINIB	FALSE	FALSE	TRUE
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	1.544343271638073	Trifarotene	rxcui:2205637	TRIFAROTENE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.3125456621172291	MELEVODOPA	ncit:C83927	MELEVODOPA	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008681824	RIFAMPICIN	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004340912	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	DTC	9/2/20	NULL	3.750547945	BERKELEYAMIDE C	chembl:CHEMBL468641	BERKELEYAMIDE C	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.004158694	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
IGFBP5	hgnc:5474	IGFBP5	NCI	14-Sep-17	NULL	2.500365296937833	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Sarizotan	ncit:C77567	SARIZOTAN	FALSE	FALSE	FALSE
KCNH8	hgnc:18864	KCNH8	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	inhibitor	0.3409589041278864	TEDATIOXETINE	ncit:C152535	TEDATIOXETINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1861974157294131	2,4-DIACETYL PHLOROGLUCINOL	chembl:CHEMBL276139	2,4-DIACETYLPHLOROGLUCINOL	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	modulator	0.046965717	ATAGABALIN	ncit:C169790	ATAGABALIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.6019397937072561	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:Q96EB6	hgnc:14929	SIRT1	TdgClinicalTrial	Jan-14	NULL	0.9053046764774912	SEN0014196	ncit:C152325	SELISISTAT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:3854	ncit:C175100	ITURELIX	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1136529680426287	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
PTBP1	hgnc:9583	PTBP1	DTC	9/2/20	NULL	0.2822993077187876	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001210747	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	SJ000018309	chembl:CHEMBL591363	CHEMBL:CHEMBL591363	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	0.1767935058440892	GOSERELIN ACETATE	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.1286952726365061	CARPHENAZINE MALEATE	ncit:C65289	CARPHENAZINE MALEATE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.5250767123569451	TUBOCURARINE CHLORIDE	rxcui:82115	TUBOCURARINE CHLORIDE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.011502228	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.051143836	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:639	iuphar.ligand:639	T-KININ	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9050	iuphar.ligand:9050	JNJ40355003	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:7393	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	2-STYRYL-QUINOLINE	chembl:CHEMBL127579	CHEMBL:CHEMBL127579	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.2461297089173179	KETOROLAC	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-2383	chembl:CHEMBL578915	CHEMBL:CHEMBL578915	FALSE	FALSE	FALSE
L-SELECTIN	hgnc:10720	SELL	TTD	2020.06.01	NULL	23.33674277141977	GMI-1070	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MENADIONE SODIUM BISULPHITE	chembl:CHEMBL2358118	MENADIONE SODIUM BISULPHITE	FALSE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	2.051080907644316	TADALAFIL	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	(S)-ROSCOVITINE	chembl:CHEMBL133342	(S)-ROSCOVITINE	FALSE	FALSE	FALSE
NCBIGENE:2366	hgnc:3874	FRA1G	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:8668	iuphar.ligand:8668	FURIN INHIBITOR PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:341	iuphar.ligand:341	ALCURONIUM	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:9537	iuphar.ligand:9537	ATRACURIUM	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9136	iuphar.ligand:9136	SB-674042	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.009471081	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	0.1342907192728759	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.012466209	tetracycline	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	CLEMIZOLE	ncit:C81139	CLEMIZOLE	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.1293292394967845	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
SRMS	hgnc:11298	SRMS	DTC	9/2/20	NULL	0.063722902	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	0.6721614540713904	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.037721028	Idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.086219493	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
UNIPROT:Q02156	hgnc:9401	PRKCE	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.048083948	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:605	iuphar.ligand:605	APELIN-13	FALSE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:8061	iuphar.ligand:8061	MK-5108	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:8473	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:2586	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1516	iuphar.ligand:1516	PYY-(13-36) (MOUSE, RAT, PIG)	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.017739078	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.2019525816757481	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
CA1	hgnc:1368	CA1	DTC	9/2/20	NULL	1.969037671338543	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
SOMATOTROPIN	hgnc:4261	GH1	TTD	2020.06.01	NULL	4.375639269641208	ACP-001	chembl:CHEMBL4297687	ACP-001	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.020328173	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	1-AMINOCYCLOPROPANE CARBOXYLIC ACID	chembl:CHEMBL265325	1-AMINOCYCLOPROPANE CARBOXYLIC ACID	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	3.500511415712966	PEXELIZUMAB	ncit:C95792	PEXELIZUMAB	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.4039051633514961	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.069454592	TARLOXOTINIB	drugbank:DB14944	TARLOXOTINIB	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.055681518	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.4565884455277782	Conteltinib	ncit:C169863	CONTELTINIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CHLOROPHACINONE	chembl:CHEMBL1874081	CHLOROPHACINONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	BUFOGENIN	ncit:C77829	BUFOGENIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	ARUNDINE	chembl:CHEMBL446452	ARUNDINE	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.4039051633514962	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P04070	hgnc:9451	PROC	TEND	1-Aug-11	NULL	15.75230137070834	SODIUM TETRADECYL SULFATE	rxcui:9913	SODIUM TETRADECYL SULFATE	TRUE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.8334550989792776	IL-4	iuphar.ligand:4996	IL-4	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.062065805	N-METHYL-D-ASPARTIC ACID (NMDA)	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	FLUVOXAMINE	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.019799273	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	0.2857560339357523	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:12387	iuphar.ligand:12387	ZONGERTINIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PROADIFEN HYDROCHLORIDE	ncit:C66468	PROADIFEN HYDROCHLORIDE	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	0.2287915957982331	Diacerein	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.1752202599633854	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.010569177	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	1.458546423213736	TRABODENOSON	ncit:C152705	TRABODENOSON	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00263434	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.014441054	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.4234489615781814	TRIPROLIDINE	rxcui:10849	TRIPROLIDINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.061197752	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.016246185	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	TCMDC-125738	chembl:CHEMBL527585	CHEMBL:CHEMBL527585	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.005403136	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:8382	iuphar.ligand:8382	VS-5584	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.018301733	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	ALPHA-NAPHTHOFLAVONE	drugbank:DB07453	ALPHA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.3684748858645228	ANTICONVULSANT	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	DIETHYLCARBAMAZINE CITRATE	rxcui:203175	DIETHYLCARBAMAZINE CITRATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012763168	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01495945	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
ATP1B1	hgnc:804	ATP1B1	ChEMBL	33	inhibitor	0.2763561643983921	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	6.300920548	TG-0054	ncit:C88323	BURIXAFOR	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:5964	iuphar.ligand:5964	EGFR/ERBB-2 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2024	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:8070	iuphar.ligand:8070	P505-15	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003053304	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	GLYCINE	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
NCBIGENE:959	hgnc:11935	CD40LG	GuideToPharmacology	2024.1	inhibitor	0.3621218705909966	IUPHAR.LIGAND:7596	ncit:C77944	DEXPROPRANOLOL	FALSE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	2.917092846427472	CD22 CAR-T	ncit:C128556	ANTI-CD22 CAR-EXPRESSING T LYMPHOCYTES	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	ChEMBL	33	inhibitor	0.7721716358190367	HYDROXYCHLOROQUINE SULFATE	rxcui:153972	HYDROXYCHLOROQUINE SULFATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	MERADIMATE	rxcui:91324	MERADIMATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	METHYLEPHEDRINE	rxcui:1739004	METHYLEPHEDRINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	PINOSYLVIN METHYL ETHER	chembl:CHEMBL186366	PINOSYLVIN METHYL ETHER	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.01036063	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1029562181092049	IPA-3	iuphar.ligand:8940	IPA-3	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	antibody	3.443125982668491	MEDI-575	ncit:C82684	TOVETUMAB	FALSE	TRUE	TRUE
EPAS1	hgnc:3374	EPAS1	DTC	9/2/20	NULL	8.751278539282415	PUUPEHENONE	chembl:CHEMBL157844	PUUPEHENONE	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11145	iuphar.ligand:11145	COMPOUND 55 [PMID: 30889352]	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1556551518844698	CARPHENAZINE	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	1.826353782111113	Ambrisentan	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
NCBIGENE:2388	hgnc:3900	FRA4A	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:7343	rxcui:1665684	EVOLOCUMAB	TRUE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:8184	iuphar.ligand:8184	COMPOUND 32 [PMID: 20471253]	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1861974157294131	CALYCOSIN	chembl:CHEMBL241608	CALYCOSIN	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	2.100306849	Tetrabenazine	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	8.751278539282415	BMS-833923	drugbank:DB16844	BMS-833923	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.1367387271762877	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	modulator	1.875273972703375	MIROGABALIN BESYLATE	ncit:C175142	MIROGABALIN BESYLATE	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.1981421556063943	IUPHAR.LIGAND:5509	rxcui:7247	NAPHAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.2917092846427472	IUPHAR.LIGAND:4167	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.2143170254518142	IUPHAR.LIGAND:10402	iuphar.ligand:10402	ZAK INHIBITOR 6P	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:2075	iuphar.ligand:2075	[125I]TYR7-SST3-ODN-8	FALSE	FALSE	FALSE
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1	hgnc:2357	CRHR1	TTD	2020.06.01	NULL	2.917092846427472	Telavancin	rxcui:473837	TELAVANCIN	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.2651902587661338	PLERIXAFOR	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
CHRM5	hgnc:1954	CHRM5	DTC	9/2/20	NULL	0.5147810905460245	VU0119498	iuphar.ligand:7632	VU0119498	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00347273	ESCITALOPRAM	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	GNF-PF-1083	chembl:CHEMBL530361	CHEMBL:CHEMBL530361	FALSE	FALSE	FALSE
DUSP1	hgnc:3064	DUSP1	NCI	14-Sep-17	NULL	0.2692701089009974	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.056826484	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.014206621	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006419031	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	NS-398	drugbank:DB14060	NS-398	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	GLYCINE	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
APOA5	hgnc:17288	APOA5	PharmGKB	4/5/24	NULL	0.630092055	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.3182283105193606	GS 6201	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	3,3',5,5'-TETRABROMOBISPHENOL A	chembl:CHEMBL184450	CHEMBL:CHEMBL184450	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.064033745	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.5556367326528517	PENICILLAMINE	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1852122442176172	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.1389091831632129	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1704794520639432	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
CDK5R1	hgnc:1775	CDK5R1	DTC	9/2/20	NULL	1.500219178	DNDI1417165	chembl:CHEMBL1406948	CHEMBL:CHEMBL1406948	FALSE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.2917092846427472	sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
TSPO	hgnc:1158	TSPO	ChEMBL	33	agonist	1.381780822	EMAPUNIL	ncit:C82906	EMAPUNIL	FALSE	FALSE	FALSE
CRTC2	hgnc:27301	CRTC2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.458546423213736	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	1.280674908	GRC-15300	chembl:CHEMBL3707319	GRC-15300	FALSE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.2536602475154323	oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.006210251	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.025929714	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003501912	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	3.750547945	HYDROFLUMETHIAZIDE	rxcui:5495	HYDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.025439763	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	OCTAVERINE	ncit:C90894	OCTAVERINE	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.2273059360852575	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.2631963470460877	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.030616718	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1040580087905162	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.052798061	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	FENDILINE HYDROCHLORIDE	rxcui:236767	FENDILINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	SJ000079774	chembl:CHEMBL601192	CHEMBL:CHEMBL601192	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.019233579	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
RPS3A	hgnc:10421	RPS3A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL10	hgnc:10298	RPL10	ChEMBL	33	modulator	0.1067229090156392	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	0.1530835896084387	AM-101	chembl:CHEMBL2364609	ESKETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00575742	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	1.019566431761058	VIA-3196	ncit:C170368	RESMETIROM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	SALSALATE	rxcui:36108	SALSALATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	BROMOCRIPTINE MESYLATE	rxcui:142426	BROMOCRIPTINE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:575	hgnc:943	ADGRB1	GuideToPharmacology	2024.1	blocker	5.250767124	IUPHAR.LIGAND:2344	iuphar.ligand:2344	BA2+	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.3547815624033412	IUPHAR.LIGAND:7393	rxcui:1490468	TASIMELTEON	TRUE	FALSE	FALSE
NCBIGENE:597	hgnc:991	BCL2A1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:8901	iuphar.ligand:8901	SR9009	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.080781033	HYDROGEN PEROXIDE	rxcui:5499	HYDROGEN PEROXIDE	TRUE	FALSE	FALSE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	0.7001022831425934	ANTIESTROGENIC	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.4773424657790409	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:1549	hgnc:2611	CYP2A7	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8128	iuphar.ligand:8128	COMPOUND 1A [PMID: 24900749]	FALSE	FALSE	FALSE
NCBIGENE:2684	ncbigene:2684	GGTL1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8979	iuphar.ligand:8979	GSK-J4	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	NELIVAPTAN	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.045579576	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
NCBIGENE:3264	hgnc:9281	PPP1CA	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:4735	iuphar.ligand:4735	MICROCYSTIN-LR	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2008	iuphar.ligand:2008	CST-17	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	1.105424657593568	AZD7762	iuphar.ligand:7713	AZD7762	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	BUTACLAMOL HYDROCHLORIDE	ncit:C81089	BUTACLAMOL HYDROCHLORIDE	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.2333674277141978	NCG-C00093820-01	chembl:CHEMBL544115	CHEMBL:CHEMBL544115	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.058799184	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
RIBONUCLEOTIDE REDUCTASE	hgnc:581	APBB1	TTD	2020.06.01	NULL	1.166837138570988	COH29	ncit:C114976	RNR INHIBITOR COH29	FALSE	FALSE	FALSE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	2.083637747448194	dantrolene	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.1166837138570988	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	THEONELLASTEROL C	chembl:CHEMBL1782599	THEONELLASTEROL C	FALSE	FALSE	FALSE
NCBIGENE:1466	hgnc:2470	CSRP2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8437	iuphar.ligand:8437	COMPOUND 101 [PMID: 21596927]	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	blocker	0.1693795846312726	IUPHAR.LIGAND:4128	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:4290	iuphar.ligand:4290	PREGNENOLONE SULPHATE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.021189536	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	BERGAPTEN	rxcui:15842	5-METHOXYPSORALEN	FALSE	FALSE	FALSE
NUMA1	hgnc:8059	NUMA1	PharmGKB	4/5/24	NULL	11.66837138570989	calcium channel blockers	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.039778539	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	SJ000032154	chembl:CHEMBL591876	CHEMBL:CHEMBL591876	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.3117023117067671	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.029170928	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
ACTIVATION B7-1 ANTIGEN	hgnc:1700	CD80	TTD	2020.06.01	NULL	2.187819634820604	HS-110	ncit:C61073	VIAGENPUMATUCEL-L	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	3.214755381777214	Coagulation Factor IX	wikidata:Q20801778	COAGULATION FACTOR IX	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	PharmGKB	4/5/24	NULL	0.026885648	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	2.634164108814105	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
BMP2	hgnc:1069	BMP2	DTC	9/2/20	NULL	26.25383561784724	BUTYL 4-ACETAMIDOBENZOATE	chembl:CHEMBL1321401	CHEMBL:CHEMBL1321401	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	DNDI1416924	chembl:CHEMBL156959	CHEMBL:CHEMBL156959	FALSE	FALSE	FALSE
CD80	hgnc:1700	CD80	PharmGKB	4/5/24	NULL	0.2500365296937833	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	THIPHENAMIL	rxcui:38150	THIPHENAMIL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	INDINAVIR	rxcui:114289	INDINAVIR	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	FUSARIC ACID	chembl:CHEMBL24510	FUSARIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	PROPIONYLPROMAZINE HYDROCHLORIDE	chembl:CHEMBL1256661	PROPIONYLPROMAZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.049864835	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.015299438	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.023151531	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.5527123287967842	RAPACURONIUM BROMIDE	rxcui:228530	RAPACURONIUM BROMIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.017859752	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1988926940746003	2-BROMO-HEXADECANOIC ACID	chembl:CHEMBL118417	CHEMBL:CHEMBL118417	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.015105774	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	0.2500365296937833	CERDULATINIB	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	modulator	0.1553481397505754	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DICHLORVOS	drugbank:DB11397	DICHLORVOS	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:7107	rxcui:149	ACEBUTOLOL	TRUE	FALSE	FALSE
NCBIGENE:1830	hgnc:3050	DSG3	GuideToPharmacology	2024.1	inhibitor	4.773424657790409	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5901	iuphar.ligand:5901	BMS COMPOUND 4C	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	TETRANITROMETHANE	chembl:CHEMBL261663	TETRANITROMETHANE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.025891357	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
CA12	hgnc:1371	CA12	PharmGKB	4/5/24	NULL	0.1704794520639432	topiramate	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
TBX21	hgnc:11599	TBX21	PharmGKB	4/5/24	NULL	0.8537832721251138	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	DERRUSTONE	chembl:CHEMBL252721	DERRUSTONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124312	chembl:CHEMBL528245	CHEMBL:CHEMBL528245	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.074797252	AZD7009	chembl:CHEMBL3545040	AZD7009	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.054243462	TETRACAINE HYDROCHLORIDE	rxcui:10391	TETRACAINE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	OncoKB	23-Jul-20	NULL	0.5672124979164529	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
OPN1LW	hgnc:9936	OPN1LW	DTC	9/2/20	NULL	21.00306849427779	CYCLOCITRAL	chembl:CHEMBL1952257	CYCLOCITRAL	FALSE	FALSE	FALSE
UNIPROT:P01138	hgnc:7808	NGF	TdgClinicalTrial	Jan-14	NULL	22.50328767	TANEZUMAB	ncit:C71522	TANEZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2937	hgnc:4624	GSS	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9562	iuphar.ligand:9562	PFK15	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.067664525	IUPHAR.LIGAND:414	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6114	iuphar.ligand:6114	GAL-B2-C14	FALSE	FALSE	FALSE
NCBIGENE:2681	hgnc:4253	GGTA1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8979	iuphar.ligand:8979	GSK-J4	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:3268	iuphar.ligand:3268	[11C]BUTYLTHIO-TZTP	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	modulator	1.312691780892362	IUPHAR.LIGAND:1026	iuphar.ligand:1026	SPINORPHIN	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	1.419126249613364	SSR240600	chembl:CHEMBL3544947	BURAPITANT	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.042898424	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1019566431761058	TDR77578	chembl:CHEMBL1364172	CHEMBL:CHEMBL1364172	FALSE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	MyCancerGenome	20-Jun-17	other/unknown	0.546954909	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.6177373086552295	SJ000040829	chembl:CHEMBL589711	CHEMBL:CHEMBL589711	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.004674828	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	DOMIPHEN BROMIDE	rxcui:49255	DOMIPHEN BROMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	TCMDC-123532	chembl:CHEMBL547833	CHEMBL:CHEMBL547833	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.4039051633514961	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	DIPHENADIONE	ncit:C75156	DIPHENADIONE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.5672124979164529	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	2.333674277141977	ANTICOAGULANT	ncit:C263	ANTICOAGULANT AGENT	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.015683295	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	IDAZOXAN HYDROCHLORIDE	chembl:CHEMBL543467	IDAZOXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	DOCONEXENT	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
KCNMB2	hgnc:6286	KCNMB2	PharmGKB	4/5/24	NULL	35.00511415712966	ritodrine	rxcui:9392	RITODRINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:307	iuphar.ligand:307	4-DAMP	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	ZOMEPIRAC SODIUM	rxcui:58331	ZOMEPIRAC SODIUM	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
NCBIGENE:1851	hgnc:9665	PTPRB	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8786	iuphar.ligand:8786	COMPOUND 13E [PMID: 16759857]	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1980	iuphar.ligand:1980	SQ-29548	FALSE	FALSE	FALSE
SYNE2	hgnc:17084	SYNE2	PharmGKB	4/5/24	NULL	1.29648571	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CINNAMALDEHYDE	rxcui:1368153	CINNAMIC ALDEHYDE	TRUE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	0.1372749574789398	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	TETRYDAMINE	ncit:C152580	TETRYDAMINE	FALSE	FALSE	FALSE
RPL23A	hgnc:10317	RPL23A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	0.2083637747448194	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	2.187819634820604	PEMTUMOMAB	drugbank:DB18563	PEMTUMOMAB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	TCMDC-125606	chembl:CHEMBL536166	CHEMBL:CHEMBL536166	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.4234489615781814	GNF-PF-3418	chembl:CHEMBL582099	CHEMBL:CHEMBL582099	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.1428780169678762	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
ITGA5	hgnc:6141	ITGA5	NCI	14-Sep-17	NULL	3.281729452230906	M-CSF	iuphar.ligand:4905	M-CSF	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.017751072	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CancerCommons	25-Jul-13	inhibitor	0.2778183663264258	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	CancerCommons	25-Jul-13	inhibitor	0.2275522047050683	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	4-DAMP	iuphar.ligand:307	4-DAMP	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	CGI	2/1/22	NULL	0.9883796938483671	Pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
ERBB4	hgnc:3432	ERBB4	CGI	2/1/22	NULL	0.1752202599633854	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	CGI	2/1/22	NULL	0.6250913242344582	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	AM-251	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	CGI	2/1/22	NULL	0.088396753	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
PTH1R	hgnc:9608	PTH1R	DTC	9/2/20	NULL	1.875273972703375	GNF-PF-5576	chembl:CHEMBL599896	CHEMBL:CHEMBL599896	FALSE	FALSE	FALSE
MLL2	hgnc:7133	KMT2D	CGI	2/1/22	NULL	2.625383561784725	Bicalutamide	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	CGI	2/1/22	NULL	0.017059022	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	0.6563458904461812	ACETAZOLAMIDE SODIUM	rxcui:91406	ACETAZOLAMIDE SODIUM	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	CGI	2/1/22	NULL	0.1131630845596864	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.062509132	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.070956312	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.074690855	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.7095631248066824	ACLIDINIUM BROMIDE	rxcui:1303097	ACLIDINIUM BROMIDE	TRUE	FALSE	FALSE
CYSLTR1	hgnc:17451	CYSLTR1	ChEMBL	33	inhibitor	1.325951293830669	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	5.000730593875666	STREPTOKINASE	rxcui:10106	STREPTOKINASE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.3062196950280639	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.9053046764774912	VALRUBICIN	rxcui:31435	VALRUBICIN	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.421837528	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	11.66837138570988	POLYTHIAZIDE	rxcui:8565	POLYTHIAZIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	PILOCARPINE NITRATE	rxcui:103244	PILOCARPINE NITRATE	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.095468493	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.5147810905460244	ELETRIPTAN HYDROBROMIDE	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1682938180631233	CARPHENAZINE MALEATE	ncit:C65289	CARPHENAZINE MALEATE	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.8078103267029924	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
GPBAR1	hgnc:19680	GPBAR1	DTC	9/2/20	NULL	1.093909817410302	URSODIOL	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1635752997996713	ESTROPIPATE	rxcui:33747	ESTROPIPATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.061340737	TRIMIPRAMINE MALEATE	rxcui:71532	TRIMIPRAMINE MALEATE	TRUE	FALSE	FALSE
GSR	hgnc:4623	GSR	ChEMBL	33	inhibitor	0.6509215442441467	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	potentiator	0.301335273	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.1434635826111871	NORETHINDRONE ACETATE	rxcui:31983	NORETHINDRONE ACETATE	TRUE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	0.2885036881082115	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	1.826353782111113	AMBRISENTAN	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	1.121958787087489	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.4930297768609811	NALBUPHINE HYDROCHLORIDE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.015429818	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	3.281729452230906	GINGKOLIC ACID	chembl:CHEMBL445177	GINGKOLIC ACID	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	negative modulator	0.2243917574174978	MEMANTINE HYDROCHLORIDE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	negative modulator	0.2160809515872201	MEMANTINE HYDROCHLORIDE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	negative modulator	0.094099769	MEMANTINE HYDROCHLORIDE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.040328473	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.2817943000126717	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1442518440541058	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.030246354	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2275522047050683	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	agonist	0.3889457128569963	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	agonist	0.1842374429322614	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1406455479527531	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.2365210416022275	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.095122593	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.069824031	DILTIAZEM HYDROCHLORIDE	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.061919424	DILTIAZEM HYDROCHLORIDE	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.08334551	VERAPAMIL HYDROCHLORIDE	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2191733444543002	ALBUTEROL SULFATE	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	LEVALBUTEROL HYDROCHLORIDE	rxcui:237159	LEVALBUTEROL	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.3256289689035318	FORMOTEROL FUMARATE	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	TERBUTALINE SULFATE	rxcui:10369	TERBUTALINE SULFATE	TRUE	FALSE	FALSE
PSMD1	hgnc:9554	PSMD1	ChEMBL	33	inhibitor	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA8	hgnc:22985	PSMA8	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB10	hgnc:9538	PSMB10	ChEMBL	33	inhibitor	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.3864200913449379	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1591141552596802	NELFINAVIR MESYLATE	rxcui:266565	NELFINAVIR MESYLATE	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.16256245	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.6250913242344582	ROCURONIUM BROMIDE	rxcui:32521	ROCURONIUM BROMIDE	TRUE	FALSE	FALSE
GLRB	hgnc:4329	GLRB	ChEMBL	33	positive modulator	0.1458546423213736	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
ATP1A1	hgnc:799	ATP1A1	ChEMBL	33	inhibitor	1.400204566285186	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
ATP1A3	hgnc:801	ATP1A3	ChEMBL	33	inhibitor	0.096521454	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.083257407	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.036925226	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.018990116	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.018521224	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	TRICLOFOS SODIUM	rxcui:104696	TRICLOFOS SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.016126435	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.013113804	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1544343271638073	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	blocker	0.1187956362798518	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	blocker	0.2243917574174979	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	blocker	0.2019525816757481	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	blocker	0.1262203635473425	BEPRIDIL HYDROCHLORIDE	rxcui:235752	BEPRIDIL HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNK18	hgnc:19439	KCNK18	ChEMBL	33	potentiator	0.3500511415712967	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
KCNK10	hgnc:6273	KCNK10	ChEMBL	33	potentiator	0.3500511415712967	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.057574201	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.039068208	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.052090944	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.027177884	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.038693936	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.023813003	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.054695491	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.057574201	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	PRILOCAINE	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.020226376	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.014206621	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	MERETHOXYLLINE PROCAINE	chembl:CHEMBL1200443	MERETHOXYLLINE PROCAINE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.047518255	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.069180068	CARPHENAZINE MALEATE	ncit:C65289	CARPHENAZINE MALEATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.041508041	LOXAPINE HYDROCHLORIDE	rxcui:91138	LOXAPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.017243899	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.028626235	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inverse agonist	0.006579909	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
KCNA6	hgnc:6225	KCNA6	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	ChEMBL	33	blocker	0.2344092465879218	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	ChEMBL	33	blocker	0.049723174	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.003116552	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCND2	hgnc:6238	KCND2	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNV1	hgnc:18861	KCNV1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCND3	hgnc:6239	KCND3	ChEMBL	33	blocker	0.1367387271762877	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCND1	hgnc:6237	KCND1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	ChEMBL	33	blocker	0.058212496	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCND1	hgnc:6237	KCND1	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	blocker	0.128067491	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNC3	hgnc:6235	KCNC3	ChEMBL	33	blocker	0.2134458180312784	GUANIDINE HYDROCHLORIDE	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNF1	hgnc:6246	KCNF1	ChEMBL	33	blocker	0.182318303	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.3704244884352345	IDELALISIB	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.042344896	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.1290114772375786	PANOBINOSTAT LACTATE	rxcui:1603349	PANOBINOSTAT LACTATE	TRUE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	1.093909817410302	PASIREOTIDE PAMOATE	rxcui:1597818	PASIREOTIDE PAMOATE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1562728310586145	IBCASERTIB	ncit:C115970	IBCASERTIB	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.2500365296937833	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1640864726115453	CM-082	chembl:CHEMBL3545427	CM-082	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.081030357	CM-082	chembl:CHEMBL3545427	CM-082	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.092443083	IBCASERTIB	ncit:C115970	IBCASERTIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1581556362520918	CM-082	chembl:CHEMBL3545427	CM-082	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1875273972703375	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.072927321	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1041818873724097	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.1093909817410302	ALTIRATINIB	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.050488145	GSK-1059615	drugbank:DB11962	GSK-1059615	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.150021918	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	1.831662950082366	LAROTRECTINIB	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.052090944	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1875273972703375	RECILISIB	ncit:C152168	RECILISIB	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.093763699	PANULISIB	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.2822993077187876	ABROCITINIB	rxcui:2591476	ABROCITINIB	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.1848861663228679	PWT-33579	chembl:CHEMBL3545323	PWT-33579	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	PS-516895	chembl:CHEMBL3545139	PS-516895	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.1093909817410302	XL-228	chembl:CHEMBL3545085	XL-228	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	agonist	1.750255707856483	SAR425899	chembl:CHEMBL3545269	SAR425899	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.3697723326457359	ZD-4190	chembl:CHEMBL281872	ZD-4190	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	inhibitor	2.282942227638891	SRX251	chembl:CHEMBL3545146	SRX251	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	2.019525817	TEDALINAB	ncit:C152534	TEDALINAB	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.2885036881082115	AZD6280	chembl:CHEMBL1783256	AZD6280	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	ChEMBL	33	inhibitor	4.039051633514961	RXDX-103	chembl:CHEMBL3545090	RXDX-103	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	2.763561643983921	RG7185	chembl:CHEMBL3544941	RG7185	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	ChEMBL	33	inhibitor	0.060008767	ULIXERTINIB	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1200175342530159	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1200175342530159	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1750255707856483	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1077080435603989	BUPARLISIB	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
INSR	hgnc:6091	INSR	ChEMBL	33	inhibitor	0.08334551	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.043756393	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	DE-104	chembl:CHEMBL3545153	DE-104	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	PELITINIB	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.3365876361262467	SAR-407899	iuphar.ligand:8910	SAR407899	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.760980743	TALMAPIMOD	ncit:C79841	TALMAPIMOD	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.1810609352954983	CANERTINIB DIHYDROCHLORIDE	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
PRKCH	hgnc:9403	PRKCH	ChEMBL	33	inhibitor	0.1325951293830669	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.01823183	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PRKCG	hgnc:9402	PRKCG	ChEMBL	33	inhibitor	0.1268301237577161	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PRKCZ	hgnc:9412	PRKCZ	ChEMBL	33	inhibitor	0.1215455352678113	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.8514757497680189	PRELADENANT	ncit:C76394	PRELADENANT	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	2.282942227638891	DARUSENTAN	ncit:C75991	DARUSENTAN	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.7095631248066824	OSEMOZOTAN	ncit:C91059	OSEMOZOTAN	FALSE	FALSE	FALSE
CALCR	hgnc:1440	CALCR	ChEMBL	33	agonist	6.563458904461812	SMC021	chembl:CHEMBL3545415	SMC021	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	ChEMBL	33	negative modulator	3.088686543276147	GEVOKIZUMAB	ncit:C97945	GEVOKIZUMAB	FALSE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	modulator	0.084146909	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	modulator	0.1262203635473425	IMAGABALIN	ncit:C83785	IMAGABALIN	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	agonist	0.05073205	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	agonist	0.055681518	GABOXADOL	ncit:C72791	GABOXADOL	FALSE	FALSE	FALSE
GDF2	hgnc:4217	GDF2	ChEMBL	33	inhibitor	1.093909817410302	DALANTERCEPT	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
KCNS1	hgnc:6300	KCNS1	ChEMBL	33	blocker	0.2187819634820604	TEDISAMIL	ncit:C72585	TEDISAMIL	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.1539814405738841	ESLICARBAZEPINE	rxcui:1482502	ESLICARBAZEPINE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.042689164	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.035719504	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.038894571	SAGOPILONE	ncit:C61072	SAGOPILONE	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.3977853881492007	ZONAMPANEL	ncit:C152963	ZONAMPANEL	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.8334550989792777	MATUZUMAB	ncit:C2012	MATUZUMAB	FALSE	FALSE	TRUE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.5645986154375752	PLACULUMAB	ncit:C170329	PLACULUMAB	FALSE	FALSE	FALSE
SELP	hgnc:10721	SELP	ChEMBL	33	inhibitor	5.250767123569449	RG-1512	chembl:CHEMBL2109487	RG-1512	FALSE	FALSE	FALSE
CALM1	hgnc:1442	CALM1	ChEMBL	33	inhibitor	1.750255707856483	BENZIODARONE	ncit:C74127	BENZIODARONE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	CLOMETACIN	ncit:C77348	CLOMETACIN	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.030598876	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.078682824	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.032252869	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.1339481409073839	MOXISYLYTE	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.2308029504865691	MOXISYLYTE	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.087222045	MOXISYLYTE	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
CCKAR	hgnc:1570	CCKAR	ChEMBL	33	inhibitor	2.625383561784724	PROGLUMIDE	rxcui:8730	PROGLUMIDE	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	2.072671233	XIMELAGATRAN	ncit:C77996	XIMELAGATRAN	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	TETRAZEPAM	rxcui:37985	TETRAZEPAM	TRUE	FALSE	FALSE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	8.751278539282415	TNX-650	chembl:CHEMBL2109466	TNX-650	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	1.265245090016735	AMG-191	chembl:CHEMBL2109325	AMG-191	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	ChEMBL	33	binder	2.917092846427472	BC8 131I	chembl:CHEMBL2109630	BC8 131I	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	positive modulator	0.4605936073306534	ALCURONIUM	rxcui:460	ALCURONIUM	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	0.6908904109959803	CANRENOATE POTASSIUM	rxcui:1981	CANRENOATE POTASSIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.03409589	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.033658764	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.032412143	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	DIBENZEPIN	rxcui:3332	DIBENZEPIN	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.028850369	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	1.500219178162699	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.023060023	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	AD-439	chembl:CHEMBL2109445	AD-439	FALSE	FALSE	FALSE
GPNMB	hgnc:4462	GPNMB	ChEMBL	33	binder	26.25383561784724	GLEMBATUMUMAB	ncit:C84520	GLEMBATUMUMAB	FALSE	FALSE	FALSE
RPS3A	hgnc:10421	RPS3A	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS13	hgnc:10386	RPS13	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS23	hgnc:10410	RPS23	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL15	hgnc:10306	RPL15	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL9P9	hgnc:30334	RPL9P8	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL9P8	hgnc:30334	RPL9P8	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL31	hgnc:10334	RPL31	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL35	hgnc:10344	RPL35	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL39	hgnc:10350	RPL39	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
HLA-DRB3	hgnc:4951	HLA-DRB3	ChEMBL	33	inhibitor	3.281729452230906	APOLIZUMAB	ncit:C2228	APOLIZUMAB	FALSE	FALSE	FALSE
RPL38	hgnc:10349	RPL38	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL36	hgnc:13631	RPL36	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	ChEMBL	33	inhibitor	0.6563458904461812	GLESATINIB	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
KCNQ1	hgnc:6294	KCNQ1	ChEMBL	33	blocker	0.056826484	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCND2	hgnc:6238	KCND2	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNA10	hgnc:6219	KCNA10	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNC3	hgnc:6235	KCNC3	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
KCNG1	hgnc:6248	KCNG1	ChEMBL	33	blocker	0.2083637747448194	AMIFAMPRIDINE	rxcui:2106338	AMIFAMPRIDINE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	TELINAVIR	ncit:C76911	TELINAVIR	FALSE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	CILUPREVIR	ncit:C76016	CILUPREVIR	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.023943307	EPHEDRINE SULFATE	rxcui:3966	EPHEDRINE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2983390411119005	DROTAVERINE	rxcui:23684	DROTAVERIN	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.007369498	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS24	hgnc:10411	RPS24	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL13	hgnc:10303	RPL13	ChEMBL	33	inhibitor	0.078958904	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL5	hgnc:10360	RPL5	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPS27A	hgnc:10417	RPS27A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL32	hgnc:10336	RPL32	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL30	hgnc:10333	RPL30	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL12	hgnc:10302	RPL12	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL7A	hgnc:10364	RPL7A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
RPL36A	hgnc:10359	RPL36A	ChEMBL	33	inhibitor	0.1105424657593568	CYCLOHEXIMIDE	ncit:C171712	CYCLOHEXIMIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	ALFLUTINIB	drugbank:DB16087	ALFLUTINIB	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1981421556063943	LERCANIDIPINE HYDROCHLORIDE	rxcui:153679	LERCANIDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2442217266776488	LERCANIDIPINE HYDROCHLORIDE	rxcui:153679	LERCANIDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	blocker	0.6250913242344582	TEGOPRAZAN	ncit:C152542	TEGOPRAZAN	FALSE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.8751278539282416	VERICIGUAT	rxcui:2475830	VERICIGUAT	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	TRANIMILAST	ncit:C171863	TRANIMILAST	FALSE	FALSE	FALSE
PMEL	hgnc:10880	PMEL	ChEMBL	33	binder	6.563458904461812	TEBENTAFUSP	rxcui:2590743	TEBENTAFUSP	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	LOTAMILAST	ncit:C170131	LOTAMILAST	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2983390411119005	DOVRAMILAST	ncit:C189964	DOVRAMILAST	FALSE	FALSE	FALSE
RPS12	hgnc:10385	RPS12	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	modulator	0.008537833	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL19	hgnc:10312	RPL19	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS29	hgnc:10419	RPS29	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL7	hgnc:10363	RPL7	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL5	hgnc:10360	RPL5	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL7A	hgnc:10364	RPL7A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS24	hgnc:10411	RPS24	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPS26	hgnc:10414	RPS26	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL9P7	hgnc:30335	RPL9P7	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL35A	hgnc:10345	RPL35A	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.2408608772279564	ORP-101	drugbank:DB16072	ORP-101	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	positive modulator	0.4234489615781814	TAK-653	drugbank:DB16304	TAK-653	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	1.166837138570988	NOMACOPAN	ncit:C167012	NOMACOPAN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.8751278539282416	EXATECAN	ncit:C66720	EXATECAN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.4375639269641208	MURELETECAN	ncit:C2234	MURELETECAN	FALSE	FALSE	FALSE
TRPM8	hgnc:17961	TRPM8	ChEMBL	33	inhibitor	5.527123287967842	ELISMETREP	ncit:C169937	ELISMETREP	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	DISTIGMINE	rxcui:3551	DISTIGMINE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.3621218705909965	ALVESPIMYCIN	ncit:C38142	ALVESPIMYCIN	FALSE	FALSE	TRUE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.5834185692854945	PENTAERYTHRITOL TETRANITRATE	rxcui:7992	PENTAERYTHRITOL TETRANITRATE	TRUE	FALSE	FALSE
SLC6A9	hgnc:11056	SLC6A9	ChEMBL	33	inhibitor	5.834185692854944	PF-03463275	drugbank:DB11993	PF-03463275	FALSE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.6177373086552295	PENTAERYTHRITOL TETRANITRATE	rxcui:7992	PENTAERYTHRITOL TETRANITRATE	TRUE	FALSE	FALSE
IL33	hgnc:16028	IL33	ChEMBL	33	inhibitor	13.12691780892362	ITEPEKIMAB	ncit:C174938	ITEPEKIMAB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	negative modulator	0.039068208	AGS-16C3F	drugbank:DB17551	AGS-16C3F	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	0.6000876712650799	PAMIPARIB	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.4015030085991933	FUTIBATINIB	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	3.088686543276147	PF-4191834	drugbank:DB11645	PF-4191834	FALSE	FALSE	FALSE
FASLG	hgnc:11936	FASLG	ChEMBL	33	binder	0.6908904109959803	ASUNERCEPT	ncit:C90562	ASUNERCEPT	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	binder	1.235474617310458	PACMILIMAB	ncit:C132192	PACMILIMAB	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	ChEMBL	33	inhibitor	0.2263261691193728	EDIFOLIGIDE SODIUM	ncit:C171738	EDIFOLIGIDE SODIUM	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	ChEMBL	33	inhibitor	0.057955487	APG115	chembl:CHEMBL4091801	APG115	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.069454592	SKLB1028	iuphar.ligand:12089	RUSERONTINIB	FALSE	FALSE	FALSE
MIF	hgnc:7097	MIF	ChEMBL	33	inhibitor	8.751278539282415	IMALUMAB	ncit:C104260	IMALUMAB	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	0.760980743	BMS-741672	iuphar.ligand:11598	BMS-741672	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.084012274	CHIGLITAZAR	iuphar.ligand:12287	CHIGLITAZAR	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	COCAINE HYDROCHLORIDE	rxcui:81985	COCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GCK	hgnc:4195	GCK	ChEMBL	33	activator	7.001022831425932	PF-04991532	drugbank:DB11765	PF-04991532	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.060772768	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.045226246	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1312691780892362	LORNOXICAM	rxcui:20890	LORNOXICAM	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.084553416	EPHEDRINE HYDROCHLORIDE	rxcui:91165	EPHEDRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.3621218705909966	DEXRAZOXANE	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	1.312691780892362	DEXRAZOXANE	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	BIVATUZUMAB MERTANSINE	chembl:CHEMBL2109288	BIVATUZUMAB MERTANSINE	FALSE	FALSE	FALSE
RSPO3	hgnc:20866	RSPO3	ChEMBL	33	inhibitor	52.50767123569449	ROSMANTUZUMAB	ncit:C122921	ROSMANTUZUMAB	FALSE	FALSE	FALSE
CPSF3	hgnc:2326	CPSF3	ChEMBL	33	inhibitor	52.50767123569449	ACOZIBOROLE	ncit:C166573	ACOZIBOROLE	FALSE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.729273212	ENOXIMONE	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.069180068	ONZIGOLIDE	ncit:C88345	ONZIGOLIDE	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.6403374540938354	PIMIVALIMAB	ncit:C157485	PIMIVALIMAB	FALSE	FALSE	FALSE
F8	hgnc:3546	F8	ChEMBL	33	positive modulator	3.088686543276147	ANTIHEMOPHILIC FACTOR, PEGYLATED (MW 20000) HUMAN SEQUENCE RECOMBINANT	ncit:C152106	ANTIHEMOPHILIC FACTOR, PEGYLATED (MW 20000) HUMAN SEQUENCE RECOMBINANT	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	ARX-788	chembl:CHEMBL4297892	ARX-788	FALSE	FALSE	FALSE
MPL	hgnc:7217	MPL	ChEMBL	33	agonist	4.773424657790408	RAFUTROMBOPAG	ncit:C188548	RAFUTROMBOPAG	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	ChEMBL	33	inhibitor	0.3697723326457359	TELAGLENASTAT	ncit:C114381	TELAGLENASTAT	FALSE	FALSE	FALSE
MYL3	hgnc:7584	MYL3	ChEMBL	33	inhibitor	1.944728564284981	MAVACAMTEN	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
MYL4	hgnc:7585	MYL4	ChEMBL	33	inhibitor	1.944728564284981	MAVACAMTEN	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
MYL2	hgnc:7583	MYL2	ChEMBL	33	inhibitor	1.944728564284981	MAVACAMTEN	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.080781033	XYLOMETAZOLINE	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
A2M	hgnc:7	A2M	ChEMBL	33	binder	0.6326225450083675	TECHNETIUM TC 99M SUCCIMER	chembl:CHEMBL1200797	TECHNETIUM TC 99M SUCCIMER	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	1.479089330582943	ORM-12741	drugbank:DB12057	ORM-12741	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.007188893	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.4734548598913698	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1541321073454828	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1396480617970598	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
CCNE1	hgnc:1589	CCNE1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.8751278539282416	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
CCND2	hgnc:1583	CCND2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3750547945406749	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1350505947420126	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
PGP	hgnc:8909	PGP	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2108741816694558	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
TLE3	hgnc:11839	TLE3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3163112725041837	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.218327115	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2465148884304905	AFURESERTIB HYDROCHLORIDE	ncit:C142902	AFURESERTIB HYDROCHLORIDE	FALSE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.015429818	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	4.118248724368196	CHEMBL2109402	chembl:CHEMBL2109402	MM-121	FALSE	TRUE	TRUE
FGFR4	hgnc:3691	FGFR4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.036038209	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4861821410712454	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.5114383561918295	BAY 869766	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2019525816757481	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
MAP2K1	hgnc:6840	MAP2K1	COSMIC	4-Sep-20	NULL	0.2678962818147679	PD0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	COSMIC	4-Sep-20	NULL	0.4906052389860809	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.039214094	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.068191781	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001886187	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	1.981421556063943	MULBERROFURAN H	chembl:CHEMBL563553	MULBERROFURAN H	FALSE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	DTC	9/2/20	NULL	0.4688184931758437	(R)-PIA	iuphar.ligand:414	(R)-PIA	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	0.577007376	SULFORAPHANE	ncit:C1424	SULFORAPHANE	FALSE	FALSE	FALSE
BMX	hgnc:1079	BMX	DTC	9/2/20	NULL	10.50153424713889	PD-168393	drugbank:DB07662	PD-168393	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.010586224	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.018699313	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	2-NITROFLUORENE	chembl:CHEMBL351487	2-NITROFLUORENE	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.026816992	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	DIPYRIDYL	chembl:CHEMBL39879	DIPYRIDYL	FALSE	FALSE	FALSE
GRM4	hgnc:4596	GRM4	DTC	9/2/20	NULL	3.750547945	N-(3,4-DIMETHOXYPHENYL)PICOLINAMIDE	chembl:CHEMBL572346	CHEMBL:CHEMBL572346	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	BRILLIANT GREEN OXALATE	chembl:CHEMBL1789985	BRILLIANT GREEN OXALATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-4364	chembl:CHEMBL528647	CHEMBL:CHEMBL528647	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.01535312	PHENYLMERCURIC ACETATE	rxcui:1426778	PHENYLMERCURIC ACETATE	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.012090184	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.013814173	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	chembl:CHEMBL1336287	3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	PARNATE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.006620561	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.039214094	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	2.019525817	NSC-640566	chembl:CHEMBL1287867	CHEMBL:CHEMBL1287867	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.037398626	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	0.1262203635473425	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	DITHIOLETHIONE	chembl:CHEMBL368700	DITHIOLETHIONE	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1166837138570989	CHLORAMBUCIL	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
DUSP3	hgnc:3069	DUSP3	DTC	9/2/20	NULL	1.875273972703375	GNF-PF-231	chembl:CHEMBL601167	CHEMBL:CHEMBL601167	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	O-DEMETHYLATED ADAPALENE	iuphar.ligand:3431	AHPN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00411841	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	chembl:CHEMBL1256180	5-(N-METHYL-N-ISOBUTYL)AMILORIDE	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.07699072	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	DTC	9/2/20	NULL	0.3125456621172291	RO-229735	chembl:CHEMBL2170369	CHEMBL:CHEMBL2170369	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	ACETOCHLOR	chembl:CHEMBL1517425	ACETOCHLOR	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.051885051	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.028929846	GNF-PF-1644	chembl:CHEMBL600734	CHEMBL:CHEMBL600734	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	OXABOLONE CIPIONATE	ncit:C81376	OXABOLONE CIPIONATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.013411921	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.009995749	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	3.088686543276147	NSC-640566	chembl:CHEMBL1287867	CHEMBL:CHEMBL1287867	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	DTC	9/2/20	NULL	1.521961485092594	CORDYCEPIN	rxcui:1989289	CORDYCEPIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.048618214	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	SJ000191886	chembl:CHEMBL601616	CHEMBL:CHEMBL601616	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	CIGLITAZONE	ncit:C72726	CIGLITAZONE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.078958904	DIFENOCONAZOLE	chembl:CHEMBL466426	DIFENOCONAZOLE	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.028850369	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	ANISINDIONE	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	TRICLABENDAZOLE	rxcui:2118525	TRICLABENDAZOLE	TRUE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	4.039051633514961	VERMISTATIN	chembl:CHEMBL1997854	VERMISTATIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	XCT790	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	ALPHA-NAPHTHOFLAVONE	drugbank:DB07453	ALPHA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.1084869240406911	HYDRASTINE	ncit:C76031	HYDRASTINE	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.069638821	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.2917092846427472	N-METHYLDOPAMINE HCL	chembl:CHEMBL1256484	CHEMBL:CHEMBL1256484	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	MERADIMATE	rxcui:91324	MERADIMATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.000434199	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	1.479089330582943	GIGANTOL	chembl:CHEMBL219553	GIGANTOL	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.019563216	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007232462	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.2333674277141978	THONZONIUM BROMIDE	rxcui:221171	THONZONIUM BROMIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.01275077	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	ORTHO-PHTHALALDEHYDE	chembl:CHEMBL160145	ORTHO-PHTHALALDEHYDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007003824	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	LAVENDUSTIN B	ncit:C1616	LAVENDUSTIN B	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.045265234	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.031861451	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	AG-99	chembl:CHEMBL296407	CHEMBL:CHEMBL296407	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.014993624	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.008418738	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	7-DEOXYPACLITAXEL	chembl:CHEMBL203365	CHEMBL:CHEMBL203365	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.08914715	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.055329474	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	NORFLOXACIN	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.039068208	CGS-21680	iuphar.ligand:375	CGS 21680	FALSE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	DTC	9/2/20	NULL	4.773424657790408	L-3,4-DEHYDROPROLINE	chembl:CHEMBL78920	CHEMBL:CHEMBL78920	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.001262355	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004384042	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	CINTAZONE	ncit:C73084	CINTAZONE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.051885051	7,12-DIMETHYL-BENZO[A]ANTHRACENE	chembl:CHEMBL329673	CHEMBL:CHEMBL329673	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1363835616511545	FUSARIC ACID	chembl:CHEMBL24510	FUSARIC ACID	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.016992774	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	CGP-60474	chembl:CHEMBL300389	CHEMBL:CHEMBL300389	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	METHOXYCHLOR	rxcui:2598123	METHOXYCHLOR	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.008899605	VANOXERINE	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	NSC-102049	chembl:CHEMBL74675	CHEMBL:CHEMBL74675	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	SPLITOMICIN	iuphar.ligand:8101	SPLITOMICIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	PHANQUONE	ncit:C90620	PHANQUONE	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.053579256	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	(S)-AMPA	drugbank:DB02057	(S)-AMPA	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	SJ000117462	chembl:CHEMBL590427	CHEMBL:CHEMBL590427	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00767656	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	GRISEOFULVIN	rxcui:5021	GRISEOFULVIN	TRUE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.093763699	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
GLI1	hgnc:4317	GLI1	DTC	9/2/20	NULL	5.834185692854944	4ALPHA-HYDROPEROXY-5-ENOVATODIOLIDE	chembl:CHEMBL512307	CHEMBL:CHEMBL512307	FALSE	FALSE	FALSE
S1PR2	hgnc:3169	S1PR2	DTC	9/2/20	NULL	0.6250913242344582	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010687497	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665886	chembl:CHEMBL532525	CHEMBL:CHEMBL532525	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.012466209	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	NSC-367089	chembl:CHEMBL1543865	CHEMBL:CHEMBL1543865	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005860885	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	3,3',4'-TRIHYDROXYFLAVONE	chembl:CHEMBL122701	CHEMBL:CHEMBL122701	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.1001290450718812	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.1244847587380144	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	ISOXABEN	chembl:CHEMBL2142789	ISOXABEN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00674559	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	SC-560	iuphar.ligand:10240	SC-560	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.045898314	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.008651783	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.007366396	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	GALLIC ACID METHYL ESTER	chembl:CHEMBL65675	GALLIC ACID METHYL ESTER	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.011152861	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	AMIDATE	chembl:CHEMBL23731	AMIDATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW589933X	chembl:CHEMBL1794055	GW589933X	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	TCMDC-123789	chembl:CHEMBL588859	CHEMBL:CHEMBL588859	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	L-162313	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	OCTABENZONE	chembl:CHEMBL1977129	OCTABENZONE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.003277632	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.026519026	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	CHLORACYZINE	ncit:C80874	CHLORACYZINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	XCT790	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.037425282	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.024141458	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.039331589	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	TCMDC-124327	chembl:CHEMBL581929	CHEMBL:CHEMBL581929	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.4930297768609811	ANDROGRAPHOLIDE	ncit:C61637	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.2734774543525755	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	0.1201548540862574	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	DNDI1417111	chembl:CHEMBL2094456	CHEMBL:CHEMBL2094456	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-5561	chembl:CHEMBL580353	CHEMBL:CHEMBL580353	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CANAVANINE	drugbank:DB01833	CANAVANINE	FALSE	FALSE	FALSE
IMPDH2	hgnc:6053	IMPDH2	DTC	9/2/20	NULL	10.50153424713889	6-CL-PRT-BIOTIN	chembl:CHEMBL1683024	CHEMBL:CHEMBL1683024	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.050488145	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012794267	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	LICOAGRONE	chembl:CHEMBL2437367	LICOAGRONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011850072	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.037081689	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001701921	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	EPIRIZOLE	ncit:C76075	EPIRIZOLE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DICHLORODIMETHYLSTANNANE	chembl:CHEMBL1076891	DICHLORODIMETHYLSTANNANE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.002706023	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
PADI3	hgnc:18337	PADI3	DTC	9/2/20	NULL	13.12691780892362	O-CL-AMIDINE	chembl:CHEMBL1910971	CHEMBL:CHEMBL1910971	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	AG-370	chembl:CHEMBL59150	CHEMBL:CHEMBL59150	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	R(+)-BUTYLINDAZONE	chembl:CHEMBL1256719	CHEMBL:CHEMBL1256719	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.064347636	XCT790	iuphar.ligand:2832	XCT790	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.051885051	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	CROMOLYN	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.041672755	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
RPS6KA1	hgnc:10430	RPS6KA1	DTC	9/2/20	NULL	8.751278539282415	SL-0101	chembl:CHEMBL240954	CHEMBL:CHEMBL240954	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IV-23E	chembl:CHEMBL1094674	CHEMBL:CHEMBL1094674	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	TCMDC-123579	chembl:CHEMBL533954	CHEMBL:CHEMBL533954	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.072927321	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.6908904109959803	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	CALMIDAZOLIUM CHLORIDE	chembl:CHEMBL1208858	CALMIDAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-1813	chembl:CHEMBL577662	CHEMBL:CHEMBL577662	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.012825518	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.050294704	ACYCLOVIR	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
RARG	hgnc:9866	RARG	DTC	9/2/20	NULL	1.323722804261206	BMS-204493	iuphar.ligand:2641	BMS493	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.031032903	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
KDM1A	hgnc:29079	KDM1A	DTC	9/2/20	NULL	5.250767123569449	TRANYLCYPROMINE HYDROCHLORIDE	chembl:CHEMBL1255743	TRANYLCYPROMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00410569	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	YOHIMBINE HYDROCHLORIDE	rxcui:133041	YOHIMBINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	GNF-PF-4227	chembl:CHEMBL585654	CHEMBL:CHEMBL585654	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	3.750547945	4-(2-TOLUYLETHYNYL)DIHYDROCINNAMIC ACID	iuphar.ligand:3952	TUG-424	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE	chembl:CHEMBL1214407	CHEMBL:CHEMBL1214407	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	ISOTHYMONIN	chembl:CHEMBL463563	ISOTHYMONIN	FALSE	FALSE	FALSE
MAPKAPK2	hgnc:6887	MAPKAPK2	DTC	9/2/20	NULL	0.3125456621172291	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.015930725	BENZETHONIUM CHLORIDE	rxcui:40036	BENZETHONIUM CHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	BIFEMELANE	rxcui:47111	BIFEMELANE	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.022249013	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.078793024	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
PADI1	hgnc:18367	PADI1	DTC	9/2/20	NULL	8.751278539282415	O-F-AMIDINE	iuphar.ligand:8625	O-F-AMIDINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.013411921	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	L-690330	iuphar.ligand:5208	L690330	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.03292017	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	HYDRALAZINE HYDROCHLORIDE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.1137761023525341	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW874091X	chembl:CHEMBL486124	GW874091X	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	GNF-PF-3582	chembl:CHEMBL606167	CHEMBL:CHEMBL606167	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
PIM2	hgnc:8987	PIM2	DTC	9/2/20	NULL	0.1075976869583903	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	1-O-ACETYLGEOPYXIN A	chembl:CHEMBL1902074	CHEMBL:CHEMBL1902074	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	3.000438356	BAS 8770945	chembl:CHEMBL478141	CHEMBL:CHEMBL478141	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	DTC	9/2/20	NULL	2.917092846427472	GHRELIN	ncit:C170105	LENOMORELIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	UNC10112764A	chembl:CHEMBL329040	CHEMBL:CHEMBL329040	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005130207	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	SJ000113211	chembl:CHEMBL602927	CHEMBL:CHEMBL602927	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	BRL-54443	iuphar.ligand:3927	BRL-54443	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	1.050153425	CHLOROQUINE-PYROLIDINYL	chembl:CHEMBL448594	CHLOROQUINE-PYROLIDINYL	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.00996918	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	GALLIC ACID METHYL ESTER	chembl:CHEMBL65675	GALLIC ACID METHYL ESTER	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.025298806	IPRONIAZID	rxcui:5981	IPRONIAZID	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.012819256	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	SULFOBROMOPHTHALEIN	rxcui:10212	SULFOBROMOPHTHALEIN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	TCMDC-124327	chembl:CHEMBL581929	CHEMBL:CHEMBL581929	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	HEXAHYDRO-SILA-DIFENIDOL HCL	chembl:CHEMBL1256647	CHEMBL:CHEMBL1256647	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TRETAZICAR	ncit:C81554	TRETAZICAR	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	PYRANTEL PAMOATE	rxcui:8985	PYRANTEL PAMOATE	TRUE	FALSE	FALSE
CASP2	hgnc:1503	CASP2	DTC	9/2/20	NULL	8.751278539282415	CETYLPYRIDINIUM CHLORIDE	rxcui:2287	CETYLPYRIDINIUM CHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.04339477	ZOXAZOLAMINE	ncit:C152966	ZOXAZOLAMINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.095122593	WHI-P154	iuphar.ligand:5993	JAK3 INHIBITOR II	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003162351	4-CHLOROMERCURIBENZOIC ACID	chembl:CHEMBL575867	4-CHLOROMERCURIBENZOIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	ETHAMSYLATE	rxcui:4112	ETHAMSYLATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	DIHYDROCAPSAICIN	rxcui:2166037	DIHYDROCAPSAICIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	1-(4-HYDROXYPHENYL)MALEIMIDE	chembl:CHEMBL565893	CHEMBL:CHEMBL565893	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.045461187	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.038467158	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	BENZAMIL	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	5-(N-ETHYL-N-ISOPROPYL)AMILORIDE	iuphar.ligand:4186	ETHYLISOPROPYLAMILORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	TRICLABENDAZOLE	rxcui:2118525	TRICLABENDAZOLE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.020510809	HYDRALAZINE HYDROCHLORIDE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.029498692	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	0.7955707762984013	FIDUXOSIN HYDROCHLORIDE	ncit:C81371	FIDUXOSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.035719504	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005039608	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.020542907	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.027855529	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	METOLACHOR	chembl:CHEMBL1884974	METOLACHOR	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.760980743	SPIRUCHOSTATIN C	chembl:CHEMBL1835659	SPIRUCHOSTATIN C	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00517674	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-3268	chembl:CHEMBL582073	CHEMBL:CHEMBL582073	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	PT-103	chembl:CHEMBL398765	CHEMBL:CHEMBL398765	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.012070729	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	CLOROPHENE	rxcui:21290	CLOROPHENE	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.2243917574174978	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	PENTAMIDINE ISETHIONATE	rxcui:7995	PENTAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	NSC-108783	chembl:CHEMBL1489812	CHEMBL:CHEMBL1489812	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.037081689	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.013613604	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
NPY2R	hgnc:7957	NPY2R	DTC	9/2/20	NULL	0.4688184931758437	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	DTC	9/2/20	NULL	0.5933070196123671	NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE	iuphar.ligand:4512	NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	DNDI1417263	chembl:CHEMBL1431115	CHEMBL:CHEMBL1431115	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1666910197958555	TCMDC-125543	chembl:CHEMBL546170	CHEMBL:CHEMBL546170	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.011176601	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.090530468	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	DNDI1417649	chembl:CHEMBL1994034	CHEMBL:CHEMBL1994034	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	GNF-PF-1577	chembl:CHEMBL600315	CHEMBL:CHEMBL600315	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	NSC-601359	chembl:CHEMBL1306524	CHEMBL:CHEMBL1306524	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001771873	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.026830696	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	SJ000040829	chembl:CHEMBL589711	CHEMBL:CHEMBL589711	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	PHENACYL CHLORIDE	iuphar.ligand:6285	OMEGA-CHLOROACETOPHENONE	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.069454592	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.016856395	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005045903	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	DNDI1417411	chembl:CHEMBL1445650	CHEMBL:CHEMBL1445650	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	NORDEFRIN	ncit:C81340	NORDEFRIN	FALSE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	DTC	9/2/20	NULL	0.8334550989792776	TRICLOCARBAN	rxcui:38609	TRICLOCARBAN	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.2500365296937833	THUNBERGINOL A	chembl:CHEMBL68810	THUNBERGINOL A	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.008599357	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.014658758	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.016807833	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	TCMDC-124266	chembl:CHEMBL124006	CHEMBL:CHEMBL124006	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.009627369	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NR2F2	hgnc:7976	NR2F2	DTC	9/2/20	NULL	1.093909817410302	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	DTC	9/2/20	NULL	0.088396753	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ENDOSULFAN SULFATE	chembl:CHEMBL2272380	ENDOSULFAN SULFATE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	CHLOROQUINE	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.015930725	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.005259182	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.007608705	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.015853765	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	TELITHROMYCIN	rxcui:274786	TELITHROMYCIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003139923	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.068369364	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00410569	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	PIPERACETAZINE	rxcui:8338	PIPERACETAZINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.801643836	LGD-5552	chembl:CHEMBL259820	CHEMBL:CHEMBL259820	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.033985548	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1750255707856483	SJ000082806	chembl:CHEMBL494668	CHEMBL:CHEMBL494668	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	TRIBUTYLCHLOROSTANNANE	chembl:CHEMBL1088186	TRIBUTYLCHLOROSTANNANE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	DIPYRITHIONE	rxcui:1362743	DIPYRITHIONE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.054243462	GNF-PF-4029	chembl:CHEMBL596633	CHEMBL:CHEMBL596633	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	DNDI1417995	chembl:CHEMBL1439833	CHEMBL:CHEMBL1439833	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	GNF-PF-4803	chembl:CHEMBL585240	CHEMBL:CHEMBL585240	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2853677784548614	AZELASTINE HYDROCHLORIDE	rxcui:235824	AZELASTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.048708415	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	0.106290832	CIANIDANOL	rxcui:1367177	CATECHIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	DYCLONINE	rxcui:23744	DYCLONINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	FASUDIL HYDROCHLORIDE	chembl:CHEMBL541388	FASUDIL HYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SALUBRINAL	chembl:CHEMBL180127	SALUBRINAL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	NSC-172033	chembl:CHEMBL238624	CHEMBL:CHEMBL238624	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	METHIOCARB	ncit:C163673	METHIOCARB	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.012211086	DEPHOSTATIN	chembl:CHEMBL269733	DEPHOSTATIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	RU-56187	chembl:CHEMBL1099140	CHEMBL:CHEMBL1099140	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.051177067	SIBUTRAMINE HYDROCHLORIDE	rxcui:1294535	SIBUTRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	0.3571950424196904	BMS-204493	iuphar.ligand:2641	BMS493	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.000813757	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.062509132	DNDI1318477	chembl:CHEMBL428064	CHEMBL:CHEMBL428064	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	NIMESULIDE	rxcui:53694	NIMESULIDE	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.6908904109959803	CEFDINIR	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	KAEMPFERITRIN	iuphar.ligand:13277	KAEMPFERITRIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	TCMDC-125784	chembl:CHEMBL581574	CHEMBL:CHEMBL581574	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	BOLDINE	chembl:CHEMBL388342	BOLDINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.084012274	ENOXOLONE	ncit:C526	ENOXOLONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-124066	chembl:CHEMBL529741	CHEMBL:CHEMBL529741	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.05486695	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	GLYCINE	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.014504882	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.093098708	GUAIAZULENE	rxcui:26290	GUAIAZULENE	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.058602312	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.4234489615781814	ISOSPAGLUMIC ACID	rxcui:236303	ISOSPAGLUMIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.006743857	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004426918	GR-127935	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.097236428	SB-216763	iuphar.ligand:8015	SB 216763	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.021554873	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	XAMOTEROL FUMARATE	rxcui:82133	XAMOTEROL FUMARATE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	4'-HYDROXYPHENYL-BENZO[D]THIAZOLE	chembl:CHEMBL47875	CHEMBL:CHEMBL47875	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.011568114	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	ZK-93423	drugbank:DB17063	ZK-93423	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.022691301	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	(S)-MEXILETINE	chembl:CHEMBL146855	(S)-MEXILETINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	(R)-FELODIPINE	chembl:CHEMBL254609	(R)-FELODIPINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW581744X	chembl:CHEMBL1909404	GW581744X	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	NAFRONYL OXALATE	ncit:C87286	NAFRONYL OXALATE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.021760328	A-23187	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.1508841127462485	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	DITHIAZANINE IODIDE	ncit:C75216	DITHIAZANINE IODIDE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	CEFOTIAM HYDROCHLORIDE	rxcui:236202	CEFOTIAM HYDROCHLORIDE	TRUE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.018719312	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	TAXIFOLIN	drugbank:DB02224	TAXIFOLIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TCMDC-123579	chembl:CHEMBL533954	CHEMBL:CHEMBL533954	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.011082244	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.01655349	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	DTC	9/2/20	NULL	0.1434635826111871	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	TRICLOCARBAN	rxcui:38609	TRICLOCARBAN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	MEBENDAZOLE	rxcui:6672	MEBENDAZOLE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	TCMDC-123641	chembl:CHEMBL532849	CHEMBL:CHEMBL532849	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	TDR77578	chembl:CHEMBL1364172	CHEMBL:CHEMBL1364172	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.2853677784548614	CRYPTOLEPINE HYDROCHLORIDE	chembl:CHEMBL92129	CRYPTOLEPINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.9723642821424906	CRYPTOLEPINE HYDROCHLORIDE	chembl:CHEMBL92129	CRYPTOLEPINE HYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-4097	chembl:CHEMBL597246	CHEMBL:CHEMBL597246	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	OXYCARBOXIN	chembl:CHEMBL1712057	OXYCARBOXIN	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.090530468	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SJ000200944	chembl:CHEMBL600173	CHEMBL:CHEMBL600173	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.2500365296937833	DNDI1417884	chembl:CHEMBL1346025	CHEMBL:CHEMBL1346025	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	LONCHOCARPIC ACID	chembl:CHEMBL1527366	LONCHOCARPIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.004399838	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	DTC	9/2/20	NULL	0.6563458904461812	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.1548898856510162	GNF-PF-3265	chembl:CHEMBL581868	CHEMBL:CHEMBL581868	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	HOMATROPINE HYDROBROMIDE	rxcui:235428	HOMATROPINE HYDROBROMIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00675253	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DIPHENADIONE	ncit:C75156	DIPHENADIONE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	GLABRONE	chembl:CHEMBL600457	GLABRONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	3,4-DIHYDROXYPHENYLACETIC ACID	chembl:CHEMBL1284	3,4-DIHYDROXYPHENYLACETIC ACID	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1256164383629055	AG-537	chembl:CHEMBL67535	CHEMBL:CHEMBL67535	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.1259176768242074	LAGASCATRIOL	chembl:CHEMBL2180482	LAGASCATRIOL	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.091159151	CLOROTEPINE	ncit:C77572	CLOROTEPINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	L-PHENYLALANINE	rxcui:8156	PHENYLALANINE	TRUE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	DTC	9/2/20	NULL	0.099446347	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	CLENBUTEROL HYDROCHLORIDE	rxcui:235955	CLENBUTEROL HYDROCHLORIDE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.001759051	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1458546423213736	TCMDC-125528	chembl:CHEMBL375673	CHEMBL:CHEMBL375673	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NSC-126757	chembl:CHEMBL228132	CHEMBL:CHEMBL228132	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.089046362	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.003949727	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	0.3409589041278864	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	0.4375639269641208	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.001807742	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.031555091	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.054695491	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	MMV006513	chembl:CHEMBL585622	CHEMBL:CHEMBL585622	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	6'-IODONONIVAMIDE	chembl:CHEMBL177809	CHEMBL:CHEMBL177809	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PROPYL GALLATE	rxcui:1311134	PROPYL GALLATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	GNF-PF-2267	chembl:CHEMBL601764	CHEMBL:CHEMBL601764	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	KETOTIFEN	rxcui:11404	KETOTIFEN FUMARATE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.1902451856365742	TRIBUTYLCHLOROSTANNANE	chembl:CHEMBL1088186	TRIBUTYLCHLOROSTANNANE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	ARUNDINE	chembl:CHEMBL446452	ARUNDINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	HYDROCOTARNINE	chembl:CHEMBL1606295	HYDROCOTARNINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	BERGAMOTTIN	chembl:CHEMBL1078442	BERGAMOTTIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CAPENSIN	chembl:CHEMBL1327256	CAPENSIN	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.2917092846427472	SJ000018309	chembl:CHEMBL591363	CHEMBL:CHEMBL591363	FALSE	FALSE	FALSE
PASK	hgnc:17270	PASK	DTC	9/2/20	NULL	0.5048814541893702	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW831091X	chembl:CHEMBL103115	GW831091X	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.022632617	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.003806283	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006096328	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	FIDUXOSIN HYDROCHLORIDE	ncit:C81371	FIDUXOSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.364636606	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	GNF-PF-2347	chembl:CHEMBL579045	CHEMBL:CHEMBL579045	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.007609807	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	MK-886	drugbank:DB16739	MK-886	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.068191781	BAS 01152706	chembl:CHEMBL2002487	CHEMBL:CHEMBL2002487	FALSE	FALSE	FALSE
NPY1R	hgnc:7956	NPY1R	DTC	9/2/20	NULL	0.3750547945406749	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-264865	chembl:CHEMBL1785002	CHEMBL:CHEMBL1785002	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.005268681	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	BW-373U86	iuphar.ligand:9002	BW373U86	FALSE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	DTC	9/2/20	NULL	2.386712328895204	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.042242696	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.036062961	NSC-663284	drugbank:DB17038	NSC-663284	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.03292017	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.025865848	MEFENAMIC ACID	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
SIRT5	hgnc:14933	SIRT5	DTC	9/2/20	NULL	0.5966780822238011	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.001939556	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.060984519	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.023524942	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	TYRPHOSTIN AG-112	iuphar.ligand:5913	AG 112	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.014832675	BIOCHANIN	iuphar.ligand:2829	BIOCHANIN A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	CEFAZOLIN	rxcui:2180	CEFAZOLIN	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	DNDI1318925	chembl:CHEMBL1390716	CHEMBL:CHEMBL1390716	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.009031247	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	THUNBERGINOL A	chembl:CHEMBL68810	THUNBERGINOL A	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	CHLOROTHALONIL	chembl:CHEMBL468167	CHLOROTHALONIL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	KRESOXIM-METHYL	chembl:CHEMBL203191	KRESOXIM-METHYL	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.026045472	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	GNF-PF-4300	chembl:CHEMBL585656	CHEMBL:CHEMBL585656	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.033985548	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	FOMOCAINE	ncit:C65747	FOMOCAINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.7242437411819931	KLUGINE	chembl:CHEMBL486004	KLUGINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.1400204566285186	FLUDIOXONIL	chembl:CHEMBL485833	FLUDIOXONIL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	PREGNENOLONE SULFATE SODIUM	chembl:CHEMBL1256742	PREGNENOLONE SULFATE SODIUM	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	2-BENZOYL-5-METHOXYBENZOQUINONE	chembl:CHEMBL1434057	2-BENZOYL-5-METHOXYBENZOQUINONE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.014206621	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.005459124	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.024108205	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	DNDI1417995	chembl:CHEMBL1439833	CHEMBL:CHEMBL1439833	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	GNF-PF-3561	chembl:CHEMBL599712	CHEMBL:CHEMBL599712	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.4134462302023188	OXAPIUM	chembl:CHEMBL1725250	OXAPIUM	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.1244257612220248	TCMDC-125086	chembl:CHEMBL532504	CHEMBL:CHEMBL532504	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	DNDI1417346	chembl:CHEMBL1490332	CHEMBL:CHEMBL1490332	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	(R)-FELODIPINE	chembl:CHEMBL254609	(R)-FELODIPINE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	MECAMYLAMINE	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	SPHAEROPSIDIN A	chembl:CHEMBL1834675	SPHAEROPSIDIN A	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.1017590527823536	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	SOLYPERTINE TARTRATE	ncit:C152391	SOLYPERTINE TARTRATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	BENZYL NICOTINATE	ncit:C83549	BENZYL NICOTINATE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	MEDRONIC ACID	rxcui:1314368	MEDRONIC ACID	TRUE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.2692701089009974	(RS)-ROSCOVITINE	chembl:CHEMBL52387	(RS)-ROSCOVITINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	chembl:CHEMBL224214	CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	MECYSTEINE HYDROCHLORIDE	rxcui:235828	MECYSTEINE HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	PILSICAINIDE	ncit:C72582	PILSICAINIDE	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.024275391	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	2,4-DIHYDROXYBENZOPHENONE	chembl:CHEMBL1392	2,4-DIHYDROXYBENZOPHENONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW643971X	chembl:CHEMBL1789962	GW643971X	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	OXYQUINOLINE	rxcui:110	OXYQUINOLINE	TRUE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-3352	chembl:CHEMBL600306	CHEMBL:CHEMBL600306	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.073540156	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.068637479	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.075333818	NSC-751382	chembl:CHEMBL1935538	CHEMBL:CHEMBL1935538	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.010726797	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	XYLOMETAZOLINE	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.2651902587661338	EMETINE HYDROCHLORIDE	rxcui:82015	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.039598545	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	AMPIROXICAM	ncit:C73073	AMPIROXICAM	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.056097939	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01150727	LY-367265	chembl:CHEMBL1079460	CHEMBL:CHEMBL1079460	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	O-DEMETHYLATED ADAPALENE	iuphar.ligand:3431	AHPN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	DNDI1417809	chembl:CHEMBL1442783	CHEMBL:CHEMBL1442783	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1029562181092048	NSC-677438	chembl:CHEMBL118678	CHEMBL:CHEMBL118678	FALSE	FALSE	FALSE
PADI2	hgnc:18341	PADI2	DTC	9/2/20	NULL	8.751278539282415	O-CL-AMIDINE	chembl:CHEMBL1910971	CHEMBL:CHEMBL1910971	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.8751278539282418	NSC-108783	chembl:CHEMBL1489812	CHEMBL:CHEMBL1489812	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	CLEBOPRIDE	rxcui:21224	CLEBOPRIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	GLABROL	chembl:CHEMBL462721	GLABROL	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.023780648	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.020383413	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.092443083	THAPSIGARGIN	ncit:C128634	THAPSIGARGIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	NORDEFRIN HYDROCHLORIDE	ncit:C99670	NORDEFRIN HYDROCHLORIDE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.025244073	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	CUCURBITACIN B	iuphar.ligand:12432	CUCURBITACIN B	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	L-165041	drugbank:DB08078	{4-[3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPOXY]PHENOXY}ACETIC ACID	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	3-PHENYLUMBELLIFERONE	chembl:CHEMBL153505	CHEMBL:CHEMBL153505	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.043611023	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.7955707762984013	PROSTAGLANDIN A2	iuphar.ligand:6279	PROSTAGLANDIN A2	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	DIFLORASONE DIACETATE	rxcui:23033	DIFLORASONE DIACETATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006780433	TYRPHOSTIN 47	chembl:CHEMBL77030	TYRPHOSTIN 47	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.040703621	AG-1879	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	TCMDC-125000	chembl:CHEMBL579742	CHEMBL:CHEMBL579742	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005574063	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007374673	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.021431703	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TESTOLACTONE	rxcui:10378	TESTOLACTONE	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010093747	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TRIPHENYLSTANNYL ACETATE	chembl:CHEMBL474376	TRIPHENYLSTANNYL ACETATE	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.026789628	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.012486961	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DINOSEB	chembl:CHEMBL1892987	DINOSEB	FALSE	FALSE	FALSE
DDR2	hgnc:2731	DDR2	DTC	9/2/20	NULL	1.615620653405984	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	PHENETHYL PHENYLCARBAMATE	chembl:CHEMBL2135268	PHENETHYL PHENYLCARBAMATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	HYDROXYZINE	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	OLIVOMYCIN I	chembl:CHEMBL576383	OLIVOMYCIN I	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-1235	chembl:CHEMBL585769	CHEMBL:CHEMBL585769	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	HOECHST 33258	chembl:CHEMBL301735	HOECHST 33258	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.09669921	GNF-PF-4674	chembl:CHEMBL584452	CHEMBL:CHEMBL584452	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.015002192	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.02339914	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	TOXYLOXANTHONE C	chembl:CHEMBL459022	TOXYLOXANTHONE C	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.012573676	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	2',3'-DIHYDROXYFLAVONE	chembl:CHEMBL242171	CHEMBL:CHEMBL242171	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.01327292	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.2734774543525755	RO-25-6981	chembl:CHEMBL305195	CHEMBL:CHEMBL305195	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	SRT-1460	chembl:CHEMBL254156	CHEMBL:CHEMBL254156	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	BENZOCAINE	rxcui:1399	BENZOCAINE	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.6563458904461813	HESPERIDIN	rxcui:5281	HESPERIDIN	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	AG-99	chembl:CHEMBL296407	CHEMBL:CHEMBL296407	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	PENTAMIDINE DIISETHIONATE	chembl:CHEMBL361506	PENTAMIDINE ISETHIONATE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	EPALRESTAT	ncit:C72762	EPALRESTAT	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.071341945	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002767057	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2403097081725148	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	CYCLOASPEPTIDE A	chembl:CHEMBL473074	CYCLOASPEPTIDE A	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	EMETINE HYDROCHLORIDE	rxcui:82015	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.01199079	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	IPA-3	iuphar.ligand:8940	IPA-3	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.1666910197958555	GNF-PF-3023	chembl:CHEMBL535331	CHEMBL:CHEMBL535331	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	RUBITECAN	ncit:C1485	RUBITECAN	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	TRIADIMEFON	chembl:CHEMBL520897	TRIADIMEFON	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.210030685	9-NITRO-ANTHRACENE	chembl:CHEMBL166112	CHEMBL:CHEMBL166112	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.048083948	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	DNDI1417099	chembl:CHEMBL1565444	CHEMBL:CHEMBL1565444	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.2792961235941196	SEMUSTINE	ncit:C827	SEMUSTINE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.037239483	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.1483267549030917	DNDI1417132	chembl:CHEMBL1492017	CHEMBL:CHEMBL1492017	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	PROSTAGLANDIN A2	iuphar.ligand:6279	PROSTAGLANDIN A2	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.016460085	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	HOE-33342	chembl:CHEMBL343002	CHEMBL:CHEMBL343002	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	DTC	9/2/20	NULL	0.2333674277141977	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.005135727	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.016206071	PYRONIN Y	chembl:CHEMBL1486690	PYRONIN Y	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.3889457128569962	BAS-0338868	chembl:CHEMBL378903	CHEMBL:CHEMBL378903	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	2-BENZOYL-5-METHOXYBENZOQUINONE	chembl:CHEMBL1434057	2-BENZOYL-5-METHOXYBENZOQUINONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	DILTIAZEM HYDROCHLORIDE	rxcui:203211	DILTIAZEM HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	LAWSONE	drugbank:DB04744	LAWSONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01256465	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.006783937	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.002450881	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	A-23187	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.010620484	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	DTC	9/2/20	NULL	0.2557191780959147	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.009349657	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.000876808	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2386712328895204	GNF-PF-5151	chembl:CHEMBL576208	CHEMBL:CHEMBL576208	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	3.000438356	BAS-8770951	chembl:CHEMBL478323	CHEMBL:CHEMBL478323	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.049817525	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003512454	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.01060761	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	QUINESTROL	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1396480617970598	METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE	chembl:CHEMBL1214407	CHEMBL:CHEMBL1214407	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.062733179	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	2-MERCAPTOBENZIMIDAZOLE	chembl:CHEMBL70141	2-MERCAPTOBENZIMIDAZOLE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	3-HYDROXYFLAVONOL	chembl:CHEMBL242172	CHEMBL:CHEMBL242172	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.3365876361262467	CLOFOCTOL	rxcui:21264	CLOFOCTOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	BOLDINE	chembl:CHEMBL388342	BOLDINE	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.009268786	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1801292323694494	PANOBINOSTAT	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	SJ000018300	chembl:CHEMBL590927	CHEMBL:CHEMBL590927	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006193403	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NU-1025	chembl:CHEMBL123904	CHEMBL:CHEMBL123904	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.084553416	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	SKIMMIANINE	chembl:CHEMBL21396	SKIMMIANINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	NSC-367089	chembl:CHEMBL1543865	CHEMBL:CHEMBL1543865	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.010819631	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	SPLITOMICIN	iuphar.ligand:8101	SPLITOMICIN	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	1.050153425	SJ000279636	chembl:CHEMBL592838	CHEMBL:CHEMBL592838	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.078958904	DIBUTYLDICHLOROSTANNANE	chembl:CHEMBL1088184	DIBUTYLDICHLOROSTANNANE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.3454452054979901	Fam-Trastuzumab Deruxtecan-nxki	rxcui:2267574	FAM-TRASTUZUMAB DERUXTECAN-NXKI	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.049349315	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.04339477	Formoterol	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.075010959	Metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.3938075342677087	Mafenide	rxcui:6572	MAFENIDE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	FDA	10-Apr-24	NULL	1.009762908	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	FDA	10-Apr-24	NULL	2.151953739167807	Olaratumab	rxcui:1855735	OLARATUMAB	TRUE	FALSE	FALSE
EPHB4	hgnc:3395	EPHB4	MyCancerGenome	20-Jun-17	inhibitor	5.469549087051511	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.1151484018326633	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.1643432589536604	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.073437302	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.041021618	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.2651902587661338	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.1077080435603989	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.1200175342530159	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.1200175342530159	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.1750255707856483	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.1312691780892362	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.1077080435603989	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.090843722	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.1312691780892362	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.088248187	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.079197091	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.049026771	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.1470803115845784	XL147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
DEPTOR	hgnc:22953	DEPTOR	MyCancerGenome	20-Jun-17	inhibitor	1.944728564284981	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.1041818873724097	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.048083948	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.1041818873724097	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.048083948	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2678962818147679	PD 0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2083637747448194	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.079236928	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1607377690888607	PKI-587	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1715936968486748	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
PDGFD	hgnc:30620	PDGFD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5357925636295356	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.252440727	ENDOSTATIN (84-114)-NH2 (JKC367)	drugbank:DB06423	ENDOSTATIN	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4906052389860809	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02321294	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.00299189	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.011810092	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.1121958787087489	LIPOSOMAL DOXORUBICIN	wikidata:Q29004943	CAELYX	FALSE	FALSE	TRUE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.1026877533944481	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.026927011	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.4039051633514962	RUTIN	rxcui:9500	RUTIN	TRUE	FALSE	FALSE
AKR1B1	hgnc:381	AKR1B1	NCI	14-Sep-17	NULL	0.2308029504865692	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
AKR1B1	hgnc:381	AKR1B1	NCI	14-Sep-17	NULL	0.6731752722524935	URACIL	rxcui:10995	URACIL	TRUE	FALSE	TRUE
AGTR2	hgnc:338	AGTR2	NCI	14-Sep-17	NULL	0.4546118721705151	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	NCI	14-Sep-17	NULL	0.068191781	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.048083948	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
APC	hgnc:583	APC	NCI	14-Sep-17	NULL	0.1432027397337122	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.2263261691193728	GANCICLOVIR	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
ATP7A	hgnc:869	ATP7A	NCI	14-Sep-17	NULL	0.2845944240417046	OXALIPLATIN	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.8537832721251137	RNA POLYMERASE INHIBITOR	ncit:C25995	RNA POLYMERASE INHIBITOR	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.042689164	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.044161204	MAO INHIBITORS	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.094864808	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.9460841664089098	PARICALCITOL	rxcui:73710	PARICALCITOL	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.079557078	INTERFERON BETA-1A	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
BTF3L1	hgnc:1126	BTF3P11	NCI	14-Sep-17	NULL	1.093909817410302	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
BTF3L1	hgnc:1126	BTF3P11	NCI	14-Sep-17	NULL	0.2224901323546377	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
CAMK2G	hgnc:1463	CAMK2G	NCI	14-Sep-17	NULL	0.1190650141398968	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
CDKN2D	hgnc:1790	CDKN2D	NCI	14-Sep-17	NULL	1.050153425	5-AZA-2&APOS;-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
CFTR	hgnc:1884	CFTR	NCI	14-Sep-17	NULL	0.082300425	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CEL	hgnc:1848	CEL	NCI	14-Sep-17	NULL	0.258658479	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.9376369863516875	GLUTAMINE	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.1123158743009508	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	1.250182648468916	ENVIRONMENTAL ESTROGEN	ncit:C1894	ENVIRONMENTAL ESTROGEN	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.4167275494896388	OPIATE	ncit:C1657	OPIATE	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.1470803115845784	NONSTEROIDAL ANTI-INFLAMMATORY DRUGS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.00804962	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP51A1	hgnc:2649	CYP51A1	NCI	14-Sep-17	NULL	3.500511415712967	FLUCONAZOLE	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.1521961485092594	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.8751278539282416	FADROZOLE	ncit:C79911	FADROZOLE	FALSE	FALSE	FALSE
CYP4B1	hgnc:2644	CYP4B1	NCI	14-Sep-17	NULL	4.375639269641208	DEXTRAN SULFATE	rxcui:40068	DEXTRAN SULFATE	FALSE	FALSE	FALSE
CYSLTR1	hgnc:17451	CYSLTR1	NCI	14-Sep-17	NULL	0.4546118721705151	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.022613123	TAXOL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.3488881809680697	PENICILLAMINE	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.037003292	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
DUSP1	hgnc:3064	DUSP1	NCI	14-Sep-17	NULL	0.33338204	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.2536602475154323	PROSTAGLANDIN E1	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.099071078	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
FCER2	hgnc:3612	FCER2	NCI	14-Sep-17	NULL	0.8078103267029924	PROTEIN TYROSINE KINASE INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.1591141552596803	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.05814803	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	2.386712328895204	BUTHIONINE SULPHOXIMINE	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.2651902587661338	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.1544343271638073	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
GPI	hgnc:4458	GPI	NCI	14-Sep-17	NULL	2.625383561784725	6-AN	ncit:C38127	6-AMINONICOTINAMIDE	FALSE	FALSE	FALSE
GLO1	hgnc:4323	GLO1	NCI	14-Sep-17	NULL	17.50255707856483	N-METHYLFORMAMIDE	ncit:C1163	N-METHYLFORMAMIDE	FALSE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	2.282942227638891	ANTITUBERCULOSIS	ncit:C280	ANTITUBERCULAR AGENT	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1250182648468916	IFOSFAMIDE	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.5147810905460245	ECHINACEA	rxcui:228041	ECHINACEA PREPARATION	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.049026771	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	GARLIC EXTRACT	ncit:C29069	GARLIC EXTRACT	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	1.029562181092049	ANTITUBERCULOSIS	ncit:C280	ANTITUBERCULAR AGENT	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1640864726115453	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1715936968486748	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
IL3RA	hgnc:6012	IL3RA	NCI	14-Sep-17	NULL	1.166837138570989	IL-3	iuphar.ligand:4994	IL-3	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1392776425349987	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
ITGA2B	hgnc:6138	ITGA2B	NCI	14-Sep-17	NULL	0.546954909	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.7242437411819932	MMF	rxcui:1546433	MONOMETHYL FUMARATE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.2430910705356226	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.067839369	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	NCI	14-Sep-17	NULL	0.2414145803939977	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	NCI	14-Sep-17	NULL	0.2853677784548614	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
KRT18	hgnc:6430	KRT18	NCI	14-Sep-17	NULL	2.917092846427472	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.8468979231563628	HMG-COA REDUCTASE INHIBITOR	ncit:C1655	HMG-COA REDUCTASE INHIBITOR	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.015219615	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.015219615	DOX	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.048958202	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.043902735	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
MARCKSL1	hgnc:7142	MARCKSL1	NCI	14-Sep-17	NULL	0.4487835148349957	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	ALTRETAMINE	rxcui:5296	ALTRETAMINE	TRUE	FALSE	FALSE
MBP	hgnc:6925	MBP	NCI	14-Sep-17	NULL	1.000146118775133	INTERFERON BETA-1A	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
MGEA5	hgnc:7056	OGA	NCI	14-Sep-17	NULL	1.141471113819445	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.093596562	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	INDIUM CHLORIDE	chembl:CHEMBL1447815	INDIUM CHLORIDE	FALSE	FALSE	FALSE
MT1H	hgnc:7400	MT1H	NCI	14-Sep-17	NULL	0.326134604	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
MT1H	hgnc:7400	MT1H	NCI	14-Sep-17	NULL	3.000438356	6-AN	ncit:C38127	6-AMINONICOTINAMIDE	FALSE	FALSE	FALSE
MYB	hgnc:7545	MYB	NCI	14-Sep-17	NULL	0.1620607136904151	TAXOL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
MXI1	hgnc:7534	MXI1	NCI	14-Sep-17	NULL	5.000730593875666	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.025183535	PROTEIN PHOSPHATASE INHIBITOR	ncit:C2159	PROTEIN PHOSPHATASE INHIBITOR	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	DTC	9/2/20	NULL	0.089298761	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.031479419	FGF-1	iuphar.ligand:4923	FGF-1	FALSE	FALSE	FALSE
NPTN	hgnc:17867	NPTN	NCI	14-Sep-17	NULL	1.500219178	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.1704794520639432	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	1.909369863116163	K-252A	drugbank:DB02152	K-252A	FALSE	FALSE	FALSE
PCNA	hgnc:8729	PCNA	NCI	14-Sep-17	NULL	1.235474617310459	CAPSAICIN	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.081030357	MILTEFOSINE	rxcui:1494066	MILTEFOSINE	TRUE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	0.068458502	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.2500365296937833	SOMATOTROPIN	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-2559	chembl:CHEMBL583584	CHEMBL:CHEMBL583584	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.041672755	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1620607136904151	ANTIVIRAL	ncit:C281	ANTIVIRAL AGENT	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.729273212	ALPHA-ADRENERGIC ANTAGONIST	ncit:C29713	ALPHA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006811217	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
RAMP3	hgnc:9845	RAMP3	NCI	14-Sep-17	NULL	0.760980743	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.1356787370431382	PREDNISONE	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	1.009762908	8-GERANYLOXY PSORALEN	chembl:CHEMBL1412710	CHEMBL:CHEMBL1412710	FALSE	FALSE	FALSE
PTPN6	hgnc:9658	PTPN6	NCI	14-Sep-17	NULL	2.500365296937833	IL-4	iuphar.ligand:4996	IL-4	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.073922431	BAY 43-9006	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.1470803115845784	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
S100B	hgnc:10500	S100B	NCI	14-Sep-17	NULL	1.141471113819445	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
RPE65	hgnc:10294	RPE65	NCI	14-Sep-17	NULL	0.7259125055625967	RETINOIC ACIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
SAG	hgnc:10521	SAG	NCI	14-Sep-17	NULL	0.5645986154375753	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.027276712	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.364636606	CGS 20267	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	0.8751278539282416	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.1187956362798518	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	2.019525817	NSC-640353	chembl:CHEMBL1288253	CHEMBL:CHEMBL1288253	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.201952582	IRBESARTAN	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.080781033	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	NCI	14-Sep-17	NULL	0.1278595890479573	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	NCI	14-Sep-17	NULL	0.095122593	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.092443083	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.03297185	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	NCI	14-Sep-17	NULL	0.027121731	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	NCI	14-Sep-17	NULL	0.027672027	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	NCI	14-Sep-17	NULL	0.08780547	TROGLITAZONE	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.005883872	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
SNW1	hgnc:16696	SNW1	NCI	14-Sep-17	NULL	4.773424657790409	TRANSFORMING GROWTH FACTOR	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	NCI	14-Sep-17	NULL	0.007906591	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	NCI	14-Sep-17	NULL	0.3889457128569963	LAVENDUSTIN A	ncit:C1142	LAVENDUSTIN A	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.3500511415712967	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.175610941	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.192335792	LITHIUM	rxcui:6448	LITHIUM	TRUE	FALSE	FALSE
SRY	hgnc:11311	SRY	NCI	14-Sep-17	NULL	1.193356164447602	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	NCI	14-Sep-17	NULL	0.1325951293830669	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	3.500511415712966	DECAPEPTYL	rxcui:38782	TRIPTORELIN	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.6035364509849942	FAMOTIDINE	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	4.200613699	ALVAC	ncit:C1479	ALVAC VACCINE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.076765601	BRL-50481	iuphar.ligand:5154	BRL50481	FALSE	FALSE	FALSE
TCN1	hgnc:11652	TCN1	NCI	14-Sep-17	NULL	157.5230137070835	VITAMIN-B12	ncit:C939	COBALAMIN	FALSE	FALSE	FALSE
TDO2	hgnc:11708	TDO2	NCI	14-Sep-17	NULL	0.4773424657790409	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	DNDI1417006	chembl:CHEMBL1415258	CHEMBL:CHEMBL1415258	FALSE	FALSE	FALSE
TFAP2A	hgnc:11742	TFAP2A	NCI	14-Sep-17	NULL	3.500511415712967	AMPRENAVIR	rxcui:228656	AMPRENAVIR	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.2419708351875322	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.042379073	CORTISOL	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.068458502	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.016916131	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.038693936	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.1282238613814273	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
TLR3	hgnc:11849	TLR3	NCI	14-Sep-17	NULL	2.625383561784724	IL-13	iuphar.ligand:4980	IL-13	FALSE	FALSE	FALSE
THY1	hgnc:11801	THY1	NCI	14-Sep-17	NULL	11.66837138570988	HEL	ncit:C1925	LYSOZYME	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.5385402178019949	BENZODIAZEPINE	ncit:C1012	BENZODIAZEPINE	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.1666910197958555	TRAIL	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.040640612	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
YY1	hgnc:12856	YY1	NCI	14-Sep-17	NULL	3.000438356	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	OncoKB	23-Jul-20	NULL	0.4022765134992723	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	DTC	9/2/20	NULL	0.138178082	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	OncoKB	23-Jul-20	NULL	0.458240639	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	1.336059069138614	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	1.282909942931453	Encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
ZRSR2	hgnc:23019	ZRSR2	OncoKB	23-Jul-20	NULL	13.12691780892362	H3B-8800	drugbank:DB14017	H3B-8800	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	TCMDC-125518	chembl:CHEMBL587772	CHEMBL:CHEMBL587772	FALSE	FALSE	FALSE
PTCH1	hgnc:9585	PTCH1	OncoKB	23-Jul-20	NULL	4.375639269641208	Sonidegib	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
SF3B1	hgnc:10768	SF3B1	OncoKB	23-Jul-20	NULL	4.375639269641208	H3B-8800	drugbank:DB14017	H3B-8800	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.6019397937072561	dacomitinib	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.006643177	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	PharmGKB	4/5/24	NULL	0.1458546423213736	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	8-AZAGUANINE	ncit:C28788	8-AZAGUANINE	FALSE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	PharmGKB	4/5/24	NULL	0.2273059360852575	eflornithine	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	1.458546423213736	8-AZAHYPOXANTHINE	chembl:CHEMBL219416	CHEMBL:CHEMBL219416	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	PharmGKB	4/5/24	NULL	0.7778914257139925	ritodrine	rxcui:9392	RITODRINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004350623	theophylline	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.3170753093942904	doxazosin	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SYMCLOSENE	rxcui:2375531	SYMCLOSENE	FALSE	FALSE	FALSE
SI	hgnc:10856	SI	PharmGKB	4/5/24	NULL	6.563458904461812	sacrosidase	rxcui:214817	SACROSIDASE	TRUE	FALSE	FALSE
LEPR	hgnc:6554	LEPR	PharmGKB	4/5/24	NULL	0.525076712	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CHLORMIDAZOLE	ncit:C78032	CHLORMIDAZOLE	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.5073204950308646	methoxamine	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
JMJD8	hgnc:14148	JMJD8	PharmGKB	4/5/24	NULL	1.500219178	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
TNFRSF11B	hgnc:11909	TNFRSF11B	PharmGKB	4/5/24	NULL	1.000146118775133	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
FDPS	hgnc:3631	FDPS	PharmGKB	4/5/24	NULL	1.633571993999384	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	ARACHIDONOYL GABA	iuphar.ligand:5494	N-ARACHIDONYL-&GAMMA;-AMINOBUTYRIC ACID	FALSE	FALSE	FALSE
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	1.000146118775133	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
COL1A1	hgnc:2197	COL1A1	PharmGKB	4/5/24	NULL	1.000146118775133	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	PharmGKB	4/5/24	NULL	0.021309932	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.9053046764774912	TRANYLCYPROMINE HYDROCHLORIDE	chembl:CHEMBL1255743	TRANYLCYPROMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	PharmGKB	4/5/24	NULL	0.1795134059339982	zoledronate	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
SLC28A3	hgnc:16484	SLC28A3	PharmGKB	4/5/24	NULL	0.5556367326528519	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	PharmGKB	4/5/24	NULL	0.042516333	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	N6-PHENYLADENOSINE	chembl:CHEMBL262083	N6-PHENYLADENOSINE	FALSE	FALSE	FALSE
E2F7	hgnc:23820	E2F7	PharmGKB	4/5/24	NULL	0.5385402178019949	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	0.064624826	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.020226376	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CCNA2	hgnc:1578	CCNA2	PharmGKB	4/5/24	NULL	0.2019525816757481	tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.015193192	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.024861587	curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
GSTA1	hgnc:4626	GSTA1	PharmGKB	4/5/24	NULL	0.8290684931951763	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.079236928	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PFDN4	hgnc:8868	PFDN4	PharmGKB	4/5/24	NULL	0.9376369863516874	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ADRA2B	hgnc:282	ADRA2B	PharmGKB	4/5/24	NULL	0.1654653505326507	yohimbine	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
ABCG1	hgnc:73	ABCG1	PharmGKB	4/5/24	NULL	0.9460841664089098	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
IL18	hgnc:5986	IL18	PharmGKB	4/5/24	NULL	0.172722603	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ABL2	hgnc:77	ABL2	DTC	9/2/20	NULL	0.080781033	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.4234489615781814	ethambutol	rxcui:142435	ETHAMBUTOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ERCC5	hgnc:3437	ERCC5	PharmGKB	4/5/24	NULL	3.938075342677087	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.022949157	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.022439176	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.00547297	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.2243917574174978	gramicidin d	rxcui:5011	GRAMICIDIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.032055965	levetiracetam	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.011906501	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.00897567	topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
IRS1	hgnc:6125	IRS1	PharmGKB	4/5/24	NULL	0.364636606	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.056097939	vitamin e	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
AOX1	hgnc:553	AOX1	PharmGKB	4/5/24	NULL	1.105424657593568	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	PharmGKB	4/5/24	NULL	0.052090944	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.1187956362798518	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.073054151	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.020672312	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.037398626	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	0.300043836	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.1682938180631233	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.074797252	ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	PharmGKB	4/5/24	NULL	0.525076712	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
MTHFD1	hgnc:7432	MTHFD1	PharmGKB	4/5/24	NULL	1.050153425	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.012466209	SB-224289	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	PharmGKB	4/5/24	NULL	0.1909369863116163	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
KL	hgnc:6344	KL	PharmGKB	4/5/24	NULL	2.561349816375341	corticosteroids	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.015599427	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	0.040235763	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	1.050153425	bilirubin	iuphar.ligand:4577	BILIRUBIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	SB-224289	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
ACSS2	hgnc:15814	ACSS2	PharmGKB	4/5/24	NULL	0.1944728564284981	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ADK	hgnc:257	ADK	PharmGKB	4/5/24	NULL	0.9546849315580819	abacavir	rxcui:190521	ABACAVIR	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	BIS(2-ETHYLHEXYL) PHTHALATE	chembl:CHEMBL1242017	BIS(2-ETHYLHEXYL) PHTHALATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.08854582	fluoxetine / olanzapine	wikidata:Q48564244	FLUOXETINE / OLANZAPINE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.017363648	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.1369170045259309	gemfibrozil	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1771513874348667	interferons	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	PharmGKB	4/5/24	NULL	0.08780547	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.018874073	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	2.838252499226729	nitrous oxide	rxcui:7486	NITROUS OXIDE	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	PharmGKB	4/5/24	NULL	0.3571950424196904	niacin	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	PharmGKB	4/5/24	NULL	0.3365876361262467	apixaban	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.033658764	carfilzomib	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.031880796	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.009327235	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.09972967	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.1296485709523321	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.08854582	vernakalant	ncit:C152864	VERNAKALANT	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.026045472	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.002683207	ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.066409365	mexiletine	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
XRCC3	hgnc:12830	XRCC3	PharmGKB	4/5/24	NULL	0.7095631248066825	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.013622434	toremifene	rxcui:38409	TOREMIFENE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	CETRIMONIUM BROMIDE	rxcui:288999	CETRIMONIUM BROMIDE	FALSE	FALSE	FALSE
FGFR3P1	hgnc:21664	FGFR3P1	PharmGKB	4/5/24	NULL	7.501095890813499	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
FIP1L1	hgnc:19124	FIP1L1	PharmGKB	4/5/24	NULL	5.834185692854944	mepolizumab	rxcui:1720597	MEPOLIZUMAB	TRUE	FALSE	FALSE
IL23R	hgnc:19100	IL23R	PharmGKB	4/5/24	NULL	0.921187215	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
FSHR	hgnc:3969	FSHR	PharmGKB	4/5/24	NULL	7.001022831425932	thyrotropin alfa	rxcui:4952	THYROTROPIN ALFA	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	METHIOCARB	ncit:C163673	METHIOCARB	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.062808219	azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	PharmGKB	4/5/24	NULL	0.028252715	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SLC30A8	hgnc:20303	SLC30A8	PharmGKB	4/5/24	NULL	3.750547945406749	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.3409589041278863	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.066005872	disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.05413162	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ABCC6	hgnc:57	ABCC6	PharmGKB	4/5/24	NULL	0.047304208	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
SPG7	hgnc:11237	SPG7	PharmGKB	4/5/24	NULL	1.419126249613364	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
CSPG4	hgnc:2466	CSPG4	PharmGKB	4/5/24	NULL	0.5676504998453459	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	NSC-645827	chembl:CHEMBL95704	CHEMBL:CHEMBL95704	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.019142425	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
BCOR	hgnc:20893	BCOR	PharmGKB	4/5/24	NULL	0.4688184931758437	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	GNF-PF-4853	chembl:CHEMBL599957	CHEMBL:CHEMBL599957	FALSE	FALSE	FALSE
SLC46A1	hgnc:30521	SLC46A1	PharmGKB	4/5/24	NULL	0.6250913242344582	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	SJ000143975	iuphar.ligand:2827	HPTE	FALSE	FALSE	FALSE
TNFAIP3	hgnc:11896	TNFAIP3	PharmGKB	4/5/24	NULL	0.9376369863516874	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
IMPDH1	hgnc:6052	IMPDH1	PharmGKB	4/5/24	NULL	0.062509132	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PERP	hgnc:17637	PERP	PharmGKB	4/5/24	NULL	0.9723642821424908	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.078136416	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.1041818873724097	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
KIR2DS4	hgnc:6336	KIR2DS4	PharmGKB	4/5/24	NULL	0.4688184931758437	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.063415062	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
RALBP1	hgnc:9841	RALBP1	PharmGKB	4/5/24	NULL	0.375054795	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
RALBP1	hgnc:9841	RALBP1	PharmGKB	4/5/24	NULL	0.3061671792168775	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.212581665	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	DOCONEXENT	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
RALBP1	hgnc:9841	RALBP1	PharmGKB	4/5/24	NULL	0.4054646427466756	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
HLA-DRB5	hgnc:4953	HLA-DRB5	PharmGKB	4/5/24	NULL	1.105424657593568	amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	PharmGKB	4/5/24	NULL	0.3365876361262467	leniolisib	rxcui:2633005	LENIOLISIB	TRUE	FALSE	FALSE
SPIDR	hgnc:28971	SPIDR	PharmGKB	4/5/24	NULL	0.3241214273808302	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.9131768910555565	edoxaban	rxcui:1599538	EDOXABAN	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	(+)-ISOBICYCLOGERMACRENAL	chembl:CHEMBL2333548	CHEMBL:CHEMBL2333548	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.4167275494896388	paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.01852776	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.04321619	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
FMO5	hgnc:3773	FMO5	PharmGKB	4/5/24	NULL	0.081597003	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
TYR	hgnc:12442	TYR	DTC	9/2/20	NULL	4.773424657790408	PHENYLTHIOUREA	drugbank:DB03694	N-PHENYLTHIOUREA	FALSE	FALSE	FALSE
CSNK1E	hgnc:2453	CSNK1E	PharmGKB	4/5/24	NULL	4.922594178346359	heroin	rxcui:3304	HEROIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.054243462	nelfinavir	rxcui:134527	NELFINAVIR	TRUE	FALSE	TRUE
CRISPLD2	hgnc:25248	CRISPLD2	PharmGKB	4/5/24	NULL	1.221108633388244	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.1013661606866689	leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
CYP2C18	hgnc:2620	CYP2C18	PharmGKB	4/5/24	NULL	0.5000730593875666	clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	GNF-PF-3537	chembl:CHEMBL601110	CHEMBL:CHEMBL601110	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	PharmGKB	4/5/24	NULL	0.1164249916534246	durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
ERICH3	hgnc:25346	ERICH3	PharmGKB	4/5/24	NULL	1.346350544504987	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.182318303	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
RXFP2	hgnc:17318	RXFP2	DTC	9/2/20	NULL	1.093909817410302	COLFORSIN	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
TPP1	hgnc:2073	TPP1	PharmGKB	4/5/24	NULL	157.5230137070835	cerliponase alfa	rxcui:1922436	CERLIPONASE ALFA	TRUE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	PharmGKB	4/5/24	NULL	1.193356164447602	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	PharmGKB	4/5/24	NULL	0.2625383561784725	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
CPA6	hgnc:17245	CPA6	PharmGKB	4/5/24	NULL	2.692701089009974	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.002864107	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
HNF1B	hgnc:11630	HNF1B	PharmGKB	4/5/24	NULL	1.346350544504987	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.1346350544504987	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
MICB	hgnc:7091	MICB	PharmGKB	4/5/24	NULL	1.093909817410302	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
MICB	hgnc:7091	MICB	PharmGKB	4/5/24	NULL	1.207072901969988	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
NRG3	hgnc:7999	NRG3	PharmGKB	4/5/24	NULL	1.000146118775133	iloperidone	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
EPHA7	hgnc:3390	EPHA7	PharmGKB	4/5/24	NULL	0.1767935058440892	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1458546423213736	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ZNRD1-AS1	hgnc:13924	POLR1HASP	PharmGKB	4/5/24	NULL	2.143170254518142	carbamazepine	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CETP	hgnc:1869	CETP	PharmGKB	4/5/24	NULL	0.2071308530007672	lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1296485709523321	rivaroxaban	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.092118721	nimodipine	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	2-(PHENOXYMETHYL)BENZOTHIAZOLE	chembl:CHEMBL233302	2-(PHENOXYMETHYL)BENZOTHIAZOLE	FALSE	FALSE	FALSE
FZD3	hgnc:4041	FZD3	PharmGKB	4/5/24	NULL	0.9723642821424907	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NME1	hgnc:7849	NME1	PharmGKB	4/5/24	NULL	0.7778914257139926	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.04464938	capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.071928317	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	5.625821918110125	vancomycin	rxcui:11124	VANCOMYCIN	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	ROSIGLITAZONE MALEATE	rxcui:253198	ROSIGLITAZONE MALEATE	TRUE	FALSE	FALSE
SOST	hgnc:13771	SOST	PharmGKB	4/5/24	NULL	1.093909817410302	alendronate	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
DCBLD1	hgnc:21479	DCBLD1	PharmGKB	4/5/24	NULL	0.8334550989792777	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.2734774543525755	dipyrone	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
BIRC2	hgnc:590	BIRC2	DTC	9/2/20	NULL	1.750255707856483	BESTATIN METHYL ESTER	chembl:CHEMBL457092	BESTATIN METHYL ESTER	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.046120045	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
ASL	hgnc:746	ASL	PharmGKB	4/5/24	NULL	2.917092846427472	glycerol phenylbutyrate	rxcui:1368451	GLYCEROL PHENYLBUTYRATE	TRUE	FALSE	FALSE
SHMT1	hgnc:10850	SHMT1	PharmGKB	4/5/24	NULL	0.5556367326528519	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SSTR2	hgnc:11331	SSTR2	PharmGKB	4/5/24	NULL	0.5834185692854945	lutetium (177Lu) oxodotreotide	rxcui:1999335	LUTETIUM LU 177 DOTATATE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	PharmGKB	4/5/24	NULL	0.024041974	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
PROS1	hgnc:9456	PROS1	PharmGKB	4/5/24	NULL	0.6819178082557728	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	PharmGKB	4/5/24	NULL	0.5250767123569451	protease inhibitors	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.7955707762984013	paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	TCMDC-125813	chembl:CHEMBL580076	CHEMBL:CHEMBL580076	FALSE	FALSE	FALSE
PARP11	hgnc:1186	PARP11	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.051731696	NSC-402083	chembl:CHEMBL1546228	CHEMBL:CHEMBL1546228	FALSE	FALSE	FALSE
MTRF1L	hgnc:21051	MTRF1L	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NT5C2	hgnc:8022	NT5C2	PharmGKB	4/5/24	NULL	0.6035364509849942	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.061992528	GS 6201	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.6241137025199848	bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
PON2	hgnc:9205	PON2	PharmGKB	4/5/24	NULL	2.019525816757481	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GLCCI1	hgnc:18713	GLCCI1	PharmGKB	4/5/24	NULL	1.909369863116163	flunisolide	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
FGFBP2	hgnc:29451	FGFBP2	PharmGKB	4/5/24	NULL	3.182283105193606	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.2430910705356227	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.03219848	primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
IKBKG	hgnc:5961	IKBKG	PharmGKB	4/5/24	NULL	2.386712328895204	primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
MYD88	hgnc:7562	MYD88	PharmGKB	4/5/24	NULL	1.591141552596803	ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.326134604	bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
FGFRL1	hgnc:3693	FGFRL1	PharmGKB	4/5/24	NULL	7.501095890813499	brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
ITGB3	hgnc:6156	ITGB3	PharmGKB	4/5/24	NULL	2.800409132570373	tirofiban	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
TK1	hgnc:11830	TK1	PharmGKB	4/5/24	NULL	0.6482428547616604	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	TALC	12-May-16	NULL	1.458546423213736	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.07631929	VARGATEF	wikidata:Q29006632	VARGATEF	FALSE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.1773907812016706	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.1682938180631233	PIVANEX	ncit:C1344	PIVALOYLOXYMETHYLBUTYRATE	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1512704997187101	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1109316997937207	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1232574442152452	ALKS 33	rxcui:2559612	SAMIDORPHAN	TRUE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.2778183663264258	AM-101	chembl:CHEMBL2364609	ESKETAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P52732	hgnc:6388	KIF11	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	ARQ-621	chembl:CHEMBL4303449	ARQ-621	FALSE	FALSE	TRUE
UNIPROT:P24385	hgnc:1582	CCND1	TdgClinicalTrial	Jan-14	NULL	0.024041974	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
UNIPROT:P05412	hgnc:6204	JUN	TdgClinicalTrial	Jan-14	NULL	0.043902735	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	2.218633995874415	ASIMADOLINE	ncit:C72137	ASIMADOLINE	FALSE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	ATI-7505	chembl:CHEMBL2103858	NARONAPRIDE	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	AZD-0837	ncit:C166758	ATECEGATRAN METOXIL	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.07767407	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1278595890479573	FLUOXETINE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P42081	hgnc:1705	CD86	TdgClinicalTrial	Jan-14	NULL	2.333674277141978	BELATACEPT	rxcui:1112973	BELATACEPT	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.4526523382387456	CAP7.1	ncit:C114977	ETOPOSIDE TONIRIBATE	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.063110182	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:P04049	hgnc:9829	RAF1	TdgClinicalTrial	Jan-14	NULL	0.4039051633514962	CHIR-265	iuphar.ligand:5674	CHIR-265	FALSE	FALSE	TRUE
UNIPROT:P15056	hgnc:1097	BRAF	TdgClinicalTrial	Jan-14	NULL	0.1099637093941246	CHIR-265	iuphar.ligand:5674	CHIR-265	FALSE	FALSE	TRUE
UNIPROT:P33765	hgnc:268	ADORA3	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	CF-102	ncit:C79826	NAMODENOSON	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.030368809	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.7395446652914718	CR665	drugbank:DB05155	CR665	FALSE	FALSE	FALSE
UNIPROT:P00326	hgnc:251	ADH1C	TdgClinicalTrial	Jan-14	NULL	0.8751278539282417	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
UNIPROT:P04053	hgnc:2983	DNTT	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	CORDYCEPIN	rxcui:1989289	CORDYCEPIN	FALSE	FALSE	FALSE
UNIPROT:P00813	hgnc:186	ADA	TdgClinicalTrial	Jan-14	NULL	0.032382159	DIPYRIDAMOLE	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.095468493	PAROXETINE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.7160136986685613	ETODOLAC	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.1442518440541057	FENRETINIDE	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
UNIPROT:P00491	hgnc:7892	PNP	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	FORODESINE	ncit:C65755	FORODESINE	FALSE	FALSE	FALSE
UNIPROT:P48051	hgnc:6267	KCNJ6	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	LE-SN38	ncit:C95717	LIPOSOMAL SN-38	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.058471794	LGD-4033	drugbank:DB13934	LIGANDROL	FALSE	FALSE	FALSE
UNIPROT:P07333	hgnc:2433	CSF1R	TdgClinicalTrial	Jan-14	NULL	0.056157937	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.022220766	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	2.143170254518142	LY-517717	drugbank:DB05713	LY-517717	FALSE	FALSE	FALSE
UNIPROT:Q04912	hgnc:7381	MST1R	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	MGCD265	ncit:C77876	GLESATINIB	FALSE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.057260274	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
UNIPROT:Q96P70	hgnc:19425	IPO9	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
UNIPROT:Q9UI26	hgnc:20628	IPO11	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	MKC-1	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	MPI-674	drugbank:DB05749	MPI-674	FALSE	FALSE	FALSE
UNIPROT:Q9NZ20	hgnc:17934	PLA2G3	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	MRX-4	iuphar.ligand:10796	CONTEZOLID ACEFOSAMIL (PARENT)	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.4930297768609811	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1591141552596802	NCX 4016	ncit:C61499	NITRIC OXIDE-RELEASING ACETYLSALICYLIC ACID DERIVATIVE	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1605739181519709	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	NI-0401	chembl:CHEMBL1743020	FORALUMAB	FALSE	FALSE	FALSE
UNIPROT:P29475	hgnc:7872	NOS1	TdgClinicalTrial	Jan-14	NULL	0.4930297768609811	NXN-188	drugbank:DB06096	NXN-188	FALSE	FALSE	FALSE
UNIPROT:P51681	hgnc:1606	CCR5	TdgClinicalTrial	Jan-14	NULL	7.876150685354174	PRO 140	ncit:C137824	LERONLIMAB	FALSE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	PRUCALOPRIDE	rxcui:2107310	PRUCALOPRIDE	TRUE	FALSE	FALSE
UNIPROT:P35499	hgnc:10591	SCN4A	TdgClinicalTrial	Jan-14	NULL	0.052116795	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	1.050153425	SAXAGLIPTIN	rxcui:1546030	SAXAGLIPTIN ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.0296486	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.3201687270469177	TESETAXEL	ncit:C37451	TESETAXEL	FALSE	FALSE	FALSE
UNIPROT:Q02127	hgnc:2867	DHODH	TdgClinicalTrial	Jan-14	NULL	5.527123287967842	TERIFLUNOMIDE	rxcui:1310520	TERIFLUNOMIDE	TRUE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	4.861821410712453	TOSITUMOMAB	rxcui:263010	TOSITUMOMAB	TRUE	FALSE	TRUE
UNIPROT:P09211	hgnc:4638	GSTP1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	CANFOSFAMIDE	ncit:C83581	CANFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.1400204566285186	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.2160809515872201	V3381	chembl:CHEMBL3707400	INDANTADOL	FALSE	FALSE	FALSE
UNIPROT:P26010	hgnc:6162	ITGB7	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	VEDOLIZUMAB	rxcui:1538097	VEDOLIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.1367387271762877	CARPHENAZINE	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.079197091	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.2375912725597036	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.207267123	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.064033745	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.070956312	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.062509132	CLORAZEPATE	rxcui:2353	CLORAZEPATE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.078510274	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.4907258993990139	DIETHYLPROPION	rxcui:3389	DIETHYLPROPION	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	EMEDASTINE	rxcui:28144	EMEDASTINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.078682824	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.038765353	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.081365193	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.064111931	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.4546118721705151	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.037734582	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
UNIPROT:P23415	hgnc:4326	GLRA1	TdgClinicalTrial	Jan-14	NULL	0.1539814405738841	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.6012328767445935	HYDROCORTAMATE	ncit:C65862	HYDROCORTAMATE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.037721028	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.4321619031744403	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.3431873936973496	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.1092771513750145	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	LISDEXAMFETAMINE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.0287871	LISURIDE	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	MARINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.061055432	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.1141471113819445	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1090501998664475	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.087512785	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	MUROMONAB	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.3547815624033412	TRIDIHEXETHYL	rxcui:38617	TRIDIHEXETHYL	TRUE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	0.078793024	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	ZUCLOPENTHIXOL	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	2.072671233	XIMELAGATRAN	ncit:C77996	XIMELAGATRAN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	TRIPELENNAMINE	rxcui:10847	TRIPELENNAMINE	TRUE	FALSE	FALSE
UNIPROT:O43570	hgnc:1371	CA12	TEND	1-Aug-11	NULL	0.8036888454443035	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.3043922970185189	DAPIPRAZOLE	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TEND	1-Aug-11	NULL	0.6141248097742047	DABIGATRAN	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	1.064344687210023	DIPHEMANIL METHYLSULFATE	rxcui:23364	DIPHEMANIL METHYLSULFATE	TRUE	FALSE	FALSE
UNIPROT:P15382	hgnc:6240	KCNE1	TEND	1-Aug-11	NULL	3.000438356	INDAPAMIDE	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.06286838	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
UNIPROT:Q07343	hgnc:8781	PDE4B	TEND	1-Aug-11	NULL	1.166837138570988	ENPROFYLLINE	ncit:C74327	ENPROFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.077827576	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.7160136986685613	ETODOLAC	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TEND	1-Aug-11	NULL	0.1873044158229292	GLIBENCLAMIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1630673019742065	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TEND	1-Aug-11	NULL	0.1223955040459079	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.4070362111294147	FENOTEROL	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.081365193	FLUNITRAZEPAM	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.4546118721705151	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	2.669881588255652	FORASARTAN	ncit:C65749	FORASARTAN	FALSE	FALSE	FALSE
UNIPROT:P47712	hgnc:9035	PLA2G4A	TEND	1-Aug-11	NULL	0.2302968036653267	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TEND	1-Aug-11	NULL	1.131630845596864	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
UNIPROT:P29474	hgnc:7876	NOS3	TEND	1-Aug-11	NULL	0.7501095890813501	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	1.790034246671403	INDECAINIDE	ncit:C65910	INDECAINIDE	TRUE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TEND	1-Aug-11	NULL	0.3195192975802911	KETAMINE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.1790034246671403	KETOROLAC	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.1591141552596803	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1090501998664475	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.087512785	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	1.875273972703375	METOLAZONE	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.066803653	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.071341945	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.051277023	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
RASGRP3	hgnc:14545	RASGRP3	DTC	9/2/20	NULL	10.50153425	[3H]-PHORBOL 12,13-DIBUTYRATE	chembl:CHEMBL27768	CHEMBL:CHEMBL27768	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.023482858	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.011601341	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	L-MIMOSINE	drugbank:DB01055	MIMOSINE	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.1935172158563679	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.046965717	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.072125922	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.068847471	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1553481397505754	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.067317527	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.2386712328895204	OXAPROZIN	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.1193356164447602	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009572521	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.051478109	GUANIDINONALTRINDOLE	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.5000730593875666	PRECLAMOL HYDROCHLORIDE	chembl:CHEMBL1255842	PRECLAMOL HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.089756703	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
NOTCH-4 RECEPTOR	hgnc:7884	NOTCH4	TTD	2020.06.01	NULL	2.917092846427472	LY3039478	ncit:C171871	CRENIGACESTAT	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	0.172722603	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.173866461	APG-115	ncit:C132991	ALRIZOMADLIN	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.022949157	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	1.381780822	AZD5153	ncit:C151943	BIVALENT BRD4 INHIBITOR AZD5153	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.5147810905460245	ARQ 531	ncit:C138066	NEMTABRUTINIB	FALSE	FALSE	FALSE
DUAL SPECIFICITY PROTEIN KINASE TTK	hgnc:10416	RPS27	TTD	2020.06.01	NULL	1.250182648468916	BOS172722	drugbank:DB15498	BOS172722	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	1.419126249613364	CPI-444	ncit:C125659	CIFORADENANT	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.01186614	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	1.909369863116163	SNDX-6352	ncit:C155813	AXATILIMAB	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 BETA	hgnc:5258	HSP90AB1	TTD	2020.06.01	NULL	1.141471113819445	SNX-5422	drugbank:DB06070	SNX-5422	FALSE	FALSE	FALSE
TANKYRASE	hgnc:11941	TNKS	TTD	2020.06.01	NULL	13.12691780892362	2X-121	drugbank:DB16063	2X-121	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	1.050153425	2X-121	drugbank:DB16063	2X-121	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	0.3431873936973496	Sym013	ncit:C131175	ANTI-EGFR/HER2/HER3 MONOCLONAL ANTIBODY MIXTURE SYM013	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.1151484018326633	Sym013	ncit:C131175	ANTI-EGFR/HER2/HER3 MONOCLONAL ANTIBODY MIXTURE SYM013	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE BRAIN	hgnc:7872	NOS1	TTD	2020.06.01	NULL	0.4930297768609811	NXN-188	drugbank:DB06096	NXN-188	FALSE	FALSE	FALSE
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	0.2853677784548614	AZD0284	iuphar.ligand:11711	AZD0284	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.1944728564284981	ITF2357	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005574063	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	1.141471113819445	LEO 124249	chembl:CHEMBL4297507	DELGOCITINIB	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.5114383561918295	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.049864835	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	CGS-12066B	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011012515	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	1.050153425	Teplizumab	rxcui:2621880	TEPLIZUMAB	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	DICHLOFENTHION	chembl:CHEMBL1396626	DICHLOFENTHION	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR A	hgnc:8799	PDGFA	TTD	2020.06.01	NULL	6.563458904461812	Squalamine	ncit:C143004	SQUALAMINE	FALSE	FALSE	FALSE
CHUK	hgnc:1974	CHUK	DTC	9/2/20	NULL	7.501095891	2,6-DIDEHYDROPEPEROMIN B	chembl:CHEMBL559876	2,6-DIDEHYDROPEPEROMIN B	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	SB-205384	chembl:CHEMBL1256667	CHEMBL:CHEMBL1256667	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.015335184	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	GLABRANIN	chembl:CHEMBL253998	GLABRANIN	FALSE	FALSE	FALSE
CARBOXYPEPTIDASE B2	hgnc:2300	CPB2	TTD	2020.06.01	NULL	7.501095891	DS-1040	ncit:C148637	TAFIA INHIBITOR DS-1040B	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.2800409132570373	HONOKIOL	rxcui:2562546	HONOKIOL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	U-37883A	iuphar.ligand:13269	PNU-37883	FALSE	FALSE	FALSE
THYMIC STROMAL LYMPHOPOIETIN	hgnc:30743	TSLP	TTD	2020.06.01	NULL	52.50767123569449	MEDI9929	rxcui:2587789	TEZEPELUMAB	TRUE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	0.750109589	S-707106	ncit:C116320	INSULIN SENSITIZER S-707106	FALSE	FALSE	FALSE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	0.5097832158805291	MB-07811	drugbank:DB15137	VK-2809	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Choline alfoscerate	rxcui:4918	GLYCERYLPHOSPHORYLCHOLINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.045265234	BENZAMIL	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
NUCLEOLIN	hgnc:7667	NCL	TTD	2020.06.01	NULL	11.66837138570988	Itarnafloxin	ncit:C71726	QUARFLOXIN	FALSE	FALSE	TRUE
MEMBRANE COPPER AMINE OXIDASE	hgnc:550	AOC3	TTD	2020.06.01	NULL	1.009762908	Clonidine	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	0.546954909	EXISULIND	ncit:C1239	EXISULIND	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.3271505995993426	Reboxetine	rxcui:60842	REBOXETINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.2191733444543002	Salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1111273465305703	BIBX-1382	ncit:C80868	FALNIDAMOL	FALSE	FALSE	FALSE
DNA TOPOISOMERASE	hgnc:38595	LINC00273	TTD	2020.06.01	NULL	17.50255707856483	Icofungipen	ncit:C65880	ICOFUNGIPEN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.05664258	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	6.300920548	ING-1	drugbank:DB05831	ING-1	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	0.1357664414626878	Tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	4.375639269641208	RUPATADINE	ncit:C73055	RUPATADINE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.044611445	Trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.008301608	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
ALBENDAZOLE MONOOXYGENASE	hgnc:2637	CYP3A4	TTD	2020.06.01	NULL	0.008390488	PMX-53	iuphar.ligand:579	PMX53	FALSE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	0.326134604	PMX-53	iuphar.ligand:579	PMX53	FALSE	FALSE	FALSE
SUBSTANCE-K RECEPTOR	hgnc:11527	TACR2	TTD	2020.06.01	NULL	1.500219178162699	PMX-53	iuphar.ligand:579	PMX53	FALSE	FALSE	FALSE
HISTAMINE N-METHYLTRANSFERASE	hgnc:5028	HNMT	TTD	2020.06.01	NULL	1.875273972703375	Amodiaquine	rxcui:720	AMODIAQUINE	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.2983390411119005	HTS-05058	chembl:CHEMBL261692	CHEMBL:CHEMBL261692	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD4	hgnc:1678	CD4	TTD	2020.06.01	NULL	9.845188356692718	Zanolimumab	ncit:C91701	ZANOLIMUMAB	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	0.092118721	AEE-788	drugbank:DB12558	AEE-788	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.075768645	Ro 31-7453	ncit:C2507	MKC-1	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.1403948428761885	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.1411496538593938	Rufinamide	rxcui:69036	RUFINAMIDE	TRUE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	1.544343271638073	Rilopirox	ncit:C75204	RILOPIROX	FALSE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.068369364	Fenoldopam	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	0.596678082	Ceruletide	ncit:C65309	CERULETIDE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	Mizolastine	rxcui:61455	MIZOLASTINE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.4375639269641208	SIMOCYCLINONE D8	chembl:CHEMBL1235969	SIMOCYCLINONE D8	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	0.8334550989792776	Levallorphan	rxcui:6370	LEVALLORPHAN	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.4717670371580817	SNDX-275	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.078510274	Clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Estriol	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.044878351	Labetalol	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	PH-011685	chembl:CHEMBL126804	CHEMBL:CHEMBL126804	FALSE	FALSE	FALSE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	0.3365876361262467	Miltefosine	rxcui:1494066	MILTEFOSINE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.033412454	Cyproterone	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.4118248724368196	P276-00	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.7242437411819931	Efungumab	ncit:C87763	EFUNGUMAB	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.035800685	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PAK-4 PROTEIN KINASE	hgnc:16059	PAK4	TTD	2020.06.01	NULL	0.6250913242344582	PF-3758309	iuphar.ligand:8937	PF-3758309	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.3860858179095183	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
HLA CLASS I ANTIGEN B-7	hgnc:4932	HLA-B	TTD	2020.06.01	NULL	1.381780822	Velimogene aliplasmid	ncit:C170392	VELIMOGENE ALIPLASMID	FALSE	FALSE	FALSE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.8078103267029924	MK-0752	drugbank:DB12852	MK-0752	FALSE	FALSE	TRUE
CYTOCHROME P450 1B1	hgnc:2597	CYP1B1	TTD	2020.06.01	NULL	1.591141552596803	PINOCEMBRIN	chembl:CHEMBL399910	PINOCEMBRIN	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.2	hgnc:1389	CACNA1B	TTD	2020.06.01	NULL	0.6563458904461813	Hesperidin	rxcui:5281	HESPERIDIN	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	5.250767123569449	PF-232798	drugbank:DB14813	PF-232798	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	HARMAN	chembl:CHEMBL12014	HARMAN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.001750956	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
TRANSFORMING GROWTH FACTOR BETA 2	hgnc:11768	TGFB2	TTD	2020.06.01	NULL	3.750547945	FANG vaccine	ncit:C90552	GEMOGENOVATUCEL-T	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 3	hgnc:11849	TLR3	TTD	2020.06.01	NULL	10.50153424713889	Rintatolimod	ncit:C1001	RINTATOLIMOD	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 2	hgnc:11848	TLR2	TTD	2020.06.01	NULL	7.501095891	OPN-305	ncit:C120554	TOMARALIMAB	FALSE	FALSE	FALSE
INTEGRIN BETA-7	hgnc:6162	ITGB7	TTD	2020.06.01	NULL	5.834185692854944	AMG-181	ncit:C139025	ABRILUMAB	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	2.151953739167807	Olaratumab	rxcui:1855735	OLARATUMAB	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	4-BENZYLOXYANILINE	chembl:CHEMBL1351571	4-BENZYLOXYANILINE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	2.625383561784724	CG-100649	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Chlophedianol	rxcui:21254	CHLOPHEDIANOL	TRUE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	Sym021	ncit:C142865	ANTI-PD-1 MONOCLONAL ANTIBODY SYM021	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.9053046764774912	Valrubicin	rxcui:31435	VALRUBICIN	TRUE	FALSE	TRUE
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	1.009762908	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1172046232939609	RAMATROBAN	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
THYROID PEROXIDASE	hgnc:12015	TPO	TTD	2020.06.01	NULL	8.751278539282415	Carbimazole	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.8204323630577265	Thymoctonan	ncit:C152593	THYMOCTONAN	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.047734247	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
ATP-BINDING CASSETTE TRANSPORTER G2	hgnc:74	ABCG2	TTD	2020.06.01	NULL	0.034184682	Sulfasalazine	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.5585922471882393	Pentolinium	ncit:C77367	PENTOLINIUM	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.2386712328895204	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	1.521961485092594	Cenicriviroc	ncit:C166464	CENICRIVIROC	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.053253216	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.8078103267029922	Florbetapir F-18	rxcui:1427224	FLORBETAPIR F-18	TRUE	FALSE	FALSE
PHOSPHODIESTERASE I BETA	hgnc:3358	ENPP3	TTD	2020.06.01	NULL	26.25383561784724	AGS-16M8F	ncit:C116626	ANTI-ENPP3/MMAF ANTIBODY-DRUG CONJUGATE AGS-16M8F	FALSE	FALSE	FALSE
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	2.386712328895204	MKC-1106-MT	ncit:C77971	IMMUNOTHERAPY REGIMEN MKC-1106-MT	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.5181678082469852	Varlitinib	ncit:C62530	VARLITINIB	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.1609430535959984	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	2.763561643983921	Trenonacog alfa	ncit:C152727	TRENONACOG ALFA	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.252440727	Abaperidone	ncit:C73280	ABAPERIDONE	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Abaperidone	ncit:C73280	ABAPERIDONE	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1988926940746003	Amfepramone	rxcui:3389	DIETHYLPROPION	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.7395446652914718	Amezinium	rxcui:17665	AMEZINIUM	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1512704997187101	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	0.301335273	Capsaicin	rxcui:1992	CAPSAICIN	TRUE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.071585127259071	Certoparin sodium	rxcui:152612	CERTOPARIN SODIUM	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.019332721	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1635752997996713	Estropipate	rxcui:33747	ESTROPIPATE	TRUE	FALSE	FALSE
TYROSINE 3-MONOOXYGENASE	hgnc:11782	TH	TTD	2020.06.01	NULL	0.6250913242344582	L-Phenylalanine	rxcui:8156	PHENYLALANINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.2308029504865691	Moxisylyte	rxcui:10561	MOXISYLYTE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	0.8204323630577265	Rhucin	wikidata:Q29006438	RHUCIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
HISTAMINE RECEPTOR	hgnc:5172	HR	TTD	2020.06.01	NULL	17.50255707856483	Repirinast	ncit:C73053	REPIRINAST	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.061412481	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
C1 ESTERASE INHIBITOR	hgnc:1228	SERPING1	TTD	2020.06.01	NULL	13.12691780892362	Rhucin	wikidata:Q29006438	RHUCIN	FALSE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.8899605294185507	Temocapril hydrochloride	ncit:C99556	TEMOCAPRIL HYDROCHLORIDE	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	STA-5312	ncit:C77066	ROSABULIN	FALSE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	1.458546423213736	AUTO3	drugbank:DB17364	AUTO3	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	3.281729452230906	CP-533536	ncit:C83707	EVATANEPAG	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.2500365296937833	LY-2875358	iuphar.ligand:7748	EMIBETUZUMAB	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	DTC	9/2/20	NULL	0.7501095890813501	BRADANICLINE	ncit:C169814	BRADANICLINE	FALSE	FALSE	FALSE
WEE1-LIKE PROTEIN KINASE	hgnc:12761	WEE1	TTD	2020.06.01	NULL	0.7212592202705288	MK-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	NVP-AUY922	iuphar.ligand:9261	LUMINESPIB	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.9907107780319716	RV001	chembl:CHEMBL1743079	TEPROTUMUMAB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	RG7845	ncit:C116844	FENEBRUTINIB	FALSE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.546954909	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
NEUROTENSIN RECEPTOR TYPE 1	hgnc:8039	NTSR1	TTD	2020.06.01	NULL	5.834185692854944	Meclinertant	ncit:C156766	MECLINERTANT	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	0.1597596487901455	Fasudil	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.6326225450083675	IUPHAR.LIGAND:3221	iuphar.ligand:3221	CP94253	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.3163112725041837	IUPHAR.LIGAND:65	iuphar.ligand:65	(R)-FLUROCARAZOLOL	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.058799184	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.1861974157294131	IUPHAR.LIGAND:67	iuphar.ligand:67	9-OH-RISPERIDONE	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.2692701089009974	IUPHAR.LIGAND:147	iuphar.ligand:147	DOI	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.062065805	IUPHAR.LIGAND:133	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01715937	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.046303061	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:158	iuphar.ligand:158	N-1-ISOPROPYL-5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:3	iuphar.ligand:3	1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.052090944	IUPHAR.LIGAND:142	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:28	iuphar.ligand:28	SB 216641	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:166	iuphar.ligand:166	RO 60-0175	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:67	iuphar.ligand:67	9-OH-RISPERIDONE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.018031481	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.029766254	IUPHAR.LIGAND:189	iuphar.ligand:189	SB 206553	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.069089041	IUPHAR.LIGAND:109	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:166	iuphar.ligand:166	RO 60-0175	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:147	iuphar.ligand:147	DOI	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.019059046	IUPHAR.LIGAND:14	iuphar.ligand:14	GR 127935	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.061412481	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.032055965	IUPHAR.LIGAND:205	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:175	iuphar.ligand:175	SPIRAMIDE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.011555385	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:232	iuphar.ligand:232	[3H]MESULERGINE	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:240	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:225	ncit:C74393	PIBOSEROD	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.072927321	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.074163377	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.034229251	IUPHAR.LIGAND:202	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.034229251	IUPHAR.LIGAND:209	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:11959	iuphar.ligand:11959	EGIS-11150	FALSE	FALSE	FALSE
NCBIGENE:1385	hgnc:2345	CREB1	GuideToPharmacology	2024.1	activator	4.773424657790408	IUPHAR.LIGAND:5183	iuphar.ligand:5183	5-LOX ACTIVATING PROTEIN	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.057574201	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8993	rxcui:7315	NEOSTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:315	hgnc:1611	ACKR4	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:811	iuphar.ligand:811	CCL21	FALSE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:10632	iuphar.ligand:10632	ITACNOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:8120	iuphar.ligand:8120	COMPOUND 13D [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1067229090156392	IUPHAR.LIGAND:7170	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:481	iuphar.ligand:481	NS-49	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:486	iuphar.ligand:486	(+)-CYCLAZOSIN	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:503	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.031479419	IUPHAR.LIGAND:49	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.025183535	IUPHAR.LIGAND:503	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.005638105	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.075550606	IUPHAR.LIGAND:5509	rxcui:7247	NAPHAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.1988926940746003	IUPHAR.LIGAND:7308	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.075550606	IUPHAR.LIGAND:7310	rxcui:10634	TOLAZOLINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.091796628	IUPHAR.LIGAND:522	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.067317527	IUPHAR.LIGAND:503	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:12574	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:11959	iuphar.ligand:11959	EGIS-11150	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:12576	rxcui:18475	ATIPAMEZOLE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.091796628	IUPHAR.LIGAND:521	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.07767407	IUPHAR.LIGAND:516	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:11151	iuphar.ligand:11151	GSK2881078	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.060146244	IUPHAR.LIGAND:425	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.060146244	IUPHAR.LIGAND:377	iuphar.ligand:377	NECA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1804387327687096	IUPHAR.LIGAND:5620	iuphar.ligand:5620	PSB-11	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:466	iuphar.ligand:466	MRS1067	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:390	iuphar.ligand:390	MRE 2029F20	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:5729	iuphar.ligand:5729	[3H]PSB-11	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:593	rxcui:69749	VALSARTAN	TRUE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8178	iuphar.ligand:8178	COMPOUND 16 [PMID: 18945615]	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:6894	iuphar.ligand:6894	ANGIOTENSIN A	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:6176	iuphar.ligand:6176	BANTAG-1	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:6176	iuphar.ligand:6176	BANTAG-1	FALSE	FALSE	FALSE
NCBIGENE:2957	hgnc:4646	GTF2A1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12414	iuphar.ligand:12414	JNJ-65234637	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:9818	iuphar.ligand:9818	ELENBECESTAT	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:6931	iuphar.ligand:6931	AZD3839	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:8699	ncit:C152868	VERUBECESTAT	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.1339481409073839	IUPHAR.LIGAND:509	rxcui:66887	RACEPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:2487	iuphar.ligand:2487	LTB4	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:7521	iuphar.ligand:7521	COMPOUND 36 [PMID: 24000170]	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:7522	iuphar.ligand:7522	COMPOUND 38 [PMID: 24000170]	FALSE	FALSE	FALSE
NCBIGENE:1947	hgnc:3226	EFNB1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:6044	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:5716	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.059397818	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:10629	ncit:C156173	ORELABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:10464	ncit:C175777	ELSUBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:654	iuphar.ligand:654	B-9858	FALSE	FALSE	FALSE
NCBIGENE:1949	hgnc:3228	EFNB3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8112	iuphar.ligand:8112	COMPOUND 2-13-1 [PMID: 24900824]	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:3765	iuphar.ligand:3765	[125I][TYR8]BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:9451	iuphar.ligand:9451	DF2593A	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:574	iuphar.ligand:574	C5A DES-ARG	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5779	iuphar.ligand:5779	C089	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:12514	iuphar.ligand:12514	BM221	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.01140975	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:1557	hgnc:2621	CYP2C19	GuideToPharmacology	2024.1	inhibitor	0.004716823	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:5770	iuphar.ligand:5770	CHIPS-(28-149)	FALSE	FALSE	FALSE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:3774	iuphar.ligand:3774	[125I]C5A (HUMAN)	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.059532507	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NCBIGENE:1999	hgnc:3318	ELF3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1997	hgnc:3316	ELF1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8050	iuphar.ligand:8050	PF-4800567	FALSE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	activator	2.917092846427472	IUPHAR.LIGAND:4318	iuphar.ligand:4318	SZ(+)-(S)-202-791	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	RIMCAZOLE	ncit:C152218	RIMCAZOLE	FALSE	FALSE	FALSE
NCBIGENE:534	hgnc:862	ATP6V1G2	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2440	iuphar.ligand:2440	CD2+	FALSE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	0.3088686543276147	IUPHAR.LIGAND:2522	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
NCBIGENE:2349	hgnc:2535	CTSH	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8613	iuphar.ligand:8613	COMPOUND 1B [PMID: 16290936]	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	modulator	0.6908904109959803	IUPHAR.LIGAND:9188	iuphar.ligand:9188	PEPCAN-12	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:11185	ncit:C175798	ILACIRNON	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.09741683	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:783	iuphar.ligand:783	TAK-779	FALSE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8217	iuphar.ligand:8217	COMPOUND 77 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4313	iuphar.ligand:4313	SULFONAMIDE-01	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	WAY-100135	iuphar.ligand:79	WAY-100135	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:7141	rxcui:20343	CARPROFEN	TRUE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:10377	iuphar.ligand:10377	CP-316,311	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:919	iuphar.ligand:919	UROCORTIN 1	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	0.5000730593875667	IUPHAR.LIGAND:758	iuphar.ligand:758	CCL5	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	SB-215505	iuphar.ligand:190	SB 215505	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8500	ncit:C169874	DANIRIXIN	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:834	iuphar.ligand:834	NSC 157449	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3677	iuphar.ligand:3677	[125I]CXCL1 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:6045	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:5952	iuphar.ligand:5952	CDK4 INHIBITOR III	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001907844	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:8176	iuphar.ligand:8176	BS-194	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:8007	iuphar.ligand:8007	BX-912	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:8114	drugbank:DB07149	(7S)-2-(2-AMINOPYRIMIDIN-4-YL)-7-(2-FLUOROETHYL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:10081	iuphar.ligand:10081	KINASE INHIBITOR 2 [PMID: 30199702]	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002861765	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:8176	iuphar.ligand:8176	BS-194	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:7379	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:1360	hgnc:2299	CPB1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8310	rxcui:2286252	OSILODROSTAT	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
NCBIGENE:1366	hgnc:2049	CLDN7	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:11381	ncit:C90792	TALAROZOLE	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:7554	rxcui:352372	DEXMETHYLPHENIDATE	TRUE	FALSE	FALSE
NCBIGENE:3002	hgnc:4709	GZMB	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9933	iuphar.ligand:9933	NSC 780521	FALSE	FALSE	FALSE
NCBIGENE:2484	ncbigene:2484	FRV1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8879	iuphar.ligand:8879	RBM2-1B	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.074163377	2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE	chembl:CHEMBL1255936	CHEMBL:CHEMBL1255936	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:1609	iuphar.ligand:1609	DSLET	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1622	iuphar.ligand:1622	DYNORPHIN B	FALSE	FALSE	FALSE
NCBIGENE:2603	hgnc:2861	DHFR	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:6837	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
NCBIGENE:1397	hgnc:2361	CRIP2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524936	IUPHAR.LIGAND:5277	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
NCBIGENE:1397	hgnc:2361	CRIP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5255	iuphar.ligand:5255	RHC80267	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	AM-404	iuphar.ligand:12556	AM404	FALSE	FALSE	FALSE
NCBIGENE:2920	hgnc:4603	CXCL2	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:11795	iuphar.ligand:11795	SLR14	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.025003653	IUPHAR.LIGAND:7279	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.009832897	IUPHAR.LIGAND:2	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.2302968036653267	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:6077	iuphar.ligand:6077	A68930	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:8127	iuphar.ligand:8127	COMPOUND 3B [PMID: 23454515]	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002447226	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
NCBIGENE:2999	hgnc:4710	GZMH	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9933	iuphar.ligand:9933	NSC 780521	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016959842	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:10689	iuphar.ligand:10689	COMPOUND 2-2C [PMID: 32003560]	FALSE	FALSE	FALSE
NCBIGENE:1831	hgnc:3051	TSC22D3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984016	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:1822	hgnc:3033	ATN1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:1828	hgnc:3048	DSG1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8141	iuphar.ligand:8141	COMPOUND 66 [PMID: 19788238]	FALSE	FALSE	FALSE
NCBIGENE:2826	hgnc:4474	CCR10	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:8025	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
TTR	hgnc:12405	TTR	DTC	9/2/20	NULL	8.751278539282415	ETHYL CAFFEATE	chembl:CHEMBL17347	ETHYL CAFFEATE	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9944	iuphar.ligand:9944	MM-433593	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10248	iuphar.ligand:10248	ASP8477	FALSE	FALSE	FALSE
NCBIGENE:2022	hgnc:3349	ENG	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9403	iuphar.ligand:9403	RO3280	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1058	rxcui:164	ACETATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	BENZTHIAZIDE	rxcui:19008	BENZTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:2365	hgnc:3873	FRA1F	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9893	iuphar.ligand:9893	COMPOUND 9 [PMID: 20718420]	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:8123	iuphar.ligand:8123	COMPOUND 1D [PMID: 21493067]	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8862	iuphar.ligand:8862	BLU-9931	FALSE	FALSE	FALSE
NCBIGENE:3175	hgnc:8138	ONECUT1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12610	iuphar.ligand:12610	COMPOUND 19B [PMID: 37058391]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:5970	iuphar.ligand:5970	FLT-3 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.019534104	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:10131	iuphar.ligand:10131	UNC4203	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:12334	iuphar.ligand:12334	COMPOUND 25C [PMID: 36649216]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:11134	iuphar.ligand:11134	TTT-3002	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:5833	iuphar.ligand:5833	AG-09/1	FALSE	FALSE	FALSE
NCBIGENE:1606	hgnc:2849	DGKA	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8659	iuphar.ligand:8659	COMPOUND 8D [PMID: 15027864]	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:5842	iuphar.ligand:5842	FMET-ILE-VAL-ILE-LEU	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	0.1136529680426287	IUPHAR.LIGAND:5826	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:3933	iuphar.ligand:3933	ASPIRIN TRIGGERED LIPOXIN A4	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.2333674277141978	IUPHAR.LIGAND:1888	iuphar.ligand:1888	U46619	FALSE	FALSE	FALSE
NCBIGENE:234	hgnc:4044	FZD6	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:3548	iuphar.ligand:3548	WNT-5A	FALSE	FALSE	FALSE
NCBIGENE:236	hgnc:425	AKR1B1P2	GuideToPharmacology	2024.1	antibody	5.250767124	IUPHAR.LIGAND:10197	iuphar.ligand:10197	VANTICTUMAB	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.045226246	IUPHAR.LIGAND:4090	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4095	iuphar.ligand:4095	&ALPHA;5IA	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:4296	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.037003292	IUPHAR.LIGAND:4193	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1565523888959287	IUPHAR.LIGAND:4348	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6076	iuphar.ligand:6076	J20 (GALANIN ANALOGUE)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6117	iuphar.ligand:6117	[125I][TYR26]GALANIN (PIG)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:3876	iuphar.ligand:3876	GALANIN(2-29) (RAT/MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6117	iuphar.ligand:6117	[125I][TYR26]GALANIN (PIG)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6109	iuphar.ligand:6109	[N-ME,DES-SAR]GAL-B2	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3900	iuphar.ligand:3900	M871	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.2035181055647073	IUPHAR.LIGAND:7068	rxcui:23033	DIFLORASONE DIACETATE	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.305277158	IUPHAR.LIGAND:2871	rxcui:3256	DESOXYCORTICOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:9715	iuphar.ligand:9715	BI 653048	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.6563458904461812	IUPHAR.LIGAND:4304	iuphar.ligand:4304	S18986	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:4141	iuphar.ligand:4141	ATPO	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.1221108633388244	IUPHAR.LIGAND:7059	rxcui:1348	BECLOMETHASONE DIPROPIONATE	TRUE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:4258	iuphar.ligand:4258	MSVIII-19	FALSE	FALSE	FALSE
NCBIGENE:453	hgnc:771	ASS1P8	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:4075	iuphar.ligand:4075	[3H]SYM2081	FALSE	FALSE	FALSE
NCBIGENE:454	hgnc:772	ASS1P9	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:4231	ncit:C79132	KAINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:5581	iuphar.ligand:5581	[D-LYS6]GNRH-II	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4491	iuphar.ligand:4491	[3H]SB-733993	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1178	iuphar.ligand:1178	NBI-42902	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	0.1166837138570988	IUPHAR.LIGAND:2820	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1187	iuphar.ligand:1178	NBI-42902	FALSE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	0.9546849315580819	IUPHAR.LIGAND:3306	iuphar.ligand:3306	OLEANOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4852	iuphar.ligand:4852	[ASU7,23']&BETA;-ANP-(7-28)	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:11118	drugbank:DB14979	MARTINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:7916	iuphar.ligand:7916	SANTACRUZAMATE A	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:11118	drugbank:DB14979	MARTINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:7491	iuphar.ligand:7491	TMP269	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.3201687270469177	IUPHAR.LIGAND:11120	iuphar.ligand:11120	ACY-738	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.3977853881492008	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:9702	iuphar.ligand:9702	TUBASTATIN A	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.1909369863116163	IUPHAR.LIGAND:9663	iuphar.ligand:9663	KA1010	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:1219	iuphar.ligand:1219	BU-E 47	FALSE	FALSE	FALSE
NCBIGENE:2034	hgnc:3374	EPAS1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8128	iuphar.ligand:8128	COMPOUND 1A [PMID: 24900749]	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1195	iuphar.ligand:1195	2-(3-CHLOROPHENYL)HISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.2573905452730122	IUPHAR.LIGAND:1241	iuphar.ligand:1241	N-[3H]METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:1265	iuphar.ligand:1265	CIPROXIFAN	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1255	iuphar.ligand:1255	PROXYFAN	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1255	iuphar.ligand:1255	PROXYFAN	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.088248187	IUPHAR.LIGAND:2424	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5562	iuphar.ligand:5562	GSK494581A	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:11210	iuphar.ligand:11210	PSB-16434	FALSE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:5135	rxcui:1311670	PIMAGEDINE	FALSE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9578	iuphar.ligand:9578	SR8185	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:12441	iuphar.ligand:12441	(&PLUSMN;)-EQUOL	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12443	iuphar.ligand:12443	ERIODICTYOL CHALCONE	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:7793	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:8309	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.041508041	IUPHAR.LIGAND:9600	iuphar.ligand:9600	MIVAVOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.069180068	IUPHAR.LIGAND:11624	iuphar.ligand:11624	NINGETINIB	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1289	iuphar.ligand:1289	KISSPEPTIN-9	FALSE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	activator	1.875273972703375	IUPHAR.LIGAND:10337	iuphar.ligand:10337	GI‐530159	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:2321	iuphar.ligand:2321	UCL1848	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:7677	iuphar.ligand:7677	PD-307243	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:10456	iuphar.ligand:10456	ZORIFERTINIB	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:2590	iuphar.ligand:2590	HMR-1556	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	0.5048814541893701	IUPHAR.LIGAND:2387	iuphar.ligand:2387	PIP2	FALSE	FALSE	FALSE
NCBIGENE:2886	hgnc:4567	GRB7	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10358	iuphar.ligand:10358	GSK065	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:12706	drugbank:DB15498	BOS172722	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:10151	iuphar.ligand:10151	NEOLYMPHOSTIN A	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:8172	iuphar.ligand:8172	COMPOUND 7 [PMID: 22464456]	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:11114	iuphar.ligand:11114	DCLK1-IN-1	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:11665	iuphar.ligand:11665	XMD-12	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8295	iuphar.ligand:8295	PF-06454589	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:11134	iuphar.ligand:11134	TTT-3002	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:11314	iuphar.ligand:11314	CPY	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:2748	iuphar.ligand:2748	DESMOSTEROL	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:11313	iuphar.ligand:11313	CPX	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8589	iuphar.ligand:8589	ONO-9780307	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:8912	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:2671	hgnc:4236	GFER	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:8229	iuphar.ligand:8229	IOX2	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11516	iuphar.ligand:11516	TAK-418	FALSE	FALSE	FALSE
NCBIGENE:2681	hgnc:4253	GGTA1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10141	iuphar.ligand:10141	KDM5 INHIBITOR N71	FALSE	FALSE	FALSE
NCBIGENE:2094	ncbigene:2094	ERVT4	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8045	drugbank:DB07430	(10R)-10-METHYL-3-(6-METHYLPYRIDIN-3-YL)-9,10,11,12-TETRAHYDRO-8H-[1,4]DIAZEPINO[5',6':4,5]THIENO[3,2-F]QUINOLIN-8-ONE	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:3827	iuphar.ligand:3827	[3H]MCH (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:7753	iuphar.ligand:7753	4-ARYLPHTHALAZIN-1(2H)-3,4-DI-F	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:3844	iuphar.ligand:3844	[125I][PHE13,TYR19]MCH	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1307	iuphar.ligand:1307	[AVA9,10,AVA14,15]-AC-HMCH6-16-NH2	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1317	iuphar.ligand:1317	[125I]S36057	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6220	iuphar.ligand:6220	MNI-136	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6348	iuphar.ligand:6348	COMPOUND 23I [PMID: 17929793]	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	inhibitor	0.1312691780892362	IUPHAR.LIGAND:6495	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:8058	iuphar.ligand:8058	JNK-IN-8	FALSE	FALSE	FALSE
NCBIGENE:2071	hgnc:3435	ERCC3	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:285	iuphar.ligand:285	(&PLUSMN;)YM796	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.092118721	IUPHAR.LIGAND:294	rxcui:194	ACETYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:12486	iuphar.ligand:12486	[3H]IPEROXO	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.138178082	IUPHAR.LIGAND:348	iuphar.ligand:348	THIOCHROME	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:8586	iuphar.ligand:8586	AE9C90CB	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:323	iuphar.ligand:323	HEXOCYCLIUM	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:330	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.099446347	IUPHAR.LIGAND:294	rxcui:194	ACETYLCHOLINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:12486	iuphar.ligand:12486	[3H]IPEROXO	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:344	iuphar.ligand:344	N-CHLOROMETHYL-BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:307	iuphar.ligand:307	4-DAMP	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:302	iuphar.ligand:302	OXOTREMORINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.054243462	IUPHAR.LIGAND:7319	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:310	iuphar.ligand:310	HEXAHYDROSILADIFENIDOL	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:3260	iuphar.ligand:318	[3H]QNB	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:330	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.054243462	IUPHAR.LIGAND:7319	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.1988926940746003	IUPHAR.LIGAND:7632	iuphar.ligand:7632	VU0119498	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.066297565	IUPHAR.LIGAND:325	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:8586	iuphar.ligand:8586	AE9C90CB	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:7483	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1353	iuphar.ligand:1353	S24014	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.072324616	IUPHAR.LIGAND:7319	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.28382525	IUPHAR.LIGAND:7712	iuphar.ligand:7712	AZD7325	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:12733	iuphar.ligand:12733	EG-1-230	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:10724	iuphar.ligand:10724	MT-45	FALSE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:2614	iuphar.ligand:2614	ATX-II	FALSE	FALSE	FALSE
NCBIGENE:3004	hgnc:4712	GZMM	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:9932	iuphar.ligand:9932	SETANAXIB	FALSE	FALSE	FALSE
NCBIGENE:1749	hgnc:2918	DLX5	GuideToPharmacology	2024.1	NULL	4.375639269641208	IUPHAR.LIGAND:4845	iuphar.ligand:4845	[125I]ANP (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	modulator	1.810609352954982	IUPHAR.LIGAND:3966	iuphar.ligand:3966	JNJ1930942	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:3965	iuphar.ligand:3965	&ALPHA;-CONOTOXIN IMI	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2113	iuphar.ligand:2113	[PHE(ME)7]NEUROKININ B	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:2126	iuphar.ligand:2126	[PRO7]NEUROKININ B	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:8867	iuphar.ligand:8867	SR16835	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1471	iuphar.ligand:1471	NEUROMEDIN U-25	FALSE	FALSE	FALSE
NCBIGENE:3057	ncbigene:3057	HCL2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10154	iuphar.ligand:10154	ML385	FALSE	FALSE	FALSE
NCBIGENE:2693	hgnc:4267	GHSR	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8783	iuphar.ligand:8783	COMPOUND 26 [PMID: 21733693]	FALSE	FALSE	FALSE
NCBIGENE:1223	hgnc:10955	SLCO2A1	GuideToPharmacology	2024.1	NULL	2.625383561784725	IUPHAR.LIGAND:1916	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:1226	hgnc:10953	SLCO4A1	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:4748	ncit:C47521	ESTROPIPATE	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.2386712328895204	IUPHAR.LIGAND:2169	ncit:C87380	ARGIPRESTOCIN	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:2192	iuphar.ligand:2192	LS-192629	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2255	iuphar.ligand:2255	[MPA1,D-TYR(ET)2,D-TIC7,AIB9]OT	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:2202	ncit:C132046	NELIVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2241	iuphar.ligand:2241	L-365,209	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	modulator	1.693795846312725	IUPHAR.LIGAND:5808	iuphar.ligand:5808	BMS COMPOUND 16 [PMID:23368907]	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1740	iuphar.ligand:1740	(N)METHANOCARBA-UTP	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2264	iuphar.ligand:2264	MAXADILAN	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2268	iuphar.ligand:2268	PG 97-269	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1851	iuphar.ligand:1851	BN 50739	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:4489	iuphar.ligand:4489	[11C]GLYSAR	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:11370	iuphar.ligand:11370	(3,5)-[19F]2-PHE-&PSI;-ALA	FALSE	FALSE	FALSE
NCBIGENE:3171	hgnc:5023	FOXA3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11399	iuphar.ligand:11399	COMPOUND 20 [PMID: 25091930]	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:2716	iuphar.ligand:2716	GW2433	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:3441	iuphar.ligand:3441	GSK0660	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2657	iuphar.ligand:2657	LY-510929	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.015627283	IUPHAR.LIGAND:1909	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:11843	iuphar.ligand:11843	COMPOUND 5 [PMID: 34779204]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.098328972	IUPHAR.LIGAND:10151	iuphar.ligand:10151	NEOLYMPHOSTIN A	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:8805	iuphar.ligand:8805	COMPOUND 82 [PMID: 21332118]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:8382	iuphar.ligand:8382	VS-5584	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:10151	iuphar.ligand:10151	NEOLYMPHOSTIN A	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:8527	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.085796848	IUPHAR.LIGAND:8059	iuphar.ligand:8059	AZD6482	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:8805	iuphar.ligand:8805	COMPOUND 82 [PMID: 21332118]	FALSE	FALSE	FALSE
NCBIGENE:1294	hgnc:2214	COL7A1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:5285	rxcui:24506	VINPOCETINE	FALSE	FALSE	FALSE
NCBIGENE:2164	ncbigene:2164	F13A3	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8444	iuphar.ligand:8444	ISA-2011B	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12003	ncit:C177065	LENRISPODUN	FALSE	FALSE	FALSE
NCBIGENE:1305	hgnc:2190	COL13A1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:5154	iuphar.ligand:5154	BRL50481	FALSE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11946	iuphar.ligand:11946	AZD9574	FALSE	FALSE	FALSE
NCBIGENE:3145	hgnc:4982	HMBS	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12020	iuphar.ligand:12020	WNT-C59	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:2803	iuphar.ligand:2803	5&BETA;-CHOLESTANE-3&ALPHA;,7&ALPHA;,12&ALPHA;-TRIOL	FALSE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7805	iuphar.ligand:7805	AZ4800	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:2769	iuphar.ligand:2769	SCHISANDRIN A	FALSE	FALSE	FALSE
NCBIGENE:2388	hgnc:3900	FRA4A	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12689	iuphar.ligand:12689	MK-0616	FALSE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12373	iuphar.ligand:12373	NARMAFOTINIB	FALSE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9763	iuphar.ligand:9763	CONTELTINIB	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1807	iuphar.ligand:1807	[PHE23]PTH-(1-34) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1800	iuphar.ligand:1800	[ILE5,TRP23]PTHRP-(3-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1801	iuphar.ligand:1801	[ILE5,TRP23]PTHRP-(4-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.02302968	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	modulator	3.088686543276147	IUPHAR.LIGAND:10643	iuphar.ligand:10643	COMPOUND 25 [ZHANG ET AL., 2020]	FALSE	FALSE	FALSE
NCBIGENE:1527	hgnc:2563	TEX28	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:8163	iuphar.ligand:8163	COMPOUND 33 [PMID: 19364658]	FALSE	FALSE	FALSE
NCBIGENE:1855	hgnc:3084	DVL1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8770	iuphar.ligand:8770	ILLUDALIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1525	hgnc:2559	CXADR	GuideToPharmacology	2024.1	inhibitor	0.8334550989792778	IUPHAR.LIGAND:12721	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:11912	iuphar.ligand:11912	DOTA/EU RELAXIN-3	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:3789	iuphar.ligand:3789	[125I]RELAXIN-3-B/INSL5 A CHIMERA	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:8346	iuphar.ligand:8346	A(4-24)(B7-24)H2	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	modulator	3.088686543276147	IUPHAR.LIGAND:9494	iuphar.ligand:9494	CYM-5541	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:9494	iuphar.ligand:9494	CYM-5541	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10311	iuphar.ligand:10311	CYM-50308	FALSE	FALSE	FALSE
NCBIGENE:2197	hgnc:3597	FAU	GuideToPharmacology	2024.1	inhibitor	0.068191781	IUPHAR.LIGAND:5678	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:3200	hgnc:5104	HOXA3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11995	ncit:C119743	UPROLESELAN	FALSE	FALSE	FALSE
NCBIGENE:2225	hgnc:11408	STK4	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12168	iuphar.ligand:12168	IHMT-MST1-58	FALSE	FALSE	FALSE
NCBIGENE:2213	hgnc:3618	FCGR2B	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9692	iuphar.ligand:9692	STK16-IN-1	FALSE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:10333	ncit:C103826	TALADEGIB	FALSE	FALSE	TRUE
NCBIGENE:3096	hgnc:4920	HIVEP1	GuideToPharmacology	2024.1	NULL	10.50153424713889	IUPHAR.LIGAND:12256	iuphar.ligand:12256	COMPOUND 37 [PMID: 36384290]	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:8070	iuphar.ligand:8070	P505-15	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3103	iuphar.ligand:3103	NB-598	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3123	iuphar.ligand:3123	COMPOUND 32 [PMID: 19191557]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5639	iuphar.ligand:5639	GA-DOTA-NOC	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2008	iuphar.ligand:2008	CST-17	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:2029	iuphar.ligand:2029	[L-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2080	iuphar.ligand:2080	H-C[CYS-PHE-LAGL(N&BETA;ME,BENZOYL)-TRP-LYS-THR-PHE-CYS]-OH	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2022	iuphar.ligand:2022	[125I]CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:2740	hgnc:4324	GLP1R	GuideToPharmacology	2024.1	NULL	0.1591141552596802	IUPHAR.LIGAND:12308	iuphar.ligand:12308	A947	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:12190	ncit:C171734	RALMITARONT	FALSE	FALSE	FALSE
NCBIGENE:2240	hgnc:11732	TESK2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8117	iuphar.ligand:8117	COMPOUND 31 [PMID: 22902653]	FALSE	FALSE	FALSE
NCBIGENE:2247	hgnc:3676	FGF2	GuideToPharmacology	2024.1	inhibitor	0.012448476	IUPHAR.LIGAND:5711	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:1795	hgnc:2989	DOCK3	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:8120	iuphar.ligand:8120	COMPOUND 13D [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:4255	iuphar.ligand:4255	ML204	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.4102161815288632	IUPHAR.LIGAND:10285	iuphar.ligand:10285	CLEMIZOLE	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:10288	iuphar.ligand:10288	M084	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.1025540453822158	IUPHAR.LIGAND:2433	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
NCBIGENE:502	hgnc:13357	MCOLN2	GuideToPharmacology	2024.1	activator	2.917092846427472	IUPHAR.LIGAND:6386	iuphar.ligand:6386	ML SA1	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.4605936073306534	IUPHAR.LIGAND:4261	iuphar.ligand:4261	NADA	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:7820	iuphar.ligand:7820	AZD1386	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4311	iuphar.ligand:4311	SB705498	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.3723948314588262	IUPHAR.LIGAND:9427	ncit:C116074	EMPESERTIB	FALSE	FALSE	FALSE
NCBIGENE:1031	hgnc:1789	CDKN2C	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:5826	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
NCBIGENE:2428	hgnc:3938	FRA9D	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:12224	iuphar.ligand:12224	COMPOUND 61 [PMID: 36221183]	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:2166	iuphar.ligand:2166	TOLYACETYL-C[DCYS-APA-DTRP-ORN-VAL-CYS]-HIS-AMIDE	FALSE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:4763	iuphar.ligand:4763	[125I]7-AZIDO-8-IODOKETANSERINE	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2275	iuphar.ligand:2275	PHV	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2258	iuphar.ligand:2258	PACAP-38	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:2274	iuphar.ligand:2274	PHM	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2778183663264258	IUPHAR.LIGAND:2185	iuphar.ligand:2185	D[D-PHE2]AVP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2216	iuphar.ligand:2216	D(CH2)5[D-TYR(ET)2,VAL4,TYR-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:1530	iuphar.ligand:1530	SR120819A	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1527	iuphar.ligand:1527	[LEU31,PRO34]PYY (HUMAN)	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	0.082043236	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.2778183663264258	ALPELISIB	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.010289569	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.1547594520630995	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.4022765134992723	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	CIViC	10-Apr-24	NULL	0.088396753	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	2.341819737097098	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	0.6241137025199848	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	CIViC	10-Apr-24	NULL	1.831662950082366	LAROTRECTINIB	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.7369497717290455	ERDAFITINIB	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.8649519486500064	ERDAFITINIB	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.5303805175322677	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	1.372749574789398	DULIGOTUZUMAB	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
FGFR4	hgnc:3691	FGFR4	CIViC	10-Apr-24	NULL	1.117184494376478	FGFR INHIBITOR ASP5878	ncit:C122719	FGFR INHIBITOR ASP5878	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.546954909	SOTORASIB	rxcui:2550714	SOTORASIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.3241214273808302	K 252A	ncit:C1382	K 252A	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.0287871	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.2160809515872201	AG1295	iuphar.ligand:5914	AG 1295	FALSE	FALSE	TRUE
NUDT15	hgnc:23063	NUDT15	CIViC	10-Apr-24	NULL	0.7955707762984016	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.042741287	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
BBOX1	hgnc:964	BBOX1	DTC	9/2/20	NULL	35.00511415712966	BENZENE SELENOIC ACID	chembl:CHEMBL39469	BENZENE SELENOIC ACID	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.061628722	PI3K/BET INHIBITOR LY294002	ncit:C148229	PI3K/BET INHIBITOR LY294002	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.3968833804663227	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.218327115	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.060772768	PHOSPHATIDYLINOSITIDE 3-KINASE INHIBITOR	ncit:C2152	PHOSPHATIDYLINOSITIDE 3-KINASE INHIBITOR	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.043180651	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.02505934	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	CIViC	10-Apr-24	NULL	0.02540284	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
XRCC1	hgnc:12828	XRCC1	CIViC	10-Apr-24	NULL	0.05751114	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
WEE1	hgnc:12761	WEE1	CIViC	10-Apr-24	NULL	0.5048814541893701	PLATINUM COMPOUND	ncit:C1450	PLATINUM COMPOUND	FALSE	FALSE	TRUE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.018540844	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
RHEB	hgnc:10011	RHEB	CIViC	10-Apr-24	NULL	0.4605936073306534	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.027811267	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
DDR2	hgnc:2731	DDR2	DoCM	10-Apr-24	NULL	1.067952635302261	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	1.336059069138614	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	DoCM	10-Apr-24	NULL	0.5672124979164529	PKC412	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	DoCM	10-Apr-24	NULL	0.3472729579080323	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.4565884455277782	MTI-31	chembl:CHEMBL4594431	MTI-31	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.038049037	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	SB590885	iuphar.ligand:9389	SB590885	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.5498185469706229	TW-37	drugbank:DB17059	TW-37	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	LTT462	ncit:C126687	RINETERKIB	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.036087747	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	VE800	ncit:C167393	COMMENSAL BACTERIAL STRAIN FORMULATION VE800	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.049983504	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2199274187882492	VX-11e	iuphar.ligand:9375	VTX-11E	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1973972602845657	Brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.021534247	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	1.105424657593568	SSR128129E	iuphar.ligand:7850	SSR128129E	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	1.467605717767858	Tofacitinib	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	2.282942227638891	Ritlecitinib	rxcui:2641595	RITLECITINIB	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.072994909	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.6721614540713904	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.019844169	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.4102161815288632	CYC065	ncit:C123902	FADRACICLIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DIGOXIGENIN	drugbank:DB03671	DIGOXIGENIN	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	1.312691780892362	GDC-0575	ncit:C116845	CHK1 INHIBITOR GDC-0575	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.100976291	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.032016873	Cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	2.763561643983921	PRT1419	ncit:C176964	MYELOID CELL LEUKEMIA 1 INHIBITOR PRT1419	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1750255707856483	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	Pegylated liposomal doxorubicin	rxcui:214525	DOXORUBICIN LIPOSOME	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.088396753	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	U0126	iuphar.ligand:5282	U0126	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.045579576	Panulisib	ncit:C104292	PANULISIB	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	BGT226	ncit:C74073	PI3K INHIBITOR BGT226	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	CCT128930	chembl:CHEMBL263664	CHEMBL:CHEMBL263664	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	AZD5991	iuphar.ligand:11783	AZD5991	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	KU-60019	iuphar.ligand:8041	KU-60019	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.3889457128569962	FLUORESCEIN DIACETATE	chembl:CHEMBL1492044	FLUORESCEIN DIACETATE	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.064505739	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.009460842	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.05913026	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CancerCommons	25-Jul-13	inhibitor	2.341819737097098	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	CLORAZEPATE DIPOTASSIUM	rxcui:2607	CLORAZEPATE DIPOTASSIUM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.033919684	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.034727296	ESZOPICLONE	rxcui:461016	ESZOPICLONE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.020351811	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.005707356	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.019447286	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.033658764	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.033232703	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.03409589	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006987979	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.075010959	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.073266518	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.073266518	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.048844345	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	METHYPRYLON	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.049457775	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.018699313	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.019710087	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.016959842	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.018006746	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	DNDI1417434	chembl:CHEMBL394883	CHEMBL:CHEMBL394883	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.055155117	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.042898424	TETRACYCLINE	rxcui:10395	TETRACYCLINE	TRUE	FALSE	FALSE
IL2RG	hgnc:6010	IL2RG	ChEMBL	33	agonist	0.5250767123569451	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	agonist	0.4039051633514962	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
CSF2RA	hgnc:2435	CSF2RA	ChEMBL	33	agonist	11.66837138570988	SARGRAMOSTIM	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.1470803115845784	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	agonist	0.3889457128569963	FINGOLIMOD HYDROCHLORIDE	rxcui:1012891	FINGOLIMOD HYDROCHLORIDE	TRUE	FALSE	FALSE
S1PR5	hgnc:14299	S1PR5	ChEMBL	33	agonist	2.625383561784725	FINGOLIMOD HYDROCHLORIDE	rxcui:1012891	FINGOLIMOD HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.025427444	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	QUINIDINE GLUCONATE	rxcui:35220	QUINIDINE GLUCONATE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.023080295	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.039068208	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	DTC	9/2/20	NULL	0.5173169579871378	GLIQUIDONE	rxcui:25793	GLIQUIDONE	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.028413242	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.039068208	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.043866058	ORPHENADRINE CITRATE	rxcui:7716	ORPHENADRINE CITRATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	PROCAINAMIDE HYDROCHLORIDE	rxcui:155056	PROCAINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.09963505	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.1103102336884338	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
TTR	hgnc:12405	TTR	ChEMBL	33	modulator	4.375639269641208	TAFAMIDIS MEGLUMINE	rxcui:1727003	TAFAMIDIS MEGLUMINE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	TRELAGLIPTIN SUCCINATE	ncit:C152724	TRELAGLIPTIN SUCCINATE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	2-AMINO-ANTHRAQUINONE	chembl:CHEMBL84685	CHEMBL:CHEMBL84685	FALSE	FALSE	FALSE
HBA2	hgnc:4824	HBA2	ChEMBL	33	negative modulator	8.751278539282415	EFAPROXIRAL	ncit:C1435	EFAPROXIRAL	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.4526523382387456	AMRUBICIN HYDROCHLORIDE	ncit:C47948	AMRUBICIN HYDROCHLORIDE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.014585464	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
NAE1	hgnc:621	NAE1	ChEMBL	33	inhibitor	10.50153425	PEVONEDISTAT	ncit:C77906	PEVONEDISTAT	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.212152207	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
UBA3	hgnc:12470	UBA3	ChEMBL	33	inhibitor	21.00306849	PEVONEDISTAT	ncit:C77906	PEVONEDISTAT	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2075402025126264	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	ChEMBL	33	inhibitor	2.386712328895204	ROXADUSTAT	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	0.3241214273808302	TALAZOPARIB	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
IDO1	hgnc:6059	IDO1	ChEMBL	33	inhibitor	3.750547945	EPACADOSTAT	ncit:C92582	EPACADOSTAT	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2651902587661338	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
PLA2G5	hgnc:9038	PLA2G5	ChEMBL	33	inhibitor	8.751278539282415	VARESPLADIB METHYL	ncit:C152833	VARESPLADIB METHYL	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
BMP10	hgnc:20869	BMP10	ChEMBL	33	inhibitor	26.25383561784724	DALANTERCEPT	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
TNFSF14	hgnc:11930	TNFSF14	ChEMBL	33	inhibitor	13.12691780892362	BAMINERCEPT	ncit:C96762	BAMINERCEPT ALFA	FALSE	FALSE	FALSE
MSLN	hgnc:7371	MSLN	ChEMBL	33	inhibitor	17.50255707856483	AMATUXIMAB	ncit:C62483	AMATUXIMAB	FALSE	FALSE	FALSE
TTR	hgnc:12405	TTR	DTC	9/2/20	NULL	0.1902451856365742	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	binder	4.200613699	OPORTUZUMAB MONATOX	ncit:C61307	OPORTUZUMAB MONATOX	FALSE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	ChEMBL	33	inhibitor	1.810609352954982	TORALIZUMAB	ncit:C152696	TORALIZUMAB	FALSE	FALSE	FALSE
MSTN	hgnc:4223	MSTN	ChEMBL	33	inhibitor	2.187819634820604	LANDOGROZUMAB	ncit:C99640	LANDOGROZUMAB	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	ChEMBL	33	inhibitor	0.6482428547616604	HUMAX-IL8	chembl:CHEMBL2109617	HUMAX-IL8	FALSE	FALSE	FALSE
SELP	hgnc:10721	SELP	ChEMBL	33	inhibitor	5.250767123569449	INCLACUMAB	ncit:C174603	INCLACUMAB	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	CONICASTEROL D	chembl:CHEMBL1782605	CONICASTEROL D	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	ChEMBL	33	modulator	0.4953553890159858	IMGATUZUMAB	ncit:C78838	IMGATUZUMAB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010678802	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	1.458546423213736	BEMIPARIN SODIUM	rxcui:436195	BEMIPARIN SODIUM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.030527716	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.020351811	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
RRM2	hgnc:10452	RRM2	ChEMBL	33	inhibitor	1.154014752432846	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	DICHLOROBENZYL ALCOHOL	rxcui:22906	DICHLOROBENZYL ALCOHOL	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	DIBENZEPIN	rxcui:3332	DIBENZEPIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00172405	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.6731752722524935	NETARSUDIL DIMESYLATE	chembl:CHEMBL4594251	NETARSUDIL DIMESYLATE	TRUE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	2.625383561784724	HGS-1025	chembl:CHEMBL2109342	HGS-1025	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	inhibitor	2.625383561784724	CROTEDUMAB	ncit:C166762	CROTEDUMAB	FALSE	FALSE	FALSE
IFNA4	hgnc:5425	IFNA4	ChEMBL	33	inhibitor	1.750255707856483	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	ChEMBL	33	agonist	29.17092846427472	LEXATUMUMAB	ncit:C64621	LEXATUMUMAB	FALSE	TRUE	TRUE
SELE	hgnc:10718	SELE	ChEMBL	33	inhibitor	4.773424657790408	CDP-850	chembl:CHEMBL2109486	CDP-850	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	binder	0.760980743	ARCITUMOMAB	ncit:C1494	ARCITUMOMAB	TRUE	FALSE	FALSE
MSLN	hgnc:7371	MSLN	ChEMBL	33	binder	11.66837138570988	ANETUMAB RAVTANSINE	ncit:C98293	ANETUMAB RAVTANSINE	FALSE	FALSE	FALSE
RPS11	hgnc:10384	RPS11	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL27	hgnc:10328	RPL27	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPL10	hgnc:10298	RPL10	ChEMBL	33	inhibitor	0.1093909817410302	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
RPS18	hgnc:10401	RPS18	ChEMBL	33	inhibitor	0.1312691780892362	DORLIMOMAB ARITOX	chembl:CHEMBL2109124	DORLIMOMAB ARITOX	FALSE	FALSE	FALSE
IL1A	hgnc:5991	IL1A	ChEMBL	33	inhibitor	5.250767123569449	LUTIKIZUMAB	ncit:C166465	LUTIKIZUMAB	FALSE	FALSE	FALSE
RPL41	hgnc:10354	RPL41	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPLP1	hgnc:10372	RPLP1	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
RPL30	hgnc:10333	RPL30	ChEMBL	33	modulator	0.128067491	ATALUREN	ncit:C169791	ATALUREN	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	EMIVIRINE	ncit:C73147	EMIVIRINE	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	positive modulator	0.3125456621172291	TAK-653	drugbank:DB16304	TAK-653	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.3697723326457359	ORP-101	drugbank:DB16072	ORP-101	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	agonist	0.1367387271762877	TAVAPADON	ncit:C174853	TAVAPADON	FALSE	FALSE	FALSE
ACACA	hgnc:84	ACACA	ChEMBL	33	negative modulator	0.5707355569097228	FIRSOCOSTAT	ncit:C169983	FIRSOCOSTAT	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.4321619031744402	FF-10101	chembl:CHEMBL4650283	FF-10101	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	GLEMBATUMUMAB VEDOTIN	ncit:C78449	GLEMBATUMUMAB VEDOTIN	FALSE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	inhibitor	0.2430910705356227	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.7955707762984014	TALAMPANEL	ncit:C38139	TALAMPANEL	FALSE	FALSE	FALSE
MTNR1A	hgnc:7463	MTNR1A	ChEMBL	33	agonist	3.750547945	PIROMELATINE	ncit:C170326	PIROMELATINE	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	ChEMBL	33	inhibitor	1.750255707856483	IDASANUTLIN	ncit:C99131	IDASANUTLIN	FALSE	FALSE	FALSE
MYH7	hgnc:7577	MYH7	ChEMBL	33	activator	2.500365296937833	DANICAMTIV	ncit:C167013	DANICAMTIV	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	negative modulator	0.041672755	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.8607814956671229	GESTODENE	rxcui:25734	GESTODENE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	negative modulator	0.042174836	T-900607	drugbank:DB12068	T-900607	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	CANTUZUMAB MERTANSINE	ncit:C95782	CANTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	LORVOTUZUMAB MERTANSINE	ncit:C38714	LORVOTUZUMAB MERTANSINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.001266832	PARAPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1071585127259071	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	2',4'-DIHYDROXYCHALCONE	chembl:CHEMBL105310	2',4'-DIHYDROXYCHALCONE	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.040989595	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	CARPHENAZINE	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	ISOKAEMPFERIDE	chembl:CHEMBL165064	ISOKAEMPFERIDE	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1693795846312726	DIMERCAPROL	rxcui:3445	DIMERCAPROL	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.022789788	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.014160645	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NU-1025	chembl:CHEMBL123904	CHEMBL:CHEMBL123904	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.026240715	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	GR-55562	iuphar.ligand:113	GR-55562	FALSE	FALSE	FALSE
CHUK	hgnc:1974	CHUK	DTC	9/2/20	NULL	0.1339481409073839	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.034229251	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	METHIOTHEPIN MESYLATE	chembl:CHEMBL1256737	METHIOTHEPIN MESYLATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	NSC-111847	chembl:CHEMBL1984884	CHEMBL:CHEMBL1984884	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.033985548	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00667527	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	L-733060	chembl:CHEMBL1256740	CHEMBL:CHEMBL1256740	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.2067231151011594	CHINIOFON	ncit:C76415	CHINIOFON	FALSE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.8204323630577265	DI-TERT-BUTYLHYDROQUINONE	chembl:CHEMBL480626	CHEMBL:CHEMBL480626	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.02339914	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.036413087	IRIGENOL	iuphar.ligand:11564	IRIGENOL	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.007329379	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	4'-METHOXYFLAVONE	chembl:CHEMBL16312	4'-METHOXYFLAVONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.000723665	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	ACETOCHLOR	chembl:CHEMBL1517425	ACETOCHLOR	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	TCMDC-125602	chembl:CHEMBL580183	CHEMBL:CHEMBL580183	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.013330203	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DIGITOXIGENIN	drugbank:DB04177	DIGITOXIGENIN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.2734774543525755	NIPECOTIC ACID	drugbank:DB08849	NIPECOTIC ACID	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	3,3',4'-TRIHYDROXYFLAVONE	chembl:CHEMBL122701	CHEMBL:CHEMBL122701	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.2169738480813822	RHEIN	drugbank:DB13174	RHEIN	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.2734774543525755	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW786460X	chembl:CHEMBL185238	GW786460X	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	NCG-C00093820-01	chembl:CHEMBL544115	CHEMBL:CHEMBL544115	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.032817295	TOPOTECAN HYDROCHLORIDE	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002936671	SB-415286	iuphar.ligand:8019	SB-415286	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.014369915	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	4-HYDROXYESTRADIOL	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.011568114	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.03729238	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004264756	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2430910705356226	SJ000018300	chembl:CHEMBL590927	CHEMBL:CHEMBL590927	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	CAMBINOL	drugbank:DB15493	CAMBINOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	FLURANDRENOLIDE	rxcui:4500	FLURANDRENOLIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01798824	SULFORAPHANE	ncit:C1424	SULFORAPHANE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	NSC-632536	chembl:CHEMBL1367933	CHEMBL:CHEMBL1367933	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.03292017	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	DTC	9/2/20	NULL	0.8334550989792776	CLIOXANIDE	ncit:C65338	CLIOXANIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.008414691	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.1207072901969988	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	CEFONICID	rxcui:2183	CEFONICID	FALSE	FALSE	FALSE
ERAP1	hgnc:18173	ERAP1	DTC	9/2/20	NULL	8.751278539282415	TCMDC-124673	chembl:CHEMBL587247	CHEMBL:CHEMBL587247	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.1084869240406911	N-(P-ISOTHIOCYANATOPHENETHYL)SPIPERONE HCL	chembl:CHEMBL1257081	CHEMBL:CHEMBL1257081	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00359617	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
TSSK2	hgnc:11401	TSSK2	DTC	9/2/20	NULL	0.2019525816757481	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	MEVASTATIN	ncit:C96285	MEVASTATIN	FALSE	FALSE	FALSE
PTK6	hgnc:9617	PTK6	DTC	9/2/20	NULL	0.1491695205559502	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	CYTARABINE HYDROCHLORIDE	ncit:C71603	CYTARABINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	CLOFOCTOL	rxcui:21264	CLOFOCTOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ALLANTODAPSONE	chembl:CHEMBL227725	ALLANTODAPSONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	TCMDC-125814	chembl:CHEMBL533082	CHEMBL:CHEMBL533082	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.005737289	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.8468979231563628	SOLYPERTINE TARTRATE	ncit:C152391	SOLYPERTINE TARTRATE	FALSE	FALSE	FALSE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	0.1810609352954982	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.07458476	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	GNF-PF-5510	chembl:CHEMBL578741	CHEMBL:CHEMBL578741	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.025003653	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.043109746	3,3',4'-TRIHYDROXYFLAVONE	chembl:CHEMBL122701	CHEMBL:CHEMBL122701	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.010586224	MERCURIC CHLORIDE	rxcui:1311634	MERCURIC CHLORIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00731101	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	CORTODOXONE	ncit:C80813	CORTODOXONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	CILNIDIPINE	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-586581A	chembl:CHEMBL230597	GSK-586581A	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.6908904109959803	NAKIJIQUINONES H	chembl:CHEMBL499608	NAKIJIQUINONES H	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	0.2187819634820604	DNDI1417132	chembl:CHEMBL1492017	CHEMBL:CHEMBL1492017	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
KDM4D	hgnc:25498	KDM4D	DTC	9/2/20	NULL	4.375639269641208	PYRIDINE-2,4-DICARBOXYLIC ACID	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	STREPTOMYCIN	rxcui:10109	STREPTOMYCIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FEBANTEL	rxcui:24805	FEBANTEL	TRUE	FALSE	FALSE
SLC28A1	hgnc:11001	SLC28A1	DTC	9/2/20	NULL	5.250767123569449	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004011894	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	TERPYRIDINE	chembl:CHEMBL89445	TERPYRIDINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	6'-IODONONIVAMIDE	chembl:CHEMBL177809	CHEMBL:CHEMBL177809	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	DTC	9/2/20	NULL	0.729273212	PD-81723	chembl:CHEMBL59532	CHEMBL:CHEMBL59532	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	TCMDC-125544	chembl:CHEMBL533602	CHEMBL:CHEMBL533602	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.2243917574174978	3,4-DIHYDROXYXANTHONE	chembl:CHEMBL446323	3,4-DIHYDROXYXANTHONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	ZM-449829	chembl:CHEMBL154580	CHEMBL:CHEMBL154580	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.053445395	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	FRENTIZOLE	ncit:C167023	FRENTIZOLE	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.075010959	COUMESTROL	iuphar.ligand:12437	COUMESTROL	FALSE	FALSE	FALSE
NPY2R	hgnc:7957	NPY2R	DTC	9/2/20	NULL	2.187819634820604	DNDI1417776	chembl:CHEMBL1585652	CHEMBL:CHEMBL1585652	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.3302369260106572	ARTESUNATE	rxcui:18346	ARTESUNATE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	1.000146118775133	MACROCARPAL A	chembl:CHEMBL396609	MACROCARPAL A	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	DIHYDREXIDINE	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.048958202	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.038608582	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007330402	GNF-PF-67	chembl:CHEMBL578512	CHEMBL:CHEMBL578512	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	GLYCYRRHIZIN	rxcui:26143	GLYCYRRHIZIC ACID	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	NSC-93401	chembl:CHEMBL452954	CHEMBL:CHEMBL452954	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.090064616	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.092118721	PECTOLINARIGENIN	chembl:CHEMBL78010	PECTOLINARIGENIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	MMV006513	chembl:CHEMBL585622	CHEMBL:CHEMBL585622	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.073540156	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.056500364	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.011568114	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.076098074	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	ALFADEX	ncit:C76093	ALFADEX	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	CETRIMIDE	rxcui:288088	CETRIMIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	BOLDINE	chembl:CHEMBL388342	BOLDINE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	TYRPHOSTIN AG-835	drugbank:DB16763	TYRPHOSTIN AG 835	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001856641	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00337822	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.3621218705909965	NEOPETROFORMYNE A	chembl:CHEMBL2177350	NEOPETROFORMYNE A	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.008773212	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	DTC	9/2/20	NULL	0.5303805175322677	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1060761035064535	DNDI1417055	chembl:CHEMBL1486366	CHEMBL:CHEMBL1486366	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.05068308	LAUROGUADINE	ncit:C80857	LAUROGUADINE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1526385791735305	DNDI1417063	chembl:CHEMBL2094422	CHEMBL:CHEMBL2094422	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.05404804	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.4412409347537352	GNF-PF-4464	chembl:CHEMBL600692	CHEMBL:CHEMBL600692	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	CADMIUM ACETATE	chembl:CHEMBL1476898	CADMIUM ACETATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000628729	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	SARCOLYSIN	ncit:C61936	SARCOLYSIN	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.045461187	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.010193685	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	GALLIC ACID METHYL ESTER	chembl:CHEMBL65675	GALLIC ACID METHYL ESTER	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	IPA-3	iuphar.ligand:8940	IPA-3	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	SJ000012773	chembl:CHEMBL589715	CHEMBL:CHEMBL589715	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.03140411	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.01555322	BENSERAZIDE HYDROCHLORIDE	rxcui:235765	BENSERAZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	METHYLDOPA (RACEMIC)	chembl:CHEMBL718	METHYLDOPA (RACEMIC)	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.010020548	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.014050755	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	PENTAMIDINE ISETHIONATE	rxcui:7995	PENTAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.091159151	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006182465	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	DTC	9/2/20	NULL	4.200613699	RISEDRONIC ACID	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.007300844	HOMIDIUM BROMIDE	ncit:C65857	HOMIDIUM BROMIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	NSC-50654	chembl:CHEMBL1372046	CHEMBL:CHEMBL1372046	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001259177	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	ESTROPIPATE	rxcui:33747	ESTROPIPATE	TRUE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	DTC	9/2/20	NULL	3.500511415712966	CIMIPRONIDINE	chembl:CHEMBL485803	CIMIPRONIDINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000422546	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PIPERONAL	rxcui:33753	PIPERONAL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.020117882	LIPOIC ACID, ALPHA	chembl:CHEMBL33864	LIPOIC ACID, ALPHA	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.008722205	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	SPLITOMICIN	iuphar.ligand:8101	SPLITOMICIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.008804103	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	SANSALVAMIDE A-AMIDE	chembl:CHEMBL192264	CHEMBL:CHEMBL192264	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	JNJ-16259685	iuphar.ligand:1385	JNJ16259685	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.596678082	5-(N,N-DIMETHYL)AMILORIDE HYDROCHLORIDE	chembl:CHEMBL1256020	5-(N,N-DIMETHYL)AMILORIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001094092	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	PILOCARPINE HYDROCHLORIDE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.011585982	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.027767145	SOTRASTAURIN	ncit:C80630	SOTRASTAURIN	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.004764329	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	0.3365876361262467	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
FES	hgnc:3657	FES	DTC	9/2/20	NULL	0.1474934585272317	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	HYDRASTININE	chembl:CHEMBL1314044	HYDRASTININE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.017456008	ISOPROTERENOL HYDROCHLORIDE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	ENNIATIN B	chembl:CHEMBL469036	ENNIATIN B	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	PROPOXYCAINE	ncit:C66492	PROPOXYCAINE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.020164236	SB-220025	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	THEONELLASTEROL B	chembl:CHEMBL1782598	THEONELLASTEROL B	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	LEVONORDEFRIN	rxcui:132889	LEVONORDEFRIN	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.036463661	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.033487035	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.00984765	SJ000044511	chembl:CHEMBL592124	CHEMBL:CHEMBL592124	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.1244257612220248	DEMECLOCYCLINE	rxcui:3154	DEMECLOCYCLINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	DNDI1417809	chembl:CHEMBL1442783	CHEMBL:CHEMBL1442783	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.004068785	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	ALDRIN	chembl:CHEMBL195953	ALDRIN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.013716738	CATECHOL	chembl:CHEMBL280998	CATECHOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	3,5-DINITROCATECHOL (OR-486)	chembl:CHEMBL168276	3,5-DINITROCATECHOL (OR-486)	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00988845	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	chembl:CHEMBL1256708	APOMORPHINE HYDROCHLORIDE HEMIHYDRATE	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.005513774	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	CGP-60474	chembl:CHEMBL300389	CHEMBL:CHEMBL300389	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001907844	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.011834048	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.022691301	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005297384	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.1653584607713247	ISOPROTERENOL HYDROCHLORIDE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.034727296	TPCK	chembl:CHEMBL60718	TPCK	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1060761035064535	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	0.8751278539282416	TCMDC-125606	chembl:CHEMBL536166	CHEMBL:CHEMBL536166	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.008224886	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	FLAVONOL	chembl:CHEMBL294009	FLAVONOL	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.048618214	CLIOQUINOL	rxcui:5942	CLIOQUINOL	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	GERONTOXANTHONE H	chembl:CHEMBL514057	GERONTOXANTHONE H	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.056097939	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	R(-)-PROPYLNORAPOMORPHINE HCL	chembl:CHEMBL538542	CHEMBL:CHEMBL538542	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.015498132	GSK-269962A	drugbank:DB17030	GSK-269962A	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.009242681	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ATROPINE METHYL BROMIDE	chembl:CHEMBL2146143	ATROPINE METHYLBROMIDE	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	ZAMPANOLIDE	chembl:CHEMBL582439	ZAMPANOLIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	DIETHYLCARBAMAZINE CITRATE	rxcui:203175	DIETHYLCARBAMAZINE CITRATE	TRUE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.04464938	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.546954909	PYRIDINE-2,4-DICARBOXYLIC ACID	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	1.193356164447602	EPIGALLOCATECHIN	drugbank:DB03823	EPIGALLOCATECHIN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.044611445	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	DTC	9/2/20	NULL	0.7501095890813498	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.048083948	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER	iuphar.ligand:5092	&ALPHA;&BETA;-METHYLENEADP	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	NSC-102029	chembl:CHEMBL74913	CHEMBL:CHEMBL74913	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	CID 667285	chembl:CHEMBL267160	CHEMBL:CHEMBL267160	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	PF-03715455	drugbank:DB12138	PF-03715455	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.00770359	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	PHENMEDIPHAM	chembl:CHEMBL1079421	PHENMEDIPHAM	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.028290771	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	PYRIDINE-2,4-DICARBOXYLIC ACID	iuphar.ligand:8744	COMPOUND 6A [PMID: 18942826]	FALSE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.091796628	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	SKF-89626	chembl:CHEMBL1256191	CHEMBL:CHEMBL1256191	FALSE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	2.386712328895204	GNF-PF-4353	chembl:CHEMBL527307	CHEMBL:CHEMBL527307	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.017352172	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	METHYLENE BLUE CHLORIDE HYDRATE	chembl:CHEMBL550495	METHYLENE BLUE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	THIETHYLPERAZINE MALATE	ncit:C66598	THIETHYLPERAZINE MALATE	TRUE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.251232877	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.6035364509849942	GNF-PF-5217	chembl:CHEMBL601970	CHEMBL:CHEMBL601970	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.011474579	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
KLF5	hgnc:6349	KLF5	DTC	9/2/20	NULL	1.640864726115453	CID 838877	chembl:CHEMBL405317	CHEMBL:CHEMBL405317	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	1,3-DIACETYLVILASININ	chembl:CHEMBL463701	CHEMBL:CHEMBL463701	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	GW9662	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010687497	EPINEPHRINE BITARTRATE	rxcui:203180	EPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002322526	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.075442056	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00475613	THIOMERSAL	rxcui:10472	THIMEROSAL	TRUE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.029498692	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.7395446652914718	NAFCILLIN SODIUM	rxcui:9893	NAFCILLIN SODIUM	TRUE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.042073455	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	NSC-753575	chembl:CHEMBL2036119	CHEMBL:CHEMBL2036119	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2430910705356226	GNF-PF-4803	chembl:CHEMBL585240	CHEMBL:CHEMBL585240	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.1084869240406911	BMS-191011	chembl:CHEMBL45349	CHEMBL:CHEMBL45349	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003689409	SU-6656	drugbank:DB08039	(3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	TCMDC-124224	chembl:CHEMBL580421	CHEMBL:CHEMBL580421	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.099446347	ACRIFLAVINE CHLORIDE	chembl:CHEMBL354349	EUFLAVINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	BERBERINE CHLORIDE	ncit:C87331	BERBERINE CHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	MMV085203	chembl:CHEMBL586031	CHEMBL:CHEMBL586031	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.011176601	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	DNDI1417346	chembl:CHEMBL1490332	CHEMBL:CHEMBL1490332	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.006252402	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
PTBP1	hgnc:9583	PTBP1	DTC	9/2/20	NULL	0.2734774543525755	ELLIPTECINE	chembl:CHEMBL123	ELLIPTECINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	7,8,3'-TRIHYDROXYFLAVONE	chembl:CHEMBL225513	CHEMBL:CHEMBL225513	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.021234525	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.012430793	CAPSAZEPINE	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.014268389	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.011355465	AG-490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.026816992	SP-600125	chembl:CHEMBL1725279	SP-600125	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	DNDI1416969	chembl:CHEMBL1453126	CHEMBL:CHEMBL1453126	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.2263261691193728	NSC-158389	chembl:CHEMBL192626	CHEMBL:CHEMBL192626	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1458546423213736	THIABENDAZOLE	rxcui:10450	THIABENDAZOLE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	NSC-102742	chembl:CHEMBL1519374	CHEMBL:CHEMBL1519374	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV396595	chembl:CHEMBL2028044	CHEMBL:CHEMBL2028044	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.018206543	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.012836492	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CEFAZOLIN	rxcui:2180	CEFAZOLIN	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007946076	PHLORETIN	rxcui:1368167	PHLORETIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	ISOQUERCETIN	ncit:C117288	ISOQUERCETIN	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.019563216	OSI-632	iuphar.ligand:7881	CP-547632	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	ICILLIN	iuphar.ligand:2429	ICILIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016780975	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.073694977	ACACETIN	chembl:CHEMBL243664	ACACETIN	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.045265234	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	GNF-PF-4463	chembl:CHEMBL584520	CHEMBL:CHEMBL584520	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.008058268	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.2983390411119005	GNF-PF-4459	chembl:CHEMBL585502	CHEMBL:CHEMBL585502	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.003371279	NSC-228155	chembl:CHEMBL505670	CHEMBL:CHEMBL505670	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	L-732138	iuphar.ligand:9461	L-732,138	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.019799273	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.009031247	NSC-9037	chembl:CHEMBL1451216	CHEMBL:CHEMBL1451216	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	BROMOENOL LACTONE	iuphar.ligand:5149	BROMOENOL LACTONE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.026858144	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	NSC-69187	chembl:CHEMBL19954	CHEMBL:CHEMBL19954	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	SCH-58261	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	KEPONE	chembl:CHEMBL462576	KEPONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.00770359	LUTEOLIN	drugbank:DB15584	LUTEOLIN	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.022949157	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009922085	TCMDC-124518	chembl:CHEMBL527584	CHEMBL:CHEMBL527584	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.596678082	BUNITROLOL	ncit:C72614	BUNITROLOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	NALOXONE METHIODIDE	chembl:CHEMBL1514361	NALOXONE METHIODIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.1389091831632129	ALOE-EMODIN	chembl:CHEMBL40275	ALOE-EMODIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.056097939	PYRILAMINE	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	CID 893238	chembl:CHEMBL473735	CHEMBL:CHEMBL473735	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	2.019525817	BERKELEYTRIONE	chembl:CHEMBL252716	BERKELEYTRIONE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.7242437411819931	ISOCEPHAELINE	chembl:CHEMBL486005	ISOCEPHAELINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	HYCANTHONE	ncit:C550	HYCANTHONE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.063415062	4-TERT-BUTYLCATECHOL	chembl:CHEMBL220845	CHEMBL:CHEMBL220845	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003307362	PURPUROGALLIN	chembl:CHEMBL66953	PURPUROGALLIN	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	SIRTINOL	chembl:CHEMBL380797	SIRTINOL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	TCMDC-125784	chembl:CHEMBL581574	CHEMBL:CHEMBL581574	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.034184682	BROXURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.2381300282797936	2,5-BIS(4-METHOXYSTYRYL)PYRAZINE	chembl:CHEMBL2181039	CHEMBL:CHEMBL2181039	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	BENOXINATE	rxcui:18889	BENOXINATE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.009242681	GNF-PF-1919	iuphar.ligand:8482	DECYNIUM 22	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	ENILCONAZOLE	rxcui:1442172	ENILCONAZOLE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.005073205	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.045265234	SJ000113972	chembl:CHEMBL591137	CHEMBL:CHEMBL591137	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	MK-212	drugbank:DB12111	MK-212	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	TYRPHOSTIN AG-112	iuphar.ligand:5913	AG 112	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	WHILE OLIVETOL	chembl:CHEMBL154533	WHILE OLIVETOL	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	1.381780822	GNF-PF-4353	chembl:CHEMBL527307	CHEMBL:CHEMBL527307	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	GYKI-52466	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.009995749	TAE-684	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.027290889	ALSTERPAULLONE	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
AKR1C1	hgnc:384	AKR1C1	DTC	9/2/20	NULL	17.50255707856483	3,5-DIBROMOSALICYLIC ACID	chembl:CHEMBL447448	CHEMBL:CHEMBL447448	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.024275391	SLAZINIC ACID	chembl:CHEMBL172439	SLAZINIC ACID	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	DNDI1417132	chembl:CHEMBL1492017	CHEMBL:CHEMBL1492017	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	SJ000294102	chembl:CHEMBL607309	CHEMBL:CHEMBL607309	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1861974157294131	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.1346350544504987	QUINALIZARIN	drugbank:DB08660	QUINALIZARIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	(S)-AMPA	drugbank:DB02057	(S)-AMPA	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MIRISTALKONIUM CHLORIDE	rxcui:236394	MIRISTALKONIUM CHLORIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	STAVUDINE	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.02339914	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003147942	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.1037701012563132	GNF-PF-3037	chembl:CHEMBL600336	CHEMBL:CHEMBL600336	FALSE	FALSE	FALSE
PROS1	hgnc:9456	PROS1	FDA	10-Apr-24	NULL	0.1595977849109255	Estradiol	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
DMD	hgnc:2928	DMD	FDA	10-Apr-24	NULL	15.00219178	Golodirsen	rxcui:2267207	GOLODIRSEN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.013281873	Imipramine	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	0.082472782	Nivolumab	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	2.500365296937833	Omacetaxine	rxcui:1546446	OMACETAXINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.010848692	Pantoprazole	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.02726255	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.012213217	Thioridazine	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
RYR1	hgnc:10483	RYR1	FDA	10-Apr-24	NULL	0.1013661606866689	Sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
IL12A	hgnc:5969	IL12A	FDA	10-Apr-24	NULL	1.050153425	Ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
IL23A	hgnc:15488	IL23A	FDA	10-Apr-24	NULL	1.640864726115453	Ustekinumab	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.007378818	Venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.021258166	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.043866058	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.172722603	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.172722603	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
RICTOR	hgnc:28611	RICTOR	MyCancerGenome	20-Jun-17	inhibitor	1.154014752432846	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
MLST8	hgnc:24825	MLST8	MyCancerGenome	20-Jun-17	inhibitor	1.009762908	AZD8055	iuphar.ligand:7714	AZD8055	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	MyCancerGenome	20-Jun-17	inhibitor	0.2333674277141978	VOLASERTIB	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	antibody	0.6908904109959803	MM-111	drugbank:DB17983	MM-111	FALSE	TRUE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1584738568481725	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	MyCancerGenome	20-Jun-17	antibody	8.751278539282417	DULANERMIN	ncit:C1685	DULANERMIN	FALSE	TRUE	TRUE
TNFSF13B	hgnc:11929	TNFSF13B	MyCancerGenome	20-Jun-17	antibody	32.81729452230906	BELIMUMAB	rxcui:1092437	BELIMUMAB	TRUE	TRUE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	antibody	1.981421556063943	BIIB022	ncit:C71530	ANTI-IGF-1R RECOMBINANT MONOCLONAL ANTIBODY BIIB022	FALSE	TRUE	TRUE
NOTCH3	hgnc:7883	NOTCH3	MyCancerGenome	20-Jun-17	other/unknown	2.100306849	RO4929097	iuphar.ligand:7338	RO4929097	FALSE	FALSE	TRUE
NOTCH1	hgnc:7881	NOTCH1	MyCancerGenome	20-Jun-17	other/unknown	3.938075342677087	RO4929097	iuphar.ligand:7338	RO4929097	FALSE	FALSE	TRUE
PARP2	hgnc:272	PARP2	MyCancerGenome	20-Jun-17	other/unknown	1.250182648468916	MK4827	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
PSMB8	hgnc:9545	PSMB8	MyCancerGenome	20-Jun-17	other/unknown	0.3182283105193606	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB1	hgnc:9537	PSMB1	MyCancerGenome	20-Jun-17	other/unknown	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB7	hgnc:9544	PSMB7	MyCancerGenome	20-Jun-17	other/unknown	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC6	hgnc:9553	PSMC6	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD10P1	hgnc:16602	PSMD10P1	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641208	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD2	hgnc:9559	PSMD2	MyCancerGenome	20-Jun-17	other/unknown	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.034018575	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.091850154	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.099220845	DACTOLISIB	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2500365296937833	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
FRK	hgnc:3955	FRK	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1136529680426288	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2500365296937833	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3642372228836055	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1043371509899543	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.079557078	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PARP2	hgnc:272	PARP2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	2.187819634820604	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.024932417	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.3443125982668492	THYMIDINE	rxcui:1372538	THYMIDINE	TRUE	FALSE	FALSE
ACADM	hgnc:89	ACADM	NCI	14-Sep-17	NULL	0.07699072	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.1259176768242074	ACYCLOVIR	rxcui:281	ACYCLOVIR	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	NCI	14-Sep-17	NULL	0.7026004179620139	ENALAPRIL MALEATE	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.035976479	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.022220766	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	1.544343271638073	GALACTITOL	chembl:CHEMBL1773904	GALACTITOL	FALSE	FALSE	FALSE
ACP5	hgnc:124	ACP5	NCI	14-Sep-17	NULL	0.2019525816757481	TPA	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
ACTC1	hgnc:143	ACTC1	NCI	14-Sep-17	NULL	0.1470803115845784	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	NCI	14-Sep-17	NULL	0.8078103267029922	METOPROLOL SUCCINATE	rxcui:221124	METOPROLOL SUCCINATE	TRUE	FALSE	FALSE
ADCYAP1	hgnc:241	ADCYAP1	NCI	14-Sep-17	NULL	13.12691780892362	ANTIPARASITIC	ncit:C276	ANTIPARASITIC AGENT	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.3860858179095183	IL-13	iuphar.ligand:4980	IL-13	FALSE	FALSE	FALSE
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	1.323722804261206	GONADOTROPINS	ncit:C527	THERAPEUTIC GONADOTROPIN	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.090843722	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
APOA2	hgnc:601	APOA2	NCI	14-Sep-17	NULL	0.3088686543276147	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
ATF2	hgnc:784	ATF2	NCI	14-Sep-17	NULL	0.5147810905460245	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.047626006	ANTISERUM	ncit:C571	ANTISERUM	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.038894571	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.053854022	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.2000292237550266	C5A	iuphar.ligand:3576	C5A	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	1.280674908	BEAUVERICIN	ncit:C1011	BEAUVERICIN	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.2561349816375342	EMD 121974	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	2.333674277141977	DNCB	ncit:C439	DINITROCHLOROBENZENE	FALSE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	0.9376369863516874	ADENOVIRAL VECTOR	ncit:C1890	ADENOVIRUS VECTOR	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.015434354	ARA-C	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CCL4	hgnc:10630	CCL4	NCI	14-Sep-17	NULL	0.4023576339899961	CYCLOSPORIN A	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CD2	hgnc:1639	CD2	NCI	14-Sep-17	NULL	1.060761035064535	COBALT	rxcui:1310300	COBALT	FALSE	FALSE	FALSE
CD27	hgnc:11922	CD27	NCI	14-Sep-17	NULL	0.7501095890813501	PROTEASE INHIBITORS	ncit:C783	PROTEASE INHIBITOR	FALSE	FALSE	FALSE
CDA	hgnc:1712	CDA	NCI	14-Sep-17	NULL	3.750547945	DEOXYCYTIDINE	rxcui:2642208	DEOXYCYTIDINE	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.052455216	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.2273059360852575	INDOLE-3-CARBINOL	rxcui:2598119	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.02783338	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.1613138901250214	L-PAM	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
CEL	hgnc:1848	CEL	NCI	14-Sep-17	NULL	0.4286340509036285	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CEL	hgnc:1848	CEL	NCI	14-Sep-17	NULL	0.3061671792168775	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
COIL	hgnc:2184	COIL	NCI	14-Sep-17	NULL	1.000146118775133	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.1852122442176172	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	1.29648571	ISOFLAVONE	drugbank:DB12007	ISOFLAVONE	FALSE	FALSE	FALSE
CR2	hgnc:2336	CR2	NCI	14-Sep-17	NULL	1.050153425	5-AZA-2-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	NCI	14-Sep-17	NULL	0.1735790784651057	PROGESTIN	ncit:C776	PROGESTIN	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	1.400204566285186	FAMCICLOVIR	rxcui:68099	FAMCICLOVIR	TRUE	FALSE	FALSE
CSF1	hgnc:2432	CSF1	NCI	14-Sep-17	NULL	0.6429510763554429	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.03043923	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CTAG1B	hgnc:2491	CTAG1B	NCI	14-Sep-17	NULL	0.2625383561784725	5-AZA-2-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
CTSD	hgnc:2529	CTSD	NCI	14-Sep-17	NULL	2.282942227638891	STREPTOZOTOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	NCI	14-Sep-17	NULL	3.850562557284263	AMD3100	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	1.250182648468916	ISOFLAVONE	drugbank:DB12007	ISOFLAVONE	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.2206204673768676	NSAIDS	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.082300425	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.1392776425349987	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.086361301	GANCICLOVIR	rxcui:4678	GANCICLOVIR	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.076765601	R115777	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.038382801	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.384671584	PENICILLAMINE	rxcui:7975	PENICILLAMINE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.019097171	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
RPE65	hgnc:10294	RPE65	NCI	14-Sep-17	NULL	0.5770073762164232	H2O2	iuphar.ligand:2448	H2O2	FALSE	FALSE	FALSE
SAMD3	hgnc:21574	SAMD3	NCI	14-Sep-17	NULL	5.000730593875666	TGFBETA1	ncit:C1293	RECOMBINANT TRANSFORMING GROWTH FACTOR-BETA 1	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.2895643634321388	GLUCOCORTICOID	ncit:C521	THERAPEUTIC GLUCOCORTICOID	FALSE	FALSE	TRUE
SLC1A5	hgnc:10943	SLC1A5	NCI	14-Sep-17	NULL	13.12691780892362	GLUTAMINE	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.090530468	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
SLC22A3	hgnc:10967	SLC22A3	NCI	14-Sep-17	NULL	39.38075342677087	SARCNU	ncit:C963	SARCNU	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.2785552850699974	GP-120	ncit:C29554	GP-120 ANTIGEN	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.068458502	4-HPR	ncit:C1098	FENRETINIDE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.048958202	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.017951341	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.300043836	5-AZA-2-DEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.3333820395917111	ANTIESTROGEN	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.2258394461750301	OK-432	ncit:C745	PICIBANIL	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.025865848	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.3922986931402463	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
TNFRSF11B	hgnc:11909	TNFRSF11B	NCI	14-Sep-17	NULL	0.5114383561918295	HORMONES	ncit:C548	THERAPEUTIC HORMONE	FALSE	FALSE	FALSE
TNFRSF1B	hgnc:11917	TNFRSF1B	NCI	14-Sep-17	NULL	0.300043836	ACTINOMYCIN D	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
TPSAB1	hgnc:12019	TPSAB1	NCI	14-Sep-17	NULL	2.187819634820604	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
TPSB2	hgnc:14120	TPSB2	NCI	14-Sep-17	NULL	1.875273972703374	SALT	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.6141248097742047	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
TYMP	hgnc:3148	TYMP	NCI	14-Sep-17	NULL	0.1103102336884338	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
TYK2	hgnc:12440	TYK2	NCI	14-Sep-17	NULL	0.065145994	IFN	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.2125816649218401	TYROSINE KINASE INHIBITOR	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	NCI	14-Sep-17	NULL	0.1881995384791917	IL-12	iuphar.ligand:4977	IL-12	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.1489579325835305	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	NCI	14-Sep-17	NULL	0.093596562	CURCUMIN	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
UBE2D1	hgnc:12474	UBE2D1	NCI	14-Sep-17	NULL	6.177373086552294	DESFERRIOXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.207267123	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UCP2	hgnc:12518	UCP2	NCI	14-Sep-17	NULL	0.6250913242344582	SALINE	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.3251536612259921	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
VCAM1	hgnc:12663	VCAM1	NCI	14-Sep-17	NULL	0.201178817	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	PHENYL ISATIN	chembl:CHEMBL117447	PHENYL ISATIN	FALSE	FALSE	FALSE
UTRN	hgnc:12635	UTRN	NCI	14-Sep-17	NULL	4.375639269641208	ENZYME INHIBITOR	ncit:C471	ENZYME INHIBITOR	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.024773612	VITAMIN K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.1802322811293861	STZ	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
VIM	hgnc:12692	VIM	NCI	14-Sep-17	NULL	0.7001022831425934	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	0.036062961	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CHRNA3	hgnc:1957	CHRNA3	PharmGKB	4/5/24	NULL	0.2447910080918158	cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	PharmGKB	4/5/24	NULL	0.3070624048871023	zilucoplan	rxcui:2672489	ZILUCOPLAN	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.087512785	pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.3977853881492008	ceftriaxone	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	0.5000730593875666	cefotaxime	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	PharmGKB	4/5/24	NULL	0.044706404	vincristine	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
OTC	hgnc:8512	OTC	PharmGKB	4/5/24	NULL	1.750255707856483	sodium phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	2.871513270702042	(S)-methadone	chembl:CHEMBL350719	ESMETHADONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-5052	chembl:CHEMBL601367	CHEMBL:CHEMBL601367	FALSE	FALSE	FALSE
PICALM	hgnc:15514	PICALM	PharmGKB	4/5/24	NULL	11.66837138570989	calcium channel blockers	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	1.750255707856483	apixaban	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.037398626	doxazosin	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.2323348284765243	st. john's wort	rxcui:1310069	HYPOXIS HEMEROCALLIDEA ROOT EXTRACT	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1161674142382621	cefuroxime	rxcui:20493	CEFUROXIME AXETIL	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.009293393	simvastatin	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.06638138	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.03319069	sulfinpyrazone	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.100976291	Analgesics	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
TCF7L2	hgnc:11641	TCF7L2	PharmGKB	4/5/24	NULL	0.5385402178019948	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.1415301111474245	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.1973972602845657	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
RAC2	hgnc:9802	RAC2	PharmGKB	4/5/24	NULL	0.9376369863516874	prednisolone	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	PharmGKB	4/5/24	NULL	0.075010959	nifedipine	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	PharmGKB	4/5/24	NULL	0.092851762	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
ATP5F1E	hgnc:838	ATP5F1E	PharmGKB	4/5/24	NULL	0.06697407	methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
SLC22A11	hgnc:18120	SLC22A11	PharmGKB	4/5/24	NULL	1.29648571	zidovudine	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
NEUROD1	hgnc:7762	NEUROD1	PharmGKB	4/5/24	NULL	2.500365296937833	repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	PharmGKB	4/5/24	NULL	0.3333820395917111	antiepileptics	ncit:C264	ANTICONVULSANT AGENT	FALSE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.6863747873946994	atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.01305187	atazanavir	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.1493817104856173	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
DAOA	hgnc:21191	DAOA	PharmGKB	4/5/24	NULL	2.763561643983921	aripiprazole	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.6364566210387212	primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.086361301	busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.2206204673768676	nefazodone	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
RPL13	hgnc:10303	RPL13	PharmGKB	4/5/24	NULL	0.4054646427466756	thalidomide	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.012325744	carfilzomib	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NBEA	hgnc:7648	NBEA	PharmGKB	4/5/24	NULL	1.009762908	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.021240967	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
PPP3R1	hgnc:9317	PPP3R1	PharmGKB	4/5/24	NULL	1.207072901969988	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
PCSK9	hgnc:20001	PCSK9	PharmGKB	4/5/24	NULL	0.8078103267029924	lomitapide	rxcui:1364478	LOMITAPIDE MESYLATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.1653584607713247	isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	16.12735616524902	desflurane	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
FHIT	hgnc:3701	FHIT	PharmGKB	4/5/24	NULL	0.3365876361262468	antidepressants	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	3.750547945	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	PharmGKB	4/5/24	NULL	0.062065805	sacituzumab govitecan-hziy	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.1325951293830669	epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
PRKAB1	hgnc:9378	PRKAB1	PharmGKB	4/5/24	NULL	1.009762908	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
DHFR	hgnc:2861	DHFR	DTC	9/2/20	NULL	1.640864726115453	TCMDC-124296	chembl:CHEMBL22148	CHEMBL:CHEMBL22148	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.086861325	stavudine	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.069180068	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
OAS1	hgnc:8086	OAS1	PharmGKB	4/5/24	NULL	1.093909817410302	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
ARHGEF10	hgnc:14103	ARHGEF10	PharmGKB	4/5/24	NULL	1.458546423213736	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
STAT3	hgnc:11364	STAT3	PharmGKB	4/5/24	NULL	0.089756703	interferons	ncit:C584	RECOMBINANT INTERFERON	FALSE	FALSE	FALSE
TRIB3	hgnc:16228	TRIB3	PharmGKB	4/5/24	NULL	7.001022831425934	indapamide	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.037884323	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.099446347	trimipramine	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.1164249916534246	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
VEGFB	hgnc:12681	VEGFB	PharmGKB	4/5/24	NULL	0.6563458904461812	bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
PRKAG3	hgnc:9387	PRKAG3	PharmGKB	4/5/24	NULL	1.795134059339982	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
SLC19A3	hgnc:16266	SLC19A3	PharmGKB	4/5/24	NULL	1.346350544504987	metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.1981421556063943	margetuximab	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
TUT7	hgnc:25817	TUT7	PharmGKB	4/5/24	NULL	1.640864726115453	peginterferon alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	PharmGKB	4/5/24	NULL	0.097236428	irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	DTC	9/2/20	NULL	1.944728564284981	TALOTREXIN	ncit:C29341	TALOTREXIN	FALSE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	PharmGKB	4/5/24	NULL	0.086219493	cyclosporine	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1312691780892362	moxifloxacin	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	PharmGKB	4/5/24	NULL	15.00219178	latanoprost	rxcui:43611	LATANOPROST	TRUE	FALSE	FALSE
USP24	hgnc:12623	USP24	PharmGKB	4/5/24	NULL	4.375639269641208	rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
HNF1B	hgnc:11630	HNF1B	PharmGKB	4/5/24	NULL	2.625383561784725	platinum	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.023493365	BRADANICLINE	ncit:C169814	BRADANICLINE	FALSE	FALSE	FALSE
METTL1	hgnc:7030	METTL1	PharmGKB	4/5/24	NULL	3.621218705909965	peginterferon alfa-2a	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
CTNNB1	hgnc:2514	CTNNB1	PharmGKB	4/5/24	NULL	0.018501646	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.010216825	acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.030527716	dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.6563458904461812	moxifloxacin	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
BCL6	hgnc:1001	BCL6	PharmGKB	4/5/24	NULL	0.921187215	polatuzumab vedotin	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	PharmGKB	4/5/24	NULL	0.1458546423213736	rofecoxib	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.035358701	warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	PharmGKB	4/5/24	NULL	0.6364566210387211	exenatide	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.1166837138570989	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.006415893	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
SPATA5	hgnc:18119	AFG2A	PharmGKB	4/5/24	NULL	0.4861821410712453	paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:O94806	hgnc:9408	PRKD3	TdgClinicalTrial	Jan-14	NULL	0.1093909817410302	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.3182283105193605	BROMFENAC	rxcui:19737	BROMFENAC	TRUE	FALSE	FALSE
UNIPROT:Q05655	hgnc:9399	PRKCD	TdgClinicalTrial	Jan-14	NULL	0.4102161815288632	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
UNIPROT:P05129	hgnc:9402	PRKCG	TdgClinicalTrial	Jan-14	NULL	0.1630673019742065	BRYOSTATIN-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
UNIPROT:Q9NY47	hgnc:1400	CACNA2D2	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	BUDIODARONE	ncit:C83563	BUDIODARONE	FALSE	FALSE	FALSE
UNIPROT:P01730	hgnc:1678	CD4	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	BT-061	iuphar.ligand:9864	TREGALIZUMAB	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.068847471	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.078276194	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:P28074	hgnc:9542	PSMB5	TdgClinicalTrial	Jan-14	NULL	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
UNIPROT:Q16602	hgnc:16709	CALCRL	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	CGRP	drugbank:DB06379	CALCITONIN GENE-RELATED PEPTIDE	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1137761023525341	OXYCODONE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.032134438	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P00325	hgnc:250	ADH1B	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.035890411	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.070860555	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.064268875	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.021422958	CNS-7056	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q96GD4	hgnc:11390	AURKB	TdgClinicalTrial	Jan-14	NULL	0.5877724392055355	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
UNIPROT:O14965	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.6674703970639131	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.1013661606866689	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:O14788	hgnc:11926	TNFSF11	TdgClinicalTrial	Jan-14	NULL	43.75639269641208	DENOSUMAB	rxcui:993449	DENOSUMAB	TRUE	FALSE	TRUE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.1769126389342806	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.1682938180631233	DIMIRACETAM	ncit:C79121	DIMIRACETAM	FALSE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	DOV 21947	chembl:CHEMBL1818442	AMITIFADINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.032492371	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.053445395	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.084146909	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	0.1339481409073839	LATREPIRDINE	ncit:C78757	LATREPIRDINE	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	DOV 21947	chembl:CHEMBL1818442	AMITIFADINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q9NY46	hgnc:10590	SCN3A	TdgClinicalTrial	Jan-14	NULL	0.070010228	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q99250	hgnc:10588	SCN2A	TdgClinicalTrial	Jan-14	NULL	0.066676408	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
UNIPROT:P08246	hgnc:3309	ELANE	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	ERDOSTEINE	rxcui:24305	ERDOSTEINE	TRUE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.072927321	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TdgClinicalTrial	Jan-14	NULL	3.454452054979901	EPLERENONE	rxcui:298869	EPLERENONE	TRUE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	1.921012362281506	OBLIMERSEN	ncit:C1870	OBLIMERSEN	FALSE	FALSE	TRUE
UNIPROT:P08648	hgnc:6141	ITGA5	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	GLPG0187	ncit:C96223	INTEGRIN RECEPTOR ANTAGONIST GLPG0187	FALSE	FALSE	FALSE
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.071341945	GLPG0634	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	GLPG0187	ncit:C96223	INTEGRIN RECEPTOR ANTAGONIST GLPG0187	FALSE	FALSE	FALSE
UNIPROT:P51168	hgnc:10600	SCNN1B	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	4.861821410712453	HUMAX-CD20	rxcui:712566	OFATUMUMAB	TRUE	TRUE	TRUE
UNIPROT:P51170	hgnc:10602	SCNN1G	TdgClinicalTrial	Jan-14	NULL	1.372749574789398	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
UNIPROT:P51787	hgnc:6294	KCNQ1	TdgClinicalTrial	Jan-14	NULL	0.059667808	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
UNIPROT:P01583	hgnc:5991	IL1A	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	RILONACEPT	rxcui:763450	RILONACEPT	TRUE	FALSE	FALSE
UNIPROT:P31785	hgnc:6010	IL2RG	TdgClinicalTrial	Jan-14	NULL	0.5250767123569451	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
UNIPROT:P14784	hgnc:6009	IL2RB	TdgClinicalTrial	Jan-14	NULL	0.4039051633514962	IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.2557191780959147	ITI-007	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.1651184630053286	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q16288	hgnc:8033	NTRK3	TdgClinicalTrial	Jan-14	NULL	0.2035181055647073	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
UNIPROT:O75899	hgnc:4507	GABBR2	TdgClinicalTrial	Jan-14	NULL	3.889457128569962	LESOGABERAN	ncit:C166751	LESOGABERAN	FALSE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	LGD-1550	drugbank:DB05785	LGD-1550	FALSE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.8643238063488805	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.081030357	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:Q8WWZ7	hgnc:35	ABCA5	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	LIM-0705	chembl:CHEMBL4297397	QUERCETIN-3'-O-PHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.07182992	CINOLAZEPAM	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1383601350084176	DROPERIDOL	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.6105543166941221	DIPIVEFRIN	rxcui:23410	DIPIVEFRIN	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.1103102336884338	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.028300937	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.055563673	FLURAZEPAM	rxcui:4501	FLURAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	PHENTERMINE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.049457775	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	2.734774543525755	PRALATREXATE	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.046518424	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.090922374	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.087512785	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.096050618	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.022606632	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.091583148	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.01858569	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.100976291	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.1166837138570989	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1221108633388244	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.661861402	RIZATRIPTAN	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.1022876712383659	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.089501712	QUAZEPAM	rxcui:35185	QUAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	0.4039051633514962	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	SECOBARBITAL	rxcui:9624	SECOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.1141471113819445	TALBUTAL	rxcui:89810	TALBUTAL	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.4922594178346359	SUPROFEN	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
UNIPROT:P30411	hgnc:1030	BDKRB2	TEND	1-Aug-11	NULL	2.187819634820604	ICATIBANT	rxcui:1148138	ICATIBANT	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TEND	1-Aug-11	NULL	0.7501095890813498	ACETAZOLAMIDE	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:P00325	hgnc:250	ADH1B	TEND	1-Aug-11	NULL	13.12691780892362	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.693795846312725	ALCAFTADINE	rxcui:1000082	ALCAFTADINE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.079197091	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:O00555	hgnc:1388	CACNA1A	TEND	1-Aug-11	NULL	0.5834185692854944	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.05387244	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.051478109	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.055155117	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.009922085	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
UNIPROT:P32238	hgnc:1570	CCKAR	TEND	1-Aug-11	NULL	2.625383561784724	CERULETIDE	ncit:C65309	CERULETIDE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.057197899	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.13086024	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	BENZODODECINIUM CHLORIDE	rxcui:1311592	BENZODODECINIUM CHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P02461	hgnc:2201	COL3A1	TEND	1-Aug-11	NULL	2.812910959055062	COLLAGENASE	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1193356164447602	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.042073455	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIP4K2A	hgnc:8997	PIP4K2A	DTC	9/2/20	NULL	3.500511415712966	TDR77225	chembl:CHEMBL1353528	CHEMBL:CHEMBL1353528	FALSE	FALSE	FALSE
UNIPROT:P02452	hgnc:2197	COL1A1	TEND	1-Aug-11	NULL	0.8036888454443035	COLLAGENASE	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P08123	hgnc:2198	COL1A2	TEND	1-Aug-11	NULL	0.6250913242344583	COLLAGENASE	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.4817217544559128	ANILERIDINE	rxcui:17933	ANILERIDINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.056826484	DNDI1417195	chembl:CHEMBL1303948	CHEMBL:CHEMBL1303948	FALSE	FALSE	FALSE
UNIPROT:Q08345	hgnc:2730	DDR1	TEND	1-Aug-11	NULL	0.7001022831425933	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P07333	hgnc:2433	CSF1R	TEND	1-Aug-11	NULL	0.089103927	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.031842129	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
UNIPROT:P24530	hgnc:3180	EDNRB	TEND	1-Aug-11	NULL	3.750547945	BOSENTAN	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.3182283105193605	BROMFENAC	rxcui:19737	BROMFENAC	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.1715936968486748	BUPROPION	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.305277158	PICROTOXIN	rxcui:2539172	PICROTOXIN	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TEND	1-Aug-11	NULL	0.087512785	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14324	hgnc:3631	FDPS	TEND	1-Aug-11	NULL	4.200613699	RISEDRONATE	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.2128689374420047	SOLIFENACIN	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TEND	1-Aug-11	NULL	0.8423690572571311	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.040452751	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:P00747	hgnc:9071	PLG	TEND	1-Aug-11	NULL	2.500365296937833	TENECTEPLASE	rxcui:259280	TENECTEPLASE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.1864177677006905	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
UNIPROT:P07101	hgnc:11782	TH	TEND	1-Aug-11	NULL	1.500219178	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TEND	1-Aug-11	NULL	2.386712328895204	TOLVAPTAN	rxcui:358257	TOLVAPTAN	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.052229116	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.028290771	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TEND	1-Aug-11	NULL	0.5321723436050118	TRANYLCYPROMINE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	GNF-PF-3286	chembl:CHEMBL581880	CHEMBL:CHEMBL581880	FALSE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TEND	1-Aug-11	NULL	1.944728564284981	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TEND	1-Aug-11	NULL	0.6731752722524935	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P22748	hgnc:1375	CA4	TEND	1-Aug-11	NULL	1.458546423213736	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	CT-1578	chembl:CHEMBL2035185	CT-1578	FALSE	FALSE	FALSE
UNIPROT:Q8N0U8	hgnc:21492	VKORC1L1	TEND	1-Aug-11	NULL	3.182283105193606	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005363398	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.3351553483129436	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
UNIPROT:P47901	hgnc:896	AVPR1B	TEND	1-Aug-11	NULL	0.5770073762164232	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	1.458546423213736	Apaxifylline	ncit:C81046	APAXIFYLLINE	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	ONO-4059	ncit:C102876	TIRABRUTINIB	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	0.546954909	Xatral	chembl:CHEMBL1723	ALFUZOSIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.5556367326528517	G1T38	ncit:C138165	LEROCICLIB	FALSE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	0.3559842117674203	M7824	ncit:C124229	BINTRAFUSP ALFA	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005366413	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	0.9723642821424906	G1T38	ncit:C138165	LEROCICLIB	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	1.193356164447602	Guadecitabine	ncit:C95209	GUADECITABINE	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	1.500219178	SKI-O-703	ncit:C170949	CEVIDOPLENIB DIMESYLATE	FALSE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	1.944728564284981	APVO414	chembl:CHEMBL4594540	APVO-414	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.3017682254924971	LYCOBETAINE	chembl:CHEMBL253553	LYCOBETAINE	FALSE	FALSE	FALSE
INACTIVE TYROSINE-PROTEIN KINASE 7	hgnc:9618	PTK7	TTD	2020.06.01	NULL	52.50767123569449	PF-06647020	ncit:C123828	COFETUZUMAB PELIDOTIN	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR-II	hgnc:5466	IGF2	TTD	2020.06.01	NULL	2.917092846427472	Dusigitumab	ncit:C82683	DUSIGITUMAB	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.4468737977505915	CYTISINE	rxcui:1723152	CYTISINE	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	2.500365296937833	NSC-119913	chembl:CHEMBL471004	CHEMBL:CHEMBL471004	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	PRN2246	ncit:C173549	TOLEBRUTINIB	FALSE	FALSE	FALSE
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	8.751278539282415	ABX-1431	drugbank:DB16036	ABX-1431	FALSE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	3.000438356	Imetelstat	ncit:C49084	IMETELSTAT	FALSE	FALSE	TRUE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	1.346350544504987	PF-04995274	drugbank:DB12675	PF-04995274	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR	hgnc:2438	CSF3	TTD	2020.06.01	NULL	8.751278539282415	LA-EP2006	ncit:C104005	PEGFILGRASTIM BIOSIMILAR LA-EP2006	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	4.200613699	GS-5745	ncit:C105803	ANDECALIXIMAB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	TCMDC-124571	chembl:CHEMBL533542	CHEMBL:CHEMBL533542	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
CHOLINE KINASE	hgnc:1937	CHKA	TTD	2020.06.01	NULL	52.50767123569449	TCD-717	chembl:CHEMBL3545084	TCD-717	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.2318219480604613	Contusugene ladenovec	ncit:C2471	CONTUSUGENE LADENOVEC	FALSE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.2	hgnc:6256	KCNJ10	TTD	2020.06.01	NULL	1.071585127259071	Glipizide	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.7026004179620139	Enalapril	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.044573575	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	PARA-SIRTINOL	chembl:CHEMBL372375	CHEMBL:CHEMBL372375	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-14	hgnc:7160	MMP14	TTD	2020.06.01	NULL	0.4412409347537353	Epigallocatechin gallate	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
LEUKOTRIENE B4 RECEPTOR 1	hgnc:6713	LTB4R	TTD	2020.06.01	NULL	3.281729452230906	CP-195543	drugbank:DB13053	CP-195543	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.040515178	Dalfampridine	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	DNDI1417777	chembl:CHEMBL1412002	CHEMBL:CHEMBL1412002	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	2.100306849	CTCE-0214	drugbank:DB05934	CTCE-0214	FALSE	FALSE	FALSE
GROWTH HORMONE-RELEASING HORMONE RECEPTOR	hgnc:4266	GHRHR	TTD	2020.06.01	NULL	19.69037671338543	Tesamorelin	rxcui:1044584	TESAMORELIN	TRUE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.060772768	CH-5132799	drugbank:DB13051	CH-5132799	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.100976291	CH-5132799	drugbank:DB13051	CH-5132799	FALSE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.2083637747448194	CH-5132799	drugbank:DB13051	CH-5132799	FALSE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	1.193356164447602	iOWH032	chembl:CHEMBL4297392	IOWH-032	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	1.193356164447602	Palifosfamide	ncit:C66990	PALIFOSFAMIDE	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	1.640864726115453	NSC-119913	chembl:CHEMBL471004	CHEMBL:CHEMBL471004	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	1.165474011072658	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
IRON	hgnc:4650	GTF2E1	TTD	2020.06.01	NULL	2.100306849	Deferiprone	rxcui:11645	DEFERIPRONE	TRUE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	0.6250913242344582	bis-triazole derivative 10	iuphar.ligand:6537	BIS-TRIAZOLE DERIVATIVE 10	FALSE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	3.281729452230906	AMG 416	rxcui:1876119	ETELCALCETIDE	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.6482428547616604	RPC-1063	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
STS	hgnc:11425	STS	DTC	9/2/20	NULL	7.001022831425932	17ALPHA-3'-BROMOBENZYL ESTRADIOL	chembl:CHEMBL1627429	CHEMBL:CHEMBL1627429	FALSE	FALSE	FALSE
5-HT 1F RECEPTOR	hgnc:5292	HTR1F	TTD	2020.06.01	NULL	14.32027397337122	Lasmiditan	rxcui:2256930	LASMIDITAN	TRUE	FALSE	FALSE
UROKINASE PLASMINOGEN ACTIVATOR SURFACE RECEPTOR	hgnc:9053	PLAUR	TTD	2020.06.01	NULL	0.3860858179095184	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.3889457128569962	GSK-356278	drugbank:DB12542	GSK-356278	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-18	hgnc:3674	FGF18	TTD	2020.06.01	NULL	52.50767123569449	AS-902330	chembl:CHEMBL2108302	SPRIFERMIN	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	4.633029815	MGN-1703	ncit:C94207	LEFITOLIMOD	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013192882	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	2.128689374420047	Tozadenant	ncit:C152704	TOZADENANT	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.8751278539282416	Etirinotecan pegol	ncit:C74069	ETIRINOTECAN PEGOL	FALSE	FALSE	TRUE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.3226277802500429	Certolizumab pegol	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.1630673019742065	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A	hgnc:7943	NPR1	TTD	2020.06.01	NULL	4.039051633514961	Ularitide	ncit:C96702	ULARITIDE	FALSE	FALSE	FALSE
STROMAL CELL-DERIVED FACTOR 1	hgnc:10672	CXCL12	TTD	2020.06.01	NULL	13.12691780892362	NOX-A12	ncit:C99379	OLAPTESED PEGOL	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	1.250182648468916	PF-05089771	drugbank:DB14856	PF-05089771	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.3088686543276147	FS118	ncit:C150734	ANTI-LAG-3/PD-L1 BISPECIFIC ANTIBODY FS118	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION GENE 3 PROTEIN	hgnc:6476	LAG3	TTD	2020.06.01	NULL	3.281729452230906	FS118	ncit:C150734	ANTI-LAG-3/PD-L1 BISPECIFIC ANTIBODY FS118	FALSE	FALSE	FALSE
PRKG1	hgnc:9414	PRKG1	DTC	9/2/20	NULL	0.040452751	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.3659071166250487	Cemiplimab	rxcui:2058825	CEMIPLIMAB-RWLC	TRUE	FALSE	TRUE
LIVER CARBOXYLESTERASE	hgnc:1863	CES1	TTD	2020.06.01	NULL	2.282942227638891	Eldacimibe	ncit:C81530	ELDACIMIBE	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.5585922471882393	Trimethaphan	rxcui:10828	TRIMETHAPHAN	TRUE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	4.039051633514961	CTS-21166	drugbank:DB06073	CTS-21166	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:42	ncit:C74391	IPSAPIRONE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.075442056	IUPHAR.LIGAND:28	iuphar.ligand:28	SB 216641	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:65	iuphar.ligand:65	(R)-FLUROCARAZOLOL	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.047734247	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.2108741816694558	IUPHAR.LIGAND:6	iuphar.ligand:6	7-METHOXY-1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.070291394	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:6	iuphar.ligand:6	7-METHOXY-1-NAPHTHYLPIPERAZINE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.1054370908347279	IUPHAR.LIGAND:129	iuphar.ligand:129	S33084	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.009442128	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.041672755	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.032899543	IUPHAR.LIGAND:134	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.052090944	IUPHAR.LIGAND:23	iuphar.ligand:23	RU 24969	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.089298761	IUPHAR.LIGAND:51	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.009329721	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.039068208	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.028413242	IUPHAR.LIGAND:97	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.032899543	IUPHAR.LIGAND:99	ncit:C66558	SPIPERONE	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.013140058	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.074478966	IUPHAR.LIGAND:5	iuphar.ligand:5	5-HYDROXYTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:3242	iuphar.ligand:3242	[18F]ALTANSERIN	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:190	iuphar.ligand:190	SB 215505	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.5527123287967841	IUPHAR.LIGAND:217	iuphar.ligand:217	(-)-NORFENFLURAMINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.092118721	IUPHAR.LIGAND:28	iuphar.ligand:28	SB 216641	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:193	iuphar.ligand:193	SB 242084	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00170159	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:3223	iuphar.ligand:3223	FR260010	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.024130364	IUPHAR.LIGAND:103	rxcui:40003	ZOTEPINE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.1023541349623674	IUPHAR.LIGAND:21	iuphar.ligand:21	LY344864	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.035430277	IUPHAR.LIGAND:209	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
NCBIGENE:1263	hgnc:2154	PLK3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5280	iuphar.ligand:5280	TOFA	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.2125816649218401	IUPHAR.LIGAND:8204	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:8204	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	MMV006937	chembl:CHEMBL580381	CHEMBL:CHEMBL580381	FALSE	FALSE	FALSE
NCBIGENE:3186	hgnc:9911	RBMXP1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:2820	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:10437	iuphar.ligand:10437	COMPOUND E22 [PMID: 31298542]	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.004621341	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.014786728	IUPHAR.LIGAND:96	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.1238388472539964	IUPHAR.LIGAND:487	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.1100789753368857	IUPHAR.LIGAND:7109	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:481	iuphar.ligand:481	NS-49	FALSE	FALSE	FALSE
NCBIGENE:1614	hgnc:13557	ACE2	GuideToPharmacology	2024.1	activator	5.250767123569449	IUPHAR.LIGAND:7867	iuphar.ligand:7867	XNT [PMID: 18391097]	FALSE	FALSE	FALSE
NCBIGENE:1933	hgnc:3208	EEF1B2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8943	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.028444026	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:606	iuphar.ligand:606	APELIN-36	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:7801	iuphar.ligand:7801	COMPOUND 1 [PMID: 25241924]	FALSE	FALSE	FALSE
NCBIGENE:1933	hgnc:3208	EEF1B2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8958	iuphar.ligand:8958	LIFIRAFENIB	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:8525	iuphar.ligand:8525	ELABELA/TODDLER-21	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:10305	iuphar.ligand:10305	PI-THERAPHOTOXIN-HM3A	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.086219493	IUPHAR.LIGAND:375	iuphar.ligand:375	CGS 21680	FALSE	FALSE	FALSE
PTBP1	hgnc:9583	PTBP1	DTC	9/2/20	NULL	0.9723642821424908	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
NCBIGENE:64	hgnc:137	ACTBP4	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:8652	iuphar.ligand:8652	CCL21B	FALSE	FALSE	FALSE
NCBIGENE:1877	hgnc:3121	E4F1	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:10067	iuphar.ligand:10067	AFM13	FALSE	FALSE	FALSE
NCBIGENE:1990	hgnc:3308	CELA1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12974	iuphar.ligand:12974	MW01	FALSE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:3422	iuphar.ligand:3422	CHEMERIN C-TERMINAL PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:8163	iuphar.ligand:8163	COMPOUND 33 [PMID: 19364658]	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:5954	iuphar.ligand:5954	CHK2 INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:82	hgnc:154	ACTG1P9	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:10573	iuphar.ligand:10573	OSTN (81-102)	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MIRIPIRIUM CHLORIDE	ncit:C166671	MIRIPIRIUM CHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:8044	iuphar.ligand:8044	CCT241533	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:8007	iuphar.ligand:8007	BX-912	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9187	iuphar.ligand:9187	CCT245737	FALSE	FALSE	FALSE
NCBIGENE:914	hgnc:1639	CD2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:4494	iuphar.ligand:4494	HEMICHOLINIUM-3	FALSE	FALSE	FALSE
NCBIGENE:1204	hgnc:2081	CLNS1AP1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4494	iuphar.ligand:4494	HEMICHOLINIUM-3	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	DNDI1417485	chembl:CHEMBL1346468	CHEMBL:CHEMBL1346468	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.1651184630053286	IUPHAR.LIGAND:10420	iuphar.ligand:10420	CHMFL-KIT-64	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:8250	iuphar.ligand:8250	SOTULETINIB	FALSE	FALSE	FALSE
NCBIGENE:1989	hgnc:1974	CHUK	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9398	iuphar.ligand:9398	PHA-408	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.038608582	IUPHAR.LIGAND:1909	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NCBIGENE:2734	hgnc:4316	GLG1	GuideToPharmacology	2024.1	activator	5.250767123569449	IUPHAR.LIGAND:12197	iuphar.ligand:12197	TTK21	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:3533	iuphar.ligand:3533	SSR125543A	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.210030685	HARMINE HYDROCHLORIDE	chembl:CHEMBL1593867	HARMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:922	iuphar.ligand:922	UROTENSIN 1 (FISH)	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.1103102336884338	IUPHAR.LIGAND:7482	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:928	iuphar.ligand:928	UROCORTIN 3	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:924	iuphar.ligand:924	[125I]ASTRESSIN	FALSE	FALSE	FALSE
NCBIGENE:1840	hgnc:3060	DTX1	GuideToPharmacology	2024.1	inhibitor	0.6731752722524936	IUPHAR.LIGAND:7476	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	AM-251	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:8497	iuphar.ligand:8497	NAVARIXIN	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:828	iuphar.ligand:828	CXCL3	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.048618214	IUPHAR.LIGAND:8473	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:5949	iuphar.ligand:5949	CDK2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:8114	drugbank:DB07149	(7S)-2-(2-AMINOPYRIMIDIN-4-YL)-7-(2-FLUOROETHYL)-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.077789143	IUPHAR.LIGAND:9923	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:7379	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:8710	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:8804	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:9893	iuphar.ligand:9893	COMPOUND 9 [PMID: 20718420]	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:6318	rxcui:1100699	LINAGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11582	ncit:C96202	ANAGLIPTIN	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:6319	rxcui:1368001	ALOGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:642	hgnc:1059	BLMH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7996	iuphar.ligand:7996	6-FLUOROMEVALONATE PYROPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2007	ncbigene:2007	ELNL1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8208	iuphar.ligand:8208	COMPOUND 5N [PMID: 20483621]	FALSE	FALSE	FALSE
NCBIGENE:2006	hgnc:3327	ELN	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11114	iuphar.ligand:11114	DCLK1-IN-1	FALSE	FALSE	FALSE
NCBIGENE:2637	hgnc:4186	GBX2	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:7069	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:3231	hgnc:5132	HOXD1	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:3306	iuphar.ligand:3306	OLEANOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:10603	iuphar.ligand:10603	TG11-77	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:10742	iuphar.ligand:10742	SKF-82958	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1400204566285186	IUPHAR.LIGAND:7671	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:946	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:9566	iuphar.ligand:9566	(R)-ZINC-3573	FALSE	FALSE	FALSE
NCBIGENE:2039	hgnc:3382	DMTN	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9398	iuphar.ligand:9398	PHA-408	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:7706	iuphar.ligand:7706	AZD3463	FALSE	FALSE	TRUE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:9382	iuphar.ligand:9382	NVP-TAE 226	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:1917	iuphar.ligand:1917	CICAPROST	FALSE	FALSE	FALSE
NCBIGENE:659	hgnc:1078	BMPR2	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:12435	iuphar.ligand:12435	L-PHE-PHE-PHE	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:12440	iuphar.ligand:12440	DATISCETIN	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:12468	iuphar.ligand:12468	GROSHEIMIN	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:8309	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:12171	iuphar.ligand:12171	COMPOUND 8L [PMID: 36053746]	FALSE	FALSE	FALSE
NCBIGENE:664	hgnc:1084	BNIP3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:12428	iuphar.ligand:12428	PARTHENOLIDE	FALSE	FALSE	FALSE
NCBIGENE:665	hgnc:1085	BNIP3L	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:4811	rxcui:8700	PROCAINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:9246	iuphar.ligand:9246	UPADACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:10000	iuphar.ligand:10000	GUSACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:8315	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:11060	iuphar.ligand:11060	PF-956980	FALSE	FALSE	FALSE
NCBIGENE:2379	hgnc:3891	FRA2G	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11347	rxcui:2467540	BEROTRALSTAT	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.02075402	IUPHAR.LIGAND:9174	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.012383885	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10677	iuphar.ligand:10677	COMPOUND 25 [PMID: 32023060]	FALSE	FALSE	FALSE
NCBIGENE:515	hgnc:840	ATP5PB	GuideToPharmacology	2024.1	activator	0.2430910705356227	IUPHAR.LIGAND:2401	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	blocker	4.773424657790408	IUPHAR.LIGAND:2310	iuphar.ligand:2310	SLOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:429	hgnc:738	ASCL1	GuideToPharmacology	2024.1	blocker	13.12691780892362	IUPHAR.LIGAND:12780	iuphar.ligand:12780	MK-8153	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	0.4167275494896388	IUPHAR.LIGAND:2322	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.8751278539282418	IUPHAR.LIGAND:2491	ncit:C1214	RESINIFERATOXIN	FALSE	FALSE	FALSE
NCBIGENE:896	hgnc:1585	CCND3	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9347	iuphar.ligand:9347	KYT-0353	FALSE	FALSE	FALSE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7507	drugbank:DB08291	N-(3-AMINOPROPYL)-2-NITROBENZENAMINE	FALSE	FALSE	FALSE
NCBIGENE:2983	hgnc:4687	GUCY1B1	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:11507	iuphar.ligand:11507	JNJ-67856633	FALSE	FALSE	FALSE
NCBIGENE:2682	hgnc:11114	KDM5C	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7027	iuphar.ligand:7027	GSK-J1	FALSE	FALSE	FALSE
NCBIGENE:2685	ncbigene:2685	GGTL2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8979	iuphar.ligand:8979	GSK-J4	FALSE	FALSE	FALSE
NCBIGENE:2685	ncbigene:2685	GGTL2	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:7027	iuphar.ligand:7027	GSK-J1	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1323	iuphar.ligand:1323	MT-II	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:1324	rxcui:2262250	AFAMELANOTIDE	TRUE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1333	iuphar.ligand:1333	&GAMMA;-MSH	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1017590527823536	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:5701	iuphar.ligand:5701	PI-103	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:7699	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.034888818	IUPHAR.LIGAND:5889	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:1573	hgnc:2634	CYP2J2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:12714	iuphar.ligand:12714	M8891	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:10131	iuphar.ligand:10131	UNC4203	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.5357925636295356	IUPHAR.LIGAND:6452	ncit:C171677	DIPRAGLURANT	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6449	iuphar.ligand:6449	COMPOUND 10 [PMID: 15482908]	FALSE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:11200	ncit:C126687	RINETERKIB	FALSE	FALSE	FALSE
NCBIGENE:1062	hgnc:1856	CENPE	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:4689	iuphar.ligand:4689	BONGKREK ACID	FALSE	FALSE	FALSE
NCBIGENE:1501	hgnc:2516	CTNND2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12122	iuphar.ligand:12122	COMPOUND 4E [PMID: 35546685]	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12122	iuphar.ligand:12122	COMPOUND 4E [PMID: 35546685]	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:7959	ncit:C143046	RALIMETINIB	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:9328	iuphar.ligand:9328	TAK-715	FALSE	FALSE	FALSE
NCBIGENE:1494	hgnc:6877	MAPK3	GuideToPharmacology	2024.1	inhibitor	0.7925686224255775	IUPHAR.LIGAND:9229	ncit:C170364	RAVOXERTINIB	FALSE	FALSE	FALSE
NCBIGENE:2078	hgnc:3446	ERG	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:8208	iuphar.ligand:8208	COMPOUND 5N [PMID: 20483621]	FALSE	FALSE	FALSE
NCBIGENE:2070	hgnc:3522	EYA4	GuideToPharmacology	2024.1	inhibitor	0.9723642821424908	IUPHAR.LIGAND:8106	iuphar.ligand:8106	URMC-099	FALSE	FALSE	FALSE
NCBIGENE:2076	ncbigene:2076	ERCM1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8218	iuphar.ligand:8218	COMPOUND 1 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:2089	ncbigene:2089	ERVT1	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:5710	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:12670	iuphar.ligand:12670	[18F]FMBP	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11815	iuphar.ligand:11815	SA-57	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:11733	iuphar.ligand:11733	COMPOUND 4F [PMID: 34328319]	FALSE	FALSE	FALSE
NCBIGENE:990	hgnc:1744	CDC6	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10405	iuphar.ligand:10405	BAY-8002	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1449	iuphar.ligand:1449	ME67	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.100976291	IUPHAR.LIGAND:344	iuphar.ligand:344	N-CHLOROMETHYL-BRUCINE	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1358	iuphar.ligand:1358	4P-PDOT	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:3366	iuphar.ligand:3366	DH97	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10271	iuphar.ligand:10271	RAG8	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:6658	iuphar.ligand:6658	GB88	FALSE	FALSE	FALSE
NCBIGENE:2878	hgnc:4555	GPX3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8685	iuphar.ligand:8685	CL-AMIDINE	FALSE	FALSE	FALSE
NCBIGENE:987	hgnc:1742	LRBA	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:4623	iuphar.ligand:4623	[14C]HISTIDINE	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:7795	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.028413242	IUPHAR.LIGAND:7933	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
NCBIGENE:2148	ncbigene:2148	F2L	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9201	iuphar.ligand:9201	PHENYLARSINE OXIDE	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:9907	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.064347636	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:8382	iuphar.ligand:8382	VS-5584	FALSE	FALSE	FALSE
NCBIGENE:2149	hgnc:3537	F2R	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:12181	iuphar.ligand:12181	COMPOUND 22 [WO2019141694A1]	FALSE	FALSE	FALSE
NCBIGENE:2148	ncbigene:2148	F2L	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:6060	drugbank:DB08059	WORTMANNIN	FALSE	FALSE	FALSE
NCBIGENE:1306	hgnc:2192	COL15A1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:5154	iuphar.ligand:5154	BRL50481	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:8115	iuphar.ligand:8115	COMPOUND 2 [PMID: 22560567]	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9373	iuphar.ligand:9373	CX-5011	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.2678962818147678	IUPHAR.LIGAND:9368	iuphar.ligand:9368	CX-6258	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:10195	iuphar.ligand:10195	COMPOUND 28 [PMID: 30624936]	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:6064	iuphar.ligand:6064	TRIAZINE COMPOUND PC1	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1866	iuphar.ligand:1866	PROKINETICIN-1	FALSE	FALSE	FALSE
NCBIGENE:1432	hgnc:6876	MAPK14	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:9796	iuphar.ligand:9796	(S)-23 [PMID: 27933945]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.013126918	IUPHAR.LIGAND:5657	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.087512785	IUPHAR.LIGAND:8013	drugbank:DB08052	PP-121	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.1500219178162699	IUPHAR.LIGAND:8183	iuphar.ligand:8183	PD166285	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:9403	iuphar.ligand:9403	RO3280	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:11743	drugbank:DB08577	3-[(3-(2-CARBOXYETHYL)-4-METHYLPYRROL-2-YL)METHYLENE]-2-INDOLINONE	FALSE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	0.3750547945406749	IUPHAR.LIGAND:8275	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12116	iuphar.ligand:12116	MRTX1719	FALSE	FALSE	FALSE
NCBIGENE:1259	hgnc:2148	CNGA1	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:8955	iuphar.ligand:8955	MS023	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:11732	iuphar.ligand:11732	BAY-8400	FALSE	FALSE	FALSE
NCBIGENE:1493	hgnc:2505	CTLA4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:8184	iuphar.ligand:8184	COMPOUND 32 [PMID: 20471253]	FALSE	FALSE	FALSE
NCBIGENE:1489	hgnc:2499	CTF1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8048	iuphar.ligand:8048	CRT 0066101	FALSE	FALSE	FALSE
NCBIGENE:1489	hgnc:2499	CTF1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9370	iuphar.ligand:9370	BPKDI	FALSE	FALSE	FALSE
NCBIGENE:2167	hgnc:3559	FABP4	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:8183	iuphar.ligand:8183	PD166285	FALSE	FALSE	FALSE
NCBIGENE:3224	hgnc:5129	HOXC8	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12480	iuphar.ligand:12480	JMS-053	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:8726	iuphar.ligand:8726	(4Z)-1-(3-FLUOROPHENYL)-4-(2-OXO-1H-INDOL-3-YLIDENE)PYRAZOLIDINE-3,5-DIONE	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	0.2169738480813822	IUPHAR.LIGAND:10155	iuphar.ligand:10155	RIPK1 INHIBITOR 22B	FALSE	FALSE	FALSE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11559	iuphar.ligand:11559	COMPOUND II [PMID: 29351497]	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:10089	iuphar.ligand:10089	PN10	FALSE	FALSE	FALSE
NCBIGENE:2413	hgnc:3924	FRA7F	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12196	iuphar.ligand:12196	SITOKIREN	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.062509132	IUPHAR.LIGAND:2645	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:2645	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:612	hgnc:10479	RXRG	GuideToPharmacology	2024.1	agonist	1.591141552596802	IUPHAR.LIGAND:10186	iuphar.ligand:10186	COMPOUND 28 [HEITEL ET AL., 2019]	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2640	iuphar.ligand:2640	AGN193109	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:10437	iuphar.ligand:10437	COMPOUND E22 [PMID: 31298542]	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.1630673019742065	IUPHAR.LIGAND:10033	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.032989113	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.025561544	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.2059124362184097	Hu5F9-G4	ncit:C117730	MAGROLIMAB	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.2019525816757481	Alvocidib	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	0.048282916	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.235474617310458	OH2	ncit:C172106	ONCOLYTIC TYPE 2 HERPES SIMPLEX VIRUS EXPRESSING GRANULOCYTE MACROPHAGE COLONY-STIMULATING FACTOR OH2	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.326134604	Pralsetinib	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.053445395	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	1.842374429322613	LY3039478	ncit:C171871	CRENIGACESTAT	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.4089382494991783	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	1.831662950082366	Debio 1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.025929714	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	BMF-500	ncit:C201247	FLT3 INHIBITOR BMF-500	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2160809515872201	PD98059	iuphar.ligand:5241	PD98059	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	OTS167	ncit:C111569	MELK INHIBITOR OTS167	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.012836492	Dovitinib	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.4605936073306534	Rigosertib Sodium	ncit:C71355	RIGOSERTIB SODIUM	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.082906849	Buparlisib	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.6908904109959803	MRTX-1133	ncit:C200319	KRAS G12D INHIBITOR MRTX1133	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.012838061	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.011670965	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.299554767	AGI-5198	iuphar.ligand:9240	AGI-5198	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.007780643	Panobinostat	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	2.187819634820604	TQB3455	ncit:C176768	IDH2 MUTANT INHIBITOR TQB3455	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.087512785	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.064190307	LY3410738	iuphar.ligand:12340	LY3410738	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.2302968036653267	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.1782942996118658	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.015219615	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.047049885	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1715936968486748	Pictilisib	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.048618214	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	Borussertib	chembl:CHEMBL4795065	BORUSSERTIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2025758921130189	Serabelisib	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.023151531	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	Prexasertib	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.018699313	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.2592971419046642	Ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	3.621218705909965	VCN-01	drugbank:DB18193	VCN-01	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.1508841127462485	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	4.699760697022038	Selpercatinib	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.072424374	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.6961244292611014	Repotrectinib	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	KU-60019	iuphar.ligand:8041	KU-60019	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.005654194	Cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.04636439	AZD7762	iuphar.ligand:7713	AZD7762	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	MK-8242	ncit:C116867	HDM2 INHIBITOR MK-8242	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.028977744	Pimasertib	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.00551957	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	PC14586	ncit:C175961	P53 Y220C MUTANT REACTIVATOR PC14586	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.016558711	Capivasertib	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	SP600125	iuphar.ligand:5273	SP600125	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.002033526	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	MOMETASONE FUROATE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.022108493	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.015193192	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CSNK1G3	hgnc:2456	CSNK1G3	DTC	9/2/20	NULL	0.9546849315580819	GS 6201	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.015263858	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	CGP-54626	iuphar.ligand:1070	CGP 54626A	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	CID 752709	chembl:CHEMBL429335	CHEMBL:CHEMBL429335	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	DTC	9/2/20	NULL	0.5738543304447485	ALISOL A-23 ACETATE	chembl:CHEMBL2059711	CHEMBL:CHEMBL2059711	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.007717177	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.2243917574174978	BRECANAVIR	ncit:C76908	BRECANAVIR	FALSE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	DTC	9/2/20	NULL	4.375639269641208	TENOVIN-6	chembl:CHEMBL1945130	CHEMBL:CHEMBL1945130	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	NSC-74859	chembl:CHEMBL477936	CHEMBL:CHEMBL477936	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	chembl:CHEMBL1322879	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.046840028	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.071928317	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CAMK2A	hgnc:1460	CAMK2A	DTC	9/2/20	NULL	0.077330885	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PRSS2	hgnc:9483	PRSS2	DTC	9/2/20	NULL	5.834185692854944	CYANOPEPTOLIN SS	chembl:CHEMBL1076839	CYANOPEPTOLIN SS	FALSE	FALSE	FALSE
OAT	hgnc:8091	OAT	DTC	9/2/20	NULL	105.0153424713889	GABACULINE	drugbank:DB02054	GABACULINE	FALSE	FALSE	FALSE
PRSS1	hgnc:9475	PRSS1	DTC	9/2/20	NULL	2.917092846427472	CYANOPEPTOLIN SS	chembl:CHEMBL1076839	CYANOPEPTOLIN SS	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.025929714	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011810092	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1131630845596864	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.023867123	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.2038341274677581	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	PROROXAN	ncit:C84119	PROROXAN	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.3889457128569962	GNF-PF-2895	chembl:CHEMBL524603	CHEMBL:CHEMBL524603	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	GW3965	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	DROMETRIZOLE	rxcui:1426903	DROMETRIZOLE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	DNDI1416975	chembl:CHEMBL1415851	CHEMBL:CHEMBL1415851	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.014222013	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	CID 2056784	chembl:CHEMBL261123	CHEMBL:CHEMBL261123	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.029833904	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	DNDI1417221	chembl:CHEMBL1459280	CHEMBL:CHEMBL1459280	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.058341857	FENOLDOPAM MESYLATE	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	AG1295	iuphar.ligand:5914	AG 1295	FALSE	FALSE	TRUE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.280789686	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	RIMCAZOLE	ncit:C152218	RIMCAZOLE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.034773292	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DANTHRON	rxcui:22293	DANTHRON	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.068907705	RAFOXANIDE	ncit:C152146	RAFOXANIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.212581665	GNF-PF-2853	chembl:CHEMBL576362	CHEMBL:CHEMBL576362	FALSE	FALSE	FALSE
PRKACB	hgnc:9381	PRKACB	DTC	9/2/20	NULL	1.810609352954982	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001670623	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	CARDAMOMIN	chembl:CHEMBL378104	CARDAMOMIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	IOBENGUANE	ncit:C87757	IOBENGUANE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	TCMDC-124571	chembl:CHEMBL533542	CHEMBL:CHEMBL533542	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.02702402	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	N-PHENETHYLCINNAMAMIDE	chembl:CHEMBL1305393	CHEMBL:CHEMBL1305393	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.3302369260106572	DNDI1417560	chembl:CHEMBL1373255	CHEMBL:CHEMBL1373255	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.010685322	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	1.750255707856483	STX-0119	chembl:CHEMBL1687979	CHEMBL:CHEMBL1687979	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-4590	chembl:CHEMBL529361	CHEMBL:CHEMBL529361	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	GNF-PF-3418	chembl:CHEMBL582099	CHEMBL:CHEMBL582099	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	AZINPHOS-ETHYL	ncit:C163587	AZINPHOS-ETHYL	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.027347745	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.071341945	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
AXIN1	hgnc:903	AXIN1	DTC	9/2/20	NULL	52.50767123569449	(+/-)-HYDNOCARPIN	chembl:CHEMBL91638	CHEMBL:CHEMBL91638	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.2885036881082115	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
FCGR1A	hgnc:3613	FCGR1A	DTC	9/2/20	NULL	1.000146118775133	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	NONOXYNOL 9	rxcui:53750	NONOXYNOL-9	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.022099188	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.031612084	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	MEDRONIC ACID	rxcui:1314368	MEDRONIC ACID	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	SJ000111093	chembl:CHEMBL585045	CHEMBL:CHEMBL585045	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	DNDI1417597	chembl:CHEMBL1330352	CHEMBL:CHEMBL1330352	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CITICOLINE SODIUM	rxcui:1099914	CITICOLINE SODIUM	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	NSC-123414	chembl:CHEMBL16751	CHEMBL:CHEMBL16751	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.034727296	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.300043836	L-755507	iuphar.ligand:3931	L 755507	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CANRENOATE POTASSIUM	rxcui:1981	CANRENOATE POTASSIUM	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	AZAMETHIPHOS	chembl:CHEMBL1867031	AZAMETHIPHOS	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.006002249	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.020737627	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	8-[3-(TRIFLUOROMETHYL)PHENOXYMETHYL]CAFFEINE	chembl:CHEMBL2088303	CHEMBL:CHEMBL2088303	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	GNF-PF-2383	chembl:CHEMBL578915	CHEMBL:CHEMBL578915	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.004589831	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003531589	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	DTC	9/2/20	NULL	3.889457128569962	4-PHENOXYPHENOL	chembl:CHEMBL224318	CHEMBL:CHEMBL224318	FALSE	FALSE	FALSE
DYRK2	hgnc:3093	DYRK2	DTC	9/2/20	NULL	5.250767124	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.2333674277141977	AZINPHOS-ETHYL	ncit:C163587	AZINPHOS-ETHYL	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	5-CHLORO-[1,10]PHENANTHROLINE	chembl:CHEMBL317115	CHEMBL:CHEMBL317115	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004216468	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1458546423213736	FLAVONE	rxcui:1536070	FLAVONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	NSC-56452	chembl:CHEMBL1358137	CHEMBL:CHEMBL1358137	FALSE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	DTC	9/2/20	NULL	3.750547945	BERKELEYAMIDE B	chembl:CHEMBL468640	BERKELEYAMIDE B	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	1R,9S-HYDRASTINE	chembl:CHEMBL475536	1R,9S-HYDRASTINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005308631	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.005117707	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	CETYLPYRIDINIUM	rxcui:2286	CETYLPYRIDINIUM	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.079920352	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.009320613	Aripiprazole Lauroxil	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.059030547	Arformoterol	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	4.200613699	SPERMINE BIS-2-NAPG	chembl:CHEMBL2347631	CHEMBL:CHEMBL2347631	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	FDA	10-Apr-24	NULL	0.5303805175322677	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.6241137025199848	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.326134604	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	2.341819737097098	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.2213645498975316	Eliglustat	rxcui:1547220	ELIGLUSTAT	TRUE	FALSE	FALSE
PROS1	hgnc:9456	PROS1	FDA	10-Apr-24	NULL	0.1271372184883644	Progesterone	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.0545251	Goserelin	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.005864158	Omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1211715490054488	Quinine Sulfate	rxcui:9071	QUININE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.00804962	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
PROS1	hgnc:9456	PROS1	FDA	10-Apr-24	NULL	0.6819178082557728	Warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.011049594	Warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	FDA	10-Apr-24	NULL	0.022078281	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	MyCancerGenome	20-Jun-17	inhibitor	0.3697723326457359	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	MyCancerGenome	20-Jun-17	inhibitor	2.407466349146467	AP26113	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.1852122442176172	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	MyCancerGenome	20-Jun-17	inhibitor	0.9723642821424906	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.052090944	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.1682938180631233	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.041540879	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.2051080907644316	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.041540879	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.015385511	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PKN1	hgnc:9405	PKN1	MyCancerGenome	20-Jun-17	inhibitor	0.3323270331373069	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PRKCG	hgnc:9402	PRKCG	MyCancerGenome	20-Jun-17	inhibitor	0.028898003	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenome	20-Jun-17	inhibitor	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.2465148884304905	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
APH1A	hgnc:29509	APH1A	MyCancerGenome	20-Jun-17	other/unknown	0.375054795	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	MyCancerGenome	20-Jun-17	other/unknown	0.760980743	RETASPIMYCIN	ncit:C80378	RETASPIMYCIN	FALSE	FALSE	TRUE
NOTCH3	hgnc:7883	NOTCH3	MyCancerGenome	20-Jun-17	other/unknown	2.100306849	REGN421	ncit:C82367	ENOTICUMAB	FALSE	FALSE	TRUE
NOTCH2	hgnc:7882	NOTCH2	MyCancerGenome	20-Jun-17	other/unknown	0.5357925636295356	PF-03084014	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
PSMA4	hgnc:9533	PSMA4	MyCancerGenome	20-Jun-17	other/unknown	0.3488881809680698	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PARP2	hgnc:272	PARP2	MyCancerGenome	20-Jun-17	other/unknown	0.3977853881492008	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PSMA7	hgnc:9536	PSMA7	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD7	hgnc:9565	PSMD7	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD12	hgnc:9557	PSMD12	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMC1	hgnc:9547	PSMC1	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD6	hgnc:9564	PSMD6	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD11	hgnc:9556	PSMD11	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB8	hgnc:9545	PSMB8	MyCancerGenome	20-Jun-17	other/unknown	0.2220197515251353	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSME3	hgnc:9570	PSME3	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD10P3	hgnc:30152	PSMD10P3	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
EDNRA	hgnc:3179	EDNRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	4.565884455277782	ZD4054	ncit:C48430	ZIBOTENTAN	FALSE	FALSE	TRUE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1767935058440892	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	2.341819737097098	GSK2118436	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1591141552596803	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2917092846427472	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.040390516	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.150021918	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1434635826111871	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.062331044	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
ABCC6	hgnc:57	ABCC6	NCI	14-Sep-17	NULL	0.1458546423213736	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	0.046725403	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.018887652	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	0.045421861	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ACTC1	hgnc:143	ACTC1	NCI	14-Sep-17	NULL	0.05814803	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
ADIPOQ	hgnc:13633	ADIPOQ	NCI	14-Sep-17	NULL	1.009762908	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
ADM	hgnc:259	ADM	NCI	14-Sep-17	NULL	0.2476776945079929	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	0.4861821410712453	ANTI-ANGIOGENIC AGENTS	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	0.3088686543276147	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
ATIC	hgnc:794	ATIC	NCI	14-Sep-17	NULL	0.8751278539282416	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.037843367	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.048282916	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
ATP7B	hgnc:870	ATP7B	NCI	14-Sep-17	NULL	0.4375639269641209	PLATINUM	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1272913242077442	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	0.1640864726115453	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.051859428	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.087512785	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.031115657	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.038808331	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.4268916360625568	HYPOXANTHINE	ncit:C29105	HYPOXANTHINE	FALSE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.3889457128569963	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	3.500511415712966	TUMOR NECROSIS FACTOR-BETA	ncit:C622	RECOMBINANT TUMOR NECROSIS FACTOR-BETA	FALSE	FALSE	FALSE
CCL11	hgnc:10610	CCL11	NCI	14-Sep-17	NULL	1.944728564284981	MOMETASONE FUROATE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
CCL11	hgnc:10610	CCL11	NCI	14-Sep-17	NULL	0.729273212	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.1136529680426287	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
CCL5	hgnc:10632	CCL5	NCI	14-Sep-17	NULL	2.763561643983921	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
CCNA2	hgnc:1578	CCNA2	NCI	14-Sep-17	NULL	0.546954909	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
CCNA2	hgnc:1578	CCNA2	NCI	14-Sep-17	NULL	0.6563458904461813	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
CD55	hgnc:2665	CD55	NCI	14-Sep-17	NULL	7.001022831425932	INTERLEUKIN-8	rxcui:1426866	INTERLEUKIN-8	FALSE	FALSE	FALSE
CD59	hgnc:1689	CD59	NCI	14-Sep-17	NULL	26.25383561784724	MBL	ncit:C1151	MANNOSE-BINDING LECTIN	FALSE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.6035364509849942	BISPECIFIC ANTIBODY	ncit:C1454	BISPECIFIC ANTIBODY	FALSE	FALSE	FALSE
CDH17	hgnc:1756	CDH17	NCI	14-Sep-17	NULL	0.2035181055647073	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	0.305277158	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	0.1436598392221464	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.2258394461750301	2-CDA	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
CDKN2D	hgnc:1790	CDKN2D	NCI	14-Sep-17	NULL	0.9376369863516874	DEPSIPEPTIDE	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.064111931	ALL-TRANS RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.2160809515872201	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	1.944728564284981	SODIUM MOLYBDATE	ncit:C1228	SODIUM MOLYBDATE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.077789143	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.3182283105193606	ATG	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.212581665	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.3671865121377238	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.4751825451194073	D4T	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.049192122	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.066409365	MEXILETINE	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.3292017005372696	BCNU	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
ERCC1	hgnc:3433	ERCC1	NCI	14-Sep-17	NULL	0.3319450480417468	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.062808219	NITROGEN MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.043180651	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
EREG	hgnc:3443	EREG	NCI	14-Sep-17	NULL	0.921187215	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.2287915957982331	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.058051599	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.7095631248066824	PYRAZOLE	drugbank:DB02757	PYRAZOLE	FALSE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.4118248724368196	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	1.346350544504987	PC4	ncit:C2651	SILICON PHTHALOCYANINE 4	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.097236428	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.4375639269641208	PEITC	ncit:C2233	PHENETHYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
HAS3	hgnc:4820	HAS3	NCI	14-Sep-17	NULL	1.250182648468916	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
HIST3H2A	hgnc:20507	H2AC25	NCI	14-Sep-17	NULL	2.333674277141978	VM-26	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	2.625383561784724	CORTISONE	rxcui:2878	CORTISONE	TRUE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.9723642821424906	SHO-SAIKO-TO	ncit:C2690	SHO-SAIKO-TO	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	NCI	14-Sep-17	NULL	0.042602573	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	NCI	14-Sep-17	NULL	0.084598826	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
HMOX1	hgnc:5013	HMOX1	NCI	14-Sep-17	NULL	0.6863747873946994	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	NCI	14-Sep-17	NULL	0.729273212	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
HP	hgnc:5141	HP	NCI	14-Sep-17	NULL	1.363835616511545	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1526385791735305	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1436598392221464	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.577007376	ANTINEOPLASTIC	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	NCI	14-Sep-17	NULL	0.043902735	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	NCI	14-Sep-17	NULL	0.053145416	ONDANSETRON	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	3.182283105193605	CASPASE INHIBITOR	ncit:C38461	CASPASE INHIBITOR	FALSE	FALSE	FALSE
IBSP	hgnc:5341	IBSP	NCI	14-Sep-17	NULL	0.8751278539282416	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.08334551	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.041214813	ALL-TRANS RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.175610941	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.096167896	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.1293292394967845	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
IGFBP4	hgnc:5473	IGFBP4	NCI	14-Sep-17	NULL	9.546849315580818	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1029562181092049	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.028184472	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.028810794	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	1.29648571	PROTECTIVE AGENT	ncit:C26170	PROTECTIVE AGENT	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.1105424657593568	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.096167896	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.2083637747448194	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.024814589	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.015019357	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.212152207	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.1495945049449985	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.2187819634820604	DMSO	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.051731696	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	ORNITHINE DECARBOXYLASE INHIBITOR	ncit:C2088	ORNITHINE DECARBOXYLASE INHIBITOR	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.033338204	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	MACROPHAGE COLONY STIMULATING FACTOR	ncit:C1290	RECOMBINANT MACROPHAGE COLONY-STIMULATING FACTOR	FALSE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.5147810905460245	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1363835616511545	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
NCF2	hgnc:7661	NCF2	NCI	14-Sep-17	NULL	2.282942227638891	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.039975387	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.1268301237577161	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1479089330582944	ANALGESICS	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.036977233	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.077846807	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	NCI	14-Sep-17	NULL	0.04715552	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	NCI	14-Sep-17	NULL	0.033401826	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.1417211099478933	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.076208521	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	1.438566335224506	CEP-2563 DIHYDROCHLORIDE	ncit:C2411	CEP-2563 DIHYDROCHLORIDE	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.3365876361262467	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.072725306	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	NCI	14-Sep-17	NULL	0.015088411	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PER1	hgnc:8845	PER1	NCI	14-Sep-17	NULL	2.715914029432474	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.015385511	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.030386384	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.013505059	PKC412	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.069454592	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.023151531	PKC412	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.6250913242344582	PHOSPHODIESTERASE INHIBITOR	ncit:C744	PHOSPHODIESTERASE INHIBITOR	FALSE	FALSE	FALSE
PLTP	hgnc:9093	PLTP	NCI	14-Sep-17	NULL	0.7001022831425933	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.2430910705356226	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	CLOMIPHENE	rxcui:2596	CLOMIPHENE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.050294704	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
PRTN3	hgnc:9495	PRTN3	NCI	14-Sep-17	NULL	1.640864726115453	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
PRLR	hgnc:9446	PRLR	NCI	14-Sep-17	NULL	0.921187215	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	NCI	14-Sep-17	NULL	0.2430910705356226	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	NCI	14-Sep-17	NULL	0.2027323213733378	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	NCI	14-Sep-17	NULL	0.2885036881082116	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.085796848	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	NCI	14-Sep-17	NULL	0.4167275494896388	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.384671584	GALLIUM NITRATE	rxcui:25544	GALLIUM NITRATE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.1583941817064691	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.1511209794852536	ALL-TRANS-RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PTPN1	hgnc:9642	PTPN1	NCI	14-Sep-17	NULL	0.079256862	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
SAG	hgnc:10521	SAG	NCI	14-Sep-17	NULL	0.6250913242344582	FK 506	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
SDS	hgnc:10691	SDS	NCI	14-Sep-17	NULL	1.221108633388244	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
SLC28A1	hgnc:11001	SLC28A1	NCI	14-Sep-17	NULL	1.105424657593568	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.172722603	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	1.842374429322613	DEFIBROTIDE	rxcui:1311089	DEFIBROTIDE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.3763990769583835	AMINOGLYCOSIDES	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.037081689	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1186614039224734	2-CDA	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
TGFBR3	hgnc:11774	TGFBR3	NCI	14-Sep-17	NULL	1.193356164447602	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.1417211099478934	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	NCI	14-Sep-17	NULL	0.5073204950308647	SAQUINAVIR	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.047049885	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.046089683	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.013589562	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	NCI	14-Sep-17	NULL	0.023652104	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.014488872	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	0.210030685	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
TPSAB1	hgnc:12019	TPSAB1	NCI	14-Sep-17	NULL	3.281729452230906	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.096967075	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.038971552	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
VAMP2	hgnc:12643	VAMP2	NCI	14-Sep-17	NULL	0.760980743	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.007962947	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
VAMP2	hgnc:12643	VAMP2	NCI	14-Sep-17	NULL	1.651184630053286	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
VAV1	hgnc:12657	VAV1	NCI	14-Sep-17	NULL	0.760980743	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.4039051633514962	ELMIRON	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.07767407	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.059030547	arformoterol	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.05454398	abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.049349315	everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.021149706	palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006525935	dronedarone	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.009838424	dronedarone	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.046303061	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CAT	hgnc:1516	CAT	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	1.432027397337122	etoricoxib	rxcui:307296	ETORICOXIB	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.010560674	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1161674142382621	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.029041854	nicardipine	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.020257589	lumiracoxib	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.058083707	minocycline	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.075010959	metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.055740628	daclatasvir	rxcui:1606218	DACLATASVIR	FALSE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.5000730593875666	metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.3977853881492006	lumiracoxib	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	PharmGKB	4/5/24	NULL	0.016856395	ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
AIFM2	hgnc:21411	AIFM2	PharmGKB	4/5/24	NULL	11.66837138570989	Vitamin K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
MIR1264	hgnc:35246	MIR1264	PharmGKB	4/5/24	NULL	0.3918482928036902	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	1.013661606866689	cyanocobalamin	rxcui:11248	VITAMIN B12	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.4118248724368196	risedronate	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.3500511415712967	isosorbide mononitrate	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
MKI67	hgnc:7107	MKI67	PharmGKB	4/5/24	NULL	1.381780822	abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.1682938180631233	Ergot alkaloids	rxcui:4023	ERGOT ALKALOIDS	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.1512704997187101	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
ZNF423	hgnc:16762	ZNF423	PharmGKB	4/5/24	NULL	1.050153425	raloxifene	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	PharmGKB	4/5/24	NULL	0.1988926940746004	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
CXCR2	hgnc:6027	CXCR2	PharmGKB	4/5/24	NULL	0.071148606	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	0.192335792	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	0.1973972602845657	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	PharmGKB	4/5/24	NULL	1.842374429322613	fluticasone/salmeterol	wikidata:Q581334	FLUTICASONE/SALMETEROL	FALSE	FALSE	FALSE
RIMS1	hgnc:17282	RIMS1	PharmGKB	4/5/24	NULL	2.917092846427472	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.105015342	raloxifene	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.3684748858645228	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
KCNH7	hgnc:18863	KCNH7	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
EYA4	hgnc:3522	EYA4	PharmGKB	4/5/24	NULL	2.500365296937833	certolizumab pegol	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.042174836	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002643159	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.1875273972703374	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
TEC	hgnc:11719	TEC	DTC	9/2/20	NULL	0.1049104320393496	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.052824619	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.104458232	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	NCI	14-Sep-17	NULL	0.2651902587661338	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.001566224	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CERS6	hgnc:23826	CERS6	PharmGKB	4/5/24	NULL	3.750547945406749	certolizumab pegol	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	TALC	12-May-16	inhibitor	0.060772768	NVP-BGT226	ncit:C74073	PI3K INHIBITOR BGT226	FALSE	FALSE	TRUE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.096167896	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.045898314	IUPHAR.LIGAND:384	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:952	iuphar.ligand:3298	[3H]PD128907	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.2134458180312784	IUPHAR.LIGAND:1913	iuphar.ligand:1913	MB-28767	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1465330360065893	Nintedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	CGI	2/1/22	NULL	0.3365876361262467	U0126	iuphar.ligand:5282	U0126	FALSE	FALSE	TRUE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.061992528	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
BCHE	hgnc:983	BCHE	PharmGKB	4/5/24	NULL	0.093763699	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
MMP7	hgnc:7174	MMP7	ChEMBL	33	inhibitor	0.6522692078968261	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1275696580070323	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.080042182	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.036237178	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:795	iuphar.ligand:795	[3H]BANYU (I)	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.019577804	darunavir	rxcui:460132	DARUNAVIR	TRUE	FALSE	FALSE
NCBIGENE:253	ncbigene:253	ALS3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:1158	iuphar.ligand:1158	FSH DEGLYCOSYLATED &ALPHA;/&BETA;	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.9460841664089098	AB928	ncit:C159564	ETRUMADENANT	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.006193403	midazolam	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:416	hgnc:721	ARSF	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:5467	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1861974157294131	GNF-PF-860	chembl:CHEMBL593254	CHEMBL:CHEMBL593254	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	NSC-45382	chembl:CHEMBL1214274	CHEMBL:CHEMBL1214274	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.088945801	Sulpiride	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:3252	iuphar.ligand:3252	[11C]WAY100635	FALSE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:8358	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
NCBIGENE:2729	hgnc:4311	GCLC	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11690	iuphar.ligand:11690	GSK852	FALSE	FALSE	FALSE
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:4270	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01036472	PIOGLITAZONE HYDROCHLORIDE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PSMB4	hgnc:9541	PSMB4	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.000562132	TCMDC-125488	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	1.009762908	2,4-DINITROPHENOL	drugbank:DB04528	2,4-DINITROPHENOL	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.05196207	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1584738568481725	Fruquintinib	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.3453256329104173	INFIGRATINIB	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
RPS27A	hgnc:10417	RPS27A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.4487835148349957	CALCITONIN	rxcui:1311287	CALCITONIN	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	1.458546423213736	Fingolimod	rxcui:1012892	FINGOLIMOD	TRUE	TRUE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:6310	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.058997383	IUPHAR.LIGAND:962	iuphar.ligand:962	[3H]NEMONAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.096167896	IUPHAR.LIGAND:7007	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:744	hgnc:1180	MPPED2	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:2459	iuphar.ligand:2459	DECAVANADATE	FALSE	FALSE	FALSE
OR10P1	hgnc:15378	OR10P1	PharmGKB	4/5/24	NULL	4.039051633514962	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SKF-83959	iuphar.ligand:8443	SKF-83959	FALSE	FALSE	FALSE
NDUFA10	hgnc:7684	NDUFA10	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10641	iuphar.ligand:10641	SLM6071469	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.1400204566285186	ALDICARB	ncit:C163578	ALDICARB	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	DNDI1417072	chembl:CHEMBL1310701	CHEMBL:CHEMBL1310701	FALSE	FALSE	FALSE
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	15.00219178	MEDI-578	chembl:CHEMBL2109527	MEDI-578	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.007962947	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:402	iuphar.ligand:402	MRS928	FALSE	FALSE	FALSE
GNAQ	hgnc:4390	GNAQ	DoCM	10-Apr-24	NULL	4.773424657790409	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1616	iuphar.ligand:1616	DIHYDROMORPHINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004894451	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:8443	iuphar.ligand:8443	SKF-83959	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	SJ000032151	chembl:CHEMBL592600	CHEMBL:CHEMBL592600	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	PHYSCION	chembl:CHEMBL42624	PHYSCION	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.2117244807890907	IZENCITINIB	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.066011799	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.1187956362798518	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
PSMC3	hgnc:9549	PSMC3	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.009788902	codeine	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.082950507	DNDI1417331	chembl:CHEMBL1092508	CHEMBL:CHEMBL1092508	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.7955707762984014	IL-8	ncit:C1289	RECOMBINANT INTERLEUKIN-8	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.546954909	PROTON PUMP INHIBITOR	ncit:C29723	PROTON PUMP INHIBITOR	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.1101693521639275	vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
B-CELL-SPECIFIC GLYCOPROTEIN B29	hgnc:1699	CD79B	TTD	2020.06.01	NULL	1.381780822	RG7596	rxcui:2174090	POLATUZUMAB VEDOTIN	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.012695278	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.018062494	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	activator	2.625383561784724	IUPHAR.LIGAND:6277	iuphar.ligand:6277	ACETALDEHYDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.019577804	nateglinide	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.4375639269641209	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.091583148	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.008899605	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.3804903712731485	olmesartan	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
EPIREGULIN	hgnc:3443	EREG	TTD	2020.06.01	NULL	4.375639269641208	LY3016859	chembl:CHEMBL4594573	FEPIXNEBART	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.021357605	dapsone	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	binder	1.944728564284981	HUJ591 177LU	chembl:CHEMBL2109678	HUJ591 177LU	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011746683	imipramine	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1131630845596864	LIPOSOMAL DOXORUBICIN	wikidata:Q29004943	CAELYX	FALSE	FALSE	TRUE
PI3KCB	hgnc:8976	PIK3CB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.066676408	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.1207072901969988	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.042619863	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	PharmGKB	4/5/24	NULL	0.0191914	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	PharmGKB	4/5/24	NULL	0.086361301	tucatinib	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.086432381	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.002669701	temazepam	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.2917092846427472	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	1.657092009619794	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	1.093909817410302	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.068727318	PD-325901	iuphar.ligand:7935	MIRDAMETINIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	2.341819737097098	dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	0.1223955040459079	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	DTC	9/2/20	NULL	0.083081758	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.073540156	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	0.5834185692854945	RG7304	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.138178082	IUPHAR.LIGAND:345	ncit:C152880	VINBURNINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	PHENAMIL	iuphar.ligand:4281	PHENAMIL	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	1.842374429322613	sulfamethoxazole / trimethoprim	wikidata:Q48566821	SULFAMETHOXAZOLE / TRIMETHOPRIM	FALSE	FALSE	FALSE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1458546423213736	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.1356787370431382	CARTEOLOL HYDROCHLORIDE	rxcui:142132	CARTEOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	GNF-PF-2671	chembl:CHEMBL578878	CHEMBL:CHEMBL578878	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.011372682	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	3,4,5-TRIHYDROXY-BENZOIC ACID PHENETHYL ESTER	chembl:CHEMBL151146	CHEMBL:CHEMBL151146	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.072125922	ANTIDEPRESSANTS	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
UNIPROT:P25103	hgnc:11526	TACR1	TdgClinicalTrial	Jan-14	NULL	1.419126249613364	VOFOPITANT	ncit:C72949	VOFOPITANT	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.061340737	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
IL5	hgnc:6016	IL5	ChEMBL	33	inhibitor	5.834185692854944	MEPOLIZUMAB	rxcui:1720597	MEPOLIZUMAB	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.2243917574174978	BISANTRENE	ncit:C1019	BISANTRENE	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.8793150685403386	dapsone	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.062509132	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2892984641085096	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.2344092465879218	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.061340737	trastuzumab deruxtecan	rxcui:2267574	FAM-TRASTUZUMAB DERUXTECAN-NXKI	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.272767123	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.029235897	METHYLTESTOSTERONE	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	0.018699313	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.012120884	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7811	iuphar.ligand:7811	COMPOUND 3 [PMID: 25408830]	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:7010	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDEIV-23C1	chembl:CHEMBL1094358	CHEMBL:CHEMBL1094358	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.063110182	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
NCBIGENE:667	hgnc:1090	DST	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:12433	iuphar.ligand:12433	DENATONIUM	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:11291	iuphar.ligand:11291	PSILOCIN	FALSE	FALSE	FALSE
UNIPROT:P08183	hgnc:40	ABCB1	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	ZOSUQUIDAR	ncit:C76198	ZOSUQUIDAR	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	inhibitor	0.027347745	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	OXOGLAUCINE	iuphar.ligand:12559	OXOGLAUCINE	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.5645986154375752	LENERCEPT	ncit:C166662	LENERCEPT	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.000995368	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.8899605294185507	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
CCDC77	hgnc:28203	CCDC77	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	15.31473744374422	Vismodegib	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.3697723326457359	LY-2456302	ncit:C170144	ATICAPRANT	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2017	iuphar.ligand:2017	NC 4-28B	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2051080907644316	arteether	ncit:C73002	ARTEMOTIL	TRUE	FALSE	FALSE
SMAD4	hgnc:6770	SMAD4	CIViC	10-Apr-24	NULL	5.250767123569449	LYSINE	rxcui:6536	LYSINE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.2778183663264259	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	1.280674908	SYL-1001	chembl:CHEMBL3707356	SYL-1001	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.08334551	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.6035364509849942	TCMDC-123749	chembl:CHEMBL524376	CHEMBL:CHEMBL524376	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.4102161815288632	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000872713	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
P2Y PURINOCEPTOR 2	hgnc:8541	P2RY2	TTD	2020.06.01	NULL	5.250767123569449	INS-37217	chembl:CHEMBL1767407	DENUFOSOL TETRASODIUM	FALSE	FALSE	FALSE
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	0.2442217266776488	Altiratinib	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
UNIPROT:Q99460	hgnc:9554	PSMD1	TdgClinicalTrial	Jan-14	NULL	0.5385402178019948	MLN-9708	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	1.009762908	SULFAMIDE	chembl:CHEMBL355001	SULFAMIDE	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.3070624048871023	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.375054795	INSULIN DEGLUDEC	rxcui:1670007	INSULIN DEGLUDEC	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.1346350544504987	IUPHAR.LIGAND:4068	iuphar.ligand:4068	(RS)-(TETRAZOL-5-YL)GLYCINE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
VEGFB	hgnc:12681	VEGFB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6731752722524936	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	NSC-659162	chembl:CHEMBL471005	CHEMBL:CHEMBL471005	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TETRAMETHRIN	drugbank:DB13752	TETRAMETHRIN	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.019896806	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.037003292	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.2573905452730122	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.068637479	APOMORPHINE HYDROCHLORIDE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	activator	2.386712328895204	ICENTICAFTOR	ncit:C174620	ICENTICAFTOR	FALSE	FALSE	FALSE
UNIPROT:Q14500	hgnc:6258	KCNJ12	TdgClinicalTrial	Jan-14	NULL	8.078103267029924	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.013716738	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CHYMASE	hgnc:2097	CMA1	TTD	2020.06.01	NULL	10.50153424713889	JNJ-10311795	iuphar.ligand:6563	JNJ-10311795	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.035418328	formoterol	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.085796848	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.022632617	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	GNF-PF-5554	chembl:CHEMBL580130	CHEMBL:CHEMBL580130	FALSE	FALSE	FALSE
TYMP	hgnc:3148	TYMP	NCI	14-Sep-17	NULL	0.546954909	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
IRS4	hgnc:6128	IRS4	PharmGKB	4/5/24	NULL	3.281729452230906	levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:3174	ncit:C65906	INCADRONIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.040515178	17-ALLYL-AMINOGELDANAMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	CLORGILINE	ncit:C77522	CLORGILINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	1,2,3,4,5,6-HEXABROMO-CYCLOHEXANE	chembl:CHEMBL444236	CHEMBL:CHEMBL444236	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	NCI	14-Sep-17	NULL	0.1640864726115453	6-HYDROXYDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.096167896	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
DDC	hgnc:2719	DDC	PharmGKB	4/5/24	NULL	5.250767123569449	carbidopa	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.09869863	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
ATG5	hgnc:589	ATG5	PharmGKB	4/5/24	NULL	3.182283105193606	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
PLEKHH2	hgnc:30506	PLEKHH2	PharmGKB	4/5/24	NULL	1.166837138570988	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.062509132	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.2220197515251353	Dexmedetomidine	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1489	hgnc:2499	CTF1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9369	iuphar.ligand:9369	KB-NB142-70	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:8464	iuphar.ligand:8464	DROXINOSTAT	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	0.5707355569097228	APROCITENTAN	ncit:C174728	APROCITENTAN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	METRAZOLINE OXALATE	chembl:CHEMBL1255866	METRAZOLINE OXALATE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.037884323	IUPHAR.LIGAND:177	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.1657439117288336	COPANLISIB	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
MT-ND3	hgnc:7458	MT-ND3	ChEMBL	33	inhibitor	0.2625383561784725	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	ChEMBL	33	inhibitor	2.187819634820604	FASITIBANT CHLORIDE	ncit:C167030	FASITIBANT CHLORIDE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	2.187819634820604	NSC-341622	chembl:CHEMBL79513	CHEMBL:CHEMBL79513	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	GNF-PF-5381	chembl:CHEMBL578109	CHEMBL:CHEMBL578109	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005669763	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	CARBOQUONE	ncit:C342	CARBOQUONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002542252	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.5556367326528517	KERACYANIN	rxcui:28165	KERACYANIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.003376265	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.1215455352678113	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:10365	iuphar.ligand:10365	COMPOUND 2Q [PMID: 30986068]	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	2-METHOXYPHENAZINE	chembl:CHEMBL1420181	CHEMBL:CHEMBL1420181	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	GNF-PF-5219	chembl:CHEMBL602012	CHEMBL:CHEMBL602012	FALSE	FALSE	FALSE
RPL37	hgnc:10347	RPL37	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
UNIPROT:Q92887	hgnc:53	ABCC2	TdgClinicalTrial	Jan-14	NULL	0.1562728310586145	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
SLC9A8	hgnc:20728	SLC9A8	PharmGKB	4/5/24	NULL	1.591141552596803	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.2917092846427472	Pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	GNF-PF-1678	chembl:CHEMBL580340	CHEMBL:CHEMBL580340	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.030832455	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	0.2800409132570373	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.1286952726365061	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.03151721	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	BEVASIRANIB	ncit:C169809	BEVASIRANIB	FALSE	FALSE	FALSE
UNIPROT:Q13200	hgnc:9559	PSMD2	TdgClinicalTrial	Jan-14	NULL	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1296	hgnc:2216	COL8A2	GuideToPharmacology	2024.1	activator	2.625383561784725	IUPHAR.LIGAND:2351	iuphar.ligand:2351	CALMODULIN	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	TYRA-200	ncit:C203336	FGFR1/2/3 INHIBITOR TYRA-200	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	FANCHININ	drugbank:DB14066	TETRANDRINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	SIB-1757	iuphar.ligand:1431	SIB-1757	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	PharmGKB	4/5/24	NULL	0.2651902587661338	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
IVL	hgnc:6187	IVL	PharmGKB	4/5/24	NULL	0.5303805175322677	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	2.234368988752957	GANTACURIUM CHLORIDE	ncit:C175789	GANTACURIUM CHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:2734	hgnc:4316	GLG1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8236	iuphar.ligand:8236	I-CBP112	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	PharmGKB	4/5/24	NULL	0.060043077	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NCBIGENE:719	hgnc:1319	C3AR1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.1389091831632129	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.1835932560688619	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.021301287	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.022949157	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.5791287268642775	GALANTAMINE HYDROBROMIDE	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	1.544343271638073	IUPHAR.LIGAND:11367	iuphar.ligand:11367	[18F]FEPPG	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.1944728564284981	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.1159109740302306	MDM2 INHIBITOR AMGMDS3	ncit:C171616	MDM2 INHIBITOR AMGMDS3	FALSE	FALSE	TRUE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	1.166837138570988	Ouabain	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	QUERCETIN DIHYDRATE	ncit:C75768	QUERCETIN DIHYDRATE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
UNIPROT:Q7Z2W7	hgnc:17961	TRPM8	TdgClinicalTrial	Jan-14	NULL	4.836232876971861	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1715936968486748	5,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484662	CHEMBL:CHEMBL484662	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	8-[(3-TRIFLUOROMETHYL)BENZYLOXY]CAFFEINE	chembl:CHEMBL602466	CHEMBL:CHEMBL602466	FALSE	FALSE	FALSE
EIF4E2	hgnc:3293	EIF4E2	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
GP1BA	hgnc:4439	GP1BA	ChEMBL	33	inhibitor	4.773424657790408	ANFIBATIDE	drugbank:DB15094	ANFIBATIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	FLAVOKAWAIN B	chembl:CHEMBL104255	FLAVOKAWAIN B	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.019949723	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	TCMDC-124317	chembl:CHEMBL586937	CHEMBL:CHEMBL586937	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.04464938	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
CXCL12	hgnc:10672	CXCL12	PharmGKB	4/5/24	NULL	0.305277158	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:3249	iuphar.ligand:3249	[11C]VOLINANSERIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	SULFADOXINE	rxcui:10173	SULFADOXINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	NCI	14-Sep-17	NULL	0.028598949	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.045898314	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.3125456621172291	TCMDC-125480	chembl:CHEMBL546257	CHEMBL:CHEMBL546257	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.033148782	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	PharmGKB	4/5/24	NULL	1.406455479527531	Antihypertensives	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
GUANYLATE CYCLASE	hgnc:4187	GC	TTD	2020.06.01	NULL	0.4375639269641209	Isosorbide Mononitrate	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001276441	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.006847636	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.036977233	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	blocker	0.172722603	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2365210416022274	KU-55933	iuphar.ligand:5928	KU-55933	FALSE	FALSE	FALSE
HMOX2	hgnc:5014	HMOX2	NCI	14-Sep-17	NULL	0.6848826682916673	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	0.3106962795011509	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
OPN1LW	hgnc:9936	OPN1LW	DTC	9/2/20	NULL	5.250767123569449	13-CIS-RETINAL	iuphar.ligand:6671	13-CIS-RETINAL	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.076840494	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1988926940746003	SIBUTRAMINE	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	0.6563458904461812	Dextromethorphan	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C9	hgnc:60	ABCC9	TTD	2020.06.01	NULL	0.596678082	Tolbutamide	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	0.8334550989792778	FUROSEMIDE	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	3.281729452230906	E 7974	chembl:CHEMBL4650465	E-7974	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ETONITAZENE	ncit:C65596	ETONITAZENE	FALSE	FALSE	FALSE
NDUFA4L2	hgnc:29836	NDUFA4L2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	ChEMBL	33	inhibitor	0.1035654265003836	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:12026	ncit:C170368	RESMETIROM	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	HEMATOXYLIN	drugbank:DB16871	HEMATOXYLIN	FALSE	FALSE	FALSE
SCD	hgnc:10571	SCD	NCI	14-Sep-17	NULL	0.6819178082557728	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.025588534	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.020591244	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.006420601	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.1215455352678113	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.020117882	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	ChEMBL	33	inhibitor	0.5707355569097228	DEFACTINIB	ncit:C79809	DEFACTINIB	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	0.5707355569097228	AZD0328	iuphar.ligand:7697	AZD0328	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.014145386	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	MECLIZINE DIHCL	chembl:CHEMBL1085765	MECLIZINE DIHCL	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	TCMDC-125785	chembl:CHEMBL588525	CHEMBL:CHEMBL588525	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1584738568481725	Fruquintinib	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE PIM-1	hgnc:8986	PIM1	TTD	2020.06.01	NULL	1.500219178	SEL-24	drugbank:DB18082	SEL-24	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.035574303	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.07699072	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1333528158366844	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1269	iuphar.ligand:1269	4-METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:12433	iuphar.ligand:12433	DENATONIUM	FALSE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.6563458904461812	TOLBUTAMIDE	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
PSMA1	hgnc:9530	PSMA1	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSEN1	hgnc:9508	PSEN1	ChEMBL	33	inhibitor	0.5048814541893701	BEGACESTAT	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
NPM1	hgnc:7910	NPM1	PharmGKB	4/5/24	NULL	0.7143900848393808	venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
UNIPROT:O60603	hgnc:11848	TLR2	TdgClinicalTrial	Jan-14	NULL	3.750547945	DIAPEP277	drugbank:DB06651	DIAPEP 277	FALSE	FALSE	FALSE
UNIPROT:P51170	hgnc:10602	SCNN1G	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	GS-9411	chembl:CHEMBL4297254	552-02	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	GNF-PF-2094	chembl:CHEMBL578928	CHEMBL:CHEMBL578928	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.3298911281823738	Ulixertinib	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.2470949234620917	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.2778183663264259	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.092443083	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	1.458546423213736	GW493838	chembl:CHEMBL3545223	GW493838	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	agonist	0.042073455	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	AGROCLAVINE	chembl:CHEMBL449081	AGROCLAVINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004252322	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	DNDI1416982	chembl:CHEMBL1479114	CHEMBL:CHEMBL1479114	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	0.7955707762984014	Triptoreline	rxcui:38782	TRIPTORELIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	(-)-PROPANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
MIA	hgnc:7076	MIA	NCI	14-Sep-17	NULL	35.00511415712966	TRP-1	ncit:C28725	RECOMBINANT TYROSINASE-RELATED PROTEIN-1	FALSE	FALSE	FALSE
PLAT	hgnc:9051	PLAT	NCI	14-Sep-17	NULL	1.363835616511545	LYMPHOKINES	ncit:C621	RECOMBINANT LYMPHOKINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	NCI	14-Sep-17	NULL	0.020836377	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
DUX1	hgnc:3079	DUX1	PharmGKB	4/5/24	NULL	0.9460841664089098	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	Desloratadine	rxcui:275635	DESLORATADINE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	DNDI1416985	chembl:CHEMBL593211	CHEMBL:CHEMBL593211	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	4-CHLOROBENZALDEHYDE	chembl:CHEMBL1474	CHEMBL:CHEMBL1474	FALSE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	NCI	14-Sep-17	NULL	5.834185692854944	OCTASTATIN	chembl:CHEMBL2218872	VAPREOTIDE ACETATE	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	inverse agonist	0.039068208	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
TNFSF4	hgnc:11934	TNFSF4	ChEMBL	33	inhibitor	26.25383561784724	KY-1005	chembl:CHEMBL4594569	KY-1005	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	modulator	0.008751279	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	ChEMBL	33	inhibitor	0.4730420832044549	EDASALONEXENT	ncit:C171665	EDASALONEXENT	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.096521454	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1374032518317239	Nintedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.030868707	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
NCBIGENE:1444	hgnc:2442	CSHL1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:5247	iuphar.ligand:5247	PROPARGYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:1003	iuphar.ligand:1003	[3H]BQ123	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:304	iuphar.ligand:304	PENTYLTHIO-TZTP	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	ChEMBL	33	inhibitor	5.000730593875666	IMD-1041	chembl:CHEMBL3545168	IMD-1041	FALSE	FALSE	FALSE
UNIPROT:P51451	hgnc:1057	BLK	TdgClinicalTrial	Jan-14	NULL	0.040328473	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:729	hgnc:1339	C6	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9332	iuphar.ligand:9332	JQEZ5	FALSE	FALSE	TRUE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:5515	iuphar.ligand:5515	COMPOUND 7E [PMID: 21571530]	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.039420174	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	ILEPCIMIDE	ncit:C72810	ILEPCIMIDE	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	0.074797252	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9074	rxcui:89778	ECOTHIOPATE	TRUE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:1379	iuphar.ligand:1379	LY367385	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.093763699	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	1.591141552596803	N-(3-CARBOXYPHENYL)RHODANINE	chembl:CHEMBL442906	CHEMBL:CHEMBL442906	FALSE	FALSE	FALSE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.7292732116068681	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	DIMETHISOQUIN	ncit:C72169	DIMETHISOQUIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002258977	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.1988926940746003	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.8468979231563628	Butacaine	rxcui:1829	BUTACAINE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.023336743	IUPHAR.LIGAND:214	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:304	iuphar.ligand:304	PENTYLTHIO-TZTP	FALSE	FALSE	FALSE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.3889457128569963	Tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.1842374429322613	Valproate	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	0.138178082	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	DIAMIDE	chembl:CHEMBL1255835	DIAMIDE	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	TALC	12-May-16	inhibitor	1.193356164447602	LY2181308	drugbank:DB05141	LY2181308	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.1994593399266647	levomethadyl acetate	rxcui:237005	LEVOMETHADYL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.022136455	umeclidinium	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	2.763561643983921	ACETYLSULFANILAMIDE	chembl:CHEMBL687	ACETYLSULFANILAMIDE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
FXYD2	hgnc:4026	FXYD2	ChEMBL	33	inhibitor	0.2302968036653267	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
TRAC	hgnc:12029	TRAC	ChEMBL	33	inhibitor	2.625383561784725	TOL-101	drugbank:DB16980	TOL-101	FALSE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	IBRITUMOMAB TIUXETAN	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.019881738	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:2754	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
NCBIGENE:1722	hgnc:7217	MPL	GuideToPharmacology	2024.1	agonist	3.182283105193605	IUPHAR.LIGAND:10032	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.01864619	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.025929714	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
UNIPROT:Q8NBP7	hgnc:20001	PCSK9	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	REGN727	rxcui:1659152	ALIROCUMAB	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005669763	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	CLORGILINE	ncit:C77522	CLORGILINE	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	0.7001022831425933	RUCAPARIB CAMSYLATE	rxcui:1862578	RUCAPARIB CAMSYLATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	ChEMBL	33	inhibitor	0.3365876361262467	ZOSUQUIDAR	ncit:C76198	ZOSUQUIDAR	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.092606122	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10220	ncit:C123826	FISOGATINIB	FALSE	FALSE	TRUE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.060984519	IUPHAR.LIGAND:4108	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.086219493	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.016418909	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
KCNK9	hgnc:6283	KCNK9	ChEMBL	33	potentiator	0.2822993077187876	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	METHAPYRILENE HYDROCHLORIDE	rxcui:235721	METHAPYRILENE HYDROCHLORIDE	TRUE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.900131507	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.001507152	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.2983390411119005	GDC-0623	drugbank:DB11982	GDC-0623	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	chembl:CHEMBL1333512	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
VIM	hgnc:12692	VIM	NCI	14-Sep-17	NULL	1.312691780892362	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
MS4A2	hgnc:7316	MS4A2	PharmGKB	4/5/24	NULL	0.037639908	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.038256955	Pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8062	iuphar.ligand:8062	MRT67307	FALSE	FALSE	FALSE
NCBIGENE:2042	hgnc:3387	EPHA3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.3860858179095183	IUPHAR.LIGAND:6222	iuphar.ligand:6222	COMPOUND 2 [PMID: 21105727]	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.029654182	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-216385	chembl:CHEMBL274863	CHEMBL:CHEMBL274863	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	1.591141552596802	DIETHYL-2-TETRADECYLIDENEMALONATE	chembl:CHEMBL257748	CHEMBL:CHEMBL257748	FALSE	FALSE	FALSE
ALDH5A1	hgnc:408	ALDH5A1	PharmGKB	4/5/24	NULL	0.6579908676152193	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	SEROTONIN	rxcui:1311214	SEROTONIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CHLOROPHENOTHANE	chembl:CHEMBL416898	CHLOROPHENOTHANE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.1375060601009582	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:1328	iuphar.ligand:1328	HS024	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.2344092465879218	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	PharmGKB	4/5/24	NULL	0.016869935	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1400204566285186	RHIL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.016156207	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011746683	vilazodone	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.022220766	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:459	iuphar.ligand:459	MRE 3008F20	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.1392776425349987	IUPHAR.LIGAND:8018	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.042006137	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:486	hgnc:4026	FXYD2	GuideToPharmacology	2024.1	blocker	0.3977853881492008	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.085378327	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.057700738	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
SRMS	hgnc:11298	SRMS	DTC	9/2/20	NULL	0.1131630845596864	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.297662535	PD-0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.2187819634820604	NAPROXCINOD	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.006210251	IUPHAR.LIGAND:7281	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2616	iuphar.ligand:2616	TETRODOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.036387853	IUPHAR.LIGAND:2399	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.003053304	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CD55	hgnc:2665	CD55	NCI	14-Sep-17	NULL	0.2308029504865692	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.032899543	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	NSC-36398	chembl:CHEMBL483206	CHEMBL:CHEMBL483206	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.1562728310586145	trastuzumab deruxtecan	rxcui:2267574	FAM-TRASTUZUMAB DERUXTECAN-NXKI	TRUE	FALSE	TRUE
METHIONINE AMINOPEPTIDASE 2	hgnc:16672	METAP2	TTD	2020.06.01	NULL	9.845188356692718	Beloranib	ncit:C90656	BELORANIB	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.043756393	ofloxacin	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
CSNK2A2	hgnc:2459	CSNK2A2	DTC	9/2/20	inhibitor	0.6563458904461813	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	3.500511415712966	ASP-9521	ncit:C133224	17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 5 INHIBITOR ASP9521	FALSE	FALSE	FALSE
DYRK4	hgnc:3095	DYRK4	DTC	9/2/20	NULL	0.3241214273808302	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	TALC	12-May-16	inhibitor	0.3453256329104173	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
UNIPROT:P16233	hgnc:9155	PNLIP	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	CETILISTAT	ncit:C77404	CETILISTAT	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.100976291	RANOLAZINE	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:5690	iuphar.ligand:5690	KI-20227	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	6-NITROQUIPAZINE	chembl:CHEMBL41140	6-NITROQUIPAZINE	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.4817217544559128	ALFENTANIL	rxcui:203203	ALFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	0.8334550989792778	Furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.1000146118775133	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.084146909	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
NCBIGENE:2757	hgnc:23177	KEAP1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8772	iuphar.ligand:8772	NRF2 PEPTIDE [PMID: 23647822]	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6447	iuphar.ligand:6447	COMPOUND 13 [PMID: 15686941]	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	inhibitor	0.5966780822238011	IUPHAR.LIGAND:12661	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.031310478	IUPHAR.LIGAND:2399	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1219690388750162	NG-MONOMETHYL-L-ARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	PharmGKB	4/5/24	NULL	0.1852122442176172	venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
UNIPROT:O43497	hgnc:1394	CACNA1G	TEND	1-Aug-11	NULL	0.097236428	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	RACEPINEPHRINE	rxcui:66887	RACEPINEPHRINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	CLOBENPROPIT	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	GNF-PF-2307	chembl:CHEMBL421088	CHEMBL:CHEMBL421088	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TRICLOFENOL	chembl:CHEMBL109095	TRICLOFENOL	FALSE	FALSE	FALSE
SIRPA	hgnc:9662	SIRPA	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.027752469	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	1.050153425	IUPHAR.LIGAND:12648	ncit:C174710	SUVECALTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:1821	iuphar.ligand:1821	[ILE5,TRP23]PTHRP-(5-36)	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:3504	iuphar.ligand:3504	JNJ-5207787	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	NEBULARINE	drugbank:DB04440	NEBULARINE	FALSE	FALSE	FALSE
RETICULON-4	hgnc:14085	RTN4	TTD	2020.06.01	NULL	21.00306849427779	ATI-355	drugbank:DB17923	ATI-355	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	1.193356164447602	ZD9331	ncit:C1629	PLEVITREXED	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	FANCHININ	drugbank:DB14066	TETRANDRINE	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8546	iuphar.ligand:8546	TG7-171	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	blocker	0.8334550989792776	IUPHAR.LIGAND:4229	iuphar.ligand:4229	JORO SPIDER TOXIN	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6335	iuphar.ligand:6335	MK-5435	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:2219	iuphar.ligand:2219	D(CH2)5[TYR(ME)2,THR4,PHE(3I,4N3)-NH29]OVT	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.2011788169949981	ANTIHISTAMINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1620607136904151	DICYCLOHEXYLCARBODIIMIDE	chembl:CHEMBL162598	DICYCLOHEXYLCARBODIIMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	PHENYL AMINOSALICYLATE	ncit:C66376	PHENYL AMINOSALICYLATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BENZO[B]TRIPHENYLENE	chembl:CHEMBL166266	BENZO[B]TRIPHENYLENE	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.546954909	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1282238613814273	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.061412481	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3A	hgnc:8778	PDE3A	TTD	2020.06.01	NULL	0.2983390411119005	VESNARINONE	ncit:C1415	VESNARINONE	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	2.625383561784724	S-555739	iuphar.ligand:11951	ASAPIPRANT	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	TCMDC-123769	chembl:CHEMBL534353	CHEMBL:CHEMBL534353	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	negative modulator	0.079197091	KETAMINE HYDROCHLORIDE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATP1B2	hgnc:805	ATP1B2	ChEMBL	33	inhibitor	0.9723642821424908	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
UCP2	hgnc:12518	UCP2	NCI	14-Sep-17	NULL	0.8334550989792776	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.063568609	SIB-1757	iuphar.ligand:1431	SIB-1757	FALSE	FALSE	FALSE
KCNH1	hgnc:6250	KCNH1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.018942161	IUPHAR.LIGAND:204	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1281	iuphar.ligand:1281	[125I]KISSPEPTIN-10 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.036718651	IUPHAR.LIGAND:2174	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:9930	iuphar.ligand:9930	HENATINIB	FALSE	FALSE	FALSE
NCBIGENE:2887	hgnc:4564	GRB10	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9016	iuphar.ligand:9016	LM10	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:2456	iuphar.ligand:2456	AMP-PNP	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.072424374	SERTACONAZOLE NITRATE	rxcui:236601	SERTACONAZOLE NITRATE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	SJ000032159	chembl:CHEMBL591361	CHEMBL:CHEMBL591361	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.1770916399180253	solanidine	iuphar.ligand:12500	SOLANIDINE	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:9283	iuphar.ligand:9283	TG6-129	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.4449802647092754	BENAZEPRIL HYDROCHLORIDE	rxcui:235758	BENAZEPRIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:8362	rxcui:2049846	ELAGOLIX	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5757	ncit:C95194	VESTIPITANT	FALSE	FALSE	FALSE
NCBIGENE:1030	hgnc:1788	CDKN2B	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:8798	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	TALC	12-May-16	inhibitor	0.42006137	NEOVASTAT	drugbank:DB05387	NEOVASTAT	FALSE	FALSE	TRUE
TTK	hgnc:12401	TTK	DTC	9/2/20	inhibitor	0.4375639269641209	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
PTBP1	hgnc:9583	PTBP1	DTC	9/2/20	NULL	0.9723642821424908	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.1909369863116163	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GUANYLYL CYCLASE C	hgnc:4688	GUCY2C	TTD	2020.06.01	NULL	19.69037671338543	MD-1100	rxcui:1307404	LINACLOTIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003162351	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	0.5000730593875666	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
KCNK18	hgnc:19439	KCNK18	ChEMBL	33	potentiator	0.3387591692625452	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.1717808219270267	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:475	iuphar.ligand:475	VUF8504	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.004951218	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV006656	chembl:CHEMBL606159	CHEMBL:CHEMBL606159	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-8186	chembl:CHEMBL122355	CHEMBL:CHEMBL122355	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00410569	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.2892984641085096	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.100976291	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
MAD1L1	hgnc:6762	MAD1L1	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005527705	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
UHRF1	hgnc:12556	UHRF1	PharmGKB	4/5/24	NULL	1.842374429322614	afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
LEPR	hgnc:6554	LEPR	PharmGKB	4/5/24	NULL	2.187819634820604	setmelanotide	rxcui:2469247	SETMELANOTIDE	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.062509132	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00267133	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1363127498330594	ESTROGENS, CONJUGATED	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.048083948	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23763	hgnc:12642	VAMP1	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	BOTULINUM TOXIN TYPE B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.081407242	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12239	iuphar.ligand:12239	JNJ-64264681	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	HURATOXIN	chembl:CHEMBL470375	HURATOXIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	ARASERTACONAZOLE	ncit:C79926	ARASERTACONAZOLE	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2892984641085096	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CancerCommons	25-Jul-13	inhibitor	0.3453256329104173	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
MSH5	hgnc:7328	MSH5	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CancerCommons	25-Jul-13	inhibitor	NULL	PLX108-01	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CancerCommons	25-Jul-13	inhibitor	NULL	PLX108-01	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	CancerCommons	25-Jul-13	inhibitor	3.000438356	ONARTUZUMAB	ncit:C82348	ONARTUZUMAB	FALSE	TRUE	TRUE
CTLA4	hgnc:2505	CTLA4	CancerCommons	25-Jul-13	antibody	0.7001022831425934	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
HGF	hgnc:4893	HGF	CancerCommons	25-Jul-13	inhibitor	7.778914257139925	AMG 102	ncit:C67079	RILOTUMUMAB	FALSE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	CancerCommons	25-Jul-13	inhibitor	0.085796848	GELFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	NULL	Fluvestrant	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	0.6050266644442165	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CGI	2/1/22	NULL	0.9842513760562132	AG-120	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
MLL	hgnc:7132	KMT2A	CGI	2/1/22	NULL	0.027047221	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.1712206670729168	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.011591097	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	1.346350544504987	RANIBIZUMAB	rxcui:595060	RANIBIZUMAB	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1773907812016706	ISOPROPAMIDE IODIDE	rxcui:6051	ISOPROPAMIDE IODIDE	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	1.381780822	DABIGATRAN ETEXILATE MESYLATE	rxcui:1037041	DABIGATRAN ETEXILATE MESYLATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.1988926940746003	SOTALOL HYDROCHLORIDE	rxcui:7008	SOTALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	BETAXOLOL HYDROCHLORIDE	rxcui:142144	BETAXOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
SIGMAR1	hgnc:8157	SIGMAR1	ChEMBL	33	agonist	0.6563458904461812	DEXTROMETHORPHAN POLISTIREX	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
CCKAR	hgnc:1570	CCKAR	ChEMBL	33	agonist	2.625383561784724	CERULETIDE DIETHYLAMINE	rxcui:20024	CERULETIDE DIETHYLAMINE	TRUE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	0.1835932560688619	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	DESVENLAFAXINE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1193356164447602	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1790034246671403	VILAZODONE HYDROCHLORIDE	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.088396753	dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	0.630092055	SITAGLIPTIN PHOSPHATE	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	agonist	0.9907107780319716	MECASERMIN RINFABATE	rxcui:616877	MECASERMIN RINFABATE	TRUE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	ChEMBL	33	agonist	6.563458904461812	SERACTIDE ACETATE	rxcui:1999801	SERACTIDE ACETATE	TRUE	FALSE	FALSE
ILES	NULL	NULL	ChEMBL	33	inhibitor	NULL	MUPIROCIN	rxcui:42372	MUPIROCIN	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.2453629496995069	AMPHETAMINE SULFATE	rxcui:81952	AMPHETAMINE SULFATE	TRUE	FALSE	FALSE
TMP1	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLUCYTOSINE	rxcui:4451	FLUCYTOSINE	TRUE	FALSE	FALSE
KCNN4	hgnc:6293	KCNN4	ChEMBL	33	potentiator	2.917092846427472	CHLORZOXAZONE	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.1110098757625676	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
MMP13	hgnc:7159	MMP13	ChEMBL	33	inhibitor	0.2853677784548614	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
MMP7	hgnc:7174	MMP7	ChEMBL	33	inhibitor	0.6522692078968261	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
MMP13	hgnc:7159	MMP13	ChEMBL	33	inhibitor	0.2853677784548614	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	15.31473744374422	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
GUCY2C	hgnc:4688	GUCY2C	ChEMBL	33	agonist	19.69037671338543	LINACLOTIDE	rxcui:1307404	LINACLOTIDE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	2.917092846427472	PITAVASTATIN CALCIUM	rxcui:861640	PITAVASTATIN CALCIUM	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.067231333	OXYMORPHONE HYDROCHLORIDE	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1751715470748774	OXYMORPHONE HYDROCHLORIDE	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.048708415	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.053038052	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.1988926940746003	CARTEOLOL HYDROCHLORIDE	rxcui:142132	CARTEOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.1620607136904151	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.100976291	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.073437302	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.067839369	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.082171629	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3571950424196904	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.4412409347537352	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1704794520639432	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1403266238077355	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.31919557	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.035083077	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.5427149481725528	ARFORMOTEROL TARTRATE	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
IL11RA	hgnc:5967	IL11RA	ChEMBL	33	agonist	10.50153425	OPRELVEKIN	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
COL4A4	hgnc:2206	COL4A4	ChEMBL	33	cleavage	0.6250913242344582	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL5A1	hgnc:2209	COL5A1	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL4A1	hgnc:2202	COL4A1	ChEMBL	33	cleavage	0.4688184931758437	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL28A1	hgnc:22442	COL28A1	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
PSMD1	hgnc:9554	PSMD1	ChEMBL	33	inhibitor	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA8	hgnc:22985	PSMA8	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
8238086	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8232915	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8231029	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8238343	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8234840	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.04339477	formoterol	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
8232678	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
SCNN1B	hgnc:10600	SCNN1B	PharmGKB	4/5/24	NULL	3.281729452230906	Farglitazar	ncit:C81693	FARGLITAZAR	FALSE	FALSE	FALSE
8237618	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8238380	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8234407	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
MTHFD1	hgnc:7432	MTHFD1	PharmGKB	4/5/24	NULL	0.2715914029432474	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
8237795	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8236088	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8236974	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8237447	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8234408	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8238085	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.1304538415793652	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
8229807	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	PharmGKB	4/5/24	NULL	0.005459124	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
8240195	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8230924	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8230507	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8233823	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8233620	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8232310	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.1801292323694494	antithymocyte globulin	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
8230937	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8236087	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8234154	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8230957	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8233619	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8235475	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1909369863116163	AMPRENAVIR	rxcui:228656	AMPRENAVIR	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.8751278539282416	LISDEXAMFETAMINE DIMESYLATE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.035358701	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.4688184931758437	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
GLRB	hgnc:4329	GLRB	ChEMBL	33	agonist	0.2386712328895204	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
EPHA1	hgnc:3385	EPHA1	ChEMBL	33	inhibitor	0.4526523382387457	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
LRP1B	hgnc:6693	LRP1B	PharmGKB	4/5/24	NULL	0.5224643904049203	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
EPHB1	hgnc:3392	EPHB1	ChEMBL	33	inhibitor	0.015088411	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GLRA1	hgnc:4326	GLRA1	ChEMBL	33	agonist	0.072324616	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1101693521639275	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NDUFB3	hgnc:7698	NDUFB3	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFB2	hgnc:7697	NDUFB2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFC2	hgnc:7706	NDUFC2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.092199598	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NDUFB10	hgnc:7696	NDUFB10	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFS3	hgnc:7710	NDUFS3	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PSMD14	hgnc:16889	PSMD14	PharmGKB	4/5/24	NULL	0.1205687054780585	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NDUFAF1	hgnc:18828	NDUFAF1	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFV2	hgnc:7717	NDUFV2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.027752469	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.026519026	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
ATP1B3	hgnc:806	ATP1B3	ChEMBL	33	inhibitor	0.9723642821424908	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
ATP1A2	hgnc:800	ATP1A2	ChEMBL	33	inhibitor	0.3947945205691315	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.059690418	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.073403082	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.066577774	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.070448575	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.07767407	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	agonist	0.037398626	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.020656047	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.020164236	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.033658764	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.104492878	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
LCK	hgnc:6524	LCK	ChEMBL	33	inhibitor	0.05348375	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.03409589	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TICARCILLIN DISODIUM	rxcui:142447	TICARCILLIN DISODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TICARCILLIN DISODIUM	rxcui:142447	TICARCILLIN DISODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TICARCILLIN DISODIUM	rxcui:142447	TICARCILLIN DISODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TICARCILLIN DISODIUM	rxcui:142447	TICARCILLIN DISODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TICARCILLIN DISODIUM	rxcui:142447	TICARCILLIN DISODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TICARCILLIN DISODIUM	rxcui:142447	TICARCILLIN DISODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TICARCILLIN DISODIUM	rxcui:142447	TICARCILLIN DISODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
TMEFF2	hgnc:11867	TMEFF2	PharmGKB	4/5/24	NULL	1.567393171214761	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN V	rxcui:7984	PENICILLIN V	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BACAMPICILLIN HYDROCHLORIDE	rxcui:327584	BACAMPICILLIN HYDROCHLORIDE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	BACAMPICILLIN HYDROCHLORIDE	rxcui:327584	BACAMPICILLIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	BACAMPICILLIN HYDROCHLORIDE	rxcui:327584	BACAMPICILLIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BACAMPICILLIN HYDROCHLORIDE	rxcui:327584	BACAMPICILLIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	BACAMPICILLIN HYDROCHLORIDE	rxcui:327584	BACAMPICILLIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	BACAMPICILLIN HYDROCHLORIDE	rxcui:327584	BACAMPICILLIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	BACAMPICILLIN HYDROCHLORIDE	rxcui:327584	BACAMPICILLIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFORANIDE	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFORANIDE	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFORANIDE	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFORANIDE	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFORANIDE	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFORANIDE	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
CCNK	hgnc:1596	CCNK	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFORANIDE	rxcui:20486	CEFORANIDE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAZOLIN SODIUM	rxcui:203171	CEFAZOLIN SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAZOLIN SODIUM	rxcui:203171	CEFAZOLIN SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAZOLIN SODIUM	rxcui:203171	CEFAZOLIN SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAZOLIN SODIUM	rxcui:203171	CEFAZOLIN SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAZOLIN SODIUM	rxcui:203171	CEFAZOLIN SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAZOLIN SODIUM	rxcui:203171	CEFAZOLIN SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAZOLIN SODIUM	rxcui:203171	CEFAZOLIN SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DORIPENEM	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DORIPENEM	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DORIPENEM	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DORIPENEM	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DORIPENEM	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DORIPENEM	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DORIPENEM	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN HYDROCHLORIDE	rxcui:281942	CEPHALEXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN HYDROCHLORIDE	rxcui:281942	CEPHALEXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN HYDROCHLORIDE	rxcui:281942	CEPHALEXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN HYDROCHLORIDE	rxcui:281942	CEPHALEXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN HYDROCHLORIDE	rxcui:281942	CEPHALEXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN HYDROCHLORIDE	rxcui:281942	CEPHALEXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHALEXIN HYDROCHLORIDE	rxcui:281942	CEPHALEXIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.077616661	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LORACARBEF	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LORACARBEF	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEROPENEM	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G BENZATHINE	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G BENZATHINE	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G BENZATHINE	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.128067491	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G BENZATHINE	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G BENZATHINE	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G BENZATHINE	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G BENZATHINE	rxcui:7982	PENICILLIN G BENZATHINE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G SODIUM	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G SODIUM	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G SODIUM	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G SODIUM	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G SODIUM	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G SODIUM	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G SODIUM	rxcui:9900	PENICILLIN G SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERACILLIN SODIUM	rxcui:203134	PIPERACILLIN SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERACILLIN SODIUM	rxcui:203134	PIPERACILLIN SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERACILLIN SODIUM	rxcui:203134	PIPERACILLIN SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERACILLIN SODIUM	rxcui:203134	PIPERACILLIN SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERACILLIN SODIUM	rxcui:203134	PIPERACILLIN SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERACILLIN SODIUM	rxcui:203134	PIPERACILLIN SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERACILLIN SODIUM	rxcui:203134	PIPERACILLIN SODIUM	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
PPP2R5D	hgnc:9312	PPP2R5D	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
FOXO1	hgnc:3819	FOXO1	PharmGKB	4/5/24	NULL	0.2561349816375341	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	PharmGKB	4/5/24	NULL	0.1715936968486748	methylprednisolone	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.3977853881492006	pilsicainide	ncit:C72582	PILSICAINIDE	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
FCGR2A	hgnc:3616	FCGR2A	PharmGKB	4/5/24	NULL	0.7778914257139925	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.2134458180312784	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	modulator	0.1875273972703375	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	modulator	0.1458546423213736	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	modulator	0.1312691780892362	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	modulator	0.1458546423213736	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	4.773424657790408	ENTECAVIR	rxcui:1546027	ENTECAVIR ANHYDROUS	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	4.773424657790408	TELBIVUDINE	rxcui:474128	TELBIVUDINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.058602312	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.021189536	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.042619863	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.016743518	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.054695491	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1041818873724097	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.1666910197958555	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.2059124362184097	PRAMIPEXOLE DIHYDROCHLORIDE	rxcui:236747	PRAMIPEXOLE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.069180068	PRAMIPEXOLE DIHYDROCHLORIDE	rxcui:236747	PRAMIPEXOLE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.1666910197958555	PRAMIPEXOLE DIHYDROCHLORIDE	rxcui:236747	PRAMIPEXOLE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.077217164	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.1029562181092048	DROPERIDOL	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
BLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVIBACTAM SODIUM	rxcui:1603833	AVIBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-3	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVIBACTAM SODIUM	rxcui:1603833	AVIBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-4	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVIBACTAM SODIUM	rxcui:1603833	AVIBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-5	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVIBACTAM SODIUM	rxcui:1603833	AVIBACTAM SODIUM	TRUE	FALSE	FALSE
BLAT-6	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVIBACTAM SODIUM	rxcui:1603833	AVIBACTAM SODIUM	TRUE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMBITASVIR	rxcui:1597371	OMBITASVIR	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	FINAFLOXACIN	rxcui:1598641	FINAFLOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FINAFLOXACIN	rxcui:1598641	FINAFLOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FINAFLOXACIN	rxcui:1598641	FINAFLOXACIN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.4375639269641208	propoxyphene	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
ANO1	hgnc:21625	ANO1	ChEMBL	33	blocker	17.50255707856483	CROFELEMER	rxcui:1364449	CROFELEMER	TRUE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	DACLATASVIR DIHYDROCHLORIDE	rxcui:1606217	DACLATASVIR DIHYDROCHLORIDE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.2083637747448194	L-21649	chembl:CHEMBL333021	L-21649	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2083637747448194	L-21649	chembl:CHEMBL333021	L-21649	FALSE	FALSE	FALSE
NDUFB6	hgnc:7701	NDUFB6	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.4667348554283955	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
NDUFA6	hgnc:7690	NDUFA6	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
SEPTIN3	hgnc:10750	SEPTIN3	PharmGKB	4/5/24	NULL	1.312691780892362	dextromethorphan	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.2792961235941196	LY-2874455	drugbank:DB13022	LY-2874455	FALSE	FALSE	FALSE
MT-ND4L	hgnc:7460	MT-ND4L	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.2853677784548614	mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
NDUFA13	hgnc:17194	NDUFA13	ChEMBL	33	inhibitor	0.2573905452730122	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB3	hgnc:7698	NDUFB3	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
IL12A	hgnc:5969	IL12A	PharmGKB	4/5/24	NULL	0.6563458904461812	mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
MT-ND5	hgnc:7461	MT-ND5	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB1	hgnc:7695	NDUFB1	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.4039051633514962	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
MT-ND2	hgnc:7456	MT-ND2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFAF1	hgnc:18828	NDUFAF1	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.3962843112127887	tocilizumab	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
NDUFV1	hgnc:7716	NDUFV1	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFA1	hgnc:7683	NDUFA1	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.2641895408085258	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
GALNT14	hgnc:22946	GALNT14	PharmGKB	4/5/24	NULL	0.2715914029432474	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NDUFS2	hgnc:7708	NDUFS2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB9	hgnc:7704	NDUFB9	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
GALNT14	hgnc:22946	GALNT14	PharmGKB	4/5/24	NULL	0.8950171233357017	mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NDUFS8	hgnc:7715	NDUFS8	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFC1	hgnc:7705	NDUFC1	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFC2	hgnc:7706	NDUFC2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.030886865	pioglitazone	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NDUFS5	hgnc:7712	NDUFS5	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1495945049449985	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.065634589	meloxicam	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.2381300282797936	RG-547	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1666910197958555	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	1.575230137070835	sulfanilamide	rxcui:10184	SULFANILAMIDE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1620607136904151	ZOTIRACICLIB	ncit:C171725	ZOTIRACICLIB	FALSE	FALSE	FALSE
GRM2	hgnc:4594	GRM2	ChEMBL	33	agonist	3.750547945	LY404039	chembl:CHEMBL375611	LY404039	FALSE	FALSE	FALSE
PAH	hgnc:8582	PAH	PharmGKB	4/5/24	NULL	0.4861821410712454	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	ChEMBL	33	inhibitor	0.28382525	XL-418	chembl:CHEMBL2016893	XL-418	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	1.458546423213736	RPR749	chembl:CHEMBL3545331	RPR749	FALSE	FALSE	FALSE
GRM2	hgnc:4594	GRM2	ChEMBL	33	agonist	3.750547945	LY2979165	chembl:CHEMBL3544939	LY2979165	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.019065966	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PRKCH	hgnc:9403	PRKCH	ChEMBL	33	inhibitor	0.280789686	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	ChEMBL	33	inhibitor	0.1544343271638073	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	ChEMBL	33	inhibitor	0.077217164	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.022099188	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	2.561349816375341	ABT-102	chembl:CHEMBL398338	ABT-102	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	ChEMBL	33	inhibitor	0.096521454	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	1.141471113819445	APN1125	chembl:CHEMBL3545013	APN1125	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	2.351089756822142	BI-811283	chembl:CHEMBL3545395	BI-811283	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	GOLVATINIB	ncit:C82363	GOLVATINIB	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.292250489	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.064111931	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.4930297768609811	IPATASERTIB	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1785975212098452	FAMITINIB	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1807492985738192	FAMITINIB	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.2459375701906065	FAMITINIB	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.046303061	FAMITINIB	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.546954909	IPATASERTIB	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	0.7095631248066824	AMP579	chembl:CHEMBL3545163	AMP579	FALSE	FALSE	FALSE
BDKRB1	hgnc:1029	BDKRB1	ChEMBL	33	inhibitor	5.834185692854944	MK0686	chembl:CHEMBL232943	MK0686	FALSE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	inhibitor	3.281729452230906	REGRELOR DISODIUM	ncit:C80841	REGRELOR DISODIUM	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.1400204566285186	ETALOCIB	ncit:C1626	ETALOCIB	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	2.561349816375341	DWP05195	chembl:CHEMBL3545229	DWP05195	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	ChEMBL	33	agonist	2.500365296937833	PF-00446687	drugbank:DB12517	PF-00446687	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	blocker	0.3061671792168775	LANICEMINE	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	blocker	0.217423069	LANICEMINE	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	1.141471113819445	AQW051	iuphar.ligand:7371	AQW051	FALSE	FALSE	FALSE
PAH	hgnc:8582	PAH	PharmGKB	4/5/24	NULL	17.50255707856483	carbocisteine	rxcui:2023	CARBOCYSTEINE	TRUE	FALSE	FALSE
TNFRSF8	hgnc:11923	TNFRSF8	ChEMBL	33	agonist	6.563458904461812	SGN-30	drugbank:DB05471	SGN-30	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.6731752722524935	AMA0076	chembl:CHEMBL3545073	AMA0076	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	positive modulator	0.596678082	FARAMPATOR	ncit:C65620	FARAMPATOR	FALSE	FALSE	FALSE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.1296485709523321	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	inverse agonist	0.040515178	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	inverse agonist	0.041540879	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	inverse agonist	0.042073455	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	PharmGKB	4/5/24	NULL	0.2083637747448194	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	inverse agonist	0.040021091	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.1022876712383659	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
KCNN4	hgnc:6293	KCNN4	ChEMBL	33	blocker	35.00511415712966	SENICAPOC	ncit:C76882	SENICAPOC	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	1.419126249613364	NALUZOTAN	ncit:C80775	NALUZOTAN	FALSE	FALSE	FALSE
CXCR1	hgnc:6026	CXCR1	ChEMBL	33	modulator	5.000730593875666	REPARIXIN	ncit:C66515	REPARIXIN	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	1.591141552596803	ELAGOLIX	rxcui:2049846	ELAGOLIX	TRUE	FALSE	FALSE
CCR9	hgnc:1610	CCR9	ChEMBL	33	inhibitor	39.38075342677087	VERCIRNON	ncit:C152858	VERCIRNON	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.3029288725136221	VOLINANSERIN	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	other/unknown	1.458546423213736	TEPLIZUMAB	rxcui:2621880	TEPLIZUMAB	TRUE	FALSE	FALSE
IL4R	hgnc:6015	IL4R	ChEMBL	33	inhibitor	8.751278539282415	DUPILUMAB	rxcui:1876376	DUPILUMAB	TRUE	FALSE	FALSE
TRBV7-9	hgnc:12243	TRBV7-9	ChEMBL	33	inhibitor	4.375639269641208	MEDI-500	chembl:CHEMBL2109592	MEDI-500	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	agonist	2.019525817	BALUGRASTIM	ncit:C134828	BALUGRASTIM	FALSE	FALSE	FALSE
TNFRSF10A	hgnc:11904	TNFRSF10A	ChEMBL	33	agonist	15.75230137070834	DULANERMIN	ncit:C1685	DULANERMIN	FALSE	TRUE	TRUE
TPH2	hgnc:20692	TPH2	ChEMBL	33	inhibitor	2.187819634820604	TELOTRISTAT	rxcui:1872382	TELOTRISTAT	TRUE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	ChEMBL	33	inhibitor	0.3125456621172291	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMA5	hgnc:9534	PSMA5	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMB8	hgnc:9545	PSMB8	ChEMBL	33	inhibitor	0.2273059360852575	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMA6	hgnc:9535	PSMA6	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMA1	hgnc:9530	PSMA1	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.5707355569097228	RETASPIMYCIN HYDROCHLORIDE	ncit:C48401	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	TRUE
PSMB6	hgnc:9543	PSMB6	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.6250913242344582	ICRUCUMAB	ncit:C79808	ICRUCUMAB	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	other/unknown	2.282942227638891	LABETUZUMAB	ncit:C2043	LABETUZUMAB	FALSE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	ChEMBL	33	inhibitor	2.019525817	AMG-108	chembl:CHEMBL2109458	AMG-108	FALSE	FALSE	FALSE
CD6	hgnc:1691	CD6	ChEMBL	33	binder	26.25383561784724	ONCOLYSIN CD6	chembl:CHEMBL2109485	ONCOLYSIN CD6	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	modulator	0.1389091831632129	MDX-447	chembl:CHEMBL2109391	MDX-447	FALSE	FALSE	FALSE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	8.751278539282415	QAX-576	chembl:CHEMBL2109465	QAX-576	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	agonist	0.029698909	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR6	hgnc:5301	HTR6	ChEMBL	33	agonist	0.2059124362184098	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	PharmGKB	4/5/24	NULL	0.2386712328895204	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
ADH1B	hgnc:250	ADH1B	ChEMBL	33	inhibitor	2.500365296937833	NITREFAZOLE	ncit:C72626	NITREFAZOLE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMAFLOXACIN HYDROCHLORIDE	rxcui:295217	TEMAFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEMAFLOXACIN HYDROCHLORIDE	rxcui:295217	TEMAFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.029715717	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.018019105	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM4	hgnc:1953	CHRM4	ChEMBL	33	inhibitor	0.062733179	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	ChEMBL	33	binder	2.917092846427472	AHN-12	chembl:CHEMBL2109480	AHN-12	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	binder	1.944728564284981	YTTRIUM Y 90 CAPROMAB PENDETIDE	chembl:CHEMBL2109552	YTTRIUM Y 90 CAPROMAB PENDETIDE	FALSE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	inhibitor	2.917092846427472	ANIFROLUMAB	rxcui:2565265	ANIFROLUMAB	TRUE	FALSE	FALSE
BOTA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GS-CDA1	chembl:CHEMBL2109314	GS-CDA1	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.2083637747448194	ALLYLESTRENOL	rxcui:525	ALLYLESTRENOL	TRUE	FALSE	FALSE
SEPTIN3	hgnc:10750	SEPTIN3	PharmGKB	4/5/24	NULL	1.750255707856483	codeine	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.051885051	BENPERIDOL	rxcui:1373	BENPERIDOL	TRUE	FALSE	FALSE
VKORC1	hgnc:23663	VKORC1	ChEMBL	33	inhibitor	4.200613698855561	ACENOCOUMAROL	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	blocker	0.130291988	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	blocker	0.1881995384791917	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	blocker	0.1693795846312726	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	blocker	0.1693795846312726	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	blocker	0.1881995384791917	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	blocker	0.1058622403945453	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	VABORBACTAM	rxcui:1945213	VABORBACTAM	TRUE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	MEDI-557	chembl:CHEMBL2109566	MEDI-557	FALSE	FALSE	FALSE
TRGV3	hgnc:12288	TRGV3	ChEMBL	33	inhibitor	4.375639269641208	MASLIMOMAB	ncit:C188519	MASLIMOMAB	FALSE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	PharmGKB	4/5/24	NULL	0.4118248724368196	cladribine	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
CD276	hgnc:19137	CD276	ChEMBL	33	binder	10.50153424713889	8H9 131I	chembl:CHEMBL2109310	8H9 131I	FALSE	FALSE	FALSE
PMEL	hgnc:10880	PMEL	ChEMBL	33	modulator	2.187819634820604	IMC-GP100	chembl:CHEMBL2109434	IMC-GP100	FALSE	FALSE	FALSE
GH	hgnc:4261	GH1	ChEMBL	33	inhibitor	8.751278539282415	SEVIRUMAB	ncit:C188584	SEVIRUMAB	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OZENOXACIN	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.056097939	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.052090944	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.048618214	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.050879526	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.053361455	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	ChEMBL	33	blocker	0.085378327	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	blocker	0.128067491	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.2019525816757481	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	PharmGKB	4/5/24	NULL	0.1182605208011137	venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	PharmGKB	4/5/24	NULL	0.1041818873724097	venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.035098711	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
WBP2NL	hgnc:28389	WBP2NL	PharmGKB	4/5/24	NULL	2.019525816757481	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	VEDROPREVIR	ncit:C152843	VEDROPREVIR	FALSE	FALSE	FALSE
REP	NULL	NULL	ChEMBL	33	inhibitor	NULL	GALIDESIVIR	ncit:C172613	GALIDESIVIR	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.2476776945079929	MANIDIPINE 6300	rxcui:29275	MANIDIPINE	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	GEPOTIDACIN	ncit:C170025	GEPOTIDACIN	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM ETZADROXIL	ncit:C87678	SULOPENEM ETZADROXIL	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	PharmGKB	4/5/24	NULL	0.2206204673768676	pioglitazone	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM ETZADROXIL	ncit:C87678	SULOPENEM ETZADROXIL	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM ETZADROXIL	ncit:C87678	SULOPENEM ETZADROXIL	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM ETZADROXIL	ncit:C87678	SULOPENEM ETZADROXIL	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM ETZADROXIL	ncit:C87678	SULOPENEM ETZADROXIL	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM ETZADROXIL	ncit:C87678	SULOPENEM ETZADROXIL	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM ETZADROXIL	ncit:C87678	SULOPENEM ETZADROXIL	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.3697723326457359	ATICAPRANT	ncit:C170144	ATICAPRANT	FALSE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	0.6177373086552295	PRALICIGUAT	ncit:C174906	PRALICIGUAT	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	TENOFOVIR EXALIDEX	ncit:C152560	TENOFOVIR EXALIDEX	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	ROVAFOVIR ETALAFENAMIDE	ncit:C170372	ROVAFOVIR ETALAFENAMIDE	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.078510274	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAZUPENEM	ncit:C84135	RAZUPENEM	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAZUPENEM	ncit:C84135	RAZUPENEM	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAZUPENEM	ncit:C84135	RAZUPENEM	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAZUPENEM	ncit:C84135	RAZUPENEM	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAZUPENEM	ncit:C84135	RAZUPENEM	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAZUPENEM	ncit:C84135	RAZUPENEM	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAZUPENEM	ncit:C84135	RAZUPENEM	FALSE	FALSE	FALSE
WBP2NL	hgnc:28389	WBP2NL	PharmGKB	4/5/24	NULL	2.187819634820604	codeine	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULOPENEM	ncit:C84189	SULOPENEM	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	PRESATOVIR	ncit:C118505	PRESATOVIR	FALSE	FALSE	FALSE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	0.1973972602845657	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
ATP2A2	hgnc:812	ATP2A2	ChEMBL	33	inhibitor	0.5707355569097228	MIPSAGARGIN	ncit:C90554	MIPSAGARGIN	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	RILEMATOVIR	ncit:C165437	RILEMATOVIR	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.1136529680426287	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
GRM2	hgnc:4594	GRM2	ChEMBL	33	positive modulator	7.501095891	JNJ-40411813	drugbank:DB12059	JNJ-40411813	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
LAG3	hgnc:6476	LAG3	ChEMBL	33	inhibitor	0.6563458904461813	RELATLIMAB	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GEPOTIDACIN	ncit:C170025	GEPOTIDACIN	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GEPOTIDACIN	ncit:C170025	GEPOTIDACIN	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	1.250182648468916	ZATOLMILAST	ncit:C175880	ZATOLMILAST	FALSE	FALSE	FALSE
METAP2	hgnc:16672	METAP2	ChEMBL	33	inhibitor	9.845188356692718	BELORANIB	ncit:C90656	BELORANIB	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2917092846427472	GSK-256066	drugbank:DB12137	GSK-256066	FALSE	FALSE	FALSE
SLC25A31	hgnc:25319	SLC25A31	PharmGKB	4/5/24	NULL	2.692701089009974	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.3125456621172291	alfentanil	rxcui:203203	ALFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	MK-0873	drugbank:DB13029	MK-0873	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.6250913242344582	MK-0873	drugbank:DB13029	MK-0873	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.9376369863516875	OGLEMILAST	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
RPL3	hgnc:10332	RPL3	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL24	hgnc:10325	RPL24	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL23	hgnc:10316	RPL23	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.108711535	atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSR1	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSR2	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ICLAPRIM	ncit:C65877	ICLAPRIM	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	ChEMBL	33	agonist	1.544343271638073	1018 ISS	chembl:CHEMBL4297680	1018 ISS	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.5385402178019948	BUNAZOSIN	rxcui:19850	BUNAZOSIN	FALSE	FALSE	FALSE
PNLIP	hgnc:9155	PNLIP	ChEMBL	33	inhibitor	4.375639269641208	CETILISTAT	ncit:C77404	CETILISTAT	FALSE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	ChEMBL	33	inhibitor	5.527123287967842	ASLAN-003	iuphar.ligand:12106	FARUDODSTAT	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.6226206075378794	JNJ-37822681	drugbank:DB12579	JNJ-37822681	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.8899605294185507	ILEPATRIL	ncit:C87731	ILEPATRIL	FALSE	FALSE	FALSE
LPTD	NULL	NULL	ChEMBL	33	inhibitor	NULL	MUREPAVADIN	ncit:C175150	MUREPAVADIN	FALSE	FALSE	FALSE
SEMA4D	hgnc:10732	SEMA4D	ChEMBL	33	inhibitor	8.751278539282415	PEPINEMAB	ncit:C96222	PEPINEMAB	FALSE	FALSE	FALSE
F11	hgnc:3529	F11	ChEMBL	33	negative modulator	2.763561643983921	OSOCIMAB	ncit:C170268	OSOCIMAB	FALSE	FALSE	FALSE
FABI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AFN-1252	drugbank:DB12658	AFN-1252	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.3846715841442821	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	3.500511415712966	AVN-944	drugbank:DB05500	AVN-944	FALSE	FALSE	FALSE
MGLL	hgnc:17038	MGLL	ChEMBL	33	inhibitor	8.751278539282415	ELCUBRAGISTAT	ncit:C148538	ELCUBRAGISTAT	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.2071308530007672	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
DXR	NULL	NULL	ChEMBL	33	inhibitor	NULL	FOSMIDOMYCIN	ncit:C65764	FOSMIDOMYCIN	FALSE	FALSE	FALSE
REVERSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TENOFOVIR EXALIDEX	ncit:C152560	TENOFOVIR EXALIDEX	FALSE	FALSE	FALSE
TRANSCRIPTASE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TENOFOVIR EXALIDEX	ncit:C152560	TENOFOVIR EXALIDEX	FALSE	FALSE	FALSE
ATP1B3	hgnc:806	ATP1B3	ChEMBL	33	inhibitor	0.9723642821424908	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
ATP1A2	hgnc:800	ATP1A2	ChEMBL	33	inhibitor	0.8334550989792778	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
ATP1B1	hgnc:804	ATP1B1	ChEMBL	33	inhibitor	0.3070624048871023	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	ChEMBL	33	agonist	0.4375639269641208	TAPINAROF	rxcui:2602286	TAPINAROF	TRUE	FALSE	FALSE
ATP1A1	hgnc:799	ATP1A1	ChEMBL	33	inhibitor	0.7778914257139926	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.1944728564284981	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.058471794	SHR3680	iuphar.ligand:12798	REZVILUTAMIDE	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	ChEMBL	33	inhibitor	3.500511415712966	M4344	chembl:CHEMBL4650286	M4344	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.037213091	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEBIPENEM PIVOXIL	ncit:C76566	TEBIPENEM PIVOXIL	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEBIPENEM PIVOXIL	ncit:C76566	TEBIPENEM PIVOXIL	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEBIPENEM PIVOXIL	ncit:C76566	TEBIPENEM PIVOXIL	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEBIPENEM PIVOXIL	ncit:C76566	TEBIPENEM PIVOXIL	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEBIPENEM PIVOXIL	ncit:C76566	TEBIPENEM PIVOXIL	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEBIPENEM PIVOXIL	ncit:C76566	TEBIPENEM PIVOXIL	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEBIPENEM PIVOXIL	ncit:C76566	TEBIPENEM PIVOXIL	FALSE	FALSE	FALSE
TFR2	hgnc:11762	TFR2	ChEMBL	33	binder	13.12691780892362	PABINAFUSP ALFA	ncit:C170281	PABINAFUSP ALFA	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.596678082	BUCINDOLOL HYDROCHLORIDE	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	ChEMBL	33	inhibitor	0.3201687270469177	APG-2575	chembl:CHEMBL4650374	APG-2575	FALSE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	modulator	1.381780822	BALCINRENONE	ncit:C188521	BALCINRENONE	FALSE	FALSE	FALSE
PCRV	NULL	NULL	ChEMBL	33	inhibitor	NULL	GREMUBAMAB	ncit:C166690	GREMUBAMAB	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	SOTROVIMAB	rxcui:2550731	SOTROVIMAB	FALSE	FALSE	FALSE
METG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CRS-3123	drugbank:DB12262	CRS-3123	FALSE	FALSE	FALSE
FGA	hgnc:3661	FGA	ChEMBL	33	positive modulator	1.591141552596802	FIBRINOGEN, HUMAN	rxcui:2264108	FIBRINOGEN, HUMAN	TRUE	FALSE	FALSE
IL2RG	hgnc:6010	IL2RG	ChEMBL	33	agonist	1.750255707856483	RECOMBINANT HUMAN INTERLEUKIN-15	ncit:C1545	RECOMBINANT HUMAN INTERLEUKIN-15	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	agonist	1.346350544504987	RECOMBINANT HUMAN INTERLEUKIN-15	ncit:C1545	RECOMBINANT HUMAN INTERLEUKIN-15	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.5585922471882393	DIANICLINE	ncit:C76073	DIANICLINE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	ODRONEXTAMAB	ncit:C119615	ODRONEXTAMAB	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	ODRONEXTAMAB	ncit:C119615	ODRONEXTAMAB	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	DIACETYLMORPHINE	ncit:C424	DIACETYLMORPHINE	TRUE	FALSE	FALSE
REVERSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CENSAVUDINE	ncit:C166942	CENSAVUDINE	FALSE	FALSE	FALSE
TRANSCRIPTASE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CENSAVUDINE	ncit:C166942	CENSAVUDINE	FALSE	FALSE	FALSE
PRKAB2	hgnc:9379	PRKAB2	ChEMBL	33	activator	1.500219178162699	ACADESINE	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	0.6177373086552294	SHR-1316	chembl:CHEMBL4297828	SHR-1316	FALSE	FALSE	FALSE
HIV1	NULL	NULL	ChEMBL	33	inhibitor	NULL	ALBUVIRTIDE	drugbank:DB15166	ALBUVIRTIDE	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	ChEMBL	33	inhibitor	0.3281729452230906	TALETRECTINIB	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
KLH1	NULL	NULL	ChEMBL	33	vaccine	NULL	SVN53-67/M57-KLH PEPTIDE VACCINE	ncit:C95705	SVN53-67/M57-KLH PEPTIDE VACCINE	FALSE	FALSE	FALSE
HMG1	hgnc:4983	HMGB1	ChEMBL	33	inhibitor	0.251232877	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	ChEMBL	33	cleavage	8.751278539282415	TRENIBOTULINUMTOXINE	chembl:CHEMBL4594539	TRENIBOTULINUMTOXINE	FALSE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	ChEMBL	33	cleavage	17.50255707856483	BOTULINUM TOXIN TYPE A	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
ATR	hgnc:882	ATR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.079557078	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.015627283	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1657439117288336	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.272767123	CABOZANTANIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.201952582	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4930297768609811	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.048379304	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
CTLA-4	hgnc:2505	CTLA4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.7001022831425934	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
ESR1	hgnc:3467	ESR1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3271505995993426	ENDOXIFEN	iuphar.ligand:10203	ENDOXIFEN	FALSE	FALSE	TRUE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.064624826	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	COSMIC	4-Sep-20	NULL	NULL	Endocrine therapy	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	COSMIC	4-Sep-20	NULL	0.085796848	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.4930297768609811	IPATASERTIB	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.006267328	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	NITROMIDE	ncit:C72599	NITROMIDE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.003821241	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	CYAZOFAMID	chembl:CHEMBL1863429	CYAZOFAMID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124448	chembl:CHEMBL588501	CHEMBL:CHEMBL588501	FALSE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	DTC	9/2/20	NULL	0.4412409347537352	ANACARDIC ACID	iuphar.ligand:6999	ANACARDIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00402481	E-DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	SPHONDIN	chembl:CHEMBL1452868	SPHONDIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.05814803	S(+)-ISOPROTERENOL-BITARTRATE	chembl:CHEMBL1257092	CHEMBL:CHEMBL1257092	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.1143957978991165	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.42006137	IPRODIONE	chembl:CHEMBL1862887	IPRODIONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	GUANFACINE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.099446347	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	ILEPCIMIDE	ncit:C72810	ILEPCIMIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	TCMDC-125556	chembl:CHEMBL587092	CHEMBL:CHEMBL587092	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	inhibitor	0.048618214	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	2-PYRIDYLCARBOXALDEHYDE ISONICOTINOYLHYDRAZONE	chembl:CHEMBL401362	CHEMBL:CHEMBL401362	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	KETANSERIN TARTRATE	ncit:C2036	KETANSERIN TARTRATE	FALSE	FALSE	FALSE
TNNI3	hgnc:11947	TNNI3	DTC	9/2/20	NULL	0.5707355569097228	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.040766825	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	OCTYL_GALLATE	chembl:CHEMBL277346	OCTYL_GALLATE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007873395	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.008334551	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.1325951293830669	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004698673	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	2.625383561784724	DIPLAMINE B	chembl:CHEMBL513108	DIPLAMINE B	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.063160791	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	TCMDC-125221	chembl:CHEMBL546649	CHEMBL:CHEMBL546649	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	ALDICARB	ncit:C163578	ALDICARB	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011850072	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIID	chembl:CHEMBL1095025	AESCULIOSIDE IIID	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	TCMDC-124278	chembl:CHEMBL534423	CHEMBL:CHEMBL534423	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.068637479	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
IDO1	hgnc:6059	IDO1	DTC	9/2/20	NULL	0.9376369863516875	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	GNF-PF-2335	chembl:CHEMBL601146	CHEMBL:CHEMBL601146	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.011316308	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	ISOFLUPREDONE ACETATE	rxcui:1364586	ISOFLUPREDONE ACETATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.014849455	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CLOFLUCARBAN	ncit:C47457	CLOFLUCARBAN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	GNF-PF-3350	chembl:CHEMBL600747	CHEMBL:CHEMBL600747	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	inhibitor	0.043756393	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.021309932	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.032412143	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.004264756	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005669763	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	PERVILLEINE B	chembl:CHEMBL486059	PERVILLEINE B	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.052090944	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.016621612	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	AGROCLAVINE	chembl:CHEMBL449081	AGROCLAVINE	FALSE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.1093909817410302	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	1.521961485092594	RADICICOL	ncit:C1462	RADICICOL	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	DNDI1417719	chembl:CHEMBL1420370	CHEMBL:CHEMBL1420370	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	DNDI1417697	chembl:CHEMBL1420457	CHEMBL:CHEMBL1420457	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.033148782	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001581175	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.035927247	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.025081286	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.013992717	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
SIRT2	hgnc:10886	SIRT2	DTC	9/2/20	NULL	8.751278539282415	PAULLONE	chembl:CHEMBL430574	PAULLONE	FALSE	FALSE	FALSE
PRSS1	hgnc:9475	PRSS1	DTC	9/2/20	NULL	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1232574442152452	EBASTINE	rxcui:23796	EBASTINE	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	PharmGKB	4/5/24	NULL	0.1372749574789398	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PYRITHIONE SODIUM	rxcui:2464540	PYRITHIONE SODIUM	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.4953553890159858	TCMDC-125150	chembl:CHEMBL534244	CHEMBL:CHEMBL534244	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	RESACTIN A	chembl:CHEMBL509617	RESACTIN A	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.003672122	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	(-)-U-50488	chembl:CHEMBL58033	(-)-U-50488	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PHENYLPYRUVATE	chembl:CHEMBL1162488	PHENYLPYRUVATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	ESOXYBUTYNIN	ncit:C166661	ESOXYBUTYNIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.03409589	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.093763699	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.1151484018326633	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	A-77636	iuphar.ligand:9637	A77636	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.596678082	GNF-PF-3176	chembl:CHEMBL582471	CHEMBL:CHEMBL582471	FALSE	FALSE	FALSE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	0.8204323630577265	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.01349118	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	DNDI1417447	chembl:CHEMBL1307453	CHEMBL:CHEMBL1307453	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.052090944	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.013814173	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	BENZOTHIAZYL DISULFIDE	chembl:CHEMBL508112	BENZOTHIAZYL DISULFIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.009205412	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.079557078	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001844705	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
EPHB4	hgnc:3395	EPHB4	TALC	12-May-16	inhibitor	5.469549087051511	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123585	chembl:CHEMBL586962	CHEMBL:CHEMBL586962	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	DNDI1417264	chembl:CHEMBL1467200	CHEMBL:CHEMBL1467200	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	GLISOFLAVONE	chembl:CHEMBL1223641	GLISOFLAVONE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.018799739	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	TRACAZOLATE	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1861974157294131	TCMDC-125785	chembl:CHEMBL588525	CHEMBL:CHEMBL588525	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002459606	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	inhibitor	0.8290684931951763	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
EEF1A1	hgnc:3189	EEF1A1	DTC	9/2/20	NULL	52.50767123569449	SPARSOMYCIN	ncit:C152413	SPARSOMYCIN	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.027177884	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.024008995	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001225383	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016273039	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.00741215	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1630673019742065	BENZO[B]FLUORANTHENE	chembl:CHEMBL1337502	BENZO[B]FLUORANTHENE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	inhibitor	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.065799087	MURAGLITAZAR	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	NSC-98938	chembl:CHEMBL1939691	CHEMBL:CHEMBL1939691	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	(S)-THIORPHAN	drugbank:DB08626	THIORPHAN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	TCMDC-125221	chembl:CHEMBL546649	CHEMBL:CHEMBL546649	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.023110771	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.1666910197958555	TALIPEXOLE HYDROCHLORIDE	chembl:CHEMBL1504869	TALIPEXOLE HYDROCHLORIDE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.009244308	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	TALC	12-May-16	inhibitor	0.3365876361262467	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.01160647	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.020351811	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008279355	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	DESOXIMETASONE	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	GNF-PF-1319	chembl:CHEMBL235891	CHEMBL:CHEMBL235891	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.065799087	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.073089743	FLUOXYMESTERONE	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.014369915	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.064824285	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	DTC	9/2/20	NULL	2.500365296937833	BENZYLPENICILLIN	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.012573676	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
HTR6	hgnc:5301	HTR6	DTC	9/2/20	NULL	8.751278539282417	SB-742457	ncit:C166572	INTEPIRDINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	4'-DEMETHYLEPIPODOPHYLLOTOXIN	chembl:CHEMBL31929	4'-DEMETHYLEPIPODOPHYLLOTOXIN	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.2778183663264259	CHR-3996	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
EP300	hgnc:3373	EP300	DTC	9/2/20	NULL	5.834185692854944	DIETHYL-2-DODECYLIDENEMALONATE	chembl:CHEMBL1797708	CHEMBL:CHEMBL1797708	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	E927A	chembl:CHEMBL28517	E927A	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.022439176	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009875432	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.1902451856365742	FLUOXASTROBIN	chembl:CHEMBL1902591	FLUOXASTROBIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	1,2-DINITRO-BENZENE	chembl:CHEMBL168075	CHEMBL:CHEMBL168075	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	ALPRENOLOL HYDROCHLORIDE	rxcui:81947	ALPRENOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.2201579506737715	CHR-3996	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
TRPV3	hgnc:18084	TRPV3	DTC	9/2/20	NULL	11.66837138570988	NSC-677436	chembl:CHEMBL120580	CHEMBL:CHEMBL120580	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	GNF-PF-2947	chembl:CHEMBL581677	CHEMBL:CHEMBL581677	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.025147352	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	TCMDC-124479	chembl:CHEMBL587259	CHEMBL:CHEMBL587259	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.5303805175322676	TCMDC-123769	chembl:CHEMBL534353	CHEMBL:CHEMBL534353	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	TALC	12-May-16	inhibitor	0.3621218705909965	ALVESPIMYCIN	ncit:C38142	ALVESPIMYCIN	FALSE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.003750548	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.00789589	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.008651783	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.039899446	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2371620200347538	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.038131933	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2701011894840252	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
XPO1	hgnc:12825	XPO1	DTC	9/2/20	NULL	5.834185692854944	OSTHOLE	iuphar.ligand:10302	OSTHOLE	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1060761035064535	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	TALC	12-May-16	antisense oligonucleotide	0.6908904109959803	ISIS 2503	drugbank:DB16181	ISIS 2503	FALSE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	LORNOXICAM	rxcui:20890	LORNOXICAM	TRUE	FALSE	FALSE
RCE1	hgnc:13721	RCE1	DTC	9/2/20	NULL	2.500365296937833	NSC-37136	chembl:CHEMBL1370674	CHEMBL:CHEMBL1370674	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006756874	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.01045553	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	DTC	9/2/20	NULL	1.640864726115453	BISINDOLYLMALEIMIDE IX	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008740353	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	GNF-PF-2335	chembl:CHEMBL601146	CHEMBL:CHEMBL601146	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	ARASERTACONAZOLE	ncit:C79926	ARASERTACONAZOLE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.030386384	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1023541349623674	(S)-PROMETHAZINE	chembl:CHEMBL251904	(S)-PROMETHAZINE	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	2.500365296937833	GERONTOXANTHONE A	chembl:CHEMBL517514	GERONTOXANTHONE A	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.011668371	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.008374429	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.070860555	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00073208	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	NSC-407228	chembl:CHEMBL74852	CHEMBL:CHEMBL74852	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004252322	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	SJ000024939	chembl:CHEMBL590691	CHEMBL:CHEMBL590691	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	FENCLONINE	ncit:C81112	FENCLONINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	NSC-172614	chembl:CHEMBL1317506	CHEMBL:CHEMBL1317506	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1019566431761058	ALAZANINE	chembl:CHEMBL578063	ALAZANINE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.027135747	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.284980577	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
MARK1	hgnc:6896	MARK1	DTC	9/2/20	inhibitor	1.312691780892362	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	CID 695758	chembl:CHEMBL260028	CHEMBL:CHEMBL260028	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	BIOALLETHRIN S-CYCLOPENTENYL ISOMER	chembl:CHEMBL1887350	BIOALLETHRIN S-CYCLOPENTENYL ISOMER	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.034184682	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.002170456	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.069454592	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	NITROMIDE	ncit:C72599	NITROMIDE	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.2938862196027677	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.013890918	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1591141552596802	NSC-3323	chembl:CHEMBL1270169	CHEMBL:CHEMBL1270169	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	GBR-12935	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.112919723	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
PRMT1	hgnc:5187	PRMT1	DTC	9/2/20	NULL	13.12691780892362	STILBAMIDINE	ncit:C200720	STILBAMIDINE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.1232574442152452	DL-CATECHIN TRIHYDRATE	chembl:CHEMBL1172228	CHEMBL:CHEMBL1172228	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.039420174	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.067231333	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NSC-747264	chembl:CHEMBL593110	CHEMBL:CHEMBL593110	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.6731752722524935	ROBUSTIC ACID	chembl:CHEMBL400777	ROBUSTIC ACID	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	AMINOPURVALANOL	iuphar.ligand:5927	AMINOPURVALANOL A	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	CORYNANTHEINE	iuphar.ligand:5345	CORYNANTHINE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.059667808	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	4,4'-DIMETHOXYDALBERGIONE	chembl:CHEMBL1436980	4,4'-DIMETHOXYDALBERGIONE	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.005483257	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	DICHLON	chembl:CHEMBL318782	DICHLON	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	E927A	chembl:CHEMBL28517	E927A	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	PYRIMETHAMINE	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV001049	chembl:CHEMBL589946	CHEMBL:CHEMBL589946	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ANETHOLTRITHION	rxcui:820	ANETHOLE TRITHIONE	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	DTC	9/2/20	NULL	3.424413341458336	SSR180711	chembl:CHEMBL559478	SSR180711	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004540615	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	AROMATICIN	chembl:CHEMBL494255	AROMATICIN	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2075402025126264	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	OSTHOLE	iuphar.ligand:10302	OSTHOLE	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1801292323694494	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	GNF-PF-3201	chembl:CHEMBL581872	CHEMBL:CHEMBL581872	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.029170928	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	TALC	12-May-16	inhibitor	0.1363835616511545	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01256465	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	SJ000201788	chembl:CHEMBL602923	CHEMBL:CHEMBL602923	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	DTC	9/2/20	NULL	0.2430910705356226	NSC-675972	chembl:CHEMBL1379243	CHEMBL:CHEMBL1379243	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	NSC-3323	chembl:CHEMBL1270169	CHEMBL:CHEMBL1270169	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009320613	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SJ000114950	chembl:CHEMBL606456	CHEMBL:CHEMBL606456	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011850072	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.016605842	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	FORMESTANE	rxcui:15070	FORMESTANE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.013964806	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	QUIPAZINE	ncit:C61919	QUIPAZINE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.010512046	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1419126249613365	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
PSMA1	hgnc:9530	PSMA1	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.023016221	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
PSMA2	hgnc:9531	PSMA2	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.011637338	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
TEK	hgnc:11724	TEK	TALC	12-May-16	inhibitor	0.3977853881492008	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PSMA8	hgnc:22985	PSMA8	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	DEXPROPRANOLOL	ncit:C77944	DEXPROPRANOLOL	FALSE	FALSE	FALSE
PSMD3	hgnc:9560	PSMD3	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	FURAZOLIDONE	rxcui:4601	FURAZOLIDONE	TRUE	FALSE	FALSE
TPPP	hgnc:24164	TPPP	TALC	12-May-16	NULL	52.50767123569449	BNC105P	ncit:C88338	VASCULAR DISRUPTING AGENT BNC105P	FALSE	FALSE	TRUE
PSMC2	hgnc:9548	PSMC2	DTC	9/2/20	NULL	0.5087952639117684	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	TALC	12-May-16	inhibitor	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
SHFM1	hgnc:10845	SEM1	DTC	9/2/20	NULL	0.3663325900164732	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	TALC	12-May-16	inhibitor	2.072671233	LY2603618	ncit:C81937	RABUSERTIB	FALSE	FALSE	TRUE
PSMD2	hgnc:9559	PSMD2	DTC	9/2/20	NULL	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD1	hgnc:9554	PSMD1	DTC	9/2/20	NULL	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD13	hgnc:9558	PSMD13	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.032858367	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	LORACARBEF HYDRATE	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	TALC	12-May-16	inhibitor	0.022949157	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	PIRIQUALONE	ncit:C74139	PIRIQUALONE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009144492	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.036413087	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PYRITHIONE SODIUM	rxcui:2464540	PYRITHIONE SODIUM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	(S)-NOMIFENSINE	chembl:CHEMBL51697	CHEMBL:CHEMBL51697	FALSE	FALSE	FALSE
KLF5	hgnc:6349	KLF5	DTC	9/2/20	NULL	0.7292732116068681	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
IDE	hgnc:5381	IDE	DTC	9/2/20	NULL	10.50153424713889	BIOTIN	rxcui:1588	BIOTIN	TRUE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.252440727	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.2243917574174978	XR-9544	chembl:CHEMBL444075	CHEMBL:CHEMBL444075	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.6019397937072561	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	1.479089330582943	EUPALININ A	chembl:CHEMBL258867	EUPALININ A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	TCMDC-123762	chembl:CHEMBL547483	CHEMBL:CHEMBL547483	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	TELENZEPINE	ncit:C75285	TELENZEPINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1810609352954982	(R)-MELPHALAN	chembl:CHEMBL250892	(R)-MELPHALAN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-4746	chembl:CHEMBL584868	CHEMBL:CHEMBL584868	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	DIBUCAINE HYDROCHLORIDE	rxcui:235402	DIBUCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	antibody	0.305277158	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.1271372184883643	SJ000001592	chembl:CHEMBL591834	CHEMBL:CHEMBL591834	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.1591141552596803	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.2465148884304905	HYDROXYSTILBAMIDINE	ncit:C65870	HYDROXYSTILBAMIDINE	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.044498026	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.069454592	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	4,4'-THIODIANILINE	chembl:CHEMBL348856	4,4'-THIODIANILINE	FALSE	FALSE	FALSE
ADRBK1	hgnc:289	GRK2	DTC	9/2/20	NULL	1.093909817410302	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	QUINOXALINE-2-CARBOXYLIC ACID	chembl:CHEMBL151797	CHEMBL:CHEMBL151797	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	TALC	12-May-16	inhibitor	2.341819737097098	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	SJ000044417	chembl:CHEMBL609438	CHEMBL:CHEMBL609438	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	FLUOCINONIDE	rxcui:4462	FLUOCINONIDE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.3684748858645227	KAEMPFERIDE	chembl:CHEMBL40919	KAEMPFERIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	CLOBETASOL	rxcui:2590	CLOBETASOL	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	PLUKENETIONE A	chembl:CHEMBL485750	PLUKENETIONE A	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	2.333674277141977	TARANABANT	ncit:C81420	TARANABANT	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ALLANTOIN	rxcui:508	ALLANTOIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004458114	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	E-FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	PSORALEN	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CHLOROETHYLCLONIDINE	chembl:CHEMBL326967	CHLOROETHYLCLONIDINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	NSC-1010	chembl:CHEMBL1688556	CHEMBL:CHEMBL1688556	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	SEPIAPTERIN	ncit:C188559	SEPIAPTERIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	A-315456	chembl:CHEMBL362863	CHEMBL:CHEMBL362863	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	GNF-PF-4085	chembl:CHEMBL528181	CHEMBL:CHEMBL528181	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.1286952726365061	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003483789	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	L-THREO-BENZYLOXY ASPARTATE	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
CAMK1D	hgnc:19341	CAMK1D	DTC	9/2/20	NULL	0.069824031	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.053579256	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FENBUCONAZOLE	chembl:CHEMBL1879687	FENBUCONAZOLE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010678802	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	DNDI1417013	chembl:CHEMBL1452227	CHEMBL:CHEMBL1452227	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.008875536	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1093909817410302	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	SJ000018298	chembl:CHEMBL591412	CHEMBL:CHEMBL591412	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.074426182	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.1002054794574322	FLUOXYMESTERONE	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.2941606231691568	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011049594	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.00961679	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.012233847	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	SJ000071854	chembl:CHEMBL602127	CHEMBL:CHEMBL602127	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	SJ000044417	chembl:CHEMBL609438	CHEMBL:CHEMBL609438	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.065799087	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006324701	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.3500511415712966	SJ000114950	chembl:CHEMBL606456	CHEMBL:CHEMBL606456	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.017380891	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.008804103	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SERTACONAZOLE NITRATE	rxcui:236601	SERTACONAZOLE NITRATE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.004684003	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	chembl:CHEMBL1348974	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	7-METHOXYISOFLAVONE	chembl:CHEMBL563919	CHEMBL:CHEMBL563919	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.046549354	NAFTOPIDIL	ncit:C72927	NAFTOPIDIL	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.049723174	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
PRKCB	hgnc:9395	PRKCB	DTC	9/2/20	NULL	0.8204323630577265	BISINDOLYLMALEIMIDE IX	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	DNDI1417773	chembl:CHEMBL1379900	CHEMBL:CHEMBL1379900	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	ROXARSONE	rxcui:1314413	ROXARSONE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	SQ-22536	chembl:CHEMBL64239	CHEMBL:CHEMBL64239	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	DIETHYLTOLUAMIDE	rxcui:3129	DIETHYLTOLUAMIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.045579576	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	NSC-50688	chembl:CHEMBL1456848	CHEMBL:CHEMBL1456848	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GNF-PF-4516	chembl:CHEMBL586029	CHEMBL:CHEMBL586029	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.1000146118775133	AGROCLAVINE	chembl:CHEMBL449081	AGROCLAVINE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.034773292	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	8.078103267029922	HYDROXYFASUDIL	drugbank:DB04707	HYDROXYFASUDIL	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.020296742	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008887554	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GALLAMINE	rxcui:4638	GALLAMINE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	TCMDC-125785	chembl:CHEMBL588525	CHEMBL:CHEMBL588525	FALSE	FALSE	FALSE
STK4	hgnc:11408	STK4	DTC	9/2/20	inhibitor	0.1875273972703375	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.182318303	VX-745	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.030004384	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	SR-59230A	iuphar.ligand:547	SR59230A	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SOBUZOXANE	ncit:C66540	SOBUZOXANE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	AGROCLAVINE	chembl:CHEMBL449081	AGROCLAVINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00731101	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	DTC	9/2/20	NULL	4.375639269641208	EPIBATIDINE	drugbank:DB07720	EPIBATIDINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	CID 94777	chembl:CHEMBL407501	CHEMBL:CHEMBL407501	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	GARDENIN	chembl:CHEMBL77705	GARDENIN	FALSE	FALSE	FALSE
RPS6KA1	hgnc:10430	RPS6KA1	DTC	9/2/20	inhibitor	0.2187819634820604	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.040766825	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.015516451	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	1.458546423213736	CID 27456	iuphar.ligand:9741	CID2745687	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.012137696	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	IMINOSTILBENE	chembl:CHEMBL243596	IMINOSTILBENE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	inhibitor	0.016206071	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	ANAZOLENE	chembl:CHEMBL1555467	ANAZOLENE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001571004	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.037081689	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV666687	chembl:CHEMBL585966	CHEMBL:CHEMBL585966	FALSE	FALSE	FALSE
NTSR1	hgnc:8039	NTSR1	DTC	9/2/20	NULL	1.750255707856483	TCMDC-125587	chembl:CHEMBL532160	CHEMBL:CHEMBL532160	FALSE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	0.3241214273808303	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DEXAMETHASONE SODIUM PHOSPHATE	rxcui:48933	DEXAMETHASONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.00340605	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.2778183663264258	TCMDC-124317	chembl:CHEMBL586937	CHEMBL:CHEMBL586937	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.036770078	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	inhibitor	0.024309107	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.02302968	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	3-METHYLCHOLANTHRENE	chembl:CHEMBL40583	3-METHYLCHOLANTHRENE	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-302042	chembl:CHEMBL1600564	CHEMBL:CHEMBL1600564	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	3.281729452230906	NSC-119910	chembl:CHEMBL487046	CHEMBL:CHEMBL487046	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	GNF-PF-860	chembl:CHEMBL593254	CHEMBL:CHEMBL593254	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.004802238	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	CHLORDANE	iuphar.ligand:2831	CHLORDANE	FALSE	FALSE	FALSE
RPS6KA5	hgnc:10434	RPS6KA5	DTC	9/2/20	NULL	0.06466462	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	TALIPEXOLE HYDROCHLORIDE	chembl:CHEMBL1504869	TALIPEXOLE HYDROCHLORIDE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.2224901323546377	GYKI-52895	chembl:CHEMBL1256984	CHEMBL:CHEMBL1256984	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008103036	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.1093909817410302	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.030176823	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.016005996	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	4-HYDROXYBENZALDEHYDE PHENYLHYDRAZONE	chembl:CHEMBL224032	CHEMBL:CHEMBL224032	FALSE	FALSE	FALSE
GAK	hgnc:4113	GAK	DTC	9/2/20	NULL	1.458546423213736	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1250182648468916	BENZO[B]FLUORANTHENE	chembl:CHEMBL1337502	BENZO[B]FLUORANTHENE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	SB-222200	iuphar.ligand:2131	SB 222200	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.039899446	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ETHYNODIOL DIACETATE	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1136529680426287	A-77636	iuphar.ligand:9637	A77636	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.1835932560688619	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003050289	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.061773731	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.056826484	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	3-MORPHOLINOSYDNONIMINE HCL	chembl:CHEMBL538104	CHEMBL:CHEMBL538104	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	25-HYDROXYCHOLECALCIFEROL	rxcui:1855064	CALCIFEDIOL ANHYDROUS	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.024814589	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	10-(4-PYRIDYL)CAMPTOTHECIN	chembl:CHEMBL1762593	CHEMBL:CHEMBL1762593	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003313623	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.004952619	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
PRSS3	hgnc:9486	PRSS3	DTC	9/2/20	NULL	5.834185692854944	CYANOPEPTOLIN S	chembl:CHEMBL1076838	CYANOPEPTOLIN S	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	ACETALDEHYDE	rxcui:1311137	ACETALDEHYDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	PROADIFEN	ncit:C84107	PROADIFEN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	ZM-336372	iuphar.ligand:9130	ZM336372	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002421494	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	2.019525817	BERKELEYDIONE	chembl:CHEMBL400514	BERKELEYDIONE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	DTC	9/2/20	NULL	0.018699313	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.032412143	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	SEW-03621	chembl:CHEMBL1271059	CHEMBL:CHEMBL1271059	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	ARISTOYUNNOLIN A	chembl:CHEMBL2333541	ARISTOYUNNOLIN A	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.729273212	HYDRASTININE HYDROCHLORIDE	ncit:C90856	HYDRASTININE HYDROCHLORIDE	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	7.501095891	2,4-DIISOBUTYRYL PHLOROGLUCINOL	chembl:CHEMBL6931	CHEMBL:CHEMBL6931	FALSE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.026626608	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.1193356164447602	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ETHYNODIOL DIACETATE	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009579944	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
PSEN1	hgnc:9508	PSEN1	DTC	9/2/20	NULL	2.019525817	LY-411575	chembl:CHEMBL392068	CHEMBL:CHEMBL392068	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	CHLOROGENIC ACID	rxcui:1311387	CHLOROGENIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004252322	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	GNF-PF-3149	chembl:CHEMBL582507	CHEMBL:CHEMBL582507	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	DTC	9/2/20	NULL	0.2000292237550266	KERACYANIN	rxcui:28165	KERACYANIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.033919684	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
ZAP70	hgnc:12858	ZAP70	DTC	9/2/20	NULL	17.50255707856483	TRIDOLGOSIR	ncit:C152742	TRIDOLGOSIR	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002522952	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.026741875	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-299115A	chembl:CHEMBL374453	GSK-299115A	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	GR-103691	chembl:CHEMBL294747	CHEMBL:CHEMBL294747	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.030386384	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.005540537	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002436325	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.010987167	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NPY1R	hgnc:7956	NPY1R	DTC	9/2/20	NULL	0.7501095890813498	TCMDC-125620	chembl:CHEMBL530291	CHEMBL:CHEMBL530291	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ESTRADIOL ENANTHATE	ncit:C76996	ESTRADIOL ENANTHATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	MEPRYLCAINE	ncit:C83931	MEPRYLCAINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.1244257612220248	3,4,5-TRIHYDROXY-BENZOIC ACID PHENETHYL ESTER	chembl:CHEMBL151146	CHEMBL:CHEMBL151146	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	CHALCONE	rxcui:2592960	CHALCONE	FALSE	FALSE	FALSE
FGF22	hgnc:3679	FGF22	DTC	9/2/20	NULL	0.6250913242344582	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	(-)-HERDMANINE I	chembl:CHEMBL2208196	CHEMBL:CHEMBL2208196	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	(-)-DICENTRINE	chembl:CHEMBL478754	CHEMBL:CHEMBL478754	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.031189588	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	GNF-PF-1731	chembl:CHEMBL581251	CHEMBL:CHEMBL581251	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.012585731	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	AZEPANE	chembl:CHEMBL1375444	AZEPANE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.053145416	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.027093742	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005208578	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	DNDI1417234	chembl:CHEMBL2094549	CHEMBL:CHEMBL2094549	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	BIFENAZATE	chembl:CHEMBL1872845	BIFENAZATE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV000570	chembl:CHEMBL590674	CHEMBL:CHEMBL590674	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	inhibitor	0.065634589	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	FERROUS SULFATE	rxcui:24947	FERROUS SULFATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	GNF-PF-3350	chembl:CHEMBL600747	CHEMBL:CHEMBL600747	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	FLAVOKAWAIN A	chembl:CHEMBL243829	FLAVOKAWAIN A	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TOSUFLOXACIN TOSYLATE	ncit:C76234	TOSUFLOXACIN TOSYLATE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	HALOFANTRINE HYDROCHLORIDE	rxcui:58130	HALOFANTRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.017059022	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
CCBL1	hgnc:1564	KYAT1	DTC	9/2/20	NULL	4.375639269641208	TRYPTOPHAN	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.009430257	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.375054795	IMINOSTILBENE	chembl:CHEMBL243596	IMINOSTILBENE	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	VOLVALERENAL D	chembl:CHEMBL1224789	VOLVALERENAL D	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	PIFEXOLE	ncit:C76774	PIFEXOLE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.3125456621172291	MORONIC ACID	chembl:CHEMBL472646	MORONIC ACID	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.00770359	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	DNDI1417447	chembl:CHEMBL1307453	CHEMBL:CHEMBL1307453	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.026227608	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	ENROFLOXACIN	rxcui:24192	ENROFLOXACIN	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.5000730593875666	SPD-128907	chembl:CHEMBL1256778	CHEMBL:CHEMBL1256778	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003906821	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004847011	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-4516	chembl:CHEMBL586029	CHEMBL:CHEMBL586029	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002459606	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.4375639269641209	DELAVIRDINE	rxcui:83816	DELAVIRDINE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	TUBERATOLIDE A	chembl:CHEMBL1668773	TUBERATOLIDE A	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.01160647	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	2-AMINOFLURENE	chembl:CHEMBL84472	CHEMBL:CHEMBL84472	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.089756703	DELAVIRDINE	rxcui:83816	DELAVIRDINE	TRUE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	1.944728564284981	NARINGIN	rxcui:31538	NARINGIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.069454592	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	GNF-PF-3909	chembl:CHEMBL599304	CHEMBL:CHEMBL599304	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.375054795	(-)-DICENTRINE	chembl:CHEMBL478754	CHEMBL:CHEMBL478754	FALSE	FALSE	FALSE
TYR	hgnc:12442	TYR	DTC	9/2/20	NULL	9.546849315580817	ALPHA-THUJAPLICIN	chembl:CHEMBL1275969	ALPHA-THUJAPLICIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002518354	ACAMPROSATE CALCIUM	rxcui:152761	ACAMPROSATE CALCIUM	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.100589408	RO-0282750	chembl:CHEMBL1397270	CHEMBL:CHEMBL1397270	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1223955040459079	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003053304	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.3671865121377238	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.009840268	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.3977853881492006	MEPINDOLOL	rxcui:29518	MEPINDOLOL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.007899454	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	1.419126249613364	RO-4583298	chembl:CHEMBL2203703	CHEMBL:CHEMBL2203703	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.014732792	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
FPR2	hgnc:3827	FPR2	DTC	9/2/20	NULL	4.375639269641208	AG-22	chembl:CHEMBL1290365	CHEMBL:CHEMBL1290365	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	TCMDC-125587	chembl:CHEMBL532160	CHEMBL:CHEMBL532160	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.021805511	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.015193192	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	SJ000262801	chembl:CHEMBL605077	CHEMBL:CHEMBL605077	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.029443554	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1367387271762877	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	NSC-125034	chembl:CHEMBL239439	CHEMBL:CHEMBL239439	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00239313	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003512454	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DICYCLOHEXYLCARBODIIMIDE	chembl:CHEMBL162598	DICYCLOHEXYLCARBODIIMIDE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	DEQUALINIUM	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.1646008502686348	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	AY-9944	chembl:CHEMBL1513392	CHEMBL:CHEMBL1513392	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.000939684	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	GNF-PF-3257	chembl:CHEMBL601768	CHEMBL:CHEMBL601768	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.060353645	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GAMMA-CYHALOTHRIN	chembl:CHEMBL1905223	GAMMA-CYHALOTHRIN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.026253836	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
RPS6KA4	hgnc:10433	RPS6KA4	DTC	9/2/20	inhibitor	0.6563458904461813	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.027929612	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	MADOLIN T	chembl:CHEMBL2333550	MADOLIN T	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	DTC	9/2/20	NULL	1.591141552596803	EOSIN_Y	chembl:CHEMBL1092023	EOSIN_Y	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	THONZONIUM	rxcui:237058	THONZONIUM	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	AROMATICIN	chembl:CHEMBL494255	AROMATICIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	BENZALDEHYDE	rxcui:1314334	BENZALDEHYDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009630901	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
TYR	hgnc:12442	TYR	DTC	9/2/20	NULL	0.3409589041278863	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.031707531	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.014500876	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	ACRISORCIN	rxcui:89729	ACRISORCIN	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	SIB-1757	iuphar.ligand:1431	SIB-1757	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.018860514	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.038049037	IMIPRAMINE HYDROCHLORIDE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	1.050153425	GNF-PF-2873	chembl:CHEMBL602400	CHEMBL:CHEMBL602400	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006978691	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
DUSP3	hgnc:3069	DUSP3	DTC	9/2/20	NULL	1.071585127259071	MESO-2,3-DIMERCAPTOSUCCINIC ACID	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.2282942227638891	TCMDC-125185	chembl:CHEMBL580819	CHEMBL:CHEMBL580819	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	GNF-PF-3201	chembl:CHEMBL581872	CHEMBL:CHEMBL581872	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	EVOXINE	chembl:CHEMBL1416006	EVOXINE	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.020575106	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003405608	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.063331621	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GABRQ	hgnc:14454	GABRQ	DTC	9/2/20	NULL	0.1252170220247087	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	KHRINONE E	chembl:CHEMBL1079959	KHRINONE E	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.02091106	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	AMOROLFINE	rxcui:17804	AMOROLFINE	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.02234369	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	DTC	9/2/20	NULL	0.1535312024435511	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PHENOXYCARB	chembl:CHEMBL15780	PHENOXYCARB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.034727296	MECLIZINE	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000679905	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	DNDI1417353	chembl:CHEMBL1481721	CHEMBL:CHEMBL1481721	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.08334551	QUINPIROLE	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	FLUOROMETHOLONE	rxcui:4491	FLUOROMETHOLONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	MONOBENZONE	rxcui:17145	MONOBENZONE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.008773212	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	LINTITRIPT	ncit:C66017	LINTITRIPT	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	NSC-407228	chembl:CHEMBL74852	CHEMBL:CHEMBL74852	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	PD-146176	iuphar.ligand:11390	PD-146176	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.085796848	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYB5R	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Isosorbide Mononitrate	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
NTRK	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.095642388	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
PROS1	hgnc:9456	PROS1	FDA	10-Apr-24	NULL	2.500365296937833	Lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.1888765152363111	Inotuzumab Ozogamicin	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
BRCA	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
CDK1	hgnc:1722	CDK1	MyCancerGenome	20-Jun-17	inhibitor	0.1544343271638073	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	0.1744440904840348	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	0.3174882446809434	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.4278402841426959	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.1374032518317239	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	MyCancerGenome	20-Jun-17	inhibitor	0.7544205637312429	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	inhibitor	0.4245903334422736	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.3163112725041837	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.1084869240406911	BI847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	MyCancerGenome	20-Jun-17	inhibitor	1.494525746746522	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.4735540335109532	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	inhibitor	0.2476776945079929	BMS-536924	iuphar.ligand:9386	BMS-536924	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.5114383561918295	PD0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.1562728310586145	GDC-0623	drugbank:DB11982	GDC-0623	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.1325951293830669	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.063331621	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.1154014752432846	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.076934317	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.093763699	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.093763699	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.09972967	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.108040476	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.046303061	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.093763699	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.015193192	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.3241214273808303	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.067317527	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.092606122	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.364636606	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.1620607136904151	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1715936968486748	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
RICTOR	hgnc:28611	RICTOR	MyCancerGenome	20-Jun-17	inhibitor	0.3409589041278864	MLN0128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1666910197958555	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5250767123569451	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
HSP90AB2	NULL	NULL	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	NULL	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
HSP90AA2	hgnc:5256	HSP90AA2P	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	7.001022831425932	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.08334551	1058137-23-7	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.201952582	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.049302978	1058137-23-7	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2944355396394084	1058137-23-7	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1657439117288336	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1860654544142257	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.089298761	BAY869766	hemonc:437	REFAMETINIB	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	NULL	CAROTENOIDS	NULL	NULL	NULL	NULL	NULL
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1158257453728555	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.272767123	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.8078103267029924	1096708-71-2	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.012466209	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.2243917574174978	GREEN TEA POLYPHENOLS	ncit:C2694	GREEN TEA EXTRACT	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02804897	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.049864835	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	1.346350544504987	UFT	ncit:C9506	TEGAFUR-URACIL	FALSE	FALSE	FALSE
ALPP	hgnc:439	ALPP	NCI	14-Sep-17	NULL	0.4167275494896388	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.1646008502686348	BUTHIONINE SULFOXIMINE	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.078722146	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.024393808	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1067229090156392	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.04573839	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.021344582	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.2134458180312784	MARIJUANA	ncit:C26659	MARIJUANA	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.4730420832044549	CALCITONIN	rxcui:1311287	CALCITONIN	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.9460841664089098	ETIDRONATE DISODIUM	rxcui:9872	ETIDRONATE DISODIUM	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.091556532	INFLIXIMAB	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.2365210416022274	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.020226376	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.033148782	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
CCKBR	hgnc:1571	CCKBR	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
CEACAM5	hgnc:1817	CEACAM5	NCI	14-Sep-17	NULL	1.141471113819445	CALCIUM GLUCONATE	rxcui:1908	CALCIUM GLUCONATE	TRUE	FALSE	FALSE
CDKN1C	hgnc:1786	CDKN1C	NCI	14-Sep-17	NULL	11.66837138570989	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
CFLAR	hgnc:1876	CFLAR	NCI	14-Sep-17	NULL	0.9376369863516874	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	0.2845944240417046	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.300043836	AMIKACIN	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
CTSC	hgnc:2528	CTSC	NCI	14-Sep-17	NULL	3.750547945	CALCIUM GLUCONATE	rxcui:1908	CALCIUM GLUCONATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.006811217	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.012649403	METOCLOPRAMIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.1770916399180253	HYDRAZINE	ncit:C29097	HYDRAZINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.011068227	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.020834311	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	NCI	14-Sep-17	NULL	0.081030357	ANTIPSYCHOTIC AGENT	ncit:C29710	ANTIPSYCHOTIC AGENT	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	NULL	CAROTENOIDS	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.013411921	CICLOSPORIN	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.093931433	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.028071463	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
DLG4	hgnc:2903	DLG4	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	0.4546118721705151	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.1704794520639431	5-FLUORODEOXYURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	NCI	14-Sep-17	NULL	0.02075402	6-HYDROXYDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.138178082	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
EIF2B1	hgnc:3257	EIF2B1	NCI	14-Sep-17	NULL	1.875273972703374	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	NULL	ENU	NULL	NULL	NULL	NULL	NULL
ERVK2	ncbigene:2087	ERVK2	NCI	14-Sep-17	NULL	0.2885036881082115	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.252440727	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.08780547	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.4953553890159858	IL-8	ncit:C1289	RECOMBINANT INTERLEUKIN-8	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	1.591141552596803	BETA-GLUCAN	ncit:C2678	BETA-GLUCAN	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.053551934	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
GCLM	hgnc:4312	GCLM	NCI	14-Sep-17	NULL	0.384671584	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
GDA	hgnc:4212	GDA	NCI	14-Sep-17	NULL	5.834185692854944	8-AZAGUANINE	ncit:C28788	8-AZAGUANINE	FALSE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.3671865121377238	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.6141248097742047	CONJUGATED ESTROGENS	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
GRM1	hgnc:4593	GRM1	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.4339476961627644	MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.3182283105193606	CEFOTAXIME	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.1767935058440892	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.2187819634820604	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.028850369	DNR	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.021087418	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
IL1A	hgnc:5991	IL1A	NCI	14-Sep-17	NULL	0.5834185692854945	IMMUNOSUPPRESSANT	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	NULL	CAROTENOIDS	NULL	NULL	NULL	NULL	NULL
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.028290771	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1893305453210138	QUININE	rxcui:9071	QUININE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.546954909	PHYTOCHEMICALS	ncit:C28269	PHYTOCHEMICAL	FALSE	FALSE	FALSE
IL5	hgnc:6016	IL5	NCI	14-Sep-17	NULL	0.1422972120208523	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
IRF1	hgnc:6116	IRF1	NCI	14-Sep-17	NULL	4.039051633514962	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.084146909	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.078840347	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
KRT10	hgnc:6413	KRT10	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
LCAT	hgnc:6522	LCAT	NCI	14-Sep-17	NULL	0.7501095890813498	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
MAP2K3	hgnc:6843	MAP2K3	NCI	14-Sep-17	NULL	0.5303805175322677	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.1500219178162699	5&APOS;-DEOXY-5-FLUOROURIDINE	ncit:C978	DOXIFLURIDINE	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.1121958787087489	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.1100789753368857	IMMUNOSUPPRESSANT	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	NULL	ENU	NULL	NULL	NULL	NULL	NULL
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.3535870116881784	ANTICARCINOGENIC	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.7955707762984014	MAFOSFAMIDE	ncit:C1150	MAFOSFAMIDE	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	NULL	GRANULOCYTE COLONY-STIMULATING FACTOR	NULL	NULL	NULL	NULL	NULL
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1521961485092594	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	NULL	DAB	NULL	NULL	NULL	NULL	NULL
MYB	hgnc:7545	MYB	NCI	14-Sep-17	NULL	0.3804903712731485	12-O-TETRADECANOYLPHORBOL-13-ACETATE	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.003147942	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.01573971	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.054581779	ANTIDEPRESSANTS	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	0.4339476961627644	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
PAX2	hgnc:8616	PAX2	NCI	14-Sep-17	NULL	0.5933070196123672	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.5000730593875667	PROTEIN KINASE INHIBITOR	ncit:C1404	PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1785975212098452	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	1.250182648468916	FAT EMULSION	ncit:C2575	FAT EMULSION	FALSE	FALSE	FALSE
PMP22	hgnc:9118	PMP22	NCI	14-Sep-17	NULL	0.8899605294185507	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PRDX1	hgnc:9352	PRDX1	NCI	14-Sep-17	NULL	0.8334550989792776	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
PXN	hgnc:9718	PXN	NCI	14-Sep-17	NULL	0.7955707762984016	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	1.166837138570989	PROTEIN KINASE INHIBITOR	ncit:C1404	PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.1440539677248134	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.014247096	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	0.7001022831425934	RECOMBINANT HUMAN GROWTH HORMONE	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.2308029504865691	GLIPIZIDE	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1468746048550895	BSO	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.040390516	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.2282942227638891	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	1.166837138570988	CALCITONIN	rxcui:1311287	CALCITONIN	TRUE	FALSE	FALSE
SOCS3	hgnc:19391	SOCS3	NCI	14-Sep-17	NULL	0.7955707762984016	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.3043922970185188	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
SYP	hgnc:11506	SYP	NCI	14-Sep-17	NULL	0.760980743	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	NCI	14-Sep-17	NULL	1.215455352678113	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
STAT6	hgnc:11368	STAT6	NCI	14-Sep-17	NULL	0.1750255707856483	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	NCI	14-Sep-17	NULL	3.125456621172291	BIM-23014	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	4.200613699	MINERAL OIL	rxcui:258439	HEAVY MINERAL OIL	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1293292394967844	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
TBX21	hgnc:11599	TBX21	NCI	14-Sep-17	NULL	1.591141552596803	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.2917092846427472	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.1168135066422569	IFN-ALPHA 2	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
TGFBR3	hgnc:11774	TGFBR3	NCI	14-Sep-17	NULL	0.1442518440541057	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.019559572	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
THBD	hgnc:11784	THBD	NCI	14-Sep-17	NULL	3.500511415712967	GINKGO BILOBA	rxcui:236809	GINKGO BILOBA EXTRACT	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.1121958787087489	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
XRCC5	hgnc:12833	XRCC5	NCI	14-Sep-17	NULL	0.4286340509036285	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	OncoKB	23-Jul-20	NULL	0.085796848	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	OncoKB	23-Jul-20	NULL	1.312691780892362	Milademetan Tosylate	ncit:C107384	MILADEMETAN TOSYLATE	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	OncoKB	23-Jul-20	NULL	0.1389091831632129	Poziotinib	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	OncoKB	23-Jul-20	NULL	0.9842513760562132	Ivosidenib	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	OncoKB	23-Jul-20	NULL	0.3070624048871023	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	OncoKB	23-Jul-20	NULL	0.1108075556053025	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	OncoKB	23-Jul-20	NULL	1.322135606654178	Asciminib	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	OncoKB	23-Jul-20	NULL	0.6050266644442165	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
CDA	hgnc:1712	CDA	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
CDA	hgnc:1712	CDA	PharmGKB	4/5/24	NULL	NULL	difluorodeoxyuridine	NULL	NULL	NULL	NULL	NULL
CHRNA3	hgnc:1957	CHRNA3	PharmGKB	4/5/24	NULL	NULL	Opium alkaloids and derivatives	NULL	NULL	NULL	NULL	NULL
CHRNB1	hgnc:1961	CHRNB1	PharmGKB	4/5/24	NULL	0.2625383561784725	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.2053085874318455	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.2263261691193728	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.1881995384791917	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
ABAT	hgnc:23	ABAT	PharmGKB	4/5/24	NULL	0.08470687	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
ABCC9	hgnc:60	ABCC9	PharmGKB	4/5/24	NULL	0.063645662	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCC9	hgnc:60	ABCC9	PharmGKB	4/5/24	NULL	0.1049104320393496	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
SLC12A3	hgnc:10912	SLC12A3	PharmGKB	4/5/24	NULL	0.4861821410712453	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	PharmGKB	4/5/24	NULL	5.000730593875666	dinutuximab	rxcui:1606274	DINUTUXIMAB	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	1.166837138570988	albendazole	rxcui:430	ALBENDAZOLE	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.2500365296937833	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.1483267549030917	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
MME	hgnc:7154	MME	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
CLOCK	hgnc:2082	CLOCK	PharmGKB	4/5/24	NULL	8.078103267029924	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.044763573	fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.040682597	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	PharmGKB	4/5/24	NULL	NULL	Corticosteroids For Systemic Use	NULL	NULL	NULL	NULL	NULL
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.070129236	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.020257589	abrocitinib	rxcui:2591476	ABROCITINIB	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.048618214	fluconazole	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
EXOC4	hgnc:30389	EXOC4	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
HNF4A	hgnc:5024	HNF4A	PharmGKB	4/5/24	NULL	0.079077818	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
HNF4A	hgnc:5024	HNF4A	PharmGKB	4/5/24	NULL	0.3281729452230906	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
UGT2B17	hgnc:12547	UGT2B17	PharmGKB	4/5/24	NULL	0.2386712328895204	vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.2344092465879218	iguratimod	ncit:C65886	IGURATIMOD	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.016408647	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TCF7L2	hgnc:11641	TCF7L2	PharmGKB	4/5/24	NULL	NULL	sulfonamides, urea derivatives	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.030598876	cabazitaxel	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.057574201	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.4375639269641208	tropisetron	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
INS-IGF2	hgnc:33527	INS-IGF2	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.729273212	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
DVL2	hgnc:3086	DVL2	PharmGKB	4/5/24	NULL	1.381780822	afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.172950169	ropinirole	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
MUCL3	hgnc:21666	MUCL3	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
MT-ND1	hgnc:7455	MT-ND1	PharmGKB	4/5/24	NULL	NULL	aminoglycoside antibacterials	NULL	NULL	NULL	NULL	NULL
MAPK11	hgnc:6873	MAPK11	PharmGKB	4/5/24	NULL	0.041872146	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MT-ND1	hgnc:7455	MT-ND1	PharmGKB	4/5/24	NULL	3.938075342677087	neomycin	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	PharmGKB	4/5/24	NULL	4.594421233123269	nutlin-3	drugbank:DB17039	NUTLIN-3	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	NULL	xenobiotics	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.019577804	blonanserin	ncit:C95920	BLONANSERIN	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.1193356164447602	flecainide	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	POSIPHEN	drugbank:DB15317	POSIPHEN	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	1.193356164447602	acebutolol	rxcui:149	ACEBUTOLOL	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.07458476	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	fluoxetine glucuronide	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.007737647	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.0135995	liothyronine	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.074797252	levofloxacin	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.02639903	(R)-methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.016027983	cimetidine	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.049864835	modafinil	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.014024485	astemizole	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
MBOAT1	hgnc:21579	MBOAT1	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
RBFOX3	hgnc:27097	RBFOX3	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
KCNMA1	hgnc:6284	KCNMA1	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
ABO	hgnc:79	ABO	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
ETV6	hgnc:3495	ETV6	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
GABRG2	hgnc:4087	GABRG2	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.043692674	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
PTGER3	hgnc:9595	PTGER3	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
PRKCQ	hgnc:9410	PRKCQ	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13705	hgnc:174	ACVR2B	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	ACE-031	chembl:CHEMBL2108674	RAMATERCEPT	FALSE	FALSE	FALSE
XPNPEP2	hgnc:12823	XPNPEP2	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
CLASP1	hgnc:17088	CLASP1	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	NULL	Ace Inhibitors, Plain	NULL	NULL	NULL	NULL	NULL
NFKB1	hgnc:7794	NFKB1	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.028009071	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	PharmGKB	4/5/24	NULL	0.073694977	flupenthixol	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.3040984820600068	milnacipran	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.033211683	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	NULL	hdl cholesterol	NULL	NULL	NULL	NULL	NULL
PCSK1	hgnc:8743	PCSK1	PharmGKB	4/5/24	NULL	3.281729452230906	setmelanotide	rxcui:2469247	SETMELANOTIDE	TRUE	FALSE	FALSE
POMC	hgnc:9201	POMC	PharmGKB	4/5/24	NULL	6.563458904461812	setmelanotide	rxcui:2469247	SETMELANOTIDE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	NULL	2-hydroxyatorvastatin	NULL	NULL	NULL	NULL	NULL
DHFR	hgnc:2861	DHFR	PharmGKB	4/5/24	NULL	NULL	Multivitamins, Plain	NULL	NULL	NULL	NULL	NULL
CXXC4	hgnc:24593	CXXC4	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.055859225	ACLIDINIUM	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
CD3EAP	hgnc:24219	POLR1G	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
DPYD	hgnc:3012	DPYD	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
TMEM167A	hgnc:28330	TMEM167A	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
APLF	hgnc:28724	APLF	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
DYNC2H1	hgnc:2962	DYNC2H1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
ERCC3	hgnc:3435	ERCC3	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
H19	hgnc:4713	H19	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.2853677784548614	AC430	iuphar.ligand:9177	AC430	FALSE	FALSE	FALSE
SPRY2	hgnc:11270	SPRY2	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
HSPA5	hgnc:5238	HSPA5	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
IGF2	hgnc:5466	IGF2	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	NULL	R-EDDP	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2734774543525755	artemisinin	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
MUTYH	hgnc:7527	MUTYH	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
OSGEP	hgnc:18028	OSGEP	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.1029562181092049	ACLIDINIUM	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
OSMR	hgnc:8507	OSMR	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
PRKCE	hgnc:9401	PRKCE	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
TGFB1	hgnc:11766	TGFB1	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
ATM	hgnc:795	ATM	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
CDK1	hgnc:1722	CDK1	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.054695491	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.064824285	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
SMAD7	hgnc:6773	SMAD7	PharmGKB	4/5/24	NULL	0.4861821410712453	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
TENM4	hgnc:29945	TENM4	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.027244868	vortioxetine	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
XRCC3	hgnc:12830	XRCC3	PharmGKB	4/5/24	NULL	0.2108741816694558	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
XRCC3	hgnc:12830	XRCC3	PharmGKB	4/5/24	NULL	0.4268916360625569	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	0.3043922970185188	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	NULL	Antimycobacterials	NULL	NULL	NULL	NULL	NULL
ATP7A	hgnc:869	ATP7A	PharmGKB	4/5/24	NULL	0.1405827877796372	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
GNA13	hgnc:4381	GNA13	PharmGKB	4/5/24	NULL	1.280674908	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
ITPA	hgnc:6176	ITPA	PharmGKB	4/5/24	NULL	2.812910959055062	interferon alfa-2b, recombinant	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
BDKRB2	hgnc:1030	BDKRB2	PharmGKB	4/5/24	NULL	0.2734774543525755	lisinopril	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
SELE	hgnc:10718	SELE	PharmGKB	4/5/24	NULL	0.2328499833068492	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	5.625821918110125	neomycin	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.023284998	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
CSMD1	hgnc:14026	CSMD1	PharmGKB	4/5/24	NULL	0.2561349816375341	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	NULL	Vitamin B-complex, Incl. Combinations	NULL	NULL	NULL	NULL	NULL
TGFB1	hgnc:11766	TGFB1	PharmGKB	4/5/24	NULL	0.2542744369767287	glatiramer acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.1091635576625665	vinorelbine	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	5.676504998453459	l-methylfolate	ncit:C107240	L-METHYLFOLATE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	4.702860988936115	alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
FMO2	hgnc:3770	FMO2	PharmGKB	4/5/24	NULL	1.207072901969988	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
KCNIP1	hgnc:15521	KCNIP1	PharmGKB	4/5/24	NULL	4.667348554283955	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.3182283105193606	granisetron	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
UNIPROT:O43653	hgnc:9500	PSCA	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	AGS-1C4D4	ncit:C71157	ANTI-PSCA MONOCLONAL ANTIBODY AGS-1C4D4	FALSE	FALSE	FALSE
F2	hgnc:3535	F2	PharmGKB	4/5/24	NULL	0.4605936073306534	lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.138178082	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1086365611772989	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	1.758630137080676	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
TAOK3	hgnc:18133	TAOK3	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
RHBDF2	hgnc:20788	RHBDF2	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
CLCC1	hgnc:29675	CLCC1	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
LKAAEAR1	hgnc:33718	LKAAEAR1	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
GAL	hgnc:4114	GAL	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
IL17A	hgnc:5981	IL17A	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
MCOLN1	hgnc:13356	MCOLN1	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
MUC16	hgnc:15582	MUC16	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.055155117	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
PDE3A	hgnc:8778	PDE3A	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
POM121L2	hgnc:13973	POM121L2	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
TACR3	hgnc:11528	TACR3	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
HNF1A	hgnc:11621	HNF1A	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
UNIPROT:P09917	hgnc:435	ALOX5	TdgClinicalTrial	Jan-14	NULL	0.3860858179095183	BALSALAZIDE	rxcui:18747	BALSALAZIDE	TRUE	FALSE	FALSE
ZNF165	hgnc:12953	ZNF165	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
IL10	hgnc:5962	IL10	PharmGKB	4/5/24	NULL	0.1842374429322613	sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.1196756039559988	lidoflazine	rxcui:6390	LIDOFLAZINE	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	NULL	clozapine 5-N-glucuronide	NULL	NULL	NULL	NULL	NULL
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.1442518440541057	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.305277158	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	sulfonamides, urea derivatives	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.018704642	dexlansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	PharmGKB	4/5/24	NULL	0.1179947668217853	aldophosphamide	chembl:CHEMBL1593	ALDOPHOSPHAMIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	11alpha-hydroxytestosterone	NULL	NULL	NULL	NULL	NULL
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	NULL	direct acting antivirals	NULL	NULL	NULL	NULL	NULL
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	NULL	direct acting antivirals	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.004339477	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.002522952	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
ATP7B	hgnc:870	ATP7B	PharmGKB	4/5/24	NULL	0.048083948	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	NULL	tamoxifen-n-glucuronide	NULL	NULL	NULL	NULL	NULL
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	2.100306849	sofosbuvir / velpatasvir	wikidata:Q25110523	SOFOSBUVIR/VELPATASVIR	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	NULL	xenobiotics	NULL	NULL	NULL	NULL	NULL
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.577007376	sotalol	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.1154014752432846	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
RAD18	hgnc:18278	RAD18	PharmGKB	4/5/24	NULL	NULL	clopidogrel thiol metabolite H4	NULL	NULL	NULL	NULL	NULL
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.1282238613814273	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.028850369	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.041214813	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
SLC15A1	hgnc:10920	SLC15A1	PharmGKB	4/5/24	NULL	0.2308029504865692	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	1.346350544504987	aprepitant	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	PharmGKB	4/5/24	NULL	0.063645662	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
IL4R	hgnc:6015	IL4R	PharmGKB	4/5/24	NULL	17.50255707856483	pitrakinra	chembl:CHEMBL2109159	PITRAKINRA	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	NULL	catecholamines	NULL	NULL	NULL	NULL	NULL
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.069454592	goserelin	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.007531221	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	NULL	non-selective monoamine reuptake inhibitors	NULL	NULL	NULL	NULL	NULL
ARRB2	hgnc:712	ARRB2	PharmGKB	4/5/24	NULL	0.1508841127462485	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	PharmGKB	4/5/24	NULL	1.750255707856483	pitavastatin	rxcui:861634	PITAVASTATIN	TRUE	FALSE	FALSE
ANKS1B	hgnc:24600	ANKS1B	PharmGKB	4/5/24	NULL	1.093909817410302	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.1691068316769549	goserelin	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
PICK1	hgnc:9394	PICK1	PharmGKB	4/5/24	NULL	4.375639269641208	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
VAC14	hgnc:25507	VAC14	PharmGKB	4/5/24	NULL	1.265245090016735	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.1640864726115453	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.1790034246671403	vilazodone	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
FTO	hgnc:24678	FTO	PharmGKB	4/5/24	NULL	0.2853677784548614	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.2651902587661338	liothyronine	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.087222045	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
GRID2	hgnc:4576	GRID2	PharmGKB	4/5/24	NULL	NULL	6-hydroxy s-warfarin	NULL	NULL	NULL	NULL	NULL
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	NULL	Drugs used in nicotine dependence	NULL	NULL	NULL	NULL	NULL
MSH5	hgnc:7328	MSH5	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	PharmGKB	4/5/24	NULL	0.009513121	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
PPCDC	hgnc:28107	PPCDC	PharmGKB	4/5/24	NULL	0.2822993077187876	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.4475085616678508	procainamide	rxcui:8700	PROCAINAMIDE	TRUE	FALSE	FALSE
MROH2A	hgnc:27936	MROH2A	PharmGKB	4/5/24	NULL	9.546849315580818	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
GPR98	hgnc:17416	ADGRV1	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
RAD52	hgnc:9824	RAD52	PharmGKB	4/5/24	NULL	0.025942525	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.105015342	BALSALAZIDE	rxcui:18747	BALSALAZIDE	TRUE	FALSE	FALSE
VASP	hgnc:12652	VASP	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
HSD3B2	hgnc:5218	HSD3B2	PharmGKB	4/5/24	NULL	2.187819634820604	cholic acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.4118248724368196	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	TALC	12-May-16	inhibitor	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NR1I3	hgnc:7969	NR1I3	PharmGKB	4/5/24	NULL	0.2206204673768676	(R)-methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.2375912725597036	(R)-methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	vaccine	NULL	RECOMBINANT HUMANEGF-RP64K/MONTANIDE	NULL	NULL	NULL	NULL	NULL
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.1389091831632129	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	NULL	TAK901	NULL	NULL	NULL	NULL	NULL
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.2333674277141978	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.201952582	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	TALC	12-May-16	inhibitor	0.2853677784548614	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
UNIPROT:Q02750	hgnc:6840	MAP2K1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	AZD-8330	drugbank:DB06061	AZD-8330	FALSE	FALSE	FALSE
ITGA5	hgnc:6141	ITGA5	TALC	12-May-16	antibody	1.640864726115453	VITAXIN	ncit:C1800	ETARACIZUMAB	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	NULL	SN-314	NULL	NULL	NULL	NULL	NULL
KIF11	hgnc:6388	KIF11	TALC	12-May-16	inhibitor	3.281729452230906	LY-2523355	chembl:CHEMBL2105661	LITRONESIB	FALSE	FALSE	TRUE
UNIPROT:Q13698	hgnc:1397	CACNA1S	TdgClinicalTrial	Jan-14	NULL	0.1320947704042629	AMLODIPINE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.3333820395917111	AMLODIPINE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
UNIPROT:P08246	hgnc:3309	ELANE	TdgClinicalTrial	Jan-14	NULL	NULL	ALPHA-1 PROTEINASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	1.400204566285186	SOMATROPIN	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
UNIPROT:P20292	hgnc:436	ALOX5AP	TdgClinicalTrial	Jan-14	NULL	NULL	AM-103	NULL	NULL	NULL	NULL	NULL
UNIPROT:P06858	hgnc:6677	LPL	TdgClinicalTrial	Jan-14	NULL	NULL	AMT-011	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04114	hgnc:603	APOB	TdgClinicalTrial	Jan-14	NULL	NULL	TKM-APOB	NULL	NULL	NULL	NULL	NULL
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	0.1312691780892362	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.029581787	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	AT13387	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.3680444245492605	ARZOXIFENE	ncit:C1805	ARZOXIFENE	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.016937958	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.036463661	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
UNIPROT:P15509	hgnc:2435	CSF2RA	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	CAM-3001	ncit:C95788	MAVRILIMUMAB	FALSE	FALSE	FALSE
UNIPROT:Q16568	hgnc:24323	CARTPT	TdgClinicalTrial	Jan-14	NULL	0.5527123287967842	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P31639	hgnc:11037	SLC5A2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	CANAGLIFLOZIN	rxcui:1373458	CANAGLIFLOZIN	TRUE	FALSE	FALSE
UNIPROT:Q14956	hgnc:4462	GPNMB	TdgClinicalTrial	Jan-14	NULL	NULL	MONOMETHYL-AURISTATIN E ADC CONJUGATE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.3017682254924971	BECATECARIN	ncit:C1620	BECATECARIN	FALSE	FALSE	FALSE
UNIPROT:P51686	hgnc:1610	CCR9	TdgClinicalTrial	Jan-14	NULL	39.38075342677087	CCX282	ncit:C152858	VERCIRNON	FALSE	FALSE	FALSE
UNIPROT:P35222	hgnc:2514	CTNNB1	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	CEQ508	drugbank:DB17911	CEQ508	FALSE	FALSE	FALSE
UNIPROT:Q96D31	hgnc:25896	ORAI1	TdgClinicalTrial	Jan-14	NULL	NULL	CM2489	NULL	NULL	NULL	NULL	NULL
UNIPROT:P16109	hgnc:10721	SELP	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	BIMOSIAMOSE	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TdgClinicalTrial	Jan-14	NULL	NULL	CPG 52364	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NR97	hgnc:15632	TLR8	TdgClinicalTrial	Jan-14	NULL	NULL	CPG 52364	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	NULL	CPG 52364	NULL	NULL	NULL	NULL	NULL
UNIPROT:P34998	hgnc:2357	CRHR1	TdgClinicalTrial	Jan-14	NULL	NULL	561679	NULL	NULL	NULL	NULL	NULL
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	BMS-582949	drugbank:DB12696	BMS-582949	FALSE	FALSE	FALSE
UNIPROT:Q9Y5Y4	hgnc:4502	PTGDR2	TdgClinicalTrial	Jan-14	NULL	NULL	CRTH2 RECEPTOR ANTAGONIST	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	CPG 10101	drugbank:DB05530	CPG 10101	FALSE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TdgClinicalTrial	Jan-14	NULL	0.4321619031744403	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P32245	hgnc:6932	MC4R	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	BREMELANOTIDE	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
UNIPROT:P26951	hgnc:6012	IL3RA	TdgClinicalTrial	Jan-14	NULL	NULL	CSL 360	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.054695491	ETILEVODOPA	rxcui:1421444	ETILEVODOPA	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.058471794	EZN-4176	ncit:C96742	ANDROGEN RECEPTOR ANTISENSE OLIGONUCLEOTIDE EZN-4176	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.2822993077187876	FEXOFENADINE	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TdgClinicalTrial	Jan-14	NULL	NULL	FSH-GEX	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.4907258993990139	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
UNIPROT:P32246	hgnc:1602	CCR1	TdgClinicalTrial	Jan-14	NULL	NULL	FX125L	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.6241137025199848	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
UNIPROT:P25024	hgnc:6026	CXCR1	TdgClinicalTrial	Jan-14	NULL	NULL	FX125L	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q92542	hgnc:17091	NCSTN	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	BMS-708163	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
UNIPROT:P25025	hgnc:6027	CXCR2	TdgClinicalTrial	Jan-14	NULL	NULL	FX125L	NULL	NULL	NULL	NULL	NULL
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	NULL	FX125L	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q99250	hgnc:10588	SCN2A	TdgClinicalTrial	Jan-14	NULL	0.151537291	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
UNIPROT:P35346	hgnc:11334	SSTR5	TdgClinicalTrial	Jan-14	NULL	3.125456621172291	LANREOTIDE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
UNIPROT:P31358	hgnc:1804	CD52	TdgClinicalTrial	Jan-14	NULL	70.01022831425932	ALEMTUZUMAB	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TdgClinicalTrial	Jan-14	NULL	0.2586584789935689	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
UNIPROT:O15392	hgnc:593	BIRC5	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	LY2181308	drugbank:DB05141	LY2181308	FALSE	FALSE	TRUE
UNIPROT:P16083	hgnc:7856	NQO2	TdgClinicalTrial	Jan-14	NULL	3.088686543276147	CARICOTAMIDE	ncit:C79915	CARICOTAMIDE	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.4907258993990139	LY-2216684	chembl:CHEMBL2103857	EDIVOXETINE	FALSE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.1544343271638073	DIHYDROERGOTAMINE	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	MAXY-G34	drugbank:DB05718	MAXY-G34	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	NULL	MCD-386	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31785	hgnc:6010	IL2RG	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	INTERLEUKIN 2	chembl:CHEMBL1201438	ALDESLEUKIN	FALSE	FALSE	FALSE
UNIPROT:P47900	hgnc:8539	P2RY1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.01354163	ACETYLSALICYLIC ACID	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:Q71U36	hgnc:20766	TUBA1A	TdgClinicalTrial	Jan-14	NULL	0.1265245090016735	MEBENDAZOLE	rxcui:6672	MEBENDAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.1290114772375786	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.2408608772279564	METHYLNALTREXONE	rxcui:29899	METHYLNALTREXONE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.025942525	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.1037701012563132	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	2.051080907644316	TADALAFIL	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.1446492320542548	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.1801292323694494	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.1164249916534246	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P05113	hgnc:6016	IL5	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	MEPOLIZUMAB	rxcui:1720597	MEPOLIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	3.000438356	METMAB	ncit:C82348	ONARTUZUMAB	FALSE	TRUE	TRUE
UNIPROT:O43193	hgnc:4495	MLNR	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	MITEMCINAL	ncit:C166967	MITEMCINAL	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.091583148	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
UNIPROT:P28074	hgnc:9542	PSMB5	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	MLN-9708	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	NULL	MPC-0920	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08648	hgnc:6141	ITGA5	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
UNIPROT:Q9NNW7	hgnc:18155	TXNRD2	TdgClinicalTrial	Jan-14	NULL	1.875273972703374	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
UNIPROT:Q16881	hgnc:12437	TXNRD1	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.2016939996249468	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:P48061	hgnc:10672	CXCL12	TdgClinicalTrial	Jan-14	NULL	NULL	MYOCELL SDF-1	NULL	NULL	NULL	NULL	NULL
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	CLAZOSENTAN	ncit:C79486	CLAZOSENTAN	FALSE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	NULL	NB-1011	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.078840347	NARATRIPTAN	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.2536602475154323	NERAMEXANE	ncit:C76781	NERAMEXANE	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.6945459158160648	NECITUMUMAB	rxcui:1723738	NECITUMUMAB	TRUE	TRUE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	NGX267	drugbank:DB05152	NGX267	FALSE	FALSE	FALSE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.2027323213733378	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
UNIPROT:P01148	hgnc:4419	GNRH1	TdgClinicalTrial	Jan-14	NULL	NULL	NORELIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	NULL	NU172	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
UNIPROT:P24557	hgnc:11609	TBXAS1	TdgClinicalTrial	Jan-14	NULL	NULL	NV-52	NULL	NULL	NULL	NULL	NULL
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.028413242	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	TIZANIDINE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P25025	hgnc:6027	CXCR2	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	PA-401	chembl:CHEMBL4298068	CANOCTAKIN	FALSE	FALSE	FALSE
UNIPROT:P48039	hgnc:7463	MTNR1A	TdgClinicalTrial	Jan-14	NULL	NULL	PD-6735	NULL	NULL	NULL	NULL	NULL
UNIPROT:P49286	hgnc:7464	MTNR1B	TdgClinicalTrial	Jan-14	NULL	NULL	PD-6735	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.070129236	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	0.041672755	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
UNIPROT:P25942	hgnc:11919	CD40	TdgClinicalTrial	Jan-14	NULL	NULL	PG102	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.3547815624033412	DARIFENACIN	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
UNIPROT:P32926	hgnc:3050	DSG3	TdgClinicalTrial	Jan-14	NULL	NULL	DESMOGLEIN-3	NULL	NULL	NULL	NULL	NULL
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.081092929	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
UNIPROT:Q15303	hgnc:3432	ERBB4	TdgClinicalTrial	Jan-14	NULL	0.7544205637312429	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.08178765	DDP225	chembl:CHEMBL5095232	DDP-225	FALSE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.1022876712383659	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
UNIPROT:P31749	hgnc:391	AKT1	TdgClinicalTrial	Jan-14	NULL	0.443726799	PERIFOSINE	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
UNIPROT:P04035	hgnc:5006	HMGCR	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	PITAVASTATIN	rxcui:861634	PITAVASTATIN	TRUE	FALSE	FALSE
UNIPROT:Q8TDV5	hgnc:19060	GPR119	TdgClinicalTrial	Jan-14	NULL	NULL	PSN821	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11217	hgnc:9726	PYGM	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	PSN357	drugbank:DB05044	PSN357	FALSE	FALSE	FALSE
UNIPROT:P31749	hgnc:391	AKT1	TdgClinicalTrial	Jan-14	NULL	0.4930297768609811	RX-0201	ncit:C88335	ARCHEXIN	FALSE	FALSE	FALSE
UNIPROT:Q9NY47	hgnc:1400	CACNA2D2	TdgClinicalTrial	Jan-14	NULL	0.2812910959055062	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	NULL	SBI-087	NULL	NULL	NULL	NULL	NULL
UNIPROT:P25103	hgnc:11526	TACR1	TdgClinicalTrial	Jan-14	NULL	NULL	HOMSPERA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	SURINABANT	ncit:C87598	SURINABANT	FALSE	FALSE	FALSE
UNIPROT:P02538	hgnc:6443	KRT6A	TdgClinicalTrial	Jan-14	NULL	NULL	TD101	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q00975	hgnc:1389	CACNA1B	TdgClinicalTrial	Jan-14	NULL	0.1230648544586589	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.4579157375205915	TRAFERMIN	ncit:C152708	TRAFERMIN	FALSE	FALSE	FALSE
UNIPROT:P45954	hgnc:91	ACADSB	TdgClinicalTrial	Jan-14	NULL	0.0287871	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
UNIPROT:P80404	hgnc:23	ABAT	TdgClinicalTrial	Jan-14	NULL	0.08470687	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.1842374429322613	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
UNIPROT:Q99460	hgnc:9554	PSMD1	TdgClinicalTrial	Jan-14	NULL	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:Q13698	hgnc:1397	CACNA1S	TdgClinicalTrial	Jan-14	NULL	0.066047385	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P00451	hgnc:3546	F8	TdgClinicalTrial	Jan-14	NULL	NULL	VON WILLEBRAND FACTOR (VWF)/COAGULATION FACTOR VIII COMPLEX	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20292	hgnc:436	ALOX5AP	TdgClinicalTrial	Jan-14	NULL	7.501095891	DG031	drugbank:DB04929	DG031	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.3029288725136221	VOLINANSERIN	ncit:C95220	VOLINANSERIN	FALSE	FALSE	FALSE
UNIPROT:Q9P0M4	hgnc:5983	IL17C	TdgClinicalTrial	Jan-14	NULL	10.50153425	VIDOFLUDIMUS	ncit:C152873	VIDOFLUDIMUS	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.267214612	DESONIDE	rxcui:3254	DESONIDE	TRUE	FALSE	FALSE
UNIPROT:Q92854	hgnc:10732	SEMA4D	TdgClinicalTrial	Jan-14	NULL	NULL	VX15/2503 VACCINE	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9UHC9	hgnc:7898	NPC1L1	TdgClinicalTrial	Jan-14	NULL	NULL	EMZETIBE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35610	hgnc:11177	SOAT1	TdgClinicalTrial	Jan-14	NULL	NULL	EMZETIBE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P36507	hgnc:6842	MAP2K2	TdgClinicalTrial	Jan-14	NULL	0.3409589041278863	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.089501712	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.017295017	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.086551106	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	CINALUKAST	ncit:C96709	CINALUKAST	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.014977128	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.041639708	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.7225826316838693	DEZOCINE	rxcui:22713	DEZOCINE	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.112919723	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P08246	hgnc:3309	ELANE	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	ELAFIN	drugbank:DB05161	ELAFIN	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.2220197515251353	DEXMEDETOMIDINE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	DESOXYCORTICOSTERONE PIVALATE	rxcui:22537	DESOXYCORTICOSTERONE PIVALATE	TRUE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q14432	hgnc:8778	PDE3A	TdgClinicalTrial	Jan-14	NULL	1.591141552596802	ENOXIMONE	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.8950171233357017	ESMOLOL	rxcui:49737	ESMOLOL	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	1.334940794127826	FOSINOPRIL	rxcui:50166	FOSINOPRIL	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.4717670371580817	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P06276	hgnc:983	BCHE	TdgClinicalTrial	Jan-14	NULL	3.938075342677087	HEXAFLURONIUM BROMIDE	rxcui:26826	HEXAFLUORENIUM	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.3663325900164732	GUANABENZ	rxcui:5033	GUANABENZ	TRUE	FALSE	FALSE
UNIPROT:P01350	hgnc:4164	GAST	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	G17DT	ncit:C1692	GASTRIN IMMUNOTOXIN	FALSE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	INTERFERON ALFACON-1	rxcui:59744	INTERFERON ALFACON-1	TRUE	TRUE	TRUE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	0.3394892536790592	INTERFERON ALFA-2A, RECOMBINANT	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.3017682254924971	INTERFERON ALFA-2A, RECOMBINANT	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.3211478363039418	LEVALLORPHAN	rxcui:6370	LEVALLORPHAN	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	2.461297089173179	MENOTROPINS	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.3723948314588262	METHANTHELINE	rxcui:6821	METHANTHELINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.546954909	MEPHENTERMINE	rxcui:6756	MEPHENTERMINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1396480617970598	METHYLSCOPOLAMINE	rxcui:89785	METHSCOPOLAMINE	TRUE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	METOLAZONE	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.085239726	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.072125922	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TdgClinicalTrial	Jan-14	NULL	1.131630845596864	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2907401508067248	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.066577774	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.061737415	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.095399112	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	0.4286340509036286	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.064944553	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.064111931	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TdgClinicalTrial	Jan-14	NULL	2.019525817	GLYCOPEG-GCSF	drugbank:DB06022	GLYCOPEG-GCSF	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.055563673	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.074797252	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.070448575	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	1.666910197958555	PANCURONIUM	rxcui:7883	PANCURONIUM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.07767407	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1704794520639432	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.083257407	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.596678082	TOCAINIDE	rxcui:42359	TOCAINIDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	TOLMETIN	rxcui:10636	TOLMETIN	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.037721028	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:P16233	hgnc:9155	PNLIP	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	GT 389-255	drugbank:DB05894	GT 389-255	FALSE	FALSE	FALSE
UNIPROT:P00519	hgnc:76	ABL1	TEND	1-Aug-11	NULL	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:Q14432	hgnc:8778	PDE3A	TEND	1-Aug-11	NULL	0.6819178082557726	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TEND	1-Aug-11	NULL	0.729273212	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.3182283105193606	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.2019525816757481	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.061340737	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TEND	1-Aug-11	NULL	0.059667808	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:O00220	hgnc:11904	TNFRSF10A	TdgClinicalTrial	Jan-14	NULL	42.00613698855559	MAPATUMUMAB	ncit:C61502	MAPATUMUMAB	FALSE	TRUE	TRUE
UNIPROT:P01589	hgnc:6008	IL2RA	TEND	1-Aug-11	NULL	1.029562181092049	DACLIZUMAB	rxcui:190353	DACLIZUMAB	TRUE	TRUE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.4234489615781814	DESLORATADINE	rxcui:275635	DESLORATADINE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.358239472	DEXTROAMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.059690418	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.2778183663264259	HUMAX-EGFR	chembl:CHEMBL2107861	ZALUTUMUMAB	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2031244535229961	DICYCLOMINE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TEND	1-Aug-11	NULL	1.312691780892362	ECHOTHIOPHATE IODIDE	rxcui:3740	ECHOTHIOPHATE IODIDE	TRUE	FALSE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TEND	1-Aug-11	NULL	1.750255707856483	ABCIXIMAB	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TEND	1-Aug-11	NULL	3.500511415712966	EPTIFIBATIDE	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.2386712328895204	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
UNIPROT:Q13489	hgnc:591	BIRC3	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	HGS1029	ncit:C78484	IAP INHIBITOR HGS1029	FALSE	FALSE	FALSE
UNIPROT:P06239	hgnc:6524	LCK	TEND	1-Aug-11	NULL	0.05348375	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2234368988752957	FESOTERODINE	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	ILOPROST	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
UNIPROT:P06870	hgnc:6357	KLK1	TEND	1-Aug-11	NULL	52.50767123569449	ECALLANTIDE	rxcui:658708	ECALLANTIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.2822993077187876	FEXOFENADINE	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.073089743	FLUOXYMESTERONE	rxcui:4494	FLUOXYMESTERONE	TRUE	FALSE	TRUE
UNIPROT:P00533	hgnc:3236	EGFR	TEND	1-Aug-11	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.157680694	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.039390601	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.080781033	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.3723948314588262	METHANTHELINE	rxcui:6821	METHANTHELINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.7778914257139926	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.053145416	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.061725319	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
UNIPROT:P46098	hgnc:5297	HTR3A	TEND	1-Aug-11	NULL	0.1166837138570989	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.1014640990061729	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.044573575	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	1.036335616	PROPARACAINE	rxcui:34905	PROPARACAINE	TRUE	FALSE	FALSE
UNIPROT:P31213	hgnc:11285	SRD5A2	TEND	1-Aug-11	NULL	13.12691780892362	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TEND	1-Aug-11	NULL	0.3513393859865807	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	MC-3001	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	0.9907107780319716	INSM-18	chembl:CHEMBL3545025	INSM-18	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	BN-DF-037	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	PF-05186462	NULL	NULL	NULL	NULL	NULL
HELODERMIN-PREFERRING VIP RECEPTOR	hgnc:12695	VIPR2	TTD	2020.06.01	NULL	NULL	RG-7103	NULL	NULL	NULL	NULL	NULL
PROTEASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	SRD-441	NULL	NULL	NULL	NULL	NULL
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	1.678633990910949	INCB18424	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
STAPHYLOCOCCUS ELONGATION FACTOR TU	NULL	NULL	TTD	2020.06.01	NULL	NULL	NAI-acne	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	CM-2395	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CM-2395	NULL	NULL	NULL	NULL	NULL
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CM-2395	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	CM-2395	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	NULL	RG-7010	NULL	NULL	NULL	NULL	NULL
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	NULL	BGS-649	NULL	NULL	NULL	NULL	NULL
UNIPROT:P16642	hgnc:11529	EPCAM	TdgClinicalTrial	Jan-14	NULL	6.300920548	ING-1	drugbank:DB05831	ING-1	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-652	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	TGFK09SD-ER	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	AZD1419	NULL	NULL	NULL	NULL	NULL
BETA-GLUCURONIDASE	hgnc:4696	GUSB	TTD	2020.06.01	NULL	NULL	PerioPatch	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAS-120	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
UNIPROT:P78536	hgnc:195	ADAM17	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	INCB7839	drugbank:DB05033	INCB7839	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.051885051	Zicronapine	ncit:C152950	ZICRONAPINE	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	MER-3001	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	NULL	MPL-containing Pollinex allergy desensitization vaccine	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 2 RECEPTOR	hgnc:4325	GLP2R	TTD	2020.06.01	NULL	26.25383561784724	Elsiglutide	ncit:C101131	ELSIGLUTIDE	FALSE	FALSE	FALSE
DELTA-LIKE PROTEIN 4	hgnc:2910	DLL4	TTD	2020.06.01	NULL	10.50153424713889	REGN-421	chembl:CHEMBL2109385	ENOTICUMAB	FALSE	FALSE	FALSE
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	NULL	EV-077	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27930	hgnc:5994	IL1R2	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
ASIALOGLYCOPROTEIN RECEPTOR 1	hgnc:742	ASGR1	TTD	2020.06.01	NULL	NULL	AMG 529	NULL	NULL	NULL	NULL	NULL
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A	hgnc:7943	NPR1	TTD	2020.06.01	NULL	NULL	PL-3994 NPR-A	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.9723642821424906	SAR247799	iuphar.ligand:10938	SAR247799	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.3241214273808302	ATI-2042	ncit:C83563	BUDIODARONE	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.5834185692854944	ATI-2042	ncit:C83563	BUDIODARONE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Estetrol	rxcui:2539031	ESTETROL	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BDB001	ncit:C156395	TLR AGONIST BDB001	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	1.944728564284981	AZD4573	ncit:C153377	CDK9 INHIBITOR AZD4573	FALSE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	INTERFERON ALPHA	chembl:CHEMBL2108506	INTERFERON ALFA	TRUE	FALSE	FALSE
ENZYME UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	BXCL702	NULL	NULL	NULL	NULL	NULL
STAT3 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	C188-9	ncit:C151932	STAT3 INHIBITOR C-188-9	FALSE	FALSE	FALSE
WNT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	CWP232291	ncit:C97663	SAM68 MODULATOR CWP232291	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 5	hgnc:11851	TLR5	TTD	2020.06.01	NULL	35.00511415712966	Entolimod	ncit:C99166	ENTOLIMOD	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	4.565884455277782	GSK1795091	iuphar.ligand:11150	GSK1795091	FALSE	FALSE	FALSE
FGFR4 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	H3B-6527	drugbank:DB15169	H3B-6527	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1790034246671403	KETOROLAC	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
ARGINASE	hgnc:77	ABL2	TTD	2020.06.01	NULL	NULL	INCB01158	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR RXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IRX-5183	drugbank:DB05653	IRX-5183	FALSE	FALSE	FALSE
UNIPROT:P19338	hgnc:7667	NCL	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	IPP-204106	ncit:C103297	NUCLEOLIN ANTAGONIST IPP-204106N	FALSE	FALSE	FALSE
PHOSPHATIDYLINOSITOL-3-PHOSPHATE 5-KINASE	hgnc:23785	PIKFYVE	TTD	2020.06.01	NULL	NULL	LAM-002	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	LTT462	ncit:C126687	RINETERKIB	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE ATR	hgnc:882	ATR	TTD	2020.06.01	NULL	3.500511415712966	M4344	chembl:CHEMBL4650286	M4344	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PRN1371	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 2 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PT2977	rxcui:2567226	BELZUTIFAN	TRUE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	0.8899605294185507	NIS793	ncit:C132250	NISEVOKITUG	FALSE	FALSE	FALSE
UNIPROT:P16615	hgnc:812	ATP2A2	TdgClinicalTrial	Jan-14	NULL	0.5073204950308647	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
TAX TRANSCRIPTIONALLY-ACTIVATED GLYCOPROTEIN 1	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	3.500511415712966	MRNA-2416	ncit:C142137	LIPID NANOPARTICLE ENCAPSULATED OX40L MRNA-2416	FALSE	FALSE	FALSE
UBIQUITIN-ACTIVATING ENZYME	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAK-243	drugbank:DB15013	TAK-243	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	Tractinostat	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRC-253	iuphar.ligand:12709	JNJ-63576253	FALSE	FALSE	FALSE
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	INCB59872	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q03181	hgnc:9235	PPARD	TdgClinicalTrial	Jan-14	NULL	1.184383561707394	KD3010	drugbank:DB05188	KD3010	FALSE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	SEL-24	drugbank:DB18082	SEL-24	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAS-120	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TG02	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.2461297089173179	KETOROLAC	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
DNA SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	acelarin	iuphar.ligand:7389	ACELARIN	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ARQ-087	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	0.1307787577476824	TPX-0005	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.1893305453210138	LURASIDONE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
INTERLEUKIN-9	hgnc:6029	IL9	TTD	2020.06.01	NULL	4.375639269641208	BNZ-1	ncit:C146636	IL-2/9/15 GAMMA CHAIN RECEPTOR INHIBITOR BNZ-1	FALSE	FALSE	FALSE
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ONC201	iuphar.ligand:9978	ONC201	FALSE	FALSE	FALSE
TUBULIN POLYMERIZATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PM184	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAK-659	ncit:C188286	MIVAVOTINIB CITRATE	FALSE	FALSE	FALSE
DOPAMINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ONC201	iuphar.ligand:9978	ONC201	FALSE	FALSE	FALSE
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	0.42006137	VISILIZUMAB	ncit:C2229	VISILIZUMAB	FALSE	FALSE	FALSE
EXPORTIN-1	hgnc:12825	XPO1	TTD	2020.06.01	NULL	NULL	Selinexor oral	NULL	NULL	NULL	NULL	NULL
STAT3-BETA-CATENIN PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	BBI-608	ncit:C96429	NAPABUCASIN	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	THX-TS01	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.693795846312725	OLOPATADINE	rxcui:135391	OLOPATADINE	TRUE	FALSE	FALSE
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	Risankizumab	rxcui:2166040	RISANKIZUMAB	TRUE	FALSE	FALSE
STAPHYLOCOCCUS ENOYL ACP REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Afabicin	ncit:C169766	AFABICIN	FALSE	FALSE	FALSE
LEUKOTRIENE A-4 HYDROLASE	hgnc:6710	LTA4H	TTD	2020.06.01	NULL	5.834185692854944	Acebilustat	ncit:C169757	ACEBILUSTAT	FALSE	FALSE	FALSE
UNIPROT:Q03431	hgnc:9608	PTH1R	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	OSTABOLIN-C	chembl:CHEMBL4802222	OSTABOLIN-C	FALSE	FALSE	FALSE
INTERLEUKIN-31	hgnc:19372	IL31	TTD	2020.06.01	NULL	52.50767123569449	KPL-716	chembl:CHEMBL4594341	VIXARELIMAB	FALSE	FALSE	FALSE
VIRUS REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	BTL-TML-001	NULL	NULL	NULL	NULL	NULL
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clobetasol propionate oral	NULL	NULL	NULL	NULL	NULL
VIRUS REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	CLS003	ncit:C162192	FUROSEMIDE/DIGOXIN TOPICAL GEL CLS003	FALSE	FALSE	FALSE
BACTERIAL PROTEIN SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lefamulin	rxcui:2198944	LEFAMULIN	TRUE	FALSE	FALSE
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	LM-030	drugbank:DB18283	LM-030	FALSE	FALSE	FALSE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
INTERLEUKIN 31 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nemolizumab	ncit:C170211	NEMOLIZUMAB	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE LYASE 1	hgnc:10817	SGPL1	TTD	2020.06.01	NULL	26.25383561784724	LX3305	iuphar.ligand:9851	LX2931	FALSE	FALSE	FALSE
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Omadacycline intravenous	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
MALONDIALDEHYDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Reproxalap	ncit:C152196	REPROXALAP	FALSE	FALSE	FALSE
BETA-KLOTHO	hgnc:15527	KLB	TTD	2020.06.01	NULL	NULL	NGM313	NULL	NULL	NULL	NULL	NULL
UNIPROT:P13612	hgnc:6140	ITGA4	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	R1295	drugbank:DB05122	R1295	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	NULL	NGM313	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	ZYDPLA 1	NULL	NULL	NULL	NULL	NULL
GHRELIN	hgnc:18129	GHRL	TTD	2020.06.01	NULL	1.544343271638073	Relamorelin	ncit:C152174	RELAMORELIN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	NULL	Clonidine topical gel	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	NULL	PF-06648671	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Veltuzumab subcutaneous	NULL	NULL	NULL	NULL	NULL
MUTATED OXALOSUCCINATE DECARBOXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AG-120	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
PARATHYROID HORMONE 1 RECEPTOR	hgnc:9608	PTH1R	TTD	2020.06.01	NULL	1.875273972703375	PCO371	drugbank:DB14946	PCO-371	FALSE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	0.4039051633514961	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	NULL	RNS-60	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	AEB701	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	ABX-0401	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RASV-Sp	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	1.518294108020081	DCC-2618	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
UNIPROT:Q00653	hgnc:7795	NFKB2	TdgClinicalTrial	Jan-14	NULL	0.3547815624033412	THYMOSIN BETA-4	drugbank:DB12003	THYMOSIN BETA-4	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	1.750255707856483	AZD1656	iuphar.ligand:7701	AZD1656	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	1.615620653405984	ALZ-801	chembl:CHEMBL4650301	VALILTRAMIPROSATE	FALSE	FALSE	FALSE
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	17.50255707856483	AZD9056	iuphar.ligand:7826	AZD9056	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	OMS405	chembl:CHEMBL5095027	OMS405	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	Pepticlere	NULL	NULL	NULL	NULL	NULL
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	SER-101	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	RPL-554	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
B7-RELATED PROTEIN 1	hgnc:17087	ICOSLG	TTD	2020.06.01	NULL	NULL	AMG 557	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-824383	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	7.501095891	BMS-830216	drugbank:DB14787	BMS-830216	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR	ncbigene:359995	mCR	TTD	2020.06.01	NULL	NULL	ASP-3291	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	RPL-554	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
MYB MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	LR3001	NULL	NULL	NULL	NULL	NULL
HISTAMINE RECEPTOR	hgnc:5172	HR	TTD	2020.06.01	NULL	NULL	ETS-6218	NULL	NULL	NULL	NULL	NULL
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	NULL	XL-499	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	TGBA01AD	NULL	NULL	NULL	NULL	NULL
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	NULL	TGBA01AD	NULL	NULL	NULL	NULL	NULL
5-HT 7 RECEPTOR	hgnc:5302	HTR7	TTD	2020.06.01	NULL	NULL	ATI-9242	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	ATI-9242	NULL	NULL	NULL	NULL	NULL
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	FPI-01	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US10022354, Example 151	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US10022354, Example 5	NULL	NULL	NULL	NULL	NULL
LEUCYL-CYSTEINYL AMINOPEPTIDASE	hgnc:6656	LNPEP	TTD	2020.06.01	NULL	NULL	US10023583, Example 13	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.760980743	TALMAPIMOD	ncit:C79841	TALMAPIMOD	FALSE	FALSE	FALSE
ANGIOPOIETIN 1 RECEPTOR	hgnc:11724	TEK	TTD	2020.06.01	NULL	0.6563458904461813	Altiratinib	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
ACTIVIN RECEPTOR TYPE IB	hgnc:172	ACVR1B	TTD	2020.06.01	NULL	NULL	US10030004, Compound 33	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US10034861, Example 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US10040779, Example 4	NULL	NULL	NULL	NULL	NULL
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	NULL	KRDULPYOVRWKMA-UHFFFAOYSA-N	NULL	NULL	NULL	NULL	NULL
CYTOMEGALOVIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10071110, Compound cCDV	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31994	hgnc:3618	FCGR2B	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	SM101	chembl:CHEMBL4298105	VALZIFLOCEPT	FALSE	FALSE	FALSE
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10087167, Compound 3003	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	AC1LDDOQ	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US10092575, Example 101	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US10092575, Example 158	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	BDBM50177019	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10149841, Compound 19	NULL	NULL	NULL	NULL	NULL
PROKINETICIN RECEPTOR-1	hgnc:4524	PROKR1	TTD	2020.06.01	NULL	NULL	ZINC19658740	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	BDBM50158755	NULL	NULL	NULL	NULL	NULL
UBIQUITIN-ACTIVATING ENZYME E1	NULL	NULL	TTD	2020.06.01	NULL	NULL	SCHEMBL15198145	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	US8470836, 6	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8481586, 5	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.4280516676822921	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
CASEIN KINASE II ALPHA PRIME	hgnc:2459	CSNK2A2	TTD	2020.06.01	NULL	NULL	US8940736, 7	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	US9006244, E2a	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	US9006244, E2b	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	US9073931, E1	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR-ALPHA	hgnc:7966	NR1H3	TTD	2020.06.01	NULL	NULL	US9073931, E2	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	SNX-5422	drugbank:DB06070	SNX-5422	FALSE	FALSE	FALSE
CASEIN KINASE I ALPHA	hgnc:2451	CSNK1A1	TTD	2020.06.01	NULL	NULL	US9096594, 3	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1117184494376478	SOLIFENACIN	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	JCXGHZCWAHCYGY-UHFFFAOYSA-N	NULL	NULL	NULL	NULL	NULL
DISCOIDIN DOMAIN-CONTAINING RECEPTOR 2	hgnc:2731	DDR2	TTD	2020.06.01	NULL	NULL	US9156852, 1	NULL	NULL	NULL	NULL	NULL
DISCOIDIN DOMAIN-CONTAINING RECEPTOR 2	hgnc:2731	DDR2	TTD	2020.06.01	NULL	NULL	US9156852, 105	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	AC1MOZOL	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	BC11-28	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.3409589041278864	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9181182, 40	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9181182, 47	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9187437, 38	NULL	NULL	NULL	NULL	NULL
PLASMODIUM HYPOXANTHINE-GUANINE PHOSPHORIBOSYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9200020, Table 3, Compound 2B	NULL	NULL	NULL	NULL	NULL
AGGRECANASE-1	hgnc:220	ADAMTS4	TTD	2020.06.01	NULL	NULL	US9206139, 5	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9216972, 94	NULL	NULL	NULL	NULL	NULL
FAP-1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9217012, 10	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	BDBM50061612	NULL	NULL	NULL	NULL	NULL
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.4565884455277783	TC-5619	ncit:C169814	BRADANICLINE	FALSE	FALSE	FALSE
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9346821, B-42	NULL	NULL	NULL	NULL	NULL
PLASMODIUM PLASMEPSIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9353089, 330	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	US9359293, TB	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	BDBM50363773	NULL	NULL	NULL	NULL	NULL
SCN1A MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9694002, 129	NULL	NULL	NULL	NULL	NULL
UNIPROT:P52333	hgnc:6193	JAK3	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	TASOCITINIB	chembl:CHEMBL459769	TASOCITINIB	FALSE	FALSE	FALSE
SRSF PROTEIN KINASE 1	hgnc:11305	SRPK1	TTD	2020.06.01	NULL	NULL	ZINC959121	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8921389, 1	NULL	NULL	NULL	NULL	NULL
CHYMOTRYPSIN-C	hgnc:2523	CTRC	TTD	2020.06.01	NULL	NULL	STK296197	NULL	NULL	NULL	NULL	NULL
CHYMOTRYPSIN-C	hgnc:2523	CTRC	TTD	2020.06.01	NULL	NULL	Z90308237	NULL	NULL	NULL	NULL	NULL
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	NULL	US10053465, 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	6EP	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	BDBM50158703	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US9714230, 12	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	US8933228, Ref 2	NULL	NULL	NULL	NULL	NULL
CYSTATHIONINE GAMMA-LYASE	hgnc:2501	CTH	TTD	2020.06.01	NULL	NULL	AKOS003197197	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	AC1LOJYQ	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
BUB1 MITOTIC CHECKPOINT SERINE/THREONINE KINASE	hgnc:1148	BUB1	TTD	2020.06.01	NULL	NULL	SCHEMBL16322760	NULL	NULL	NULL	NULL	NULL
BUB1 MITOTIC CHECKPOINT SERINE/THREONINE KINASE	hgnc:1148	BUB1	TTD	2020.06.01	NULL	NULL	SCHEMBL16365841	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	NULL	SKF-110679	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	3.500511415712966	Tivantinib	ncit:C62437	TIVANTINIB	FALSE	FALSE	TRUE
PHENYLALANINE HYDROXYLASE	hgnc:8582	PAH	TTD	2020.06.01	NULL	NULL	HepaStem	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR RECEPTOR TYPE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	Drug 2862277	NULL	NULL	NULL	NULL	NULL
OX40L RECEPTOR	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	NULL	Anti-OX40 mab	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.06970816	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
B-RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MLN2480	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASP-015K	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	APD-403	NULL	NULL	NULL	NULL	NULL
FREE FATTY ACID RECEPTOR 2	hgnc:4501	FFAR2	TTD	2020.06.01	NULL	NULL	HL-018	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 21 RECEPTOR	hgnc:6006	IL21R	TTD	2020.06.01	NULL	NULL	Ab-01	NULL	NULL	NULL	NULL	NULL
FACTOR XII MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	methyl 5-[(4-tert-butylbenzoyl)amino]-2H-1,2,4-triazole-3-carboxylate	iuphar.ligand:6553	METHYL 5-[(4-TERT-BUTYLBENZOYL)AMINO]-2H-1,2,4-TRIAZOLE-3-CARBOXYLATE	FALSE	FALSE	FALSE
PROSTATE SPECIFIC ANTIGEN	hgnc:6364	KLK3	TTD	2020.06.01	NULL	NULL	ProstaVac	NULL	NULL	NULL	NULL	NULL
PCSK9 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MPSK3169A	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	DWP-09031	NULL	NULL	NULL	NULL	NULL
PI3-KINASE BETA	hgnc:8976	PIK3CB	TTD	2020.06.01	NULL	0.1389091831632129	PQR309	ncit:C111898	BIMIRALISIB	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	NULL	PEP-223/CoVaccine HT	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-2/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAR-339658	chembl:CHEMBL1743086	VATELIZUMAB	FALSE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	NULL	Factor 8	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	NULL	Plasma derived factor VIII PEGylated liposomal	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	ATM AVI	NULL	NULL	NULL	NULL	NULL
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	NULL	T2c-003	NULL	NULL	NULL	NULL	NULL
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	ZYGK-1	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	Laevo-Bambuterol	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP4	hgnc:9596	PTGER4	TTD	2020.06.01	NULL	NULL	EP4-R antagonist	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	NULL	SPD-556	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	NULL	NSD-788	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	NULL	Dexpirronium	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.046965717	Zolpidem	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	GTU-TB vaccine	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NS3 HELICASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VBY-376	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	GMZ-2	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	Affitope AD-01	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	DAC-060	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	TTP-054	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	Cyt-1010	NULL	NULL	NULL	NULL	NULL
CCR5 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	DdRNAi therapy rHIV7-shl-TAR-CCR5RZ, stem cells	NULL	NULL	NULL	NULL	NULL
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	1.500219178	Metformin glycinate	ncit:C170168	METFORMIN GLYCINATE	FALSE	FALSE	FALSE
UROTENSIN II RECEPTOR	hgnc:4468	UTS2R	TTD	2020.06.01	NULL	NULL	GSK1440115	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	CAF-01	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	TPM-1/Morphine	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	TPM-1/Morphine	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	TPM-1/Morphine	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL ABSORPTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	KT6-971	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS LEUCYL-TRNA SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AN-2718	drugbank:DB12810	AN-2718	FALSE	FALSE	FALSE
BETA-HEMATIN FORMATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Artemisone	ncit:C87431	ARTEMISONE	FALSE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	2.157849503	MIM-D3	chembl:CHEMBL3544981	TAVILERMIDE	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	3.750547945	RO-4995819	chembl:CHEMBL3301593	DECOGLURANT	FALSE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	4.375639269641208	EC-145	ncit:C62525	VINTAFOLIDE	FALSE	FALSE	TRUE
BACTERIAL RIBOSOME	NULL	NULL	TTD	2020.06.01	NULL	NULL	Omadacycline intravenous	NULL	NULL	NULL	NULL	NULL
HEPCIDIN	hgnc:15598	HAMP	TTD	2020.06.01	NULL	NULL	Hepcidin mab	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	CVX 096	NULL	NULL	NULL	NULL	NULL
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	ADV-1002401	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amikacin	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lincomycin	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
VEGFR1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
S-ADENOSYLMETHIONINE DECARBOXYLASE PROENZYME	hgnc:457	AMD1	TTD	2020.06.01	NULL	NULL	ORG 34517/34850	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	5.834185692854944	BIO-1211	iuphar.ligand:6589	BIO1211	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazolidinedione	chembl:CHEMBL85398	THIAZOLIDINEDIONE	FALSE	FALSE	FALSE
STAPHYLOCOCCUS ELONGATION FACTOR TU	NULL	NULL	TTD	2020.06.01	NULL	NULL	GE-1170A	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY 86-5044	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	BAY 86-5044	NULL	NULL	NULL	NULL	NULL
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	NULL	BAY 86-5044	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	NULL	HF-0299	NULL	NULL	NULL	NULL	NULL
BACTERIAL DD-CARBOXYPEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cephalosporin	chembl:CHEMBL1235646	CEPHALOSPORIN	FALSE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	JES-9501	NULL	NULL	NULL	NULL	NULL
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lefradafiban	ncit:C81565	LEFRADAFIBAN	FALSE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NP-2	NULL	NULL	NULL	NULL	NULL
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	R0-93877	NULL	NULL	NULL	NULL	NULL
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	NULL	SB-207266A	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	SoRI-9409	NULL	NULL	NULL	NULL	NULL
BACTERIAL HYDROXYMETHYL-DIHYDROPTERIN PYROPHOSPHOKINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-157695	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.6105543166941221	SARIPIDEM	ncit:C74381	SARIPIDEM	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.1491695205559502	LOMERIZINE	ncit:C66029	LOMERIZINE	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.4234489615781814	LOMERIZINE	ncit:C66029	LOMERIZINE	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	5.250767123569449	Vanadate	chembl:CHEMBL86473	VANADATE	FALSE	FALSE	FALSE
NUCLEAR RECEPTOR UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	FLUASTERONE	ncit:C63639	FLUASTERONE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ampicillin	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.8899605294185507	Enalaprilat	rxcui:1545989	ENALAPRILAT ANHYDROUS	TRUE	FALSE	FALSE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.1108075556053025	STI571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
STEROID 11-BETA-HYDROXYLASE	hgnc:2591	CYP11B1	TTD	2020.06.01	NULL	5.250767123569449	Metyrapone	rxcui:6923	METYRAPONE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydrocodeine	rxcui:23088	DIHYDROCODEINE	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	S-06911	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	ICO-25	NULL	NULL	NULL	NULL	NULL
SYNAPTOSOMAL-ASSOCIATED PROTEIN 25	hgnc:11132	SNAP25	TTD	2020.06.01	NULL	17.50255707856483	Botulinum Toxin Type A	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.046221542	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	NULL	BVT.2733	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	WF-11605	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chlorhexidine	rxcui:20791	CHLORHEXIDINE GLUCONATE	TRUE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	MK-8808	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	SMT-D002	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M2	hgnc:1951	CHRM2	TTD	2020.06.01	NULL	NULL	SMT-D002	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	NULL	SMT-D002	NULL	NULL	NULL	NULL	NULL
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	Gene therapy, IFN-b	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	UCB-35440	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	UCB-35440	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	SULFAMIDE	chembl:CHEMBL355001	SULFAMIDE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sodium pyruvate	rxcui:1358847	SODIUM PYRUVATE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceftizoxime	rxcui:2192	CEFTIZOXIME	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID UPTAKE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tiagabine	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GAP JUNCTION PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	ROTIGAPTIDE	ncit:C152260	ROTIGAPTIDE	FALSE	FALSE	FALSE
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AEOL-10150	drugbank:DB05874	AEOL-10150	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.045791574	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
GLIOMA PATHOGENESIS-RELATED PROTEIN 1	hgnc:17001	GLIPR1	TTD	2020.06.01	NULL	NULL	AdRTVP-1	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GW-695634	chembl:CHEMBL1233182	GW-695634	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	NULL	KB-6806	NULL	NULL	NULL	NULL	NULL
TNF RELATED APOPTOSIS INDUCING LIGAND	hgnc:11925	TNFSF10	TTD	2020.06.01	NULL	17.50255707856483	Ad5-TRAIL	ncit:C116879	RECOMBINANT ADENOVIRUS 5 ENCODING TUMOR NECROSIS FACTOR-RELATED APOPTOSIS-INDUCING LIGAND	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	0.1973972602845657	MELAGATRAN	ncit:C66077	MELAGATRAN	FALSE	FALSE	FALSE
DEHYDROPEPTIDASE I	hgnc:3002	DPEP1	TTD	2020.06.01	NULL	17.50255707856483	Cilastatin	rxcui:2540	CILASTATIN	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	BIM23A760	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	ONO-6126	NULL	NULL	NULL	NULL	NULL
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	NULL	SB-265610	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pinaverium bromide	rxcui:54743	PINAVERIUM BROMIDE	FALSE	FALSE	FALSE
SUBSTANCE-K RECEPTOR	hgnc:11527	TACR2	TTD	2020.06.01	NULL	NULL	SLV-332	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	DTI-015	ncit:C2602	CARMUSTINE IN ETHANOL	FALSE	FALSE	FALSE
LEUKOTRIENE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	0.2386712328895204	METHYLENEDIOXYMETHAMPHETAMINE	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flucytosine	rxcui:4451	FLUCYTOSINE	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Naveglitazar	ncit:C75191	NAVEGLITAZAR	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bacampicillin	rxcui:18687	BACAMPICILLIN	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Balsalazide	rxcui:18747	BALSALAZIDE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lymecycline	rxcui:6513	LYMECYCLINE	FALSE	FALSE	FALSE
EXTRACELLULAR MATRIX RECEPTOR III	hgnc:1681	CD44	TTD	2020.06.01	NULL	NULL	BIWA 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL DEOXY-MANNO-OCTULOSONATE CYTIDYLYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	UX-001	chembl:CHEMBL152452	SIALIC ACID	FALSE	FALSE	FALSE
INFLUENZA NEURAMINIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	UX-001	chembl:CHEMBL152452	SIALIC ACID	FALSE	FALSE	FALSE
NETRIN	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	CERE-120	NULL	NULL	NULL	NULL	NULL
STERYL-SULFATASE	hgnc:11425	STS	TTD	2020.06.01	NULL	NULL	STX-140	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	P2B-001	NULL	NULL	NULL	NULL	NULL
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Plevitrexed (R)-isomer	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cloxacillin	rxcui:2625	CLOXACILLIN	FALSE	FALSE	FALSE
STAPHYLOCOCCUS ENOYL ACP REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CG-400549	drugbank:DB12347	CG-400549	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefotetan	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
CARNITINE O-PALMITOYLTRANSFERASE I	hgnc:2329	CPT1B	TTD	2020.06.01	NULL	0.2206204673768676	Perhexiline	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	0.2734774543525755	Iloprost	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	BIO-306	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1111273465305703	CI-1033	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	11C-6-Me-BTA-1	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	ORG 34517/34850	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	ZD-6126	drugbank:DB11872	ZD-6126	FALSE	FALSE	FALSE
BRAIN-DERIVED NEUROTROPHIC FACTOR	hgnc:1033	BDNF	TTD	2020.06.01	NULL	NULL	PYM-50028	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	CYSTEMUSTINE	ncit:C1167	CYSTEMUSTINE	FALSE	FALSE	FALSE
REGULATORY PROTEIN UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Visilizumab	ncit:C2229	VISILIZUMAB	FALSE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE ENDOTHELIAL	hgnc:7876	NOS3	TTD	2020.06.01	NULL	NULL	MTR105	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.035083077	Nilutamide	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	1.193356164447602	Iodipamide	rxcui:5936	IODIPAMIDE	FALSE	FALSE	FALSE
RIBONUCLEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ranpirnase	ncit:C1183	RANPIRNASE	FALSE	FALSE	FALSE
INTERFERON ALPHA/BETA RECEPTOR 2	hgnc:5433	IFNAR2	TTD	2020.06.01	NULL	NULL	Alfa-interferon	NULL	NULL	NULL	NULL	NULL
HEPATOCYTE GROWTH FACTOR	hgnc:4893	HGF	TTD	2020.06.01	NULL	NULL	VM-202	NULL	NULL	NULL	NULL	NULL
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cethromycin	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefacetrile	ncit:C81037	CEPHACETRILE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefradine	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	ESBA-105	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dapivirine	ncit:C73205	DAPIVIRINE	FALSE	FALSE	FALSE
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrolides	ncit:C261	MACROLIDE ANTIBIOTIC	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Meglitinides	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Procarbazine	rxcui:8702	PROCARBAZINE	TRUE	FALSE	FALSE
LEUTINIZING-HORMONE-RELEASING HORMONE	hgnc:4419	GNRH1	TTD	2020.06.01	NULL	0.3070624048871023	Goserelin	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.8899605294185507	Quinapril	rxcui:35208	QUINAPRIL	TRUE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valganciclovir	rxcui:275891	VALGANCICLOVIR	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC KAINATE 1	hgnc:4579	GRIK1	TTD	2020.06.01	NULL	NULL	NS 1209	NULL	NULL	NULL	NULL	NULL
INTERFERON-ALPHA 5	hgnc:5426	IFNA5	TTD	2020.06.01	NULL	NULL	Interferon alpha 5	NULL	NULL	NULL	NULL	NULL
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	2.838252499226729	Aprepitant	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1376949420516464	Cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
MULTIDRUG RESISTANCE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	BN82451	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	BN82451	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.1884246575443582	Flunitrazepam	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
LIPASE UNSPECIFIC	hgnc:30045	SMG1	TTD	2020.06.01	NULL	NULL	Bisquaternary salt	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	ISF-402	NULL	NULL	NULL	NULL	NULL
GUANYLATE CYCLASE	hgnc:4187	GC	TTD	2020.06.01	NULL	0.2302968036653267	Methylene blue	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	0.6403374540938354	A-425619	iuphar.ligand:4117	A425619	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.5585922471882393	Clidinium	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
DNA REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chlorambucil	rxcui:2346	CHLORAMBUCIL	TRUE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	TRELANSERIN	ncit:C90946	TRELANSERIN	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fosamprenavir	rxcui:358262	FOSAMPRENAVIR	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HER2/neu peptide vaccine	NULL	NULL	NULL	NULL	NULL
UNIPROT:O00254	hgnc:3539	F2RL2	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	VORAPAXAR	rxcui:1537034	VORAPAXAR	TRUE	FALSE	FALSE
T-LYMPHOCYTE ACTIVATION ANTIGEN CD86	NULL	NULL	TTD	2020.06.01	NULL	NULL	Abatacept	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Exeporfinium chloride topical	NULL	NULL	NULL	NULL	NULL
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	0.750109589	Dendritic cell vaccine	ncit:C28310	DENDRITIC CELL VACCINE	FALSE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR ALPHA	hgnc:6008	IL2RA	TTD	2020.06.01	NULL	NULL	CHT-25	NULL	NULL	NULL	NULL	NULL
ERYTHROPOIETIN	hgnc:3415	EPO	TTD	2020.06.01	NULL	NULL	MK-2578	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxeglitazar	ncit:C66259	OXEGLITAZAR	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
UNIPROT:P12931	hgnc:11283	SRC	TdgClinicalTrial	Jan-14	NULL	0.4167275494896389	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE XIV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.082559232	AXL-1717	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
CARBONIC ANHYDRASE XII	hgnc:1371	CA12	TTD	2020.06.01	NULL	0.056826484	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Intravenous minocycline	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-4/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	R411	drugbank:DB05468	R411	FALSE	FALSE	FALSE
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.1618941559168381	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.1959241464018451	AMG 900	ncit:C82349	AURORA KINASE INHIBITOR AMG 900	FALSE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	0.074797252	ABT-229	ncit:C81349	ALEMCINAL	FALSE	FALSE	FALSE
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Epristeride	ncit:C81621	EPRISTERIDE	FALSE	FALSE	FALSE
UNIPROT:P01584	hgnc:5992	IL1B	TdgClinicalTrial	Jan-14	NULL	3.088686543276147	GEVOKIZUMAB	ncit:C97945	GEVOKIZUMAB	FALSE	FALSE	FALSE
TRYPTOPHAN 5-HYDROXYLASE	hgnc:12008	TPH1	TTD	2020.06.01	NULL	NULL	LX-1031	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 2	hgnc:11848	TLR2	TTD	2020.06.01	NULL	NULL	MALP-2S	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 6	hgnc:16711	TLR6	TTD	2020.06.01	NULL	NULL	MALP-2S	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	FPL-62064	NULL	NULL	NULL	NULL	NULL
APOPTOSIS MEDIATING SURFACE ANTIGEN FAS	hgnc:11920	FAS	TTD	2020.06.01	NULL	NULL	APO-010	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-9164	drugbank:DB12115	AZD-9164	FALSE	FALSE	FALSE
UNIPROT:P30939	hgnc:5292	HTR1F	TdgClinicalTrial	Jan-14	NULL	0.9546849315580819	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	tideglusib	ncit:C97364	TIDEGLUSIB	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HER-2 Protein AutoVac	NULL	NULL	NULL	NULL	NULL
ION CHANNEL UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATI-2042	ncit:C83563	BUDIODARONE	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	NKP 608	NULL	NULL	NULL	NULL	NULL
RELAXIN RECEPTOR 1	hgnc:19718	RXFP1	TTD	2020.06.01	NULL	3.750547945	RLX030	chembl:CHEMBL2108358	SERELAXIN	FALSE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	0.8078103267029924	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
COMPLEMENT FACTOR H	hgnc:4883	CFH	TTD	2020.06.01	NULL	NULL	TT-30	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.4861821410712453	BENZTROPINE	rxcui:1424	BENZTROPINE	TRUE	FALSE	FALSE
COMPLEMENT RECEPTOR TYPE 2	hgnc:2336	CR2	TTD	2020.06.01	NULL	NULL	TT-30	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAZ AVI	NULL	NULL	NULL	NULL	NULL
STROMAL CELL-DERIVED FACTOR 1	hgnc:10672	CXCL12	TTD	2020.06.01	NULL	NULL	SDF-1	NULL	NULL	NULL	NULL	NULL
MULTIDRUG RESISTANCE PROTEIN 1	hgnc:40	ABCB1	TTD	2020.06.01	NULL	NULL	W-198	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.041085815	VE-822	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1396480617970598	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	E-1224	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV1.5	hgnc:6224	KCNA5	TTD	2020.06.01	NULL	NULL	XEN-D0101	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	870086 (topical, atopic dermatitis), GlaxoSmithKline	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	0.9001315068976199	Mirabegron	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.099446347	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE MELK	hgnc:16870	MELK	TTD	2020.06.01	NULL	5.250767123569449	OTSSP167	iuphar.ligand:8046	OTSSP167	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-135	chembl:CHEMBL4783446	VX-135	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	BUCLIZINE	rxcui:59636	BUCLIZINE	TRUE	FALSE	FALSE
PROGESTERONE	hgnc:6207	JUP	TTD	2020.06.01	NULL	NULL	BAY 86-5044	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR RECEPTOR TYPE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK1995057	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD4	hgnc:1678	CD4	TTD	2020.06.01	NULL	NULL	LIPO-4	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD8	hgnc:1706	CD8A	TTD	2020.06.01	NULL	NULL	LIPO-4	NULL	NULL	NULL	NULL	NULL
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	1.009762908	AZ-4217	iuphar.ligand:6939	AZ-4217	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.077827576	CABERGOLINE	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.6226206075378794	JNJ-37822681	drugbank:DB12579	JNJ-37822681	FALSE	FALSE	FALSE
PLATELET GLYCOPROTEIN IB ALPHA	hgnc:4439	GP1BA	TTD	2020.06.01	NULL	NULL	ZK-001	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	Intravenous carbamazepine	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.1158257453728555	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-5885	rxcui:1591922	LEDIPASVIR	TRUE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	4.039051633514961	MAXY-G34	drugbank:DB05718	MAXY-G34	FALSE	FALSE	FALSE
DICKKOPF-RELATED PROTEIN 3	hgnc:2893	DKK3	TTD	2020.06.01	NULL	NULL	REIC gene therapy	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-267	rxcui:1597371	OMBITASVIR	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.084689792	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-6620	drugbank:DB15222	GS-6620	FALSE	FALSE	FALSE
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-7655	rxcui:2184137	RELEBACTAM	TRUE	FALSE	FALSE
IDURONATE 2-SULFATASE	hgnc:5389	IDS	TTD	2020.06.01	NULL	NULL	Recombinant human iduronate-2-sulfatase	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	RBP-7000	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dimiracetam	ncit:C79121	DIMIRACETAM	FALSE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	CIPEMASTAT	ncit:C96297	CIPEMASTAT	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	8.751278539282415	LY2605541	chembl:CHEMBL2108569	INSULIN PEGLISPRO	FALSE	FALSE	FALSE
LEUKOTRIENE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PIRODOMAST	ncit:C82230	PIRODOMAST	FALSE	FALSE	FALSE
OXALOSUCCINATE DECARBOXYLASE	hgnc:5382	IDH1	TTD	2020.06.01	NULL	0.9842513760562132	AG-120	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	AMG 595	ncit:C99222	ANTI-EGFRVIII ANTIBODY DRUG CONJUGATE AMG 595	FALSE	FALSE	FALSE
MYELOPEROXIDASE	hgnc:7218	MPO	TTD	2020.06.01	NULL	1.750255707856483	AZD-3241	ncit:C152861	VERDIPERSTAT	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,2,4-triazole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,5-diphenylpyrrolidin-2-one derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,5-diphenylpyrrolidin-2-one derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	4-methyl-4,5-dihydro-1H-pyrazole-3-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 7	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 9	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Azetidine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Azetidine derivative 4	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q08493	hgnc:8782	PDE4C	TdgClinicalTrial	Jan-14	NULL	0.7759754369807069	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diaryl morpholine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diaryl piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Furopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Heterocyclic-substituted 3-alkyl azetidine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Heterocyclic-substituted 3-alkyl azetidine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazolidine-2,4-dione derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	N-phenyl-5-phenyl-pyrazolin-3-yl amide derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	N-phenyl-5-phenyl-pyrazolin-3-yl amide derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	PMID26161824-Compound-68	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 12	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 18	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 35	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.5000730593875666	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 39	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 5	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 53	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 54	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 58	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazoline derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazoline derivative 5	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.3170753093942904	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyridotriazolopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyridotriazolopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 5	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Sulfonylated piperazine derivative 4	NULL	NULL	NULL	NULL	NULL
HGF/MET SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.158793361	DIPHENHYDRAMINE	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
ENDOTHELIN B RECEPTOR	hgnc:3180	EDNRB	TTD	2020.06.01	NULL	2.812910959055062	Macitentan	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.081281225	Cinolazepam	ncit:C77635	CINOLAZEPAM	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	4.375639269641208	Insulin degludec	rxcui:1670007	INSULIN DEGLUDEC	TRUE	FALSE	FALSE
DNA REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ozenoxacin	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
UNIPROT:Q13946	hgnc:8791	PDE7A	TdgClinicalTrial	Jan-14	NULL	3.000438356325399	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS DNA GYRASE A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ozenoxacin	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAFINAMIDE MESYLATE	rxcui:1922449	SAFINAMIDE MESYLATE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sofosbuvir + velpatasvir + voxilaprevir	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sofosbuvir + velpatasvir + voxilaprevir	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS SERINE PROTEASE NS3/4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sofosbuvir + velpatasvir + voxilaprevir	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-14	hgnc:7160	MMP14	TTD	2020.06.01	NULL	NULL	BT-1718	NULL	NULL	NULL	NULL	NULL
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.2206204673768676	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
PSEUDOMONAS LPS-ASSEMBLY PROTEIN LPTD	NULL	NULL	TTD	2020.06.01	NULL	NULL	Murepavadin	ncit:C175150	MUREPAVADIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3A	hgnc:8778	PDE3A	TTD	2020.06.01	NULL	1.591141552596802	Enoximone	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	NULL	Segesterone acetate and ethinyl estradiol vaginal system	NULL	NULL	NULL	NULL	NULL
POTASSIUM	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sodium zirconium cyclosilicate	rxcui:2047628	SODIUM ZIRCONIUM CYCLOSILICATE	TRUE	FALSE	FALSE
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tildrakizumab	rxcui:2053436	TILDRAKIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.076263865	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lacosamide	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	NULL	Lumacaftor + ivacaftor	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.2375912725597036	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL F508 DELETION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lumacaftor + ivacaftor	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	DWJ-208	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.2625383561784725	FENOPROFEN	rxcui:4331	FENOPROFEN	TRUE	FALSE	FALSE
GABA(A) RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAGE-324	NULL	NULL	NULL	NULL	NULL
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1583941817064691	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.1	hgnc:1388	CACNA1A	TTD	2020.06.01	NULL	NULL	XEN007	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BLZ-100	chembl:CHEMBL3990023	TOZULERISTIDE	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	BIZELESIN	ncit:C1472	BIZELESIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	349U85.HCL	NULL	NULL	NULL	NULL	NULL
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	NULL	G-619	NULL	NULL	NULL	NULL	NULL
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	NULL	G-619	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.079197091	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
TROMBOXANE A2 SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazole salicylate	ncit:C65894	IMIDAZOLE SALICYLATE	FALSE	FALSE	FALSE
LIPOXYGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TZI-41078	NULL	NULL	NULL	NULL	NULL
BACTERIAL DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nitrofurantoin	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
INOSITOL 1,4,5-TRISPHOSPHATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nitroprusside	rxcui:7476	NITROPRUSSIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.089501712	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
VASOPRESSIN V1 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Menadione	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P23786	hgnc:2330	CPT2	TdgClinicalTrial	Jan-14	NULL	0.326134604	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	E-6700	NULL	NULL	NULL	NULL	NULL
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	NULL	E-6700	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATEVIRDINE	ncit:C73840	ATEVIRDINE	FALSE	FALSE	FALSE
PITUITARY ADENYLATE CYCLASE-ACTIVATING 38	NULL	NULL	TTD	2020.06.01	NULL	NULL	PACAP38	drugbank:DB17073	PACAP38	FALSE	FALSE	FALSE
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	CYCLOPLATAM	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PTI-202	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PHE-377	NULL	NULL	NULL	NULL	NULL
WNT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	SM-04690	chembl:CHEMBL4297639	LORECIVIVINT	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	NULL	EGT-0001474	NULL	NULL	NULL	NULL	NULL
ENZYME UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	HTI-101	NULL	NULL	NULL	NULL	NULL
UNIPROT:P50416	hgnc:2328	CPT1A	TdgClinicalTrial	Jan-14	NULL	1.154014752432846	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
GLUTAMYL AMINOPEPTIDASE	hgnc:3355	ENPEP	TTD	2020.06.01	NULL	6.563458904461812	QGC-001	drugbank:DB13107	QGC-001	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	NULL	R4996	NULL	NULL	NULL	NULL	NULL
PLACENTA GROWTH FACTOR	hgnc:8893	PGF	TTD	2020.06.01	NULL	NULL	R7334	NULL	NULL	NULL	NULL	NULL
A-RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7304	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
B-RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7304	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7304	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7304	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	T-607	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-V/BETA-6	NULL	NULL	TTD	2020.06.01	NULL	NULL	STX-100	drugbank:DB16334	STX-100	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	PICROTOXIN	rxcui:2539172	PICROTOXIN	FALSE	FALSE	FALSE
MICROTUBULE-ASSOCIATED PROTEIN	hgnc:25228	SGSM3	TTD	2020.06.01	NULL	2.917092846427472	RG7304	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	TOL-3021	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	HPP404	NULL	NULL	NULL	NULL	NULL
AGOUTI-RELATED PROTEIN	hgnc:330	AGRP	TTD	2020.06.01	NULL	NULL	TTP435	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-222	chembl:CHEMBL3039503	LOMIBUVIR	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	ZYOG1	NULL	NULL	NULL	NULL	NULL
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	NULL	BI-135585	NULL	NULL	NULL	NULL	NULL
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	NULL	RG-4929	NULL	NULL	NULL	NULL	NULL
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lu-AA34893	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.4605936073306534	PROCYCLIDINE	rxcui:8718	PROCYCLIDINE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	Lu-AA34893	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1325951293830669	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
T-CELL-SPECIFIC PROTEIN RANTES	hgnc:10632	CCL5	TTD	2020.06.01	NULL	NULL	NI-0701	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR VII	hgnc:3544	F7	TTD	2020.06.01	NULL	NULL	Activated recombinant FVII-albumin fusion protein	NULL	NULL	NULL	NULL	NULL
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	NULL	Activated recombinant FVII-albumin fusion protein	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	PBSVax	NULL	NULL	NULL	NULL	NULL
CONNECTING PEPTIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CBX-129801	chembl:CHEMBL4594533	CBX-129801	FALSE	FALSE	FALSE
ALPHA-MANNOSIDASE	hgnc:6827	MAN2C1	TTD	2020.06.01	NULL	NULL	M-0011	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.16256245	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE BRAIN	hgnc:7872	NOS1	TTD	2020.06.01	NULL	NULL	NXN-462	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	IC9-GD2-CD28-OX40	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.1635752997996713	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
HORMONE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD4901	ncit:C166698	PAVINETANT	FALSE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	Autologous T cells transfected with chimeric anti-mesothelin immunoreceptor SS1	NULL	NULL	NULL	NULL	NULL
ENZYME UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASC-101	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 specific CAR T cells	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	K-103-IP	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-GD2-CAR engineered T cells	NULL	NULL	NULL	NULL	NULL
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	8.751278539282417	QUINETHAZONE	rxcui:59743	QUINETHAZONE	TRUE	FALSE	FALSE
HAEMOPHILUS INFLUENZAE CRM197	NULL	NULL	TTD	2020.06.01	NULL	NULL	NU300	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting CD19	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD22	NULL	NULL	NULL	NULL	NULL
ACTIVATION B7-1 ANTIGEN	hgnc:1700	CD80	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD80/86	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting HER2	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	CD123-specific gene-engineered T cells	NULL	NULL	NULL	NULL	NULL
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	NULL	CD38-specific gene-engineered T cells	NULL	NULL	NULL	NULL	NULL
NEURAL CELL ADHESION MOLECULE 1	hgnc:7656	NCAM1	TTD	2020.06.01	NULL	NULL	CD56-specific gene-engineered T cells	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.089501712	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	Muc1-specific gene-engineered T cells	NULL	NULL	NULL	NULL	NULL
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting CEA	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting EGFRvIII	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting HER2	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Humanized CD19 CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	PZ01 CAR-T cells	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	CART-117 cells	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	CART-33 cells	NULL	NULL	NULL	NULL	NULL
NEURAL CELL ADHESION MOLECULE 1	hgnc:7656	NCAM1	TTD	2020.06.01	NULL	NULL	CART-56 cells	NULL	NULL	NULL	NULL	NULL
UNIPROT:P18825	hgnc:283	ADRA2C	TEND	1-Aug-11	NULL	0.1848861663228679	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
CLAUDIN-18	hgnc:2039	CLDN18	TTD	2020.06.01	NULL	NULL	CAR-CLD18 T cell	NULL	NULL	NULL	NULL	NULL
MYELOID INHIBITORY C-TYPE LECTIN-LIKE RECEPTOR	hgnc:31713	CLEC12A	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CLL1	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting PSMA	NULL	NULL	NULL	NULL	NULL
MELANOMA-ASSOCIATED ANTIGEN 1	hgnc:6796	MAGEA1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting MAGE-A1	NULL	NULL	NULL	NULL	NULL
MELANOMA-ASSOCIATED ANTIGEN 4	hgnc:6802	MAGEA4	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting MAGE-A4	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-CAR T cell	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	GD2-CART01	hemonc:117107	GD2-CART01	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CARCIK-CD19	NULL	NULL	NULL	NULL	NULL
NEUROTROPHIC TYROSINE KINASE ROR2	hgnc:10257	ROR2	TTD	2020.06.01	NULL	NULL	CCT301-38 (targeting ROR2)	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.010128795	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	MUC-1 CART cell immunotherapy	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	EGFR806-specific CAR T cell	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	Anti-C-met CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.921012362281506	KYMRIAH	rxcui:1986438	TISAGENLECLEUCEL	TRUE	FALSE	TRUE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	1.640864726115453	ATLCAR.CD30.CCR4 cells	ncit:C155293	AUTOLOGOUS CCR4-CD30CAR-CD28-CD3ZETA-EXPRESSING T-LYMPHOCYTES	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Human CD19 targeted T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-TriCAR-T	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA-UCART	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	CD38 and BCMA CAR-T Cells	NULL	NULL	NULL	NULL	NULL
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	NULL	CD38 and BCMA CAR-T Cells	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	GSK-958108	NULL	NULL	NULL	NULL	NULL
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	NULL	SCH-1359113	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	CD19.CAR-aNKT cells	ncit:C177533	ALLOGENEIC ANTI-CD19-CAR-CD28-IL-15-EXPRESSING NATURAL KILLER T-CELLS	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	2.212697851403848	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indeloxazine	rxcui:1311673	INDELOXAZINE	FALSE	FALSE	FALSE
SEROTONINNOREPINEPHRINEDOPAMINE REUPTAKE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Olanzapine/fluoxetine combination	NULL	NULL	NULL	NULL	NULL
RIBOSOME A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Omacetaxine mepesuccinate	rxcui:27100	OMACETAXINE MEPESUCCINATE	TRUE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
PROTEASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Prolastin	rxcui:535	ALPHA 1-ANTITRYPSIN	TRUE	FALSE	FALSE
IMMUNOGLOBULIN UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vaccinia immune globulin	chembl:CHEMBL2108699	VACCINIA IMMUNE GLOBULIN	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	EFEGATRAN SULFATE HYDRATE	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	LB-30870	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	SR-46559A	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 3A	hgnc:8778	PDE3A	TTD	2020.06.01	NULL	2.386712328895204	BEMORADAN	ncit:C76314	BEMORADAN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	13.12691780892362	Oxilofrine	rxcui:32639	OXILOFRINE	FALSE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis(olanzapine) pamoate monohydrate	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Bis(olanzapine) pamoate monohydrate	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	FASORACETAM	ncit:C65623	FASORACETAM	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Adefovir Dipivoxil	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amoxicillin	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
ACID-SENSING ION CHANNEL 1	hgnc:100	ASIC1	TTD	2020.06.01	NULL	0.081281225	Amiloride	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
FUNGAL 1,3-BETA-GLUCAN SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Caspofungin	rxcui:140108	CASPOFUNGIN	TRUE	FALSE	FALSE
CALCIUM	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cellulose Sodium Phosphate	rxcui:342965	CELLULOSE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dapagliflozin Propanediol; Saxagliptin Hydrochloride	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.6105543166941221	Methyldopate Hydrochloride	rxcui:91241	METHYLDOPATE HYDROCHLORIDE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Enoximone	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	4SC-203	drugbank:DB12669	4SC-203	FALSE	FALSE	FALSE
POSITIVE TRANSCRIPTION ELONGATION FACTOR B	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY1143572	ncit:C121456	ATUVECICLIB	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.4039051633514961	CLR457	ncit:C117230	PAN-PI3K INHIBITOR CLR457	FALSE	FALSE	FALSE
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	1.944728564284981	CEP-37440	drugbank:DB13060	CEP-37440	FALSE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	Medusa IL-2	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	Liposomal encapsulated doxorubicin (LED)	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-ornithine phenylacetate	NULL	NULL	NULL	NULL	NULL
POLY-N-ACETYL GLUCOSAMINE	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAR279356	NULL	NULL	NULL	NULL	NULL
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	TC-6499-12	chembl:CHEMBL4594254	SIMPINICLINE	FALSE	FALSE	FALSE
HEPATITIS C VIRUS SERINE PROTEASE NS4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	TG-2349	chembl:CHEMBL4297647	FURAPREVIR	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	Roclatan	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Roclatan	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	MC-3002	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MC-3002	NULL	NULL	NULL	NULL	NULL
STREPTOCOCCUS STREPTOKINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Streptokinase rectal suppository	NULL	NULL	NULL	NULL	NULL
AMP-ACTIVATED PROTEIN KINASE	hgnc:9377	PRKAA2	TTD	2020.06.01	NULL	NULL	MB-11055	NULL	NULL	NULL	NULL	NULL
BACTERIAL 70S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Viomycin sulfate	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
LOW-AFFINITY NERVE GROWTH FACTOR RECEPTOR	hgnc:7809	NGFR	TTD	2020.06.01	NULL	NULL	SPI-205	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROFOLATE REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Iclaprim	ncit:C65877	ICLAPRIM	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Arbaclofen placarbil	ncit:C76088	ARBACLOFEN PLACARBIL	FALSE	FALSE	FALSE
BACTERIAL 70S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Capreomycin Sulfate	rxcui:1987	CAPREOMYCIN SULFATE	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	SSR-181507	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	SSR-181507	NULL	NULL	NULL	NULL	NULL
SOMATOSTATIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Somatoprim	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
APOPTOSIS INHIBITOR SURVIVIN	hgnc:593	BIRC5	TTD	2020.06.01	NULL	NULL	ISIS 23722	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.2885036881082115	PF-03084014	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
INTEGRIN ALPHA-4/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Firategrast	ncit:C76692	FIRATEGRAST	FALSE	FALSE	FALSE
NEUROMEDIN-K RECEPTOR	hgnc:11528	TACR3	TTD	2020.06.01	NULL	NULL	GSK1144814	NULL	NULL	NULL	NULL	NULL
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	GSK1144814	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	Nalbuphine hydrochloride ER	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	Nalbuphine hydrochloride ER	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.3182283105193605	Lixisenatide	rxcui:1440051	LIXISENATIDE	TRUE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoline derivative 18	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoline derivative 20	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Heteroaryl-pyrazole derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-16	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-16	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-25	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-38	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-41	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-49	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-50	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-52	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 77	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 5	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 7	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	2,2-bipyridyl derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	2,2-bipyridyl derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	Disulfiram analog 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Hydroxyqunoline analog 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Hydroxyqunoline analog 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 8	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 9	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-47	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-53	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Pyridine-2,4-dicarboxylic acid analog 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Pyridine-2,4-dicarboxylic acid analog 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	Selenium compound 1	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 3	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Lactam derivative 3	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Lactam derivative 5	NULL	NULL	NULL	NULL	NULL
ACETOACETYL-COA THIOLASE	hgnc:93	ACAT1	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-K-604	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-PF-04620110	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 28	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo cyclohexylamine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo cyclohexylamine derivative 3	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 47	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-13	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-17	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-18	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-38	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-71	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 30	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 31	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 32	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidinedione derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[1,2-f]triazine derivative 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazole piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyrimidinedione derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-11	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-Figure3	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-10	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-13	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-117	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-123	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-126	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-127	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-131	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-133	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-140	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-142	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-152	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-155	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-157	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-18	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-2	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-20	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-21	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-22	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-25	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-31	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-33	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-39	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-5	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-50	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-55	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-60	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-64	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-66	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-68	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-70	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-74	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-75	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-79	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-8	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-83	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-87	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-88	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-92	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-93	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-95	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzonaphthyridine derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 5	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 12	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 13	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 15	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 16	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 17	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 19	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 5	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Aromatic ring compound 1	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Aromatic ring compound 2	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Biphenyl carboxamidopropanoic acid derivative 3	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Heterocycle-containing compound 1	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Picolinamido propanoic acid derivative 3	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	PMID25828189-Compound-19	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 6	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 8	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Quinolinyl compound 1	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Spiroimidazolone derivative 2	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-11	NULL	NULL	NULL	NULL	NULL
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	0.9053046764774912	PG-102	chembl:CHEMBL2109475	PG-102	FALSE	FALSE	FALSE
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-16	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-22	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-22	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-27	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 2	hgnc:591	BIRC3	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-27	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-27	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-31	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-37	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-37	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-45	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-6	NULL	NULL	NULL	NULL	NULL
MELANOMA INHIBITOR OF APOPTOSIS PROTEIN	hgnc:13702	BIRC7	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-6	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-6	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 7	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A10	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A10	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A7	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A7	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A8	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A8	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A9	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A9	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-C1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-E1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-E2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-G4	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J3	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J6	NULL	NULL	NULL	NULL	NULL
JNK-INTERACTING PROTEIN PEPTIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-L1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	N-(pyridin-2-yl)pyrimidin-4-amine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	N-(pyridin-2-yl)pyrimidin-4-amine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Naphthyridine and isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Naphthyridine and isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	Naphthyridine and isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 3	hgnc:1772	CDK3	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	Oxazolyl methylthiothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 3	hgnc:1772	CDK3	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-17	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-17	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-25	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-25	NULL	NULL	NULL	NULL	NULL
CDC7-RELATED KINASE	hgnc:1745	CDC7	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-44	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-44	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Purine derivative 4	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Pyrazinylpyridine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	NULL	Pyrazolo-triazine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Tricyclic benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	Tricyclic benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	NULL	Tricyclic benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 8	hgnc:1779	CDK8	TTD	2020.06.01	NULL	NULL	Tricyclic benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Tricyclic benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl compound 2	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl compound 4	NULL	NULL	NULL	NULL	NULL
NF-KAPPA-B-ACTIVATING KINASE	hgnc:11584	TBK1	TTD	2020.06.01	NULL	NULL	Pyrimidinyl compound 6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 2	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 4	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin analog 2	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Curcumin analog 2	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 2	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 3	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Gold-complexed thiosaccharide derivative 2	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Gold-complexed thiosaccharide derivative 3	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 4	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 1	hgnc:11362	STAT1	TTD	2020.06.01	NULL	NULL	Platinum IV complexe 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Platinum IV complexe 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 5	hgnc:11366	STAT5A	TTD	2020.06.01	NULL	NULL	Platinum IV complexe 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-50	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-54	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 63	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Salicylic acid derivative 2	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Salicylic acid derivative 3	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Salicylic acid derivative 6	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Aryl urea derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azetidine urea derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Benzoxazole derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Boronic acid derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Boronic acid derivative 4	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Boronic acid derivative 5	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Boronic acid derivative 6	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-34	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 11	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 11	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 12	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 12	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 15	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 15	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 16	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 16	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 18	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 18	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 19	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 19	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 2	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 2	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 20	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 20	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 13	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 20	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-cyclodextrin conjugate derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 13	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 18	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 30	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 31	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 13	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 15	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 16	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 17	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 5	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 8	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-128	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-50	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5d	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-6b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-7c	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-8a	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-8d	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-9d	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-9e	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-9f	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 1	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 2	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	3-(phenoxymethyl) benzylamine derivative 6	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Aromatic hydrazine carboxyimidoamide derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Aromatic hydrazine carboxyimidoamide derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Aromatic hydrazine carboxyimidoamide derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Aromatic hydrazine carboxyimidoamide derivative 6	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzoic acid linked peptide analog 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzoic acid linked peptide analog 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzothiazole analog 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzothiazoline derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 10	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 12	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 14	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 6	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 6	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Diamine derivative 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Aryl methoxyacrylate derivative 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Matairesinol derivative 1	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-15	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Steroid derivative 4	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Aminocyclopentenone compound 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Aminocyclopentenone compound 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 11	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 11	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 12	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-53	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-57	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrazole and thiophene derivative 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Pyrimido-indole derivative 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrrolone derivative 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Quinazolinone derivative 4	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Tetra-hydro-quinoline derivative 4	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Amidine compound 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 9	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-20a	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-20a	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-37a	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-42a	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-43a	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-43c	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-45	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-46	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-30	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-30	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-32	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-34	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-38	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-39	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	2-cycloalkyl resorcinol cannabinoid ligand derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	2-cycloalkyl resorcinol cannabinoid ligand derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	2-cycloalkyl resorcinol cannabinoid ligand derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	2-cycloalkyl resorcinol cannabinoid ligand derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Adamantyl derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Carbazole-3-carboxamide analog 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Carbazole-3-carboxamide analog 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-12	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-19	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 6	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 6	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo triazine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo triazine derivative 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27321640-Compound-58	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Figure3CG	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-422	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-422	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3B	hgnc:2979	DNMT3B	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-422	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-424	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-424	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3B	hgnc:2979	DNMT3B	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-424	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-PG-11048	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-PG-11048	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Table1Example11	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Table1Example30	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-Table1Example4	NULL	NULL	NULL	NULL	NULL
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	NULL	PMID27387065-Compound-6	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-1	hgnc:10430	RPS6KA1	TTD	2020.06.01	NULL	NULL	1,6-diazanaphthalenes and pyrido[2,3-d] pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-1	hgnc:10430	RPS6KA1	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 26	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE BETA-1	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	NULL	PMID27410995-Compound-Figure3c	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-82	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 12	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 4	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 5	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 6	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 9	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Aryl oxyanilide derivative 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Aryl oxyanilide derivative 3	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzimidazolone acetamide derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 7	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Bidentate pyrazolopyrimidine acetamide analog 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine acetamide derivative 3	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine acetamide derivative 4	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 7	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Phenylpyrrolidinone derivative 1	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Phenylpyrrolidinone derivative 4	NULL	NULL	NULL	NULL	NULL
DUAL SPECIFICITY PROTEIN KINASE TTK	hgnc:10416	RPS27	TTD	2020.06.01	NULL	NULL	Tricyclic isoxazoloquinazoline derivative 3	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Tricyclic isoxazoloquinazoline derivative 3	NULL	NULL	NULL	NULL	NULL
DUAL SPECIFICITY PROTEIN KINASE TTK	hgnc:10416	RPS27	TTD	2020.06.01	NULL	NULL	Tricyclic isoxazoloquinazoline derivative 4	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Tricyclic isoxazoloquinazoline derivative 4	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Benzo(b)carbazol-11-one compound 1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Dihydropyridine compound 2	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Dihydropyridine compound 6	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Indole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	PMID27724045-Compound-14	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	PMID27724045-Compound-15	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	PMID27724045-Compound-29	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	PMID27724045-Compound-33	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Quinoline derivative 12	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 12	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Thiazole derivative 5	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Triazolo-pyrazinone derivative 1	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	Indole-based analog 1	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	Indole-based analog 3	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	NULL	Indole-based analog 3	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	Indole-based analog 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridone derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridone derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic compound 11	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic compound 11	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Tricyclic compound 11	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Tricyclic compound 11	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclohexyl azetidine derivative 1	NULL	NULL	NULL	NULL	NULL
JAK-STAT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure3Example18	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure3Example18	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure3Example18	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure3Example18	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure5Example13	NULL	NULL	NULL	NULL	NULL
EGFR T790M MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2down	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2down	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2down	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2down	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2down	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2down	NULL	NULL	NULL	NULL	NULL
B LYMPHOCYTE KINASE	hgnc:1057	BLK	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
T-CELL-SPECIFIC KINASE	hgnc:6171	ITK	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE TEC	hgnc:11719	TEC	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidopyridazinone derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	NULL	Pyrimidopyridazinone derivative 1	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-132	NULL	NULL	NULL	NULL	NULL
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zithromax	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-3	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-39	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-42	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-43	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-neotuberostemonine	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine-caffeic acid hybrid derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-43	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-48	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Terpyridineplatinum(II) complexe 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Terpyridineplatinum(II) complexe 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Terpyridineplatinum(II) complexe 3	NULL	NULL	NULL	NULL	NULL
GLUTATHIONE REDUCTASE	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	Terpyridineplatinum(II) complexe 3	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-11	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-12	NULL	NULL	NULL	NULL	NULL
CATHEPSIN F	hgnc:2531	CTSF	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-12	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-12	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-12	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-12	NULL	NULL	NULL	NULL	NULL
CATHEPSIN V	hgnc:2538	CTSV	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-12	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-2	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-9	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-9	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-9	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-9	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hexahydro azepinone derivative 1	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoquinoline sulfonyl derivative 3	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-2	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-2	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-6	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-6	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	Tricyclic compound 5	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	Tricyclic compound 7	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	STM 434	iuphar.ligand:8991	STM 434	FALSE	FALSE	FALSE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	1,2,4-triazole derivative 3	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Aryl alkanolamine derivative 2	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Bicyclo-heptan-2-amine derivative 2	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Bicyclo-heptan-2-amine derivative 3	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	N-substituted 9-azabicyclo[3.3.1]nonan-3alpha-yl-phenylcarbamate analog 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	N-substituted 9-azabicyclo[3.3.1]nonan-3alpha-yl-phenylcarbamate analog 3	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Phenylpropylamine derivative 2	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Piperidine derivative 4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID28051882-Compound-Figure9	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 86	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	2-(substituted ethynyl)quinoline derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	6-aryl-imidazopyridine and 6-aryl-triazolopyridine carboxamide analog 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Bicarboxylic and tricarboxylic ethynyl derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl carboxamide analog 1	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33e	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33e	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33f	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33f	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33h	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33h	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33i	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33i	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33k	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33k	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33l	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33l	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33m	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33m	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Aminopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2 G2019S MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-arylmethyl-N-phenyl cyclic urea derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure16-a	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure16-b-1	NULL	NULL	NULL	NULL	NULL
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure24-a	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure24-a	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-3	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21918	hgnc:3026	DRD5	TEND	1-Aug-11	NULL	0.097236428	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 18	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 21	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 23	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 10	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 3	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 8	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpiperidine ether derivative 4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpiperidine ether derivative 5	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpyrrolidine ether derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2010077680 103	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2010077680 201	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2010077680 803	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2013009582Example76	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2014078408Example1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2014078408Example26	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2016054807Example112	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[4,3-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-b]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[3,2-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Six-membered heterocyclic benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Six-membered heterocyclic benzamide derivative 7	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-21	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-35	NULL	NULL	NULL	NULL	NULL
EZH2 Y641F MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-11	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.01354163	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-15	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-17	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-18	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-23	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-27	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-31	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE 1	hgnc:6840	MAP2K1	TTD	2020.06.01	NULL	NULL	Pyridic ketone derivative 1	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27487	hgnc:3009	DPP4	TEND	1-Aug-11	NULL	1.050153425	SAXAGLIPTIN	rxcui:1546030	SAXAGLIPTIN ANHYDROUS	TRUE	FALSE	FALSE
ERK ACTIVATOR KINASE 2	hgnc:6842	MAP2K2	TTD	2020.06.01	NULL	NULL	Pyridic ketone derivative 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	3-phenyl-5-ureidoisothiazole-4-carboximide and 3-amino-5-phenylisothiazole derivative 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 11	NULL	NULL	NULL	NULL	NULL
GREMLIN-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Antibodie derivative 5	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Antibodie derivative 6	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 7	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00374	hgnc:2861	DHFR	TEND	1-Aug-11	NULL	0.525076712	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 8	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 14	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Oxetane 3,3-dicarboxamide compound 2	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 4	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 6	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 12	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 7	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 9	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzamide derivative 14	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzamide derivative 18	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 14	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 15	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 16	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 17	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 5	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	PMID28627961-Compound-30	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	PMID28627961-Compound-31	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14324	hgnc:3631	FDPS	TEND	1-Aug-11	NULL	1.458546423213736	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
FUNGAL PROTON PUMP	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrithione Zinc	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Benzodihydroisofuran derivative 1	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Benzodihydroisofuran derivative 2	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Cyclohexane carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Cyclopentane carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Cyclopentane carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl pyrazole derivative 2	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl triazole derivative 1	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl triazole derivative 2	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Pyrrolidine carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08709	hgnc:3544	F7	TEND	1-Aug-11	NULL	1.250182648468916	COAGULATION FACTOR VIIA	rxcui:2386863	COAGULATION FACTOR VIIA (RECOMBINANT)-JNCW	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 16	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 17	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 18	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 31	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 33	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme12-2	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme14BINDY	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme14BINDY	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 2	hgnc:3093	DYRK2	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme14BINDY	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme15-2	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure11(3)	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure11(3)	NULL	NULL	NULL	NULL	NULL
GELATINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure14(5)	NULL	NULL	NULL	NULL	NULL
GELATINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure14(6)	NULL	NULL	NULL	NULL	NULL
UNIPROT:P18825	hgnc:283	ADRA2C	TEND	1-Aug-11	NULL	0.2465148884304905	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure16(9a)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure16(9a)	NULL	NULL	NULL	NULL	NULL
KALLIKREIN-4	hgnc:6365	KLK4	TTD	2020.06.01	NULL	NULL	Benzoxazinone derivative 2	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1204304386139782	BUPRENORPHINE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzoxazinone derivative 2	NULL	NULL	NULL	NULL	NULL
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 11	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Tacrine-coumarin hybrid derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tacrine-coumarin hybrid derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	4-benzylidene-1-(cyclobutylo)piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazol-2(3H)-one derivative 2	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazol-2(3H)-one derivative 2	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazol-2(3H)-one derivative 3	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazol-2(3H)-one derivative 3	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylsulfonyl derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylsulfonyl derivative 3	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine carbamate/urea derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine carbamate/urea derivative 2	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine carbamate/urea derivative 4	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-25	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	BROMODIPHENHYDRAMINE	rxcui:19759	BROMODIPHENHYDRAMINE	TRUE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-28	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-58	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-benzodiazepine derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-13	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-15	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-20	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-22	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-23	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-24	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-27	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.2282942227638891	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-28	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-33	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-40	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-44	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-48	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-49	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Amide derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Biphenyl 1,2-diamine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Biphenyl derivative 3	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Imidazo isoindole derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Imidazoleisoindoles derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Indazole derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Monoaryl-1,2-diamine derivative 2	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Monoaryl-1,2-diamine derivative 3	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.047886613	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-14	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-16	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-72b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-9	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-9	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-9	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-9	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-7	NULL	NULL	NULL	NULL	NULL
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.068637479	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-7	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8b	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8b	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.2234368988752957	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-isoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 10	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 13	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 13	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 17	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 17	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 22	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 38	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 38	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 38	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 41	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 41	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 41	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 41	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 41	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 42	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-38	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-39	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-45	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-46	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-46	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-46	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-46	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-52	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-54	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclic peptidomimetic derivative 3	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocyclic peptide analog 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-phenyl-pyridine-2-carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylate derivative 2	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example12	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example12	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example14	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2015035128	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2015150568	NULL	NULL	NULL	NULL	NULL
KERATINOCYTE GROWTH FACTOR	hgnc:3685	FGF7	TTD	2020.06.01	NULL	NULL	Keratinocyte growth factor (KGF)	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PF-3864086	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.921012362281506	CTL019	rxcui:1986438	TISAGENLECLEUCEL	TRUE	FALSE	TRUE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	INTOPLICINE	ncit:C1495	INTOPLICINE	FALSE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	TAK-114	NULL	NULL	NULL	NULL	NULL
DELTA-AMINOLEVULINIC ACID DEHYDRATASE	hgnc:395	ALAD	TTD	2020.06.01	NULL	NULL	Aminolevulinic acid hci	NULL	NULL	NULL	NULL	NULL
THYROTROPIN-RELEASING HORMONE RECEPTOR	hgnc:12299	TRHR	TTD	2020.06.01	NULL	17.50255707856483	protirelin	rxcui:10580	THYROTROPIN-RELEASING HORMONE	TRUE	FALSE	FALSE
VITAMIN K EPOXIDE REDUCTASE COMPLEX 1	hgnc:23663	VKORC1	TTD	2020.06.01	NULL	4.200613698855561	Acenocoumarol	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
BETA-HEMATIN FORMATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Arteether	ncit:C73002	ARTEMOTIL	TRUE	FALSE	FALSE
PLASMODIUM DIHYDROOROTATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Atovaquone	rxcui:60212	ATOVAQUONE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	Belotecan hydrocholoride	NULL	NULL	NULL	NULL	NULL
AMIDOPHOSPHORIBOSYLTRANSFERASE	hgnc:9238	PPAT	TTD	2020.06.01	NULL	0.921187215	Azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Besifloxacin	rxcui:819911	BESIFLOXACIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Besifloxacin	rxcui:819911	BESIFLOXACIN	TRUE	FALSE	FALSE
VESICLE-ASSOCIATED MEMBRANE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Botulinum Toxin Type B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.272767123	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Cimetropium bromide	ncit:C90696	CIMETROPIUM BROMIDE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	Dhaq diacetate	NULL	NULL	NULL	NULL	NULL
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Efinaconazole	rxcui:1539753	EFINACONAZOLE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.03849536	Doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	2.258394462	Golimumab	rxcui:819300	GOLIMUMAB	TRUE	TRUE	FALSE
CYTOMEGALOVIRUS TERMINASE UL56	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-8228	rxcui:1988648	LETERMOVIR	TRUE	FALSE	FALSE
HEPATITIS B VIRUS LARGE ENVELOPE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nabi-HB (intramuscular)	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Naltrexone	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	Oral paclitaxel	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	Oral paclitaxel	NULL	NULL	NULL	NULL	NULL
INFLUENZA NEURAMINIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oseltamivir	rxcui:259275	OSELTAMIVIR PHOSPHATE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	1.193356164447602	Morniflumate	rxcui:30225	MORNIFLUMATE	FALSE	FALSE	FALSE
BACTERIAL FATTY ACID SYNTHETASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	Prothionamide	rxcui:8871	PROTHIONAMIDE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.5427149481725528	Procaterol	rxcui:34530	PROCATEROL	FALSE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1B	hgnc:7464	MTNR1B	TTD	2020.06.01	NULL	10.50153424713889	Ramelteon	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
LYSOSOMAL ACID LIPASE	hgnc:6617	LIPA	TTD	2020.06.01	NULL	8.751278539282415	SBC-102	rxcui:1726975	SEBELIPASE ALFA	TRUE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	2.187819634820604	Sulodexide	ncit:C152467	SULODEXIDE	TRUE	FALSE	FALSE
ADENOSINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Theophylline	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valproate	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1101693521639275	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE	hgnc:30092	NAMPT	TTD	2020.06.01	NULL	21.00306849427779	GMX1777	drugbank:DB05217	GMX1777	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	PF-4603629	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	R-1663	NULL	NULL	NULL	NULL	NULL
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	ROCICLOVIR	ncit:C73204	ROCICLOVIR	FALSE	FALSE	FALSE
PROLYL ENDOPEPTIDASE	hgnc:9358	PREP	TTD	2020.06.01	NULL	NULL	S-17092-1	NULL	NULL	NULL	NULL	NULL
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.3918482928036902	MK-5108	drugbank:DB12556	MK-5108	FALSE	FALSE	FALSE
MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE	hgnc:16870	MELK	TTD	2020.06.01	NULL	5.250767123569449	OTSSP167	iuphar.ligand:8046	OTSSP167	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	NULL	SDZ-LAV-694	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	SSR-125329A	NULL	NULL	NULL	NULL	NULL
OXIDATIVE STRESS	hgnc:7095	MID1	TTD	2020.06.01	NULL	NULL	SUN-N8075	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.093763699	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
GLYCINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ZD-9379	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD8	hgnc:1706	CD8A	TTD	2020.06.01	NULL	NULL	Anti-VEGFR2 CD8 cell therapy	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	Anti-VEGFR2 CD8 cell therapy	NULL	NULL	NULL	NULL	NULL
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.075333818	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.079197091	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	CHLOPHEDIANOL	rxcui:21254	CHLOPHEDIANOL	TRUE	FALSE	FALSE
COMPLEMENT FACTOR D	hgnc:2771	CFD	TTD	2020.06.01	NULL	8.751278539282415	Anti-Factor D	iuphar.ligand:8294	LAMPALIZUMAB	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 7	hgnc:1778	CDK7	TTD	2020.06.01	NULL	2.100306849	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	CAP1-6D	NULL	NULL	NULL	NULL	NULL
ERBB4 TYROSINE KINASE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CI-1033	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
CASPASE-1	hgnc:1499	CASP1	TTD	2020.06.01	NULL	4.039051633514961	Belnacasan	ncit:C171755	BELNACASAN	FALSE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	4.565884455277782	BQ-123	drugbank:DB12054	BQ-123	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.1367387271762877	CARPHENAZINE	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
CD40L RECEPTOR	hgnc:11919	CD40	TTD	2020.06.01	NULL	1.093909817410302	CFZ533	iuphar.ligand:9802	CFZ533	FALSE	FALSE	FALSE
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-745,870	iuphar.ligand:3303	L745870	FALSE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	Labetuzumab I-131	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	LCAR-B38M CAR-T Cell	NULL	NULL	NULL	NULL	NULL
FARNESYL PROTEIN TRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lonafarnib	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1556551518844698	CARPHENAZINE	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
INDUCIBLE T-CELL COSTIMULATOR	hgnc:5351	ICOS	TTD	2020.06.01	NULL	35.00511415712966	JTX-2011	ncit:C129876	VOPRATELIMAB	FALSE	FALSE	FALSE
ATP PHOSPHATASE	hgnc:2952	DNAH8	TTD	2020.06.01	NULL	NULL	LYC-30937	NULL	NULL	NULL	NULL	NULL
NICOTINIC ACID RECEPTOR	hgnc:24827	HCAR2	TTD	2020.06.01	NULL	NULL	MK-1903	NULL	NULL	NULL	NULL	NULL
RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MLN2480	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	OCFENTANIL	ncit:C84024	OCFENTANIL	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Org-30029	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	MGA012	ncit:C142168	RETIFANLIMAB	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.054243462	METHYLENEDIOXYMETHAMPHETAMINE	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	S-15535	iuphar.ligand:26	S-15535	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	SSR-180575	NULL	NULL	NULL	NULL	NULL
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tempol	drugbank:DB12449	TEMPOL	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRAXOPRODIL MESYLATE	ncit:C61981	TRAXOPRODIL MESYLATE	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	TZI-41078	NULL	NULL	NULL	NULL	NULL
CAMP FORMATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	UCB-11056	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.1539814405738841	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	1.193356164447602	ASP1941	ncit:C166685	IPRAGLIFLOZIN	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	AVP-786	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clazosentan	ncit:C79486	CLAZOSENTAN	FALSE	FALSE	FALSE
CLUSTERIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Custirsen	ncit:C169869	CUSTIRSEN	FALSE	FALSE	TRUE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TEND	1-Aug-11	NULL	0.2344092465879218	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
GLUTAMATE DECARBOXYLASE 2	hgnc:4093	GAD2	TTD	2020.06.01	NULL	NULL	Diamyd	NULL	NULL	NULL	NULL	NULL
FUNGAL PAPULACANDIN B RESISTANCE PROTEIN 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Eraxis/Vfend	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCTION UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Forigerimod	ncit:C166505	FORIGERIMOD	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.4930297768609811	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Grippol Plus	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Grippol TC	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDDBCP161883	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	ketoprofen patch	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Low dose ITI-007	NULL	NULL	NULL	NULL	NULL
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	NULL	NT0202	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	NULL	PGF2ALPHA-IE	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:80	iuphar.ligand:3251	[3H]WAY100635	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.090634645	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.3163112725041837	IUPHAR.LIGAND:117	ncit:C77255	ALNIDITAN	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.063262255	IUPHAR.LIGAND:60	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:145	iuphar.ligand:145	5-MEO-DMT	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1346350544504987	IUPHAR.LIGAND:60	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1121958787087489	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.046303061	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.046303061	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.046303061	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:160	iuphar.ligand:160	AL-37350A	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:159	iuphar.ligand:159	N-1-ISOPROPYLTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.08334551	IUPHAR.LIGAND:167	iuphar.ligand:167	S 16924	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.050246575	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:173	ncit:C61919	QUIPAZINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.02271093	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.035098711	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.032173818	IUPHAR.LIGAND:130	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.4449802647092754	IUPHAR.LIGAND:141	drugbank:DB01488	DIMETHYLTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.042379073	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.3547815624033412	DARIFENACIN	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:792	hgnc:74	ABCG2	GuideToPharmacology	2024.1	inhibitor	0.066011799	IUPHAR.LIGAND:1024	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:8121	iuphar.ligand:8121	ML347	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.1158257453728555	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:80	hgnc:153	ACTG1P8	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:836	iuphar.ligand:836	CXCL11	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:8959	iuphar.ligand:8959	ENSARTINIB	FALSE	FALSE	FALSE
NCBIGENE:2611	hgnc:4147	GAPDHP69	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4642	ncit:C87373	DUVOGLUSTAT	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:490	iuphar.ligand:490	A-119637	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.6403374540938354	IUPHAR.LIGAND:480	iuphar.ligand:480	A61603	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.066297565	IUPHAR.LIGAND:7207	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	0.6058577450272442	DIHYDROERGOTAMINE	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.032252869	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.070197421	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2857	ncit:C166564	METRIBOLONE	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:6459	rxcui:21102	CILAZAPRIL	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:5606	iuphar.ligand:5606	FK-453	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:417	iuphar.ligand:417	APNEA	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1875273972703375	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.063110182	IUPHAR.LIGAND:380	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:399	iuphar.ligand:399	MRS1093	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:585	iuphar.ligand:585	ANGIOTENSIN III	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:11931	iuphar.ligand:11931	COMPOUND 2 [PMID: 28379944]	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:8466	iuphar.ligand:8466	COMPOUND 10 [PMID: 19402633]	FALSE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:7733	iuphar.ligand:7733	GDC-0152	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:10394	iuphar.ligand:10394	COMPOUND 3L [PMID: 30637955]	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.017295017	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:534	ncit:C77934	DENOPAMINE	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:569	rxcui:20192	CARAZOLOL	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:12582	rxcui:2580	CLENBUTEROL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	LEVOCABASTINE	rxcui:28627	LEVOCABASTINE	TRUE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.1785975212098452	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:3399	iuphar.ligand:3399	20-HYDROXY-LTB4	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.0287871	LISURIDE	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:1786	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:8155	iuphar.ligand:8155	COMPOUND 13A [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11690	iuphar.ligand:11690	GSK852	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:7034	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.4449802647092754	LISINOPRIL	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7514	iuphar.ligand:7514	GW841819X	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7809	iuphar.ligand:7809	COMPOUND 1 [PMID: 25408830]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:7512	iuphar.ligand:7512	MS417	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:7514	iuphar.ligand:7514	GW841819X	FALSE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TEND	1-Aug-11	NULL	1.121958787087489	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
NCBIGENE:2726	hgnc:14310	BRD7	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9522	iuphar.ligand:9522	TP-472	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:9391	iuphar.ligand:9391	COMPOUND 36 [PMID: 21958547]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:11983	iuphar.ligand:11983	EXAMPLE A225 [WO2012170976A2]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9516	iuphar.ligand:9516	CHMFL-BTK-11	FALSE	FALSE	FALSE
UNIPROT:P47712	hgnc:9035	PLA2G4A	TEND	1-Aug-11	NULL	1.093909817410302	MEDRYSONE	rxcui:29439	MEDRYSONE	TRUE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:647	iuphar.ligand:647	[DES-PHE9,DES-ARG10]KALLIDIN	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:656	iuphar.ligand:656	JMV1431	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:659	iuphar.ligand:659	NVP-SAA164	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:640	iuphar.ligand:640	[D-LYS1,DES-ARG10]KALLIDIN	FALSE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TEND	1-Aug-11	NULL	0.2243917574174978	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:663	iuphar.ligand:663	[DES-ARG10]ICATIBANT	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:679	ncit:C79554	ANATIBANT	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:9746	iuphar.ligand:9746	NDT9513727	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:10228	iuphar.ligand:10228	LACTOMEDIN 1	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:3915	iuphar.ligand:3915	E7	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.2692701089009974	IUPHAR.LIGAND:6807	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
UNIPROT:P09884	hgnc:9173	POLA1	TEND	1-Aug-11	NULL	1.036335616	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
NCBIGENE:2599	hgnc:1375	CA4	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:6807	rxcui:3353	DICHLORPHENAMIDE	TRUE	FALSE	FALSE
NCBIGENE:531	hgnc:1393	CACNA1F	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2511	iuphar.ligand:2511	BAYK 8644	FALSE	FALSE	FALSE
NCBIGENE:534	hgnc:862	ATP6V1G2	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:2476	iuphar.ligand:2476	NI2+	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11643	iuphar.ligand:11643	CALPEPTIN	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.4782119420372905	MEGESTROL	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
NCBIGENE:2353	hgnc:3796	FOS	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:9855	ncit:C174598	PETESICATIB	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:9430	iuphar.ligand:9430	BMS-681	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:760	iuphar.ligand:760	FLU-CCL3	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.1363835616511545	MECLOFENAMIC ACID	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
NCBIGENE:1990	hgnc:3308	CELA1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8162	iuphar.ligand:8162	ML315	FALSE	FALSE	FALSE
NCBIGENE:1990	hgnc:3308	CELA1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12975	iuphar.ligand:12975	MW05	FALSE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TEND	1-Aug-11	NULL	0.9546849315580819	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
NCBIGENE:2473	hgnc:3883	FRA22A	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6668	iuphar.ligand:6668	NVP 231	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.053361455	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:715	hgnc:1246	C1R	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:723	hgnc:4283	GJB1	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1041818873724097	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TEND	1-Aug-11	NULL	1.591141552596803	NAFARELIN	rxcui:28656	NAFARELIN	TRUE	FALSE	FALSE
NCBIGENE:724	hgnc:1327	C4BPAP2	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:723	hgnc:4283	GJB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:729	hgnc:1339	C6	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:728	hgnc:1338	C5AR1	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
UNIPROT:P23921	hgnc:10451	RRM1	TEND	1-Aug-11	NULL	0.487687349	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12584	iuphar.ligand:12584	ACT-777991	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:8185	iuphar.ligand:8185	COMPOUND 3 [PMID: 19097791]	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:7806	iuphar.ligand:7806	PURVALANOL B	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:5969	iuphar.ligand:5969	FASCAPLYSIN	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:12079	iuphar.ligand:12079	ULECACICLIB	FALSE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.4605936073306534	BENZOCAINE	rxcui:1399	BENZOCAINE	TRUE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:7806	iuphar.ligand:7806	PURVALANOL B	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.049026771	IUPHAR.LIGAND:5670	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.1646008502686348	IUPHAR.LIGAND:7938	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:11885	iuphar.ligand:11885	TANUXICICLIB	FALSE	FALSE	FALSE
UNIPROT:P21817	hgnc:10483	RYR1	TEND	1-Aug-11	NULL	2.083637747448194	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12079	iuphar.ligand:12079	ULECACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:7806	iuphar.ligand:7806	PURVALANOL B	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:8052	iuphar.ligand:8052	THZ1	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.280789686	IUPHAR.LIGAND:7938	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:9171	iuphar.ligand:9171	COMPOUND 20 [BERGERON ET AL., 2016]	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.1065064325267637	IUPHAR.LIGAND:5670	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
NCBIGENE:2027	hgnc:3354	ENO3	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:7792	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
NCBIGENE:1329	hgnc:2269	COX5B	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8746	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TEND	1-Aug-11	NULL	4.039051633514961	PEGFILGRASTIM	rxcui:2048018	PEGFILGRASTIM-JMDB	TRUE	FALSE	FALSE
NCBIGENE:1320	hgnc:2597	CYP1B1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:8789	iuphar.ligand:8789	CHRYSIN	FALSE	FALSE	FALSE
NCBIGENE:1326	hgnc:6860	MAP3K8	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10559	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
UNIPROT:P51172	hgnc:10601	SCNN1D	TEND	1-Aug-11	NULL	2.059124362184098	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:3352	iuphar.ligand:3352	LTE4	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:4797	rxcui:6664	MAZINDOL	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:9006	iuphar.ligand:9006	UFP-512	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.060077427	IUPHAR.LIGAND:7236	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.4646696569530486	IUPHAR.LIGAND:4060	iuphar.ligand:4060	[D-ALA2]DELTORPHIN II	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1161674142382621	IUPHAR.LIGAND:8870	iuphar.ligand:8870	AT-076	FALSE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12238	iuphar.ligand:12238	ICED-2	FALSE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TEND	1-Aug-11	NULL	7.001022831425932	PHENINDIONE	rxcui:8130	PHENINDIONE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.003470434	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.039331589	IUPHAR.LIGAND:7556	ncit:C66358	PEROSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.019739726	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.1628144844517658	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:2832	hgnc:4530	NPBWR2	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8454	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
NCBIGENE:1249	hgnc:7876	NOS3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8759	iuphar.ligand:8759	L-NNA	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.032899543	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:1567	hgnc:29499	ERAP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9682	iuphar.ligand:9682	COMPOUND 2G [PMID: 27390066]	FALSE	FALSE	FALSE
NCBIGENE:1615	hgnc:2678	DARS1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8617	iuphar.ligand:8617	PD159790	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:12615	ncit:C167347	TULMIMETOSTAT	FALSE	FALSE	FALSE
UNIPROT:P55011	hgnc:10911	SLC12A2	TEND	1-Aug-11	NULL	5.834185692854945	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:12164	iuphar.ligand:12164	BI-4142	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	0.1988926940746004	IUPHAR.LIGAND:7259	rxcui:11473	PAMIDRONATE	TRUE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:9601	iuphar.ligand:9601	CATEQUENTINIB	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:9789	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:12485	iuphar.ligand:12485	COMPOUND 7 [NGUYEN ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:11619	ncit:C80870	TOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:12485	iuphar.ligand:12485	COMPOUND 7 [NGUYEN ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:9789	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:9786	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.068369364	IUPHAR.LIGAND:9601	iuphar.ligand:9601	CATEQUENTINIB	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.002707698	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:3175	hgnc:8138	ONECUT1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11481	iuphar.ligand:11481	SAFIT1	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:10549	iuphar.ligand:10549	COMPOUND 18E [PMID: 31670517]	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.004310975	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:5834	iuphar.ligand:5834	COMPOUND R-(-)-5F [PMID: 22607879]	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:5841	iuphar.ligand:5841	FMET-ILE-VAL-THR-LEU-PHE	FALSE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	11.66837138570988	POLYTHIAZIDE	rxcui:8565	POLYTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.020002922	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	0.018288983	IUPHAR.LIGAND:1024	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6265	iuphar.ligand:6265	QUIN-C1	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:3383	iuphar.ligand:3383	ATLA2	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1034	iuphar.ligand:1034	LXA4	FALSE	FALSE	FALSE
NCBIGENE:253	ncbigene:253	ALS3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:1157	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
NCBIGENE:235	hgnc:4045	FZD7	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:10323	iuphar.ligand:10323	SRI37892	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4299	iuphar.ligand:4299	RO4938581	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:4346	iuphar.ligand:4346	ZK93423	FALSE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.1304538415793652	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4326	iuphar.ligand:4326	TP003	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:11942	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.050879526	IUPHAR.LIGAND:4297	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	blocker	0.067839369	IUPHAR.LIGAND:4369	iuphar.ligand:4369	[35S]TBPS	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6106	iuphar.ligand:6106	GAL-B2-DPEG24	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6100	iuphar.ligand:6100	M617	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.023943307	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:3899	iuphar.ligand:3899	M40	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6102	iuphar.ligand:6102	M1151	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3189	iuphar.ligand:3189	BPH-742	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.05309168	IUPHAR.LIGAND:2870	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
NCBIGENE:451	hgnc:769	ASS1P6	GuideToPharmacology	2024.1	modulator	3.750547945	IUPHAR.LIGAND:4162	iuphar.ligand:4162	CONCANAVALIN A	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:4274	iuphar.ligand:4274	NS3763	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.1635752997996713	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4155	ncit:C152322	SELFOTEL	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	blocker	0.079197091	IUPHAR.LIGAND:4233	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1162	iuphar.ligand:1162	GNRH I	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.2191733444543002	SALBUTAMOL	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.2692701089009974	TAMSULOSIN	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.167488584	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4603	iuphar.ligand:4603	[3H]N-METHYL-SSR504734	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.187193124	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:9078	iuphar.ligand:9078	COMPOUND 15 [PMID: 25411721]	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1180	iuphar.ligand:1180	D-23487	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	modulator	0.7955707762984014	IUPHAR.LIGAND:1182	iuphar.ligand:1182	FD-1	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1182	iuphar.ligand:1182	FD-1	FALSE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:726	rxcui:9671	SERINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.3535870116881784	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:1468	hgnc:10980	SLC25A10	GuideToPharmacology	2024.1	inhibitor	4.039051633514962	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:1470	hgnc:2474	CST2	GuideToPharmacology	2024.1	inhibitor	4.039051633514962	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:2031	ncbigene:2031	ENUR1	GuideToPharmacology	2024.1	activator	26.25383561784724	IUPHAR.LIGAND:9165	iuphar.ligand:9165	GUANYLYL CYCLASE-ACTIVATING PROTEIN 2	FALSE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TEND	1-Aug-11	NULL	2.100306849	TETRABENAZINE	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
NCBIGENE:2904	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:10118	iuphar.ligand:10118	GRP94 INHIBITOR 54	FALSE	FALSE	FALSE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:12609	iuphar.ligand:12609	COMPOUND 30 [PMID: 37057760]	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:7007	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:8464	iuphar.ligand:8464	DROXINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:7504	iuphar.ligand:7504	NEXTURASTAT A	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.060353645	IUPHAR.LIGAND:11976	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1196	iuphar.ligand:1196	2-(3-IODOPHENYL)HISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.060353645	IUPHAR.LIGAND:6063	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:7157	rxcui:275635	DESLORATADINE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	agonist	0.9211872146613068	IUPHAR.LIGAND:1229	iuphar.ligand:1229	BURIMAMIDE	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1226	iuphar.ligand:1226	IMPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1221	ncit:C72108	ARPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:1216	iuphar.ligand:1216	A-317920	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1259	iuphar.ligand:1259	FUB 349	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:7991	iuphar.ligand:7991	COMPOUND 2 [DREYER ET AL., 1991]	FALSE	FALSE	FALSE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:4837	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TEND	1-Aug-11	NULL	0.1325951293830669	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:101	hgnc:215	ADAM8	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:4064	iuphar.ligand:4064	LYSOPHOSPHATIDYLSERINE	FALSE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:10567	iuphar.ligand:10567	GPR15L	FALSE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	0.6482428547616605	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
UNIPROT:P29274	hgnc:263	ADORA2A	TEND	1-Aug-11	NULL	0.157680694	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:1453	hgnc:2452	CSNK1D	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8844	iuphar.ligand:8844	COMPOUND 5 [NOBLE ET AL., 1992]	FALSE	FALSE	FALSE
NCBIGENE:744	hgnc:1180	MPPED2	GuideToPharmacology	2024.1	activator	0.2625383561784725	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
UNIPROT:P21964	hgnc:2228	COMT	TEND	1-Aug-11	NULL	2.500365296937833	TOLCAPONE	rxcui:72937	TOLCAPONE	TRUE	FALSE	FALSE
NCBIGENE:745	hgnc:1181	MYRF	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:2459	iuphar.ligand:2459	DECAVANADATE	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12444	iuphar.ligand:12444	HOMOERIODICTYOL	FALSE	FALSE	FALSE
NCBIGENE:745	hgnc:1181	MYRF	GuideToPharmacology	2024.1	activator	0.4375639269641209	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:12318	iuphar.ligand:12318	GDC-0214	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:6977	iuphar.ligand:6977	COMPOUND 19A [PMID: 24359159]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:1656	iuphar.ligand:1655	U69593	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.2365210416022274	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1620	iuphar.ligand:1620	DYNORPHIN A	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1666	iuphar.ligand:1666	SALVINORIN A	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.069180068	IUPHAR.LIGAND:7886	iuphar.ligand:7886	FAMITINIB	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.00178914	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.023060023	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:9601	iuphar.ligand:9601	CATEQUENTINIB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:9301	iuphar.ligand:9301	CHMFL-KIT-8140	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.3547815624033412	TRIDIHEXETHYL	rxcui:38617	TRIDIHEXETHYL	TRUE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:12249	iuphar.ligand:12249	COMPOUND 6LI [CHAN ET AL., 2022]	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:7886	iuphar.ligand:7886	FAMITINIB	FALSE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	activator	0.375054795	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	modulator	4.773424657790408	IUPHAR.LIGAND:12649	ncit:C171756	RIMTUZALCAP	FALSE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TEND	1-Aug-11	NULL	0.078793024	VINBLASTINE	rxcui:11198	VINBLASTINE	TRUE	FALSE	TRUE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	2.625383561784724	IUPHAR.LIGAND:9314	iuphar.ligand:9314	CM-TPMF	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	activator	0.062509132	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:2605	iuphar.ligand:2605	E4031	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:7659	iuphar.ligand:7659	KB-130015	FALSE	FALSE	FALSE
NCBIGENE:540	hgnc:870	ATP7B	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:2555	iuphar.ligand:2555	CORREOLIDE	FALSE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TEND	1-Aug-11	NULL	0.421837528	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9815	iuphar.ligand:9815	CCT196969	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9393	iuphar.ligand:9393	GNE-0877	FALSE	FALSE	FALSE
NCBIGENE:2380	hgnc:3892	FRA2H	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8633	iuphar.ligand:8633	COMPOUND 7U [PMID: 24775305]	FALSE	FALSE	FALSE
NCBIGENE:1271	hgnc:2170	CNTFR	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:5116	iuphar.ligand:5116	3-HYDROXYBENZYLHYDRAZINE	FALSE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TEND	1-Aug-11	NULL	0.3062196950280639	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9964	iuphar.ligand:9964	NIK SMI1	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:2753	iuphar.ligand:2753	ACETYL-PODOCARPIC DIMER	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:2936	iuphar.ligand:2936	2-OLEOYL-LPA	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:2936	iuphar.ligand:2936	2-OLEOYL-LPA	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9391	iuphar.ligand:9391	COMPOUND 36 [PMID: 21958547]	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.347732922	Kevetrin	ncit:C102881	THIOUREIDOBUTYRONITRILE	FALSE	FALSE	FALSE
NCBIGENE:2983	hgnc:4687	GUCY1B1	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:11589	iuphar.ligand:11589	COMPOUND 20C [PMID: 34181850]	FALSE	FALSE	FALSE
NCBIGENE:2102	hgnc:16870	MELK	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8046	iuphar.ligand:8046	OTSSP167	FALSE	FALSE	FALSE
NCBIGENE:2104	hgnc:3474	ESRRG	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:12385	iuphar.ligand:12385	TINODASERTIB	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.212152207	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:283	hgnc:483	ANG	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:1327	iuphar.ligand:1327	ASIP [90-132 (L89Y)]	FALSE	FALSE	FALSE
NCBIGENE:281	hgnc:479	AMYP1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1290	iuphar.ligand:1290	AC-HMCH-(6-16)-NH2	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6340	iuphar.ligand:6340	CFMMC	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6212	iuphar.ligand:6212	[11C]MMTP	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:1391	iuphar.ligand:1391	[3H]R214127	FALSE	FALSE	FALSE
PROTEIN KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	0.2187819634820604	LY2801653	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1392	iuphar.ligand:1392	(2R,3R)-APDC	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6330	iuphar.ligand:6330	JNJ-40068782	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	modulator	0.4735540335109532	IUPHAR.LIGAND:5665	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:2080	hgnc:6857	MAP3K5	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8076	iuphar.ligand:8076	MSC2032964A	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:5436	iuphar.ligand:5436	BQCA	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	2.282942227638891	G100	drugbank:DB17244	G100	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.276356164	IUPHAR.LIGAND:3262	iuphar.ligand:3262	LY2033298	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:327	iuphar.ligand:327	METHOCTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:7449	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:290	iuphar.ligand:290	MCN-A-343	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:3262	iuphar.ligand:3262	LY2033298	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:326	iuphar.ligand:326	LITHOCHOLYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.049723174	IUPHAR.LIGAND:360	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:328	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:327	iuphar.ligand:327	METHOCTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.066297565	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	BTK inhibitor	ncit:C124801	BTK INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:8583	iuphar.ligand:8583	UH-AH 37	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	1.419126249613364	IUPHAR.LIGAND:7775	iuphar.ligand:7775	2-METHOXY-&ALPHA;,&BETA;-DIDEHYDRO-AGOMELATINE	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:12324	iuphar.ligand:12324	UCM1341	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1620	iuphar.ligand:1620	DYNORPHIN A	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:9006	iuphar.ligand:9006	UFP-512	FALSE	FALSE	FALSE
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	1.009762908	ABBV-257	chembl:CHEMBL4297682	ABBV-257	FALSE	FALSE	FALSE
NCBIGENE:3004	hgnc:4712	GZMM	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9935	iuphar.ligand:9935	GKT136901	FALSE	FALSE	FALSE
NCBIGENE:3001	hgnc:4708	GZMA	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9935	iuphar.ligand:9935	GKT136901	FALSE	FALSE	FALSE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	blocker	0.1750255707856483	IUPHAR.LIGAND:2616	iuphar.ligand:2616	TETRODOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:12643	iuphar.ligand:12643	RELUTRIGINE	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:12643	iuphar.ligand:12643	RELUTRIGINE	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:2616	iuphar.ligand:2616	TETRODOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:585	hgnc:969	BBS4	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:11864	iuphar.ligand:11864	PF-04885614	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	activator	0.1250182648468916	IUPHAR.LIGAND:2619	iuphar.ligand:2619	BATRACHOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:5731	iuphar.ligand:5731	PYRROLOPYRIMIDINE 48 [PMID: 22318156]	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.6482428547616604	GSK3179106	chembl:CHEMBL3355009	GSK-3179106	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:12643	iuphar.ligand:12643	RELUTRIGINE	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	blocker	0.9376369863516875	IUPHAR.LIGAND:3963	ncit:C75979	HEXAMETHONIUM	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:3998	iuphar.ligand:3998	PHA-543613	FALSE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:2125	iuphar.ligand:2125	PD157672	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1474	iuphar.ligand:1474	[125I]NEUROMEDIN U-25 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1470	iuphar.ligand:1470	NEUROMEDIN U-25	FALSE	FALSE	FALSE
MUCOSAL ADDRESSIN CELL ADHESION MOLECULE 1	hgnc:6765	MADCAM1	TTD	2020.06.01	NULL	17.50255707856483	SHP647	iuphar.ligand:9340	ONTAMALIMAB	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	inhibitor	0.076098074	IUPHAR.LIGAND:4844	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	inhibitor	0.1909369863116163	IUPHAR.LIGAND:4743	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	inhibitor	0.1909369863116163	IUPHAR.LIGAND:4743	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	NULL	2.100306849	IUPHAR.LIGAND:4765	iuphar.ligand:4765	[3H]CCK-8 (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2243	iuphar.ligand:2243	L-366,682	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2256	iuphar.ligand:2256	[MPA1,D-TYR(ET)2,D-TIC7]OT	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1752	iuphar.ligand:1752	MRS2567	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6078	ncit:C77947	BEPAFANT	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2259	iuphar.ligand:2259	RO 25-1553	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	1.235474617310458	CX-072	ncit:C132192	PACMILIMAB	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:12492	iuphar.ligand:12492	ISOX-CHA-CHG-ALA-ARG-DPR(4FB)-NH2	FALSE	FALSE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	NULL	1.346350544504987	IUPHAR.LIGAND:4659	iuphar.ligand:4659	[3H]GLYSAR	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:12737	ncit:C166556	LANIFIBRANOR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2692	iuphar.ligand:2692	15-DEOXY-&DELTA;-12,14-PROSTAGLANDIN J2	FALSE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	5.250767123569449	MB-102	ncit:C165435	AUTOLOGOUS CD123CAR-CD28-CD3ZETA-EGFRT-EXPRESSING T LYMPHOCYTES MB-102	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2705	iuphar.ligand:2705	FMOC-L-LEUCINE	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:10489	iuphar.ligand:10489	COMPOUND 12B [PMID: 31465220]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.012040282	IUPHAR.LIGAND:7950	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:9571	iuphar.ligand:9571	ECF309	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1966579447029756	IUPHAR.LIGAND:10649	iuphar.ligand:10649	COMPOUND 7 [PMID: 31955578]	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:9636	iuphar.ligand:9636	INAVOLISIB	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	1.117184494376478	RPI-MN	drugbank:DB17957	RPI-MN	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.032055965	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.2949869170544634	IUPHAR.LIGAND:12903	iuphar.ligand:12903	STX-478	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:8918	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:9425	ncit:C174798	NEMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.075768645	IUPHAR.LIGAND:7965	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:10702	iuphar.ligand:10702	COMPOUND 15A [PMID: 32069401]	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.085796848	IUPHAR.LIGAND:8003	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.022062047	IUPHAR.LIGAND:7955	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:10365	iuphar.ligand:10365	COMPOUND 2Q [PMID: 30986068]	FALSE	FALSE	FALSE
NCBIGENE:1311	hgnc:2227	COMP	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:6559	iuphar.ligand:6559	BC11-38	FALSE	FALSE	FALSE
NCBIGENE:1296	hgnc:2216	COL8A2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:5270	iuphar.ligand:5270	SCH51866	FALSE	FALSE	FALSE
NCBIGENE:1297	hgnc:2217	COL9A1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:5147	iuphar.ligand:5147	BAY607550	FALSE	FALSE	FALSE
NCBIGENE:1294	hgnc:2214	COL7A1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:5270	iuphar.ligand:5270	SCH51866	FALSE	FALSE	FALSE
NCBIGENE:1299	hgnc:2219	COL9A3	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:7148	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11865	iuphar.ligand:11865	ENSIFENTRINE	FALSE	FALSE	FALSE
NCBIGENE:1307	hgnc:2193	COL16A1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9659	iuphar.ligand:9659	PF-04957325	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:5270	iuphar.ligand:5270	SCH51866	FALSE	FALSE	FALSE
NCBIGENE:1309	hgnc:8795	PDE9A	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5270	iuphar.ligand:5270	SCH51866	FALSE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:7519	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:2772	iuphar.ligand:2772	(+)-S20	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.027010119	IUPHAR.LIGAND:2770	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	0.1093909817410302	IUPHAR.LIGAND:7335	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1875	iuphar.ligand:1875	[125I]PRRP-20 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1873	iuphar.ligand:1873	PRRP-31	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1791	iuphar.ligand:1791	[125I][NLE8,21,TYR34]PTH-(1-34)-NH2 (RAT)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:4448	rxcui:32915	TERIPARATIDE	TRUE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:1819	iuphar.ligand:1819	[D-TRP12,TYR34]PTH-(7-34) (BOVINE)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1822	iuphar.ligand:1822	PTHRP-(1-34) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:1821	iuphar.ligand:1821	[ILE5,TRP23]PTHRP-(5-36)	FALSE	FALSE	FALSE
NCBIGENE:2143	hgnc:8811	PDK3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9350	iuphar.ligand:9350	VER-246608	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:12351	iuphar.ligand:12351	COMPOUND 14 [SCHNUTE ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9322	rxcui:1992864	NETARSUDIL	TRUE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:11908	iuphar.ligand:11908	H3 AC-B10-27(13-17 HC)	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:6992	iuphar.ligand:6992	VPC03090-P	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:11494	iuphar.ligand:11494	BMS-986104 DERIVATIVE 12	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:12569	iuphar.ligand:12569	ST-2191	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:6992	iuphar.ligand:6992	VPC03090-P	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:9320	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:12573	iuphar.ligand:12573	COMPOUND 15 [PMID: 33738061]	FALSE	FALSE	FALSE
NCBIGENE:2197	hgnc:3597	FAU	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9581	iuphar.ligand:9581	ARN-3236	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:9289	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
NCBIGENE:3103	hgnc:10721	SELP	GuideToPharmacology	2024.1	inhibitor	8.751278539282417	IUPHAR.LIGAND:8307	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.081407242	IUPHAR.LIGAND:201	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:2219	hgnc:3623	FCN1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:2632	hgnc:4180	GBE1	GuideToPharmacology	2024.1	activator	0.3281729452230906	IUPHAR.LIGAND:4214	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
NCBIGENE:2399	hgnc:3910	FRA5F	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:7897	iuphar.ligand:7897	BPTI-K15R/R17G	FALSE	FALSE	FALSE
NCBIGENE:2553	hgnc:4074	GABPB1	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:6681	iuphar.ligand:6681	PB-28	FALSE	FALSE	FALSE
NCBIGENE:3096	hgnc:4920	HIVEP1	GuideToPharmacology	2024.1	NULL	3.500511415712966	IUPHAR.LIGAND:12061	iuphar.ligand:12061	BI-3406	FALSE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:8376	rxcui:1992672	ERTUGLIFLOZIN	TRUE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3128	iuphar.ligand:3128	COMPOUND 8 [PMID: 19191557]	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3125	iuphar.ligand:3125	COMPOUND 14 [PMID: 19191557]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2052	iuphar.ligand:2052	NC 8-12	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.086361301	IUPHAR.LIGAND:2018	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:2028	iuphar.ligand:2028	[D-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5642	iuphar.ligand:5642	IN-NODAGATOC	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2792961235941196	IUPHAR.LIGAND:2012	iuphar.ligand:2012	DES-AA5-[D-TRP8]SRIF	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.1595977849109255	IUPHAR.LIGAND:8487	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:2028	iuphar.ligand:2028	[D-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2057	iuphar.ligand:2057	[111IN,90Y]DOTA-NOC	FALSE	FALSE	FALSE
NCBIGENE:2740	hgnc:4324	GLP1R	GuideToPharmacology	2024.1	inhibitor	0.1060761035064535	IUPHAR.LIGAND:12206	iuphar.ligand:12206	GNE-064	FALSE	FALSE	FALSE
NCBIGENE:1885	ncbigene:1885	EBR4	GuideToPharmacology	2024.1	NULL	17.50255707856483	IUPHAR.LIGAND:5069	iuphar.ligand:5069	BAFF	FALSE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:12239	iuphar.ligand:12239	JNJ-64264681	FALSE	FALSE	FALSE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11082	iuphar.ligand:11082	OM-1700	FALSE	FALSE	FALSE
NCBIGENE:1752	hgnc:11848	TLR2	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:9408	iuphar.ligand:9408	TOMARALIMAB	FALSE	FALSE	FALSE
NCBIGENE:1758	hgnc:2932	DMP1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11989	iuphar.ligand:11989	COMPOUND 15 [PMID: 35450354]	FALSE	FALSE	FALSE
NCBIGENE:1752	hgnc:11848	TLR2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:10341	iuphar.ligand:10341	DIPROVOCIM-1	FALSE	FALSE	FALSE
NCBIGENE:2421	hgnc:3931	FRA8C	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11956	iuphar.ligand:11956	N-0385	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.596678082	IUPHAR.LIGAND:10293	iuphar.ligand:10293	POLYGODIAL	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.2075402025126264	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.4102161815288632	IUPHAR.LIGAND:2828	iuphar.ligand:2828	DAIDZEIN	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.043180651	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.7721716358190367	IUPHAR.LIGAND:2436	iuphar.ligand:2436	OAG	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.1544343271638073	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.041672755	IUPHAR.LIGAND:5338	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	activator	4.836232876971861	IUPHAR.LIGAND:2430	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.750109589	IUPHAR.LIGAND:4129	iuphar.ligand:4129	AMG517	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4076	iuphar.ligand:4076	[3H]A778317	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.750109589	IUPHAR.LIGAND:4117	iuphar.ligand:4117	A425619	FALSE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	blocker	0.5966780822238011	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	0.2778183663264258	IUPHAR.LIGAND:6310	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:1836	hgnc:10994	SLC26A2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8135	iuphar.ligand:8135	COMPOUND 21 [PMID: 23312943]	FALSE	FALSE	FALSE
NCBIGENE:2837	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	antibody	1.810609352954982	IUPHAR.LIGAND:12978	iuphar.ligand:12978	HIMB1636-MMAE	FALSE	FALSE	FALSE
NCBIGENE:2272	hgnc:3701	FHIT	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11340	iuphar.ligand:11340	SBP-7455	FALSE	FALSE	FALSE
NCBIGENE:2428	hgnc:3938	FRA9D	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11964	iuphar.ligand:11964	KSQ-4279	FALSE	FALSE	FALSE
NCBIGENE:2273	hgnc:3702	FHL1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8220	iuphar.ligand:8220	COMPOUND 15 [PMID: 24900237]	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:3293	iuphar.ligand:3293	[ARG16]CHICKEN SECRETIN	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:1155	iuphar.ligand:1155	SECRETIN	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1152	iuphar.ligand:1152	VIP	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:1512	iuphar.ligand:1512	PANCREATIC POLYPEPTIDE	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	CIViC	10-Apr-24	NULL	0.2651902587661338	ANTI-PD-L1 MONOCLONAL ANTIBODY	ncit:C128057	ANTI-PD-L1 MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
GROWTH/DIFFERENTIATION FACTOR 2	hgnc:4217	GDF2	TTD	2020.06.01	NULL	1.093909817410302	ACE-041	ncit:C88296	DALANTERCEPT	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.00172405	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
TLK2	hgnc:11842	TLK2	CIViC	10-Apr-24	NULL	NULL	GO6983	NULL	NULL	NULL	NULL	NULL
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	1.322135606654178	ASCIMINIB	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
FN1	hgnc:3778	FN1	CIViC	10-Apr-24	NULL	8.078103267029922	L19IL2	chembl:CHEMBL2109608	L19IL2	FALSE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.012430793	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.4579157375205915	DERAZANTINIB	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	CIViC	10-Apr-24	NULL	0.3846715841442821	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.01535312	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
MBD4	hgnc:6919	MBD4	CIViC	10-Apr-24	NULL	26.25383561784724	PD1 INHIBITOR	ncit:C124946	PD1 INHIBITOR	FALSE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	CIViC	10-Apr-24	NULL	0.055329474	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	NULL	R3MAB	NULL	NULL	NULL	NULL	NULL
H3C2	hgnc:4776	H3C2	CIViC	10-Apr-24	NULL	17.50255707856483	AKT/ERK INHIBITOR ONC201	ncit:C113792	DORDAVIPRONE	FALSE	FALSE	TRUE
ERCC2	hgnc:3434	ERCC2	CIViC	10-Apr-24	NULL	0.054243462	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	RG5	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1565212775308858	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.1984416902331613	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.228073862	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.020158043	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NBN	hgnc:7652	NBN	CIViC	10-Apr-24	NULL	NULL	GPI-15427	NULL	NULL	NULL	NULL	NULL
ASS1	hgnc:758	ASS1	CIViC	10-Apr-24	NULL	0.017363648	TAXOL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.022466607	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
GNAQ	hgnc:4390	GNAQ	CIViC	10-Apr-24	NULL	2.625383561784725	SOTRASTAURIN ACETATE	ncit:C80631	SOTRASTAURIN ACETATE	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	NULL	GSK321	NULL	NULL	NULL	NULL	NULL
NT5C2	hgnc:8022	NT5C2	CIViC	10-Apr-24	NULL	4.375639269641208	NELARABINE	rxcui:274771	NELARABINE	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	CIViC	10-Apr-24	NULL	NULL	DVP REGMEN	NULL	NULL	NULL	NULL	NULL
DRD5	hgnc:3026	DRD5	CIViC	10-Apr-24	NULL	0.8751278539282416	AKT/ERK INHIBITOR ONC201	ncit:C113792	DORDAVIPRONE	FALSE	FALSE	TRUE
SMO	hgnc:11119	SMO	DoCM	10-Apr-24	NULL	15.31473744374422	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	1.544343271638073	AZD8329	iuphar.ligand:7715	AZD8329	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	DoCM	10-Apr-24	NULL	1.494525746746522	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	DoCM	10-Apr-24	NULL	0.057841988	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	CEP-28122	NULL	NULL	NULL	NULL	NULL
MAPK-ACTIVATED PROTEIN KINASE 2	hgnc:6887	MAPKAPK2	TTD	2020.06.01	NULL	4.375639269641208	CBP-501	drugbank:DB17277	CBP-501	FALSE	FALSE	FALSE
GNA11	hgnc:4379	GNA11	DoCM	10-Apr-24	NULL	1.750255707856483	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
HERC2	hgnc:4868	HERC2	DoCM	10-Apr-24	NULL	7.501095890813499	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	G007-LK	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.008153365	Methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1141471113819445	Filgotinib	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.010618336	Dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1826353782111113	Milademetan	ncit:C141432	MILADEMETAN	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	CGP049090	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	RM-018	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	Trifluridine-tipiracil hydrochloride	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.023905154	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	UNC2025	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	TGX-221	iuphar.ligand:8244	TGX-221	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.030545475	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	WEHI-539	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.1060761035064535	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	NVP-TNKS656	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	NULL	CEP-28122	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	NULL	XMU-MP-5	NULL	NULL	NULL	NULL	NULL
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.2853677784548614	Filgotinib	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	5.527123287967842	RP-6306	chembl:CHEMBL5095288	RP-6306	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.167488584	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.1004931506903244	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.2631963470460877	Entinostat	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.075496292	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	0.6731752722524935	PLX7486	iuphar.ligand:9104	PLX7486	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	1.831662950082366	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	1.050153425	Telaglenastat	ncit:C114381	TELAGLENASTAT	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.010569177	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	SEL201	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	G007-LK	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	DCC-3009	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.01562031	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.1725334213659184	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.2083637747448194	Encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.2344092465879218	I-BET151	iuphar.ligand:7518	I-BET151	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.1875273972703375	Ulixertinib	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	NULL	AQ-101	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	2.282942227638891	AZD-2423	iuphar.ligand:7825	AZD2423	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	NULL	YF438	NULL	NULL	NULL	NULL	NULL
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.33338204	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.1250182648468916	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.072026984	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.3241214273808303	Tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.054020238	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.071148606	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	2.812910959055062	Dostarlimab-gxly	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.060772768	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.094099769	Tivozanib	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1	hgnc:2357	CRHR1	TTD	2020.06.01	NULL	2.917092846427472	GSK561679	ncit:C152869	VERUCERFONT	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1176247115494948	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	Ulixertinib	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	UNC2025	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	ERAS-007	ncit:C150248	ERK1/2 INHIBITOR ERAS-007	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.065145994	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.013505059	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.038382801	PI-103	drugbank:DB17046	PI-103	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.032412143	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	0.2625383561784725	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	0.2187819634820604	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1419126249613365	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.078840347	Idelalisib	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	WEHI-539	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.053217234	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.078840347	Encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	RER	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.8468979231563628	GSK1014802	iuphar.ligand:12645	VIXOTRIGINE	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	DHM25	NULL	NULL	NULL	NULL	NULL
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	1.166837138570988	Belzutifan	rxcui:2567226	BELZUTIFAN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CancerCommons	25-Jul-13	inhibitor	0.1657439117288336	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	CancerCommons	25-Jul-13	inhibitor	0.1232574442152452	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.2890330526735477	ALVIMOPAN	rxcui:1516803	ALVIMOPAN ANHYDROUS	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.1226814748497534	Sulfatinib	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	VILANTEROL TRIFENATATE	rxcui:1424883	VILANTEROL TRIFENATATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	ANTHRANILIC ACID	drugbank:DB04166	ANTHRANILIC ACID	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.010685322	melphalan	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	0.1666910197958555	melphalan	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
ALOX5	hgnc:435	ALOX5	PharmGKB	4/5/24	NULL	0.1403948428761885	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.210030685	ropivacaine	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	4.375639269641208	Yttrium (90Y) clivatuzumab tetraxetan	iuphar.ligand:8087	YTTRIUM (90Y) CLIVATUZUMAB TETRAXETAN	FALSE	FALSE	FALSE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.2442217266776488	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.021846337	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE RAF	hgnc:18513	ZHX2	TTD	2020.06.01	NULL	1.166837138570989	LY3009120	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.4636438961209227	APR-246	ncit:C85465	EPRENETAPOPT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:84	rxcui:21877	CYAMEMAZINE	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:8644	iuphar.ligand:8644	GSK1511931	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.4730420832044549	IUPHAR.LIGAND:12766	ncit:C171708	TOLUDESVENLAFAXINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	DNDI1417413	chembl:CHEMBL1343568	CHEMBL:CHEMBL1343568	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	0.6977763619361395	ACY-1215	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	GNF-PF-2335	chembl:CHEMBL601146	CHEMBL:CHEMBL601146	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	HALOPROGIN	rxcui:26422	HALOPROGIN	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.015534814	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.596678082	TOCAINIDE	rxcui:42359	TOCAINIDE	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.081281225	Adinazolam	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P04049	hgnc:9829	RAF1	TEND	1-Aug-11	NULL	0.159436249	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4604	iuphar.ligand:4603	[3H]N-METHYL-SSR504734	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9610	iuphar.ligand:9610	CBS-3595	FALSE	FALSE	FALSE
HISTAMINE N-METHYLTRANSFERASE	hgnc:5028	HNMT	TTD	2020.06.01	NULL	0.9376369863516875	Diphenhydramine	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:8591	iuphar.ligand:8591	ML381	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	CIViC	10-Apr-24	NULL	0.002861765	SAPANISERTIB	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
ATP1B1	hgnc:804	ATP1B1	ChEMBL	33	inhibitor	0.3070624048871023	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.029106248	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.596678082	MK-0873	drugbank:DB13029	MK-0873	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Cinoxacin	rxcui:2550	CINOXACIN	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	AZD-3759	drugbank:DB14795	AZD-3759	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.1346350544504987	BUCINDOLOL HYDROCHLORIDE	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
ACO1	hgnc:117	ACO1	NCI	14-Sep-17	NULL	2.333674277141977	N-ACETYLCYSTEINE	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	CIViC	10-Apr-24	NULL	1.184383561707394	BIRABRESIB	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	inhibitor	0.5000730593875666	CARTEOLOL HYDROCHLORIDE	rxcui:142132	CARTEOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	1.123158743009508	Tazarotene	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
NCBIGENE:1359	hgnc:2298	CPA3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8871	iuphar.ligand:8871	(2S,4S)-KETOCONAZOLE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.055271233	IUPHAR.LIGAND:286	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:9253	iuphar.ligand:9253	PEPTIDE 30 [PMID: 27019010]	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.049337723	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.027177884	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	CAULIBUGULONE B	chembl:CHEMBL508779	CAULIBUGULONE B	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	6-BENZYLAMINOPURINE	chembl:CHEMBL228862	6-BENZYLAMINOPURINE	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	0.085796848	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	GNF-PF-4516	chembl:CHEMBL586029	CHEMBL:CHEMBL586029	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.014832675	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.099446347	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.05814803	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	5.834185692854944	SB-649868	drugbank:DB14822	SB-649868	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.1831662950082366	Oxymetazoline	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:9636	iuphar.ligand:9636	INAVOLISIB	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	OLEAMIDE	iuphar.ligand:284	OLEAMIDE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.040235763	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:426	ncit:C87285	METRIFUDIL	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	PYRAZOLOACRIDINE	ncit:C1564	PYRAZOLOACRIDINE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.525076712	Articaine	rxcui:592464	ARTICAINE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	13.12691780892362	CP-461	chembl:CHEMBL4068108	CP-461	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	ChEMBL	33	inhibitor	1.154014752432846	BIRABRESIB	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.032899543	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.1973972602845657	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	(-)-DEMECOLCINE	ncit:C419	DEMECOLCINE	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2917092846427472	DICHLON	chembl:CHEMBL318782	DICHLON	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.021933029	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
MAPK/ERK KINASE KINASE 1	hgnc:6848	MAP3K1	TTD	2020.06.01	NULL	0.3241214273808303	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	Tafluposide	ncit:C152490	TAFLUPOSIDE	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.3387591692625452	Permethrin	rxcui:33199	PERMETHRIN	TRUE	FALSE	FALSE
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A	hgnc:7943	NPR1	TTD	2020.06.01	NULL	4.039051633514961	Nesiritide	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR BETA-2	hgnc:4082	GABRB2	TTD	2020.06.01	NULL	0.05814803	ALLOPREGNANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	3.750547945	calcium	rxcui:1895	CALCIUM	TRUE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-2	hgnc:4087	GABRG2	TTD	2020.06.01	NULL	0.059532507	ALLOPREGNANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
UNIPROT:P29279	hgnc:2500	CCN2	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	FG-3019	ncit:C92577	PAMREVLUMAB	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.2625383561784725	IUPHAR.LIGAND:2012	iuphar.ligand:2012	DES-AA5-[D-TRP8]SRIF	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.021440454	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.045461187	Pramlintide	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.5625821918110124	ACIVICIN	ncit:C986	ACIVICIN	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1458546423213736	NORETHISTERONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
CHST3	hgnc:1971	CHST3	PharmGKB	4/5/24	NULL	0.6326225450083675	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NALCN	hgnc:19082	NALCN	PharmGKB	4/5/24	NULL	1.693795846312725	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.009368006	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
RIBOSOMAL PROTEIN S6 KINASE ALPHA-2	hgnc:10432	RPS6KA3	TTD	2020.06.01	NULL	0.2143170254518142	BI-D1870	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	PharmGKB	4/5/24	NULL	0.1842374429322613	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	1.009762908	flurbiprofen	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.358239472	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.1346350544504987	PQR309	ncit:C111898	BIMIRALISIB	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	0.364636606	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.6563458904461813	IUPHAR.LIGAND:4177	iuphar.ligand:4177	DIDS	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6111	iuphar.ligand:6111	GAL-B2-C8	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.3968833804663227	HKI-272	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
NCBIGENE:1762	hgnc:2936	DMWD	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:5021	iuphar.ligand:5021	MESO-DAP	FALSE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.1166837138570989	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
INTERFERON-GAMMA	hgnc:5438	IFNG	TTD	2020.06.01	NULL	0.4688184931758437	Emapalumab	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.084689792	Phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.3500511415712966	LACTULOSE	rxcui:6218	LACTULOSE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.182318303	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	0.546954909	IUPHAR.LIGAND:2308	iuphar.ligand:2308	NS1643	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	RMC-5552	iuphar.ligand:12338	RMC-5552	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.2059124362184098	Felodipine	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1111665587205952	OXYCODONE HYDROCHLORIDE	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.024709492	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1389091831632129	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
ROTAMASE A	hgnc:9253	PPIA	TTD	2020.06.01	NULL	3.750547945	L-Proline	rxcui:8737	PROLINE	TRUE	FALSE	FALSE
ILF3	hgnc:6038	ILF3	NCI	14-Sep-17	NULL	0.6035364509849942	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.02234369	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.5556367326528519	RO5083945	chembl:CHEMBL2109389	IMGATUZUMAB	FALSE	TRUE	TRUE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	BI-836858	drugbank:DB17267	BI-836858	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.04907259	Ethinyl Estradiol	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.090530468	Novobiocin	rxcui:7538	NOVOBIOCIN	FALSE	FALSE	FALSE
NCBIGENE:1275	ncbigene:1275	COD2	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8779	iuphar.ligand:8779	COMPOUND 10H [PMID: 20832306]	FALSE	FALSE	FALSE
NCBIGENE:2739	hgnc:4323	GLO1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12206	iuphar.ligand:12206	GNE-064	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DINITRO CRESOL	chembl:CHEMBL419564	DINITRO CRESOL	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.1562728310586145	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.1416573864272333	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
GRM4	hgnc:4596	GRM4	DTC	9/2/20	NULL	7.501095891	N-(3,4-DICHLOROPHENYL)PICOLINAMIDE	chembl:CHEMBL549330	CHEMBL:CHEMBL549330	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.01535312	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	OncoKB	23-Jul-20	NULL	0.1154860804304131	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PRKCE	hgnc:9401	PRKCE	PharmGKB	4/5/24	NULL	0.046059361	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.068191781	DIDANOSINE	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	0.364636606	Tonapofylline	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	ChEMBL	33	inhibitor	0.5087952639117684	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.5834185692854945	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:322	iuphar.ligand:322	HEXAHYDRODIFENIDOL	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	TCMDC-124746	chembl:CHEMBL524407	CHEMBL:CHEMBL524407	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	OncoKB	23-Jul-20	NULL	0.029416062	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.059667808	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.048083948	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
MEK1	hgnc:6840	MAP2K1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4735540335109532	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	5.250767123569449	LGD-6972	drugbank:DB14779	LGD-6972	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	1.875273972703375	BCI-838	chembl:CHEMBL4594408	MGS-0210	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	0.3547815624033412	LY2780301	ncit:C95737	AKT INHIBITOR LY2780301	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.048083948	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.084553416	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.020575106	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1500219178162699	SJ000071854	chembl:CHEMBL602127	CHEMBL:CHEMBL602127	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.026789628	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.033295923	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	2.763561643983921	SCH-900776	chembl:CHEMBL2386889	SCH-900776	FALSE	FALSE	FALSE
INFLAMMATION PATHOGENESIS	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	26.25383561784724	HMPL-004	chembl:CHEMBL186141	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
GLUCOSYLCERAMIDASE	hgnc:4177	GBA1	TTD	2020.06.01	NULL	3.000438356	Velaglucerase alfa	rxcui:901805	VELAGLUCERASE ALFA	TRUE	FALSE	FALSE
PIP4K2A	hgnc:8997	PIP4K2A	DTC	9/2/20	NULL	2.625383561784724	SJ000201788	chembl:CHEMBL602923	CHEMBL:CHEMBL602923	FALSE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	DTC	9/2/20	NULL	2.187819634820604	LY-411575	chembl:CHEMBL392068	CHEMBL:CHEMBL392068	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.3088686543276147	Pidilizumab	ncit:C71014	PIDILIZUMAB	FALSE	TRUE	TRUE
CD40	hgnc:11919	CD40	ChEMBL	33	agonist	4.375639269641208	SOTIGALIMAB	ncit:C123734	SOTIGALIMAB	FALSE	FALSE	FALSE
TRBV7-9	hgnc:12243	TRBV7-9	ChEMBL	33	inhibitor	3.500511415712967	TOL-101	drugbank:DB16980	TOL-101	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	SJ000001592	chembl:CHEMBL591834	CHEMBL:CHEMBL591834	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	DNDI1417025	chembl:CHEMBL1320453	CHEMBL:CHEMBL1320453	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.100976291	BGT226	ncit:C74073	PI3K INHIBITOR BGT226	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.007406922	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10343	iuphar.ligand:10343	GSK8612	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:1998	iuphar.ligand:1998	R3/I5	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	DNDI1417234	chembl:CHEMBL2094549	CHEMBL:CHEMBL2094549	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	2.972132334095915	CIXUTUMUMAB	ncit:C79828	CIXUTUMUMAB	FALSE	TRUE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	3.500511415712966	MEDI-3617	chembl:CHEMBL2109298	MEDI-3617	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.032055965	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002796829	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.024354207	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	NSC-327705	chembl:CHEMBL1317986	CHEMBL:CHEMBL1317986	FALSE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE	hgnc:1189	AHSA1	TTD	2020.06.01	NULL	1.250182648468916	GSK2269557	ncit:C174798	NEMIRALISIB	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1363835616511545	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
GPX3	hgnc:4555	GPX3	PharmGKB	4/5/24	NULL	0.2885036881082115	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.093596562	liothyronine	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1962903597596056	Chlorotrianisene	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.1620607136904151	Minoxidil	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.2734774543525755	PI3KBETA INHIBITOR AZD8186	ncit:C107684	PI3KBETA INHIBITOR AZD8186	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.3454452054979901	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.055271233	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	METHIDATHION	ncit:C163672	METHIDATHION	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1286952726365061	PALMITOYL-CARNITINE	chembl:CHEMBL301722	PALMITOYL-CARNITINE	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.4118248724368196	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.1271372184883643	IUPHAR.LIGAND:5979	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.017751072	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	CICLOPIROX OLAMINE	rxcui:52172	CICLOPIROX OLAMINE	TRUE	FALSE	FALSE
DEFA4	hgnc:2763	DEFA4	NCI	14-Sep-17	NULL	4.039051633514962	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.276356164	IUPHAR.LIGAND:8598	iuphar.ligand:8598	CY3B-TELENZEPINE	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.048083948	IUPHAR.LIGAND:7794	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:11940	iuphar.ligand:11940	MAP855	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.025865848	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.023274677	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.1544343271638073	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.034590034	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	INDOLE-3-CARBINOL	rxcui:2598119	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.1495945049449985	SCUTELLARIN	iuphar.ligand:13075	SCUTELLARIN	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.041672755	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
COL1A1	hgnc:2197	COL1A1	PharmGKB	4/5/24	NULL	1.071585127259071	etidronic acid	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.057700738	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
SPG7	hgnc:11237	SPG7	PharmGKB	4/5/24	NULL	0.6326225450083675	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:2443	hgnc:3841	FRA11F	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11488	ncit:C90673	ZAURATEGRAST	FALSE	FALSE	FALSE
NDUFAF2	hgnc:28086	NDUFAF2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.089298761	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.182318303	STEPHOLIDINE	iuphar.ligand:8370	(-)-STEPHOLIDINE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.030598876	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.024008995	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	PharmGKB	4/5/24	NULL	1.944728564284981	botulinum toxin type a	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
VEGFC	hgnc:12682	VEGFC	PharmGKB	4/5/24	NULL	3.889457128569962	uric acid	rxcui:1427088	URIC ACID	FALSE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	PharmGKB	4/5/24	NULL	1.166837138570988	esomeprazole	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.2442217266776488	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:157	iuphar.ligand:157	(R)-DOI	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.1132444383228493	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.089298761	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:6698	iuphar.ligand:6698	PF0998425	FALSE	FALSE	FALSE
NCBIGENE:720	hgnc:1323	C4A	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.2027323213733378	IUPHAR.LIGAND:1346	iuphar.ligand:1346	6-CL-MLT	FALSE	FALSE	FALSE
BCR	hgnc:1014	BCR	TALC	12-May-16	inhibitor	0.1298891063344329	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	inhibitor	0.1615620653405984	IUPHAR.LIGAND:3439	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
UNIPROT:P47872	hgnc:10608	SCTR	TEND	1-Aug-11	NULL	15.75230137070834	SECRETIN	rxcui:9627	SECRETIN	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.2408608772279564	MEPTAZINOL	rxcui:6761	MEPTAZINOL	TRUE	FALSE	FALSE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TEND	1-Aug-11	NULL	0.4023576339899962	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.078136416	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
LEUKOTRIENE CYSLT2 RECEPTOR	hgnc:18274	CYSLTR2	TTD	2020.06.01	NULL	26.25383561784724	BAY-X-7195	chembl:CHEMBL314115	CHEMBL:CHEMBL314115	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.09745299	NANDROLONE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.28382525	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	FDA	10-Apr-24	NULL	0.4605936073306534	Lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	CHRYSOPHANOL	chembl:CHEMBL41092	CHRYSOPHANOL	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.042174836	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	1.009762908	CINACIGUAT	ncit:C87280	CINACIGUAT	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005412046	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.010819631	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.2885036881082115	GNF-PF-4085	chembl:CHEMBL528181	CHEMBL:CHEMBL528181	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.087222045	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.1000146118775133	ETHER	ncit:C29819	ETHER	FALSE	FALSE	FALSE
INTERLEUKIN 15 RECEPTOR ALPHA	hgnc:5978	IL15RA	TTD	2020.06.01	NULL	13.12691780892362	ALT-803	iuphar.ligand:9615	ALT-803	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.1250182648468916	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.325124899	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.073403082	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:3950	ncit:C73038	SITAXENTAN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	LAPACHOL	chembl:CHEMBL15193	LAPACHOL	FALSE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	ChEMBL	33	blocker	0.058212496	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
RPS21	hgnc:10409	RPS21	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:4040	iuphar.ligand:4040	ER819762	FALSE	FALSE	FALSE
KCNK2	hgnc:6277	KCNK2	ChEMBL	33	potentiator	0.2419708351875322	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.032899543	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
PSMA5	hgnc:9534	PSMA5	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	GNF-PF-2776	chembl:CHEMBL578294	CHEMBL:CHEMBL578294	FALSE	FALSE	FALSE
FASTKD3	hgnc:28758	FASTKD3	PharmGKB	4/5/24	NULL	0.9460841664089098	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003566492	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.8334550989792776	glucose	rxcui:349730	ANHYDROUS DEXTROSE	TRUE	FALSE	FALSE
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.012185582	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:Q14432	hgnc:8778	PDE3A	TEND	1-Aug-11	NULL	1.591141552596802	ENOXIMONE	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.054187483	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	4.375639269641208	JNJ-479655	iuphar.ligand:7538	JNJ-47965567	FALSE	FALSE	FALSE
NCBIGENE:2991	ncbigene:2991	GUSM	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:9833	iuphar.ligand:9833	BSAB (CD89-CD20)	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6450	iuphar.ligand:6450	COMPOUND 10 [PMID: 15482906]	FALSE	FALSE	FALSE
NCBIGENE:1216	hgnc:25588	SLC47A1	GuideToPharmacology	2024.1	NULL	0.5385402178019948	IUPHAR.LIGAND:4503	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	agonist	0.040021091	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	DNDI1417215	chembl:CHEMBL1390650	CHEMBL:CHEMBL1390650	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.2524407270946851	OXYTOCIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.010939098	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6100	iuphar.ligand:6100	M617	FALSE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:12661	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	CIViC	10-Apr-24	NULL	0.046965717	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MT-ND4	hgnc:7459	MT-ND4	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:4513	iuphar.ligand:4513	NBTGR	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.086361301	IUPHAR.LIGAND:5933	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
DCK	hgnc:2704	DCK	NCI	14-Sep-17	NULL	0.760980743	2,3-DIDEOXYADENOSINE	ncit:C429	DIDEOXYADENOSINE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	NCI	14-Sep-17	NULL	0.031822831	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.1396480617970598	CARISOPRODOL	rxcui:2101	CARISOPRODOL	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.3500511415712966	DIFLUBENZURON	rxcui:1665336	DIFLUBENZURON	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6258	iuphar.ligand:6258	4-APPES	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2272	iuphar.ligand:2272	PG 99-465	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2272	iuphar.ligand:2272	PG 99-465	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.013890918	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.095122593	NICOTINE GUM	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
RXRB	hgnc:10478	RXRB	ChEMBL	33	agonist	1.944728564284981	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	GSK2140944	ncit:C170025	GEPOTIDACIN	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.2333674277141977	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.2734774543525755	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
UNIPROT:P11168	hgnc:11006	SLC2A2	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9359	iuphar.ligand:9359	CP466722	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	TRIAMCINOLONE HEXACETONIDE	rxcui:38546	TRIAMCINOLONE HEXACETONIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.093763699	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.3059887601147698	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	0.1298891063344329	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2035181055647073	RIMITEROL	rxcui:9388	RIMITEROL	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.08334551	IUPHAR.LIGAND:161	iuphar.ligand:161	BW723C86	FALSE	FALSE	FALSE
UNIPROT:P42263	hgnc:4573	GRIA3	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	TALAMPANEL	ncit:C38139	TALAMPANEL	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:931	iuphar.ligand:931	ANTISAUVAGINE	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:1885	iuphar.ligand:1885	PGJ2	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5747	iuphar.ligand:5747	COMPOUND 36 [PMID: 21273063]	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	NULL	0.1037701012563132	IUPHAR.LIGAND:5089	iuphar.ligand:5089	VEGFE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	2.763561643983921	N9-GP	rxcui:1990855	COAGULATION FACTOR IX (RECOMBINANT), GLYCOPEGYLATED	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.169927739	CAULIBUGULONE B	chembl:CHEMBL508779	CAULIBUGULONE B	FALSE	FALSE	FALSE
NFATC2	hgnc:7776	NFATC2	PharmGKB	4/5/24	NULL	0.9723642821424908	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	CARBARIL	ncit:C76389	CARBARIL	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	1.944728564284981	NS-8	chembl:CHEMBL42661	CHEMBL:CHEMBL42661	FALSE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TEND	1-Aug-11	NULL	0.305277158	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	THIOLUTIN	ncit:C64175	THIOLUTIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	QUERCETIN DIHYDRATE	ncit:C75768	QUERCETIN DIHYDRATE	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	2.100306849	ASN06356088	chembl:CHEMBL1290361	ASN06356088	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	1.419126249613364	V81444	ncit:C125659	CIFORADENANT	FALSE	FALSE	FALSE
HOXC10	hgnc:5122	HOXC10	CIViC	10-Apr-24	NULL	1.312691780892362	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.7395446652914718	CEFATRIZINE	rxcui:2179	CEFATRIZINE	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	MyCancerGenome	20-Jun-17	other/unknown	0.5966780822238011	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.08780547	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.028413242	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2098	iuphar.ligand:2098	SUBSTANCE P	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.031765076	IUPHAR.LIGAND:7216	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.760980743	IUPHAR.LIGAND:2438	iuphar.ligand:2438	BTP2	FALSE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TEND	1-Aug-11	NULL	0.7143900848393808	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:1924	iuphar.ligand:1924	SC-51322	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:1733	iuphar.ligand:1733	MRS2698	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9919	iuphar.ligand:9919	SELATINIB	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	1.479089330582943	12-EPI-SALVINORIN A	chembl:CHEMBL458235	12-EPI-SALVINORIN A	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
NCBIGENE:1232	hgnc:1604	CCR3	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:5092	iuphar.ligand:5092	&ALPHA;&BETA;-METHYLENEADP	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9768	ncit:C120102	ROBLITINIB	FALSE	FALSE	FALSE
NCBIGENE:925	hgnc:1706	CD8A	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:4757	iuphar.ligand:4757	PHLORIZIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	DNDI1417155	chembl:CHEMBL1548739	CHEMBL:CHEMBL1548739	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.3125456621172291	METHYSERGIDE MALEATE	rxcui:203190	METHYSERGIDE MALEATE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	2.212697851403848	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.061055432	TCMDC-125185	chembl:CHEMBL580819	CHEMBL:CHEMBL580819	FALSE	FALSE	FALSE
GDNF	hgnc:4232	GDNF	NCI	14-Sep-17	NULL	0.351221881	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.0191914	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
MONOCYTE CHEMOTACTIC AND ACTIVATING FACTOR	hgnc:10618	CCL2	TTD	2020.06.01	NULL	17.50255707856483	Carlumab	ncit:C71010	CARLUMAB	FALSE	FALSE	FALSE
UGT1A	hgnc:12529	UGT1A	CIViC	10-Apr-24	NULL	1.640864726115453	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	CGI	2/1/22	NULL	0.6471533709721451	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.5321723436050118	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1591141552596802	IBUFENAC	ncit:C96750	IBUFENAC	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.027121731	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1448	iuphar.ligand:1448	ME4	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.032817295	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	0.2333674277141978	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.1108075556053025	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	MEDRYSONE	rxcui:29439	MEDRYSONE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.009702083	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	0.6177373086552295	EPOETIN BETA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
LPAR5	hgnc:13307	LPAR5	DTC	9/2/20	NULL	52.50767123569449	(S)-CARBA CYCLIC-PHOSPHATIDIC ACID	chembl:CHEMBL1630084	CHEMBL:CHEMBL1630084	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	GNF-PF-860	chembl:CHEMBL593254	CHEMBL:CHEMBL593254	FALSE	FALSE	FALSE
ERAP2	hgnc:29499	ERAP2	DTC	9/2/20	NULL	1.458546423213736	SCOPOLETIN	chembl:CHEMBL71851	SCOPOLETIN	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	6.300920548	TG-0054	ncit:C88323	BURIXAFOR	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.05486695	IUPHAR.LIGAND:384	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:6893	iuphar.ligand:6893	NOVOKININ	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	0.2075402025126264	IUPHAR.LIGAND:5668	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	MMV007764	chembl:CHEMBL609628	CHEMBL:CHEMBL609628	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.064111931	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.07631929	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.087222045	IUPHAR.LIGAND:8918	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.073954467	SJ000089001	chembl:CHEMBL591618	CHEMBL:CHEMBL591618	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	PharmGKB	4/5/24	NULL	0.006353015	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.182318303	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.3571950424196904	BIRABRESIB	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	SULFADOXINE	rxcui:10173	SULFADOXINE	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:535	rxcui:3616	DOBUTAMINE	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:2110	ncit:C170264	OSANETANT	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.000146118775133	Beperminogene perplasmid	chembl:CHEMBL2108332	BEPERMINOGENE PERPLASMID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.7721716358190367	PIDNARULEX	ncit:C126798	PIDNARULEX	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
NDUFA1	hgnc:7683	NDUFA1	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	0.6250913242344582	PF-05241328	drugbank:DB15124	PF-05241328	FALSE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	modulator	0.1458546423213736	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	1.040600372117402	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:245	ncit:C152942	ZACOPRIDE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.019889269	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	ALEXIDINE DIHYDROCHLORIDE	chembl:CHEMBL554041	ALEXIDINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TEND	1-Aug-11	NULL	0.3394892536790592	INTERFERON ALFA-2A, RECOMBINANT	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.2083637747448194	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.008152099	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.272767123	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:9522	iuphar.ligand:9522	TP-472	FALSE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	2.917092846427472	BMS-753493	chembl:CHEMBL4297749	EPOFOLATE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4299	iuphar.ligand:4299	RO4938581	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:4344	iuphar.ligand:4344	XESTOSPONGIN C	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	ASTX029	iuphar.ligand:11727	ASTX029	FALSE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	0.074797252	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.2263261691193728	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	PharmGKB	4/5/24	NULL	0.159436249	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.3571950424196904	HMBA	ncit:C1125	HEXAMETHYLENE BISACETAMIDE	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	0.1767935058440892	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.3804903712731485	ezetimibe	rxcui:341248	EZETIMIBE	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.7955707762984014	NITROBLUE TETRAZOLIUM	chembl:CHEMBL1185260	NITROBLUE TETRAZOLIUM	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.048618214	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
JUN N TERMINAL KINASE	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	0.3431873936973496	CC-930	ncit:C152510	TANZISERTIB	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.032173818	IUPHAR.LIGAND:221	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.013313304	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:12513	iuphar.ligand:12513	BM213	FALSE	FALSE	FALSE
PXN	hgnc:9718	PXN	DTC	9/2/20	NULL	13.12691780892362	1,2,4,5-BENZENETETRAAMINE TETRAHYDROCHLORIDE	chembl:CHEMBL456559	CHEMBL:CHEMBL456559	FALSE	FALSE	FALSE
CHLORIDE CHANNEL UNSPECIFIC	hgnc:2014	CLC	TTD	2020.06.01	NULL	13.12691780892362	TM-601	drugbank:DB15210	CHLOROTOXIN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.037505479	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.2983390411119005	TD-9855	chembl:CHEMBL4297646	AMPRELOXETINE	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.3431873936973496	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.034318739	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
PGP	hgnc:8909	PGP	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2966535098061836	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.036770078	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.059397818	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:7912	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	Olodaterol	rxcui:1546059	OLODATEROL	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2690	iuphar.ligand:2690	L-165461	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.095295229	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	IBI-308	hemonc:61131	SINTILIMAB	FALSE	FALSE	FALSE
FHL2	hgnc:3703	FHL2	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	0.8334550989792777	APG-1387	drugbank:DB16095	APG-1387	FALSE	FALSE	FALSE
TTC37	hgnc:23639	SKIC3	PharmGKB	4/5/24	NULL	4.039051633514962	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.01160647	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.192335792	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DESOXYCORTICOSTERONE	rxcui:3256	DESOXYCORTICOSTERONE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.051177067	FEXOFENADINE HYDROCHLORIDE	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.015662243	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.6482428547616605	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
BRD4	hgnc:13575	BRD4	ChEMBL	33	inhibitor	0.9211872146613068	MOLIBRESIB	ncit:C101538	MOLIBRESIB	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.036847489	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	1.831662950082366	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1610	iuphar.ligand:1610	ETHYLKETOCYCLAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	1.591141552596802	IUPHAR.LIGAND:10302	iuphar.ligand:10302	OSTHOLE	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.043756393	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.2792961235941196	L-METHIONINE-SULFOXIMINE	chembl:CHEMBL1627202	CHEMBL:CHEMBL1627202	FALSE	FALSE	FALSE
OXALOSUCCINATE DECARBOXYLASE	hgnc:5382	IDH1	TTD	2020.06.01	NULL	0.9842513760562132	Ivosidenib	rxcui:2049873	IVOSIDENIB	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	N,N-HEXAMETHYLENEAMILORIDE	iuphar.ligand:1192	5-(N,N-HEXAMETHYLENE)-AMILORIDE	FALSE	FALSE	FALSE
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	8.078103267029922	SGN-70	chembl:CHEMBL2108673	VORSETUZUMAB	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.065716735	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.2983390411119005	IUPHAR.LIGAND:2430	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Pheniramine	rxcui:8132	PHENIRAMINE	TRUE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	2.282942227638891	CeaVac	ncit:C2424	MONOCLONAL ANTIBODY 3H1 ANTI-IDIOTYPE VACCINE	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.2465148884304905	LY-25582	chembl:CHEMBL300662	CHEMBL:CHEMBL300662	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.038693936	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
KIF11	hgnc:6388	KIF11	DTC	9/2/20	NULL	6.563458904461812	NSC-123138	chembl:CHEMBL409102	CHEMBL:CHEMBL409102	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.7225826316838693	DEZOCINE	rxcui:22713	DEZOCINE	TRUE	FALSE	FALSE
GUANYLYL CYCLASE C	hgnc:4688	GUCY2C	TTD	2020.06.01	NULL	19.69037671338543	Linaclotide	rxcui:1307404	LINACLOTIDE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.028413242	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	Carmoxirole	ncit:C81077	CARMOXIROLE	FALSE	FALSE	FALSE
SLC39A6	hgnc:18607	SLC39A6	ChEMBL	33	binder	3.281729452230906	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	1.346350544504987	FELCISETRAG	ncit:C171900	FELCISETRAG	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP1	hgnc:9593	PTGER1	TTD	2020.06.01	NULL	3.750547945	AS-013	chembl:CHEMBL2104574	ECRAPROST	FALSE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	ChEMBL	33	inhibitor	1.591141552596802	PACTIMIBE	ncit:C66290	PACTIMIBE	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.020195258	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P48058	hgnc:4574	GRIA4	TdgClinicalTrial	Jan-14	NULL	1.790034246671403	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
UNIPROT:Q9Y251	hgnc:5164	HPSE	TdgClinicalTrial	Jan-14	NULL	0.091159151	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.2706580991530644	IUPHAR.LIGAND:429	iuphar.ligand:429	MRS1088	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.00809554	IUPHAR.LIGAND:4139	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.3454452054979901	S-222611	chembl:CHEMBL3545200	S-222611	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.1483267549030917	IUPHAR.LIGAND:5947	iuphar.ligand:5947	CDK1/5 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:8870	iuphar.ligand:8870	AT-076	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	0.2430910705356227	IUPHAR.LIGAND:2597	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:9441	iuphar.ligand:9441	UROLININ	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	NSC-45382	chembl:CHEMBL1214274	CHEMBL:CHEMBL1214274	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.315046027	GW501516	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	13.12691780892362	HBV vaccine	wikidata:Q117749	HEPATITIS B VACCINE	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1680	iuphar.ligand:1680	AC-RYYRWK-NH2	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2034	iuphar.ligand:2034	BIM 23030	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	4-HYDROXYEVODIAMINE	chembl:CHEMBL2171794	CHEMBL:CHEMBL2171794	FALSE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	1.334940794127826	Fosinopril	rxcui:50166	FOSINOPRIL	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.073266518	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1389091831632129	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
PROHEPARIN-BINDING EGF-LIKE GROWTH FACTOR	hgnc:3059	HBEGF	TTD	2020.06.01	NULL	3.387591692625451	KHK-2866	chembl:CHEMBL2109437	KHK-2866	FALSE	FALSE	FALSE
RPL23A	hgnc:10317	RPL23A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	inhibitor	2.625383561784724	MK-3577	drugbank:DB14957	MK-3577	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2333674277141978	1207456-01-6	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
PML	hgnc:9113	PML	FDA	10-Apr-24	NULL	0.384671584	Tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	Desirudin Recombinant	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:10387	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.2051080907644316	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.045778266	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	TDR77585	chembl:CHEMBL1333386	CHEMBL:CHEMBL1333386	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	1.591141552596802	ETHER	ncit:C29819	ETHER	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	ChEMBL	33	inhibitor	4.922594178346359	DELCASERTIB	ncit:C101384	DELCASERTIB	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.8468979231563628	Dexchlorpheniramine Maleate	rxcui:54828	DEXCHLORPHENIRAMINE MALEATE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.049723174	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:Q03431	hgnc:9608	PTH1R	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	ALX1-11	chembl:CHEMBL2108078	PARATHYROID HORMONE	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:577	iuphar.ligand:577	L-156,602	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.5585922471882393	Diphemanil Methylsulfate	rxcui:23364	DIPHEMANIL METHYLSULFATE	TRUE	FALSE	FALSE
NCBIGENE:717	hgnc:1248	C2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	DNDI1417719	chembl:CHEMBL1420370	CHEMBL:CHEMBL1420370	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.3621218705909966	Dexrazoxane	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.052246439	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	GABAZINE	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.591141552596803	Elagolix	rxcui:2049846	ELAGOLIX	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.2900976311364336	2'-HYDROXYGENISTEIN	chembl:CHEMBL6665	CHEMBL:CHEMBL6665	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.1495945049449986	Dofetilide	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
UNIPROT:Q99250	hgnc:10588	SCN2A	TEND	1-Aug-11	NULL	0.053771297	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:5690	iuphar.ligand:5690	KI-20227	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.3125456621172291	PAPAVERINE HYDROCHLORIDE	rxcui:203132	PAPAVERINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	1,7-O-DIACETYLGEOPYXIN A	chembl:CHEMBL1873045	CHEMBL:CHEMBL1873045	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.1058622403945453	Ethopropazine	rxcui:4134	PROFENAMINE	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	PharmGKB	4/5/24	NULL	0.4375639269641209	metreleptin	rxcui:1491625	METRELEPTIN	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	NSC-95909	chembl:CHEMBL1547715	CHEMBL:CHEMBL1547715	FALSE	FALSE	FALSE
ITGB5	hgnc:6160	ITGB5	ChEMBL	33	inhibitor	8.751278539282415	INTETUMUMAB	ncit:C61070	INTETUMUMAB	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:12556	iuphar.ligand:12556	AM404	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1852122442176172	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.1074020548002842	Indomethacin	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	3.750547945	esuberaprost	ncit:C166506	ESUBERAPROST	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	CYCLOVALONE	ncit:C81040	CYCLOVALONE	FALSE	FALSE	FALSE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.1666910197958555	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.00901574	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
MEMBRANE COPPER AMINE OXIDASE	hgnc:550	AOC3	TTD	2020.06.01	NULL	1.312691780892362	Hydralazine	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.01103914	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.546954909	NICERGOLINE	rxcui:7398	NICERGOLINE	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:5244	iuphar.ligand:5244	PF750	FALSE	FALSE	FALSE
NCBIGENE:2685	ncbigene:2685	GGTL2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9960	iuphar.ligand:9960	COMPOUND 3 [PMID: 29633584]	FALSE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.060984519	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	inhibitor	1.193356164447602	SATAVAPTAN	ncit:C80380	SATAVAPTAN	FALSE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	1.250182648468916	SITAXENTAN	ncit:C73038	SITAXENTAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	BENZPIPERYLON	ncit:C83547	BENZPIPERYLON	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:6222	iuphar.ligand:6222	COMPOUND 2 [PMID: 21105727]	FALSE	FALSE	FALSE
HISTAMINE RECEPTOR	hgnc:5172	HR	TTD	2020.06.01	NULL	8.751278539282415	Histamine Phosphate	rxcui:26925	HISTAMINE PHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:2080	hgnc:6857	MAP3K5	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9040	ncit:C121943	SELONSERTIB	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.059297201	METOCLOPRAMIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.1151484018326633	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-3876	chembl:CHEMBL596631	CHEMBL:CHEMBL596631	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.066011799	CICLOSPORIN	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.3621218705909965	AT13387	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.5114383561918295	Nadolol	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.069240885	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.1426838892274307	IZENCITINIB	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	3.281729452230906	Methotrexate Sodium	rxcui:287734	METHOTREXATE SODIUM	TRUE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	ChEMBL	33	activator	1.093909817410302	INDOXIMOD	ncit:C71535	INDOXIMOD	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2659	iuphar.ligand:2659	LY-465608	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	PENTAMETHYLQUERCETIN	chembl:CHEMBL19032	PENTAMETHYLQUERCETIN	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.3663325900164732	GUANABENZ	rxcui:5033	GUANABENZ	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	5-HYDROXYINDOLACETIC ACID	iuphar.ligand:11900	5-HYDROXYINDOLEACETIC ACID	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.0055883	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.801643836	Methylprednisolone Acetate	rxcui:155323	METHYLPREDNISOLONE ACETATE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.016829382	CLADRIBINE	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.028598949	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1037701012563132	MESORIDAZINE BESYLATE	rxcui:203186	MESORIDAZINE BESYLATE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.358239472	DEXTROAMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
COL11A2	hgnc:2187	COL11A2	ChEMBL	33	cleavage	0.1875273972703374	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	1.544343271638073	Prolixin decanoate	drugsatfda.nda:016727	DRUGSATFDA.NDA:016727	FALSE	FALSE	FALSE
MT-ND6	hgnc:7462	MT-ND6	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CACNG8	hgnc:13628	CACNG8	ChEMBL	33	blocker	0.1881995384791917	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	0.1750255707856483	TENELIGLIPTIN	ncit:C87623	TENELIGLIPTIN	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	AZATADINE	rxcui:18600	AZATADINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.005524797	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	2.386712328895204	4-N-BENZYLCYTOSINE	chembl:CHEMBL2063052	CHEMBL:CHEMBL2063052	FALSE	FALSE	FALSE
APOLIPOPROTEIN C-III	hgnc:610	APOC3	TTD	2020.06.01	NULL	0.9376369863516875	ISIS-APOCIIIRx	rxcui:2637345	VOLANESORSEN	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	OncoKB	23-Jul-20	NULL	0.7440358272264402	Abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
V-SET IMMUNOREGULATORY RECEPTOR	hgnc:30085	VSIR	TTD	2020.06.01	NULL	26.25383561784724	JNJ-61610588	ncit:C127124	ONVATILIMAB	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1226814748497534	ESTROGENS, CONJUGATED SYNTHETIC A	chembl:CHEMBL1201466	ESTROGENS, CONJUGATED SYNTHETIC A	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.2983390411119005	Flurbiprofen	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
NDUFA12	hgnc:23987	NDUFA12	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.073437302	BAY 80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.2365210416022275	Caffeine	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.2408608772279564	OLICERIDINE	rxcui:2392230	OLICERIDINE	TRUE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P06280	hgnc:4296	GLA	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	MIGALASTAT	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8981	iuphar.ligand:8981	CONESSINE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 3	hgnc:10912	SLC12A3	TTD	2020.06.01	NULL	5.834185692854944	Bendroflumethiazide	rxcui:1369	BENDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:2808	drugbank:DB01941	LG-100268	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1029562181092048	NSC-36398	chembl:CHEMBL483206	CHEMBL:CHEMBL483206	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	DNDI1417013	chembl:CHEMBL1452227	CHEMBL:CHEMBL1452227	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	ERGOCORNINE	chembl:CHEMBL1385840	ERGOCORNINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.009443826	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.1682938180631234	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	PharmGKB	4/5/24	NULL	0.1864619006949378	clobazam	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.1672218829162245	Doxercalciferol	rxcui:11516	DOXERCALCIFEROL	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	3.000438356	boceprevir	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	1-HYDROXY-4-ETHOXYBENZENE	chembl:CHEMBL225153	1-HYDROXY-4-ETHOXYBENZENE	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.1136529680426287	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
TCN1	hgnc:11652	TCN1	NCI	14-Sep-17	NULL	7.501095890813499	CYANOCOBALAMIN	rxcui:11248	VITAMIN B12	TRUE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	ChEMBL	33	inhibitor	0.048618214	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.4102161815288632	IUPHAR.LIGAND:4270	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.3547815624033412	Darifenacin	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
NCBIGENE:78	hgnc:151	ACTG1P6	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:810	iuphar.ligand:810	CCL19	FALSE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:724	rxcui:6536	LYSINE	TRUE	FALSE	TRUE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	1.615620653405984	Epalrestat	ncit:C72762	EPALRESTAT	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:1238	iuphar.ligand:1238	(S)-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:1251	hgnc:7872	NOS1	GuideToPharmacology	2024.1	inhibitor	0.2465148884304905	IUPHAR.LIGAND:8759	iuphar.ligand:8759	L-NNA	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	CIViC	10-Apr-24	NULL	1.494525746746522	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.5357925636295356	AMIKACIN	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.016005996	tamatinib	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.5073204950308646	estrone sulfate	ncit:C1091	ESTRONE SULFATE	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.060077427	Estazolam	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q96GD4	hgnc:11390	AURKB	TdgClinicalTrial	Jan-14	NULL	0.07463777	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.03070624	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:569	rxcui:20192	CARAZOLOL	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:7349	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:5908	iuphar.ligand:5908	MRS2905	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PIPERIDOLATE	rxcui:59064	PIPERIDOLATE	FALSE	FALSE	FALSE
ACYL-COA DESATURASE	hgnc:10571	SCD	TTD	2020.06.01	NULL	7.501095891	Isoxyl	ncit:C152637	TIOCARLIDE	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.4953553890159858	MAFOSFAMIDE	ncit:C1150	MAFOSFAMIDE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	DTC	9/2/20	NULL	0.016669102	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	GRAVEOLINE	chembl:CHEMBL1371756	GRAVEOLINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	7-NITROINDAZOLE	drugbank:DB02207	7-NITROINDAZOLE	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	2.051080907644316	Tadalafil	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	CancerCommons	25-Jul-13	inhibitor	0.09003373	PF00562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.4773424657790409	pitavastatin	rxcui:861634	PITAVASTATIN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	PAPAVERINE HYDROCHLORIDE	rxcui:203132	PAPAVERINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AKT1S1	hgnc:28426	AKT1S1	MyCancerGenome	20-Jun-17	inhibitor	0.5966780822238011	MLN0128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	3.889457128569962	DIETHYL-2-DODECYLIDENEMALONATE	chembl:CHEMBL1797708	CHEMBL:CHEMBL1797708	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.053771297	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.074797252	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.018062494	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.01495945	flupenthixol	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:2393	hgnc:3905	FRA5A	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6497	iuphar.ligand:6497	UPAMOSTAT	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	agonist	0.040515178	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.1930429089547591	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	HYDRASTININE HYDROCHLORIDE	ncit:C90856	HYDRASTININE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:943	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
NCBIGENE:924	hgnc:1695	CD7	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4757	iuphar.ligand:4757	PHLORIZIN	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	DEL-22379	wikidata:Q21044462	DEL-22379	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.056826484	TDR77585	chembl:CHEMBL1333386	CHEMBL:CHEMBL1333386	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.4930297768609811	ARQ 092	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.04593847	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.044611445	METHYLENEDIOXYMETHAMPHETAMINE	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	negative modulator	0.042174836	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.056097939	IUPHAR.LIGAND:7207	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:8969	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
ACE	hgnc:2707	ACE	NCI	14-Sep-17	NULL	0.044498026	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
COMPLEMENT C3	hgnc:7422	MT-CO3	TTD	2020.06.01	NULL	13.12691780892362	APL-2	rxcui:2557372	PEGCETACOPLAN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	HARMALINE	drugbank:DB13875	HARMALINE	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.07458476	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	1.346350544504987	M-1095	chembl:CHEMBL4298023	M-1095	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
RFC1	hgnc:9969	RFC1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	17.50255707856483	PRALATREXATE	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	0.089756703	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
NCBIGENE:1877	hgnc:3121	E4F1	GuideToPharmacology	2024.1	NULL	17.50255707856483	IUPHAR.LIGAND:5080	iuphar.ligand:5080	CD30 LIGAND	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:6126	iuphar.ligand:6126	SNAP 37889	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.085239726	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	DTC	9/2/20	NULL	0.3409589041278863	TCMDC-124059	chembl:CHEMBL530733	CHEMBL:CHEMBL530733	FALSE	FALSE	FALSE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	0.4375639269641208	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.002480521	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
JUNB	hgnc:6205	JUNB	NCI	14-Sep-17	NULL	1.346350544504987	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
NCBIGENE:721	hgnc:1324	C4B	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
ATP1A3	hgnc:801	ATP1A3	ChEMBL	33	inhibitor	0.172722603	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	ETHOPROPAZINE HYDROCHLORIDE	rxcui:6541	ETHOPROPAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	DTC	9/2/20	NULL	0.07458476	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.7955707762984013	XANTHOHUMOL	ncit:C121950	XANTHOHUMOL	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	DTC	9/2/20	NULL	0.1988926940746003	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	MERCAPTOPURINE HYDRATE	chembl:CHEMBL1200751	MERCAPTOPURINE	FALSE	FALSE	FALSE
UNIPROT:P68871	hgnc:4827	HBB	TdgClinicalTrial	Jan-14	NULL	1.810609352954982	AES-103	chembl:CHEMBL185885	AES-103	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.090530468	IUPHAR.LIGAND:17	ncit:C76104	LYSERGIDE	FALSE	FALSE	FALSE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	0.056581542	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:1488	hgnc:2495	CTBP2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9349	iuphar.ligand:9349	COMPOUND 41 [PMID: 25000588]	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.019461702	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
ASS1	hgnc:758	ASS1	CIViC	10-Apr-24	NULL	0.021309932	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.036463661	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.112919723	CEFOTAXIME	rxcui:203117	CEFOTAXIME SODIUM	TRUE	FALSE	FALSE
SOST	hgnc:13771	SOST	ChEMBL	33	inhibitor	6.563458904461812	AMG-167	chembl:CHEMBL2109571	AMG-167	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	CancerCommons	25-Jul-13	inhibitor	0.030945115	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
EIF4E	hgnc:3287	EIF4E	CancerCommons	25-Jul-13	inhibitor	NULL	ISIS-EIF4ERX	NULL	NULL	NULL	NULL	NULL
DPYD	hgnc:3012	DPYD	CGI	2/1/22	NULL	NULL	Flourouracil	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	NULL	Chemotherapy	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.2917092846427472	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
DNMT3A	hgnc:2978	DNMT3A	CGI	2/1/22	NULL	0.021370644	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.3454452054979901	HSP90 inhibitor	ncit:C156880	HSP90 INHIBITOR	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.2917092846427472	Pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	NULL	Chemotherapy	NULL	NULL	NULL	NULL	NULL
PALB2	hgnc:26144	PALB2	CGI	2/1/22	NULL	NULL	Mytomycin C	NULL	NULL	NULL	NULL	NULL
NPM1	hgnc:7910	NPM1	CGI	2/1/22	NULL	0.082429625	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CGI	2/1/22	NULL	NULL	Chemotherapy	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	CGI	2/1/22	NULL	NULL	Chemotherapy	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	CGI	2/1/22	NULL	0.015768069	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
MICRORNA HSA-MIR-155	hgnc:31542	MIR155	TTD	2020.06.01	NULL	26.25383561784724	Cobomarsen	ncit:C124225	COBOMARSEN	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	CARBINOXAMINE MALEATE	rxcui:91066	CARBINOXAMINE MALEATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	FLUPHENAZINE DECANOATE	rxcui:25190	FLUPHENAZINE DECANOATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.059297201	METOCLOPRAMIDE HYDROCHLORIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	1.779921058837101	SARALASIN ACETATE	rxcui:7830	SARALASIN ACETATE	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	1.988926940746003	ABARELIX	rxcui:301739	ABARELIX	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.2373228078449469	CANDESARTAN CILEXETIL	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	ChEMBL	33	agonist	16.40864726115453	LUTROPIN ALFA	rxcui:388084	LUTROPIN ALFA	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	2.386712328895204	GANIRELIX ACETATE	rxcui:259264	GANIRELIX ACETATE	TRUE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	0.159436249	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.2014360789093139	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
SCTR	hgnc:10608	SCTR	ChEMBL	33	agonist	31.50460274141669	SECRETIN SYNTHETIC HUMAN	rxcui:606396	SECRETIN HUMAN, SYNTHETIC	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.063331621	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.059667808	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.179119736	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.6731752722524935	ALMOTRIPTAN MALATE	rxcui:283792	ALMOTRIPTAN MALATE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.100976291	TRAZODONE HYDROCHLORIDE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
PTGIR	hgnc:9602	PTGIR	ChEMBL	33	agonist	0.8334550989792778	TREPROSTINIL	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
SV2A	hgnc:20566	SV2A	ChEMBL	33	modulator	4.500657534	LEVETIRACETAM	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
PPPK-DHPS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFACYTINE	rxcui:78902	SULFACYTINE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.4861821410712453	AMPHETAMINE SULFATE	rxcui:81952	AMPHETAMINE SULFATE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.358239472	DEXTROAMPHETAMINE SULFATE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	HEXAFLUORENIUM BROMIDE	rxcui:53017	HEXAFLUORENIUM BROMIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.7225826316838693	DEZOCINE	rxcui:22713	DEZOCINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.1717808219270267	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	PREDNICARBATE	rxcui:34369	PREDNICARBATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.039778539	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.067059606	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.1389091831632129	ESTROGENS, CONJUGATED	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	HYDROCODONE POLISTIREX	rxcui:221107	HYDROCODONE POLISTIREX	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.02875557	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.3513393859865807	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.5000730593875666	ISOPROTERENOL SULFATE	rxcui:82031	ISOPROTERENOL SULFATE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	negative modulator	0.09963505	KETAMINE HYDROCHLORIDE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.2651902587661338	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.2220197515251353	DEXMEDETOMIDINE HYDROCHLORIDE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.085239726	DEXMEDETOMIDINE HYDROCHLORIDE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1178056726441863	IBUPROFEN SODIUM	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	BALSALAZIDE DISODIUM	rxcui:153718	BALSALAZIDE DISODIUM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1193356164447602	BALSALAZIDE DISODIUM	rxcui:153718	BALSALAZIDE DISODIUM	TRUE	FALSE	FALSE
ABCC9	hgnc:60	ABCC9	ChEMBL	33	potentiator	0.3977853881492006	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.054695491	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.09055649	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	0.061791905	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
GB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
GG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
GJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
GN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
GI	hgnc:4384	GNAI1	ChEMBL	33	inhibitor	6.563458904461812	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	2.917092846427472	CRILVASTATIN	ncit:C90865	CRILVASTATIN	FALSE	FALSE	FALSE
GK	hgnc:4289	GK	ChEMBL	33	inhibitor	6.563458904461812	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
PBP4	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHICILLIN SODIUM	rxcui:267073	METHICILLIN SODIUM	TRUE	FALSE	FALSE
PBPF	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHICILLIN SODIUM	rxcui:267073	METHICILLIN SODIUM	TRUE	FALSE	FALSE
MECA	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHICILLIN SODIUM	rxcui:267073	METHICILLIN SODIUM	TRUE	FALSE	FALSE
PBP2	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHICILLIN SODIUM	rxcui:267073	METHICILLIN SODIUM	TRUE	FALSE	FALSE
PBPA	NULL	NULL	ChEMBL	33	inhibitor	NULL	METHICILLIN SODIUM	rxcui:267073	METHICILLIN SODIUM	TRUE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	1.250182648468916	Troplasminogen alfa	ncit:C152767	TROPLASMINOGEN ALFA	FALSE	FALSE	FALSE
PSMA2	hgnc:9531	PSMA2	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMC3	hgnc:9549	PSMC3	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA5	hgnc:9534	PSMA5	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
EPHRIN TYPE-B RECEPTOR 4	hgnc:3395	EPHB4	TTD	2020.06.01	NULL	5.469549087051511	KD019	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
8230819	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8231511	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE	hgnc:38595	LINC00273	TTD	2020.06.01	NULL	8.751278539282415	Nemonoxacin	ncit:C174838	NEMONOXACIN	FALSE	FALSE	FALSE
8236100	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8233621	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
8230508	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
NCBIGENE:2464	hgnc:3861	FRA16E	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4821	rxcui:14851	VIGABATRIN	TRUE	FALSE	FALSE
8238404	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
PSMD2	hgnc:9559	PSMD2	ChEMBL	33	inhibitor	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD3	hgnc:9560	PSMD3	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SEM1	hgnc:10845	SEM1	ChEMBL	33	inhibitor	0.3663325900164732	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD13	hgnc:9558	PSMD13	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.041150213	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
8239920	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIPERONYL BUTOXIDE	rxcui:8345	PIPERONYL BUTOXIDE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	ECONAZOLE NITRATE	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	SERTACONAZOLE NITRATE	rxcui:236601	SERTACONAZOLE NITRATE	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	BUTOCONAZOLE NITRATE	rxcui:19884	BUTOCONAZOLE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.7501095890813501	MIVACURIUM CHLORIDE	rxcui:52796	MIVACURIUM CHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.025304902	IUPHAR.LIGAND:22	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
NDUFB5	hgnc:7700	NDUFB5	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MT-ND4	hgnc:7459	MT-ND4	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.05751114	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NDUFB7	hgnc:7702	NDUFB7	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.6049270879688307	TOFACITINIB CITRATE	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.6326225450083675	IUPHAR.LIGAND:3231	iuphar.ligand:3231	SB236057	FALSE	FALSE	FALSE
NDUFS4	hgnc:7711	NDUFS4	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.2344092465879218	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.056826484	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
RXRG	hgnc:10479	RXRG	ChEMBL	33	agonist	1.988926940746004	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.2381300282797936	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
RXRG	hgnc:10479	RXRG	ChEMBL	33	agonist	0.2983390411119005	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
RXRG	hgnc:10479	RXRG	ChEMBL	33	agonist	0.9092237443410301	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.061992528	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:120	ncit:C77255	ALNIDITAN	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.064505739	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.061197752	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.058931169	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.073266518	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.076840494	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.030850571	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.084553416	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.05309168	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.039390601	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.031254566	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.021715331	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXIFLOXACIN HYDROCHLORIDE	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
TOPB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ENOXACIN	rxcui:3925	ENOXACIN	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFATHIAZOLE	rxcui:10193	SULFATHIAZOLE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFALENE	rxcui:10175	SULFALENE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFISOXAZOLE ACETYL	rxcui:40595	ACETYL SULFISOXAZOLE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAMERAZINE	rxcui:10176	SULFAMERAZINE	TRUE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TRIMETHOPRIM SULFATE	rxcui:221176	TRIMETHOPRIM SULFATE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIBUTEN	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIBUTEN	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.008224886	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIBUTEN	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIBUTEN	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIBUTEN	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIBUTEN	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTIBUTEN	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.04468738	IUPHAR.LIGAND:22	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMOXICILLIN	rxcui:1297882	AMOXICILLIN ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:211	ncit:C152343	SERGOLEXOLE	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.276356164	IUPHAR.LIGAND:183	iuphar.ligand:183	LY53857	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMPICILLIN SODIUM	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LORACARBEF	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LORACARBEF	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LORACARBEF	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LORACARBEF	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LORACARBEF	rxcui:28981	LORACARBEF	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.03070624	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
FOLP1	NULL	NULL	ChEMBL	33	inhibitor	NULL	DAPSONE	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
FOLP1	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFOXONE SODIUM	ncit:C66574	SULFOXONE SODIUM	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:194	iuphar.ligand:194	SB 243213	FALSE	FALSE	FALSE
CPS1	hgnc:2323	CPS1	ChEMBL	33	positive modulator	7.501095891	CARGLUMIC ACID	rxcui:401713	CARGLUMIC ACID	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:2941	rxcui:1300701	LORCASERIN	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:171	iuphar.ligand:171	ORG-37684	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:191	iuphar.ligand:191	SB 221284	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.077217164	IUPHAR.LIGAND:206	ncit:C83940	MESULERGINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.020320306	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.099446347	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.088996053	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.011710007	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.1779921058837101	IUPHAR.LIGAND:206	ncit:C83940	MESULERGINE	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
NCBIGENE:779	hgnc:1397	CACNA1S	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:11741	ncit:C71621	BIRICODAR	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	0.1025540453822158	PEGINTERFERON ALFA-2B	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.3889457128569963	INTERFERON BETA-1A	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXIFLOXACIN HYDROCHLORIDE	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MOXIFLOXACIN HYDROCHLORIDE	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEVOFLOXACIN	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEVOFLOXACIN	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ENOXACIN	rxcui:3925	ENOXACIN	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ENOXACIN	rxcui:3925	ENOXACIN	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.130291988	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.068458502	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.062139256	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
PFOR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEVOFLOXACIN	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
KCNK3	hgnc:6278	KCNK3	ChEMBL	33	potentiator	0.2419708351875322	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.3017682254924971	LEVOFLOXACIN	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR1	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSR2	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB1	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMB2	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG1	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMG2	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	SOFOSBUVIR	rxcui:1484911	SOFOSBUVIR	TRUE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	ChEMBL	33	agonist	2.461297089173179	MENOTROPINS	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	2.812910959055062	MACITENTAN	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.061055432	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.2910624791335615	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.2892984641085096	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEDIZOLID PHOSPHATE	rxcui:1540824	TEDIZOLID PHOSPHATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.2408608772279564	NALOXEGOL OXALATE	rxcui:1551777	NALOXEGOL	TRUE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	4.039051633514961	ALIROCUMAB	rxcui:1659152	ALIROCUMAB	TRUE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	5.527123287967842	ARRY-502	drugbank:DB16053	ARRY-502	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.4579157375205915	DERAZANTINIB	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.3125456621172291	AS-703988	chembl:CHEMBL3545243	AS-703988	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	ChEMBL	33	inhibitor	1.591141552596802	AR-12	iuphar.ligand:8005	OSU-03012	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.4167275494896388	CAL-263	chembl:CHEMBL3545247	CAL-263	FALSE	FALSE	FALSE
NDUFA1	hgnc:7683	NDUFA1	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFAB1	hgnc:7694	NDUFAB1	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
MT-ND4L	hgnc:7460	MT-ND4L	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA4	hgnc:7687	NDUFA4	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.1232574442152452	PKI-179	drugbank:DB13109	PKI-179	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.4773424657790409	PLX-5622	chembl:CHEMBL3545079	PLX-5622	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	SCIO-323	chembl:CHEMBL1614702	SCIO-323	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	ChEMBL	33	inhibitor	1.029562181092048	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.6250913242344582	AZD3161	chembl:CHEMBL3545208	AZD3161	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.2586584789935689	DELUCEMINE	ncit:C76776	DELUCEMINE	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.1389091831632129	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	inhibitor	0.2453629496995069	SR16234	chembl:CHEMBL3545210	SR16234	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.1400204566285186	SODELGLITAZAR	ncit:C75193	SODELGLITAZAR	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.105015342	FARGLITAZAR	ncit:C81693	FARGLITAZAR	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.2641230947469542	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.079376676	SAPITINIB	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.4234489615781814	FILGOTINIB	ncit:C155799	FILGOTINIB	TRUE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.3387591692625452	SOLCITINIB	ncit:C152385	SOLCITINIB	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.2237542808339254	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.04464938	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.3070624048871023	ABEMACICLIB	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1607377690888607	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.088248187	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.09972967	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.079197091	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.089298761	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.046303061	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.2465148884304905	TRICIRIBINE PHOSPHATE	ncit:C1262	TRICIRIBINE PHOSPHATE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2500365296937833	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PTK2	hgnc:9611	PTK2	ChEMBL	33	inhibitor	2.917092846427472	DEFACTINIB	ncit:C79809	DEFACTINIB	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1875273972703375	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.030386384	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1041818873724097	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	inhibitor	0.3860858179095183	GSK163090	chembl:CHEMBL1631540	GSK163090	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	1.750255707856483	UBROGEPANT	rxcui:2268216	UBROGEPANT	TRUE	FALSE	FALSE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	6.563458904461812	TALADEGIB	ncit:C103826	TALADEGIB	FALSE	FALSE	TRUE
CRHR1	hgnc:2357	CRHR1	ChEMBL	33	inhibitor	2.917092846427472	CRINECERFONT	ncit:C174708	CRINECERFONT	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.458546423213736	CP-601927	drugbank:DB12244	CP-601927	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	agonist	0.040021091	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	agonist	0.038159645	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	inverse agonist	0.03729238	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.3409589041278863	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.1544343271638073	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.6806549974997433	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
FNTB	hgnc:3785	FNTB	ChEMBL	33	inhibitor	2.333674277141978	TIPIFARNIB	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
CETP	hgnc:1869	CETP	ChEMBL	33	inhibitor	6.058577450272442	ANACETRAPIB	ncit:C75251	ANACETRAPIB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.041672755	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
XPNPEP1	hgnc:12822	XPNPEP1	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
XPNPEP2	hgnc:12823	XPNPEP2	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
RNPEP	hgnc:10078	RNPEP	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
RNPEPL1	hgnc:10079	RNPEPL1	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PSMB3	hgnc:9540	PSMB3	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
SEM1	hgnc:10845	SEM1	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMD6	hgnc:9564	PSMD6	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMD12	hgnc:9557	PSMD12	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMA1	hgnc:9530	PSMA1	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMA2	hgnc:9531	PSMA2	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB10	hgnc:9538	PSMB10	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB7	hgnc:9544	PSMB7	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMA5	hgnc:9534	PSMA5	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMD11	hgnc:9556	PSMD11	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.2885036881082115	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.3040984820600068	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	CARMEGLIPTIN	ncit:C81698	CARMEGLIPTIN	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.3125456621172292	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.2744303374687866	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
CHRNA9	hgnc:14079	CHRNA9	ChEMBL	33	inhibitor	2.917092846427472	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.042174836	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	negative modulator	0.038894571	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	negative modulator	0.1530835896084387	ESKETAMINE HYDROCHLORIDE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.4434769530041765	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	FALDAPREVIR	ncit:C171746	FALDAPREVIR	FALSE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	ChEMBL	33	binder	4.375639269641208	VINTAFOLIDE	ncit:C62525	VINTAFOLIDE	FALSE	FALSE	TRUE
EGLN1	hgnc:1232	EGLN1	ChEMBL	33	inhibitor	0.9546849315580819	DAPRODUSTAT	rxcui:2628210	DAPRODUSTAT	TRUE	FALSE	FALSE
EGLN3	hgnc:14661	EGLN3	ChEMBL	33	inhibitor	2.100306849	DAPRODUSTAT	rxcui:2628210	DAPRODUSTAT	TRUE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.093909817410302	BEXAGLIFLOZIN	rxcui:2627044	BEXAGLIFLOZIN	TRUE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.2243917574174978	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.2011788169949981	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.2027323213733378	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1190650141398968	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
MGAM2	hgnc:28101	MGAM2	ChEMBL	33	inhibitor	6.563458904461812	VOGLIBOSE	ncit:C95221	VOGLIBOSE	TRUE	FALSE	FALSE
RBX1	hgnc:9928	RBX1	ChEMBL	33	inhibitor	1.875273972703375	POMALIDOMIDE	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.3580068493342807	DEXIBUPROFEN	ncit:C166907	DEXIBUPROFEN	TRUE	FALSE	FALSE
VEGFC	hgnc:12682	VEGFC	ChEMBL	33	inhibitor	1.166837138570989	CONBERCEPT	ncit:C162879	CONBERCEPT	FALSE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	TAPLITUMOMAB PAPTOX	ncit:C203065	TAPLITUMOMAB PAPTOX	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	0.2019525816757481	CONBERCEPT	ncit:C162879	CONBERCEPT	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	2.333674277141977	INTETUMUMAB	ncit:C61070	INTETUMUMAB	FALSE	FALSE	FALSE
CCN2	hgnc:2500	CCN2	ChEMBL	33	inhibitor	4.039051633514961	PAMREVLUMAB	ncit:C92577	PAMREVLUMAB	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	ChEMBL	33	inhibitor	1.458546423213736	MLNM-2201	chembl:CHEMBL2109332	MLNM-2201	FALSE	FALSE	FALSE
KIR2DL2	hgnc:6330	KIR2DL2	ChEMBL	33	inhibitor	7.876150685354174	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	VELPATASVIR	rxcui:1799206	VELPATASVIR	TRUE	FALSE	FALSE
TRGV3	hgnc:12288	TRGV3	ChEMBL	33	inhibitor	3.500511415712967	TOL-101	drugbank:DB16980	TOL-101	FALSE	FALSE	FALSE
TCDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MK-3415	chembl:CHEMBL2109312	MK-3415	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	0.2187819634820604	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	agonist	0.760980743	ARGIPRESSIN TANNATE	ncit:C166779	ARGIPRESSIN TANNATE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.032016873	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.100976291	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OZENOXACIN	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OZENOXACIN	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	TUVIRUMAB	ncit:C166625	TUVIRUMAB	FALSE	FALSE	FALSE
FGB	hgnc:3662	FGB	ChEMBL	33	binder	3.500511415712966	BICIROMAB BRALLOBARBITAL	chembl:CHEMBL2109283	BICIROMAB BRALLOBARBITAL	FALSE	FALSE	FALSE
TNFRSF1A	hgnc:11916	TNFRSF1A	ChEMBL	33	inhibitor	17.50255707856483	GSK-1995057	chembl:CHEMBL2109590	GSK-1995057	FALSE	FALSE	FALSE
KCNA6	hgnc:6225	KCNA6	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNH3	hgnc:6252	KCNH3	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
MPL	hgnc:7217	MPL	ChEMBL	33	agonist	3.182283105193605	LUSUTROMBOPAG	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	ChEMBL	33	inhibitor	0.6731752722524935	MOLIBRESIB	ncit:C101538	MOLIBRESIB	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	ChEMBL	33	inhibitor	1.184383561707394	BIRABRESIB	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
HSPA1B	hgnc:5233	HSPA1B	ChEMBL	33	inhibitor	8.751278539282415	CD24FC	chembl:CHEMBL4297717	CD24FC	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.1902451856365742	CD24FC	chembl:CHEMBL4297717	CD24FC	FALSE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	VEDROPREVIR	ncit:C152843	VEDROPREVIR	FALSE	FALSE	FALSE
PIKFYVE	hgnc:23785	PIKFYVE	ChEMBL	33	inhibitor	8.751278539282415	APILIMOD	ncit:C90808	APILIMOD	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	1.346350544504987	TOLOXATONE	rxcui:38382	TOLOXATONE	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.6563458904461812	MOFEZOLAC	rxcui:11469	MOFEZOLAC	FALSE	FALSE	FALSE
L	NULL	NULL	ChEMBL	33	inhibitor	NULL	GALIDESIVIR	ncit:C172613	GALIDESIVIR	FALSE	FALSE	FALSE
HELI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMENAMEVIR	ncit:C90782	AMENAMEVIR	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	BENZHYDROCODONE HYDROCHLORIDE	rxcui:2122776	BENZHYDROCODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CASR	hgnc:1514	CASR	ChEMBL	33	positive modulator	1.640864726115453	EVOCALCET	ncit:C153105	EVOCALCET	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.7369497717290455	PEMIGATINIB	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
CHRM4	hgnc:1953	CHRM4	ChEMBL	33	inhibitor	0.3241214273808302	SOFPIRONIUM BROMIDE	ncit:C152384	SOFPIRONIUM BROMIDE	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.1535312024435511	SOFPIRONIUM BROMIDE	ncit:C152384	SOFPIRONIUM BROMIDE	FALSE	FALSE	FALSE
CHRM5	hgnc:1954	CHRM5	ChEMBL	33	inhibitor	0.1715936968486748	SOFPIRONIUM BROMIDE	ncit:C152384	SOFPIRONIUM BROMIDE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	2.187819634820604	POTASSIUM OXYBATE	rxcui:2387309	POTASSIUM OXYBATE	TRUE	FALSE	FALSE
CRBN	hgnc:30185	CRBN	ChEMBL	33	modulator	1.458546423213736	IBERDOMIDE	ncit:C129048	IBERDOMIDE	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.4817217544559128	GSK-1521498	drugbank:DB12886	GSK-1521498	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	SERPLULIMAB	ncit:C156738	SERPLULIMAB	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	2.282942227638891	BMS-813160	drugbank:DB16240	BMS-813160	FALSE	FALSE	FALSE
CUL4A	hgnc:2554	CUL4A	ChEMBL	33	modulator	3.281729452230906	IBERDOMIDE	ncit:C129048	IBERDOMIDE	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	1.544343271638073	MM-111	drugbank:DB17983	MM-111	FALSE	TRUE	TRUE
IL17A	hgnc:5981	IL17A	ChEMBL	33	binder	2.019525817	CJM-112	chembl:CHEMBL4297926	CJM-112	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.2885036881082115	PERZINFOTEL	ncit:C72122	PERZINFOTEL	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	agonist	0.038159645	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	agonist	0.042073455	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	negative modulator	0.3889457128569963	TAS-117	drugbank:DB15054	TAS-117	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	agonist	0.044347695	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
REVERSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ISLATRAVIR	ncit:C174896	ISLATRAVIR	FALSE	FALSE	FALSE
TRANSCRIPTASE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ISLATRAVIR	ncit:C174896	ISLATRAVIR	FALSE	FALSE	FALSE
RPS6	hgnc:10429	RPS6	ChEMBL	33	modulator	0.1093909817410302	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL9	hgnc:10369	RPL9	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL21	hgnc:10313	RPL21	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL10	hgnc:10298	RPL10	ChEMBL	33	modulator	0.1093909817410302	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL26	hgnc:10327	RPL26	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL4	hgnc:10353	RPL4	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL18A	hgnc:10311	RPL18A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL38	hgnc:10349	RPL38	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL35A	hgnc:10345	RPL35A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL39	hgnc:10350	RPL39	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TALAMPICILLIN	rxcui:10322	TALAMPICILLIN	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TALAMPICILLIN	rxcui:10322	TALAMPICILLIN	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TALAMPICILLIN	rxcui:10322	TALAMPICILLIN	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TALAMPICILLIN	rxcui:10322	TALAMPICILLIN	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TALAMPICILLIN	rxcui:10322	TALAMPICILLIN	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TALAMPICILLIN	rxcui:10322	TALAMPICILLIN	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TALAMPICILLIN	rxcui:10322	TALAMPICILLIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMB1	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMB2	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMG1	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMG2	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.035719504	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	ABT-072	drugbank:DB15156	ABT-072	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	FILIBUVIR	ncit:C83717	FILIBUVIR	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	ChEMBL	33	inhibitor	0.1190650141398968	ZAGOTENEMAB	ncit:C171842	ZAGOTENEMAB	FALSE	FALSE	FALSE
TAT	hgnc:11573	TAT	ChEMBL	33	inhibitor	3.500511415712966	RO-24-7429	chembl:CHEMBL2360841	RO-24-7429	FALSE	FALSE	FALSE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	1.312691780892362	TRIAPINE	ncit:C2242	TRIAPINE	FALSE	FALSE	TRUE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	0.8751278539282416	ATN-161	drugbank:DB05491	ATN-161	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
TACR2	hgnc:11527	TACR2	ChEMBL	33	inhibitor	5.250767123569449	SAREDUTANT	ncit:C152301	SAREDUTANT	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
ITGB1	hgnc:6153	ITGB1	ChEMBL	33	inhibitor	1.093909817410302	ATN-161	drugbank:DB05491	ATN-161	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM MEDOXOMIL	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM MEDOXOMIL	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM MEDOXOMIL	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM MEDOXOMIL	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM MEDOXOMIL	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM MEDOXOMIL	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM MEDOXOMIL	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
ATP1A3	hgnc:801	ATP1A3	ChEMBL	33	inhibitor	0.364636606	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	ChEMBL	33	inhibitor	0.1419126249613365	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.068637479	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.087222045	E-7090	iuphar.ligand:11414	TASURGRATINIB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.2282942227638891	LUMINESPIB	ncit:C71467	LUMINESPIB	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.072424374	LUMINESPIB	ncit:C71467	LUMINESPIB	FALSE	FALSE	FALSE
VWF	hgnc:12726	VWF	ChEMBL	33	inhibitor	5.527123287967842	EGAPTIVON PEGOL	ncit:C95742	EGAPTIVON PEGOL	FALSE	FALSE	FALSE
REVERSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	RO-0622	chembl:CHEMBL519846	RO-0622	FALSE	FALSE	FALSE
TRANSCRIPTASE	NULL	NULL	ChEMBL	33	inhibitor	NULL	RO-0622	chembl:CHEMBL519846	RO-0622	FALSE	FALSE	FALSE
TBXAS1	hgnc:11609	TBXAS1	ChEMBL	33	inhibitor	1.640864726115453	PICOTAMIDE	ncit:C73157	PICOTAMIDE	TRUE	FALSE	FALSE
OPG071	NULL	NULL	ChEMBL	33	inhibitor	NULL	BRINCIDOFOVIR	rxcui:2599518	BRINCIDOFOVIR	TRUE	FALSE	FALSE
REP	NULL	NULL	ChEMBL	33	inhibitor	NULL	RO-0622	chembl:CHEMBL519846	RO-0622	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	TEGOBUVIR	ncit:C152541	TEGOBUVIR	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	EPCORITAMAB	rxcui:2637392	EPCORITAMAB	TRUE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	ChEMBL	33	inhibitor	4.039051633514961	MARALIXIBAT CHLORIDE	rxcui:2571073	MARALIXIBAT CHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	RO-0622	chembl:CHEMBL519846	RO-0622	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	binder	0.7955707762984014	EP-100	chembl:CHEMBL4297748	EP-100	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOMOXEF	ncit:C65693	FLOMOXEF	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOMOXEF	ncit:C65693	FLOMOXEF	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOMOXEF	ncit:C65693	FLOMOXEF	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOMOXEF	ncit:C65693	FLOMOXEF	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOMOXEF	ncit:C65693	FLOMOXEF	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOMOXEF	ncit:C65693	FLOMOXEF	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	FLOMOXEF	ncit:C65693	FLOMOXEF	FALSE	FALSE	FALSE
HA	NULL	NULL	ChEMBL	33	inhibitor	NULL	GEDIVUMAB	ncit:C166943	GEDIVUMAB	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.1268301237577161	BUCINDOLOL HYDROCHLORIDE	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	potentiator	1.250182648468916	EZOGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
INT	hgnc:29239	INTU	ChEMBL	33	inhibitor	52.50767123569449	BMS-707035	chembl:CHEMBL486226	BMS-707035	FALSE	FALSE	FALSE
FLNA	hgnc:3754	FLNA	ChEMBL	33	positive modulator	26.25383561784724	SIMUFILAM	ncit:C180661	SIMUFILAM	FALSE	FALSE	FALSE
PRMT5	hgnc:10894	PRMT5	ChEMBL	33	inhibitor	11.66837138570988	PEMRAMETOSTAT	ncit:C142177	PEMRAMETOSTAT	FALSE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	inhibitor	0.8751278539282416	BAZLITORAN	ncit:C114975	BAZLITORAN	FALSE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	ChEMBL	33	inhibitor	2.187819634820604	ENPATORAN	ncit:C177069	ENPATORAN	FALSE	FALSE	FALSE
CTAG1B	hgnc:2491	CTAG1B	ChEMBL	33	vaccine	2.187819634820604	RASDEGAFUSP ALFA	ncit:C170362	RASDEGAFUSP ALFA	FALSE	FALSE	FALSE
ADAM17	hgnc:195	ADAM17	ChEMBL	33	inhibitor	3.500511415712967	APRATASTAT	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
SV2A	hgnc:20566	SV2A	ChEMBL	33	modulator	21.00306849427779	SELETRACETAM	ncit:C66534	SELETRACETAM	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.2476776945079929	LACIDIPINE	rxcui:28382	LACIDIPINE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	ChEMBL	33	inhibitor	0.1190650141398968	BEPRANEMAB	ncit:C174583	BEPRANEMAB	FALSE	FALSE	FALSE
LEPR	hgnc:6554	LEPR	ChEMBL	33	agonist	8.751278539282415	MIBAVADEMAB	ncit:C179103	MIBAVADEMAB	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
C-MET	hgnc:7029	MET	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.272767123	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
CDK1	hgnc:1722	CDK1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3431873936973496	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3409589041278863	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
IL-1R2	hgnc:5994	IL1R2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	5.834185692854945	ANAKINRA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
PARP2	hgnc:272	PARP2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.5966780822238011	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
VEGFC	hgnc:12682	VEGFC	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4487835148349958	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	COSMIC	4-Sep-20	NULL	0.1108075556053025	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	COSMIC	4-Sep-20	NULL	0.1766118064547324	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.039899446	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007378818	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.003150019	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	DTC	9/2/20	NULL	0.4688184931758437	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	DIMETHISOQUIN	ncit:C72169	DIMETHISOQUIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	SJ000117451	chembl:CHEMBL592123	CHEMBL:CHEMBL592123	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	OXOPURPUREINE	chembl:CHEMBL456295	OXOPURPUREINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CERIVASTATIN SODIUM	rxcui:221072	CERIVASTATIN SODIUM	TRUE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.025390557	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	GNF-PF-1399	chembl:CHEMBL578504	CHEMBL:CHEMBL578504	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.347732922	FUCHSIN, BASIC	chembl:CHEMBL1979636	FUCHSIN, BASIC	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-4078	chembl:CHEMBL584883	CHEMBL:CHEMBL584883	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1591141552596803	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.004185879	TCMDC-125488	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1025540453822158	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1988926940746003	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.006627246	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CGA	hgnc:1885	CGA	DTC	9/2/20	NULL	6.563458904461812	4-{([(4'-CHLOROPHENYL)AMINO]CARBONYLAMINO)}BENZENESULFONAMIDE	chembl:CHEMBL1446150	CHEMBL:CHEMBL1446150	FALSE	FALSE	FALSE
SLC22A2	hgnc:10966	SLC22A2	DTC	9/2/20	NULL	1.875273972703374	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	THIORPHAN	drugbank:DB08626	THIORPHAN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.031822831	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	SJ000032152	chembl:CHEMBL590665	CHEMBL:CHEMBL590665	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004698673	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.040235763	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.016460085	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
CRYZ	hgnc:2419	CRYZ	DTC	9/2/20	NULL	17.50255707856483	2'-HYDROXYCHALCONE	chembl:CHEMBL32147	2'-HYDROXYCHALCONE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2703097618311171	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	PHENSERINE	drugbank:DB04892	PHENSERINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	3,5-DICHLORO-BENZOIC ACID	chembl:CHEMBL118280	CHEMBL:CHEMBL118280	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	PROFLAVINE	rxcui:8723	PROFLAVINE	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	NSC-728558	chembl:CHEMBL457246	CHEMBL:CHEMBL457246	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.078958904	TPKI-24	iuphar.ligand:9403	RO3280	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.059667808	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	GRAVEOLINE	chembl:CHEMBL1371756	GRAVEOLINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	2'-HYDROXYCHALCONE	chembl:CHEMBL32147	2'-HYDROXYCHALCONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	2,4-DINITROPHENOL	drugbank:DB04528	2,4-DINITROPHENOL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	MESO-2,3-DIMERCAPTOSUCCINIC ACID	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	GNF-PF-1000	chembl:CHEMBL600554	CHEMBL:CHEMBL600554	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.010685322	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.010001461	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.000562132	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	TCMDC-125185	chembl:CHEMBL580819	CHEMBL:CHEMBL580819	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.059330702	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.002899535	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-4789	chembl:CHEMBL583351	CHEMBL:CHEMBL583351	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.032412143	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001631484	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.8751278539282416	TEPOTINIB	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	IOPHENOXIC ACID	chembl:CHEMBL1551165	IOPHENOXIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
IDO1	hgnc:6059	IDO1	DTC	9/2/20	NULL	7.501095891	S-(4-CHLOROBENZYL)ISOTHIOUREA HCL	chembl:CHEMBL1224312	CHEMBL:CHEMBL1224312	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000002502	chembl:CHEMBL591630	CHEMBL:CHEMBL591630	FALSE	FALSE	FALSE
TRPM8	hgnc:17961	TRPM8	DTC	9/2/20	NULL	4.836232876971861	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.05293112	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.4934931507114145	GW501516	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1181274943435196	ANACARDIC ACID	iuphar.ligand:6999	ANACARDIC ACID	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.018619742	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.034453853	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.03043923	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.013022736	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	GNF-PF-3501	chembl:CHEMBL581910	CHEMBL:CHEMBL581910	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.015184405	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	SJ000047240	chembl:CHEMBL590706	CHEMBL:CHEMBL590706	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	25-HYDROXYCHOLECALCIFEROL	rxcui:1855064	CALCIFEDIOL ANHYDROUS	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	MMV007363	chembl:CHEMBL601528	CHEMBL:CHEMBL601528	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	DTC	9/2/20	NULL	0.088396753	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	2.442217266776488	NICOXAMAT	ncit:C77068	NICOXAMAT	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	URAPIDIL	rxcui:39230	URAPIDIL	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.015215205	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.025390557	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	GNF-PF-1529	chembl:CHEMBL586078	CHEMBL:CHEMBL586078	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	CLOBENPROPIT	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
AKR1B10	hgnc:382	AKR1B10	DTC	9/2/20	NULL	5.250767124	OLEANOLIC_ACID	iuphar.ligand:3306	OLEANOLIC ACID	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.025588534	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2778183663264259	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ALTRENOGEST	rxcui:1314612	ALTRENOGEST	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TRIFLUPROMAZINE HYDROCHLORIDE	rxcui:91125	TRIFLUPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	MURUCOIDIN V	chembl:CHEMBL505000	MURUCOIDIN V	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	METHYL ISOBUTYL KETONE	rxcui:1362929	METHYL ISOBUTYL KETONE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.010554306	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	TCMDC-124022	chembl:CHEMBL548017	CHEMBL:CHEMBL548017	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.023620185	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	DTC	9/2/20	NULL	2.917092846427472	AZD-9272	iuphar.ligand:6439	AZD9272	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.2592971419046642	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	IDEBENONE	rxcui:51296	IDEBENONE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.036925226	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	5-HYDROXYINDOLACETIC ACID	iuphar.ligand:11900	5-HYDROXYINDOLEACETIC ACID	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	2.019525817	BERKELEYACETAL C	chembl:CHEMBL400716	BERKELEYACETAL C	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.013964806	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002784371	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.2500365296937833	ERGOCORNINE	chembl:CHEMBL1385840	ERGOCORNINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	CLADRIBINE	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	AM580	iuphar.ligand:2647	RO 40-6055	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	NSC-125034	chembl:CHEMBL239439	CHEMBL:CHEMBL239439	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.3281729452230906	TCMDC-125221	chembl:CHEMBL546649	CHEMBL:CHEMBL546649	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	GALANGIN	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.039899446	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	DTC	9/2/20	NULL	0.2224901323546377	CGS-27023A	iuphar.ligand:8846	CGS-27023A	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.02726255	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	GNF-PF-710	chembl:CHEMBL596839	CHEMBL:CHEMBL596839	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.00453826	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1562728310586145	DIHYDROERGOCRISTINE MESYLATE	ncit:C75939	DIHYDROERGOCRISTINE MESYLATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	TCMDC-125773	chembl:CHEMBL528451	CHEMBL:CHEMBL528451	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	LINTITRIPT	ncit:C66017	LINTITRIPT	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	NAFTIDROFURYL	ncit:C87212	NAFTIDROFURYL	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	THEONELLASTEROL G	chembl:CHEMBL1782602	THEONELLASTEROL G	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	SJ000201287	chembl:CHEMBL590900	CHEMBL:CHEMBL590900	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.093098708	TANSHINONE IIA SULFONATE	chembl:CHEMBL1473252	TANSHINONE IIA SULFONATE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	PERVILLEINE D	chembl:CHEMBL446465	PERVILLEINE D	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.3281729452230906	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.233887177	ENOBOSARM	rxcui:2168587	ENOBOSARM	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	IODOFORM	rxcui:27748	IODOFORM	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00475613	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	0.1973972602845657	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.4526523382387456	DOBUTAMINE HYDROCHLORIDE	rxcui:203121	DOBUTAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.0287871	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.009734459	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.052090944	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002951527	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.020025809	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	inhibitor	0.033658764	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	TESMILIFENE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
TACR3	hgnc:11528	TACR3	DTC	9/2/20	NULL	5.834185692854944	RO-4583298	chembl:CHEMBL2203703	CHEMBL:CHEMBL2203703	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.010975684	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	OXOPURPUREINE	chembl:CHEMBL456295	OXOPURPUREINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002663877	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	FLUOXASTROBIN	chembl:CHEMBL1902591	FLUOXASTROBIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	SERTACONAZOLE NITRATE	rxcui:236601	SERTACONAZOLE NITRATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	URAPIDIL	rxcui:39230	URAPIDIL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	SCLAREOL	chembl:CHEMBL294740	SCLAREOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	FURAZOLIDONE	rxcui:4601	FURAZOLIDONE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	TREQUINSIN	ncit:C152731	TREQUINSIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.084963869	QUINALDINE BLUE	chembl:CHEMBL1433292	QUINALDINE BLUE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.076098074	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
HEXA	hgnc:4878	HEXA	DTC	9/2/20	NULL	10.50153424713889	THIOCORALINE	chembl:CHEMBL487913	THIOCORALINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	7-NITROINDAZOLE	drugbank:DB02207	7-NITROINDAZOLE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	8-[(3-TRIFLUOROMETHYL)BENZYLOXY]CAFFEINE	chembl:CHEMBL602466	CHEMBL:CHEMBL602466	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.083744292	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TOLYLFLUANID	chembl:CHEMBL3189057	TOLYLFLUANID	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.047561296	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
PLD1	hgnc:9067	PLD1	DTC	9/2/20	NULL	1.250182648468916	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	NIMUSTINE	ncit:C693	NIMUSTINE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.2542744369767287	ANACARDIC ACID	iuphar.ligand:6999	ANACARDIC ACID	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.1984416902331613	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.105015342	FLUOXASTROBIN	chembl:CHEMBL1902591	FLUOXASTROBIN	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	4.773424657790408	DIETHYL-2-PENTADECYLMALONATE	chembl:CHEMBL1797713	CHEMBL:CHEMBL1797713	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2628011573358083	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.2160809515872201	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
EIF2AK3	hgnc:3255	EIF2AK3	DTC	9/2/20	NULL	35.00511415712966	GSK2606414	iuphar.ligand:6740	GSK2606414	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010588359	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.029399592	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.7001022831425933	SPHINGOSINE	drugbank:DB03203	SPHINGOSINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	ZUCLOPENTHIXOL	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.006200717	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DNDI1417607	chembl:CHEMBL1588679	CHEMBL:CHEMBL1588679	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.005184407	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE	chembl:CHEMBL460508	CHEMBL:CHEMBL460508	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.03292017	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	METOPRINE	ncit:C1161	METOPRINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.013411921	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
GLI1	hgnc:4317	GLI1	DTC	9/2/20	NULL	5.834185692854944	4-METHYLENE-5BETA-HYDROPEROXYOVATODIOLIDE	chembl:CHEMBL471694	CHEMBL:CHEMBL471694	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.010777437	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.049723174	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	NIALAMIDE	rxcui:7394	NIALAMIDE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.010952789	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	CYCLOVALONE	ncit:C81040	CYCLOVALONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.008899605	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	PSORALEN	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-125150	chembl:CHEMBL534244	CHEMBL:CHEMBL534244	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	HEMATOXYLIN	drugbank:DB16871	HEMATOXYLIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE	chembl:CHEMBL152028	N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.095122593	NELFINAVIR MESYLATE	rxcui:266565	NELFINAVIR MESYLATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.009803523	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.038382801	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	SHINFLAVANONE	chembl:CHEMBL590635	SHINFLAVANONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BROMODIOLONE	chembl:CHEMBL1165553	BROMODIOLONE	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.020257589	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.077789143	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.007899454	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.021189536	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	GNF-PF-1000	chembl:CHEMBL600554	CHEMBL:CHEMBL600554	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	5,7-DIHYDROXY-4-METHYLCOUMARIN	chembl:CHEMBL12252	5,7-DIHYDROXY-4-METHYLCOUMARIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010541895	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	GALANGIN	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	DRONEDARONE	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	DTC	9/2/20	NULL	0.078136416	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	2-(P-HYDROXYBENZYL)PRODIGIOSIN	chembl:CHEMBL578220	CHEMBL:CHEMBL578220	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.3889457128569962	NSC-164459	chembl:CHEMBL1567041	CHEMBL:CHEMBL1567041	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007063179	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1666910197958555	PHENELZINE SULFATE	rxcui:8124	PHENELZINE SULFATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009009552	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.01555322	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.076098074	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1750255707856483	QUESTIOMYCIN B	chembl:CHEMBL28319	QUESTIOMYCIN B	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	OXOPURPUREINE	chembl:CHEMBL456295	OXOPURPUREINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	N-(2,4-DIMETHYLPHENYL)BENZENESULFONAMIDE	chembl:CHEMBL492651	CHEMBL:CHEMBL492651	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	ANISOMYCIN	ncit:C95312	ANISOMYCIN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIE	chembl:CHEMBL1095337	AESCULIOSIDE IIE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.018846975	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	NALOXONE HYDROCHLORIDE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.2778183663264259	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
DDO	hgnc:2727	DDO	DTC	9/2/20	NULL	35.00511415712966	5-AMINONICOTINIC ACID	chembl:CHEMBL1491941	CHEMBL:CHEMBL1491941	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002932079	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.062509132	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
HTR4	hgnc:5299	HTR4	DTC	9/2/20	NULL	2.692701089009974	6-BROMOTRYPTOPHANARGININE	chembl:CHEMBL401607	CHEMBL:CHEMBL401607	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1651184630053286	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.1902451856365742	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2365210416022274	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.035005114	IMIPRAMINE HYDROCHLORIDE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.014092236	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.1875273972703375	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.2397610558707511	HEPTACHLOR	chembl:CHEMBL194400	HEPTACHLOR	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.022099188	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00449706	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	TREQUINSIN	ncit:C152731	TREQUINSIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	HYDROCORTISONE PROBUTATE	rxcui:27196	HYDROCORTISONE PROBUTATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006555265	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.2897774350755767	NUTLIN-3	drugbank:DB17039	NUTLIN-3	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	4.594421233123269	NUTLIN-3	drugbank:DB17039	NUTLIN-3	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	DTC	9/2/20	NULL	0.2243917574174978	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.4102161815288632	5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB]	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CARBOQUONE	ncit:C342	CARBOQUONE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.2143170254518142	TCMDC-125620	chembl:CHEMBL530291	CHEMBL:CHEMBL530291	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	LEVISOPRENALINE	ncit:C74197	LEVISOPRENALINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	NITROFURAZONE	rxcui:7455	NITROFURAZONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NITROBLUE TETRAZOLIUM CHLORIDE	chembl:CHEMBL403063	NITROBLUE TETRAZOLIUM CHLORIDE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	ALAZANINE	chembl:CHEMBL578063	ALAZANINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.095122593	CHLORDANE	iuphar.ligand:2831	CHLORDANE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	NSC-50688	chembl:CHEMBL1456848	CHEMBL:CHEMBL1456848	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	2-ACETYLAMINOFLUORENE	chembl:CHEMBL311469	2-ACETYLAMINOFLUORENE	FALSE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.037239483	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	DIBUCAINE HYDROCHLORIDE	rxcui:235402	DIBUCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	DTC	9/2/20	NULL	0.3170753093942904	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	TRACAZOLATE	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	1.810609352954982	2-BENZYLIDENEHYDRAZINECARBOXIMIDAMIDE	chembl:CHEMBL1183425	CHEMBL:CHEMBL1183425	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.018860514	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	D-64131	chembl:CHEMBL140220	CHEMBL:CHEMBL140220	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.07699072	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-2776	chembl:CHEMBL578294	CHEMBL:CHEMBL578294	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	NSC-8186	chembl:CHEMBL122355	CHEMBL:CHEMBL122355	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.045265234	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GNF-PF-1509	chembl:CHEMBL576412	CHEMBL:CHEMBL576412	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1458546423213736	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	DTC	9/2/20	NULL	1.521961485092594	CARBETOCIN	ncit:C96858	CARBETOCIN	TRUE	FALSE	FALSE
RCE1	hgnc:13721	RCE1	DTC	9/2/20	NULL	3.750547945	GNF-PF-763	chembl:CHEMBL1576338	CHEMBL:CHEMBL1576338	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	OXOTREMORINE METHIODIDE	chembl:CHEMBL23957	OXOTREMORINE METHIODIDE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.002801007	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009579944	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	ICI-199,441	iuphar.ligand:11691	ICI-199441	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.013631275	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	1.400204566285186	SCUTELLARIN	iuphar.ligand:13075	SCUTELLARIN	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	2.187819634820604	NOR-BINALTORPHIMINE DIHYDROCHLORIDE	chembl:CHEMBL2374078	CHEMBL:CHEMBL2374078	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.009673484	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	ARASERTACONAZOLE	ncit:C79926	ARASERTACONAZOLE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.157680694	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00389812	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PENTOSALEN	ncit:C63672	PENTOSALEN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	EPINASTINE	rxcui:39684	EPINASTINE	TRUE	FALSE	FALSE
RCE1	hgnc:13721	RCE1	DTC	9/2/20	NULL	0.9376369863516875	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	L-687384	chembl:CHEMBL1256916	CHEMBL:CHEMBL1256916	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	DTC	9/2/20	NULL	4.375639269641208	PURMORPHAMINE	iuphar.ligand:10356	PURMORPHAMINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	SJ000201681	chembl:CHEMBL602135	CHEMBL:CHEMBL602135	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	VINPOCETINE	rxcui:24506	VINPOCETINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	TCMDC-124059	chembl:CHEMBL530733	CHEMBL:CHEMBL530733	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	CID 695758	chembl:CHEMBL260028	CHEMBL:CHEMBL260028	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013192882	IMIPRAMINE HYDROCHLORIDE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.009009552	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.010952789	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	PESUDOGINSENOSIDE RP1 METHYL ESTER	chembl:CHEMBL1288831	PESUDOGINSENOSIDE RP1 METHYL ESTER	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	7-METHOXYISOFLAVONE	chembl:CHEMBL563919	CHEMBL:CHEMBL563919	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	AZARIBINE	ncit:C1008	AZARIBINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002796829	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	GNF-PF-763	chembl:CHEMBL1576338	CHEMBL:CHEMBL1576338	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	FENITROTHION	ncit:C65655	FENITROTHION	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	TCMDC-124479	chembl:CHEMBL587259	CHEMBL:CHEMBL587259	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.004583821	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	GNF-PF-2335	chembl:CHEMBL601146	CHEMBL:CHEMBL601146	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	3-MORPHOLINOSYDNONIMINE HCL	chembl:CHEMBL538104	CHEMBL:CHEMBL538104	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1693795846312726	CHLORPYRIFOS	ncit:C163641	CHLORPYRIFOS	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	GNF-PF-1319	chembl:CHEMBL235891	CHEMBL:CHEMBL235891	FALSE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	DTC	9/2/20	NULL	0.060423097	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.4565884455277783	NOVOBIOCIN	rxcui:7538	NOVOBIOCIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	AGROCLAVINE	chembl:CHEMBL449081	AGROCLAVINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.039899446	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	A-315456	chembl:CHEMBL362863	CHEMBL:CHEMBL362863	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	3.500511415712966	VERNOLIDE-B	chembl:CHEMBL2062868	CHEMBL:CHEMBL2062868	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	GNF-PF-1731	chembl:CHEMBL581251	CHEMBL:CHEMBL581251	FALSE	FALSE	FALSE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.081030357	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.027276712	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CHLOROTRIPHENYLSTANNANE	chembl:CHEMBL515580	CHLOROTRIPHENYLSTANNANE	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.596678082	DICHLOROISOPROTERENOL	drugbank:DB12803	DICHLOROISOPROTERENOL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.015268296	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	TOLUENE DIISOCYANATE	chembl:CHEMBL1086446	TOLUENE DIISOCYANATE	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.00741215	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.045461187	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.1881995384791917	DIACEREIN	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	INDOCATE	ncit:C65912	INDOCATE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.004810597	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.004857324	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE	chembl:CHEMBL460508	CHEMBL:CHEMBL460508	FALSE	FALSE	FALSE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	0.7501095890813498	MESO-2,3-DIMERCAPTOSUCCINIC ACID	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.006466462	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1232574442152452	TCMDC-124166	chembl:CHEMBL528712	CHEMBL:CHEMBL528712	FALSE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.3500511415712967	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.015744429	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.011086924	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001844705	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.01609924	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.008103036	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	DOLASTATIN 12	chembl:CHEMBL448114	DOLASTATIN 12	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	GNF-PF-840	chembl:CHEMBL601605	CHEMBL:CHEMBL601605	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.004296863	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1988926940746003	2-(2-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL112060	CHEMBL:CHEMBL112060	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.3271505995993426	ENDOXIFEN	iuphar.ligand:10203	ENDOXIFEN	FALSE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.019607047	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	SJ000059275	chembl:CHEMBL603952	CHEMBL:CHEMBL603952	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SJ000296655	chembl:CHEMBL589734	CHEMBL:CHEMBL589734	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.007758226	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00282664	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.016590101	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	(S)-FELODIPINE	chembl:CHEMBL428768	(S)-FELODIPINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	PNU-99194A	chembl:CHEMBL16410	PNU-99194A	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.019889269	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	DIACEREIN	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
RPS6KA5	hgnc:10434	RPS6KA5	DTC	9/2/20	inhibitor	0.1875273972703375	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.072524408	HTS-05057	chembl:CHEMBL372629	CHEMBL:CHEMBL372629	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.028413242	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.2625383561784725	SJ000201681	chembl:CHEMBL602135	CHEMBL:CHEMBL602135	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	BUPRENORPHINE HYDROCHLORIDE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	A-315456	chembl:CHEMBL362863	CHEMBL:CHEMBL362863	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	NITROFURAZONE	rxcui:7455	NITROFURAZONE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	SKF-83959	iuphar.ligand:8443	SKF-83959	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.009571212	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.760980743	SR-13668	chembl:CHEMBL245030	SR-13668	FALSE	FALSE	FALSE
EPHA5	hgnc:3389	EPHA5	DTC	9/2/20	inhibitor	0.2625383561784725	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	ALBENDAZOLE	rxcui:430	ALBENDAZOLE	TRUE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.016764901	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	7-METHOXYISOFLAVONE	chembl:CHEMBL563919	CHEMBL:CHEMBL563919	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.002299841	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.045579576	A-77636	iuphar.ligand:9637	A77636	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	2-MERCAPTOPYRIMIDINE	chembl:CHEMBL1688952	2-MERCAPTOPYRIMIDINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	TRYPTOPHAN	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.02726255	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-4237	chembl:CHEMBL600701	CHEMBL:CHEMBL600701	FALSE	FALSE	FALSE
SPHK2	hgnc:18859	SPHK2	DTC	9/2/20	NULL	8.751278539282415	DIMETHYLSPINGOSINE	chembl:CHEMBL322333	DIMETHYLSPINGOSINE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.058602312	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.005310242	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	NAPHAZOLINE	rxcui:7247	NAPHAZOLINE	TRUE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	DTC	9/2/20	NULL	2.838252499226729	BANOXANTRONE	ncit:C79528	BANOXANTRONE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.081407242	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	CITRONELLOL	chembl:CHEMBL395827	CITRONELLOL	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1112450661773188	DIHYDREXIDINE HYDROCHLORIDE	chembl:CHEMBL1256832	DIHYDREXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004191225	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004427291	SKF-82526	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.0287871	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2703097618311171	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.3659071166250487	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2778183663264258	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.042619863	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	NSC-3323	chembl:CHEMBL1270169	CHEMBL:CHEMBL1270169	FALSE	FALSE	FALSE
PTK6	hgnc:9617	PTK6	DTC	9/2/20	NULL	0.081030357	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.01439355	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	GNF-PF-2947	chembl:CHEMBL581677	CHEMBL:CHEMBL581677	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	(+)-TETRAHYDROBERBERINE	chembl:CHEMBL476501	CHEMBL:CHEMBL476501	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	DNDI1417013	chembl:CHEMBL1452227	CHEMBL:CHEMBL1452227	FALSE	FALSE	FALSE
GLA	hgnc:4296	GLA	DTC	9/2/20	NULL	4.039051633514961	L-GLUTAMIC ACID, N-PHTHALOYL	chembl:CHEMBL1256390	CHEMBL:CHEMBL1256390	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007378818	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	ACRIDONE	chembl:CHEMBL436589	ACRIDONE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.014160645	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004120188	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	DTC	9/2/20	NULL	4.773424657790408	3-FORMYLINDOLE	chembl:CHEMBL147741	3-FORMYLINDOLE	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	0.3571950424196904	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	SJ000024939	chembl:CHEMBL590691	CHEMBL:CHEMBL590691	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	ALLITRIDIN	chembl:CHEMBL123040	ALLITRIDIN	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.036237178	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.095122593	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	LEMILDIPINE	ncit:C170102	LEMILDIPINE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.048349605	GNF-PF-3501	chembl:CHEMBL581910	CHEMBL:CHEMBL581910	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.009368006	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	THIOSALICYLIC ACID	rxcui:322165	THIOSALICYLIC ACID	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-739452	chembl:CHEMBL408564	CHEMBL:CHEMBL408564	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.017059022	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.1704794520639432	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	inhibitor	0.026789628	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.7395446652914718	BISLEUCONOTHINE A	chembl:CHEMBL1077259	BISLEUCONOTHINE A	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	SJ000001592	chembl:CHEMBL591834	CHEMBL:CHEMBL591834	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.004764761	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	TCMDC-124354	chembl:CHEMBL546344	CHEMBL:CHEMBL546344	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIIC	chembl:CHEMBL1095341	AESCULIOSIDE IIIC	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	TCMDC-125653	chembl:CHEMBL580918	CHEMBL:CHEMBL580918	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	GNF-PF-3350	chembl:CHEMBL600747	CHEMBL:CHEMBL600747	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.026626608	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.019799273	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BENORILATE	rxcui:1372	BENORILATE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	GNF-PF-710	chembl:CHEMBL596839	CHEMBL:CHEMBL596839	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	0.092606122	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	SCOPOLETIN	chembl:CHEMBL71851	SCOPOLETIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	5,7-DIHYDROXY-4-METHYLCOUMARIN	chembl:CHEMBL12252	5,7-DIHYDROXY-4-METHYLCOUMARIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	SOBUZOXANE	ncit:C66540	SOBUZOXANE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.053253216	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	NELFINAVIR MESYLATE	rxcui:266565	NELFINAVIR MESYLATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.6863747873946993	TRIDOLGOSIR	ncit:C152742	TRIDOLGOSIR	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1293292394967844	NSC-8186	chembl:CHEMBL122355	CHEMBL:CHEMBL122355	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.007869855	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.024008995	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.032055965	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.01787191	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004674828	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-3949	chembl:CHEMBL528390	CHEMBL:CHEMBL528390	FALSE	FALSE	FALSE
POLD1	hgnc:9175	POLD1	DTC	9/2/20	NULL	4.375639269641208	HYMENOIC ACID	chembl:CHEMBL494213	HYMENOIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	MMV007764	chembl:CHEMBL609628	CHEMBL:CHEMBL609628	FALSE	FALSE	FALSE
BBOX1	hgnc:964	BBOX1	DTC	9/2/20	NULL	1.521961485092594	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.010405801	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	NSC-119889	chembl:CHEMBL516616	CHEMBL:CHEMBL516616	FALSE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.045265234	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2910624791335615	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	0.6819178082557728	OXYMORPHONE	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.3059887601147698	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.024008995	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001169436	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	OXYPHENISATIN ACETATE	ncit:C170278	OXYPHENISATIN ACETATE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.01644462	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	METHYLTESTOSTERONE	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
AGTR2	hgnc:338	AGTR2	DTC	9/2/20	NULL	3.182283105193605	AZD-4017	drugbank:DB14875	AZD-4017	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	SJ000032151	chembl:CHEMBL592600	CHEMBL:CHEMBL592600	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	ISOCARBOXAZID	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.022730594	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	DIENOCHLOR	chembl:CHEMBL1355965	DIENOCHLOR	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-625137A	chembl:CHEMBL230911	GSK-625137A	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	TRIBROMSALAN	ncit:C47768	TRIBROMSALAN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	D-64131	chembl:CHEMBL140220	CHEMBL:CHEMBL140220	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.036463661	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	DTC	9/2/20	NULL	11.66837138570988	4-(4-ETHOXYPHENOXY)PHENOL	chembl:CHEMBL455078	CHEMBL:CHEMBL455078	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.033875917	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	BENZIODARONE	ncit:C74127	BENZIODARONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	KINETIN RIBOSIDE	chembl:CHEMBL411066	KINETIN RIBOSIDE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.02896975	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	MONASTROL	drugbank:DB04331	MONASTROL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	AVOCADYNE ACETATE	chembl:CHEMBL1396170	AVOCADYNE ACETATE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.096123883	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	CID 695758	chembl:CHEMBL260028	CHEMBL:CHEMBL260028	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	DTC	9/2/20	NULL	0.1136529680426287	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	HALOPROGIN	rxcui:26422	HALOPROGIN	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1715936968486748	PROCATEROL	rxcui:34530	PROCATEROL	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.046059361	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	CLOBENPROPIT	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.065964411	DIENOCHLOR	chembl:CHEMBL1355965	DIENOCHLOR	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.038270897	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.8751278539282416	GNF-PF-4328	chembl:CHEMBL597452	CHEMBL:CHEMBL597452	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	TELENZEPINE	ncit:C75285	TELENZEPINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	GNF-PF-2307	chembl:CHEMBL421088	CHEMBL:CHEMBL421088	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	L-701324	iuphar.ligand:4240	L701324	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.042863405	GNF-PF-3201	chembl:CHEMBL581872	CHEMBL:CHEMBL581872	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	GALUTEOLIN	chembl:CHEMBL233929	GALUTEOLIN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	LICOFLAVANONE A	chembl:CHEMBL506929	LICOFLAVANONE A	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.002977807	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
TSSK2	hgnc:11401	TSSK2	DTC	9/2/20	NULL	0.1117184494376478	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	DTC	9/2/20	NULL	0.025244073	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1013661606866689	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	7,3'-DIHYDROXYFLAVONE	chembl:CHEMBL253786	CHEMBL:CHEMBL253786	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.2476776945079929	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2651902587661338	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
HRH4	hgnc:17383	HRH4	DTC	9/2/20	NULL	9.546849315580817	VUF-10497	chembl:CHEMBL452847	CHEMBL:CHEMBL452847	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.023274677	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011738804	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	TCMDC-123769	chembl:CHEMBL534353	CHEMBL:CHEMBL534353	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.036847489	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	DTC	9/2/20	NULL	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	1.500219178	BAS-8770931	chembl:CHEMBL515495	CHEMBL:CHEMBL515495	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.014545061	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.1105424657593568	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011850072	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	DTC	9/2/20	NULL	0.1172046232939609	TCMDC-124059	chembl:CHEMBL530733	CHEMBL:CHEMBL530733	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.04464938	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.046303061	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	DNDI1417447	chembl:CHEMBL1307453	CHEMBL:CHEMBL1307453	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NS-1619	iuphar.ligand:4272	NS1619	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	A-315456	chembl:CHEMBL362863	CHEMBL:CHEMBL362863	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2117244807890907	DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE	iuphar.ligand:5445	N-DOCOSATETRA-7,10,13,16-ENOYLETHANOLAMINE	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.2763561643983921	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.1458546423213736	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	GNF-PF-704	chembl:CHEMBL597449	CHEMBL:CHEMBL597449	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	THEONELLASTEROL G	chembl:CHEMBL1782602	THEONELLASTEROL G	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.08334551	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	SJ000047240	chembl:CHEMBL590706	CHEMBL:CHEMBL590706	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	DEHYDROEPIANDROSTERONE ACETATE	chembl:CHEMBL1480686	DEHYDROEPIANDROSTERONE ACETATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003840807	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	1.615620653405984	2-(4-NITROPHENYL)BENZO[D]THIAZOLE	chembl:CHEMBL477841	CHEMBL:CHEMBL477841	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	LAPACHOL	chembl:CHEMBL15193	LAPACHOL	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	QUINOLIN-6-YLAMINE	chembl:CHEMBL99408	CHEMBL:CHEMBL99408	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.016764901	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	THIOLUTIN	ncit:C64175	THIOLUTIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004540811	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.062509132	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.1835932560688619	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	4,4'-DIMETHOXYDALBERGIONE	chembl:CHEMBL1436980	4,4'-DIMETHOXYDALBERGIONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007699637	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1296485709523321	QUESTIOMYCIN B	chembl:CHEMBL28319	QUESTIOMYCIN B	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.035430277	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	TANGERETIN	chembl:CHEMBL73930	TANGERETIN	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.045461187	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	PHYLLODULCIN	chembl:CHEMBL303483	PHYLLODULCIN	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1750255707856483	NAPHTHOQUINONE	chembl:CHEMBL55934	NAPHTHOQUINONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	ISRAPAFANT	ncit:C65987	ISRAPAFANT	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.7242437411819931	CH-5015765	chembl:CHEMBL1834096	CHEMBL:CHEMBL1834096	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	DTC	9/2/20	NULL	0.1143957978991165	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	GNF-PF-3350	chembl:CHEMBL600747	CHEMBL:CHEMBL600747	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	(+)-CIS-DIOXOLANE IODIDE	chembl:CHEMBL387632	CHEMBL:CHEMBL387632	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	DTC	9/2/20	NULL	0.1018248310970158	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW829115X	chembl:CHEMBL188794	GW829115X	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.9907107780319716	GNF-PF-1609	chembl:CHEMBL600956	CHEMBL:CHEMBL600956	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.019065966	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.061412481	FRAXETIN	chembl:CHEMBL54909	FRAXETIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	THIOPERAMIDE	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	2.386712328895204	TETRAHYDROCURCUMIN	chembl:CHEMBL318743	TETRAHYDROCURCUMIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	4,4'-DIHYDROXYDIPHENYLMETHANE	chembl:CHEMBL138061	CHEMBL:CHEMBL138061	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.072927321	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	THIDIAZURON	chembl:CHEMBL505661	THIDIAZURON	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	DIFLUBENZURON	rxcui:1665336	DIFLUBENZURON	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.150021918	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	1.500219178	TCMDC-125278	chembl:CHEMBL588327	CHEMBL:CHEMBL588327	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.038894571	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	NSC-119889	chembl:CHEMBL516616	CHEMBL:CHEMBL516616	FALSE	FALSE	FALSE
PML-RARA	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Arsenic Trioxide	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.1535312024435511	Ado-Trastuzumab Emtansine	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	4.702860988936115	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.01402074	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	ETHOPROPAZINE HYDROCHLORIDE	rxcui:6541	ETHOPROPAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.5000730593875667	Blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
HBB	hgnc:4827	HBB	FDA	10-Apr-24	NULL	1.810609352954982	Crizanlizumab-tmca	rxcui:2262279	CRIZANLIZUMAB	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	FDA	10-Apr-24	NULL	0.364636606	Eltrombopag	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
STX11	hgnc:11429	STX11	FDA	10-Apr-24	NULL	13.12691780892362	Emapalumab-lzsg	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
UNC13D	hgnc:23147	UNC13D	FDA	10-Apr-24	NULL	13.12691780892362	Emapalumab-lzsg	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.015702055	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	FDA	10-Apr-24	NULL	0.076765601	Oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.01090502	Pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	3.150460274	Velpatasvir	rxcui:1799206	VELPATASVIR	TRUE	FALSE	FALSE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Tipiracil	rxcui:10803	TRIFLURIDINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1312691780892362	Tolbutamide	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
AURKC	hgnc:11391	AURKC	MyCancerGenome	20-Jun-17	inhibitor	0.3182283105193606	BI847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.142490288	BI847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	MyCancerGenome	20-Jun-17	inhibitor	0.07463777	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.1984416902331613	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	MyCancerGenome	20-Jun-17	inhibitor	0.6806549974997433	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.079376676	AZD8931	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	MyCancerGenome	20-Jun-17	inhibitor	0.1022876712383659	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	MyCancerGenome	20-Jun-17	inhibitor	0.5834185692854945	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	MyCancerGenome	20-Jun-17	inhibitor	0.159436249	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	antibody	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	antibody	0.2917092846427472	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.03043923	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2108741816694558	4'-N-BENZOYLSTAUROSPORINE	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	MyCancerGenome	20-Jun-17	other/unknown	15.31473744374422	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.063331621	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.159436249	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.6050266644442165	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.076934317	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1154014752432846	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ABCC6	hgnc:57	ABCC6	NCI	14-Sep-17	NULL	0.1944728564284981	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
ACO1	hgnc:117	ACO1	NCI	14-Sep-17	NULL	1.666910197958555	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	NULL	CHELATORS	NULL	NULL	NULL	NULL	NULL
ADAMTS4	hgnc:220	ADAMTS4	NCI	14-Sep-17	NULL	11.66837138570989	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
ADIPOQ	hgnc:13633	ADIPOQ	NCI	14-Sep-17	NULL	1.640864726115453	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.098513454	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.252440727	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.029698909	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.2536602475154323	FUROSEMIDE	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
ATF3	hgnc:785	ATF3	NCI	14-Sep-17	NULL	0.2542744369767288	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.016869935	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.040005845	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.080781033	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1909369863116163	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.015386863	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	0.1141471113819445	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.082364974	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	NCI	14-Sep-17	NULL	0.051885051	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CCL1	hgnc:10609	CCL1	NCI	14-Sep-17	NULL	3.182283105193606	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.080471527	CICLOSPORIN	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CCK	hgnc:1569	CCK	NCI	14-Sep-17	NULL	0.9460841664089098	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.3684748858645228	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.2258394461750301	INFLIXIMAB	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.024041974	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.1389091831632129	CHEMOPREVENTIVE	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
CCR3	hgnc:1604	CCR3	NCI	14-Sep-17	NULL	0.4487835148349958	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	NCI	14-Sep-17	NULL	14.58546423213736	HLL2	ncit:C1887	EPRATUZUMAB	FALSE	FALSE	FALSE
CD4	hgnc:1678	CD4	NCI	14-Sep-17	NULL	0.1988926940746004	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	0.100589408	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.048282916	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	0.1458546423213736	RECOMBINANT HUMAN IL-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
CD83	hgnc:1703	CD83	NCI	14-Sep-17	NULL	2.187819634820604	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.014987205	DNR	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CDKN2C	hgnc:1789	CDKN2C	NCI	14-Sep-17	NULL	0.6364566210387212	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	NCI	14-Sep-17	NULL	0.1383601350084176	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
CGA	hgnc:1885	CGA	NCI	14-Sep-17	NULL	0.3201687270469177	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CRMP1	hgnc:2365	CRMP1	NCI	14-Sep-17	NULL	0.2500365296937833	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.006324701	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.3409589041278864	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	0.6731752722524935	ETHER	ncit:C29819	ETHER	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.9053046764774912	RAS INHIBITORS	ncit:C1902	RAS INHIBITOR	FALSE	FALSE	FALSE
EPO	hgnc:3415	EPO	NCI	14-Sep-17	NULL	NULL	CHELATORS	NULL	NULL	NULL	NULL	NULL
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.0191914	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.049349315	FLUORODEOXYURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1238388472539964	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	NCI	14-Sep-17	NULL	1.312691780892362	IL-5	iuphar.ligand:4997	IL-5	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.3535870116881784	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.7955707762984014	LACTULOSE	rxcui:6218	LACTULOSE	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.7955707762984014	MAFOSFAMIDE	ncit:C1150	MAFOSFAMIDE	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.7955707762984014	POLY I:C	ncit:C758	POLY IC	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	NCI	14-Sep-17	NULL	2.234368988752957	FGF-6	iuphar.ligand:4927	FGF-6	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.315361389	CALCIUM CHANNEL BLOCKER	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.1750255707856483	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.7001022831425934	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.2470949234620917	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	NULL	CAROTENE	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	NULL	ETHYLNITROSOUREA	NULL	NULL	NULL	NULL	NULL
GADD45A	hgnc:4095	GADD45A	NCI	14-Sep-17	NULL	NULL	CHELATORS	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.2500365296937833	SULFORAPHANE	ncit:C1424	SULFORAPHANE	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1416573864272333	IUPHAR.LIGAND:5691	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
H2AFX	hgnc:4739	H2AX	NCI	14-Sep-17	NULL	1.000146118775133	N-ACETYLCYSTEINE	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.4039051633514962	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	NCI	14-Sep-17	NULL	0.7242437411819931	PIMONIDAZOLE	ncit:C1196	PIMONIDAZOLE	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	NULL	CHELATORS	NULL	NULL	NULL	NULL	NULL
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	0.2983390411119005	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	NCI	14-Sep-17	NULL	1.500219178162699	LYMPHOKINES	ncit:C621	RECOMBINANT LYMPHOKINE	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	0.7292732116068681	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.325124899	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	2.763561643983921	AUTOLOGOUS DENDRITIC CELLS	ncit:C2594	THERAPEUTIC AUTOLOGOUS DENDRITIC CELLS	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.034544521	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	NULL	CHELATORS	NULL	NULL	NULL	NULL	NULL
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.092851762	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
HSPA8	hgnc:5241	HSPA8	NCI	14-Sep-17	NULL	0.3860858179095184	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	NCI	14-Sep-17	NULL	0.051782713	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
HUS1	hgnc:5309	HUS1	NCI	14-Sep-17	NULL	1.500219178	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	2.625383561784724	LISOFYLLINE	ncit:C1516	LISOFYLLINE	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	1.312691780892362	PROTON PUMP INHIBITOR	ncit:C29723	PROTON PUMP INHIBITOR	FALSE	FALSE	FALSE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	0.3977853881492008	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	NCI	14-Sep-17	NULL	NULL	GRANULOCYTE COLONY-STIMULATING FACTOR	NULL	NULL	NULL	NULL	NULL
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.6908904109959803	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.1348078850723864	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.5357925636295356	METRONIDAZOLE	rxcui:6922	METRONIDAZOLE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.024932417	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.2592971419046642	CI-1033	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
LOH19CR1	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.577007376	METOCLOPRAMIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	NCI	14-Sep-17	NULL	NULL	OPIOID	NULL	NULL	NULL	NULL	NULL
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.5357925636295356	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.1715936968486748	LGD1069	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.024163678	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	1.591141552596803	NITROSOUREAS	ncit:C699	NITROSOUREA COMPOUND	FALSE	FALSE	FALSE
MDH2	hgnc:6971	MDH2	NCI	14-Sep-17	NULL	1.250182648468916	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	1.166837138570988	TOLMETIN	rxcui:10636	TOLMETIN	TRUE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:10662	iuphar.ligand:10662	BMS-986260	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1666910197958555	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.037505479	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	NULL	EF-1	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.007869855	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	NULL	PHOSPHATE BUFFER	NULL	NULL	NULL	NULL	NULL
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.03607535	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.6482428547616605	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.4930297768609811	GREEN TEA EXTRACT	rxcui:283567	GREEN TEA LEAF EXTRACT	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	NCI	14-Sep-17	NULL	NULL	ENU	NULL	NULL	NULL	NULL	NULL
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.077066054	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	0.3153613888029699	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	1.166837138570989	NORETHISTERONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.009723643	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.054020238	SELECTIVE ESTROGEN RECEPTOR MODULATOR	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.014126358	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.023813003	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	NCI	14-Sep-17	NULL	0.017679351	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
NCBIGENE:1662	hgnc:2735	DDX10	GuideToPharmacology	2024.1	inhibitor	0.42006137	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
PMAIP1	hgnc:9108	PMAIP1	NCI	14-Sep-17	NULL	1.221108633388244	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PPA1	hgnc:9226	PPA1	NCI	14-Sep-17	NULL	52.50767123569449	GUANIDINIUM	ncit:C1375	GUANIDINIUM CATION	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	0.364636606	CHEMOPREVENTIVE AGENT	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.2430910705356226	CALCIUM CHANNEL BLOCKER	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	NULL	CAROTENOIDS	NULL	NULL	NULL	NULL	NULL
RPE65	hgnc:10294	RPE65	NCI	14-Sep-17	NULL	0.1648592503475494	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.088996053	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	NCI	14-Sep-17	NULL	0.5357925636295356	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
TBXA2R	hgnc:11608	TBXA2R	NCI	14-Sep-17	NULL	0.4167275494896389	FUROSEMIDE	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	NCI	14-Sep-17	NULL	0.060008767	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.6731752722524935	IL-8	ncit:C1289	RECOMBINANT INTERLEUKIN-8	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.045639002	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12112	iuphar.ligand:12112	NTQ1062	FALSE	FALSE	FALSE
THBS2	hgnc:11786	THBS2	NCI	14-Sep-17	NULL	1.312691780892362	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.094099769	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.2822993077187876	PROTON PUMP INHIBITOR	ncit:C29723	PROTON PUMP INHIBITOR	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.066423367	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	NULL	DAB	NULL	NULL	NULL	NULL	NULL
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.025865848	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.061725319	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.1159109740302306	L-744,832	ncit:C1682	L-744,832	FALSE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.1049104320393496	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.06584034	CDDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.064033745	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
NCBIGENE:2595	hgnc:4139	GANC	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6919	iuphar.ligand:6919	PRUNETIN	FALSE	FALSE	FALSE
TPO	hgnc:12015	TPO	NCI	14-Sep-17	NULL	0.2885036881082115	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.055859225	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
TSPYL2	hgnc:24358	TSPYL2	NCI	14-Sep-17	NULL	0.2885036881082115	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	1.117184494376478	ENILURACIL	ncit:C1773	ENILURACIL	FALSE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	NCI	14-Sep-17	NULL	0.16256245	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.012386806	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.006370357	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
VIM	hgnc:12692	VIM	NCI	14-Sep-17	NULL	NULL	ENU	NULL	NULL	NULL	NULL	NULL
CHRNA3	hgnc:1957	CHRNA3	PharmGKB	4/5/24	NULL	0.1591141552596803	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.012794267	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
SLC22A16	hgnc:20302	SLC22A16	PharmGKB	4/5/24	NULL	NULL	doxorubicinol	NULL	NULL	NULL	NULL	NULL
AKR1A1	hgnc:380	AKR1A1	PharmGKB	4/5/24	NULL	NULL	doxorubicinol	NULL	NULL	NULL	NULL	NULL
CBR1	hgnc:1548	CBR1	PharmGKB	4/5/24	NULL	NULL	doxorubicinol	NULL	NULL	NULL	NULL	NULL
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.3125456621172291	rasagiline	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.546954909	lumefantrine	rxcui:847728	LUMEFANTRINE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.095122593	erythromycin	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:7890	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	NULL	vitamin b-complex, plain	NULL	NULL	NULL	NULL	NULL
MTRR	hgnc:7473	MTRR	PharmGKB	4/5/24	NULL	NULL	vitamin b-complex, plain	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	Phenothiazine derivatives	NULL	NULL	NULL	NULL	NULL
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	0.364636606	eltrombopag	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.027121731	felbamate	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	NULL	clozapine n-oxide	NULL	NULL	NULL	NULL	NULL
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.5645986154375752	alirocumab	rxcui:1659152	ALIROCUMAB	TRUE	FALSE	FALSE
CHST13	hgnc:21755	CHST13	PharmGKB	4/5/24	NULL	3.621218705909965	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	NULL	17beta-estradiol glucuronide	NULL	NULL	NULL	NULL	NULL
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	NULL	purine analogues	NULL	NULL	NULL	NULL	NULL
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.016023092	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.038722471	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	NULL	xenobiotics	NULL	NULL	NULL	NULL	NULL
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.03319069	phenylbutazone	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.029041854	miconazole	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.051629962	modafinil	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	6.300920548	ledipasvir	rxcui:1591922	LEDIPASVIR	TRUE	FALSE	FALSE
CLCN6	hgnc:2024	CLCN6	PharmGKB	4/5/24	NULL	0.3500511415712966	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	NULL	cabotegravir / rilpivirine	NULL	NULL	NULL	NULL	NULL
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	NULL	cabotegravir / rilpivirine	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.002132378	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	Paracetamol, combinations excl. Psycholeptics (Vicks MediNait Sirup)	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	Paracetamol, combinations excl. Psycholeptics (Vicks MediNait Sirup)	NULL	NULL	NULL	NULL	NULL
COL1A1	hgnc:2197	COL1A1	PharmGKB	4/5/24	NULL	0.2631963470460877	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	NULL	n-desethyl sunitinib	NULL	NULL	NULL	NULL	NULL
SLC26A8	hgnc:14468	SLC26A8	PharmGKB	4/5/24	NULL	2.917092846427472	adefovir dipivoxil	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
SLCO3A1	hgnc:10952	SLCO3A1	PharmGKB	4/5/24	NULL	11.66837138570988	darunavir	rxcui:460132	DARUNAVIR	TRUE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:11838	iuphar.ligand:11838	BMS-986224	FALSE	FALSE	FALSE
ANO2	hgnc:1183	ANO2	PharmGKB	4/5/24	NULL	4.039051633514962	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GPX3	hgnc:4555	GPX3	PharmGKB	4/5/24	NULL	0.1750255707856483	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	1.193356164447602	bucillamine	ncit:C83561	BUCILLAMINE	FALSE	FALSE	FALSE
TCF7L2	hgnc:11641	TCF7L2	PharmGKB	4/5/24	NULL	0.7369497717290455	sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NT5C	hgnc:17144	NT5C	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NT5C1A	hgnc:17819	NT5C1A	PharmGKB	4/5/24	NULL	0.3763990769583835	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.2169738480813822	cabazitaxel	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
ZNF804A	hgnc:21711	ZNF804A	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.9010915075351876	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:1614	hgnc:13557	ACE2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:12820	iuphar.ligand:12820	BCY15291	FALSE	FALSE	FALSE
BTC	hgnc:1121	BTC	PharmGKB	4/5/24	NULL	0.182318303	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NRG3	hgnc:7999	NRG3	PharmGKB	4/5/24	NULL	0.2917092846427472	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.7001022831425934	ropivacaine	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
GATA4	hgnc:4173	GATA4	PharmGKB	4/5/24	NULL	NULL	Drugs used in alcohol dependence	NULL	NULL	NULL	NULL	NULL
FSTL5	hgnc:21386	FSTL5	PharmGKB	4/5/24	NULL	NULL	purine analogues	NULL	NULL	NULL	NULL	NULL
IL6ST	hgnc:6021	IL6ST	PharmGKB	4/5/24	NULL	NULL	purine analogues	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6375	rxcui:1546196	BENAZEPRILAT	TRUE	FALSE	FALSE
PACSIN2	hgnc:8571	PACSIN2	PharmGKB	4/5/24	NULL	NULL	purine analogues	NULL	NULL	NULL	NULL	NULL
RAC1	hgnc:9801	RAC1	PharmGKB	4/5/24	NULL	NULL	purine analogues	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.011591097	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.006439499	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
SULT1A1	hgnc:11453	SULT1A1	PharmGKB	4/5/24	NULL	NULL	desmethylnaproxen	NULL	NULL	NULL	NULL	NULL
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	NULL	catecholamines	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	lidocaine / prilocaine	NULL	NULL	NULL	NULL	NULL
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
RGS19	hgnc:13735	RGS19	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
ADRA1D	hgnc:280	ADRA1D	PharmGKB	4/5/24	NULL	NULL	Alpha-adrenoreceptor antagonists	NULL	NULL	NULL	NULL	NULL
NCBIGENE:696	hgnc:1135	BTN1A1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	NULL	Alpha-adrenoreceptor antagonists	NULL	NULL	NULL	NULL	NULL
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	NULL	Alpha-adrenoreceptor antagonists	NULL	NULL	NULL	NULL	NULL
NPPA-AS1	hgnc:37635	NPPA-AS1	PharmGKB	4/5/24	NULL	2.917092846427472	torasemide	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	PharmGKB	4/5/24	NULL	0.729273212	torasemide	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.022249013	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
MDGA2	hgnc:19835	MDGA2	PharmGKB	4/5/24	NULL	5.000730593875666	milnacipran	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
IGH	hgnc:5477	IGH	PharmGKB	4/5/24	NULL	6.563458904461812	pirtobrutinib	rxcui:2629338	PIRTOBRUTINIB	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.729273212	daniquidone	ncit:C66984	DANIQUIDONE	FALSE	FALSE	FALSE
DVL2	hgnc:3086	DVL2	PharmGKB	4/5/24	NULL	0.4449802647092754	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NUP107	hgnc:29914	NUP107	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NCBIGENE:693	hgnc:1129	BTF3P1	GuideToPharmacology	2024.1	activator	5.250767124	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.007179391	chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	0.3977853881492006	roflumilast	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.3633748874442526	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.2853677784548614	bleomycin	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
PARP14	hgnc:29232	PARP14	PharmGKB	4/5/24	NULL	NULL	6-hydroxy s-warfarin	NULL	NULL	NULL	NULL	NULL
NKX2-5	hgnc:2488	NKX2-5	PharmGKB	4/5/24	NULL	0.2983390411119005	levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
NCBIGENE:1244	hgnc:53	ABCC2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8806	iuphar.ligand:8806	A1P	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.095122593	levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	activator	0.2125816649218401	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:5603	iuphar.ligand:5603	CPFPX	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.05486695	IUPHAR.LIGAND:372	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	NULL	2-hydroxyatorvastatin	NULL	NULL	NULL	NULL	NULL
AXIN2	hgnc:904	AXIN2	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1207072901969988	IUPHAR.LIGAND:5595	ncit:C174671	BINODENOSON	FALSE	FALSE	FALSE
CRYBG2	hgnc:17295	CRYBG2	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:10235	iuphar.ligand:10235	MRS7469	FALSE	FALSE	FALSE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.2561349816375341	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	bisoprolol fumarate / perindopril arginine	NULL	NULL	NULL	NULL	NULL
APCDD1	hgnc:15718	APCDD1	PharmGKB	4/5/24	NULL	NULL	Dihydropyridine derivatives	NULL	NULL	NULL	NULL	NULL
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.017751072	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
NUMA1	hgnc:8059	NUMA1	PharmGKB	4/5/24	NULL	NULL	Dihydropyridine derivatives	NULL	NULL	NULL	NULL	NULL
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.040235763	IUPHAR.LIGAND:2844	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	PharmGKB	4/5/24	NULL	NULL	methylcholanthrene	NULL	NULL	NULL	NULL	NULL
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	0.017951341	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2A7P1	hgnc:2612	CYP2A7P1	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
DHCR7	hgnc:2860	DHCR7	PharmGKB	4/5/24	NULL	4.375639269641208	cholic acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:389	iuphar.ligand:389	L-97-1	FALSE	FALSE	FALSE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	NULL	aminoglycoside antibacterials	NULL	NULL	NULL	NULL	NULL
CACNA2D3	hgnc:15460	CACNA2D3	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
TTR	hgnc:12405	TTR	PharmGKB	4/5/24	NULL	4.375639269641208	eplontersen	rxcui:2671939	EPLONTERSEN	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.2476776945079929	halothane	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.066172238	erythromycin	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.078136416	fruquintinib	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.060737619	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CPS1	hgnc:2323	CPS1	PharmGKB	4/5/24	NULL	3.000438356	methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.251232877	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	vindesine	rxcui:11204	VINDESINE	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	NULL	norfentanyl	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	NULL	2-hydroxyatorvastatin	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	lumefantrine	rxcui:847728	LUMEFANTRINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.015662243	tropisetron	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006525935	lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.019577804	teneligliptin	ncit:C87623	TENELIGLIPTIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.010678802	granisetron	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
HLA-DOB	hgnc:4937	HLA-DOB	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:396	iuphar.ligand:396	MRS1066	FALSE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.076934317	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.1296485709523321	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.070690956	pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MALAT1	hgnc:29665	MALAT1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	NULL	Analgesics and anesthetics	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.039688338	geldanamycin	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.04427291	albendazole	rxcui:430	ALBENDAZOLE	TRUE	FALSE	FALSE
IGF2-AS	hgnc:14062	IGF2-AS	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:405	drugbank:DB08770	4-{2-[(7-AMINO-2-FURAN-2-YL[1,2,4]TRIAZOLO[1,5-A][1,3,5]TRIAZIN-5-YL)AMINO]ETHYL}PHENOL	FALSE	FALSE	FALSE
IL16	hgnc:5980	IL16	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
RRM1	hgnc:10451	RRM1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
PPP1R13L	hgnc:18838	PPP1R13L	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
XPA	hgnc:12814	XPA	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.061992528	IUPHAR.LIGAND:372	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
CCN4	hgnc:12769	CCN4	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
YAP1	hgnc:16262	YAP1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
WNT5B	hgnc:16265	WNT5B	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
WIF1	hgnc:18081	WIF1	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
ATP7A	hgnc:869	ATP7A	PharmGKB	4/5/24	NULL	NULL	Platinum compounds	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	PharmGKB	4/5/24	NULL	0.179119736	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	NULL	lamivudine / abacavir	NULL	NULL	NULL	NULL	NULL
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	NULL	dolutegravir / abacavir / lamivudine	NULL	NULL	NULL	NULL	NULL
MAPK7	hgnc:6880	MAPK7	PharmGKB	4/5/24	NULL	0.4605936073306534	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.6819178082557726	IUPHAR.LIGAND:434	iuphar.ligand:434	AB-NECA	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1312691780892362	binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	PharmGKB	4/5/24	NULL	0.063331621	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.3070624048871023	isoniazid	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
AREG	hgnc:651	AREG	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.028290771	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.8204323630577265	efavirenz / emtricitabine / tenofovir disoproxil	wikidata:Q2869808	EMTRICITABINE/TENOFOVIR/EFAVIRENZ	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.1369170045259309	captopril	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1136529680426287	IUPHAR.LIGAND:5596	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	NULL	Dihydropyridine derivatives	NULL	NULL	NULL	NULL	NULL
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1363835616511545	IUPHAR.LIGAND:5595	ncit:C174671	BINODENOSON	FALSE	FALSE	FALSE
DDX58	hgnc:19102	RIGI	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
TANC1	hgnc:29364	TANC1	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
TMEM167A	hgnc:28330	TMEM167A	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
APEX1	hgnc:587	APEX1	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
CDH2	hgnc:1759	CDH2	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
CXCL8	hgnc:6025	CXCL8	PharmGKB	4/5/24	NULL	NULL	radiotherapy	NULL	NULL	NULL	NULL	NULL
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.017679351	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NSUN3	hgnc:26208	NSUN3	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
SELE	hgnc:10718	SELE	PharmGKB	4/5/24	NULL	0.1767935058440892	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.036087747	IUPHAR.LIGAND:2844	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
LMNTD1	hgnc:26683	LMNTD1	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	1.458546423213736	methazolamide	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	Vitamin B-complex with vitamin C	NULL	NULL	NULL	NULL	NULL
CSMD1	hgnc:14026	CSMD1	PharmGKB	4/5/24	NULL	1.615620653405984	anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
CSMD1	hgnc:14026	CSMD1	PharmGKB	4/5/24	NULL	0.4565884455277782	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1193356164447602	hydralazine	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	PharmGKB	4/5/24	NULL	0.1666910197958555	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
PTPRD	hgnc:9668	PTPRD	PharmGKB	4/5/24	NULL	0.2917092846427472	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
SCNN1B	hgnc:10600	SCNN1B	PharmGKB	4/5/24	NULL	0.4526523382387457	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:5610	iuphar.ligand:5610	MSX-2	FALSE	FALSE	FALSE
EIF2AK4	hgnc:19687	EIF2AK4	PharmGKB	4/5/24	NULL	0.5645986154375753	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	NULL	xenobiotics	NULL	NULL	NULL	NULL	NULL
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
ZNF568	hgnc:25392	ZNF568	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
CNIH3	hgnc:26802	CNIH3	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
BDNF-AS	hgnc:20608	BDNF-AS	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
ADGRV1	hgnc:17416	ADGRV1	PharmGKB	4/5/24	NULL	NULL	opioids	NULL	NULL	NULL	NULL	NULL
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.305277158	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
TTR	hgnc:12405	TTR	PharmGKB	4/5/24	NULL	4.375639269641208	vutrisiran	rxcui:2604578	VUTRISIRAN	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	PharmGKB	4/5/24	NULL	0.1037701012563132	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	NULL	Drugs used in nicotine dependence	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.052181537	pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PROS1	hgnc:9456	PROS1	PharmGKB	4/5/24	NULL	2.500365296937833	lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
TRIB3	hgnc:16228	TRIB3	PharmGKB	4/5/24	NULL	5.834185692854944	perindopril	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
PRRC2A	hgnc:13918	PRRC2A	PharmGKB	4/5/24	NULL	0.3763990769583835	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
FCGR2A	hgnc:3616	FCGR2A	PharmGKB	4/5/24	NULL	0.1166837138570988	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CRTC2	hgnc:27301	CRTC2	PharmGKB	4/5/24	NULL	NULL	hdl cholesterol	NULL	NULL	NULL	NULL	NULL
ZSCAN25	hgnc:21961	ZSCAN25	PharmGKB	4/5/24	NULL	10.50153425	lopinavir	rxcui:195088	LOPINAVIR	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	2.333674277141977	faldaprevir	ncit:C171746	FALDAPREVIR	FALSE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	1.400204566285186	faldaprevir	ncit:C171746	FALDAPREVIR	FALSE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	PharmGKB	4/5/24	NULL	0.8334550989792778	chlorthalidone	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
SLC22A3	hgnc:10967	SLC22A3	PharmGKB	4/5/24	NULL	NULL	catecholamines	NULL	NULL	NULL	NULL	NULL
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.3088686543276147	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	PharmGKB	4/5/24	NULL	1.250182648468916	remifentanil	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
PADI4	hgnc:18368	PADI4	PharmGKB	4/5/24	NULL	8.751278539282415	uric acid	rxcui:1427088	URIC ACID	FALSE	FALSE	FALSE
SLC9A9	hgnc:20653	SLC9A9	PharmGKB	4/5/24	NULL	8.751278539282415	remifentanil	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.3818739726232327	telmisartan	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	1.575230137070835	pamaquine	ncit:C73003	PAMAQUINE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.525076712	metabutethamine	ncit:C81413	METABUTETHAMINE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	NULL	Dihydropyridine derivatives	NULL	NULL	NULL	NULL	NULL
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	NULL	Dihydropyridine derivatives	NULL	NULL	NULL	NULL	NULL
RYR3	hgnc:10485	RYR3	PharmGKB	4/5/24	NULL	NULL	Dihydropyridine derivatives	NULL	NULL	NULL	NULL	NULL
IL1A	hgnc:5991	IL1A	PharmGKB	4/5/24	NULL	0.138178082	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
ATP1A2	hgnc:800	ATP1A2	PharmGKB	4/5/24	NULL	0.1973972602845657	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.5413161983061289	IUPHAR.LIGAND:458	iuphar.ligand:458	I-ABA	FALSE	FALSE	FALSE
CHAT	hgnc:1912	CHAT	PharmGKB	4/5/24	NULL	0.1535312024435511	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NPIPB8	hgnc:37490	NPIPB8	PharmGKB	4/5/24	NULL	NULL	desmethylnaproxen	NULL	NULL	NULL	NULL	NULL
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.070010228	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.1131630845596864	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.028850369	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.2853677784548614	galantamine	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
SLCO6A1	hgnc:23613	SLCO6A1	PharmGKB	4/5/24	NULL	0.3500511415712966	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
COL1A2	hgnc:2198	COL1A2	PharmGKB	4/5/24	NULL	0.077789143	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.049210563	IUPHAR.LIGAND:5615	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
MSH2	hgnc:7325	MSH2	PharmGKB	4/5/24	NULL	0.038894571	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.006731753	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.017502557	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
IMPDH1	hgnc:6052	IMPDH1	PharmGKB	4/5/24	NULL	0.3182283105193606	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1944728564284981	esomeprazole	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	PharmGKB	4/5/24	NULL	2.917092846427472	anifrolumab	rxcui:2565265	ANIFROLUMAB	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	NULL	Drugs used in nicotine dependence	NULL	NULL	NULL	NULL	NULL
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.1470803115845784	naloxone	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	2.12152207	artemisinin	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
CPS1	hgnc:2323	CPS1	PharmGKB	4/5/24	NULL	3.000438356	l-methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	0.7501095890813501	pantoprazole	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.050488145	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.172722603	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.2616661357260523	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:405	drugbank:DB08770	4-{2-[(7-AMINO-2-FURAN-2-YL[1,2,4]TRIAZOLO[1,5-A][1,3,5]TRIAZIN-5-YL)AMINO]ETHYL}PHENOL	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	TALC	12-May-16	NULL	5.250767123569449	CVX-060	chembl:CHEMBL4594470	CVX-060	FALSE	FALSE	TRUE
HDAC11	hgnc:19086	HDAC11	TALC	12-May-16	inhibitor	0.3182283105193606	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:12070	iuphar.ligand:12070	VIC 1911	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.1875273972703375	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.1981421556063943	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	NULL	SN-314	NULL	NULL	NULL	NULL	NULL
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.1712206670729168	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.2580229544751573	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.3659071166250487	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.064413418	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	NULL	JNJ38877605	NULL	NULL	NULL	NULL	NULL
AURKC	hgnc:11391	AURKC	TALC	12-May-16	inhibitor	NULL	SN-314	NULL	NULL	NULL	NULL	NULL
MFGE8	hgnc:7036	MFGE8	TALC	12-May-16	vaccine	NULL	MONOCLONAL ANTIBODY11D10 ANTI-IDIOTYPE VACCINE	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:9397	iuphar.ligand:9397	SNS-314	FALSE	FALSE	FALSE
MMP12	hgnc:7158	MMP12	TALC	12-May-16	inhibitor	1.166837138570989	NEOVASTAT	drugbank:DB05387	NEOVASTAT	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.5000730593875666	ARQ197	hemonc:499	TIVANTINIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.1458546423213736	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	TALC	12-May-16	inhibitor	0.1438566335224506	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	TALC	12-May-16	agonist	0.42006137	EFATUTAZONE	ncit:C83819	EFATUTAZONE	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	TALC	12-May-16	inhibitor	0.2401265452851882	OBATOCLAX	ncit:C60770	OBATOCLAX	FALSE	FALSE	TRUE
RPTOR	hgnc:30287	RPTOR	TALC	12-May-16	inhibitor	0.2524407270946851	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	TALC	12-May-16	inhibitor	0.4268916360625568	AT-101	ncit:C187300	ANTI-CD19 CAR T CELLS AT101	FALSE	FALSE	TRUE
RXRG	hgnc:10479	RXRG	TALC	12-May-16	NULL	1.988926940746004	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
RXRB	hgnc:10478	RXRB	TALC	12-May-16	NULL	1.944728564284981	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:12375	iuphar.ligand:12375	ADRIXETINIB	FALSE	FALSE	FALSE
TNFRSF10A	hgnc:11904	TNFRSF10A	TALC	12-May-16	agonist	15.75230137070834	DULANERMIN	ncit:C1685	DULANERMIN	FALSE	TRUE	TRUE
TUSC2	hgnc:17034	TUSC2	TALC	12-May-16	NULL	NULL	DOTAP:CHOL-FUS1	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	TALC	12-May-16	inhibitor	NULL	ARQ736	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	NULL	MM111	NULL	NULL	NULL	NULL	NULL
CTLA4	hgnc:2505	CTLA4	TALC	12-May-16	antibody	0.7001022831425934	IPILIMUMAB	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
CLU	hgnc:2095	CLU	TALC	12-May-16	antisense oligonucleotide	17.50255707856483	CUSTIRSEN	ncit:C169869	CUSTIRSEN	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	TALC	12-May-16	inhibitor	0.012398506	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P08174	hgnc:2665	CD55	TdgClinicalTrial	Jan-14	NULL	NULL	ONYVAX-105 (105AD7)	NULL	NULL	NULL	NULL	NULL
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:6170	iuphar.ligand:6170	MK-5046	FALSE	FALSE	FALSE
UNIPROT:P11532	hgnc:2928	DMD	TdgClinicalTrial	Jan-14	NULL	NULL	DYSTROPHIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	NULL	NOT DISCLOSED	NULL	NULL	NULL	NULL	NULL
UNIPROT:O95264	hgnc:5298	HTR3B	TdgClinicalTrial	Jan-14	NULL	NULL	NOT DISCLOSED	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.023716202	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:Q8WXI7	hgnc:15582	MUC16	TdgClinicalTrial	Jan-14	NULL	11.25164383622025	ABAGOVOMAB	ncit:C26449	ABAGOVOMAB	FALSE	FALSE	FALSE
UNIPROT:P29474	hgnc:7876	NOS3	TdgClinicalTrial	Jan-14	NULL	NULL	ORGANIC NITRATE + L-ARGININE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	NULL	ACCCRETROPIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.084383562	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	1.166837138570988	ADL5859	drugbank:DB05050	ADL5859	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.4817217544559128	ADL5945	chembl:CHEMBL3039511	BEVENOPRAN	FALSE	FALSE	FALSE
UNIPROT:Q02643	hgnc:4266	GHRHR	TdgClinicalTrial	Jan-14	NULL	NULL	AKL-0707	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q99705	hgnc:4479	MCHR1	TdgClinicalTrial	Jan-14	NULL	NULL	ALB-127158(A)	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9GZT9	hgnc:1232	EGLN1	TdgClinicalTrial	Jan-14	NULL	1.909369863116163	AKB-6548	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:612	iuphar.ligand:612	GASTRIN-RELEASING PEPTIDE	FALSE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	0.3061671792168775	AZD-6765	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.217423069	AZD-6765	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
UNIPROT:P62993	hgnc:4566	GRB2	TdgClinicalTrial	Jan-14	NULL	NULL	LIPOSOMAL GRB-2	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20839	hgnc:6052	IMPDH1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
UNIPROT:P20701	hgnc:6148	ITGAL	TdgClinicalTrial	Jan-14	NULL	NULL	CYTOLIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q03181	hgnc:9235	PPARD	TdgClinicalTrial	Jan-14	NULL	NULL	DB-959	NULL	NULL	NULL	NULL	NULL
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	NULL	DB-959	NULL	NULL	NULL	NULL	NULL
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6180	iuphar.ligand:6180	[D-PHE6]BOMBESIN(6-13)METHYL ESTER	FALSE	FALSE	FALSE
UNIPROT:P10253	hgnc:4065	GAA	TdgClinicalTrial	Jan-14	NULL	0.5469549087051511	DEOXYNOJIRIMYCIN	ncit:C87373	DUVOGLUSTAT	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1640864726115453	DERSALAZINE	ncit:C77949	DERSALAZINE	FALSE	FALSE	FALSE
UNIPROT:P41231	hgnc:8541	P2RY2	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	DENUFOSOL	ncit:C78118	DENUFOSOL	FALSE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	NULL	DG071	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	NULL	DG071	NULL	NULL	NULL	NULL	NULL
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	DEXANABINOL	ncit:C99381	DEXANABINOL	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.3017682254924971	DEXANABINOL	ncit:C99381	DEXANABINOL	FALSE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.1121958787087489	DEXANABINOL	ncit:C99381	DEXANABINOL	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	NULL	BETANECHOL	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TdgClinicalTrial	Jan-14	NULL	NULL	DV1179	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	NULL	DV1179	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.035145697	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.084383562	FLUTICASONE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	E-10030	chembl:CHEMBL3301576	PEGPLERANIB SODIUM	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.1093909817410302	E-10030	chembl:CHEMBL3301576	PEGPLERANIB SODIUM	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.039390601	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P07333	hgnc:2433	CSF1R	TdgClinicalTrial	Jan-14	NULL	0.061592576	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	EPTIFIBATIDE	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
UNIPROT:P12931	hgnc:11283	SRC	TdgClinicalTrial	Jan-14	NULL	0.03136659	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	EPINASTINE	rxcui:39684	EPINASTINE	TRUE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	NULL	ESBA105	NULL	NULL	NULL	NULL	NULL
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.5791287268642775	GALANTAMINE	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
UNIPROT:P10242	hgnc:7545	MYB	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	G4460	drugbank:DB06359	G4460	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:7854	iuphar.ligand:7854	COMPOUND J [PMID: 21907142]	FALSE	FALSE	FALSE
UNIPROT:P14672	hgnc:11009	SLC2A4	TdgClinicalTrial	Jan-14	NULL	0.100976291	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:Q9NY91	hgnc:11039	SLC5A4	TdgClinicalTrial	Jan-14	NULL	0.596678082	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	NULL	HERZYME	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23921	hgnc:10451	RRM1	TdgClinicalTrial	Jan-14	NULL	3.088686543276147	GTI-2501	drugbank:DB05406	GTI-2501	FALSE	FALSE	FALSE
UNIPROT:Q92542	hgnc:17091	NCSTN	TdgClinicalTrial	Jan-14	NULL	0.6819178082557726	GSI-136	drugbank:DB12819	GSI-136	FALSE	FALSE	FALSE
UNIPROT:P04141	hgnc:2434	CSF2	TdgClinicalTrial	Jan-14	NULL	0.043756393	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
UNIPROT:Q9NZ42	hgnc:30100	PSENEN	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	GSI-136	drugbank:DB12819	GSI-136	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:12747	ncit:C166726	UMIBECESTAT	FALSE	FALSE	FALSE
UNIPROT:P28907	hgnc:1667	CD38	TdgClinicalTrial	Jan-14	NULL	0.3889457128569963	HUMAX-CD38	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	2.316514907	HUPERZINE-A	rxcui:2267703	HUPERZINE A	FALSE	FALSE	FALSE
UNIPROT:O14763	hgnc:11905	TNFRSF10B	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	HGS-TR2J	drugbank:DB05895	HGS-TR2J	FALSE	FALSE	FALSE
UNIPROT:P51787	hgnc:6294	KCNQ1	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	ICA-105665	drugbank:DB06089	ICA-105665	FALSE	FALSE	FALSE
UNIPROT:O43526	hgnc:6296	KCNQ2	TdgClinicalTrial	Jan-14	NULL	1.050153425	ICA-105665	drugbank:DB06089	ICA-105665	FALSE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	NULL	ANTI-CD20 (HA20) MONOCLONAL ANTIBODY	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NYK1	hgnc:15631	TLR7	TdgClinicalTrial	Jan-14	NULL	NULL	IMO-3100	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	NULL	IMO-3100	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13007	hgnc:11346	IL24	TdgClinicalTrial	Jan-14	NULL	NULL	INGN 242	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q99062	hgnc:2439	CSF3R	TdgClinicalTrial	Jan-14	NULL	NULL	INS-19	NULL	NULL	NULL	NULL	NULL
UNIPROT:P09874	hgnc:270	PARP1	TdgClinicalTrial	Jan-14	NULL	4.200613699	INIPARIB	ncit:C62526	INIPARIB	FALSE	FALSE	TRUE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:533	iuphar.ligand:533	T-0509	FALSE	FALSE	FALSE
UNIPROT:P47871	hgnc:4192	GCGR	TdgClinicalTrial	Jan-14	NULL	NULL	ISIS 325568	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	INTERFERON BETA	chembl:CHEMBL2108510	INTERFERON BETA	TRUE	FALSE	FALSE
UNIPROT:P00749	hgnc:9052	PLAU	TdgClinicalTrial	Jan-14	NULL	NULL	MRX-801	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
UNIPROT:O00519	hgnc:3553	FAAH	TdgClinicalTrial	Jan-14	NULL	NULL	IW-6118	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08648	hgnc:6141	ITGA5	TdgClinicalTrial	Jan-14	NULL	NULL	JSM 6427	NULL	NULL	NULL	NULL	NULL
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	NULL	JSM 6427	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	NULL	KB3305	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11775	iuphar.ligand:11775	COMPOUND 6 [PMID: 34553947]	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	NULL	PLATELET-DERIVED GROWTH FACTOR (PDGF)	NULL	NULL	NULL	NULL	NULL
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	NULL	PLATELET-DERIVED GROWTH FACTOR (PDGF)	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q02156	hgnc:9401	PRKCE	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	KAI-1455	drugbank:DB06064	KAI-1455	FALSE	FALSE	FALSE
UNIPROT:Q7L0J3	hgnc:20566	SV2A	TdgClinicalTrial	Jan-14	NULL	4.500657534	LEVETIRACETAM	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	NULL	LINAGLIPTON	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31350	hgnc:10452	RRM2	TdgClinicalTrial	Jan-14	NULL	NULL	LOR-2040	NULL	NULL	NULL	NULL	NULL
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.1875273972703375	IUPHAR.LIGAND:7445	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
UNIPROT:Q7LG56	hgnc:17296	RRM2B	TdgClinicalTrial	Jan-14	NULL	NULL	LOR-2040	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14765	hgnc:11365	STAT4	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	LISOFYLLINE	ncit:C1516	LISOFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P25092	hgnc:4688	GUCY2C	TdgClinicalTrial	Jan-14	NULL	19.69037671338543	LINACLOTIDE	rxcui:1307404	LINACLOTIDE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.061725319	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:3464	rxcui:34530	PROCATEROL	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.029465584	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.026227608	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.029106248	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:CARDIAC MYSOIN	NULL	NULL	TdgClinicalTrial	Jan-14	NULL	NULL	OMECAMTIV MECARBIL	ncit:C166579	OMECAMTIV MECARBIL	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P22894	hgnc:7175	MMP8	TdgClinicalTrial	Jan-14	NULL	NULL	DOXYCYKLIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	OSI-461	drugbank:DB05415	OSI-461	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:543	iuphar.ligand:543	ICI 118551	FALSE	FALSE	FALSE
UNIPROT:P78348	hgnc:100	ASIC1	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9UHC3	hgnc:101	ASIC3	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:554	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
UNIPROT:Q96FT7	hgnc:21263	ASIC4	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q16515	hgnc:99	ASIC2	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
UNIPROT:P37088	hgnc:10599	SCNN1A	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
UNIPROT:P51168	hgnc:10600	SCNN1B	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
UNIPROT:P51172	hgnc:10601	SCNN1D	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
UNIPROT:P51170	hgnc:10602	SCNN1G	TdgClinicalTrial	Jan-14	NULL	NULL	P-552	NULL	NULL	NULL	NULL	NULL
UNIPROT:P07288	hgnc:6364	KLK3	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	PRX302	chembl:CHEMBL2364656	TOPSALYSIN	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	NULL	NOT DISCLOSED	NULL	NULL	NULL	NULL	NULL
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	NULL	NOT DISCLOSED	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	NULL	NOT DISCLOSED	NULL	NULL	NULL	NULL	NULL
UNIPROT:P56159	hgnc:4243	GFRA1	TdgClinicalTrial	Jan-14	NULL	NULL	PYM50028	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08138	hgnc:7809	NGFR	TdgClinicalTrial	Jan-14	NULL	NULL	PYM50028	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04629	hgnc:8031	NTRK1	TdgClinicalTrial	Jan-14	NULL	NULL	PYM50028	NULL	NULL	NULL	NULL	NULL
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:532	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
UNIPROT:Q16620	hgnc:8032	NTRK2	TdgClinicalTrial	Jan-14	NULL	NULL	PYM50028	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43405	hgnc:11491	SYK	TdgClinicalTrial	Jan-14	NULL	NULL	R343	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9Y6A2	hgnc:2641	CYP46A1	TdgClinicalTrial	Jan-14	NULL	NULL	RC-8800	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.081407242	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.076098074	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.1060761035064535	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P05155	hgnc:1228	SERPING1	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT HUMAN C1 ESTERASE INHIBITOR	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:8148	iuphar.ligand:8148	COMPOUND 31 [PMID: 24915291]	FALSE	FALSE	FALSE
UNIPROT:Q02153	hgnc:4687	GUCY1B1	TdgClinicalTrial	Jan-14	NULL	1.235474617310459	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	0.8751278539282416	ROLOFYLLINE	ncit:C96195	ROLOFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P33402	hgnc:4684	GUCY1A2	TdgClinicalTrial	Jan-14	NULL	1.166837138570989	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TdgClinicalTrial	Jan-14	NULL	NULL	SA4503	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	0.7740688634254718	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
UNIPROT:Q86V86	hgnc:19310	PIM3	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TdgClinicalTrial	Jan-14	NULL	NULL	GAMMA HYDROXYBUTYRIC ACID	NULL	NULL	NULL	NULL	NULL
UNIPROT:O75899	hgnc:4507	GABBR2	TdgClinicalTrial	Jan-14	NULL	NULL	GAMMA HYDROXYBUTYRIC ACID	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9HAB3	hgnc:30224	SLC52A2	TdgClinicalTrial	Jan-14	NULL	NULL	GAMMA HYDROXYBUTYRIC ACID	NULL	NULL	NULL	NULL	NULL
UNIPROT:O15392	hgnc:593	BIRC5	TdgClinicalTrial	Jan-14	NULL	NULL	SPC-3042	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04114	hgnc:603	APOB	TdgClinicalTrial	Jan-14	NULL	NULL	SPC4955	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00797	hgnc:9958	REN	TdgClinicalTrial	Jan-14	NULL	NULL	SPP635	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	NULL	TC-2696	NULL	NULL	NULL	NULL	NULL
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	NULL	TC-2696	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08183	hgnc:40	ABCB1	TdgClinicalTrial	Jan-14	NULL	0.5609793935437446	TARIQUIDAR	ncit:C2246	TARIQUIDAR	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	NULL	TGAAC94	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.045778266	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.033002936	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	NULL	TNF-ALPHA ADENOVECTOR	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q92847	hgnc:4267	GHSR	TdgClinicalTrial	Jan-14	NULL	8.751278539282417	TZP-101	ncit:C102755	ULIMORELIN HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	TROSPIUM	rxcui:236778	TROSPIUM	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	NULL	VA106483	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q13163	hgnc:6845	MAP2K5	TdgClinicalTrial	Jan-14	NULL	0.9376369863516874	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
UNIPROT:P02724	hgnc:4702	GYPA	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	WX-G250	ncit:C1960	GIRENTUXIMAB	FALSE	FALSE	FALSE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	0.272767123	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.1136529680426288	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
UNIPROT:P50579	hgnc:16672	METAP2	TdgClinicalTrial	Jan-14	NULL	9.845188356692718	BELORANIB	ncit:C90656	BELORANIB	FALSE	FALSE	FALSE
UNIPROT:P13945	hgnc:288	ADRB3	TdgClinicalTrial	Jan-14	NULL	0.9001315068976199	YM-178	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
UNIPROT:P14174	hgnc:7097	MIF	TdgClinicalTrial	Jan-14	NULL	NULL	ANTI-MIF MONOCLONAL ANTIBODY	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	NULL	CHF 6001	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	NULL	CHF 6001	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	NULL	DEUTERATED DEXTROMETHORPHAN	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TdgClinicalTrial	Jan-14	NULL	NULL	DEUTERATED DEXTROMETHORPHAN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P19793	hgnc:10477	RXRA	TdgClinicalTrial	Jan-14	NULL	0.1166837138570988	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.2344092465879218	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.2890330526735477	ALVIMOPAN	rxcui:1516803	ALVIMOPAN ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P48443	hgnc:10479	RXRG	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.05814803	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.060984519	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.064111931	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	BROMPHENIRAMINE	rxcui:1767	BROMPHENIRAMINE	TRUE	FALSE	FALSE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.1534190540122556	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.033243223	DRONEDARONE	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.8468979231563628	DIMENHYDRINATE	rxcui:3444	DIMENHYDRINATE	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TdgClinicalTrial	Jan-14	NULL	0.7001022831425934	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.067839369	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1035654265003836	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.1555782851427985	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	PENBUTOLOL	rxcui:7973	PENBUTOLOL	TRUE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:9285	iuphar.ligand:9285	PRN694	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.03140411	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	PHENIRAMINE	rxcui:8132	PHENIRAMINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.060077427	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.079557078	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1835932560688619	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.091796628	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.088396753	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.083257407	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.072125922	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.078682824	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q02643	hgnc:4266	GHRHR	TdgClinicalTrial	Jan-14	NULL	19.69037671338543	SERMORELIN	rxcui:56188	SERMORELIN	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.079557078	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	1.193356164447602	ACEBUTOLOL	rxcui:149	ACEBUTOLOL	TRUE	FALSE	FALSE
UNIPROT:P48443	hgnc:10479	RXRG	TEND	1-Aug-11	NULL	0.9092237443410301	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
UNIPROT:Q13698	hgnc:1397	CACNA1S	TEND	1-Aug-11	NULL	0.066047385	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P10276	hgnc:9864	RARA	TEND	1-Aug-11	NULL	0.2381300282797936	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	AZATADINE	rxcui:18600	AZATADINE	TRUE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TEND	1-Aug-11	NULL	4.773424657790408	CINALUKAST	ncit:C96709	CINALUKAST	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.4070362111294147	BENZPHETAMINE	rxcui:1422	BENZPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.693795846312725	BEPOTASTINE	rxcui:658552	BEPOTASTINE BESILATE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1282238613814273	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.060984519	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TEND	1-Aug-11	NULL	0.1275696580070323	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:7880	iuphar.ligand:7880	AGERAFENIB	FALSE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TEND	1-Aug-11	NULL	0.179119736	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P09038	hgnc:3676	FGF2	TEND	1-Aug-11	NULL	1.135300999690692	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TEND	1-Aug-11	NULL	10.50153424713889	CHORIOGONADOTROPIN ALFA	rxcui:283550	CHORIOGONADOTROPIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1643432589536604	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.092606122	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.091476779	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1282238613814273	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.094950581	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.8140724222588294	CLENBUTEROL	rxcui:2580	CLENBUTEROL	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1376949420516464	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7510	iuphar.ligand:7510	BIC1	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.091583148	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.4565884455277783	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.04724037	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TEND	1-Aug-11	NULL	0.3017682254924971	INTERFERON ALFA-2A, RECOMBINANT	rxcui:120608	PEGINTERFERON ALFA-2A	TRUE	TRUE	TRUE
UNIPROT:P50406	hgnc:5301	HTR6	TEND	1-Aug-11	NULL	0.33338204	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.040682597	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.9814517987980279	GUANETHIDINE	rxcui:5036	GUANETHIDINE	TRUE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TEND	1-Aug-11	NULL	3.938075342677087	HEXAFLURONIUM BROMIDE	rxcui:26826	HEXAFLUORENIUM	FALSE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	1.250182648468916	GLIPIZIDE	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
UNIPROT:P16083	hgnc:7856	NQO2	TEND	1-Aug-11	NULL	0.1065064325267636	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TEND	1-Aug-11	NULL	0.2419708351875322	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1615620653405984	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:3093	hgnc:4914	UBE2K	GuideToPharmacology	2024.1	activator	1.346350544504987	IUPHAR.LIGAND:1204	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
UNIPROT:P08709	hgnc:3544	F7	TEND	1-Aug-11	NULL	0.021554873	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:O60733	hgnc:9039	PLA2G6	TEND	1-Aug-11	NULL	2.019525816757481	NIFLUMIC ACID	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
UNIPROT:P04070	hgnc:9451	PROC	TEND	1-Aug-11	NULL	0.1810609352954982	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.074690855	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.056097939	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.2051080907644316	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.091583148	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.1325951293830669	MOMETASONE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
UNIPROT:P43088	hgnc:9600	PTGFR	TEND	1-Aug-11	NULL	2.812910959055062	BIMATOPROST	rxcui:283810	BIMATOPROST	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	0.4861821410712454	NATEGLINIDE	rxcui:274332	NATEGLINIDE	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TEND	1-Aug-11	NULL	0.1555782851427985	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	1.666910197958555	PANCURONIUM	rxcui:7883	PANCURONIUM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.2734774543525755	PHENDIMETRAZINE	rxcui:33272	PHENDIMETRAZINE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	1.458546423213736	PHENMETRAZINE	rxcui:8133	PHENMETRAZINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.031929262	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TEND	1-Aug-11	NULL	1.750255707856483	PITAVASTATIN	rxcui:861634	PITAVASTATIN	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.100976291	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
UNIPROT:P30988	hgnc:1440	CALCR	TEND	1-Aug-11	NULL	1.875273972703374	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
UNIPROT:P04035	hgnc:5006	HMGCR	TEND	1-Aug-11	NULL	0.4321619031744403	PRAVASTATIN	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.8899605294185507	QUINAPRIL	rxcui:35208	QUINAPRIL	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.5933070196123671	RAMIPRIL	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
NCBIGENE:3055	hgnc:4840	HCK	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:10434	iuphar.ligand:10434	COMPOUND 5B  [PMID: 31287314]	FALSE	FALSE	FALSE
UNIPROT:P02671	hgnc:3661	FGA	TEND	1-Aug-11	NULL	4.773424657790408	RETEPLASE	rxcui:76895	RETEPLASE	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TEND	1-Aug-11	NULL	2.500365296937833	RETEPLASE	rxcui:76895	RETEPLASE	TRUE	FALSE	FALSE
UNIPROT:P30531	hgnc:11042	SLC6A1	TEND	1-Aug-11	NULL	0.8078103267029924	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.172950169	ROPINIROLE	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TEND	1-Aug-11	NULL	0.09055649	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TEND	1-Aug-11	NULL	0.1403266238077355	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TEND	1-Aug-11	NULL	0.063331621	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P21802	hgnc:3689	FGFR2	TEND	1-Aug-11	NULL	0.033002936	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:P01375	hgnc:11892	TNF	TEND	1-Aug-11	NULL	0.045778266	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.1164249916534246	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P00918	hgnc:1373	CA2	TEND	1-Aug-11	NULL	0.1376949420516464	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.4070362111294147	TIZANIDINE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P22748	hgnc:1375	CA4	TEND	1-Aug-11	NULL	0.3977853881492008	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.1049104320393496	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TEND	1-Aug-11	NULL	0.546954909	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.6908904109959803	ZALEPLON	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
UNIPROT:O14786	hgnc:8004	NRP1	TEND	1-Aug-11	NULL	17.50255707856483	PEGAPTANIB	rxcui:498509	PEGAPTANIB	TRUE	FALSE	FALSE
UNIPROT:Q8N0U8	hgnc:21492	VKORC1L1	TEND	1-Aug-11	NULL	1.810609352954982	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TEND	1-Aug-11	NULL	4.200613698855561	ACENOCOUMAROL	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1221108633388244	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.2763561643983921	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.6177373086552295	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.022889133	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.048859496	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
C-X-C MOTIF CHEMOKINE 10	hgnc:10637	CXCL10	TTD	2020.06.01	NULL	6.177373086552294	NI-0801	chembl:CHEMBL2109379	NI-0801	FALSE	FALSE	FALSE
INTERLEUKIN-11	hgnc:5966	IL11	TTD	2020.06.01	NULL	NULL	VM-501	NULL	NULL	NULL	NULL	NULL
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	NULL	DSP-0565	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	XP-23829	iuphar.ligand:9770	TEPILAMIDE FUMARATE	FALSE	FALSE	FALSE
VIRAL MATURATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Drug 2838232	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	ANAVEX 1-41	NULL	NULL	NULL	NULL	NULL
PLK1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TKM-PLK1	ncit:C116889	LIPID ENCAPSULATED ANTI-PLK1 SIRNA TKM-PLK1	FALSE	FALSE	FALSE
HAEMOPHILUS INFLUENZAE OUTER MEMBRANE PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	NTHI vaccine	NULL	NULL	NULL	NULL	NULL
HEPATITIS B VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clevudine	ncit:C95210	CLEVUDINE	FALSE	FALSE	FALSE
NCBIGENE:528	hgnc:856	ATP6V1C1	GuideToPharmacology	2024.1	activator	2.625383561784724	IUPHAR.LIGAND:4065	iuphar.ligand:4065	(-)-(S)-BAYK8644	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SUN-101	drugbank:DB17238	SUN-101	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	CLR-3001	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	CLR-3001	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	COL-1077	NULL	NULL	NULL	NULL	NULL
HEPARIN-BINDING GROWTH FACTOR 1	hgnc:3665	FGF1	TTD	2020.06.01	NULL	NULL	CVBT-141H	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	SSR-128428	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	SSR-128428	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	FP-1097	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M2	hgnc:1951	CHRM2	TTD	2020.06.01	NULL	NULL	FP-1097	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	TT-100	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	NULL	TT-100	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 6 RECEPTOR	hgnc:6019	IL6R	TTD	2020.06.01	NULL	12.11715490054488	SAR153191	rxcui:1923319	SARILUMAB	TRUE	FALSE	FALSE
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1	hgnc:2357	CRHR1	TTD	2020.06.01	NULL	1.458546423213736	SSR125543	iuphar.ligand:3533	SSR125543A	FALSE	FALSE	FALSE
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	0.5707355569097228	LYC-55716	ncit:C131294	CINTIRORGON	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	1.193356164447602	ASTX727	ncit:C115102	DECITABINE AND CEDAZURIDINE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	0.7369497717290455	INCB54828	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.100976291	TGR-1202	rxcui:2478439	UMBRALISIB	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Darolutamide	rxcui:2180325	DAROLUTAMIDE	TRUE	FALSE	TRUE
GUANINE NUCLEOTIDE EXCHANGE FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Plinabulin	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
NCBIGENE:1621	hgnc:2689	DBH	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:8654	iuphar.ligand:8654	M826	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Rubraca rucaparib	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Talabostat	ncit:C48264	TALABOSTAT	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Talabostat	ncit:C48264	TALABOSTAT	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	AC0058TA	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD9567	iuphar.ligand:9812	AZD9567	FALSE	FALSE	FALSE
DNA TOPOISOMERASE	hgnc:38595	LINC00273	TTD	2020.06.01	NULL	8.751278539282415	Karenitecin	chembl:CHEMBL1743260	KARENITECIN	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	0.5164688974002737	DCC-2618	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	NULL	Gerilimzumab	NULL	NULL	NULL	NULL	NULL
CELL ADHESION MOLECULE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PRX003	iuphar.ligand:9805	IMAPRELIMAB	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.4070362111294147	IUPHAR.LIGAND:7718	iuphar.ligand:7718	Z944	FALSE	FALSE	FALSE
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	NULL	PTG-100	NULL	NULL	NULL	NULL	NULL
INTEGRIN BETA-7	hgnc:6162	ITGB7	TTD	2020.06.01	NULL	NULL	PTG-100	NULL	NULL	NULL	NULL	NULL
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	NULL	VTP-43742	NULL	NULL	NULL	NULL	NULL
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	3.621218705909965	Dapirolizumab pegol	ncit:C174737	DAPIROLIZUMAB PEGOL	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.2573905452730122	TAK-020	iuphar.ligand:11730	TAK-020	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	Topical ruxolitinib	NULL	NULL	NULL	NULL	NULL
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	AMG 211	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	1.166837138570988	Ponesimod	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	MVT-5873	chembl:CHEMBL4297791	MVT-5873	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	AU105	NULL	NULL	NULL	NULL	NULL
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	NULL	AD04	NULL	NULL	NULL	NULL	NULL
MITOCHONDRIAL ALDEHYDE DEHYDROGENASE	hgnc:404	ALDH2	TTD	2020.06.01	NULL	NULL	ANS-6637	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Apimostinel	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	OPNT001	NULL	NULL	NULL	NULL	NULL
SEROTONINNOREPINEPHRINEDOPAMINE REUPTAKE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dasotraline	ncit:C166750	DASOTRALINE	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Esketamine	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Lu AF35700	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PH94B NS	NULL	NULL	NULL	NULL	NULL
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	NULL	PU-AD	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BHV-5000	drugbank:DB17817	BHV-5000	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	CA-011	NULL	NULL	NULL	NULL	NULL
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA2	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAD-1833	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	NULL	CNTX-6970	NULL	NULL	NULL	NULL	NULL
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	DSP-6745	NULL	NULL	NULL	NULL	NULL
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	EPX-100	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	NULL	M4 agonist	NULL	NULL	NULL	NULL	NULL
SYNUCLEIN ALPHA	hgnc:11138	SNCA	TTD	2020.06.01	NULL	NULL	MEDI1341	NULL	NULL	NULL	NULL	NULL
BETA-SECRETASE 1	hgnc:933	BACE1	TTD	2020.06.01	NULL	NULL	Selective BACE 1 inhibitor	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C1S COMPONENT	hgnc:1247	C1S	TTD	2020.06.01	NULL	5.250767123569449	ANX005	chembl:CHEMBL4650442	ANX-005	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	0.5707355569097228	BNC375	iuphar.ligand:10693	BNC375	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	TRV250	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	NULL	VX-128	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	WST-057	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED T-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	CX-8998	ncit:C174710	SUVECALTAMIDE	FALSE	FALSE	FALSE
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Edasalonexent	ncit:C171665	EDASALONEXENT	FALSE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	EPX-300	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	1.166837138570988	SHAPE	ncit:C97513	REMETINOSTAT	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.4667348554283956	Revamilast	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	1.141471113819445	Tiprelestat	ncit:C152650	TIPRELESTAT	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS CAPSID P24	NULL	NULL	TTD	2020.06.01	NULL	NULL	F4co vaccine	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS MATRIX P17	NULL	NULL	TTD	2020.06.01	NULL	NULL	F4co vaccine	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS NEGATIVE FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	F4co vaccine	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	F4co vaccine	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	HO/03/03	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TMC-647055	drugbank:DB11822	TMC-647055	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-333	rxcui:1597381	DASABUVIR	TRUE	FALSE	FALSE
TRANSTHYRETIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Patisiran	rxcui:2053490	PATISIRAN	TRUE	FALSE	FALSE
TRANSTHYRETIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALN-TTR02	rxcui:2053490	PATISIRAN	TRUE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	Anti-N3pG-Abeta antibody	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG1577	chembl:CHEMBL3707394	SEMBRAGILINE	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	LC-150444	chembl:CHEMBL3707235	GEMIGLIPTIN	FALSE	FALSE	FALSE
INTERLEUKIN-9	hgnc:6029	IL9	TTD	2020.06.01	NULL	35.00511415712966	MEDI-528	iuphar.ligand:8934	ENOKIZUMAB	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.2983390411119005	BL-1021	chembl:CHEMBL1187120	BL-1021	FALSE	FALSE	FALSE
TGF BETA-2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Belagenpumatucel-L	ncit:C73438	BELAGENPUMATUCEL-L	FALSE	FALSE	TRUE
PROGRAMMED CELL DEATH PROTEIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	RHIgM12B7	chembl:CHEMBL2109309	RHIGM12B7	FALSE	FALSE	FALSE
ERBB4 TYROSINE KINASE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK3052230	ncit:C77970	FGF RECEPTOR ANTAGONIST HGS1036	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.1389091831632129	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
GLUTATHIONE S-TRANSFERASE P	hgnc:4638	GSTP1	TTD	2020.06.01	NULL	1.750255707856483	Ezatiostat	ncit:C83709	EZATIOSTAT	FALSE	FALSE	FALSE
INHIBITOR OF APOPTOSIS PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	LCL161	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	DNA vaccine, University of Southampton/Inovio	NULL	NULL	NULL	NULL	NULL
UBIQUITIN-ACTIVATING ENZYME	NULL	NULL	TTD	2020.06.01	NULL	NULL	MLN7243	ncit:C113788	UAE INHIBITOR TAK-243	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	NULL	PS-938285	NULL	NULL	NULL	NULL	NULL
MACROPHAGE MIGRATION INHIBITORY FACTOR	hgnc:7097	MIF	TTD	2020.06.01	NULL	NULL	COR100140	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	DS-1093	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	0.3596415838061266	DS-6051	chembl:CHEMBL4650989	TALETRECTINIB	FALSE	FALSE	FALSE
SUPPRESSOR OF TUMORIGENICITY 14 PROTEIN	hgnc:11344	ST14	TTD	2020.06.01	NULL	NULL	US8569313, Inhibitor 18	NULL	NULL	NULL	NULL	NULL
SUPPRESSOR OF TUMORIGENICITY 14 PROTEIN	hgnc:11344	ST14	TTD	2020.06.01	NULL	NULL	US8569313, Inhibitor 19	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US8586571, 36	NULL	NULL	NULL	NULL	NULL
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.086361301	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
ACETYL-COA TRANSPORTER	hgnc:95	SLC33A1	TTD	2020.06.01	NULL	NULL	US8592431, 181	NULL	NULL	NULL	NULL	NULL
ACETYL-COA TRANSPORTER	hgnc:95	SLC33A1	TTD	2020.06.01	NULL	NULL	US8592431, 457	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8592455, 90	NULL	NULL	NULL	NULL	NULL
KYNURENINE OXOGLUTARATE TRANSAMINASE II	hgnc:17929	AADAT	TTD	2020.06.01	NULL	NULL	US8933095, 14	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	US8614253, 32-5	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8669361, 103	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8669361, 107	NULL	NULL	NULL	NULL	NULL
GALECTIN-1	hgnc:6561	LGALS1	TTD	2020.06.01	NULL	NULL	US8703720, 15	NULL	NULL	NULL	NULL	NULL
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:10058	ncit:C166825	OLORINAB	FALSE	FALSE	FALSE
INTEGRIN-LINKED PROTEIN KINASE 1	hgnc:6040	ILK	TTD	2020.06.01	NULL	NULL	US8754233, (4-Benzothiazol-2-yl-1H-pyrazol-3-yl)-[2-(1H-imidazol-4-yl)-ethyl]-amine	NULL	NULL	NULL	NULL	NULL
INTEGRIN-LINKED PROTEIN KINASE 1	hgnc:6040	ILK	TTD	2020.06.01	NULL	NULL	US8754233, 2-(3-Amino-1H-pyrazol-4-yl)-5-fluoro-benzothiazole-6-sulfonic acid amide	NULL	NULL	NULL	NULL	NULL
INTEGRIN-LINKED PROTEIN KINASE 1	hgnc:6040	ILK	TTD	2020.06.01	NULL	NULL	US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl)-5-(2-fluoro-phenyl)-2H-pyrazol-3-ylamine	NULL	NULL	NULL	NULL	NULL
BACTERIAL NICOTINATE-NUCLEOTIDE ADENYLYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AC1LJNG0	NULL	NULL	NULL	NULL	NULL
NCBIGENE:391	hgnc:672	RHOG	GuideToPharmacology	2024.1	activator	0.3804903712731485	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
CASEIN KINASE II ALPHA PRIME	hgnc:2459	CSNK2A2	TTD	2020.06.01	NULL	NULL	US8791257, 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	US8846654, 11	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	US8846654, 251	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	US8846654, 294	NULL	NULL	NULL	NULL	NULL
PRKACA MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	XHPNYYOUZWOWNT-PYUWXLGESA-N	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	A1-10438	NULL	NULL	NULL	NULL	NULL
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9232	ncit:C84034	OTENABANT	FALSE	FALSE	FALSE
REGULATOR OF G-PROTEIN SIGNALING 8	hgnc:16810	RGS8	TTD	2020.06.01	NULL	NULL	1-Benzyl-3-bromo-1H-pyrrole-2,5-dione	NULL	NULL	NULL	NULL	NULL
REGULATOR OF G-PROTEIN SIGNALING 8	hgnc:16810	RGS8	TTD	2020.06.01	NULL	NULL	1-Benzyl-3-p-tolyl-1H-pyrrole-2,5-dione	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8921389, 123	NULL	NULL	NULL	NULL	NULL
KYNURENINE OXOGLUTARATE TRANSAMINASE II	hgnc:17929	AADAT	TTD	2020.06.01	NULL	NULL	US8933095, 16	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	Unii-I92MU0V408	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9409892, 136	NULL	NULL	NULL	NULL	NULL
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:742	iuphar.ligand:742	LY320135	FALSE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9409892, 19	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9422240, 1-282	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9422240, 1-286	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9422240, 1-298	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9434725, 285	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US9434727, 120	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US9434727, 153	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE D1	hgnc:9067	PLD1	TTD	2020.06.01	NULL	NULL	ML272	NULL	NULL	NULL	NULL	NULL
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:12754	iuphar.ligand:12754	AZD1940	FALSE	FALSE	FALSE
PHOSPHOLIPASE D1	hgnc:9067	PLD1	TTD	2020.06.01	NULL	NULL	US9453017, 1	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE D1	hgnc:9067	PLD1	TTD	2020.06.01	NULL	NULL	US9453017, 2	NULL	NULL	NULL	NULL	NULL
BETA-ADRENERGIC RECEPTOR KINASE 1	hgnc:289	GRK2	TTD	2020.06.01	NULL	NULL	US9493490, D	NULL	NULL	NULL	NULL	NULL
PROTEIN-TYROSINE PHOSPHATASE SHP-1	hgnc:9658	PTPN6	TTD	2020.06.01	NULL	NULL	BDBM50054344	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9522888, 575	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9522888, 695	NULL	NULL	NULL	NULL	NULL
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	BDBM50080408	NULL	NULL	NULL	NULL	NULL
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:11693	iuphar.ligand:11693	PF-514273	FALSE	FALSE	FALSE
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	US9567304, Compound F-54	NULL	NULL	NULL	NULL	NULL
EPITHELIAL DISCOIDIN DOMAIN RECEPTOR 1	hgnc:2730	DDR1	TTD	2020.06.01	NULL	NULL	US9567304, Compound N-9	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9580418, Example 11	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9586945, 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US9611221, Example 9	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	BDBM50080563	NULL	NULL	NULL	NULL	NULL
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	NULL	BDBM50444059	NULL	NULL	NULL	NULL	NULL
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	NULL	BDBM50444062	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE EIF2AK2	hgnc:20932	POLD3	TTD	2020.06.01	NULL	NULL	US9650366, 12	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE EIF2AK2	hgnc:20932	POLD3	TTD	2020.06.01	NULL	NULL	US9650366, 2	NULL	NULL	NULL	NULL	NULL
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3781	iuphar.ligand:3781	[125I]GASTRIN	FALSE	FALSE	FALSE
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9024044, 2	NULL	NULL	NULL	NULL	NULL
ENTEROPEPTIDASE	hgnc:9490	TMPRSS15	TTD	2020.06.01	NULL	NULL	US9024044, 4	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9656955, Example 540	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE C4 SYNTHASE	hgnc:6719	LTC4S	TTD	2020.06.01	NULL	NULL	US20160326143, 38	NULL	NULL	NULL	NULL	NULL
ACTIVIN RECEPTOR TYPE IB	hgnc:172	ACVR1B	TTD	2020.06.01	NULL	NULL	US9682983, 1	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US9434727, 40	NULL	NULL	NULL	NULL	NULL
SODIUM/HYDROGEN EXCHANGER 3	hgnc:11073	SLC9A3	TTD	2020.06.01	NULL	NULL	AZD1772//RDX5791	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	GPX-150D	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Rituxan Hemotalogy/oncology	NULL	NULL	NULL	NULL	NULL
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:866	iuphar.ligand:866	GLAXO-11P	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tegobuvir	ncit:C152541	TEGOBUVIR	FALSE	FALSE	FALSE
ZINC FINGER PROTEIN	hgnc:23717	ZNF501	TTD	2020.06.01	NULL	NULL	PCL-016	NULL	NULL	NULL	NULL	NULL
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	antibody	1.458546423213736	IUPHAR.LIGAND:10752	iuphar.ligand:10752	LERONLIMAB	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	NULL	SAR-389644	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	MCP-201	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	MCP-201	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	MCP-201	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rosiglitazone XR	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	1.202465753489187	GW685698X	rxcui:705022	FLUTICASONE FUROATE	TRUE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	NULL	Triciribine prodrug	NULL	NULL	NULL	NULL	NULL
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:800	iuphar.ligand:800	TAK-220	FALSE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	MT-112	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Teneligliptin	ncit:C87623	TENELIGLIPTIN	FALSE	FALSE	FALSE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	Colorectal cancer vaccine	NULL	NULL	NULL	NULL	NULL
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	NULL	AS-1670542	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	MGN-1706	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	HER-2/HER-1 vaccine	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	SN-32793	NULL	NULL	NULL	NULL	NULL
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	NULL	AMG888/U3-1287	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	NULL	1.640864726115453	IUPHAR.LIGAND:11253	iuphar.ligand:11253	AX-024	FALSE	FALSE	FALSE
ERBB4 TYROSINE KINASE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7388	ncit:C99131	IDASANUTLIN	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Insulin oral sublingual	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	DM-71	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDX-189	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GLYCOPROTEIN 41	NULL	NULL	TTD	2020.06.01	NULL	NULL	ITV-1	NULL	NULL	NULL	NULL	NULL
HUMAN PAPILLOMAVIRUS PROTEIN E7	NULL	NULL	TTD	2020.06.01	NULL	NULL	ADXS-HPV	drugbank:DB16692	AXALIMOGENE FILOLISBAC	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	INCB24360	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2836	hgnc:1817	CEACAM5	GuideToPharmacology	2024.1	antibody	2.282942227638891	IUPHAR.LIGAND:8251	iuphar.ligand:8251	LABETUZUMAB	FALSE	FALSE	FALSE
TERT MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
THYMIDYLATE SYNTHASE MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
MCL-1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
GLUCAGON RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS 325568	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2840	hgnc:4471	GPR17	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:8267	iuphar.ligand:8267	MILATUZUMAB	FALSE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA 2	hgnc:11768	TGFB2	TTD	2020.06.01	NULL	NULL	AP12009	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	Low dose ITI-007	NULL	NULL	NULL	NULL	NULL
TRANSTHYRETIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-TTR	NULL	NULL	NULL	NULL	NULL
EIF4E-BP2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-EIF4E	NULL	NULL	NULL	NULL	NULL
FGFR4 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-FGFR4	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	NULL	CPG 52364	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 8	hgnc:15632	TLR8	TTD	2020.06.01	NULL	NULL	CPG 52364	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	CPG 52364	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	CXL	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-5172	rxcui:1734630	GRAZOPREVIR	TRUE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	NULL	MER-102	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2602	hgnc:1804	CD52	GuideToPharmacology	2024.1	antibody	70.01022831425932	IUPHAR.LIGAND:6770	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
ENDOSIALIN	hgnc:18219	CD248	TTD	2020.06.01	NULL	NULL	OntecizumabAmatuximab	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	MP-124	NULL	NULL	NULL	NULL	NULL
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BC-7013	iuphar.ligand:11034	BC-7013	FALSE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	WCK-2349	ncit:C166823	ALALEVONADIFLOXACIN	FALSE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	1.458546423213736	KW-3357	chembl:CHEMBL1201554	ANTITHROMBIN ALFA	FALSE	FALSE	FALSE
NFKB MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	DIMS-0150	chembl:CHEMBL5095448	COBITOLIMOD SODIUM	FALSE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	JTZ-951	ncit:C169944	ENARODUSTAT	FALSE	FALSE	FALSE
NCBIGENE:82	hgnc:154	ACTG1P9	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:2945	iuphar.ligand:2945	CHEMERIN	FALSE	FALSE	FALSE
CYTOSINE DEAMINASE	hgnc:13203	AICDA	TTD	2020.06.01	NULL	NULL	JX-929	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	TS-032	NULL	NULL	NULL	NULL	NULL
HEAT SHOCK PROTEIN 70	hgnc:5232	HSPA1A	TTD	2020.06.01	NULL	NULL	AEG-33773	NULL	NULL	NULL	NULL	NULL
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	NULL	LY-2599506	NULL	NULL	NULL	NULL	NULL
GLUCOSE TRANSPORTER TYPE 4	hgnc:11009	SLC2A4	TTD	2020.06.01	NULL	NULL	DS-1150b	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD6423	NULL	NULL	NULL	NULL	NULL
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12979	iuphar.ligand:12979	S-26D [PMID: 37883692]	FALSE	FALSE	FALSE
CANCER/TESTIS ANTIGEN 1	hgnc:2491	CTAG1B	TTD	2020.06.01	NULL	NULL	NY-ESO-1 vaccine	NULL	NULL	NULL	NULL	NULL
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alfimeprase	ncit:C79877	ALFIMEPRASE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	DG-17	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	NULL	PS-178990	NULL	NULL	NULL	NULL	NULL
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	NULL	SBC-014	NULL	NULL	NULL	NULL	NULL
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PC-SOD	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	ATHX-105	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK-625433	chembl:CHEMBL2024212	GSK-625433	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	CR-845 iv infusion	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.2375912725597036	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	CTAP-201	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	DM-CHOC-PEN	ncit:C90539	MIPICOLEDINE	FALSE	FALSE	FALSE
RESPIRATORY SYNCYTIAL VIRUS PROTEIN F	NULL	NULL	TTD	2020.06.01	NULL	NULL	MEDI-557	chembl:CHEMBL2109566	MEDI-557	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	NULL	OP-R003	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	NULL	192C86	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	LY-2428757	NULL	NULL	NULL	NULL	NULL
INFLUENZA M2 PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	TCN-032	chembl:CHEMBL2109619	TCN-032	FALSE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:2901	iuphar.ligand:2901	[3H]RESOLVIN E1	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	CYT-609	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-492	rxcui:1927663	DELAFLOXACIN	TRUE	FALSE	FALSE
PROSTAGLANDIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Iclaprim	ncit:C65877	ICLAPRIM	FALSE	FALSE	FALSE
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	7.001022831425932	SYN-120	chembl:CHEMBL1082508	LANDIPIRDINE	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	9.845188356692718	Iratumumab	ncit:C26441	IRATUMUMAB	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	2.019525817	PLX-5622	chembl:CHEMBL3545079	PLX-5622	FALSE	FALSE	FALSE
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lotilibcin dermatological cream	NULL	NULL	NULL	NULL	NULL
EBOLA VIRUS VP24 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-6003	NULL	NULL	NULL	NULL	NULL
EBOLA VIRUS VP35 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-6003	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAND-5	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-2836	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE C	hgnc:5273	HSPG2	TTD	2020.06.01	NULL	NULL	D-20133	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.2206204673768676	IUPHAR.LIGAND:10357	iuphar.ligand:10357	CDK INHIBITOR 4.35	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	NULL	PRT6207	NULL	NULL	NULL	NULL	NULL
EXPORTIN-1	hgnc:12825	XPO1	TTD	2020.06.01	NULL	NULL	KOS-1815	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VM-1500	NULL	NULL	NULL	NULL	NULL
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Delamanid	ncit:C157406	DELAMANID	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	NC-4016	ncit:C113175	DACH-PLATIN MICELLE NC-4016	FALSE	FALSE	FALSE
FUNGAL CELL MEMBRANE ERGOSTEROL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Candicidin	ncit:C87461	CANDICIDIN	TRUE	FALSE	FALSE
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	activator	0.1773907812016706	IUPHAR.LIGAND:4279	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
RENAL CARCINOMA ANTIGEN NY-REN-56	hgnc:8874	PFKFB3	TTD	2020.06.01	NULL	52.50767123569449	PFK-158	chembl:CHEMBL4303611	PFK-158	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION GENE 3 PROTEIN	hgnc:6476	LAG3	TTD	2020.06.01	NULL	0.6563458904461813	BMS-986016	rxcui:1597876	NIVOLUMAB	TRUE	TRUE	TRUE
IMMUNOGLOBULIN G1K	NULL	NULL	TTD	2020.06.01	NULL	NULL	NKTT-120	drugbank:DB17730	NKTT-120	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAK-063	chembl:CHEMBL3989972	BALIPODECT	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	SAR342434	NULL	NULL	NULL	NULL	NULL
GLUCOSE-DEPENDENT INSULINOTROPIC RECEPTOR	hgnc:19060	GPR119	TTD	2020.06.01	NULL	NULL	DS-8500	NULL	NULL	NULL	NULL	NULL
NEUROPILIN-1	hgnc:8004	NRP1	TTD	2020.06.01	NULL	NULL	RG7347	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-2/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valetizumab	NULL	NULL	NULL	NULL	NULL
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	NULL	MK-8109	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	WY-50295-tromethamine	NULL	NULL	NULL	NULL	NULL
EOSINOPHIL/LYMPHOCYTE-RICH ACCUMULATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PNU-142731A	NULL	NULL	NULL	NULL	NULL
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	blocker	0.2983390411119005	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Colistin	rxcui:2709	COLISTIN	TRUE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:6390	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
CATHEPSIN D	hgnc:2529	CTSD	TTD	2020.06.01	NULL	NULL	PMID10498202C1	NULL	NULL	NULL	NULL	NULL
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	NULL	Demogastrin	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Insulin-lispro	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.079077818	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
BACTERIAL FATTY ACID SYNTHETASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazinamide	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:11869	ncit:C162676	ELZOVANTINIB	FALSE	FALSE	FALSE
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	Staurosporine	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Spectinomycin	rxcui:270	SPECTINOMYCIN	FALSE	FALSE	FALSE
BACTERIAL FUMARATE REDUCTASE FLAVOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxantel pamoate	rxcui:1871176	OXANTEL PAMOATE	FALSE	FALSE	FALSE
PARATHYROID HORMONE RECEPTOR	hgnc:9609	PTH2R	TTD	2020.06.01	NULL	NULL	GSK768974	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzylpenicillin	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
SODIUM/POTASSIUM-TRANSPORTING ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Digitoxin	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
PROTEIN KINASE C EPSILON	hgnc:9401	PRKCE	TTD	2020.06.01	NULL	0.3750547945406749	Bryostatin-1	drugbank:DB11752	BRYOSTATIN 1	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.082559232	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
THYMIDYLATE SYNTHASE	hgnc:12441	TYMS	TTD	2020.06.01	NULL	NULL	Plevitrexed (R)-isomer	NULL	NULL	NULL	NULL	NULL
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	NULL	PD-157695	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triptolide	drugbank:DB12025	TRIPTOLIDE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzylpenicillin	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Kanamycin	rxcui:1727573	KANAMYCIN A	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gentamicine sulfate	NULL	NULL	NULL	NULL	NULL
URIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pegadricase	ncit:C166797	PEGADRICASE	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:7220	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	CHF-4227	NULL	NULL	NULL	NULL	NULL
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.093098708	Mecamylamine	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Insulin transdermal	NULL	NULL	NULL	NULL	NULL
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Josamycin	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	18F-FEDAA-1106	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	Pc4 (topical formulation	NULL	NULL	NULL	NULL	NULL
GLYCINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	MDL-27531	NULL	NULL	NULL	NULL	NULL
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	NULL	DC/I540/KLH vaccine	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD4	hgnc:1678	CD4	TTD	2020.06.01	NULL	NULL	Protein vaccines	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD8	hgnc:1706	CD8A	TTD	2020.06.01	NULL	NULL	Protein vaccines	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1426838892274307	IUPHAR.LIGAND:7220	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
TNF/IL-10 RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PUR-0110	NULL	NULL	NULL	NULL	NULL
RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	LErafAON	drugbank:DB04973	LERAFAON	FALSE	FALSE	FALSE
NITRIC OXIDE ELIMINATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	NOX-700	drugbank:DB05464	NOX-700	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Metformin arginine-hemisuccinimide	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxytetracycline	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Estrogen receptor beta-selective phytoestrogenic formulation	NULL	NULL	NULL	NULL	NULL
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Recombinant batroxobin	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1840	hgnc:3060	DTX1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984016	IUPHAR.LIGAND:10316	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenyltoloxamine	rxcui:33408	PHENYLTOLOXAMINE	TRUE	FALSE	FALSE
DOPAMINE D5 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenyltoloxamine	rxcui:33408	PHENYLTOLOXAMINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Phenyltoloxamine	rxcui:33408	PHENYLTOLOXAMINE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ertapenem	rxcui:325642	ERTAPENEM	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefaclor	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hemoglobin raffimer	ncit:C166918	HEMOGLOBIN RAFFIMER	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.087707691	CB-03-01	rxcui:2474340	CLASCOTERONE	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	Morphine-6-glucuronide	ncit:C166899	MORPHINE GLUCURONIDE	FALSE	FALSE	FALSE
NCBIGENE:715	hgnc:1246	C1R	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	AG140699	NULL	NULL	NULL	NULL	NULL
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Faropenem	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oritavancin	rxcui:1547611	ORITAVANCIN	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-3304	drugbank:DB12149	S-3304	FALSE	FALSE	TRUE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.09745299	Nandrolone	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
FRUCTOSE-1,6-BISPHOSPHATASE	hgnc:3606	FBP1	TTD	2020.06.01	NULL	26.25383561784724	Managlinat dialanetil	ncit:C166705	MANAGLINAT DIALANETIL	FALSE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dalfopristin	rxcui:229369	DALFOPRISTIN	TRUE	FALSE	FALSE
SOMATOTROPIN	hgnc:4261	GH1	TTD	2020.06.01	NULL	NULL	YPEG-Somatropin	NULL	NULL	NULL	NULL	NULL
CATECHOL-O-METHYL-TRANSFERASE	hgnc:2228	COMT	TTD	2020.06.01	NULL	NULL	Entacapone+levodopa+carbidopa	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Entacapone+levodopa+carbidopa	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	AZ-40140	NULL	NULL	NULL	NULL	NULL
CHOLECYSTOKININ RECEPTOR TYPE A	hgnc:1570	CCKAR	TTD	2020.06.01	NULL	NULL	AR-R-1589	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 2	hgnc:7957	NPY2R	TTD	2020.06.01	NULL	NULL	BMS-192548	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	CP-114271	NULL	NULL	NULL	NULL	NULL
PERIPHERAL CAROTID CHEMORECEPTOR	hgnc:2411	CRYGD	TTD	2020.06.01	NULL	26.25383561784724	Doxapram	rxcui:3637	DOXAPRAM	TRUE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	NULL	IDDBCP-150101	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	L-742791	NULL	NULL	NULL	NULL	NULL
MELANOCORTIN RECEPTOR 3	hgnc:6931	MC3R	TTD	2020.06.01	NULL	NULL	Melanotetan II	NULL	NULL	NULL	NULL	NULL
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	NULL	Melanotetan II	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE Y RECEPTOR TYPE 5	hgnc:7958	NPY5R	TTD	2020.06.01	NULL	NULL	NPY antagonist	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	Low dose fentanyl	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	HER1-VSSP vaccine	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ANDROSTERONE	rxcui:1312359	ANDROSTERONE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Meticillin	rxcui:2181306	METHICILLIN	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	1.346350544504987	Ranibizumab	rxcui:595060	RANIBIZUMAB	TRUE	FALSE	FALSE
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	6.563458904461812	PRX-08066	drugbank:DB05607	PRX-08066	FALSE	FALSE	FALSE
WISKOTT-ALDRICH SYNDROME PROTEIN	hgnc:12731	WAS	TTD	2020.06.01	NULL	NULL	Hematopoietic stem cell gene therapy	NULL	NULL	NULL	NULL	NULL
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-0865	chembl:CHEMBL497011	LINAPRAZAN	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	11C-PBR-28	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mesalazine	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Varenicline	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	NOX-F37	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	GPI-16072	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Retapamulin	rxcui:642274	RETAPAMULIN	TRUE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	Recombinant RGD-hirudin	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	RO-26-2853	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	1192U90	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	1192U90	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	1192U90	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BL-1020	drugbank:DB05687	BL-1020	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	BL-1020	drugbank:DB05687	BL-1020	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	0.596678082	Oral azacitidine	ncit:C118288	ORAL AZACITIDINE	FALSE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	NULL	D1 agonist D2 antagonist	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	D1 agonist D2 antagonist	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Org-23366	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Org-23366	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	NULL	Org-23366	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PD-157695	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-157695	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	PD-158771	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PD-158771	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-158771	NULL	NULL	NULL	NULL	NULL
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD-165167	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	SSR-504734	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	U-99194A	NULL	NULL	NULL	NULL	NULL
BACTERIAL RNA POLYMERASE SWITCH REGION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rifalazil	ncit:C152213	RIFALAZIL	FALSE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	5.834185692854944	Organon	chembl:CHEMBL427683	ORGANON	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.1479089330582944	CI-1033	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.2917092846427472	Procaine	rxcui:8701	PROCAINE	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.5645986154375752	Benzocaine	rxcui:1399	BENZOCAINE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.7395446652914718	Alacizumab pegol	ncit:C61438	ALACIZUMAB PEGOL	FALSE	FALSE	FALSE
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	Ad-IFN-alpha	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	NULL	STX-140	NULL	NULL	NULL	NULL	NULL
DNA SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nelarabine	rxcui:274771	NELARABINE	TRUE	FALSE	TRUE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3661	iuphar.ligand:3661	[125I]CXCL11 (HUMAN)	FALSE	FALSE	FALSE
INTERLEUKIN-1	hgnc:5991	IL1A	TTD	2020.06.01	NULL	NULL	K-832	NULL	NULL	NULL	NULL	NULL
PHENYLALANINE HYDROXYLASE	hgnc:8582	PAH	TTD	2020.06.01	NULL	8.751278539282415	Sapropterin hydrochloride	chembl:CHEMBL1201775	SAPROPTERIN DIHYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2900	iuphar.ligand:2900	ISOTHIOUREA-1A	FALSE	FALSE	FALSE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.637458239	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
ALBENDAZOLE MONOOXYGENASE	hgnc:2637	CYP3A4	TTD	2020.06.01	NULL	0.0008899	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	GPC-3298306	NULL	NULL	NULL	NULL	NULL
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RQ-00000004	ncit:C152542	TEGOPRAZAN	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:852	iuphar.ligand:852	T134	FALSE	FALSE	FALSE
ASPERGILLUS MANNITOL 2-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannitol	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
NCBIGENE:1374	hgnc:2328	CPT1A	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:10548	iuphar.ligand:10548	COMPOUND 10 [PMID: 31663733]	FALSE	FALSE	FALSE
ASPERGILLUS MANNITOL-1-PHOSPHATE 5-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannitol	rxcui:6628	MANNITOL	TRUE	FALSE	FALSE
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rottlerin	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	NULL	AIKO-150	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	AIKO-150	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	1.280674908	GRC-6211	chembl:CHEMBL3545107	GRC-6211	FALSE	FALSE	FALSE
ERYTHROPOIETIN	hgnc:3415	EPO	TTD	2020.06.01	NULL	NULL	Erythropoietin-transfected autologous cell therapy	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pivmecillinam	rxcui:627	AMDINOCILLIN PIVOXIL	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	0.6563458904461812	Tolbutamide	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1356	hgnc:2295	CP	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:8795	iuphar.ligand:8795	COMPOUND 7P [PMID: 7861416]	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	0.031822831	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bendamustine hydrochloride	rxcui:1114693	BENDAMUSTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HEPATITIS B VIRUS POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Telbivudine	rxcui:474128	TELBIVUDINE	TRUE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penciclovir	rxcui:59839	PENCICLOVIR	TRUE	FALSE	FALSE
NCBIGENE:1374	hgnc:2328	CPT1A	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8799	ncit:C79817	AZALANSTAT	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valaciclovir	rxcui:73645	VALACYCLOVIR	TRUE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.8751278539282416	Rolofylline	ncit:C96195	ROLOFYLLINE	FALSE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	2.983390411119005	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceftibuten	rxcui:20492	CEFTIBUTEN	TRUE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	5.527123287967842	IUPHAR.LIGAND:6844	rxcui:1310520	TERIFLUNOMIDE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Methylene blue	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
RESPIRATORY SYNCYTIAL VIRUS PROTEIN F	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lasofoxifene	ncit:C80679	LASOFOXIFENE	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ketoconazole	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	NRT inhibitor	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:6286	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
KERATIN 6A MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TD-101	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD1480	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3B	hgnc:2979	DNMT3B	TTD	2020.06.01	NULL	0.1325951293830669	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8301	iuphar.ligand:8301	COMPOUND 1 [XIAO ET AL. 2014]	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.2187819634820604	Pazopanib HCl	chembl:CHEMBL1201733	PAZOPANIB HYDROCHLORIDE	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	0.054243462	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1232574442152452	Pazopanib HCl	chembl:CHEMBL1201733	PAZOPANIB HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:2650	hgnc:4203	GCNT1	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7018	iuphar.ligand:7018	BROMO-DEAZA-SAH	FALSE	FALSE	FALSE
S100 CALCIUM-BINDING PROTEIN A4	hgnc:10494	S100A4	TTD	2020.06.01	NULL	NULL	SP-MET-1	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	SULFAMIDE	chembl:CHEMBL355001	SULFAMIDE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	SULFAMIDE	chembl:CHEMBL355001	SULFAMIDE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	EQ-917	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE XIV	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRIENTINE	rxcui:10798	TRIENTINE	TRUE	FALSE	FALSE
NCBIGENE:2006	hgnc:3327	ELN	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8057	iuphar.ligand:8057	XMD8-92	FALSE	FALSE	FALSE
BACTERIAL PROTECTIVE ANTIGEN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Raxibacumab	rxcui:1366567	RAXIBACUMAB	TRUE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	LEISH-F1	NULL	NULL	NULL	NULL	NULL
ACTIVATION B7-1 ANTIGEN	hgnc:1700	CD80	TTD	2020.06.01	NULL	NULL	MAXY-4	NULL	NULL	NULL	NULL	NULL
T-LYMPHOCYTE ACTIVATION ANTIGEN CD86	NULL	NULL	TTD	2020.06.01	NULL	NULL	MAXY-4	NULL	NULL	NULL	NULL	NULL
PLATELET GLYCOPROTEIN VI	hgnc:14388	GP6	TTD	2020.06.01	NULL	NULL	Revacept	NULL	NULL	NULL	NULL	NULL
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	CP-601927	drugbank:DB12244	CP-601927	FALSE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	Iofolastat I-124	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2605	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:7018	iuphar.ligand:7018	BROMO-DEAZA-SAH	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	NULL	PF-4455242	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-V/BETA-3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Intetumumab	ncit:C61070	INTETUMUMAB	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AR-12286	ncit:C152866	VEROSUDIL	FALSE	FALSE	FALSE
ACETALDEHYDE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Calcium carbimide	rxcui:1902	CALCIUM CARBIMIDE	FALSE	FALSE	FALSE
NCBIGENE:1505	hgnc:2933	DMPK	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
GLUCOSE-DEPENDENT INSULINOTROPIC RECEPTOR	hgnc:19060	GPR119	TTD	2020.06.01	NULL	NULL	APD-597	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS SERINE PROTEASE NS4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PHX-1766	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Aflunov	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-6186	drugbank:DB12999	MK-6186	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	XMT-1001	drugbank:DB06069	XMT-1001	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	INM-176	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GAG PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN	NULL	NULL	NULL	NULL	NULL
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1877	iuphar.ligand:1877	15-DEOXY-&DELTA;12,14-PGJ2	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS NEGATIVE FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ad35-GRIN	NULL	NULL	NULL	NULL	NULL
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	NULL	PMID22911925C2	NULL	NULL	NULL	NULL	NULL
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nitrofurazone	rxcui:7455	NITROFURAZONE	TRUE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TDZD-8	iuphar.ligand:5977	GSK-3BETA INHIBITOR I	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:1881	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
GROWTH/DIFFERENTIATION FACTOR 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	ACE-031	chembl:CHEMBL2108674	RAMATERCEPT	FALSE	FALSE	FALSE
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	IFN alpha kinoid	NULL	NULL	NULL	NULL	NULL
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.044878351	VE-822	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ME-1071	NULL	NULL	NULL	NULL	NULL
PI3K/AKT/MTOR PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	ON-01210.Na	chembl:CHEMBL2219410	RECILISIB SODIUM	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:1891	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
BETA-SITE APP-CLEAVING ENZYME 2	hgnc:934	BACE2	TTD	2020.06.01	NULL	NULL	example 98 (WO2011020806)	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	MVA HER-2 AutoVac	NULL	NULL	NULL	NULL	NULL
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MSC1936369B	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	NULL	Remogli ozin-etabonate	NULL	NULL	NULL	NULL	NULL
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:10170	iuphar.ligand:10170	AM-461	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	0.7721716358190367	Darbufelone	ncit:C81061	DARBUFELONE	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	NULL	ASCJ-9 topical	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	TGFK08AA-ER	NULL	NULL	NULL	NULL	NULL
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
THYROID HORMONE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	VIA-3196	ncit:C170368	RESMETIROM	TRUE	FALSE	FALSE
PROLIFERATING CELL NUCLEAR ANTIGEN	hgnc:8729	PCNA	TTD	2020.06.01	NULL	10.50153424713889	ATX-101	drugbank:DB05780	ATX-101	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:7650	iuphar.ligand:7650	UNC9975	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-3102	ncit:C174662	OMARIGLIPTIN	FALSE	FALSE	FALSE
PLASMODIAL PHOSPHOLIPID METABOLISM	NULL	NULL	TTD	2020.06.01	NULL	NULL	CDRI-97/78	iuphar.ligand:10399	CDRI-97/78	FALSE	FALSE	FALSE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-494	iuphar.ligand:9246	UPADACITINIB	FALSE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-852927	chembl:CHEMBL3545047	BMS-852927	FALSE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CS-8080	chembl:CHEMBL3545238	CS-8080	FALSE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	LXR 623	NULL	NULL	NULL	NULL	NULL
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.046425881	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pitolisant	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	RAD-140	drugbank:DB13939	RAD-140	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1481697953740938	AZD9291	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:8161	iuphar.ligand:8161	COMPOUND 17 [PMID: 23642479]	FALSE	FALSE	FALSE
ENDOGENOUS GUT PEPTIDE	hgnc:8524	OVGP1	TTD	2020.06.01	NULL	NULL	GSK2890457	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XIII	hgnc:3534	F13B	TTD	2020.06.01	NULL	NULL	NN1841	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Azlocillin	rxcui:1266	AZLOCILLIN	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9352	iuphar.ligand:9352	HARMINE	FALSE	FALSE	FALSE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	5.104912481248077	LDE225	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
INTERFERON-GAMMA	hgnc:5438	IFNG	TTD	2020.06.01	NULL	NULL	AMG 811	NULL	NULL	NULL	NULL	NULL
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	UFT/leucovorin calcium	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8055	drugbank:DB08691	ETHYL 3-[(E)-2-AMINO-1-CYANOETHENYL]-6,7-DICHLORO-1-METHYL-1H-INDOLE-2-CARBOXYLATE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 39 MEMBER 6	hgnc:18607	SLC39A6	TTD	2020.06.01	NULL	NULL	SGN LIV1A	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS LEUCYL-TRNA SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK-2251052	ncit:C166950	EPETRABOROLE	FALSE	FALSE	FALSE
PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9	hgnc:20001	PCSK9	TTD	2020.06.01	NULL	4.039051633514961	LY3015014	chembl:CHEMBL4298016	FROVOCIMAB	FALSE	FALSE	FALSE
PSEUDOMONAS PCRV PROTEIN TYPE III	NULL	NULL	TTD	2020.06.01	NULL	NULL	MEDI3902	chembl:CHEMBL4298031	GREMUBAMAB	FALSE	FALSE	FALSE
PSEUDOMONAS PSL EXOPOLYSACCHARIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MEDI3902	chembl:CHEMBL4298031	GREMUBAMAB	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pennvax-G	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rhopressa	rxcui:1992864	NETARSUDIL	TRUE	FALSE	FALSE
FUSION PROTEIN FGFR3-TACC3	NULL	NULL	TTD	2020.06.01	NULL	NULL	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	2.187819634820604	ImMucin	drugbank:DB17403	IMMUCIN	FALSE	FALSE	FALSE
TGF-BETA RECEPTOR TYPE I	hgnc:11772	TGFBR1	TTD	2020.06.01	NULL	2.500365296937833	LY2157299	ncit:C116891	GALUNISERTIB	FALSE	FALSE	FALSE
ADVANCED GLYCOSYLATION END PRODUCT RECEPTOR	hgnc:320	AGER	TTD	2020.06.01	NULL	NULL	TTP-448	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	CT 327	NULL	NULL	NULL	NULL	NULL
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	DPK-060	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Intedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.1312691780892362	Intedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.4773424657790409	Dulaglutide	rxcui:1551291	DULAGLUTIDE	TRUE	FALSE	FALSE
UTROPHIN	hgnc:12635	UTRN	TTD	2020.06.01	NULL	26.25383561784724	SMT-C1100	ncit:C166897	EZUTROMID	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.1374032518317239	Intedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
KAPPA MYELOMA ANTIGEN	NULL	NULL	TTD	2020.06.01	NULL	NULL	MDX-1097	drugbank:DB18383	MDX-1097	FALSE	FALSE	FALSE
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK2586184	ncit:C152385	SOLCITINIB	FALSE	FALSE	FALSE
HEPATITIS C VIRUS SERINE PROTEASE NS4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-6325	drugbank:DB15249	MK-6325	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-21	hgnc:3678	FGF21	TTD	2020.06.01	NULL	NULL	PF-05231023	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	CNT0-1959	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.8751278539282416	MSC2156119	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	7.501095891	JNJ-40411813	drugbank:DB12059	JNJ-40411813	FALSE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	CDX-301	chembl:CHEMBL4650387	CDX-301	FALSE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	LY2963016	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	BL-7040	NULL	NULL	NULL	NULL	NULL
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	NULL	UNBS-1450	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Plasma derived human butyrylcholinesterase	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,2,3-triazole derivative 1	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	1.944728564284981	MT-1303	ncit:C166641	AMISELIMOD	FALSE	FALSE	FALSE
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	8.751278539282415	GSK2879552	iuphar.ligand:9116	GSK2879552	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Elvitegravir	rxcui:1306286	ELVITEGRAVIR	TRUE	FALSE	FALSE
HEPATITIS C VIRUS SERINE PROTEASE NS3/4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Simeprevir	rxcui:1482790	SIMEPREVIR	FALSE	FALSE	FALSE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	NULL	Testogen TDS	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Meropenem + vaborbactam	NULL	NULL	NULL	NULL	NULL
CYTOMEGALOVIRUS TERMINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-8228	rxcui:1988648	LETERMOVIR	TRUE	FALSE	FALSE
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sarecycline	rxcui:2059018	SARECYCLINE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bictegravir, emtricitabine and tenofovir alafenamide	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bictegravir, emtricitabine and tenofovir alafenamide	NULL	NULL	NULL	NULL	NULL
G-PROTEIN COUPLED ESTROGEN RECEPTOR 1	hgnc:4485	GPER1	TTD	2020.06.01	NULL	NULL	Segesterone acetate and ethinyl estradiol vaginal system	NULL	NULL	NULL	NULL	NULL
CHLORIDE CHANNEL UNSPECIFIC	hgnc:2014	CLC	TTD	2020.06.01	NULL	6.563458904461812	BLZ-100	chembl:CHEMBL3990023	TOZULERISTIDE	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.130291988	Lacosamide	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
TWIK-RELATED ACID-SENSITIVE POTASSIUM CHANNEL 1	hgnc:6278	KCNK3	TTD	2020.06.01	NULL	NULL	BAY-2253651a	NULL	NULL	NULL	NULL	NULL
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA2	NULL	NULL	TTD	2020.06.01	NULL	NULL	AP-30663	NULL	NULL	NULL	NULL	NULL
CALCIUM-ACTIVATED POTASSIUM CHANNEL KCA2	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAD-1883	ncit:C171756	RIMTUZALCAP	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	NULL	Intravenous glibenclamide	NULL	NULL	NULL	NULL	NULL
LONG TRANSIENT RECEPTOR POTENTIAL CHANNEL 4	hgnc:17993	TRPM4	TTD	2020.06.01	NULL	NULL	Intravenous glibenclamide	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2010	hgnc:3331	EMD	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9352	iuphar.ligand:9352	HARMINE	FALSE	FALSE	FALSE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	NULL	MDAM (y-methylene-10-deazaaminopterin)	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	NULL	Anisodine	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	NULL	Anisodine	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bleomycin	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.045898314	Ajmalicine	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	VAL-083	chembl:CHEMBL3137322	DIANHYDROGALACTITOL	FALSE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Netilmicin	rxcui:7337	NETILMICIN	FALSE	FALSE	FALSE
APOLIPOPROTEIN A-I	hgnc:600	APOA1	TTD	2020.06.01	NULL	NULL	MDCO-216	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	VCL-1M01	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lenapenem hydrochloride hydrate	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	ONO-2506	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clidinium	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
CHOLINERGIC RECEPTOR UNSPECIFIC	ncbigene:1125	CHR	TTD	2020.06.01	NULL	3.281729452230906	Cisatracurium	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	P2B-001	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	P2B-001	NULL	NULL	NULL	NULL	NULL
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	OXY-111A	NULL	NULL	NULL	NULL	NULL
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.2051080907644316	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.012974468	Rapamycin	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefmetazole	rxcui:2182	CEFMETAZOLE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefoperazone	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	SNN-0031	NULL	NULL	NULL	NULL	NULL
WNT PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ipafricept	ncit:C102565	IPAFRICEPT	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	CKD602	hemonc:64	BELOTECAN	FALSE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	NULL	SK-NBP601	NULL	NULL	NULL	NULL	NULL
GRANULOCYTE COLONY-STIMULATING FACTOR	hgnc:2438	CSF3	TTD	2020.06.01	NULL	4.375639269641208	SPI-2012	rxcui:2612526	EFLAPEGRASTIM	TRUE	FALSE	FALSE
GALACTOSYLTRANSFERASE	hgnc:4135	GALT	TTD	2020.06.01	NULL	NULL	HyperAcute vaccine	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ADENOVECTOR AD35	NULL	NULL	TTD	2020.06.01	NULL	NULL	VRC-HIVDNA016-00-VP	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	AFO-18	NULL	NULL	NULL	NULL	NULL
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Plasmin	rxcui:4388	PLASMIN	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	NPC-01	NULL	NULL	NULL	NULL	NULL
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	NULL	NPC-01	NULL	NULL	NULL	NULL	NULL
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	NULL	GSK-1322888	NULL	NULL	NULL	NULL	NULL
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	NNC-0123-0000-0338	NULL	NULL	NULL	NULL	NULL
ACID-SENSING ION CHANNEL 1	hgnc:100	ASIC1	TTD	2020.06.01	NULL	NULL	PPC-5650	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:7646	ncit:C80868	FALNIDAMOL	FALSE	FALSE	FALSE
N-SULPHOGLUCOSAMINE SULPHOHYDROLASE	hgnc:10818	SGSH	TTD	2020.06.01	NULL	52.50767123569449	HGT-1410	chembl:CHEMBL4297976	N-SULFOGLUCOSAMINE SULFOHYDROLASE RECOMBINANT	FALSE	FALSE	FALSE
MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN	hgnc:7467	MTTP	TTD	2020.06.01	NULL	8.751278539282415	JNJ-16269110	chembl:CHEMBL2103860	USISTAPIDE	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR T Cells	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	GSK2339345	NULL	NULL	NULL	NULL	NULL
WNT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	SM04755	ncit:C122693	WNT SIGNALING INHIBITOR SM04755	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	CART30	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-7	hgnc:6023	IL7	TTD	2020.06.01	NULL	NULL	GSK2618960	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Chimeric Antigen Receptor Modified T cells Targeting CD19	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	HuCART19	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	ICasp9M28z T cell	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR T-cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART-19 autologous T-cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-targeting CAR T Cells	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	Anti-meso-CAR vector transduced T cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CART22 cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Anti-CD20-CAR-transduced T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19CART	NULL	NULL	NULL	NULL	NULL
CO-STIMULATORY MOLECULE 4-1BB	hgnc:11924	TNFRSF9	TTD	2020.06.01	NULL	NULL	MG7-CART	NULL	NULL	NULL	NULL	NULL
GASTRIC CARCINOMA-ASSOCIATED ANTIGEN MG7	NULL	NULL	TTD	2020.06.01	NULL	NULL	MG7-CART	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	GLYCAR T cells	NULL	NULL	NULL	NULL	NULL
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	NULL	CAR-T cells recognizing EpCAM	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	NULL	Anti-PD-L1 CSR T cells	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	Anti-BCMA-CAR-transduced T cells	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	4SCAR-GD2	ncit:C128896	4SCAR-GD2-MODIFIED T-LYMPHOCYTES	FALSE	FALSE	FALSE
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting EpCAM	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	Anti-CD30-CAR T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19/20-CAR vector-transduced T cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Anti-CD19/20-CAR vector-transduced T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 targeted chimeric antigen receptor T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR30	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR30	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR38	NULL	NULL	NULL	NULL	NULL
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR38	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR70	NULL	NULL	NULL	NULL	NULL
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	NULL	4SCAR19 and 4SCAR70	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	GPC3-CART cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	ARI-0001 cells	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR VARIANT III	NULL	NULL	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting EGFRviii	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CD20-CART	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-CAR T Cells	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD117	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting Mucl	NULL	NULL	NULL	NULL	NULL
SYNDECAN-1	hgnc:10658	SDC1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD138	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	TriCAR-T-CD19	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HER2-specific CAR T cell	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA CART	NULL	NULL	NULL	NULL	NULL
DELTA-LIKE PROTEIN 3	hgnc:2909	DLL3	TTD	2020.06.01	NULL	26.25383561784724	AMG 119	ncit:C150586	CAR T-CELLS AMG 119	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-CAR-T Cells	NULL	NULL	NULL	NULL	NULL
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	NULL	Dapagliflozin Propanediol; Saxagliptin Hydrochloride	NULL	NULL	NULL	NULL	NULL
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Desonide	rxcui:3254	DESONIDE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ergoloid mesylate	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Esomeprazole	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fluconazole	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flumethasone Pivalate	rxcui:25113	FLUMETHASONE PIVALATE	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	Insulin-aspart	NULL	NULL	NULL	NULL	NULL
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-3/BETA-4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Levopropoxyphene Napsylate Anhydrous	ncit:C90775	LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Meropenem	rxcui:1546029	MEROPENEM ANHYDROUS	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Miconazole	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Norfloxacin	rxcui:7517	NORFLOXACIN	TRUE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ofloxacin	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
GASTRIC H(+)/K(+) ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
RESPIRATORY SYNCYTIAL VIRUS PROTEIN F	NULL	NULL	TTD	2020.06.01	NULL	NULL	Palivizumab	rxcui:194279	PALIVIZUMAB	TRUE	FALSE	FALSE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Prednicarbate	rxcui:34369	PREDNICARBATE	TRUE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sparfloxacin	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sparfloxacin	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
INTERLEUKIN 6 RECEPTOR	hgnc:6019	IL6R	TTD	2020.06.01	NULL	12.11715490054488	Sarilumab	rxcui:1923319	SARILUMAB	TRUE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valacyclovir Hydrochloride	rxcui:236081	VALACYCLOVIR HYDROCHLORIDE	TRUE	FALSE	FALSE
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vadimezan	ncit:C2504	VADIMEZAN	FALSE	FALSE	TRUE
MUTATED KRAS	NULL	NULL	TTD	2020.06.01	NULL	NULL	GI-4000 in combination with gemcitabine	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	PMI-005	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	CZEN-002	NULL	NULL	NULL	NULL	NULL
APOLIPOPROTEIN A MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-APO(a)	NULL	NULL	NULL	NULL	NULL
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	0.6177373086552295	Zolmitriptan	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.008621949	IUPHAR.LIGAND:5717	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
DMPK MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-DMPK	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	MK-866	NULL	NULL	NULL	NULL	NULL
SOMATOSTATIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	FK-962	chembl:CHEMBL4802206	FK-962	FALSE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Grepafloxacin	rxcui:83719	GREPAFLOXACIN	FALSE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ozenoxacin	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ozenoxacin	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	MEDI7814	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PPI-461	NULL	NULL	NULL	NULL	NULL
C-X-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1060	CXCR5	TTD	2020.06.01	NULL	NULL	SAR113244	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C1S COMPONENT	hgnc:1247	C1S	TTD	2020.06.01	NULL	NULL	TS01	NULL	NULL	NULL	NULL	NULL
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.091317689	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	NULL	ZYT-1	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II BETA	hgnc:11990	TOP2B	TTD	2020.06.01	NULL	NULL	XK-469	NULL	NULL	NULL	NULL	NULL
NEUROMEDIN-K RECEPTOR	hgnc:11528	TACR3	TTD	2020.06.01	NULL	5.834185692854944	AZD2624	ncit:C166698	PAVINETANT	FALSE	FALSE	FALSE
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-288	drugbank:DB15192	ABT-288	FALSE	FALSE	FALSE
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 10	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 9	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 2	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 8	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 9	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.2500365296937833	LY3164530	ncit:C118281	ANTI-MET/EGFR MONOCLONAL ANTIBODY LY3164530	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.6403374540938354	AFM-11	chembl:CHEMBL4297874	AFM-11	FALSE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clorgyline	drugbank:DB04017	CLORGILINE	FALSE	FALSE	FALSE
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	(-)-deprenyl	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	3-Hydroxy-2-butanone	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	HouttuynoidA	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	KadcoccitoneA	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	MyriberineA	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure1-Aphanamixoid A	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure1-Sarcaboside B	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure3-Aspeverin	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 5-O-methyl-M30	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-10	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-10	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C12	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C16	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C20	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C4	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C7	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 8	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 8	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MRL20	iuphar.ligand:6742	MRL20	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylpropionic acid derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-H	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-H	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2013059587(VI, 2nd set)	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-17	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-19	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-22	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-29	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-32	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-34	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-39	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-47	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-7	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.3	hgnc:10590	SCN3A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Cyclopropyl-spiro piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Methylsulfonylbenzamide derivative 2	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Pyrrolo-benzo-diazine derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.3	hgnc:10590	SCN3A	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 6	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	NULL	0.2500365296937833	IUPHAR.LIGAND:4918	iuphar.ligand:4918	EPIREGULIN	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 6	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-quinolin-benzene sulphonamide derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2012832440110	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US20138552206 4	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2013082253 32	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tihourea derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	6,6-fused nitrogenous heterocyclic compound 1	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.1312691780892362	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Aminopyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Azaindole derivative 1	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-13	hgnc:5973	IL13	TTD	2020.06.01	NULL	8.751278539282415	Anrukinzumab	ncit:C95781	ANRUKINZUMAB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Azaindole derivative 2	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Deuterated 3-cyanoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Deuterated 3-cyanoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-11a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-11b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-11c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-15b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-16b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-21a	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:10494	iuphar.ligand:10494	SWE101	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-21a	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-21a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-23c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-25	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-26b	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-28b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-29b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-31a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-31b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-37b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-37b	NULL	NULL	NULL	NULL	NULL
ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-42	NULL	NULL	NULL	NULL	NULL
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:10315	ncit:C170253	OMIDENEPAG	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-42	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-46	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-5	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-1	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-102	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-104	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-109	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-110	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20120277229 39(1.1)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20120277229 44(1.4)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20130053382 38(5-7)	NULL	NULL	NULL	NULL	NULL
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.2430910705356226	IUPHAR.LIGAND:1936	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2011137219 35(1-11)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolopyridines and imidazopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrido[4,3-d]pyrimidin-5(6H)-one derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidinone derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 11	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 12	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 14	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 18	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 19	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 20	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 22	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 24	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 29	NULL	NULL	NULL	NULL	NULL
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.1988926940746003	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 30	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 9	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Bicyclic hexapeptide derivative 1	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Bicyclic hexapeptide derivative 2	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 5	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Imidazo bicyclic iminium derivative 6	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-11	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-12	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-13	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-24	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-26	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-27	NULL	NULL	NULL	NULL	NULL
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1935	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-32	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-34	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-35	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-38	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-43	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-44	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-50	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-50	NULL	NULL	NULL	NULL	NULL
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1936	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-50	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-50	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-62	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-63	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-64	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 22	NULL	NULL	NULL	NULL	NULL
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.1067229090156392	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750M2	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750TG7-112-2	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750TG8-15	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	PMID25776143-Compound-1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.6403374540938354	IUPHAR.LIGAND:1952	iuphar.ligand:1952	L-161,982 (EP4A)	FALSE	FALSE	FALSE
INTEGRIN ALPHA-5/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMEP	ncit:C90537	PLASMID ENCODING ANTIANGIOGENIC METARGIDIN PEPTIDE	FALSE	FALSE	FALSE
INTEGRIN ALPHA-V/BETA-3	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMEP	ncit:C90537	PLASMID ENCODING ANTIANGIOGENIC METARGIDIN PEPTIDE	FALSE	FALSE	FALSE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	3-substituted-2-furancarboxylic acid hydrazide derivative 1	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	3-substituted-2-furancarboxylic acid hydrazide derivative 5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.6403374540938354	IUPHAR.LIGAND:1912	iuphar.ligand:1912	17-PHENYL-&OMEGA;-TRINOR-PGE2	FALSE	FALSE	FALSE
JUN N TERMINAL KINASE	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-Q1	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-Q1	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140031349A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140031349B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140031349C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140142115B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140336177E	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2010129379C	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.1367387271762877	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2012058116A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013028474A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013028474B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014015495B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014015495D	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014150132B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014150132C	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:7422	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
UBIQUITIN CARBOXYL-TERMINAL HYDROLASE 14	hgnc:12612	USP14	TTD	2020.06.01	NULL	NULL	PMID26077642-Compound-Figure3A	NULL	NULL	NULL	NULL	NULL
UBIQUITIN C-TERMINAL HYDROLASE UCH37	hgnc:19678	UCHL5	TTD	2020.06.01	NULL	NULL	PMID26077642-Compound-Figure3A	NULL	NULL	NULL	NULL	NULL
ZINC FINGER-CONTAINING UBIQUITIN PEPTIDASE 1	hgnc:21224	ZUP1	TTD	2020.06.01	NULL	NULL	PMID26077642-Compound-Figure3G	NULL	NULL	NULL	NULL	NULL
ZINC FINGER-CONTAINING UBIQUITIN PEPTIDASE 1	hgnc:21224	ZUP1	TTD	2020.06.01	NULL	NULL	PMID26077642-Compound-Figure3H	NULL	NULL	NULL	NULL	NULL
HERPESVIRUS UBIQUITIN-SPECIFIC PROTEASE	hgnc:12630	USP7	TTD	2020.06.01	NULL	NULL	PMID26077642-Compound-Vif1	NULL	NULL	NULL	NULL	NULL
UBIQUITIN CARBOXYL-TERMINAL HYDROLASE 14	hgnc:12612	USP14	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 4	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	2-pyrazinone derivative 3	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	2-pyrazinone derivative 4	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	2-pyrazinone derivative 5	NULL	NULL	NULL	NULL	NULL
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:12896	ncit:C174042	IMLUNESTRANT	FALSE	FALSE	FALSE
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 57	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 57	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 66	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 69	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	4-(thiazol-5-yl)-pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	4-(thiazol-5-yl)-pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	4-(thiazol-5-yl)-pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	4-(thiazol-5-yl)-pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Aniline derivative 1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3911	iuphar.ligand:3911	RES7011	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	Aniline derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Enol carbamate derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Isoxazoline derivative 4	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Ketoheterocycle derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Ketoheterocycle derivative 4	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Tetrazolyl urea derivative 1	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2015	hgnc:3336	ADGRE1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8168	iuphar.ligand:8168	COMPOUND 27 [PMID: 19854648]	FALSE	FALSE	FALSE
STAPHYLOCOCCUS ALPHA-HEMOLYSIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASN100	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS FIVE LEUKOCIDIN TOXINS	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASN100	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	Indole and benzimidazole derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Dihydroisoxazole derivative 2	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Dipeptide analog 2	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Dipeptide analog 3	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Peptide analog 53	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-16	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-24	NULL	NULL	NULL	NULL	NULL
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	blocker	0.051885051	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 4	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 4	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 5	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 5	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 6	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 6	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 7	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 7	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Benzazepine derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Benzazepine derivative 4	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Benzazepine derivative 5	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Benzazepine derivative 6	NULL	NULL	NULL	NULL	NULL
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.1151484018326633	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Benzoyl-piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Benzoyl-piperidine derivative 2	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Diarylamine and arylheteroarylamine pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 10	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 3	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 8	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Piperazine derivative 3	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Piperazine derivative 4	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	PMID26609882-Compound-58	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	PMID26609882-Compound-83	NULL	NULL	NULL	NULL	NULL
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	blocker	0.1201548540862574	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 68	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 74	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 75	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 25	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 25	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 25	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Quinoline derivative 2	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Quinoline derivative 2	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolidine derivative 3	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolidine derivative 4	NULL	NULL	NULL	NULL	NULL
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.1256164383629055	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 12	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 2	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 10	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	C-linked disaccharide biphenyl mannoside derivative 6	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 9	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-113	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-114	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-117a	NULL	NULL	NULL	NULL	NULL
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.1067229090156392	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-117b	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 3	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 3	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 4	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 4	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 5	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 5	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 8	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 8	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure11topright	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure12bottommiddle02	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure12topmiddile	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle05	NULL	NULL	NULL	NULL	NULL
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.2561349816375342	IUPHAR.LIGAND:4156	iuphar.ligand:4156	CGS8216	FALSE	FALSE	FALSE
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle08	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9topright01	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	3-(phenoxymethyl) benzylamine derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	P-coumaric acid derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	P-coumaric acid derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-115	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-122	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-126	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-30	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-32	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-50	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-51	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Polyhydroxy benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Polyhydroxy benzamide derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 10	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 14	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 16	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 18	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 22	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 31	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 8	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Thiazolidine derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Thiazolidine derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Thiazoline derivative 2	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	2,2-dimethylbenzopyran derivative 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 13	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 5	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 8	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-23	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-31	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 6	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 8	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Peptide analog 71	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Peptide analog 72	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Piperidine derivative 2	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 12	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 13	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Aryl cyclopropylamine derivative 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 13	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 13	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 9	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1B	hgnc:21577	KDM1B	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-46	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 17	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-1	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-13	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-13	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-14	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-14	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-17	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-17	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-20	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-20	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 3	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 3	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 5	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 5	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 5	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 6	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 6	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 6	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 8	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 8	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 8	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 1	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 3	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Isoxazoles and isoxazoline derivative 1	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Isoxazoles and isoxazoline derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-31	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-32	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-33	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Tricyclic phytocannabinoid derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Tricyclic phytocannabinoid derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Tricyclic phytocannabinoid derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Tricyclic phytocannabinoid derivative 2	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Amidopyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Amidopyrazole derivative 4	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Amidopyrazole derivative 6	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Indazole amide derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [1,5-a]pyrimidin-7-yl derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	PMID27321640-Compound-58	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Triazolo-phthalazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-14	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE BETA-1	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	NULL	Pyrimido[4,5-d] pyrimidines and pyrido[4,3-d] pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-1	hgnc:10430	RPS6KA1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	3-benzyloxyphenyloxoacetic acid derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Phenylthioacetate derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	PMID27414413-Compound-Figure6right	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Ring-fused compound 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 10	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-93	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-94	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-99	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	2-cyclopropyl-4-substituted-phenoxy-quinoline derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Lactol derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Lactol derivative 2	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	PMID27537201-Compound-Figure13c	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Sterol derivative 1	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	2-piperidine thiazole derivative 1	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-13	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-17	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-6	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-9	NULL	NULL	NULL	NULL	NULL
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	PMID27551786-Compound-I	NULL	NULL	NULL	NULL	NULL
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	PMID27551786-Compound-III	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-52	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-10	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-141	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-162	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 4	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 6	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 5	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 7	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 8	NULL	NULL	NULL	NULL	NULL
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	NULL	Pyridine derivative 19	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 19	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyridine derivative 19	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	Pyridine derivative 19	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 1	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 3	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 14	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	Indolizine derivative 1	NULL	NULL	NULL	NULL	NULL
PLATELET-ACTIVATING FACTOR ACETYLHYDROLASE	hgnc:9040	PLA2G7	TTD	2020.06.01	NULL	NULL	Indolizine derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Benzamide derivative 12	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Benzamide derivative 13	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl amide derivative 1	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-4	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkynyl-substituted pyrimidinyl-pyrrole derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE LYN	hgnc:6735	LYN	TTD	2020.06.01	NULL	NULL	Alkynyl-substituted pyrimidinyl-pyrrole derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyanomethyl pypazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyanomethyl pypazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloalkyl nitrile pyrazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloalkyl nitrile pyrazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Five-and-six-membered heterocyclic compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Five-and-six-membered heterocyclic compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Five-and-six-membered heterocyclic compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Geminally-substituted cyanoethylpypazolo pyridone derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Geminally-substituted cyanoethylpypazolo pyridone derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Geminally-substituted cyanoethylpypazolo pyridone derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Geminally-substituted cyanoethylpypazolo pyridone derivative 2	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure2Example4-3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure6Example3	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure9Example15	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 5	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Tricyclic heterocycle derivative 5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolopyridine compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolopyridine compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolopyridine compound 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Tricyclic pyrrolopyridine compound 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Tricyclic compound 2	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3H)-one derivative 2	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3H)-one derivative 3	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Indandione derivative 1	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Indandione derivative 2	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Indandione derivative 3	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Oxazolo[3,4-a]pyrazine derivative 6	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-5a	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-5b	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-6	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-6c	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoline derivative 14	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TDZD-8	iuphar.ligand:5977	GSK-3BETA INHIBITOR I	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 5	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	3-phenyl isoquinolin-1(2H) derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	4-Carboxamido-isoindolinone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	4-Carboxamido-isoindolinone derivative 3	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 8	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Dihydrodiazepinocarbazolone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 2	hgnc:272	PARP2	TTD	2020.06.01	NULL	NULL	Dihydrodiazepinocarbazolone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Phthalazine derivative 3	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Phthalazine ketone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-33	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-36	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Tetra/penta-cyclic pyridophthalazinone derivative 1	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 2	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 9	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine-dihydropyridine hybrid derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine-indole hybrid derivative 3	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	4-aryl quinol derivative 3	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	4-aryl quinol derivative 5	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Acyl oxymethyl acrylamide ester derivative 1	NULL	NULL	NULL	NULL	NULL
GLUTATHIONE REDUCTASE	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	Acyl oxymethyl acrylamide ester derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Benzisoselenazolone difluorocytidine derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Binuclear gold(I) compound 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Binuclear gold(I) compound 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Disulfide compound 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-19	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-28	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-31	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl carboxamide analog 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Diazepinone derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Ethynyl compound 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Ethynyl compound 6	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Heterocyclic derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Imidazopyridine and triazolopyridine compound 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 5	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 6	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-pyrazolopyrazine derivative 3	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 10	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 8	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 12	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 9	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20100022547C80	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20100022547C81	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20100022547C82	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20120264760C82	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20120264760C83	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20128202889C90	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20158969342C84	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20169447134C85	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 13	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 15	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 2	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 4	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	Diaryl amine derivative 4	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32d	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32d	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32g	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32g	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32m	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32m	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32p	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32p	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32q	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32q	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32r	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32r	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32v	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32v	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32y	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32y	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Hydrazide derivative 3	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Hydrazide derivative 5	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Oxindole derivative 3	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2 G2019S MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxindole derivative 3	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	PMID28117607-Compound-20	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyridopyrimidinone derivative 2	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 11	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 9	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 2	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-33	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-37	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-41	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-44	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-49	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-54	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-Figure3bII	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Complex heterocyclic compound 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydropyrido pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaromatic ring derivative 1	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaromatic ring derivative 4	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine derivative 8	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-10	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-14	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DLG] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-phenyl-1,3,4-triazole derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	1-phenyl-1,3,4-triazole derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	4-(2-cyclohexylethoxy) aniline derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazole derivative 4	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chalcone derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Chalcone derivative 3	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chalcone derivative 4	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Chalcone derivative 4	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-13	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-13	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-32	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-32	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-33	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-33	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-49	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-49	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-94	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 2	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 4	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Pyrazino[2,1-a]isoquinolin derivative 4	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	NULL	PMID28460551-Compound-1	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	Azetidine derivative 2	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	Benzoheterocyclic compound 1	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	PMID28594589-Compound-TABLE3C14	NULL	NULL	NULL	NULL	NULL
MICROTUBULE-ASSOCIATED PROTEIN TAU PHOSPHORYLATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme22Middle	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme24Paprotrain	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme25-4	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme25-4	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme27LeucettineL41	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme27LeucettineL41derivatives	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme4Bottom	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme4Bottom	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme7WO2012/098070bottom	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme7WO2012/098070bottom	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT6840	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT6840	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-40	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-43	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-45	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-47	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-48	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-50	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-62	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-69	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	PMID28906174-Compound-figure1g	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	PMID28906174-Compound-figure1g	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Pyrrolidine derivative 11	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Triazole derivative 4	NULL	NULL	NULL	NULL	NULL
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	NULL	Triazole derivative 7	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidinyl-piperazine derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 17	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 17	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamide derivative 24	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamide derivative 24	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamide derivative 25	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamide derivative 25	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamide derivative 26	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamide derivative 26	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-11d	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-11d	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-11d	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-17	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-7d	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-7f	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 80	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 80	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 80	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 81	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 81	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 81	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-41	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-47	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-50	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-54	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-70	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Pyrrolo[1,2-c]pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 6	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 7	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-19	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-22	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-29	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-38	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-5	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-9	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-24	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-24	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 10	hgnc:18128	HDAC10	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 11	hgnc:19086	HDAC11	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 5	hgnc:14068	HDAC5	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 9	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-25	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 10	hgnc:18128	HDAC10	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 11	hgnc:19086	HDAC11	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 5	hgnc:14068	HDAC5	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 9	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-43	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-47a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-53	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-61	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-61	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-61	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-61	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-61	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-61	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-68b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-68b	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-62	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-8	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-8	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imatinib and nilotinib derivative 1	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imatinib and nilotinib derivative 2	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30074415-Compound-21	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	1,2,4-oxadiazole derivative 2	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	1,3,4-oxadiazole derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3,4-oxadiazole derivative 3	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,3,4-oxadiazole derivative 6	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	3-substituted-1,2,4-oxadiazole derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	3-substituted-1,2,4-oxadiazole derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzyl phenyl ether derivative 2	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl compound 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl compound 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bromo benzyl ether derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bromo benzyl ether derivative 2	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example41	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example45	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example46	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example49	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example57	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example58	NULL	NULL	NULL	NULL	NULL
5-HT 1 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 15	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 15	NULL	NULL	NULL	NULL	NULL
5-HT 1 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 16	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 16	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 6	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 6	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 6	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 6	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-13TABLE4	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-13TABLE4	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-13TABLE4	NULL	NULL	NULL	NULL	NULL
5-HT 7 RECEPTOR	hgnc:5302	HTR7	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-13TABLE4	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-13TABLE4	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-34TABLE4	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-34TABLE4	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-34TABLE4	NULL	NULL	NULL	NULL	NULL
5-HT 7 RECEPTOR	hgnc:5302	HTR7	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-34TABLE4	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-34TABLE4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Aryl azepine derivative 2	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Benzamide derivative 10	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 10	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Benzamide derivative 11	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 11	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Fused aryl carbocycle derivative 3	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Fused aryl carbocycle derivative 4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Fused aryl carbocycle derivative 8	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 5	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 5	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 5	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-63	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID30259754-Compound-INT-767	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-37	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-38	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2008009652	NULL	NULL	NULL	NULL	NULL
CATHELICIDIN ANTIMICROBIAL PEPTIDE	hgnc:1472	CAMP	TTD	2020.06.01	NULL	NULL	Colforsin daropate hci	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.8140724222588294	Clenbuterol	rxcui:2580	CLENBUTEROL	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Erythromycin	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
BACTERIAL FATTY ACID SYNTHETASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ethionamide	rxcui:4127	ETHIONAMIDE	TRUE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	2.812910959055062	Epoprostenol	rxcui:8814	EPOPROSTENOL	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.2822993077187876	Fexofenadine	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Incruse Ellipta	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lestaurtinib	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Leucovorin/5-fluorouracil	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.032769506	Lisuride	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	Lmw heparin	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	Loxoprofen gel	NULL	NULL	NULL	NULL	NULL
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Luliconazole	rxcui:1482680	LULICONAZOLE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Meglitinides	NULL	NULL	NULL	NULL	NULL
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mianserin	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.059297201	Metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxybutynin hydrochloride	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Paromomycin	rxcui:66912	PAROMOMYCIN SULFATE	TRUE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Perospirone	ncit:C66358	PEROSPIRONE	FALSE	FALSE	FALSE
ANGIOGENESIS/MYELOMA CELL GROWTH	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pomalidomide	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Premarin/Trimegestone	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Pramiracetam	ncit:C84171	PRAMIRACETAM	FALSE	FALSE	FALSE
PEDICULUS HUMANUS NICOTINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Spinosad	rxcui:299081	SPINOSAD	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	SR141716A	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS LEUCYL-TRNA SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tavaborole	rxcui:1543173	TAVABOROLE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1193356164447602	Sertraline	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	NULL	AIKO-150	NULL	NULL	NULL	NULL	NULL
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	NULL	ALO-1567	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR-LIKE PROTEIN 7	hgnc:20594	EGFL7	TTD	2020.06.01	NULL	NULL	Anti-EGFL7	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	ATI-9242	NULL	NULL	NULL	NULL	NULL
GHR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATL1103	chembl:CHEMBL3989982	ATESIDORSEN	FALSE	FALSE	FALSE
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	1.312691780892362	ALRN-6924	ncit:C118669	SULANEMADLIN	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.1000146118775133	Altiratinib	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	CAR.CD30 cells	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting MucI	NULL	NULL	NULL	NULL	NULL
EPHRIN TYPE-A RECEPTOR 2	hgnc:3386	EPHA2	TTD	2020.06.01	NULL	NULL	DS-8895	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	ELOMOTECAN HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	NULL	F-15845	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	DRF-1042	drugbank:DB17152	DRF-1042	FALSE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	3.621218705909965	CDP-7657	ncit:C174737	DAPIROLIZUMAB PEGOL	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	IC9-CAR19 cells	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	IMC-EB10	chembl:CHEMBL2109328	IMC-EB10	FALSE	FALSE	FALSE
INTEGRIN ALPHA-5	hgnc:6141	ITGA5	TTD	2020.06.01	NULL	NULL	JSM 6427	NULL	NULL	NULL	NULL	NULL
INTEGRIN BETA-1	hgnc:6153	ITGB1	TTD	2020.06.01	NULL	NULL	JSM 6427	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	M1 agonist	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	IM19	ncit:C155888	AUTOLOGOUS ANTI-CD19 CAR T-CELLS IM19	FALSE	FALSE	FALSE
FK506-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Timcodar dimesilate	ncit:C2443	TIMCODAR DIMESYLATE	FALSE	FALSE	FALSE
WISKOTT-ALDRICH SYNDROME PROTEIN	hgnc:12731	WAS	TTD	2020.06.01	NULL	NULL	WASP gene therapy	NULL	NULL	NULL	NULL	NULL
ICAM1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alicaforsen	ncit:C169771	ALICAFORSEN	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.801643836	CORT-125134	ncit:C127838	RELACORILANT	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	6.300920548	Ulocuplumab	ncit:C95755	ULOCUPLUMAB	FALSE	FALSE	FALSE
SYK MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASN002	ncit:C166736	GUSACITINIB	FALSE	FALSE	FALSE
TNF-RELATED WEAK INDUCER OF APOPTOSIS	hgnc:11927	TNFSF12	TTD	2020.06.01	NULL	NULL	BIIB 023	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	BIM23A760	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gallopamil	rxcui:4648	GALLOPAMIL	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.2302968036653267	Ertumaxomab	ncit:C2658	ERTUMAXOMAB	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	0.7001022831425933	Ertumaxomab	ncit:C2658	ERTUMAXOMAB	FALSE	FALSE	FALSE
SUPEROXIDE DISMUTASE MN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imisopasem manganese	ncit:C111684	IMISOPASEM MANGANESE	FALSE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	JKB-122	NULL	NULL	NULL	NULL	NULL
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	VOFOPITANT HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
NEUROMEDIN-K RECEPTOR	hgnc:11528	TACR3	TTD	2020.06.01	NULL	5.834185692854944	Talnetant	ncit:C76464	TALNETANT	FALSE	FALSE	FALSE
T-CELL ACTIVATION ANTIGEN CD27	hgnc:11922	CD27	TTD	2020.06.01	NULL	15.00219178	Varlilumab	ncit:C99127	VARLILUMAB	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	ZK-91587	NULL	NULL	NULL	NULL	NULL
S100 CALCIUM-BINDING PROTEIN B	hgnc:10500	S100B	TTD	2020.06.01	NULL	NULL	ONO-2506	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	AVP-786	NULL	NULL	NULL	NULL	NULL
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	7.876150685354174	Hematide	rxcui:1248798	PEGINESATIDE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Recombinant acidic fibroblast growth factor	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	SaxaDapa FDC	NULL	NULL	NULL	NULL	NULL
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	NULL	SaxaDapa FDC	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19-CAR vector-transduced T cells	NULL	NULL	NULL	NULL	NULL
PRESYNAPTIC DENSITY PROTEIN 95	hgnc:2903	DLG4	TTD	2020.06.01	NULL	17.50255707856483	Tat-NR2B9c	ncit:C170212	NERINETIDE	FALSE	FALSE	FALSE
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	8.751278539282417	SB-742457	ncit:C166572	INTEPIRDINE	FALSE	FALSE	FALSE
SECRETORY PHOSPHOLIPASE A2	hgnc:9031	PLA2G2A	TTD	2020.06.01	NULL	2.917092846427472	Varespladib methyl	ncit:C152833	VARESPLADIB METHYL	FALSE	FALSE	FALSE
CI MAN-6-P RECEPTOR	hgnc:5467	IGF2R	TTD	2020.06.01	NULL	NULL	EP-128504	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PHENSERINE TARTRATE	NULL	NULL	NULL	NULL	NULL
NEUROMEDIN-K RECEPTOR	hgnc:11528	TACR3	TTD	2020.06.01	NULL	NULL	SB222200	NULL	NULL	NULL	NULL	NULL
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	NULL	ZK-thiazolidinone	NULL	NULL	NULL	NULL	NULL
NCBIGENE:1388	hgnc:2349	ATF6B	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10263	iuphar.ligand:10263	ML351	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.06466462	IUPHAR.LIGAND:62	iuphar.ligand:62	(+)-BUTACLAMOL	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:70	iuphar.ligand:70	GR 218,231	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.090530468	IUPHAR.LIGAND:71	iuphar.ligand:71	MPDT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.090530468	IUPHAR.LIGAND:167	iuphar.ligand:167	S 16924	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.050294704	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.056581542	IUPHAR.LIGAND:73	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.005955952	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.045265234	IUPHAR.LIGAND:60	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.026626608	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:74	iuphar.ligand:74	REC 15/3079	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.018860514	IUPHAR.LIGAND:63	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.027177884	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.078136416	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:144	drugbank:DB01445	BUFOTENINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.008224886	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:7227	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.276356164	IUPHAR.LIGAND:208	iuphar.ligand:208	NORFLUOXETINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.042898424	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.048260727	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.032173818	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:229	iuphar.ligand:229	WAY-163909	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.080905503	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.1779921058837101	IUPHAR.LIGAND:71	iuphar.ligand:71	MPDT	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:101	ncit:C73303	TIOSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.024896952	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.037775303	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.3777530304726222	IUPHAR.LIGAND:5699	drugbank:DB02567	PD173955	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1162317016838838	IUPHAR.LIGAND:7731	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1259176768242074	IUPHAR.LIGAND:12383	iuphar.ligand:12383	RISVODETINIB	FALSE	FALSE	FALSE
NCBIGENE:3068	hgnc:4856	HDGF	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10216	iuphar.ligand:10216	KH7	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	modulator	0.9211872146613068	IUPHAR.LIGAND:7945	iuphar.ligand:7945	MK-2206	FALSE	FALSE	FALSE
NCBIGENE:1678	hgnc:11817	TIMM8A	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12778	ncit:C175739	ALDUMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1673	hgnc:2767	DEFB4A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8680	iuphar.ligand:8680	IK-862	FALSE	FALSE	FALSE
NCBIGENE:874	hgnc:1549	CBR3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:4501	iuphar.ligand:4501	BENZYLCYSTEINE	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:502	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	0.090843722	IUPHAR.LIGAND:2714	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6560	iuphar.ligand:6560	5-CL-5-DEOXY-(&PLUSMN;)-ENBA	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:382	iuphar.ligand:382	AS70	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:8419	iuphar.ligand:8419	WRC-0571	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:5607	iuphar.ligand:5607	LUF5981	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:431	iuphar.ligand:403	SCH 58261	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1804387327687096	IUPHAR.LIGAND:5622	iuphar.ligand:5622	MRS5151	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:5607	iuphar.ligand:5607	LUF5981	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	modulator	0.5413161983061289	IUPHAR.LIGAND:9447	iuphar.ligand:9447	LUF6096	FALSE	FALSE	FALSE
NCBIGENE:3245	hgnc:115	ACLY	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12854	iuphar.ligand:12854	NDI-091143	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6917	iuphar.ligand:6917	5-BUTYL-METHYL IMMIDAZOLE CARBOXYLATE 30	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12319	iuphar.ligand:12319	LARTESERTIB	FALSE	FALSE	FALSE
NCBIGENE:2594	hgnc:59	ABCC8	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:6801	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:9388	iuphar.ligand:9388	GSK143	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:8358	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.019980088	IUPHAR.LIGAND:5718	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:615	iuphar.ligand:615	[PHE13]BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8502	iuphar.ligand:8502	MK-7725	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:567	iuphar.ligand:567	BRL 37344	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.5645986154375752	IUPHAR.LIGAND:569	rxcui:20192	CARAZOLOL	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.4234489615781814	IUPHAR.LIGAND:9512	ncit:C96754	SOLABEGRON	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:568	ncit:C77932	AMIBEGRON	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:552	iuphar.ligand:552	CICLOPROLOL	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:9176	iuphar.ligand:9176	WZ4002	FALSE	FALSE	TRUE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6154	iuphar.ligand:6154	BIIL 260	FALSE	FALSE	FALSE
NCBIGENE:2724	ncbigene:2724	GLC1D	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9524	iuphar.ligand:9524	BAY-299	FALSE	FALSE	FALSE
NCBIGENE:2722	ncbigene:2722	GLC1B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8571	iuphar.ligand:8571	BAZ2-ICR	FALSE	FALSE	FALSE
NCBIGENE:2730	hgnc:4312	GCLM	GuideToPharmacology	2024.1	NULL	1.346350544504987	IUPHAR.LIGAND:8573	iuphar.ligand:8573	NI-57	FALSE	FALSE	FALSE
NCBIGENE:3055	hgnc:4840	HCK	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:10433	iuphar.ligand:10433	COMPOUND 5A [PMID: 31287314]	FALSE	FALSE	FALSE
NCBIGENE:3092	hgnc:4913	HIP1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:10433	iuphar.ligand:10433	COMPOUND 5A [PMID: 31287314]	FALSE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	1.050153425	IUPHAR.LIGAND:12648	ncit:C174710	SUVECALTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.4884434533552977	IUPHAR.LIGAND:12648	ncit:C174710	SUVECALTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.03591496	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:388	hgnc:668	RHOB	GuideToPharmacology	2024.1	activator	0.2917092846427472	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:9237	iuphar.ligand:9237	GAT100	FALSE	FALSE	FALSE
NCBIGENE:391	hgnc:672	RHOG	GuideToPharmacology	2024.1	activator	0.4375639269641209	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	modulator	1.009762908	IUPHAR.LIGAND:10273	iuphar.ligand:10273	COMPOUND C2 [PMID: 29990428]	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:877	iuphar.ligand:877	JNJ-17156516	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:890	ncit:C66017	LINTITRIPT	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:751	iuphar.ligand:751	SR144528	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:773	iuphar.ligand:773	HIV-TAT	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:762	iuphar.ligand:762	[125I]CCL2 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:774	iuphar.ligand:774	VCCL4	FALSE	FALSE	FALSE
NCBIGENE:63	hgnc:136	ACTBP3	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:809	iuphar.ligand:809	CCL20-SEAP(HIS)6	FALSE	FALSE	FALSE
NCBIGENE:65	ncbigene:65	ACTBP5	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:812	iuphar.ligand:812	CCL1	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:768	iuphar.ligand:768	VMIP-II	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:807	ncit:C73589	VICRIVIROC	FALSE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:12229	iuphar.ligand:12229	ZWB67	FALSE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:8162	iuphar.ligand:8162	ML315	FALSE	FALSE	FALSE
NCBIGENE:1993	hgnc:3313	ELAVL2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12975	iuphar.ligand:12975	MW05	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:8159	iuphar.ligand:8159	COMPOUND 25 [PMID: 20855207]	FALSE	FALSE	FALSE
NCBIGENE:698	ncbigene:698	BTS1	GuideToPharmacology	2024.1	blocker	7.501095891	IUPHAR.LIGAND:4098	iuphar.ligand:4098	S-(-)CPP	FALSE	FALSE	FALSE
NCBIGENE:702	hgnc:2021	CLCN3	GuideToPharmacology	2024.1	blocker	2.625383561784725	IUPHAR.LIGAND:4285	drugbank:DB07810	PHLORETIN	FALSE	FALSE	FALSE
NCBIGENE:700	hgnc:1153	BVR1	GuideToPharmacology	2024.1	blocker	3.500511415712967	IUPHAR.LIGAND:4177	iuphar.ligand:4177	DIDS	FALSE	FALSE	FALSE
NCBIGENE:1255	ncbigene:1255	CNA1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9258	iuphar.ligand:9258	BIIB021	FALSE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:6388	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:6385	rxcui:15202	ARGATROBAN	TRUE	FALSE	FALSE
NCBIGENE:2364	hgnc:3872	FRA1E	GuideToPharmacology	2024.1	antibody	6.563458904461812	IUPHAR.LIGAND:9744	rxcui:1989794	EMICIZUMAB	TRUE	FALSE	FALSE
NCBIGENE:1255	ncbigene:1255	CNA1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9529	iuphar.ligand:9529	MS049	FALSE	FALSE	FALSE
NCBIGENE:1255	ncbigene:1255	CNA1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7031	iuphar.ligand:7031	COMPOUND 17F [PMID: 19632837]	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	antibody	0.9907107780319716	IUPHAR.LIGAND:8944	iuphar.ligand:8944	EMACTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.010952789	IUPHAR.LIGAND:4139	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:607	hgnc:1008	BCL9	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:2759	iuphar.ligand:2759	5&BETA;-PREGNANE-3,20-DIONE	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:917	iuphar.ligand:917	[125I]UROCORTIN 1 (MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:3890	iuphar.ligand:3890	K31440	FALSE	FALSE	FALSE
NCBIGENE:1840	hgnc:3060	DTX1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:12392	iuphar.ligand:12392	ZIDESAMTINIB	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:810	iuphar.ligand:810	CCL19	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:820	iuphar.ligand:820	CXCL6	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.068637479	IUPHAR.LIGAND:5670	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.2333674277141978	IUPHAR.LIGAND:11885	iuphar.ligand:11885	TANUXICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:6310	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:3230	hgnc:5131	HOXD@	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12658	iuphar.ligand:12658	ART812	FALSE	FALSE	FALSE
NCBIGENE:2650	hgnc:4203	GCNT1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9205	iuphar.ligand:9205	COMPOUND 13 [CHEN ET AL., 2016]	FALSE	FALSE	FALSE
NCBIGENE:2650	hgnc:4203	GCNT1	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7020	iuphar.ligand:7020	SGC0946	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:1898	iuphar.ligand:1898	S-5751	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.061197752	IUPHAR.LIGAND:204	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.070860555	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	modulator	0.3500511415712966	IUPHAR.LIGAND:7694	iuphar.ligand:7694	SB269652	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.050007306	IUPHAR.LIGAND:960	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.2333674277141977	IUPHAR.LIGAND:7556	ncit:C66358	PEROSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.011799477	IUPHAR.LIGAND:11976	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.058997383	IUPHAR.LIGAND:952	iuphar.ligand:3298	[3H]PD128907	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.007866318	IUPHAR.LIGAND:948	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.081533651	IUPHAR.LIGAND:960	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:988	iuphar.ligand:988	BETA-ERGOCRIPTINE	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:7001	iuphar.ligand:7001	GARCINOL	FALSE	FALSE	FALSE
NCBIGENE:2888	hgnc:4565	GRB14	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:12103	ncit:C171450	PERENOSTOBART	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.333674277141978	IUPHAR.LIGAND:7012	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:5965	iuphar.ligand:5965	EGFR/ERBB-2/ERBB-4 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:10194	iuphar.ligand:10194	COMPOUND 6G [PMID: 30633509]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.004951218	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:7966	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1890	iuphar.ligand:1890	ZK118182	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:3360	iuphar.ligand:3360	GW848687X	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.3241214273808302	IUPHAR.LIGAND:1913	iuphar.ligand:1913	MB-28767	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.1422972120208523	IUPHAR.LIGAND:5820	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.064033745	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.2651902587661338	IUPHAR.LIGAND:5820	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:1924	iuphar.ligand:1924	SC-51322	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:9845	iuphar.ligand:9845	CR6086	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.2344092465879218	IUPHAR.LIGAND:5675	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.2344092465879218	IUPHAR.LIGAND:7717	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:1929	ncit:C83707	EVATANEPAG	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:9176	iuphar.ligand:9176	WZ4002	FALSE	FALSE	TRUE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:5965	iuphar.ligand:5965	EGFR/ERBB-2/ERBB-4 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.056826484	IUPHAR.LIGAND:2818	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:2817	drugbank:DB04468	AFIMOXIFENE	FALSE	FALSE	FALSE
NCBIGENE:2652	hgnc:4206	OPN1MW	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8389	iuphar.ligand:8389	UNC0321	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:3886	ncit:C74027	SOVATELTIDE	FALSE	FALSE	FALSE
NCBIGENE:2651	hgnc:4204	GCNT2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8238	iuphar.ligand:8238	A-366	FALSE	FALSE	FALSE
NCBIGENE:2016	hgnc:3340	EMX1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:5988	iuphar.ligand:5988	INDIRUBIN DERIVATIVE E804	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:12910	iuphar.ligand:12910	HPG1860	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4299	iuphar.ligand:4299	RO4938581	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	blocker	0.2302968036653267	IUPHAR.LIGAND:4369	iuphar.ligand:4369	[35S]TBPS	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.1315981735230438	IUPHAR.LIGAND:4108	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.09869863	IUPHAR.LIGAND:10773	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4179	iuphar.ligand:4179	DMCM	FALSE	FALSE	FALSE
NCBIGENE:412	hgnc:11425	STS	GuideToPharmacology	2024.1	modulator	3.500511415712966	IUPHAR.LIGAND:7336	ncit:C72768	ETAZOLATE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:4107	iuphar.ligand:4107	5-ME-IAA	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6129	iuphar.ligand:6129	GALANIN	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6090	iuphar.ligand:6090	GALANIN(2-30) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:5391	iuphar.ligand:5391	[125I][TYR26]GALANIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:3899	iuphar.ligand:3899	M40	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6107	iuphar.ligand:6107	GAL-B5	FALSE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:6513	iuphar.ligand:6513	(S)-EF-1520	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3052	drugbank:DB07841	GERANYLGERANYL DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:4251	iuphar.ligand:4251	LY503430	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.4688184931758437	IUPHAR.LIGAND:4166	iuphar.ligand:4166	CX546	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.6563458904461812	IUPHAR.LIGAND:4249	iuphar.ligand:4249	LY404187	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:13017	drugbank:DB12280	AZD-5423	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:4140	iuphar.ligand:4140	ATPA	FALSE	FALSE	FALSE
NCBIGENE:2978	hgnc:4678	GUCA1A	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:10697	iuphar.ligand:10697	NCGC607	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.05309168	IUPHAR.LIGAND:2867	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
NCBIGENE:2798	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	activator	0.3977853881492007	IUPHAR.LIGAND:7701	iuphar.ligand:7701	AZD1656	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1521961485092594	IUPHAR.LIGAND:4082	iuphar.ligand:4082	[3H]CPP	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.1521961485092594	IUPHAR.LIGAND:4068	iuphar.ligand:4068	(RS)-(TETRAZOL-5-YL)GLYCINE	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4154	iuphar.ligand:4154	CGP37849	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.09963505	IUPHAR.LIGAND:4233	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	modulator	0.6819178082557728	IUPHAR.LIGAND:731	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	modulator	0.5527123287967842	IUPHAR.LIGAND:4164	iuphar.ligand:4164	CU2+	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	modulator	0.3182283105193606	IUPHAR.LIGAND:4164	iuphar.ligand:4164	CU2+	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:731	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:5980	iuphar.ligand:5980	TWS119	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:5976	drugbank:DB08454	N-(5-METHYL-1H-PYRAZOL-3-YL)-2-PHENYLQUINAZOLIN-4-AMINE	FALSE	FALSE	FALSE
NCBIGENE:1707	hgnc:2435	CSF2RA	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:7785	iuphar.ligand:7785	MAVRILIMUMAB	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:12418	drugbank:DB02494	(S)-3-PHENYLLACTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5792	iuphar.ligand:5792	COMPOUND 1Q  [PMID: 18029181]	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:2933	iuphar.ligand:2933	3-HYDROXYOCTANOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2032	ncbigene:2032	ENUR2	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:8136	iuphar.ligand:8136	COMPOUND 2 [PMID: 15546730]	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:12609	iuphar.ligand:12609	COMPOUND 30 [PMID: 37057760]	FALSE	FALSE	FALSE
NCBIGENE:2615	hgnc:4161	LRRC32	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:9276	ncit:C152698	TOREFORANT	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1271	iuphar.ligand:1271	N-ETHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5755	iuphar.ligand:5755	COMPOUND 36J [PMID: 21536438]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5723	iuphar.ligand:5723	AS1907417	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5653	iuphar.ligand:5653	AR231453	FALSE	FALSE	FALSE
NCBIGENE:145	hgnc:276	PARP1P2	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:4064	iuphar.ligand:4064	LYSOPHOSPHATIDYLSERINE	FALSE	FALSE	FALSE
NCBIGENE:203	hgnc:361	AK1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:3639	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
NCBIGENE:123	hgnc:248	PLIN2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:10031	iuphar.ligand:10031	RTI-13951-33	FALSE	FALSE	FALSE
NCBIGENE:156	hgnc:289	GRK2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:10567	iuphar.ligand:10567	GPR15L	FALSE	FALSE	FALSE
NCBIGENE:2625	hgnc:4172	GATA3	GuideToPharmacology	2024.1	inhibitor	0.251232877	IUPHAR.LIGAND:6845	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
NCBIGENE:2453	hgnc:3850	FRA13A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12736	iuphar.ligand:12736	GSK3008348	FALSE	FALSE	FALSE
NCBIGENE:2443	hgnc:3841	FRA11F	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11486	drugbank:DB12732	FIRATEGRAST	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	inhibitor	0.1576806944014849	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.057574201	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:12464	iuphar.ligand:12464	THEAFLAVIN	FALSE	FALSE	FALSE
NCBIGENE:674	ncbigene:674	BRAFPS1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:412	iuphar.ligand:412	SAKURANETIN	FALSE	FALSE	FALSE
NCBIGENE:682	hgnc:1116	BSG	GuideToPharmacology	2024.1	inhibitor	0.5966780822238011	IUPHAR.LIGAND:4357	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.3088686543276147	IUPHAR.LIGAND:4285	drugbank:DB07810	PHLORETIN	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12470	iuphar.ligand:12470	CYCLAMATE	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:5432	rxcui:9509	SACCHARIN	TRUE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:12499	iuphar.ligand:12499	LACTUCOPICRIN	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	modulator	0.2917092846427472	IUPHAR.LIGAND:10432	rxcui:2612087	DEUCRAVACITINIB	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:11565	iuphar.ligand:11565	COMPOUND 13AC [PMID: 33256400]	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:11304	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:10549	iuphar.ligand:10549	COMPOUND 18E [PMID: 31670517]	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:6977	iuphar.ligand:6977	COMPOUND 19A [PMID: 24359159]	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.09869863	IUPHAR.LIGAND:12609	iuphar.ligand:12609	COMPOUND 30 [PMID: 37057760]	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:11613	ncit:C180657	ROPSACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2379	hgnc:3891	FRA2G	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11754	ncit:C175138	MILVEXIAN	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:7471	rxcui:1516803	ALVIMOPAN ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:968	hgnc:1693	CD68	GuideToPharmacology	2024.1	inhibitor	0.9723642821424908	IUPHAR.LIGAND:4837	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	antibody	0.034590034	IUPHAR.LIGAND:7390	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.2075402025126264	IUPHAR.LIGAND:8096	iuphar.ligand:8096	BIBF-1202	FALSE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:208	iuphar.ligand:208	NORFLUOXETINE	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	activator	0.375054795	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	modulator	1.640864726115453	IUPHAR.LIGAND:10447	iuphar.ligand:10447	LUF7244	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.2344092465879218	IUPHAR.LIGAND:7200	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.4102161815288632	IUPHAR.LIGAND:7167	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
NCBIGENE:573	hgnc:937	BAG1	GuideToPharmacology	2024.1	activator	5.834185692854944	IUPHAR.LIGAND:2308	iuphar.ligand:2308	NS1643	FALSE	FALSE	FALSE
NCBIGENE:546	hgnc:886	ATRX	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:2569	iuphar.ligand:2569	3-BICYCLO[2.2.1]HEPT-2-YL-BENZENE-1,2-DIOL	FALSE	FALSE	FALSE
NCBIGENE:552	hgnc:895	AVPR1A	GuideToPharmacology	2024.1	blocker	0.047561296	IUPHAR.LIGAND:2416	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
NCBIGENE:547	hgnc:888	KIF1A	GuideToPharmacology	2024.1	blocker	0.182318303	IUPHAR.LIGAND:2416	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
NCBIGENE:545	hgnc:882	ATR	GuideToPharmacology	2024.1	blocker	0.036463661	IUPHAR.LIGAND:2416	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
NCBIGENE:1243	ncbigene:1243	CMM	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:5117	iuphar.ligand:5117	3-IODOTYROSINE	FALSE	FALSE	FALSE
NCBIGENE:2627	hgnc:4174	GATA6	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4842	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:3804	iuphar.ligand:3804	[125I]SHU9119	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1356787370431382	IUPHAR.LIGAND:8003	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:3136	hgnc:4965	HLA-H	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11133	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:10489	iuphar.ligand:10489	COMPOUND 12B [PMID: 31465220]	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:12248	iuphar.ligand:12248	D6808	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3049	iuphar.ligand:3049	DIMETHYLALLYL DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	NULL	0.6177373086552294	IUPHAR.LIGAND:8585	iuphar.ligand:8585	GE-137	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	0.5834185692854944	IUPHAR.LIGAND:6234	iuphar.ligand:6234	VU0364770	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6229	iuphar.ligand:6229	VU0092145	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1411	ncit:C169894	DEXFOSFOSERINE	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	modulator	2.500365296937833	IUPHAR.LIGAND:1441	iuphar.ligand:1441	AMN082	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.034590034	IUPHAR.LIGAND:5668	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:7815	ncit:C96531	DILMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:6059	iuphar.ligand:6059	VX-702	FALSE	FALSE	FALSE
NCBIGENE:2093	ncbigene:2093	ERVT3	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10183	iuphar.ligand:10183	BAY-885	FALSE	FALSE	FALSE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:2074	hgnc:3438	ERCC6	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9964	iuphar.ligand:9964	NIK SMI1	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:11083	iuphar.ligand:11083	COMPOUND 36 [PMID: 32429662]	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9481	iuphar.ligand:9481	JJKK 048	FALSE	FALSE	FALSE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6636	iuphar.ligand:6636	CLORGILINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.045898314	IUPHAR.LIGAND:355	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1360	iuphar.ligand:1360	S20928	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:7771	iuphar.ligand:7771	[125I]DIV880	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.1666910197958555	IUPHAR.LIGAND:1346	iuphar.ligand:1346	6-CL-MLT	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:1356	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.03394161	IUPHAR.LIGAND:1639	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.3547815624033412	IUPHAR.LIGAND:7551	rxcui:6465	LOFEPRAMINE	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.094608417	IUPHAR.LIGAND:201	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:3214	hgnc:5115	HOXB4	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:13013	iuphar.ligand:13013	COMPOUND 22 [PMID: 30457869]	FALSE	FALSE	FALSE
NCBIGENE:631	hgnc:1040	BFSP1	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:12997	iuphar.ligand:12997	COMPOUND 111 [PMID: 37918435]	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3997	iuphar.ligand:3997	PHA-709829	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2098	iuphar.ligand:2098	SUBSTANCE P	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:8869	iuphar.ligand:8869	SCH486757	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	0.3201687270469177	IUPHAR.LIGAND:8870	iuphar.ligand:8870	AT-076	FALSE	FALSE	FALSE
NCBIGENE:310	hgnc:545	ANXA7	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1568	iuphar.ligand:1568	JMV2004	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:4021	iuphar.ligand:4021	[3H]EYF	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9305	iuphar.ligand:9305	NAG 26	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:6169	iuphar.ligand:6169	5-OXO-20-HETE	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:6167	iuphar.ligand:6167	5-OXO-15-HETE	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1701	iuphar.ligand:1701	JNJ-10397049	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:9302	rxcui:2272403	LEMBOREXANT	TRUE	FALSE	FALSE
NCBIGENE:2136	hgnc:16059	PAK4	GuideToPharmacology	2024.1	inhibitor	0.2430910705356227	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	2.187819634820604	IUPHAR.LIGAND:9021	iuphar.ligand:9021	AZ10606120	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:9021	iuphar.ligand:9021	AZ10606120	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10502	iuphar.ligand:10502	COMPOUND 16I [PMID: 31525963]	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	0.2187819634820604	IUPHAR.LIGAND:6063	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	2.187819634820604	IUPHAR.LIGAND:4235	iuphar.ligand:4235	KN62	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641209	IUPHAR.LIGAND:2459	iuphar.ligand:2459	DECAVANADATE	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:1739	iuphar.ligand:1739	REACTIVE BLUE-2	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:10340	iuphar.ligand:10340	COMPOUND 58L [PMID: 30843696]	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:1716	iuphar.ligand:1716	2-CHLOROADENOSINE-5-TRIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1731	iuphar.ligand:1731	5BRUTP	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1749	drugbank:DB03435	URIDINE-5'-DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:3293	iuphar.ligand:3293	[ARG16]CHICKEN SECRETIN	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:4049	iuphar.ligand:4049	2-FUROYL-LIGRL[N[3H]PROPIONYL]-O-NH2	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:6660	iuphar.ligand:6660	[3H]2-FUROYL-LIGRL-NH2	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9458	iuphar.ligand:9458	YD-3	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.024041974	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:8012	iuphar.ligand:8012	PIK-75	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:9571	iuphar.ligand:9571	ECF309	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:8012	iuphar.ligand:8012	PIK-75	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:7963	iuphar.ligand:7963	PILARALISIB	FALSE	FALSE	FALSE
NCBIGENE:641	hgnc:1058	BLM	GuideToPharmacology	2024.1	inhibitor	0.5097832158805291	IUPHAR.LIGAND:3047	iuphar.ligand:3047	(R)-5-DIPHOSPHOMEVALONATE	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:8214	iuphar.ligand:8214	COMPOUND 14K [PMID: 21982499]	FALSE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.1495945049449985	IUPHAR.LIGAND:2399	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.010397559	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.009053047	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.1500219178162699	IUPHAR.LIGAND:8170	iuphar.ligand:8170	COMPOUND 8H [PMID: 21561767]	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.080781033	IUPHAR.LIGAND:7816	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
NCBIGENE:2388	hgnc:3900	FRA4A	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11539	iuphar.ligand:11539	SBC-115,337	FALSE	FALSE	FALSE
NCBIGENE:1259	hgnc:2148	CNGA1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9529	iuphar.ligand:9529	MS049	FALSE	FALSE	FALSE
NCBIGENE:1257	ncbigene:1257	CNC2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9529	iuphar.ligand:9529	MS049	FALSE	FALSE	FALSE
NCBIGENE:2408	hgnc:9545	PSMB8	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:9031	iuphar.ligand:9031	ONX-0914	FALSE	FALSE	FALSE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12477	iuphar.ligand:12477	CHLOROGENIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:10387	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12311	iuphar.ligand:12311	SZM679	FALSE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:13017	drugbank:DB12280	AZD-5423	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8725	iuphar.ligand:8725	CCG-63808	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.1630673019742065	IUPHAR.LIGAND:8170	iuphar.ligand:8170	COMPOUND 8H [PMID: 21561767]	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:2653	drugbank:DB07031	3-FLUORO-4-{[(2R)-2-HYDROXY-2-(5,5,8,8-TETRAMETHYL-5,6,7,8-TETRAHYDRO-2-NAPHTHALENYL)ACETYL]AMINO}BENZOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:8276	iuphar.ligand:8276	PALOVAROTENE	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:10318	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.095295229	IUPHAR.LIGAND:5181	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10425	iuphar.ligand:10425	ROCK INHIBITOR 3	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:12381	iuphar.ligand:12381	RESENCATINIB	FALSE	FALSE	FALSE
NCBIGENE:1527	hgnc:2563	TEX28	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9356	iuphar.ligand:9356	GSK429286A	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	activator	0.1312691780892362	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	inhibitor	0.1312691780892362	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	activator	0.1290114772375786	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:2000	iuphar.ligand:2000	INSL5	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:8326	iuphar.ligand:8326	MINIMISED RELAXIN-3 ANALOGUE 3	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:9491	iuphar.ligand:9491	AMISELIMOD PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10641	iuphar.ligand:10641	SLM6071469	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9388	iuphar.ligand:9388	GSK143	FALSE	FALSE	FALSE
NCBIGENE:1417	hgnc:2400	CRYBB3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:6703	iuphar.ligand:6703	KH064	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:2010	iuphar.ligand:2010	DES-ALA1,2,5-[D-TRP8,IAMP9]SRIF	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2058	iuphar.ligand:2058	[111IN,90Y]DOTA-OC	FALSE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10671	iuphar.ligand:10671	MC2050	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.1244257612220248	IUPHAR.LIGAND:8062	iuphar.ligand:8062	MRT67307	FALSE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10671	iuphar.ligand:10671	MC2050	FALSE	FALSE	FALSE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2636	iuphar.ligand:2636	RT3	FALSE	FALSE	FALSE
NCBIGENE:1722	hgnc:7217	MPL	GuideToPharmacology	2024.1	agonist	2.045753424767318	IUPHAR.LIGAND:9953	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
NCBIGENE:1754	hgnc:11850	TLR4	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5019	iuphar.ligand:5019	LPS	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1987	ncit:C81570	IFETROBAN	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1973	iuphar.ligand:1973	[125I]BOP	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1977	iuphar.ligand:1977	KW-3635	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:10279	iuphar.ligand:10279	GSK417651A	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:10286	iuphar.ligand:10286	HC-070	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.760980743	IUPHAR.LIGAND:4232	iuphar.ligand:4232	KB-R7943	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.760980743	IUPHAR.LIGAND:10283	iuphar.ligand:10283	SAR7334	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	0.069089041	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.7721716358190367	IUPHAR.LIGAND:10279	iuphar.ligand:10279	GSK417651A	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.1403948428761885	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:9968	iuphar.ligand:9968	SH045	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.5147810905460244	IUPHAR.LIGAND:9968	iuphar.ligand:9968	SH045	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.1325951293830669	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	1.875273972703375	IUPHAR.LIGAND:4114	iuphar.ligand:4114	9-PHENANTHROL	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	activator	0.046881849	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:4188	iuphar.ligand:4188	EPIPREGNANOLONE SULPHATE	FALSE	FALSE	FALSE
NCBIGENE:504	hgnc:828	ATP5F1AP2	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:2476	iuphar.ligand:2476	NI2+	FALSE	FALSE	FALSE
NCBIGENE:504	hgnc:828	ATP5F1AP2	GuideToPharmacology	2024.1	activator	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:502	hgnc:13357	MCOLN2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11862	iuphar.ligand:11862	PRU-12	FALSE	FALSE	FALSE
NCBIGENE:2887	hgnc:4564	GRB10	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9019	iuphar.ligand:9019	NAVOXIMOD	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	blocker	0.4773424657790409	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1209854175937661	IUPHAR.LIGAND:12609	iuphar.ligand:12609	COMPOUND 30 [PMID: 37057760]	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2791	rxcui:73710	PARICALCITOL	TRUE	FALSE	FALSE
NCBIGENE:1011	hgnc:1752	CDH12P2	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:4834	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2215	iuphar.ligand:2215	D(CH2)5[D-ILE2,ILE4,ALA-NH2]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.097236428	IUPHAR.LIGAND:2181	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:2831	hgnc:4522	NPBWR1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:11999	iuphar.ligand:11999	COMPOUND 41 [PMID: 35436124]	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2196	iuphar.ligand:2196	OPC-21268	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2238	ncit:C74429	LIXIVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1513	iuphar.ligand:1513	PANCREATIC POLYPEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:587	hgnc:977	BCAT2	GuideToPharmacology	2024.1	modulator	8.751278539282415	IUPHAR.LIGAND:12563	iuphar.ligand:12563	TTFB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	0.096123883	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	CIViC	10-Apr-24	NULL	0.007749066	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	AS602868	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	0.2108741816694558	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.4947116523181093	GILTERITINIB	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.9211872146613068	ANTI-PD-L1 MONOCLONAL ANTIBODY	ncit:C128057	ANTI-PD-L1 MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
APC	hgnc:583	APC	CIViC	10-Apr-24	NULL	NULL	JW55	NULL	NULL	NULL	NULL	NULL
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.3860858179095183	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.035083077	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	NULL	ERBB3 INHIBITOR	NULL	NULL	NULL	NULL	NULL
CTAG2	hgnc:2492	CTAG2	CIViC	10-Apr-24	NULL	26.25383561784724	LETETRESGENE AUTOLEUCEL	ncit:C121379	LETETRESGENE AUTOLEUCEL	FALSE	FALSE	TRUE
FGF19	hgnc:3675	FGF19	CIViC	10-Apr-24	NULL	26.25383561784724	FGFR4 INHIBITOR H3B-6527	ncit:C128862	FGFR4 INHIBITOR H3B-6527	FALSE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	CIViC	10-Apr-24	NULL	0.6806549974997433	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.2083637747448194	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
XRCC1	hgnc:12828	XRCC1	CIViC	10-Apr-24	NULL	0.1627303860610366	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	CIViC	10-Apr-24	NULL	0.058341857	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	XMU-MP-5	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.096123883	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1141471113819445	Onalespib	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	NVP-TNKS656	NULL	NULL	NULL	NULL	NULL
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	1.591141552596803	PLX2853	ncit:C146825	BRD4 INHIBITOR PLX2853	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.431569901	E7449	ncit:C102746	PARP/TANKYRASE INHIBITOR 2X-121	FALSE	FALSE	TRUE
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	0.1526385791735305	Bortezomib	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.03366236	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	CLM3	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.063440602	Saracatinib	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1099637093941246	RO4987655	ncit:C82696	MEK INHIBITOR RO4987655	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	LSN3074753	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	Sintilimab	ncit:C132992	SINTILIMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.1544343271638073	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6471533709721451	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.07330914	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.049418985	Eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	1.346350544504987	PF3644022	drugbank:DB07430	(10R)-10-METHYL-3-(6-METHYLPYRIDIN-3-YL)-9,10,11,12-TETRAHYDRO-8H-[1,4]DIAZEPINO[5',6':4,5]THIENO[3,2-F]QUINOLIN-8-ONE	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	1.009762908	PF-00477736	chembl:CHEMBL3545137	PF-00477736	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.2647445608522412	Anlotinib	ncit:C138997	ANLOTINIB	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	2.019525817	HMN-214	chembl:CHEMBL3545431	HMN-214	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	NULL	ZK 304709	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	Mps-BAY2b	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	NTRC 0066-0	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	NULL	G007-LK	NULL	NULL	NULL	NULL	NULL
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.251232877	Belinostat	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	1.141471113819445	HJC0152	iuphar.ligand:12140	HJC0152	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.4565884455277783	Milademetan	ncit:C141432	MILADEMETAN	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	AZ6089	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	ABSK061	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.2442217266776488	RO4987655	ncit:C82696	MEK INHIBITOR RO4987655	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1110098757625676	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	NULL	ABSK061	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	UNC2025	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.5527123287967841	TYRA-300	ncit:C190779	FGFR3 INHIBITOR TYRA-300	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	CG-806	ncit:C162573	LUXEPTINIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.056020987	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1579178082276526	PRN1371	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1842374429322613	Sintilimab	ncit:C132992	SINTILIMAB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2160809515872201	ONO-7475	chembl:CHEMBL4650414	ONO-7475	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	FTI-277	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	RM-018	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.035430277	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.3851418428046051	DS-1001b	chembl:CHEMBL4650282	DS-1001B	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.086361301	AZD8186	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.001584946	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	1.494525746746522	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.057073556	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	NULL	NIBR3049	NULL	NULL	NULL	NULL	NULL
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	NULL	MSU38225	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.03136659	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	N-Arachidonoyl Dopamine	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	RM-018	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	3144	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	LSN3074753	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.018699313	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	DHM25	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	SHR-A1307	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	T-2143	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	WEHI-539	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	PWT33597	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	STX-478	iuphar.ligand:12903	STX-478	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.069454592	Vistusertib	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	AT13148	ncit:C101786	MULTI-AGC KINASE INHIBITOR AT13148	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	PW12	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	OSU-T315	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	HG-6-63-01	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	SYHA1815	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.1375060601009582	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	NULL	Unspecified VEGFR inhibitor	NULL	NULL	NULL	NULL	NULL
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.067059606	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.4167275494896388	Hydroxyurea	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.008693323	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.025757994	Idelalisib	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.00799386	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	CEP-8983	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	CTX-1	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	unspecified EGFR antibody	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	Unspecified VEGFR inhibitor	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	AZ31	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.028977744	CG-806	ncit:C162573	LUXEPTINIB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.019318496	Methylprednisolone	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	CPUY201112	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.2318219480604613	Siremadlin	ncit:C116325	SIREMADLIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.012878997	Encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.057955487	PF-00477736	chembl:CHEMBL3545137	PF-00477736	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	AQ-101	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	SLMP53-2	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.010537361	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	binder	0.8334550989792777	DEPATUXIZUMAB MAFODOTIN	ncit:C105612	DEPATUXIZUMAB MAFODOTIN	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.039538909	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	DBPR-108	chembl:CHEMBL1082462	DBPR-108	FALSE	FALSE	FALSE
BIRC2	hgnc:590	BIRC2	DTC	9/2/20	NULL	1.875273972703375	AT-406	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.031612084	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.037884323	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	SJ000047240	chembl:CHEMBL590706	CHEMBL:CHEMBL590706	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ORSELLINIC ACID	chembl:CHEMBL457583	ORSELLINIC ACID	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.015193192	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	7.001022831425932	DSG	ncit:C1598	GUSPERIMUS TRIHYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	1.607377690888607	BETRIXABAN	rxcui:1927851	BETRIXABAN	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.2465148884304905	TIZANIDINE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.037363144	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:488	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:630	iuphar.ligand:630	COMPOUND 21B [PMID: 12723954]	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.070574827	IUPHAR.LIGAND:564	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	HARMALINE	drugbank:DB13875	HARMALINE	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.1640864726115453	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.33338204	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.025613498	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.3571950424196904	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
SYP	hgnc:11506	SYP	NCI	14-Sep-17	NULL	1.750255707856483	6-HYDROXYDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	BUNOLOL	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
UNIPROT:Q969P6	hgnc:29787	TOP1MT	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	PEG-SN38	ncit:C70651	FIRTECAN PEGOL	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:223	iuphar.ligand:223	[3H]RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:4209	iuphar.ligand:4209	GYKI53655	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:10034	iuphar.ligand:10034	IMB-808	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.025584378	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001701921	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.1086365611772989	CDDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.3621218705909965	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE	hgnc:4141	GAPDH	TTD	2020.06.01	NULL	1.346350544504987	Omigapil	ncit:C97362	OMIGAPIL	FALSE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.1172046232939609	Dihydrexidine	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
TISSUE FACTOR PATHWAY INHIBITOR	hgnc:11760	TFPI	TTD	2020.06.01	NULL	2.763561643983921	NN-7415	chembl:CHEMBL4297730	CONCIZUMAB	FALSE	FALSE	FALSE
D-AMINO ACID OXIDASE	hgnc:2671	DAO	TTD	2020.06.01	NULL	10.50153424713889	TAK-831	chembl:CHEMBL2338801	LUVADAXISTAT	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	1.009762908	LY3202626	iuphar.ligand:11557	LY3202626	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.031479419	IUPHAR.LIGAND:5386	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.067664525	IUPHAR.LIGAND:408	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	AMYLMETACRESOL	rxcui:236248	AMYLMETACRESOL	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.2430910705356226	ALBENDAZOLE	rxcui:430	ALBENDAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002159654	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.031851787	boceprevir	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	NAPHTHOQUINONE	chembl:CHEMBL55934	NAPHTHOQUINONE	FALSE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	0.2143170254518142	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
UNIPROT:P38435	hgnc:4247	GGCX	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	PHYTONADIONE	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TEND	1-Aug-11	NULL	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.046059361	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.064824285	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	MOLINATE	chembl:CHEMBL1865916	MOLINATE	FALSE	FALSE	FALSE
PROC	hgnc:9451	PROC	PharmGKB	4/5/24	NULL	1.750255707856483	lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
TBXA2R	hgnc:11608	TBXA2R	ChEMBL	33	inhibitor	1.875273972703375	TERUTROBAN	ncit:C90753	TERUTROBAN	FALSE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	21.00306849427779	METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA	rxcui:729596	METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	ChEMBL	33	inhibitor	2.692701089009974	TOPIROXOSTAT	ncit:C96311	TOPIROXOSTAT	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.056826484	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.1744440904840348	milnacipran	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.018081154	abrocitinib	rxcui:2591476	ABROCITINIB	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:768	iuphar.ligand:768	VMIP-II	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4326	iuphar.ligand:4326	TP003	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1411496538593938	IUPHAR.LIGAND:4240	iuphar.ligand:4240	L701324	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.029465584	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.010397559	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:7666	iuphar.ligand:7666	ML277	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:11221	ncit:C87279	CAPADENOSON	FALSE	FALSE	FALSE
POLRMT	hgnc:9200	POLRMT	DTC	9/2/20	NULL	105.0153424713889	2',2'-DIFLUORODEOXYCYTIDINE 5'-TRIPHOSPHATE	chembl:CHEMBL1201383	GEMCITABINE TRIPHOSPHATE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.010952789	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	DTC	9/2/20	NULL	0.1187956362798518	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
NCBIGENE:2605	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:11750	iuphar.ligand:11750	GSK3685032	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	COSMIC	4-Sep-20	NULL	0.5509279467829125	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.014622019	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	0.375054795	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
EGR2	hgnc:3239	EGR2	NCI	14-Sep-17	NULL	0.5770073762164231	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
HFE	hgnc:4886	HFE	PharmGKB	4/5/24	NULL	26.25383561784724	iron	rxcui:262150	IRON CARBONYL	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.1553481397505754	oxazepam	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O75343	hgnc:4686	GUCY1B2	TdgClinicalTrial	Jan-14	NULL	1.615620653405984	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	METHSCOPOLAMINE BROMIDE	rxcui:56092	METHSCOPOLAMINE BROMIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.077827576	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
EGLN3	hgnc:14661	EGLN3	ChEMBL	33	inhibitor	2.100306849	MOLIDUSTAT	rxcui:2637535	MOLIDUSTAT	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.009630901	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1426838892274307	2,4-DINITROPHENOL	drugbank:DB04528	2,4-DINITROPHENOL	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.5509279467829125	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
UPB1	hgnc:16297	UPB1	PharmGKB	4/5/24	NULL	0.9723642821424907	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.364636606	Tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
ATP2A1	hgnc:811	ATP2A1	ChEMBL	33	inhibitor	1.312691780892362	MIPSAGARGIN	ncit:C90554	MIPSAGARGIN	FALSE	FALSE	FALSE
RPS29	hgnc:10419	RPS29	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.00822231	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:602	iuphar.ligand:602	[125I]APELIN-13	FALSE	FALSE	FALSE
NCBIGENE:1295	hgnc:2215	COL8A1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:5270	iuphar.ligand:5270	SCH51866	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
CLCN3	hgnc:2021	CLCN3	DTC	9/2/20	NULL	13.12691780892362	CINOBUFAGIN	ncit:C95021	CINOBUFAGIN	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.2447910080918158	MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	ZARDAVERINE	ncit:C66686	ZARDAVERINE	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	4.200613699	GSK2578215A	chembl:CHEMBL2204495	CHEMBL:CHEMBL2204495	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.075333818	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:966	ncit:C65572	ETICLOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:7865	drugbank:DB06973	BISPHENOL A	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:92	rxcui:33739	PIPAMPERONE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.055271233	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
NDUFA9	hgnc:7693	NDUFA9	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.3125456621172291	E-6201	drugbank:DB11687	E-6201	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	1.071585127259071	IDRABIOTAPARINUX SODIUM	ncit:C170050	IDRABIOTAPARINUX SODIUM	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.05068308	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.036463661	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	7-NITROINDAZOLE	drugbank:DB02207	7-NITROINDAZOLE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.010777437	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
UNIPROT:P01375	hgnc:11892	TNF	TEND	1-Aug-11	NULL	0.3226277802500429	CERTOLIZUMAB PEGOL	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.1312691780892362	IUPHAR.LIGAND:2018	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
CCR5	hgnc:1606	CCR5	PharmGKB	4/5/24	NULL	0.7501095890813498	glatiramer acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
SLC10A1	hgnc:10905	SLC10A1	ChEMBL	33	inhibitor	8.751278539282415	HEPALATIDE	chembl:CHEMBL4650398	HEPALATIDE	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.082171629	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE ATR	hgnc:882	ATR	TTD	2020.06.01	NULL	0.9723642821424907	VE-822	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.3938075342677087	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PRF1	hgnc:9360	PRF1	FDA	10-Apr-24	NULL	4.375639269641208	Emapalumab-lzsg	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
RXRG	hgnc:10479	RXRG	ChEMBL	33	agonist	1.591141552596802	IRX-4204	chembl:CHEMBL75133	IRX-4204	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	2.500365296937833	IUPHAR.LIGAND:2329	iuphar.ligand:2329	CHARYBDOTOXIN-GLU32 ANALOG	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	5-FLUOROURIDINE	drugbank:DB01629	5-FLUOROURIDINE	FALSE	FALSE	FALSE
UNIPROT:Q99795	hgnc:4445	GPA33	TdgClinicalTrial	Jan-14	NULL	39.38075342677087	KRN-330	chembl:CHEMBL2109293	KRN-330	FALSE	FALSE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	1.312691780892362	P-1101	rxcui:2587059	ROPEGINTERFERON ALFA-2B	TRUE	FALSE	FALSE
PLCG1	hgnc:9065	PLCG1	DTC	9/2/20	NULL	0.3365876361262468	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.290901226	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
NCBIGENE:2421	hgnc:3931	FRA8C	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11533	iuphar.ligand:11533	MM3122	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.2800409132570373	HYPERBARIC OXYGEN	ncit:C2351	HYPERBARIC OXYGEN	FALSE	FALSE	FALSE
STAT5B	hgnc:11367	STAT5B	NCI	14-Sep-17	NULL	1.400204566285186	RECOMBINANT HUMAN GROWTH HORMONE	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.837888371	Oxyphenonium	rxcui:7818	OXYPHENONIUM	TRUE	FALSE	FALSE
MAPK4	hgnc:6878	MAPK4	PharmGKB	4/5/24	NULL	0.9211872146613069	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.3621218705909965	DEBIO 0932	ncit:C92572	HSP90 INHIBITOR DEBIO 0932	FALSE	FALSE	FALSE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:10559	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:12164	iuphar.ligand:12164	BI-4142	FALSE	FALSE	FALSE
NCBIGENE:547	hgnc:888	KIF1A	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7760	iuphar.ligand:7760	GXTX-1E	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:9101	iuphar.ligand:9101	BRIMAPITIDE	FALSE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	2.917092846427472	POTASSIUM OXYBATE	rxcui:2387309	POTASSIUM OXYBATE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.014891569	Guanidine Hydrochloride	rxcui:50676	GUANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	RACEPINEPHRINE	rxcui:66887	RACEPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:154	iuphar.ligand:154	(+)-LSD	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	QUINOSOL	chembl:CHEMBL451260	QUINOSOL	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	0.49187514	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.071928317	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008581087	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.014732792	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.003920824	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.075333818	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5112	iuphar.ligand:5112	2-OLEOYL GLYCEROL	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.4102161815288632	IUPHAR.LIGAND:2605	iuphar.ligand:2605	E4031	FALSE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	ChEMBL	33	blocker	0.1600843635234588	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
RPL36	hgnc:13631	RPL36	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	DAMNACANTHAL	ncit:C1480	DAMNACANTHAL	FALSE	FALSE	FALSE
E-SELECTIN	hgnc:10718	SELE	TTD	2020.06.01	NULL	1.591141552596802	GMI-1359	drugbank:DB18092	GMI-1359	FALSE	FALSE	FALSE
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	2.100306849	DUTOGLIPTIN	ncit:C87492	DUTOGLIPTIN	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	CARBINOXAMINE	rxcui:20220	CARBINOXAMINE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1442518440541058	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	0.8751278539282417	Interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	PharmGKB	4/5/24	NULL	0.023620185	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
B7 HOMOLOG 3	hgnc:19137	CD276	TTD	2020.06.01	NULL	10.50153424713889	Omburtamab I-131	drugbank:DB17124	OMBURTAMAB I-131	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	(R)-MELPHALAN	chembl:CHEMBL250892	(R)-MELPHALAN	FALSE	FALSE	FALSE
NCBIGENE:1822	hgnc:3033	ATN1	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8170	iuphar.ligand:8170	COMPOUND 8H [PMID: 21561767]	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:9610	iuphar.ligand:9610	CBS-3595	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.4817217544559128	SB-0304	chembl:CHEMBL409225	CHEMBL:CHEMBL409225	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.059667808	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.012504804	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.017520077	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	SJ000024939	chembl:CHEMBL590691	CHEMBL:CHEMBL590691	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	modulator	0.3804903712731485	IUPHAR.LIGAND:12050	iuphar.ligand:12050	SAGE-718	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	0.9376369863516875	Ethacrynic acid	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1888765152363111	IUPHAR.LIGAND:8147	iuphar.ligand:8147	COMPOUND 24 [PMID: 23441572]	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:2052	iuphar.ligand:2052	NC 8-12	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.054355767	Hydroxyurea	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.012932924	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	PharmGKB	4/5/24	NULL	0.049723174	levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2670	ncit:C98152	REGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:11304	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1019566431761058	CIRAZOLINE	ncit:C77294	CIRAZOLINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CYPRODINIL	chembl:CHEMBL521027	CYPRODINIL	FALSE	FALSE	FALSE
FCN2	hgnc:3624	FCN2	PharmGKB	4/5/24	NULL	2.019525816757481	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2702	iuphar.ligand:2701	AD5075	FALSE	FALSE	FALSE
NCBIGENE:414	hgnc:717	ARSD	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.8204323630577265	ADAGRASIB	rxcui:2625882	ADAGRASIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002646023	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
SLC9A3	hgnc:11073	SLC9A3	ChEMBL	33	inhibitor	13.12691780892362	TENAPANOR HYDROCHLORIDE	rxcui:2199673	TENAPANOR HYDROCHLORIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.012360563	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.009481342	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.061055432	IUPHAR.LIGAND:4798	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	blocker	6.563458904461812	IUPHAR.LIGAND:12547	iuphar.ligand:12547	SET2	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.3182283105193605	INDINAVIR SULFATE	rxcui:203153	INDINAVIR SULFATE	TRUE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.089756703	IUPHAR.LIGAND:8018	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NB-ACETYLTRYPTAMINE	chembl:CHEMBL33171	NB-ACETYLTRYPTAMINE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	PEG-CAMPTOTHECIN	chembl:CHEMBL3989476	PEGAMOTECAN	FALSE	FALSE	FALSE
NCBIGENE:932	hgnc:7317	MS4A3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6513	iuphar.ligand:6513	(S)-EF-1520	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	0.4039051633514962	IUPHAR.LIGAND:772	iuphar.ligand:772	CCL8	FALSE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:5672	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:304	iuphar.ligand:304	PENTYLTHIO-TZTP	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.044347695	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	SJ000120081	chembl:CHEMBL606532	CHEMBL:CHEMBL606532	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.089298761	DNDI1417413	chembl:CHEMBL1343568	CHEMBL:CHEMBL1343568	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.2226788432387383	MOMETASONE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TEND	1-Aug-11	NULL	0.1346350544504987	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:281	hgnc:479	AMYP1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:1304	iuphar.ligand:1304	ATC0065	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.056826484	IUPHAR.LIGAND:7965	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.084146909	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.008310806	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.085239726	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.068191781	Escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	0.4412409347537352	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2917092846427472	CYPRODINIL	chembl:CHEMBL521027	CYPRODINIL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	5-FLUOROURIDINE	drugbank:DB01629	5-FLUOROURIDINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009084372	SKF-82526	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	GBR-12935	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.3889457128569962	TCMDC-125322	chembl:CHEMBL580324	CHEMBL:CHEMBL580324	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.091796628	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.085239726	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:966	ncit:C65572	ETICLOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:2448	hgnc:6145	ITGA9	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12045	iuphar.ligand:12045	BOP	FALSE	FALSE	FALSE
CR2	hgnc:2336	CR2	NCI	14-Sep-17	NULL	0.4449802647092754	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:1678	hgnc:11817	TIMM8A	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8553	iuphar.ligand:8553	COMPOUND 15C [PMID: 21536437]	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	inhibitor	0.3125456621172291	APROTININ	rxcui:1056	APROTININ	TRUE	FALSE	FALSE
PSMC3	hgnc:9549	PSMC3	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.1356787370431382	DILEVALOL HYDROCHLORIDE	ncit:C174786	DILEVALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.1356787370431382	DILEVALOL HYDROCHLORIDE	ncit:C174786	DILEVALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
OPN1LW	hgnc:9936	OPN1LW	DTC	9/2/20	NULL	21.00306849427779	1,3-DIMETHYLCYCLOHEXANE	chembl:CHEMBL1952259	CHEMBL:CHEMBL1952259	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	OncoKB	23-Jul-20	NULL	0.3509871071904712	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.051885051	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
CYP7A1	hgnc:2651	CYP7A1	PharmGKB	4/5/24	NULL	0.729273212	cholic acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.050007306	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	activator	0.082043236	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.596678082	IUPHAR.LIGAND:6277	iuphar.ligand:6277	ACETALDEHYDE	FALSE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	DTC	9/2/20	NULL	1.093909817410302	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.1403948428761885	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	0.4884434533552977	IL-5	iuphar.ligand:4997	IL-5	FALSE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	NCI	14-Sep-17	NULL	0.1909369863116163	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
NCBIGENE:1467	hgnc:2471	CSRP2P1	GuideToPharmacology	2024.1	inhibitor	2.019525816757481	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	NCI-10777	chembl:CHEMBL189724	CHEMBL:CHEMBL189724	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.3241214273808303	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.007072693	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.040112812	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	DTC	9/2/20	NULL	3.750547945	BERKELEYACETAL C	chembl:CHEMBL400716	BERKELEYACETAL C	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DNDI1417447	chembl:CHEMBL1307453	CHEMBL:CHEMBL1307453	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	HYDROXYSTILBAMIDINE ISETHIONATE	ncit:C65871	HYDROXYSTILBAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	2-METHYL-5,7,8-TRIMETHOXYISOFLAVONE	chembl:CHEMBL1559418	2-METHYL-5,7,8-TRIMETHOXYISOFLAVONE	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.2778183663264259	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.064111931	rasagiline	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.3040984820600068	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
NCBIGENE:1880	hgnc:3128	GPR183	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:5065	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:10140	iuphar.ligand:10140	SPARTALIZUMAB	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.010199625	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003307362	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	TCMDC-125204	chembl:CHEMBL588028	CHEMBL:CHEMBL588028	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.009481342	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GLUTARAL	rxcui:4888	GLUTARAL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	CYCLOVALONE	ncit:C81040	CYCLOVALONE	FALSE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	DTC	9/2/20	inhibitor	0.1193356164447602	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
ALDH1L1	hgnc:3978	ALDH1L1	PharmGKB	4/5/24	NULL	10.50153425	l-methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
NDUFS5	hgnc:7712	NDUFS5	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:417	hgnc:723	ART1	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.039390601	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPL37A	hgnc:10348	RPL37A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
FFAR2	hgnc:4501	FFAR2	ChEMBL	33	inhibitor	26.25383561784724	GLPG-0974	drugbank:DB15406	GLPG-0974	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	ChEMBL	33	positive modulator	1.312691780892362	TOLIMIDONE	ncit:C152683	TOLIMIDONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	BENZYL ISOTHIOCYANATE	drugbank:DB16860	BENZYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PENCYCURON	chembl:CHEMBL2229452	PENCYCURON	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1643432589536604	CHEMOPREVENTIVE	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.010718039	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00202529	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
FK506-BINDING PROTEIN 1A	hgnc:3711	FKBP1A	TTD	2020.06.01	NULL	0.5373592085524291	Rapamycin	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	0.7955707762984013	TG003	iuphar.ligand:5942	CDC2-LIKE KINASE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:998	iuphar.ligand:998	FR139317	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.056097939	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.5834185692854945	PRALICIGUAT	ncit:C174906	PRALICIGUAT	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	ChEMBL	33	inhibitor	0.021608095	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1992	iuphar.ligand:1992	RELAXIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	MyCancerGenome	20-Jun-17	antibody	1.413668071730236	ZIV-AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-180736A	chembl:CHEMBL384073	GSK-180736A	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.007012242	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.008518441	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
MHC CLASS I NK CELL RECEPTOR 3DL2	hgnc:6330	KIR2DL2	TTD	2020.06.01	NULL	6.563458904461812	IPH4102	ncit:C124999	LACUTAMAB	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.020041096	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.030176823	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1961070821127712	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	2.917092846427472	MAGNESIUM SULFATE	rxcui:1311625	MAGNESIUM SULFATE ANHYDROUS	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	2-METHOXYPHENAZINE	chembl:CHEMBL1420181	CHEMBL:CHEMBL1420181	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.017409705	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.3165837197673226	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	0.9376369863516875	Cisatracurium	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
UNIPROT:P00750	hgnc:9051	PLAT	TEND	1-Aug-11	NULL	3.182283105193605	TRANEXAMIC ACID	rxcui:10691	TRANEXAMIC ACID	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.058997383	IUPHAR.LIGAND:950	iuphar.ligand:3296	[3H]7-OH-DPAT	FALSE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	ChEMBL	33	inhibitor	0.1790034246671403	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
BRDT	hgnc:1105	BRDT	ChEMBL	33	inhibitor	0.6250913242344582	MOLIBRESIB	ncit:C101538	MOLIBRESIB	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1325951293830669	ISOSORBIDE DINITRATE	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011746683	alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	2.983390411119005	Ivacaftor	rxcui:1243041	IVACAFTOR	TRUE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	PharmGKB	4/5/24	NULL	0.1049104320393496	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005208578	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.2561349816375342	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.2692701089009974	Oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:10417	iuphar.ligand:10417	COMPOUND 31 [PMID: 31259550]	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:9148	iuphar.ligand:9148	COMPOUND 4 [PMID: 27074625]	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1041818873724097	CARBARIL	ncit:C76389	CARBARIL	TRUE	FALSE	FALSE
NCBIGENE:1353	hgnc:2261	COX11	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:5175	ncit:C171920	DAZOXIBEN	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	4.200613699	SPERMINE TRIS-1-NAPG	chembl:CHEMBL2347632	CHEMBL:CHEMBL2347632	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.007806671	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.2051080907644316	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
SERPINH1	hgnc:1546	SERPINH1	NCI	14-Sep-17	NULL	0.5303805175322677	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.4518732464345482	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.082300425	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.078276194	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
PSMB11	hgnc:31963	PSMB11	ChEMBL	33	inhibitor	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	1.050153425	TALAZOPARIB TOSYLATE	rxcui:2099703	TALAZOPARIB TOSYLATE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	binder	0.062509132	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.071928317	TALETRECTINIB	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.049723174	regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	antibody	0.6177373086552294	IUPHAR.LIGAND:8966	iuphar.ligand:8966	ONARTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2707	ncit:C72822	NETOGLITAZONE	FALSE	FALSE	FALSE
PSMB1	hgnc:9537	PSMB1	DTC	9/2/20	NULL	3.214755381777214	MG-132	iuphar.ligand:8616	MG-132	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:8982	iuphar.ligand:8982	INCB-38579	FALSE	FALSE	FALSE
NCBIGENE:442	hgnc:755	ASNSP2	GuideToPharmacology	2024.1	activator	1.093909817410302	IUPHAR.LIGAND:4254	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.023616644	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.036463661	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.201952582	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.026519026	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	TCMDC-125620	chembl:CHEMBL530291	CHEMBL:CHEMBL530291	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	(E)-2-STYRYLCHROMONE	chembl:CHEMBL388823	CHEMBL:CHEMBL388823	FALSE	FALSE	FALSE
OR4D6	hgnc:15175	OR4D6	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.015219615	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	REVERSETRIIODOTHYRONINE	iuphar.ligand:2636	RT3	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.015516451	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.018613141	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
NCBIGENE:3236	hgnc:5133	HOXD10	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12748	iuphar.ligand:12748	PF-06835919	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	ICI-199,441	iuphar.ligand:11691	ICI-199441	FALSE	FALSE	FALSE
APEH	hgnc:586	APEH	PharmGKB	4/5/24	NULL	0.1083749664307419	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.01795748	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.2548916079402645	1,4,5,8-TETRAAMINO-ANTHRAQUINONE	chembl:CHEMBL87568	CHEMBL:CHEMBL87568	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	GNF-PF-4876	chembl:CHEMBL585444	CHEMBL:CHEMBL585444	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.038131933	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.025244073	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003541833	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	PERFLUNAFENE	rxcui:2462501	PERFLUNAFENE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.055504938	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:265	iuphar.ligand:265	5-BENZYLOXYTRYPTAMINE	FALSE	FALSE	FALSE
CLDN11	hgnc:8514	CLDN11	PharmGKB	4/5/24	NULL	8.078103267029924	anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:4099	iuphar.ligand:4099	TRANS-3-ACPBPA	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	TALC	12-May-16	inhibitor	0.7242437411819931	EZN-2968	ncit:C68930	ANTI-HIF-1ALPHA LNA ANTISENSE OLIGONUCLEOTIDE EZN-2968	FALSE	FALSE	TRUE
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	0.4688184931758437	ABT-263	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	NCI	14-Sep-17	NULL	0.01097339	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	3.889457128569962	DIETHYL-2-TETRADECYLIDENEMALONATE	chembl:CHEMBL257748	CHEMBL:CHEMBL257748	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.012932924	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	GNF-PF-3257	chembl:CHEMBL601768	CHEMBL:CHEMBL601768	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	GANODERIC ACID TR	chembl:CHEMBL1097474	GANODERIC ACID TR	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	CetuGEX	ncit:C94221	ANTI-EGFR MONOCLONAL ANTIBODY GT-MAB 5.2-GEX	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.1160818081850283	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	CancerCommons	25-Jul-13	inhibitor	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.3409589041278864	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
GUCY1B1	hgnc:4687	GUCY1B1	ChEMBL	33	activator	1.544343271638073	CINACIGUAT	ncit:C87280	CINACIGUAT	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:5928	iuphar.ligand:5928	KU-55933	FALSE	FALSE	FALSE
NCBIGENE:1358	hgnc:2297	CPA2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8871	iuphar.ligand:8871	(2S,4S)-KETOCONAZOLE	FALSE	FALSE	FALSE
NCBIGENE:622	hgnc:1027	BDH1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:2828	iuphar.ligand:2828	DAIDZEIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006199253	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.2047082699247349	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
TRGV3	hgnc:12288	TRGV3	ChEMBL	33	inhibitor	4.375639269641208	MEDI-500	chembl:CHEMBL2109592	MEDI-500	FALSE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	inhibitor	2.692701089009974	INTETUMUMAB	ncit:C61070	INTETUMUMAB	FALSE	FALSE	FALSE
UNIPROT:P13500	hgnc:10618	CCL2	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	NOX-E36	ncit:C171710	EMAPTICAP PEGOL	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6083	iuphar.ligand:6083	GALANIN(7-29) (PIG)	FALSE	FALSE	FALSE
XPC	hgnc:12816	XPC	PharmGKB	4/5/24	NULL	0.7001022831425933	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	2.019525817	E2012	iuphar.ligand:7358	E2012	FALSE	FALSE	FALSE
GC	hgnc:4187	GC	PharmGKB	4/5/24	NULL	0.2430910705356227	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NEUROPEPTIDE Y RECEPTOR TYPE 1	hgnc:7956	NPY1R	TTD	2020.06.01	NULL	1.750255707856483	PD-160170	chembl:CHEMBL422942	CHEMBL:CHEMBL422942	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.026748686	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
COL1A1	hgnc:2197	COL1A1	ChEMBL	33	cleavage	0.8036888454443035	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.076690854	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
PTGDR	hgnc:9591	PTGDR	ChEMBL	33	inhibitor	2.917092846427472	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	NABILONE	rxcui:31447	NABILONE	TRUE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	2.386712328895204	Roxadustat	ncit:C141436	ROXADUSTAT	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	NSC-45382	chembl:CHEMBL1214274	CHEMBL:CHEMBL1214274	FALSE	FALSE	FALSE
UNIPROT:Q9UI33	hgnc:10583	SCN11A	TEND	1-Aug-11	NULL	0.130291988	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6113	iuphar.ligand:6113	GAL-B2-C12	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.6141248097742047	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	GW0742	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	DIOXYBENZONE	rxcui:23350	DIOXYBENZONE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
UNIPROT:Q05586	hgnc:4584	GRIN1	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	DEXANABINOL	ncit:C99381	DEXANABINOL	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.595325071	RIVAROXABAN	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:71	iuphar.ligand:71	MPDT	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.021988137	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.075768645	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006488837	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.076263865	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.105947682	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006397133	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000775559	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.5707355569097228	CIPROFIBRATE	rxcui:21149	CIPROFIBRATE	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.280789686	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.028444026	ANTIDEPRESSANTS	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.002278979	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.1041818873724097	LY3023414	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.157680694	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	1,4,5,8-TETRAAMINO-ANTHRAQUINONE	chembl:CHEMBL87568	CHEMBL:CHEMBL87568	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.99446347	BETAXOLOL	rxcui:1520	BETAXOLOL	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.101562227	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.5048814541893701	CHOLIC ACID	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.108040476	CHLORDANE	iuphar.ligand:2831	CHLORDANE	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	MyCancerGenome	20-Jun-17	inhibitor	0.525076712	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.116943588	DROMOSTANOLONE PROPIONATE	rxcui:23678	DROMOSTANOLONE	TRUE	FALSE	TRUE
UNIPROT:P05362	hgnc:5344	ICAM1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	HYALURONAN	rxcui:5463	HYALURONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:7524	iuphar.ligand:7524	XD14	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	blocker	0.6563458904461812	IUPHAR.LIGAND:4138	iuphar.ligand:4138	ARGIOTOXIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	Z-PRO-PROLINAL	drugbank:DB03535	Z-PRO-PROLINAL	FALSE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TEND	1-Aug-11	NULL	0.4688184931758437	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000991047	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TRIBROMSALAN	ncit:C47768	TRIBROMSALAN	TRUE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	1.105424657593568	Belzutifan	rxcui:2567226	BELZUTIFAN	TRUE	FALSE	FALSE
PSMC5	hgnc:9552	PSMC5	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
MT-ND3	hgnc:7458	MT-ND3	ChEMBL	33	inhibitor	0.2573905452730122	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	DTC	9/2/20	NULL	0.2273059360852575	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	BENZYL ISOTHIOCYANATE	drugbank:DB16860	BENZYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.005873341	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
UNIPROT:P33527	hgnc:51	ABCC1	TdgClinicalTrial	Jan-14	NULL	0.1844531776429549	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.5000730593875666	IUPHAR.LIGAND:2422	rxcui:1297880	CAMPHOR OIL	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.012211086	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.046466966	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6103	iuphar.ligand:6103	M1152	FALSE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	modulator	0.1458546423213736	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:7975	iuphar.ligand:7975	BPH-675	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.7095631248066824	MEBANAZINE	ncit:C80969	MEBANAZINE	TRUE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.305277158	IUPHAR.LIGAND:2476	iuphar.ligand:2476	NI2+	FALSE	FALSE	FALSE
NCBIGENE:1329	hgnc:2269	COX5B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9883	iuphar.ligand:9883	COMPOUND 46C [PMID: 29350534]	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:5933	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	FRAXETIN	chembl:CHEMBL54909	FRAXETIN	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.2083637747448194	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
P-SELECTIN	hgnc:10721	SELP	TTD	2020.06.01	NULL	10.50153424713889	RPSGL-Ig	drugbank:DB06256	RPSGL-IG	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.020873652	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:1097	iuphar.ligand:1097	[35S]IBUTAMOREN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.092443083	TCMDC-125465	chembl:CHEMBL536151	CHEMBL:CHEMBL536151	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.6482428547616604	GSK-2018682	drugbank:DB11987	GSK-2018682	FALSE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	2.282942227638891	FE-202158	ncit:C152319	SELEPRESSIN	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1392776425349986	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.049210563	IUPHAR.LIGAND:5617	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
CXCR2	hgnc:6027	CXCR2	ChEMBL	33	modulator	1.944728564284981	REPARIXIN	ncit:C66515	REPARIXIN	FALSE	FALSE	FALSE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:8973	iuphar.ligand:8973	HUMAN GIP(1-30)NH2	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	ACEMETACIN	rxcui:16695	ACEMETACIN	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	FDA	10-Apr-24	NULL	2.983390411119005	Ivacaftor	rxcui:1243041	IVACAFTOR	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.028290771	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:1134	iuphar.ligand:1134	[125I]GLP-1-(7-36)-AMIDE	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:4077	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.029074015	IUPHAR.LIGAND:2868	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
UNIPROT:P10827	hgnc:11796	THRA	TEND	1-Aug-11	NULL	1.875273972703375	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1988926940746003	7,2'-DIHYDROXYFLAVONE	chembl:CHEMBL475908	CHEMBL:CHEMBL475908	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.1356787370431382	IUPHAR.LIGAND:9029	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
FNTA	hgnc:3782	FNTA	MyCancerGenome	20-Jun-17	other/unknown	2.917092846427472	TIPIFARNIB	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1715936968486748	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
INTERLEUKIN-13	hgnc:5973	IL13	TTD	2020.06.01	NULL	6.563458904461812	Tralokinumab	rxcui:2589225	TRALOKINUMAB	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PARAOXON	ncit:C99562	PARAOXON	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:9650	ncit:C174807	DAGROCORAT	FALSE	FALSE	FALSE
NCBIGENE:734	hgnc:1355	OSGIN2	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.057700738	IUPHAR.LIGAND:7221	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	Chlorpheniramine	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
IL5	hgnc:6016	IL5	NCI	14-Sep-17	NULL	0.1341192113299987	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	inhibitor	0.043611023	IUPHAR.LIGAND:2805	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
ICAM1	hgnc:5344	ICAM1	DTC	9/2/20	NULL	6.563458904461812	LIFITEGRAST	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.063722902	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.073266518	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.4070362111294147	IUPHAR.LIGAND:9812	iuphar.ligand:9812	AZD9567	FALSE	FALSE	FALSE
QUINONE REDUCTASE 2	hgnc:7856	NQO2	TTD	2020.06.01	NULL	0.6177373086552295	NSC-645809	chembl:CHEMBL338604	C-1311	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	SJ000024939	chembl:CHEMBL590691	CHEMBL:CHEMBL590691	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	NCI	14-Sep-17	NULL	0.2734774543525755	CORTICOTROPIN	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.011152861	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	1.093909817410302	TCMDC-123749	chembl:CHEMBL524376	CHEMBL:CHEMBL524376	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4208	iuphar.ligand:4208	GV196771A	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.004428785	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.021234525	9-CRA	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	STROPHANTHIDIN	chembl:CHEMBL111743	STROPHANTHIDIN	FALSE	FALSE	FALSE
NDUFS2	hgnc:7708	NDUFS2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
ATP1A4	hgnc:14073	ATP1A4	ChEMBL	33	inhibitor	0.2917092846427472	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.076098074	IUPHAR.LIGAND:3309	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:5777	iuphar.ligand:5777	FLTCHAAR	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4154	iuphar.ligand:4154	CGP37849	FALSE	FALSE	FALSE
PSMA3	hgnc:9532	PSMA3	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.1086365611772989	CIS-PLATINUM	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.1411496538593938	IUPHAR.LIGAND:727	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.6731752722524935	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.1121958787087489	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.2117244807890907	IUPHAR.LIGAND:4260	iuphar.ligand:4260	N1-DANSYL-SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:5852	iuphar.ligand:5852	MRE-269	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:3480	ncit:C170264	OSANETANT	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	1.334940794127826	SPIRAPRIL	rxcui:36908	SPIRAPRIL	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.052090944	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.1411496538593938	IUPHAR.LIGAND:4084	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	PharmGKB	4/5/24	NULL	0.2206204673768676	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
ADENOSINE DEAMINASE	hgnc:186	ADA	TTD	2020.06.01	NULL	2.282942227638891	Elapegademase	rxcui:2059218	ELAPEGADEMASE-LVLR	TRUE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:4079	iuphar.ligand:4079	[3H]CGP61594	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-3438	chembl:CHEMBL582276	CHEMBL:CHEMBL582276	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.023336743	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	0.8899605294185507	OLMESARTAN	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.018062494	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	modulator	0.072324616	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
PTHLH	hgnc:9607	PTHLH	NCI	14-Sep-17	NULL	1.093909817410302	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	NSC-747266	chembl:CHEMBL609570	CHEMBL:CHEMBL609570	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.064347636	PERGOLIDE	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.6908904109959803	MM-111	drugbank:DB17983	MM-111	FALSE	TRUE	TRUE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.4884434533552977	PROTEIN KINASE INHIBITOR	ncit:C1404	PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:3239	hgnc:5136	HOXD13	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12800	iuphar.ligand:12800	ML162	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	3.000438356	LANRAPLENIB	ncit:C174607	LANRAPLENIB	FALSE	FALSE	FALSE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.100976291	PKI-589	ncit:C84837	PI3K/MTOR KINASE INHIBITOR PF-04691502	FALSE	FALSE	TRUE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:257	iuphar.ligand:257	SB 207710	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.012695278	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.1521961485092594	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	1.944728564284981	Moxetumomab pasudotox	rxcui:2099295	MOXETUMOMAB PASUDOTOX	TRUE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	ChEMBL	33	agonist	6.563458904461812	CHORIOGONADOTROPIN ALFA	rxcui:283550	CHORIOGONADOTROPIN ALFA	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.041672755	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
NCBIGENE:3110	hgnc:4979	MNX1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10718	iuphar.ligand:10718	COMPOUND 25 [PMID: 32105470]	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.1973972602845657	ELAFIBRANOR	ncit:C166574	ELAFIBRANOR	FALSE	FALSE	FALSE
SP7	hgnc:17321	SP7	NCI	14-Sep-17	NULL	4.039051633514962	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1025540453822158	TRACAZOLATE	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004762601	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.020465128	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	blocker	0.175610941	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
UNIPROT:P08514	hgnc:6138	ITGA2B	TEND	1-Aug-11	NULL	3.646366058	ABCIXIMAB	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:260	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	0.8204323630577265	Triflupromazine	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P14784	hgnc:6009	IL2RB	TEND	1-Aug-11	NULL	0.4039051633514962	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
CYP4B1	hgnc:2644	CYP4B1	PharmGKB	4/5/24	NULL	0.3163112725041837	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:4286	iuphar.ligand:4286	PICROTIN	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1848861663228679	NSC-37642	chembl:CHEMBL1707907	CHEMBL:CHEMBL1707907	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.9053046764774912	NEBULARINE	drugbank:DB04440	NEBULARINE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	TULOBUTEROL	rxcui:38967	TULOBUTEROL	TRUE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:7958	iuphar.ligand:7958	LY2090314	FALSE	FALSE	FALSE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.077789143	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.6326225450083675	IUPHAR.LIGAND:106	iuphar.ligand:106	5-(NONYLOXY)-TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.03251249	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1739	iuphar.ligand:1739	REACTIVE BLUE-2	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:8481	iuphar.ligand:8481	LDN-214117	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	TCMDC-124022	chembl:CHEMBL548017	CHEMBL:CHEMBL548017	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:10688	iuphar.ligand:10688	GNF4877	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.082043236	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.030176823	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.022606632	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6407	iuphar.ligand:6407	COMPOUND 30 [PMID: 21757343]	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:11548	iuphar.ligand:11548	COMPOUND 4-3 [PMID: 34027661]	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	ChEMBL	33	inhibitor	0.8751278539282416	CERALASERTIB	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	negative modulator	0.9546849315580818	DORAVIRINE	rxcui:2055755	DORAVIRINE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3125456621172291	LACIDIPINE	rxcui:28382	LACIDIPINE	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:3203	iuphar.ligand:3203	CINNAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2198	ncbigene:2198	FAUNA@	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:12157	ncit:C175865	TILPISERTIB	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:2016	iuphar.ligand:2016	L-817,818	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:9634	iuphar.ligand:9634	(S)-CHLOROSUCCINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:402	hgnc:693	ARL2	GuideToPharmacology	2024.1	blocker	2.100306849	IUPHAR.LIGAND:2359	iuphar.ligand:2359	ZD7288	FALSE	FALSE	FALSE
NCBIGENE:2940	hgnc:4628	GSTA3	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:12361	iuphar.ligand:12361	SABATOLIMAB	FALSE	FALSE	FALSE
APC	hgnc:583	APC	NCI	14-Sep-17	NULL	0.1403948428761885	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1595	ncit:C81534	ACIFRAN	FALSE	FALSE	FALSE
TSPO	hgnc:1158	TSPO	NCI	14-Sep-17	NULL	0.6908904109959803	METRONIDAZOLE	rxcui:6922	METRONIDAZOLE	TRUE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.072324616	WARFARIN	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	ZM-336372	iuphar.ligand:9130	ZM336372	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.09972967	prenylamine	rxcui:8674	PRENYLAMINE	TRUE	FALSE	FALSE
NCBIGENE:2032	ncbigene:2032	ENUR2	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	S-222611	chembl:CHEMBL3545200	S-222611	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.3777530304726222	RADOTINIB	ncit:C98110	RADOTINIB	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
UNIPROT:P20292	hgnc:436	ALOX5AP	TdgClinicalTrial	Jan-14	NULL	7.501095891	AM-803	chembl:CHEMBL1922660	FIBOFLAPON	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.097308509	XL880	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:5662	iuphar.ligand:5662	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:9170	iuphar.ligand:9170	COMPOUND 51 [MALLINGER ET AL., 2016]	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:3381	iuphar.ligand:3381	BAYU9773	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3381	iuphar.ligand:3381	BAYU9773	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:11220	iuphar.ligand:11220	SUPRASTAT	FALSE	FALSE	FALSE
NCBIGENE:2013	hgnc:3334	EMP2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8167	iuphar.ligand:8167	LEUCETTINE L41	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.029416062	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004616465	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1274	iuphar.ligand:1274	VUF 8430	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.010777437	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.1035654265003836	IUPHAR.LIGAND:1204	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	DTC	9/2/20	NULL	0.5834185692854944	TCMDC-125454	chembl:CHEMBL535714	CHEMBL:CHEMBL535714	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.2243917574174978	IUPHAR.LIGAND:1250	iuphar.ligand:1250	IMETIT	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.063160791	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.060249766	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.037081689	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	BIFENAZATE	chembl:CHEMBL1872845	BIFENAZATE	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.026418954	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004585022	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	FRAXETIN	chembl:CHEMBL54909	FRAXETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.073089743	GALETERONE	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:5281	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.006496866	IUPHAR.LIGAND:2181	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.009860596	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.039199456	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.046303061	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5652	iuphar.ligand:5652	LYSOPHOSPHATIDYLETHANOLAMINE	FALSE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.3889457128569963	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	inhibitor	3.281729452230906	PRASUGREL HYDROCHLORIDE	rxcui:847020	PRASUGREL HYDROCHLORIDE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.042310775	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	CID 3241690	chembl:CHEMBL259103	CHEMBL:CHEMBL259103	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10535	iuphar.ligand:10535	DD-03-171	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5745	iuphar.ligand:5745	COMPOUND 1 [PMID: 21273063]	FALSE	FALSE	FALSE
FBXL17	hgnc:13615	FBXL17	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	TIRABRUTINIB	ncit:C102876	TIRABRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8775	iuphar.ligand:8775	NCRW0005-F05	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:2090	iuphar.ligand:2090	NEUROKININ B	FALSE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	GLYCODIAZINE	rxcui:102848	GLYMIDINE	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:5947	iuphar.ligand:5947	CDK1/5 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.059397818	IUPHAR.LIGAND:5670	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.1017590527823536	IUPHAR.LIGAND:4346	iuphar.ligand:4346	ZK93423	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	SJ000114950	chembl:CHEMBL606456	CHEMBL:CHEMBL606456	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.027929612	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.024108205	labetalol	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.012713722	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	1.166837138570988	PHYTOCHEMICALS	ncit:C28269	PHYTOCHEMICAL	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.075010959	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.1651184630053286	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	BETAMETHASONE DIPROPIONATE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
CDK4	hgnc:1773	CDK4	CancerCommons	25-Jul-13	inhibitor	0.1190650141398968	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	0.2524407270946851	IUPHAR.LIGAND:2919	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	CancerCommons	25-Jul-13	inhibitor	30.00438356	ORTERONEL	ncit:C90582	ORTERONEL	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.1805819381121768	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
NCBIGENE:150	hgnc:281	ADRA2A	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:11280	iuphar.ligand:11280	AR291903	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	CGI	2/1/22	NULL	0.058341857	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CGI	2/1/22	NULL	0.020465128	Flutamide	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.074163377	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	CGI	2/1/22	NULL	0.2651902587661338	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
CA1	hgnc:1368	CA1	ChEMBL	33	inhibitor	0.4375639269641208	METHOCARBAMOL	rxcui:6845	METHOCARBAMOL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.077273983	AZD6738	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:12819	iuphar.ligand:12819	PBI-4547	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	2.019525817	PEGAPTANIB SODIUM	rxcui:498509	PEGAPTANIB	TRUE	FALSE	FALSE
CYSLTR1	hgnc:17451	CYSLTR1	ChEMBL	33	inhibitor	1.084869240406911	MONTELUKAST SODIUM	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.7026004179620139	ENALAPRIL MALEATE	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	2.500365296937833	TENECTEPLASE	rxcui:259280	TENECTEPLASE	TRUE	FALSE	FALSE
PNLIP	hgnc:9155	PNLIP	ChEMBL	33	inhibitor	3.029288725136221	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1396480617970598	METHSCOPOLAMINE BROMIDE	rxcui:56092	METHSCOPOLAMINE BROMIDE	TRUE	FALSE	FALSE
NCBIGENE:2039	hgnc:3382	DMTN	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9357	iuphar.ligand:9357	BI605906	FALSE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ChEMBL	33	inhibitor	0.5000730593875666	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1331836936859721	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.3642372228836055	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:1402	hgnc:736	NAAA	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:5161	iuphar.ligand:5161	CCP	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	ChEMBL	33	agonist	0.9309870786470656	THYROTROPIN ALFA	rxcui:4952	THYROTROPIN ALFA	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.084146909	DROPERIDOL	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN PURIFIED PORK	chembl:CHEMBL1201630	INSULIN PURIFIED PORK	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.08178765	LISDEXAMFETAMINE DIMESYLATE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:4972	iuphar.ligand:4972	INSULIN-LIKE GROWTH FACTOR 2	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.059481927	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.2453629496995069	PHENYLPROPANOLAMINE HYDROCHLORIDE	rxcui:3266	PHENYLPROPANOLAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	inhibitor	1.591141552596802	CROFELEMER	rxcui:1364449	CROFELEMER	TRUE	FALSE	FALSE
FRK	hgnc:3955	FRK	ChEMBL	33	inhibitor	0.1136529680426288	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.091636424	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	modulator	1.721562991334245	ULIPRISTAL ACETATE	rxcui:1005920	ULIPRISTAL ACETATE	TRUE	FALSE	FALSE
NCBIGENE:2453	hgnc:3850	FRA13A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12108	ncit:C188615	BEXOTEGRAST	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	HYDROCODONE BITARTRATE	rxcui:142439	HYDROCODONE BITARTRATE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.078276194	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	inhibitor	0.1023541349623674	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	potentiator	0.4526523382387456	PINACIDIL	rxcui:33717	PINACIDIL	TRUE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.5321723436050118	TRANYLCYPROMINE SULFATE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.6731752722524935	TRANYLCYPROMINE SULFATE	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.3488881809680697	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
NCBIGENE:2042	hgnc:3387	EPHA3	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:9655	iuphar.ligand:9655	TAKINIB	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.032899543	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
RRM2	hgnc:10452	RRM2	ChEMBL	33	inhibitor	0.384671584	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
COL3A1	hgnc:2201	COL3A1	ChEMBL	33	cleavage	2.812910959055062	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL4A2	hgnc:2203	COL4A2	ChEMBL	33	cleavage	0.6250913242344582	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL11A1	hgnc:2186	COL11A1	ChEMBL	33	cleavage	0.1172046232939609	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	ChEMBL	33	inhibitor	0.4579157375205915	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB10	hgnc:9538	PSMB10	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB3	hgnc:9540	PSMB3	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.4039051633514962	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
NCBIGENE:1697	ncbigene:1697	DFNB5	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:7574	rxcui:1876376	DUPILUMAB	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.9546849315580818	VALDECOXIB	rxcui:278567	VALDECOXIB	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.251232877	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	4.861821410712453	OFATUMUMAB	rxcui:712566	OFATUMUMAB	TRUE	TRUE	TRUE
EPHA3	hgnc:3387	EPHA3	ChEMBL	33	inhibitor	0.100589408	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9666	iuphar.ligand:9666	PF-06426779	FALSE	FALSE	FALSE
EPHA5	hgnc:3389	EPHA5	ChEMBL	33	inhibitor	0.1810609352954982	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
EPHA8	hgnc:3391	EPHA8	ChEMBL	33	inhibitor	0.069638821	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:2460	hgnc:6161	ITGB6	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:10450	iuphar.ligand:10450	COMPOUND 7 [PMID: 31381331]	FALSE	FALSE	FALSE
NDUFA5	hgnc:7688	NDUFA5	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFB4	hgnc:7699	NDUFB4	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFB9	hgnc:7704	NDUFB9	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFV3	hgnc:7719	NDUFV3	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.030598876	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.030211548	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
NCBIGENE:2462	hgnc:3859	FRA16C	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:10450	iuphar.ligand:10450	COMPOUND 7 [PMID: 31381331]	FALSE	FALSE	FALSE
ATP1A1	hgnc:799	ATP1A1	ChEMBL	33	inhibitor	1.555782851427985	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
ATP1A1	hgnc:799	ATP1A1	ChEMBL	33	inhibitor	0.5527123287967842	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.027121731	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.063160791	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.066241806	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.073885091	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.07767407	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	agonist	0.099446347	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	agonist	0.033919684	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	agonist	0.036013492	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.056826484	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.058212496	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.021715331	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.018819954	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:5853	iuphar.ligand:5853	EP 157	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.093763699	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	modulator	0.1312691780892362	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	modulator	0.100976291	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	modulator	0.030527716	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	modulator	0.100976291	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
NCBIGENE:667	hgnc:1090	DST	GuideToPharmacology	2024.1	agonist	3.750547945406749	IUPHAR.LIGAND:7163	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.079557078	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.2237542808339254	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.064111931	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.036977233	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.057073556	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.059667808	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.061055432	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:674	ncbigene:674	BRAFPS1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9112	iuphar.ligand:9112	GIV3727	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.073954467	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.076098074	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.054695491	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.084553416	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.060772768	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.066297565	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.067839369	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1383601350084176	DROPERIDOL	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	1.458546423213736	PARAMETHADIONE	rxcui:32894	PARAMETHADIONE	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.6250913242344582	TRIMETHADIONE	rxcui:10827	TRIMETHADIONE	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	2.187819634820604	TRIMETHADIONE	rxcui:10827	TRIMETHADIONE	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.305277158	TRIMETHADIONE	rxcui:10827	TRIMETHADIONE	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	FINAFLOXACIN	rxcui:1598641	FINAFLOXACIN	TRUE	FALSE	FALSE
NCBIGENE:676	hgnc:1105	BRDT	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9112	iuphar.ligand:9112	GIV3727	FALSE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.3571950424196904	MIBEFRADIL DIHYDROCHLORIDE	rxcui:83214	MIBEFRADIL DIHYDROCHLORIDE	TRUE	FALSE	FALSE
FYN	hgnc:4037	FYN	ChEMBL	33	inhibitor	0.3241214273808303	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.1458546423213736	HMN-214	chembl:CHEMBL3545431	HMN-214	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.100589408	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.1226814748497534	LY-2874455	drugbank:DB13022	LY-2874455	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.5707355569097228	LS-104	chembl:CHEMBL5095023	LS-104	FALSE	FALSE	FALSE
ARAF	hgnc:646	ARAF	ChEMBL	33	inhibitor	0.3182283105193605	LY-3009120	chembl:CHEMBL3545195	LY-3009120	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	1.381780822	LY-2606368	chembl:CHEMBL3545377	LY-2606368	FALSE	FALSE	FALSE
NDUFA8	hgnc:7692	NDUFA8	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFV3	hgnc:7719	NDUFV3	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFC1	hgnc:7705	NDUFC1	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB5	hgnc:7700	NDUFB5	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFS6	hgnc:7713	NDUFS6	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFA8	hgnc:7692	NDUFA8	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
MT-ND5	hgnc:7461	MT-ND5	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA12	hgnc:23987	NDUFA12	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA9	hgnc:7693	NDUFA9	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFB2	hgnc:7697	NDUFB2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA13	hgnc:17194	NDUFA13	ChEMBL	33	inhibitor	0.2625383561784725	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.305277158	PLX-7486	chembl:CHEMBL3545381	PLX-7486	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.044878351	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.1798207919030633	PLX-7486	chembl:CHEMBL3545381	PLX-7486	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.2083637747448194	AVUTOMETINIB	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.5707355569097228	TRICETAMIDE	ncit:C74378	TRICETAMIDE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.2430910705356226	PKI-179	drugbank:DB13109	PKI-179	FALSE	FALSE	FALSE
SMO	hgnc:11119	SMO	ChEMBL	33	inhibitor	8.751278539282415	LEQ506	chembl:CHEMBL3133037	LEQ506	FALSE	FALSE	FALSE
RPS6KB2	hgnc:10437	RPS6KB2	ChEMBL	33	inhibitor	2.625383561784725	XL-418	chembl:CHEMBL2016893	XL-418	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.1479089330582944	XL-418	chembl:CHEMBL2016893	XL-418	FALSE	FALSE	FALSE
GRM3	hgnc:4595	GRM3	ChEMBL	33	agonist	5.250767123569449	LY404039	chembl:CHEMBL375611	LY404039	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	modulator	0.2075402025126264	SERIDOPIDINE	ncit:C152345	SERIDOPIDINE	FALSE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	5.834185692854944	LAS101057	chembl:CHEMBL1672627	LAS101057	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	GSK159802	chembl:CHEMBL3545087	GSK159802	FALSE	FALSE	FALSE
PDE10A	hgnc:21160	LINC00473	ChEMBL	33	inhibitor	4.375639269641208	PBF-999	iuphar.ligand:13188	PBF-999	FALSE	FALSE	FALSE
HRH4	hgnc:17383	HRH4	ChEMBL	33	inhibitor	14.32027397337122	ADRIFORANT	ncit:C169765	ADRIFORANT	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.059667808	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1363835616511545	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.038131933	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.1902451856365742	BMS-582949	drugbank:DB12696	BMS-582949	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1848861663228679	GOLVATINIB	ncit:C82363	GOLVATINIB	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.4167275494896389	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.3472729579080324	ROCILETINIB	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
CDK5	hgnc:1774	CDK5	ChEMBL	33	inhibitor	0.085239726	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1785975212098452	FAMITINIB	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.3125456621172291	FADOLMIDINE HYDROCHLORIDE	ncit:C77297	FADOLMIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2465148884304905	FADOLMIDINE HYDROCHLORIDE	ncit:C77297	FADOLMIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
LTB4R	hgnc:6713	LTB4R	ChEMBL	33	inhibitor	1.093909817410302	ETALOCIB	ncit:C1626	ETALOCIB	FALSE	FALSE	FALSE
PTAFR	hgnc:9582	PTAFR	ChEMBL	33	inhibitor	8.751278539282415	MINOPAFANT	ncit:C170178	MINOPAFANT	FALSE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	agonist	2.282942227638891	SELEPRESSIN	ncit:C152319	SELEPRESSIN	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.8468979231563628	ITACITINIB	ncit:C116855	ITACITINIB	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	blocker	0.5173169579871378	LANICEMINE	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	blocker	0.192335792	LANICEMINE	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.5556367326528519	NAZARTINIB	ncit:C115109	NAZARTINIB	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	positive modulator	0.3125456621172291	FARAMPATOR	ncit:C65620	FARAMPATOR	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.3977853881492007	BECAMPANEL	ncit:C79860	BECAMPANEL	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.4234489615781814	BECAMPANEL	ncit:C79860	BECAMPANEL	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	0.596678082	BECAMPANEL	ncit:C79860	BECAMPANEL	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	positive modulator	0.4234489615781814	MIBAMPATOR	ncit:C174617	MIBAMPATOR	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	positive modulator	0.3977853881492007	MIBAMPATOR	ncit:C174617	MIBAMPATOR	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	inverse agonist	0.036463661	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	inverse agonist	0.042619863	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
TRPV3	hgnc:18084	TRPV3	ChEMBL	33	inhibitor	8.751278539282415	GRC-15300	chembl:CHEMBL3707319	GRC-15300	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.1461794856227575	APALUTAMIDE	rxcui:1999574	APALUTAMIDE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.036770078	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.036770078	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	inhibitor	1.419126249613364	LECOZOTAN HYDROCHLORIDE	ncit:C72813	LECOZOTAN HYDROCHLORIDE	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	7.001022831425932	TELCAGEPANT	ncit:C152545	TELCAGEPANT	FALSE	FALSE	FALSE
RXFP2	hgnc:17318	RXFP2	ChEMBL	33	activator	4.375639269641208	SERELAXIN	ncit:C152342	SERELAXIN	FALSE	FALSE	FALSE
OPRL1	hgnc:8155	OPRL1	ChEMBL	33	agonist	0.7292732116068681	CEBRANOPADOL	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	agonist	1.973972602845657	PICLIDENOSON	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.1296485709523321	CEBRANOPADOL	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
PTGDR	hgnc:9591	PTGDR	ChEMBL	33	inhibitor	5.250767123569449	ASAPIPRANT	ncit:C171866	ASAPIPRANT	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	binder	2.423430980108977	GANTENERUMAB	ncit:C88580	GANTENERUMAB	FALSE	FALSE	FALSE
TRAV29DV5	hgnc:12127	TRAV29DV5	ChEMBL	33	inhibitor	4.375639269641208	MEDI-500	chembl:CHEMBL2109592	MEDI-500	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
CTSK	hgnc:2536	CTSK	ChEMBL	33	inhibitor	23.33674277141977	ODANACATIB	ncit:C66981	ODANACATIB	FALSE	FALSE	TRUE
AOPEP	hgnc:1361	AOPEP	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
GUCY2C	hgnc:4688	GUCY2C	ChEMBL	33	agonist	19.69037671338543	PLECANATIDE	rxcui:1873752	PLECANATIDE	TRUE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	ChEMBL	33	inhibitor	0.3571950424196904	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMB5	hgnc:9542	PSMB5	ChEMBL	33	inhibitor	0.7501095890813498	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.071439008	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	2.187819634820604	CANTUZUMAB RAVTANSINE	ncit:C61576	CANTUZUMAB RAVTANSINE	FALSE	FALSE	FALSE
CD200	hgnc:7203	CD200	ChEMBL	33	inhibitor	157.5230137070835	SAMALIZUMAB	ncit:C77891	SAMALIZUMAB	FALSE	FALSE	FALSE
CD14	hgnc:1628	CD14	ChEMBL	33	inhibitor	14.32027397337122	IC14	chembl:CHEMBL2109330	IC14	FALSE	FALSE	FALSE
FCGR1A	hgnc:3613	FCGR1A	ChEMBL	33	modulator	15.75230137070834	MDX-447	chembl:CHEMBL2109391	MDX-447	FALSE	FALSE	FALSE
MADCAM1	hgnc:6765	MADCAM1	ChEMBL	33	inhibitor	17.50255707856483	ONTAMALIMAB	ncit:C166947	ONTAMALIMAB	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	agonist	0.068637479	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.079197091	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	FENCLOFENAC	ncit:C65643	FENCLOFENAC	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	METHAPYRILENE FUMARATE	ncit:C83953	METHAPYRILENE FUMARATE	TRUE	FALSE	FALSE
ADH1C	hgnc:251	ADH1C	ChEMBL	33	inhibitor	0.1666910197958555	NITREFAZOLE	ncit:C72626	NITREFAZOLE	TRUE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	1.521961485092594	SITAXENTAN	ncit:C73038	SITAXENTAN	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	VERALIPRIDE	rxcui:39468	VERALIPRIDE	TRUE	FALSE	FALSE
CHRM5	hgnc:1954	CHRM5	ChEMBL	33	inhibitor	0.033211683	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	inhibitor	2.187819634820604	LUCATUMUMAB	ncit:C48405	LUCATUMUMAB	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.1110098757625676	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.101562227	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.091583148	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.092443083	CELIPROLOL	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.1172046232939609	CELIPROLOL	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.036038209	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	blocker	0.09963505	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.5527123287967841	RG-7444	chembl:CHEMBL2109411	RG-7444	FALSE	FALSE	FALSE
TRAV29DV5	hgnc:12127	TRAV29DV5	ChEMBL	33	inhibitor	4.375639269641208	MASLIMOMAB	ncit:C188519	MASLIMOMAB	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	binder	2.282942227638891	90Y-CT84.66	chembl:CHEMBL2109369	90Y-CT84.66	FALSE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	0.8204323630577265	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.05913026	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.033919684	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
BHMT2	hgnc:1048	BHMT2	ChEMBL	33	other/unknown	5.250767124	BETAINE	rxcui:1512	BETAINE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.054020238	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	blocker	0.128067491	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNC3	hgnc:6235	KCNC3	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCND2	hgnc:6238	KCND2	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	positive modulator	0.729273212	ROPEGINTERFERON ALFA-2B	rxcui:2587059	ROPEGINTERFERON ALFA-2B	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.037213091	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3125456621172291	MANIDIPINE 6300	rxcui:29275	MANIDIPINE	FALSE	FALSE	FALSE
F12	hgnc:3530	F12	ChEMBL	33	inhibitor	2.187819634820604	HUMAN C1-ESTERASE INHIBITOR	ncit:C87730	HUMAN C1-ESTERASE INHIBITOR	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.305277158	MANIDIPINE 6300	rxcui:29275	MANIDIPINE	FALSE	FALSE	FALSE
GUCY1B2	hgnc:4686	GUCY1B2	ChEMBL	33	activator	0.8078103267029924	PRALICIGUAT	ncit:C174906	PRALICIGUAT	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.1260688385010672	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	2.059124362184098	BMS-986142	drugbank:DB15291	BMS-986142	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2983390411119005	GSK-256066	drugbank:DB12137	GSK-256066	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	1.193356164447602	OGLEMILAST	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
RPS11	hgnc:10384	RPS11	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS3A	hgnc:10421	RPS3A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL29	hgnc:10331	RPL29	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL14	hgnc:10305	RPL14	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS26	hgnc:10414	RPS26	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL31	hgnc:10334	RPL31	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL9P7	hgnc:30335	RPL9P7	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.3977853881492007	ELAFIBRANOR	ncit:C166574	ELAFIBRANOR	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.039538909	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
LGALS3	hgnc:6563	LGALS3	ChEMBL	33	inhibitor	26.25383561784724	BELAPECTIN	ncit:C115111	BELAPECTIN	FALSE	FALSE	FALSE
IL3RA	hgnc:6012	IL3RA	ChEMBL	33	binder	2.625383561784724	FLOTETUZUMAB	ncit:C117238	FLOTETUZUMAB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	ChEMBL	33	positive modulator	0.2318219480604613	CONTUSUGENE LADENOVEC	ncit:C2471	CONTUSUGENE LADENOVEC	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.5147810905460245	ABIVERTINIB MALEATE	ncit:C169756	ABIVERTINIB MALEATE	FALSE	FALSE	FALSE
IL3RA	hgnc:6012	IL3RA	ChEMBL	33	binder	10.50153424713889	TALACOTUZUMAB	ncit:C102784	TALACOTUZUMAB	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.2817943000126717	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.218327115	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	1.591141552596803	ACYLINE	drugbank:DB11906	ACYLINE	FALSE	FALSE	FALSE
ENPEP	hgnc:3355	ENPEP	ChEMBL	33	inhibitor	13.12691780892362	FIRIBASTAT	ncit:C166894	FIRIBASTAT	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	ZIMBERELIMAB	ncit:C159549	ZIMBERELIMAB	FALSE	FALSE	FALSE
RPS6KA6	hgnc:10435	RPS6KA6	ChEMBL	33	inhibitor	0.8751278539282418	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	binder	0.3241214273808302	AMG553	chembl:CHEMBL4650295	AMG553	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.078958904	E-7090	iuphar.ligand:11414	TASURGRATINIB	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	FLOTETUZUMAB	ncit:C117238	FLOTETUZUMAB	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.2075402025126264	PF-00217830	drugbank:DB12998	PF-00217830	FALSE	FALSE	FALSE
NCBP2	hgnc:7659	NCBP2	ChEMBL	33	modulator	26.25383561784724	OBEFAZIMOD	ncit:C158506	OBEFAZIMOD	FALSE	FALSE	FALSE
NCBP1	hgnc:7658	NCBP1	ChEMBL	33	modulator	26.25383561784724	OBEFAZIMOD	ncit:C158506	OBEFAZIMOD	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	inhibitor	1.193356164447602	IOWH-032	drugbank:DB12959	IOWH-032	FALSE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	ChEMBL	33	inhibitor	2.187819634820604	BAZLITORAN	ncit:C114975	BAZLITORAN	FALSE	FALSE	FALSE
NCBIGENE:662	hgnc:1082	BNIP1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:12425	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.3182283105193605	PEGAPAMODUTIDE	ncit:C170294	PEGAPAMODUTIDE	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.6403374540938354	RO-7121661	chembl:CHEMBL4594602	RO-7121661	FALSE	FALSE	FALSE
PRKAG1	hgnc:9385	PRKAG1	ChEMBL	33	activator	2.500365296937833	ACADESINE	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.057574201	IUPHAR.LIGAND:7949	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
LY75	hgnc:6729	LY75	ChEMBL	33	binder	17.50255707856483	RASDEGAFUSP ALFA	ncit:C170362	RASDEGAFUSP ALFA	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:10631	iuphar.ligand:10631	LORPUCITINIB	FALSE	FALSE	FALSE
LILRA4	hgnc:15503	LILRA4	ChEMBL	33	inhibitor	52.50767123569449	DAXDILIMAB	ncit:C174660	DAXDILIMAB	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	ChEMBL	33	inhibitor	4.039051633514961	AZENOSERTIB	ncit:C167064	AZENOSERTIB	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	TOLEBRUTINIB	ncit:C173549	TOLEBRUTINIB	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.7095631248066824	AZD-9164	drugbank:DB12115	AZD-9164	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.040640612	IUPHAR.LIGAND:5688	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1269527834518725	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2739530673166669	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.068369364	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1621858570986702	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.043180651	IUPHAR.LIGAND:7081	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:9285	iuphar.ligand:9285	PRN694	FALSE	FALSE	FALSE
P53	hgnc:11998	TP53	ClearityFoundationClinicalTrial	15-Jun-13	activator	0.010537361	GRANISETRON	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
IL-1R1	hgnc:5993	IL1R1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	3.141484604	ANAKINRA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.047518255	GDC-0943	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
NCBIGENE:971	hgnc:1696	CD72	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4589	iuphar.ligand:4589	DIOA	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.086861325	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	(+)-TETRAHYDROBERBERINE	chembl:CHEMBL476501	CHEMBL:CHEMBL476501	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.006504109	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.030996264	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	SJ000201287	chembl:CHEMBL590900	CHEMBL:CHEMBL590900	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	SJ000201788	chembl:CHEMBL602923	CHEMBL:CHEMBL602923	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.1037701012563132	QUINPIROLE	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	0.093098708	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	ETHACRIDINE LACTATE	rxcui:4107	ETHACRIDINE LACTATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	2,4,5,10-TETRAHYDROPYRAZOLO[3,4-A]CARBAZOLE	chembl:CHEMBL512649	CHEMBL:CHEMBL512649	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	agonist	0.1037701012563132	IUPHAR.LIGAND:5085	iuphar.ligand:5085	VEGFA	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.1930429089547591	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	0.087512785	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.017975923	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	SB-200646	chembl:CHEMBL85194	CHEMBL:CHEMBL85194	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.011530011	IUPHAR.LIGAND:7426	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	FALNIDAMOL	ncit:C80868	FALNIDAMOL	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.010526799	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	OXOPURPUREINE	chembl:CHEMBL456295	OXOPURPUREINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	TOSUFLOXACIN TOSYLATE	ncit:C76234	TOSUFLOXACIN TOSYLATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	CHLORDANE	iuphar.ligand:2831	CHLORDANE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	CYCLOFENIL	rxcui:2983	CYCLOFENIL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002188184	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
TNNC1	hgnc:11943	TNNC1	DTC	9/2/20	NULL	0.4565884455277782	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.008609226	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	0.095468493	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:11190	ncit:C175876	VIMSELTINIB	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	TCMDC-124354	chembl:CHEMBL546344	CHEMBL:CHEMBL546344	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.031707531	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	6ALPHA-METHYLPREDNISOLONE ACETATE	chembl:CHEMBL1364144	METHYLPREDNISOLONE ACETATE	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:2318	iuphar.ligand:2318	NS8593	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.093763699	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
CLCN3	hgnc:2021	CLCN3	DTC	9/2/20	NULL	26.25383561784724	BUFALIN	ncit:C107555	BUFALIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.093098708	GNF-PF-3501	chembl:CHEMBL581910	CHEMBL:CHEMBL581910	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.003116552	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.01151484	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	GNF-PF-704	chembl:CHEMBL597449	CHEMBL:CHEMBL597449	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	DNDI1417300	chembl:CHEMBL1401091	CHEMBL:CHEMBL1401091	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	3.750547945	IUPHAR.LIGAND:2390	drugbank:DB03566	SPERMIDINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.039778539	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1861974157294131	PT-101	chembl:CHEMBL316796	CHEMBL:CHEMBL316796	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.041021618	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	DNDI1417932	chembl:CHEMBL1334191	CHEMBL:CHEMBL1334191	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	GALANGIN	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	ARASERTACONAZOLE	ncit:C79926	ARASERTACONAZOLE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1033615575505797	HALOPROGIN	rxcui:26422	HALOPROGIN	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.003864268	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	0.1704794520639432	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010058941	OXIDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.075768645	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	(S,S)-(+)-FENOTEROL	chembl:CHEMBL389390	CHEMBL:CHEMBL389390	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006557721	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01495945	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:437	hgnc:6266	KCNJ5	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:2340	iuphar.ligand:2340	NA+	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.036062961	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	8-(3-BROMOPHENOXYMETHYL)CAFFEINE	chembl:CHEMBL2088301	CHEMBL:CHEMBL2088301	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-376719	chembl:CHEMBL156263	CHEMBL:CHEMBL156263	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	SEROTONIN	rxcui:1311214	SEROTONIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	BENZTROPINE MESYLATE	rxcui:18927	BENZTROPINE MESYLATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	MELENGESTROL ACETATE	rxcui:1537798	MELENGESTROL ACETATE	TRUE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.1715936968486748	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.03574382	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	7-NITROINDAZOLE	drugbank:DB02207	7-NITROINDAZOLE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	OXOTREMORINE	iuphar.ligand:302	OXOTREMORINE	FALSE	FALSE	FALSE
NCBIGENE:539	hgnc:850	ATP5PO	GuideToPharmacology	2024.1	blocker	5.834185692854944	IUPHAR.LIGAND:2547	iuphar.ligand:2547	MARGATOXIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	ANISOMYCIN	ncit:C95312	ANISOMYCIN	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	DEMETHYLZEYLASTERONE	chembl:CHEMBL465251	DEMETHYLZEYLASTERONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.1396480617970598	HOMOVANILLIC ACID	chembl:CHEMBL1562	HOMOVANILLIC ACID	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.005388718	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.026599631	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1693795846312726	PHENYLSTIBONIC ACID	chembl:CHEMBL1369257	PHENYLSTIBONIC ACID	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.005453643	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	2-PICOLINIC ACID	chembl:CHEMBL72628	2-PICOLINIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	SNC-80	iuphar.ligand:1611	SNC80	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	DNDI1417025	chembl:CHEMBL1320453	CHEMBL:CHEMBL1320453	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	IDEBENONE	rxcui:51296	IDEBENONE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.017189329	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.052090944	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	NELFINAVIR MESYLATE	rxcui:266565	NELFINAVIR MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	0.4102161815288632	IUPHAR.LIGAND:7658	iuphar.ligand:7658	GINSENOSIDE RG3	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.2143170254518142	GNF-PF-4085	chembl:CHEMBL528181	CHEMBL:CHEMBL528181	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	OXOGLAUCINE	iuphar.ligand:12559	OXOGLAUCINE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	3-EPI-ISOCUCURBITACIN D	chembl:CHEMBL2022241	CHEMBL:CHEMBL2022241	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.009696708	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:2686	hgnc:4259	GGT7	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:7025	iuphar.ligand:7025	DAMINOZIDE	FALSE	FALSE	FALSE
POLG	hgnc:9179	POLG	DTC	9/2/20	NULL	35.00511415712966	KASANOSIN B	chembl:CHEMBL457091	KASANOSIN B	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.130291988	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00292359	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.057197899	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	NSC-19029	chembl:CHEMBL483835	CHEMBL:CHEMBL483835	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	0.017490896	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.00854061	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.010148371	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1325	iuphar.ligand:1325	SHU9119	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.4412409347537352	NSC-119889	chembl:CHEMBL516616	CHEMBL:CHEMBL516616	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.062509132	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	ANAZOLENE	chembl:CHEMBL1555467	ANAZOLENE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	PHENAMIL	iuphar.ligand:4281	PHENAMIL	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.02302968	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	chembl:CHEMBL284028	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	DNDI1417025	chembl:CHEMBL1320453	CHEMBL:CHEMBL1320453	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003654487	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
PON1	hgnc:9204	PON1	DTC	9/2/20	NULL	0.6646540662746139	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:1325	iuphar.ligand:1325	SHU9119	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	METHYL 2-(2-METHOXYBENZAMIDO)BENZOATE	chembl:CHEMBL249190	CHEMBL:CHEMBL249190	FALSE	FALSE	FALSE
PTPN11	hgnc:9644	PTPN11	DTC	9/2/20	NULL	1.071585127259071	MESO-2,3-DIMERCAPTOSUCCINIC ACID	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	OXOGLAUCINE	iuphar.ligand:12559	OXOGLAUCINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	SAPPANONE A DIMETHYL ETHER	chembl:CHEMBL1489223	SAPPANONE A DIMETHYL ETHER	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	LAVENDUSTIN C	ncit:C1487	LAVENDUSTIN C	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.047561296	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	7-METHOXY-BAPTIGENIN	chembl:CHEMBL583578	CHEMBL:CHEMBL583578	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.001609332	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	QUESTIOMYCIN B	chembl:CHEMBL28319	QUESTIOMYCIN B	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.010156223	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	inhibitor	0.012268147	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
NCBIGENE:3136	hgnc:4965	HLA-H	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12941	drugbank:DB15257	MILADEMETAN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.1037701012563132	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	MUNDULONE ACETATE	chembl:CHEMBL1372368	MUNDULONE ACETATE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.008109293	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.037693949	QUERCETIN DIHYDRATE	ncit:C75768	QUERCETIN DIHYDRATE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	REVERSETRIIODOTHYRONINE	iuphar.ligand:2636	RT3	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	GNF-PF-3964	chembl:CHEMBL599088	CHEMBL:CHEMBL599088	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.026775967	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2187819634820604	1,5-NAPHTHALENEDIAMINE	chembl:CHEMBL538965	CHEMBL:CHEMBL538965	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	P-HYDROXYCINNAMALDEHYDE	chembl:CHEMBL431836	P-HYDROXYCINNAMALDEHYDE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.028536778	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	GNF-PF-1319	chembl:CHEMBL235891	CHEMBL:CHEMBL235891	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.008475815	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1286952726365061	5-HYDROXYINDOLACETIC ACID	iuphar.ligand:11900	5-HYDROXYINDOLEACETIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.2210849315187137	SORBINIL	ncit:C97357	SORBINIL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	TCMDC-124055	chembl:CHEMBL546576	CHEMBL:CHEMBL546576	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	TDR78277	chembl:CHEMBL1308346	CHEMBL:CHEMBL1308346	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	MECARBAM	chembl:CHEMBL1417951	MECARBAM	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1025540453822158	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	1,2,3,4,5,6-HEXABROMO-CYCLOHEXANE	chembl:CHEMBL444236	CHEMBL:CHEMBL444236	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	DTC	9/2/20	NULL	1.093909817410302	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NSC-747259	chembl:CHEMBL561679	CHEMBL:CHEMBL561679	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1909369863116163	GALUTEOLIN	chembl:CHEMBL233929	GALUTEOLIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004762601	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.2419708351875322	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	chembl:CHEMBL1333512	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	TOSUFLOXACIN TOSYLATE	ncit:C76234	TOSUFLOXACIN TOSYLATE	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.00915725	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.030386384	SKF-38393	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	ZAPA	chembl:CHEMBL20562	ZAPA	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008176218	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007149737	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	DTC	9/2/20	NULL	2.917092846427472	AZD-6538	iuphar.ligand:6440	AZD6538	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	ISOFENPHOS	ncit:C163668	ISOFENPHOS	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1033615575505797	ALLITRIDIN	chembl:CHEMBL123040	ALLITRIDIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	2'-HYDROXYCHALCONE	chembl:CHEMBL32147	2'-HYDROXYCHALCONE	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.0191914	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	SPERMIDINE	rxcui:1483262	SPERMIDINE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	MMV006587	chembl:CHEMBL597857	CHEMBL:CHEMBL597857	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	QUERCETIN DIHYDRATE	ncit:C75768	QUERCETIN DIHYDRATE	FALSE	FALSE	FALSE
CAMK1D	hgnc:19341	CAMK1D	DTC	9/2/20	NULL	0.1151484018326633	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002170994	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.057574201	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.072927321	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00908123	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	PANTOPRAZOLE	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	SB-200646	chembl:CHEMBL85194	CHEMBL:CHEMBL85194	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	RS-100329	iuphar.ligand:7381	RS-100329	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2628011573358083	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	OBTUSAQUINONE	chembl:CHEMBL1333653	OBTUSAQUINONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.009423487	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FENBUCONAZOLE	chembl:CHEMBL1879687	FENBUCONAZOLE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002858494	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	PHENYLSTIBONIC ACID	chembl:CHEMBL1369257	PHENYLSTIBONIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.020721259	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	GNF-PF-2671	chembl:CHEMBL578878	CHEMBL:CHEMBL578878	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.008746905	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	chembl:CHEMBL284028	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.091159151	SK&F-82958	iuphar.ligand:10742	SKF-82958	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.02646556	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.029465584	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001432522	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	GNF-PF-4798	chembl:CHEMBL584635	CHEMBL:CHEMBL584635	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	0.6403374540938354	ALLYL ISOTHIOCYANATE	iuphar.ligand:2420	ALLYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000260261	chembl:CHEMBL602552	CHEMBL:CHEMBL602552	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1293292394967844	GNF-PF-1399	chembl:CHEMBL578504	CHEMBL:CHEMBL578504	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.007758226	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001244081	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	2.019525817	NSC-640556	chembl:CHEMBL1983317	CHEMBL:CHEMBL1983317	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.014537008	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	SJ000120081	chembl:CHEMBL606532	CHEMBL:CHEMBL606532	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	1,2-DIPHENYLDISULFANE	chembl:CHEMBL462861	CHEMBL:CHEMBL462861	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004287741	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.035216413	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.07631929	CCG-63802	iuphar.ligand:8724	CCG-63802	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.022249013	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.099446347	GW0742	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2273059360852575	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.212152207	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	MAPROTILINE HYDROCHLORIDE	rxcui:203126	MAPROTILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	SKF-38393	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	OXICONAZOLE NITRATE	rxcui:32638	OXICONAZOLE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	3,4-DIMETHOXYDALBERGIONE	chembl:CHEMBL1591258	3,4-DIMETHOXYDALBERGIONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	TANSHINONE IIA SULFONATE	chembl:CHEMBL1473252	TANSHINONE IIA SULFONATE	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.006173741	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.061773731	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ANETHOLTRITHION	rxcui:820	ANETHOLE TRITHIONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.050048162	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
PSMB11	hgnc:31963	PSMB11	DTC	9/2/20	NULL	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA6	hgnc:9535	PSMA6	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB5	hgnc:9542	PSMB5	DTC	9/2/20	NULL	0.4273880216858854	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB3	hgnc:9540	PSMB3	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB10	hgnc:9538	PSMB10	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CYP24A1	hgnc:2602	CYP24A1	DTC	9/2/20	NULL	0.9723642821424906	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.043611023	IUPHAR.LIGAND:7940	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.002680057	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.03043923	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.015184405	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	7-METHOXYISOFLAVONE	chembl:CHEMBL563919	CHEMBL:CHEMBL563919	FALSE	FALSE	FALSE
LAT	hgnc:18874	LAT	DTC	9/2/20	NULL	35.00511415712966	TRIDOLGOSIR	ncit:C152742	TRIDOLGOSIR	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.1110098757625676	IUPHAR.LIGAND:10097	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	2-ETHYLANTHRAQUINONE	chembl:CHEMBL42355	CHEMBL:CHEMBL42355	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.044573575	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	HARMALOL HYDROCHLORIDE	chembl:CHEMBL486816	HARMALOL HYDROCHLORIDE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.305277158	PENICILLIOL A	chembl:CHEMBL457041	PENICILLIOL A	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.062509132	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	NOLATREXED	ncit:C143088	NOLATREXED	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	TCMDC-125185	chembl:CHEMBL580819	CHEMBL:CHEMBL580819	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	CYSTAMINE	rxcui:1426401	CYSTAMINE	FALSE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	0.5250767123569451	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.032173818	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-1000163A	chembl:CHEMBL1096290	GSK-1000163A	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1483267549030917	GALLAMINE	rxcui:4638	GALLAMINE	FALSE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	DTC	9/2/20	NULL	3.750547945	BERKELEYDIONE	chembl:CHEMBL400514	BERKELEYDIONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	ZAPA	chembl:CHEMBL20562	ZAPA	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.051885051	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.7395446652914718	2-PYRIDYLCARBOXALDEHYDE P-NITROBENZOYL HYDRAZONE	chembl:CHEMBL255067	CHEMBL:CHEMBL255067	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	CHLORDANE	iuphar.ligand:2831	CHLORDANE	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.6908904109959803	HTS-05057	chembl:CHEMBL372629	CHEMBL:CHEMBL372629	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	inhibitor	0.041021618	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.02321294	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	3-MORPHOLINOSYDNONIMINE HCL	chembl:CHEMBL538104	CHEMBL:CHEMBL538104	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.005585922	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	BERBERINE	rxcui:1437	BERBERINE	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:8974	iuphar.ligand:8974	OMIPALISIB	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	PROPANTHELINE	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.1058622403945453	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2386712328895204	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.007561589	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00551957	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.023759127	IUPHAR.LIGAND:4903	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.010966514	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007003824	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	0.1944728564284981	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:12088	iuphar.ligand:12088	DALMELITINIB	FALSE	FALSE	FALSE
SAP130	hgnc:29813	SAP130	DTC	9/2/20	NULL	35.00511415712966	SPLICEOSTATIN-A	chembl:CHEMBL1221944	CHEMBL:CHEMBL1221944	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.192335792	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.3251536612259921	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1458546423213736	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:3048	drugbank:DB04714	ISOPENTENYL PYROPHOSPHATE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.010620484	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	BW-28C51	iuphar.ligand:6600	BW284C51	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.1029562181092049	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	2.692701089009974	CID 27456	iuphar.ligand:9741	CID2745687	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.075333818	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.1260688385010672	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003531589	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.069089041	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6341	iuphar.ligand:6341	CFMTI	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.058931169	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1363835616511545	SPERMIDINE	rxcui:1483262	SPERMIDINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.047561296	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012977675	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:7678	iuphar.ligand:7678	AZD8529	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.007804351	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003378437	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	CID 660258	chembl:CHEMBL259805	CHEMBL:CHEMBL259805	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.049723174	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	BIOALLETHRIN S-CYCLOPENTENYL ISOMER	chembl:CHEMBL1887350	BIOALLETHRIN S-CYCLOPENTENYL ISOMER	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.017608206	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:3323	iuphar.ligand:3323	VU0155041	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.015286076	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.063568609	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.2966535098061835	GNF-PF-2307	chembl:CHEMBL421088	CHEMBL:CHEMBL421088	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.012683012	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	0.7501095890813498	TCMDC-125620	chembl:CHEMBL530291	CHEMBL:CHEMBL530291	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	SB-222200	iuphar.ligand:2131	SB 222200	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	BERGAPTOL	chembl:CHEMBL242711	BERGAPTOL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.036463661	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	NANDROLONE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.010594768	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	1,5-NAPHTHALENEDIAMINE	chembl:CHEMBL538965	CHEMBL:CHEMBL538965	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.305277158	MK-912	iuphar.ligand:12577	MK-912	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.525076712	DIHYDRODAPHNODORIN B	chembl:CHEMBL1532097	DIHYDRODAPHNODORIN B	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	0.8751278539282416	IUPHAR.LIGAND:1426	iuphar.ligand:1426	MPEP	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.076208521	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	EBASTINE	rxcui:23796	EBASTINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	GNF-PF-3350	chembl:CHEMBL600747	CHEMBL:CHEMBL600747	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	DNDI1417719	chembl:CHEMBL1420370	CHEMBL:CHEMBL1420370	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	4,4'-DIMETHOXYDALBERGIONE	chembl:CHEMBL1436980	4,4'-DIMETHOXYDALBERGIONE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.004543365	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	ARSANILIC ACID	ncit:C29883	ARSANILIC ACID	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6235	iuphar.ligand:6235	COMPOUND 11 [PMID: 20638279]	FALSE	FALSE	FALSE
SETD7	hgnc:30412	SETD7	DTC	9/2/20	NULL	17.50255707856483	EOSIN	drugbank:DB13706	EOSIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	CYCLOVALONE	ncit:C81040	CYCLOVALONE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.002069839	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
CDC42	hgnc:1736	CDC42	DTC	9/2/20	NULL	8.751278539282415	ZU-4194738	chembl:CHEMBL554475	CHEMBL:CHEMBL554475	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.5801952622728673	EDGEWORIN	chembl:CHEMBL259025	EDGEWORIN	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.006402594	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	GNF-PF-4876	chembl:CHEMBL585444	CHEMBL:CHEMBL585444	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	GNF-PF-2413	chembl:CHEMBL578515	CHEMBL:CHEMBL578515	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006489639	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00347273	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.5556367326528517	KERACYANIN	rxcui:28165	KERACYANIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	SB-200646	chembl:CHEMBL85194	CHEMBL:CHEMBL85194	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.074443768	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.028977744	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
STK36	hgnc:17209	STK36	DTC	9/2/20	NULL	1.458546423213736	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9731	iuphar.ligand:9731	BENZODROCORTISONE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.052824619	SJ000071854	chembl:CHEMBL602127	CHEMBL:CHEMBL602127	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	GNF-PF-5183	chembl:CHEMBL577660	CHEMBL:CHEMBL577660	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.1187956362798518	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.013749063	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.1151484018326633	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.023080295	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	DNDI1417719	chembl:CHEMBL1420370	CHEMBL:CHEMBL1420370	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	modulator	2.500365296937833	IUPHAR.LIGAND:8545	iuphar.ligand:8545	XAP044	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.729273212	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
PAK7	hgnc:15916	PAK5	DTC	9/2/20	inhibitor	1.312691780892362	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.001308407	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	TCMDC-124354	chembl:CHEMBL546344	CHEMBL:CHEMBL546344	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1902451856365742	TRIFLUPROMAZINE HYDROCHLORIDE	rxcui:91125	TRIFLUPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.038608582	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	BENOXATHIAN HYDROCHLORIDE	chembl:CHEMBL544713	BENOXATHIAN HYDROCHLORIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-122400	chembl:CHEMBL2059067	CHEMBL:CHEMBL2059067	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.032472277	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002258977	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	GNF-PF-4791	chembl:CHEMBL583555	CHEMBL:CHEMBL583555	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.023039786	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:1378	iuphar.ligand:1378	LY341495	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00517215	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	inhibitor	0.025739055	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	HYDROXYTYROSOL	rxcui:1314227	HYDROXYTYROSOL	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1060761035064535	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	PSB-1115	iuphar.ligand:3286	PSB1115	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.028536778	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.072927321	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002542744	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2097	hgnc:3464	ESB3	GuideToPharmacology	2024.1	inhibitor	2.019525816757481	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	AG-126	chembl:CHEMBL77387	CHEMBL:CHEMBL77387	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	DIHYDREXIDINE HYDROCHLORIDE	chembl:CHEMBL1256832	DIHYDREXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	EUPARIN	chembl:CHEMBL503938	EUPARIN	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.364636606	CYCLOFENIL	rxcui:2983	CYCLOFENIL	TRUE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.06466462	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-2094	chembl:CHEMBL578928	CHEMBL:CHEMBL578928	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.036413087	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	R(-)-APOCODEINE HCL	chembl:CHEMBL1256735	CHEMBL:CHEMBL1256735	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.024041974	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.012070729	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	GW0742	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
NCBIGENE:3023	ncbigene:3023	H4F3	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10917	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-4325	chembl:CHEMBL598263	CHEMBL:CHEMBL598263	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	ACRISORCIN	rxcui:89729	ACRISORCIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	chembl:CHEMBL1333512	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	KARANJIN	chembl:CHEMBL208484	KARANJIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	E-FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.8468979231563628	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:8056	iuphar.ligand:8056	SCH772984	FALSE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.023780648	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	LINTITRIPT	ncit:C66017	LINTITRIPT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	PIFEXOLE	ncit:C76774	PIFEXOLE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PROCYMIDONE	chembl:CHEMBL513678	PROCYMIDONE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.034118045	RS-17053	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002042305	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.027093742	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.035358701	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.0191914	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ACLARUBICIN HYDROCHLORIDE	ncit:C95830	ACLARUBICIN HYDROCHLORIDE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	MMV007363	chembl:CHEMBL601528	CHEMBL:CHEMBL601528	FALSE	FALSE	FALSE
NCBIGENE:2103	hgnc:3473	ESRRB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8179	iuphar.ligand:8179	PF-03715455	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.089298761	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
TACR3	hgnc:11528	TACR3	DTC	9/2/20	NULL	11.66837138570988	GSK256471	chembl:CHEMBL479463	CHEMBL:CHEMBL479463	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.036413087	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.2651902587661338	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
MAP2K6	hgnc:6846	MAP2K6	DTC	9/2/20	NULL	0.8751278539282416	VX-745	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	TCMDC-124278	chembl:CHEMBL534423	CHEMBL:CHEMBL534423	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-4384	chembl:CHEMBL602763	CHEMBL:CHEMBL602763	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.049349315	IUPHAR.LIGAND:2866	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	DTC	9/2/20	NULL	2.386712328895204	LY-411575	chembl:CHEMBL392068	CHEMBL:CHEMBL392068	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	ACEPROMAZINE	rxcui:155	ACEPROMAZINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	SERTACONAZOLE NITRATE	rxcui:236601	SERTACONAZOLE NITRATE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.173866461	MIRIPIRIUM	chembl:CHEMBL1393904	MIRIPIRIUM	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.016067219	IUPHAR.LIGAND:2768	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	TG100-115	drugbank:DB05552	TG100-115	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	DAMNACANTHAL	ncit:C1480	DAMNACANTHAL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002188184	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.073540156	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	RHETSININE	chembl:CHEMBL508030	RHETSININE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00158739	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.012713722	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	ALDISIN	chembl:CHEMBL357047	ALDISIN	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:7687	iuphar.ligand:7687	AZD6703	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9915	ncit:C90996	PAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:5273	iuphar.ligand:5273	SP600125	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:9915	ncit:C90996	PAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:5273	iuphar.ligand:5273	SP600125	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	DTC	9/2/20	NULL	0.03140411	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	N-(4-NITROPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1574420	CHEMBL:CHEMBL1574420	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00399693	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	PUTRESCINE DIHYDROCHLORIDE	chembl:CHEMBL1528028	PUTRESCINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003874533	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CYAZOFAMID	chembl:CHEMBL1863429	CYAZOFAMID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	KINETIN RIBOSIDE	chembl:CHEMBL411066	KINETIN RIBOSIDE	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	inhibitor	0.1093909817410302	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.066803653	METHYLTESTOSTERONE	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.025663573	IUPHAR.LIGAND:6038	drugbank:DB04338	SB220025	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	MECETRONIUM	ncit:C87264	MECETRONIUM	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	NSC-102042	chembl:CHEMBL273103	CHEMBL:CHEMBL273103	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.01439355	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9453	iuphar.ligand:9453	COMPOUND 12 [PMID: 27448772]	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.015498132	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.025087277	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.025644772	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.031189588	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.040766825	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:2070	hgnc:3522	EYA4	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8173	iuphar.ligand:8173	CEP-1347	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	GNF-PF-1319	chembl:CHEMBL235891	CHEMBL:CHEMBL235891	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.036770078	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.015791781	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.003973038	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	GNF-PF-1339	chembl:CHEMBL600353	CHEMBL:CHEMBL600353	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	JNK INHIBITOR VIII	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.729273212	SQ-22536	chembl:CHEMBL64239	CHEMBL:CHEMBL64239	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.02302968	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	TYRPHOSTIN AG-1478	iuphar.ligand:4862	AG1478	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	5,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484662	CHEMBL:CHEMBL484662	FALSE	FALSE	FALSE
NCBIGENE:2068	hgnc:3434	ERCC2	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:9989	iuphar.ligand:9989	COMPOUND 11 [PMID: 26431428]	FALSE	FALSE	FALSE
EGR1	hgnc:3238	EGR1	DTC	9/2/20	NULL	52.50767123569449	GENIPIN	chembl:CHEMBL459016	GENIPIN	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.042481935	QUINPIROLE	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DINITRO CRESOL	chembl:CHEMBL419564	DINITRO CRESOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	MAHANIMBINE	chembl:CHEMBL495873	MAHANIMBINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	THIAMINE CHLORIDE	chembl:CHEMBL1588	THIAMINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	SAPPANONE A DIMETHYL ETHER	chembl:CHEMBL1489223	SAPPANONE A DIMETHYL ETHER	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	TANGERETIN	chembl:CHEMBL73930	TANGERETIN	FALSE	FALSE	FALSE
FPR1	hgnc:3826	FPR1	DTC	9/2/20	NULL	3.500511415712966	AG-22	chembl:CHEMBL1290365	CHEMBL:CHEMBL1290365	FALSE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	DTC	9/2/20	NULL	0.1325951293830669	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	GRAVEOLINE	chembl:CHEMBL1371756	GRAVEOLINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ANDROSTENEDIOL	ncit:C95979	ANDROSTENEDIOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	AMINOPURVALANOL	iuphar.ligand:5927	AMINOPURVALANOL A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	DEOXYSAPPANONE B TRIMETHYL ETHER	chembl:CHEMBL1482446	DEOXYSAPPANONE B TRIMETHYL ETHER	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.008016438	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	DTC	9/2/20	NULL	0.5834185692854944	SNC-80	iuphar.ligand:1611	SNC80	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1141471113819445	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	SJ000044417	chembl:CHEMBL609438	CHEMBL:CHEMBL609438	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006397133	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
EPHB1	hgnc:3392	EPHB1	DTC	9/2/20	inhibitor	0.021878196	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	TCMDC-125293	chembl:CHEMBL548629	CHEMBL:CHEMBL548629	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.3409589041278863	OXOGLAUCINE	iuphar.ligand:12559	OXOGLAUCINE	FALSE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	3.750547945	TRIPHENYL PHOSPHATE	chembl:CHEMBL454511	TRIPHENYL PHOSPHATE	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.2419708351875322	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DEXAMETHASONE DIPROPIONATE	ncit:C77417	DEXAMETHASONE DIPROPIONATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	5-FLUOROURIDINE	drugbank:DB01629	5-FLUOROURIDINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CROCIN	rxcui:2262278	CROCIN	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.9907107780319716	CID 646303	chembl:CHEMBL505807	CHEMBL:CHEMBL505807	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006381584	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.03233231	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	GRAVEOLINE	chembl:CHEMBL1371756	GRAVEOLINE	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.1000146118775133	CCT018159	chembl:CHEMBL399530	CHEMBL:CHEMBL399530	FALSE	FALSE	FALSE
MERTK	hgnc:7027	MERTK	DTC	9/2/20	inhibitor	0.2625383561784725	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.7001022831425933	CHLORHEXIDINE DIACETATE	rxcui:133054	CHLORHEXIDINE DIACETATE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.032412143	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.004251633	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	GW0742	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1274458039701322	3-METHYLCHOLANTHRENE	chembl:CHEMBL40583	3-METHYLCHOLANTHRENE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	ROBUSTIC ACID	chembl:CHEMBL400777	ROBUSTIC ACID	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	SJ000089001	chembl:CHEMBL591618	CHEMBL:CHEMBL591618	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.046549354	NSC-3323	chembl:CHEMBL1270169	CHEMBL:CHEMBL1270169	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.043976274	HEMATOXYLIN	drugbank:DB16871	HEMATOXYLIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011049594	MONTELUKAST	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	TCMDC-123749	chembl:CHEMBL524376	CHEMBL:CHEMBL524376	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124919	chembl:CHEMBL546168	CHEMBL:CHEMBL546168	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.4234489615781814	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.015123177	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
BMP2K	hgnc:18041	BMP2K	DTC	9/2/20	inhibitor	0.2625383561784725	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-125539	chembl:CHEMBL533388	CHEMBL:CHEMBL533388	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.006452952	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	CHLORPYRIFOS	ncit:C163641	CHLORPYRIFOS	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE	chembl:CHEMBL460508	CHEMBL:CHEMBL460508	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	DNDI1417413	chembl:CHEMBL1343568	CHEMBL:CHEMBL1343568	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	QUINPIROLE	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
NOD1	hgnc:16390	NOD1	DTC	9/2/20	NULL	52.50767123569449	TRACHEAL CYTOTOXIN	chembl:CHEMBL1765916	TRACHEAL CYTOTOXIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.001996565	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.016491103	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1215455352678113	MIGALASTAT	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
F12	hgnc:3530	F12	DTC	9/2/20	NULL	0.2035181055647073	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.2169738480813822	CLODRONIC ACID	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.006793592	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	CARBOXYMETHYL-TRIMETHYL-ARSONIUM	chembl:CHEMBL2448348	CARBOXYMETHYL-TRIMETHYL-ARSONIUM	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.016206071	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	ALDOSTERONE	rxcui:1312358	ALDOSTERONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	FOSPIRATE	chembl:CHEMBL1873189	FOSPIRATE	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.023274677	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.069454592	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.008418738	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.525076712	MMV006587	chembl:CHEMBL597857	CHEMBL:CHEMBL597857	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.030386384	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.03070624	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	BISINDOLYLMALEIMIDE IX	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.026830696	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.069638821	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	2.763561643983921	1,3-BIS(3-NITROPHENYL)UREA	chembl:CHEMBL1443422	CHEMBL:CHEMBL1443422	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	CCG-63802	iuphar.ligand:8724	CCG-63802	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	SJ000112730	chembl:CHEMBL591178	CHEMBL:CHEMBL591178	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.016206071	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004427291	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.105947682	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.3621218705909966	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.040452751	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.099446347	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	PIRETANIDE	rxcui:33770	PIRETANIDE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.7778914257139925	CHOLESTAN-3BETA,5ALPHA,6BETA-TRIOL	chembl:CHEMBL1278089	CHOLESTAN-3BETA,5ALPHA,6BETA-TRIOL	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	LORECLEZOLE	ncit:C66036	LORECLEZOLE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	chembl:CHEMBL1333512	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	FDA	10-Apr-24	NULL	0.4861821410712453	Lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
PROC	hgnc:9451	PROC	FDA	10-Apr-24	NULL	1.750255707856483	Lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.1215455352678113	Meloxicam	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.022305723	Ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.078252863	Ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.081030357	Lesinurad	rxcui:1731031	LESINURAD	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.023744802	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.05553429	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.039126432	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.2827336143460473	Nitrofurantoin	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	MyCancerGenome	20-Jun-17	inhibitor	0.2941606231691568	AZD8931	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.053445395	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	0.1852122442176172	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.05348829	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.4605936073306534	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	MyCancerGenome	20-Jun-17	inhibitor	0.652269208	SAR302503	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.0504235	MLN0128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.3281729452230906	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.035719504	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.08572681	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3C3	hgnc:8974	PIK3C3	MyCancerGenome	20-Jun-17	inhibitor	0.093763699	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.025244073	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.084146909	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.108040476	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.2500365296937833	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.2500365296937833	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.08334551	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.047712559	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.060492709	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2917092846427472	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
AKT2	hgnc:392	AKT2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.097236428	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.055563673	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.010939098	SIMVASTIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.033338204	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3431873936973496	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1363835616511545	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.075768645	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1894216134043813	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.150021918	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.09753747	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
ABCA1	hgnc:29	ABCA1	NCI	14-Sep-17	NULL	0.01160647	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.012822386	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.037398626	ANTHRACYCLINES	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.1495945049449985	ANTIFOLATES	ncit:C511	FOLATE ANTAGONIST	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.018193926	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.049864835	LONAFARNIB	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.089756703	GINKGO BILOBA	rxcui:236809	GINKGO BILOBA EXTRACT	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	NCI	14-Sep-17	NULL	0.078276194	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.100976291	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
ALDH1A2	hgnc:15472	ALDH1A2	NCI	14-Sep-17	NULL	0.4616059009731384	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	NCI	14-Sep-17	NULL	0.052824619	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.020458863	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.06714536	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	0.1018248310970158	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.045421861	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	2.386712328895204	ST 638	ncit:C1235	ST 638	FALSE	FALSE	FALSE
ANXA5	hgnc:543	ANXA5	NCI	14-Sep-17	NULL	0.057700738	DNR	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.1902451856365742	3TC	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.9053046764774912	LUTEIN	rxcui:11359	LUTEIN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.009927712	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.040656346	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.018560506	12-O-TETRADECANOYLPHORBOL-13-ACETATE	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
BCL2L2	hgnc:995	BCL2L2	NCI	14-Sep-17	NULL	0.1526385791735305	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.053361455	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.034151331	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.1013661606866689	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.1351548809155585	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
BHLHB2	hgnc:1046	BHLHE40	NCI	14-Sep-17	NULL	0.5770073762164231	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.039778539	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
BLK	hgnc:1057	BLK	NCI	14-Sep-17	NULL	0.075768645	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
BTF3L1	hgnc:1126	BTF3P11	NCI	14-Sep-17	NULL	0.3201687270469177	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.069824031	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
CALR	hgnc:1455	CALR	NCI	14-Sep-17	NULL	0.5707355569097228	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
CARTPT	hgnc:24323	CARTPT	NCI	14-Sep-17	NULL	0.3559842117674203	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CEL	hgnc:1848	CEL	NCI	14-Sep-17	NULL	1.071585127259071	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	NCI	14-Sep-17	NULL	0.088396753	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	3.889457128569962	CARDIOPROTECTIVE AGENT	ncit:C2079	CARDIOPROTECTIVE AGENT	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	FAA	ncit:C1101	MITOFLAXONE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	FLAVONE ACETIC ACID	ncit:C1101	MITOFLAXONE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.053854022	ETANERCEPT	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NCBIGENE:2071	hgnc:3435	ERCC3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8195	iuphar.ligand:8195	COMPOUND 8 [PMID: 24044867]	FALSE	FALSE	FALSE
CYP11B2	hgnc:2592	CYP11B2	NCI	14-Sep-17	NULL	1.250182648468916	METOCLOPRAMIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.1770916399180253	PROPYLENE GLYCOL	rxcui:34693	PROPYLENE GLYCOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.004319308	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.08854582	LUTEIN	rxcui:11359	LUTEIN	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.1767935058440892	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.059030547	GREEN TEA EXTRACT	rxcui:283567	GREEN TEA LEAF EXTRACT	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.035418328	GINKGO BILOBA	rxcui:236809	GINKGO BILOBA EXTRACT	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.031555091	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1162960603226899	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.8751278539282416	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.2035181055647073	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.028397875	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	4.773424657790408	NM-3	drugbank:DB12818	NM-3	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	NCI	14-Sep-17	NULL	0.009023487	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
EPHB1	hgnc:3392	EPHB1	NCI	14-Sep-17	NULL	0.029665351	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.040640612	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	NCI	14-Sep-17	NULL	2.386712328895204	MACROLIDES	ncit:C261	MACROLIDE ANTIBIOTIC	FALSE	FALSE	FALSE
EVI1	hgnc:3498	MECOM	NCI	14-Sep-17	NULL	1.419126249613364	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
NCBIGENE:2072	hgnc:3436	ERCC4	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9989	iuphar.ligand:9989	COMPOUND 11 [PMID: 26431428]	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.069638821	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.1508841127462485	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.086007651	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.08780547	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.2375912725597036	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.596678082	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.3535870116881784	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.097236428	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	NCI	14-Sep-17	NULL	0.046590658	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.105015342	5-AZADEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.041182487	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1628	hgnc:2697	DBP	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	DIDEMNIN B	ncit:C1364	DIDEMNIN B	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	2.059124362184098	R24	ncit:C2349	MONOCLONAL ANTIBODY R24	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	2.059124362184098	L-778,123	ncit:C1840	FARNESYLTRANSFERASE/GERANYLGERANYLTRANSFERASE INHIBITOR L-778,123	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	1.029562181092049	HEPATITIS B VACCINE	ncit:C29091	HEPATITIS B VACCINE	FALSE	FALSE	FALSE
IRS1	hgnc:6125	IRS1	NCI	14-Sep-17	NULL	1.640864726115453	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.1715936968486748	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.050294704	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.072927321	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	2.917092846427472	RECOMBINANT C5A	ncit:C388	RECOMBINANT C5A	FALSE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	NCI	14-Sep-17	NULL	0.596678082	DOLASETRON	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.1539814405738841	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:9655	iuphar.ligand:9655	TAKINIB	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.325124899	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.049629179	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.096167896	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.022593662	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
MT1G	hgnc:7399	MT1G	NCI	14-Sep-17	NULL	9.546849315580818	BSO	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.035598421	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	1.200175343	5-AZADEOXYCYTIDINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1071585127259071	4-HYDROXY-TAMOXIFEN	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
NME1	hgnc:7849	NME1	NCI	14-Sep-17	NULL	2.625383561784724	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.098605955	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NRIP1	hgnc:8001	NRIP1	NCI	14-Sep-17	NULL	0.8655110643246345	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PAPPA	hgnc:8602	PAPPA	NCI	14-Sep-17	NULL	2.386712328895204	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
PCSK1	hgnc:8743	PCSK1	NCI	14-Sep-17	NULL	4.375639269641208	CALCITONIN	rxcui:1311287	CALCITONIN	TRUE	FALSE	FALSE
PDHX	hgnc:21350	PDHX	NCI	14-Sep-17	NULL	2.500365296937833	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
NCBIGENE:1648	hgnc:2725	GADD45AP1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.033658764	ICI 182,780	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.042516333	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.010770804	STI571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PPIA	hgnc:9253	PPIA	NCI	14-Sep-17	NULL	0.4310974649892816	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
PZP	hgnc:9750	PZP	NCI	14-Sep-17	NULL	1.750255707856483	NORETHISTERONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.3125456621172291	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.028184472	12-O-TETRADECANOYLPHORBOL-13-ACETATE	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:6464	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
RTN4	hgnc:14085	RTN4	NCI	14-Sep-17	NULL	4.200613698855561	HYPERBARIC OXYGEN	ncit:C2351	HYPERBARIC OXYGEN	FALSE	FALSE	FALSE
RNASEH2A	hgnc:18518	RNASEH2A	NCI	14-Sep-17	NULL	0.4449802647092754	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
SAG	hgnc:10521	SAG	NCI	14-Sep-17	NULL	0.4375639269641209	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
SILV	hgnc:10880	PMEL	NCI	14-Sep-17	NULL	2.500365296937833	HMBA	ncit:C1125	HEXAMETHYLENE BISACETAMIDE	FALSE	FALSE	FALSE
SERPINH1	hgnc:1546	SERPINH1	NCI	14-Sep-17	NULL	17.50255707856483	11D10	ncit:C2446	MONOCLONAL ANTIBODY 11D10	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.4412409347537352	RECOMBINANT INTERLEUKIN	ncit:C593	RECOMBINANT INTERLEUKIN	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.3860858179095183	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.5385402178019948	GREEN TEA EXTRACT	rxcui:283567	GREEN TEA LEAF EXTRACT	TRUE	FALSE	FALSE
SLPI	hgnc:11092	SLPI	NCI	14-Sep-17	NULL	1.009762908	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.1521961485092594	12-O-TETRADECANOYLPHORBOL-13-ACETATE	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.2500365296937833	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.076934317	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:10827	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
SRI	hgnc:11292	SRI	NCI	14-Sep-17	NULL	0.4039051633514962	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.8751278539282416	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.084758146	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.123644438	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10028	iuphar.ligand:10028	MJN110	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	NCI	14-Sep-17	NULL	0.077217164	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.033243223	VCR	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	1.666910197958555	DENSPM	ncit:C1168	DIETHYLNORSPERMINE	FALSE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	NCI	14-Sep-17	NULL	0.8678953923255289	MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	OncoKB	23-Jul-20	NULL	0.4861821410712453	GDC-0077	ncit:C132166	INAVOLISIB	FALSE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.084553416	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
NPPA-AS1	hgnc:37635	NPPA-AS1	PharmGKB	4/5/24	NULL	1.944728564284981	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.4375639269641208	astemizole	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.046673486	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	0.091317689	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
SPOPL	hgnc:27934	SPOPL	PharmGKB	4/5/24	NULL	1.381780822	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	0.7343730242754476	arachidonic acid	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
COL22A1	hgnc:22989	COL22A1	PharmGKB	4/5/24	NULL	8.078103267029924	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.1065064325267636	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
PAPPA2	hgnc:14615	PAPPA2	PharmGKB	4/5/24	NULL	8.078103267029924	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
CAMK4	hgnc:1464	CAMK4	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1447	iuphar.ligand:1447	ME36	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.1553481397505754	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.011365297	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.042619863	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	PharmGKB	4/5/24	NULL	0.076765601	encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.051885051	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003037935	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CXCL12	hgnc:10672	CXCL12	PharmGKB	4/5/24	NULL	0.3860858179095184	fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00133485	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
HFE	hgnc:4886	HFE	PharmGKB	4/5/24	NULL	0.4526523382387457	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	PharmGKB	4/5/24	NULL	0.012486961	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	PharmGKB	4/5/24	NULL	4.699760697022038	selpercatinib	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8812	iuphar.ligand:8812	COMPOUND 30 [PMID: 15953724]	FALSE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.502465753	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	1.032937794800547	etonogestrel	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	PharmGKB	4/5/24	NULL	0.1331836936859721	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.081030357	lesinurad	rxcui:1731031	LESINURAD	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.004191225	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.1491695205559502	telmisartan	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.4102161815288632	dolutegravir	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.018031481	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.01439355	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.2734774543525755	levofloxacin	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.086361301	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NUP62	hgnc:8066	NUP62	PharmGKB	4/5/24	NULL	1.842374429322614	afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	1.166837138570989	cannabidiol	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.018046974	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
ARF1	hgnc:652	ARF1	PharmGKB	4/5/24	NULL	1.842374429322614	afatinib	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
SLC15A1	hgnc:10920	SLC15A1	PharmGKB	4/5/24	NULL	2.333674277141978	cannabidiol	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	PharmGKB	4/5/24	NULL	0.1096651446025365	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
CD96	hgnc:16892	CD96	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.064111931	boceprevir	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.074797252	aliskiren	rxcui:325646	ALISKIREN	TRUE	FALSE	FALSE
REV3L	hgnc:9968	REV3L	PharmGKB	4/5/24	NULL	0.9723642821424907	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NPPA	hgnc:7939	NPPA	PharmGKB	4/5/24	NULL	2.917092846427472	chlorthalidone	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.005059761	primidone	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.026927011	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	0.1613138901250215	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ORM2	hgnc:8499	ORM2	PharmGKB	4/5/24	NULL	1.265245090016735	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.089756703	terazosin	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.100976291	IUPHAR.LIGAND:336	drugbank:DB02152	K-252A	FALSE	FALSE	FALSE
ACSS2	hgnc:15814	ACSS2	PharmGKB	4/5/24	NULL	0.253049018	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.1779921058837101	nitrendipine	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
AREG	hgnc:651	AREG	PharmGKB	4/5/24	NULL	0.3889457128569963	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NECTIN4	hgnc:19688	NECTIN4	PharmGKB	4/5/24	NULL	4.118248724368196	enfortumab vedotin	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TMEM131L	hgnc:29146	TMEM131L	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.009838424	eletriptan	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
SLC22A6	hgnc:10970	SLC22A6	PharmGKB	4/5/24	NULL	1.312691780892362	pantoprazole	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	PharmGKB	4/5/24	NULL	4.861821410712453	ofatumumab	rxcui:712566	OFATUMUMAB	TRUE	TRUE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:7391	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	PharmGKB	4/5/24	NULL	0.1061833594250647	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.053361455	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.074690855	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.1795134059339982	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	PharmGKB	4/5/24	NULL	0.089756703	anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.092118721	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
CYP51A1	hgnc:2649	CYP51A1	PharmGKB	4/5/24	NULL	1.207072901969988	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:3264	iuphar.ligand:3264	AFDX384	FALSE	FALSE	FALSE
SUMO4	hgnc:21181	SUMO4	PharmGKB	4/5/24	NULL	3.750547945406749	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
CPS1	hgnc:2323	CPS1	PharmGKB	4/5/24	NULL	0.2631963470460877	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	0.1405827877796372	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	PharmGKB	4/5/24	NULL	0.4054646427466756	serotonin	rxcui:1311214	SEROTONIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.5983780197799943	terodiline	rxcui:37815	TERODILINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.1105424657593568	IUPHAR.LIGAND:343	iuphar.ligand:343	BRUCINE N-OXIDE	FALSE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	3.182283105193605	glucose	rxcui:349730	ANHYDROUS DEXTROSE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.4817217544559128	remifentanil	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.003740928	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
YEATS4	hgnc:24859	YEATS4	PharmGKB	4/5/24	NULL	3.424413341458336	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.018081154	methylphenobarbital	rxcui:6758	MEPHOBARBITAL	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	0.011715232	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.070010228	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.2409837027645336	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
ERICH3	hgnc:25346	ERICH3	PharmGKB	4/5/24	NULL	5.000730593875666	serotonin	rxcui:1311214	SEROTONIN	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.021215221	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
AKR1C3	hgnc:386	AKR1C3	PharmGKB	4/5/24	NULL	0.076934317	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MAN1B1	hgnc:6823	MAN1B1	PharmGKB	4/5/24	NULL	1.154014752432846	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:3264	iuphar.ligand:3264	AFDX384	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.017409705	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.017709164	flecainide	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.06466462	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.2386712328895204	flecainide	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1166837138570989	flecainide	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
SLCO4C1	hgnc:23612	SLCO4C1	PharmGKB	4/5/24	NULL	0.2333674277141977	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.5527123287967841	IUPHAR.LIGAND:354	rxcui:3267	DEXETIMIDE	FALSE	FALSE	FALSE
FASLG	hgnc:11936	FASLG	PharmGKB	4/5/24	NULL	0.009211872	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.2386712328895204	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:313	iuphar.ligand:313	MUSCARINIC TOXIN 3	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.025003653	eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.013442824	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.020446912	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.2651902587661338	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.4150804050252529	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.016365177	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	1.186614039224734	perindopril	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.2685814385457519	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:291	iuphar.ligand:291	NNC 11-1314	FALSE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.08780547	oxazepam	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	4.200613699	dasabuvir	rxcui:1597381	DASABUVIR	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.1744440904840349	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
PPCDC	hgnc:28107	PPCDC	PharmGKB	4/5/24	NULL	0.3163112725041837	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
LIPC	hgnc:6619	LIPC	PharmGKB	4/5/24	NULL	1.458546423213736	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
ZNF613	hgnc:25827	ZNF613	PharmGKB	4/5/24	NULL	2.692701089009974	anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
PSORS1C1	hgnc:17202	PSORS1C1	PharmGKB	4/5/24	NULL	0.2258394461750301	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	PharmGKB	4/5/24	NULL	0.043430663	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SLC25A31	hgnc:25319	SLC25A31	PharmGKB	4/5/24	NULL	0.760980743	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
AKR1A1	hgnc:380	AKR1A1	PharmGKB	4/5/24	NULL	52.50767123569449	daunorubicinol	ncit:C1062	DUBORIMYCIN	FALSE	FALSE	FALSE
GNMT	hgnc:4415	GNMT	PharmGKB	4/5/24	NULL	7.001022831425934	l-methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	PharmGKB	4/5/24	NULL	0.1355619739303644	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	1.981421556063943	BIIB022	ncit:C71530	ANTI-IGF-1R RECOMBINANT MONOCLONAL ANTIBODY BIIB022	FALSE	TRUE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.2465148884304905	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1584738568481725	BRIVANIB	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
KIF11	hgnc:6388	KIF11	TALC	12-May-16	inhibitor	6.563458904461812	SB-743921	drugbank:DB05546	SB-743921	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.1405827877796372	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
UNIPROT:Q08289	hgnc:1402	CACNB2	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	AMLODIPINE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	ALOSETRON	rxcui:85248	ALOSETRON	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:7770	iuphar.ligand:7770	[125I]SD6	FALSE	FALSE	FALSE
UNIPROT:P63027	hgnc:12643	VAMP2	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	BOTULINUM TOXIN TYPE B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TdgClinicalTrial	Jan-14	NULL	2.100306849	ANAVEX 2-73	ncit:C171846	BLARCAMESINE	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	1.514644363	APD125	ncit:C83996	NELOTANSERIN	FALSE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.087512785	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.028382525	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.061773731	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	1.413668071730236	AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.2465148884304905	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.0296486	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	BAZEDOXIFENE	rxcui:1441386	BAZEDOXIFENE	TRUE	FALSE	FALSE
UNIPROT:P31639	hgnc:11037	SLC5A2	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	DAPAGLIFLOZIN	rxcui:1486966	DAPAGLIFLOZIN PROPANEDIOL	TRUE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.007714909	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	2.838252499226729	BVT.115959	chembl:CHEMBL3545409	BVT.115959	FALSE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	0.8899605294185507	OLMESARTAN	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.1458546423213736	IUPHAR.LIGAND:198	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.13086024	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.3818739726232327	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	RALOXIFEN	chembl:CHEMBL1079109	RALOXIFEN	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.041508041	ETILEVODOPA	rxcui:1421444	ETILEVODOPA	FALSE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.6364566210387211	EXENATIDE	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:1629	iuphar.ligand:1629	NALORPHINE	FALSE	FALSE	FALSE
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	0.276356164	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	FOSPROPOFOL	rxcui:828682	FOSPROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	1.211715490054488	FROVATRIPTAN	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.2027323213733378	FLIBANSERIN	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
UNIPROT:P30872	hgnc:11330	SSTR1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	LANREOTIDE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
UNIPROT:P62942	hgnc:3711	FKBP1A	TdgClinicalTrial	Jan-14	NULL	0.5373592085524291	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.2885036881082115	IUPHAR.LIGAND:1613	iuphar.ligand:1613	[LEU]ENKEPHALIN	FALSE	FALSE	FALSE
UNIPROT:P30939	hgnc:5292	HTR1F	TdgClinicalTrial	Jan-14	NULL	14.32027397337122	LASMIDITAN	rxcui:2256930	LASMIDITAN	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1625	ncit:C80578	ETORPHINE	FALSE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	1.019566431761058	MB07811	drugbank:DB05192	MB07811	FALSE	FALSE	FALSE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	2.019525817	PEGAPTANIB	rxcui:498509	PEGAPTANIB	TRUE	FALSE	FALSE
UNIPROT:P41231	hgnc:8541	P2RY2	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
NCBIGENE:3144	ncbigene:3144	HMAB	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11155	iuphar.ligand:11155	COMPOUND 5 [STECULA ET AL., 2020]	FALSE	FALSE	FALSE
UNIPROT:P43657	hgnc:15520	LPAR6	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.035982643	MDV3100	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.1223955040459079	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.2347585897273971	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.2273059360852575	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	0.5770073762164231	MOSAPRIDE	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.031536139	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P31350	hgnc:10452	RRM2	TdgClinicalTrial	Jan-14	NULL	1.154014752432846	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:11880	iuphar.ligand:11880	PALTIMATRECTINIB	FALSE	FALSE	FALSE
UNIPROT:P15309	hgnc:125	ACP3	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	MVA-BN	rxcui:2464823	MODIFIED VACCINIA ANKARA-BAVARIAN NORDIC	TRUE	FALSE	FALSE
UNIPROT:P07288	hgnc:6364	KLK3	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	MVA-BN	rxcui:2464823	MODIFIED VACCINIA ANKARA-BAVARIAN NORDIC	TRUE	FALSE	FALSE
UNIPROT:P30939	hgnc:5292	HTR1F	TdgClinicalTrial	Jan-14	NULL	1.060761035064535	NARATRIPTAN	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.2243917574174978	NERAMEXANE	ncit:C76781	NERAMEXANE	FALSE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	0.4487835148349957	NARATRIPTAN	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.061197752	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
NCBIGENE:1251	hgnc:7872	NOS1	GuideToPharmacology	2024.1	NULL	0.7395446652914718	IUPHAR.LIGAND:12316	iuphar.ligand:12316	ZZL-7	FALSE	FALSE	FALSE
UNIPROT:P25024	hgnc:6026	CXCR1	TdgClinicalTrial	Jan-14	NULL	3.750547945	PA-401	chembl:CHEMBL4298068	CANOCTAKIN	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.075442056	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.4605936073306534	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	3.088686543276147	PF-3512676	ncit:C28580	AGATOLIMOD SODIUM	FALSE	FALSE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.8140724222588294	PF-00610355	drugbank:DB11871	PF-00610355	FALSE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	0.1406455479527531	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	PLASMIN	rxcui:4388	PLASMIN	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.1426838892274307	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:1251	hgnc:7872	NOS1	GuideToPharmacology	2024.1	inhibitor	0.7395446652914718	IUPHAR.LIGAND:5113	iuphar.ligand:5113	3-BROMO-7NI	FALSE	FALSE	FALSE
UNIPROT:Q9Y243	hgnc:393	AKT3	TdgClinicalTrial	Jan-14	NULL	0.546954909	RX-0201	ncit:C88335	ARCHEXIN	FALSE	FALSE	FALSE
UNIPROT:P07101	hgnc:11782	TH	TdgClinicalTrial	Jan-14	NULL	1.500219178	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:O14695	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.105947682	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
UNIPROT:P41594	hgnc:4597	GRM5	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	STX107	chembl:CHEMBL3642985	STX107	FALSE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.3697723326457359	TAFA-93	drugbank:DB05887	TAFA-93	FALSE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	1.166837138570988	TM38837	iuphar.ligand:8705	TM38837	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:12396	iuphar.ligand:12396	CZS-241	FALSE	FALSE	FALSE
UNIPROT:P49146	hgnc:7957	NPY2R	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	OBINEPITIDE	ncit:C175168	OBINEPITIDE	FALSE	FALSE	FALSE
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	0.138178082	TRAFERMIN	ncit:C152708	TRAFERMIN	FALSE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	FILGRASTIM	rxcui:1433764	TBO-FILGRASTIM	TRUE	FALSE	FALSE
NCBIGENE:470	ncbigene:470	ATHS	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3996	iuphar.ligand:3996	MUSCARINE	FALSE	FALSE	FALSE
UNIPROT:Q99973	hgnc:11726	TEP1	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	V934/V935	ncit:C80055	HTERT VACCINE V934/V935	FALSE	FALSE	FALSE
UNIPROT:Q13324	hgnc:2358	CRHR2	TdgClinicalTrial	Jan-14	NULL	7.501095891	UROCORTIN 2	iuphar.ligand:3545	UROCORTIN 2	FALSE	FALSE	FALSE
UNIPROT:Q01668	hgnc:1391	CACNA1D	TdgClinicalTrial	Jan-14	NULL	0.081407242	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278864	IUPHAR.LIGAND:10316	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
UNIPROT:P16422	hgnc:11529	EPCAM	TdgClinicalTrial	Jan-14	NULL	6.300920548	VB6-845	ncit:C71694	CITATUZUMAB BOGATOX	FALSE	FALSE	FALSE
UNIPROT:P28074	hgnc:9542	PSMB5	TdgClinicalTrial	Jan-14	NULL	0.4273880216858854	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:Q9UHF5	hgnc:5982	IL17B	TdgClinicalTrial	Jan-14	NULL	10.50153425	VIDOFLUDIMUS	ncit:C152873	VIDOFLUDIMUS	FALSE	FALSE	FALSE
NCBIGENE:470	ncbigene:470	ATHS	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:4008	iuphar.ligand:4008	&ALPHA;-CONOTOXIN RGIA	FALSE	FALSE	FALSE
UNIPROT:Q02127	hgnc:2867	DHODH	TdgClinicalTrial	Jan-14	NULL	1.658136986390352	VIDOFLUDIMUS	ncit:C152873	VIDOFLUDIMUS	FALSE	FALSE	FALSE
UNIPROT:Q08289	hgnc:1402	CACNB2	TdgClinicalTrial	Jan-14	NULL	0.1458546423213736	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:Q02641	hgnc:1401	CACNB1	TdgClinicalTrial	Jan-14	NULL	0.1666910197958555	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	CARBINOXAMINE	rxcui:20220	CARBINOXAMINE	TRUE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:7700	iuphar.ligand:7700	AZD1332	FALSE	FALSE	FALSE
UNIPROT:P08123	hgnc:2198	COL1A2	TdgClinicalTrial	Jan-14	NULL	0.6250913242344583	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.029260335	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:3987	iuphar.ligand:3987	TC-2559	FALSE	FALSE	FALSE
UNIPROT:P02461	hgnc:2201	COL3A1	TdgClinicalTrial	Jan-14	NULL	2.812910959055062	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P02452	hgnc:2197	COL1A1	TdgClinicalTrial	Jan-14	NULL	0.8036888454443035	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:4011	iuphar.ligand:4011	&ALPHA;-CONOTOXIN TXIA	FALSE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.3231241306811969	DAPIPRAZOLE	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P03886	hgnc:7455	MT-ND1	TdgClinicalTrial	Jan-14	NULL	0.3500511415712967	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	0.4487835148349958	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.044611445	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	1.479089330582943	DEZOCINE	rxcui:22713	DEZOCINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.040703621	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	blocker	0.1325951293830669	IUPHAR.LIGAND:356	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.1653584607713247	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
UNIPROT:O75762	hgnc:497	TRPA1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
UNIPROT:P14780	hgnc:7176	MMP9	TdgClinicalTrial	Jan-14	NULL	0.42006137	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
UNIPROT:P49286	hgnc:7464	MTNR1B	TdgClinicalTrial	Jan-14	NULL	1.086365611772989	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2713574740862764	METIPRANOLOL	rxcui:10824	METIPRANOLOL	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	5.000730593875666	METOCURINE	rxcui:29950	METOCURINE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.0701037	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.1396480617970598	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	NEPAFENAC	rxcui:298665	NEPAFENAC	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.108711535	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	0.729273212	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
UNIPROT:O00555	hgnc:1388	CACNA1A	TdgClinicalTrial	Jan-14	NULL	0.4118248724368196	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.056826484	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.087903467	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3988	iuphar.ligand:3988	PNU-282987	FALSE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	NITROPRUSSIDE	rxcui:7476	NITROPRUSSIDE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.060984519	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.075732218	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	0.8078103267029924	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.192335792	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.07767407	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.073885091	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.076934317	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:467	hgnc:785	ATF3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3970	iuphar.ligand:3970	&ALPHA;-CONOTOXIN MII	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.087318744	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.2864054794674245	TENOXICAM	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
UNIPROT:P16473	hgnc:12373	TSHR	TdgClinicalTrial	Jan-14	NULL	0.9309870786470656	THYROTROPIN ALFA	rxcui:4952	THYROTROPIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.052229116	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
UNIPROT:Q9NPF7	hgnc:15488	IL23A	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	USTEKINUMAB	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10700	iuphar.ligand:10700	SUVN-911	FALSE	FALSE	FALSE
UNIPROT:Q9UNQ0	hgnc:74	ABCG2	TEND	1-Aug-11	NULL	0.01864619	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	TRIMEPRAZINE	rxcui:10825	TRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:O43497	hgnc:1394	CACNA1G	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	TRIMETHADIONE	rxcui:10827	TRIMETHADIONE	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	blocker	0.1508841127462485	IUPHAR.LIGAND:3990	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.2386712328895204	CLOCORTOLONE	rxcui:21249	CLOCORTOLONE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1293292394967845	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.069638821	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TEND	1-Aug-11	NULL	1.458546423213736	ENOXAPARIN	rxcui:221095	ENOXAPARIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	blocker	0.3125456621172291	IUPHAR.LIGAND:3990	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:2089	iuphar.ligand:2089	NEUROKININ A	FALSE	FALSE	FALSE
UNIPROT:P20701	hgnc:6148	ITGAL	TEND	1-Aug-11	NULL	2.414145803939977	EFALIZUMAB	rxcui:356988	EFALIZUMAB	TRUE	TRUE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	0.8975670296699915	ELETRIPTAN	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TEND	1-Aug-11	NULL	6.563458904461812	CHORIOGONADOTROPIN ALFA	rxcui:283550	CHORIOGONADOTROPIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	1.032937794800547	ETONOGESTREL	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:3824	iuphar.ligand:3824	[3H]LEU-N/OFQ	FALSE	FALSE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TEND	1-Aug-11	NULL	2.763561643983921	FLUDROCORTISONE	rxcui:4452	FLUDROCORTISONE	TRUE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TEND	1-Aug-11	NULL	1.795134059339982	ISOCARBOXAZID	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.020465128	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	1.211715490054488	FROVATRIPTAN	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TEND	1-Aug-11	NULL	1.640864726115453	LERCANIDIPINE	rxcui:135056	LERCANIDIPINE	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TEND	1-Aug-11	NULL	0.3977853881492007	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1479	iuphar.ligand:1479	NEUROPEPTIDE FF	FALSE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.1658136986390352	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.08914715	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.048844345	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.2713574740862764	METIPRANOLOL	rxcui:10824	METIPRANOLOL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.047049885	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TEND	1-Aug-11	NULL	3.500511415712966	NABILONE	rxcui:31447	NABILONE	TRUE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1688	iuphar.ligand:1688	[3H]N/OFQ	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.077217164	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TEND	1-Aug-11	NULL	1.084869240406911	MONTELUKAST	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.09814518	NORGESTIMATE	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:1498	iuphar.ligand:1498	[125I][TYR11]DES-BR-NPB-23	FALSE	FALSE	FALSE
UNIPROT:O60896	hgnc:9845	RAMP3	TEND	1-Aug-11	NULL	5.000730593875666	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
UNIPROT:O00555	hgnc:1388	CACNA1A	TEND	1-Aug-11	NULL	0.4039051633514961	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.2047082699247349	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.096967075	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.080103236	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.040640612	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.06502498	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.057574201	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:3797	iuphar.ligand:3797	[125I]NPFF	FALSE	FALSE	FALSE
UNIPROT:P23415	hgnc:4326	GLRA1	TEND	1-Aug-11	NULL	0.1290114772375786	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.072125922	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TEND	1-Aug-11	NULL	0.7095631248066824	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9168	iuphar.ligand:9168	NCGC 84	FALSE	FALSE	FALSE
UNIPROT:O14788	hgnc:11926	TNFSF11	TEND	1-Aug-11	NULL	43.75639269641208	DENOSUMAB	rxcui:993449	DENOSUMAB	TRUE	FALSE	TRUE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:1572	iuphar.ligand:1572	JMV458	FALSE	FALSE	FALSE
EPHRIN TYPE-A RECEPTOR 3	hgnc:3387	EPHA3	TTD	2020.06.01	NULL	11.66837138570988	KB-004	chembl:CHEMBL2109398	KB-004	FALSE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	5.834185692854944	RG7882	ncit:C147031	ANTI-MUC16/MMAE ANTIBODY-DRUG CONJUGATE DMUC4064A	FALSE	FALSE	FALSE
ASPARTYL AMINOPEPTIDASE	hgnc:2981	DNPEP	TTD	2020.06.01	NULL	13.12691780892362	QGC-001	drugbank:DB13107	QGC-001	FALSE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	AMG 673	ncit:C175778	EMERFETAMAB	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	4.039051633514961	BI 894999	ncit:C160257	AMREDOBRESIB	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:11648	rxcui:2591497	DARIDOREXANT	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 4	hgnc:1605	CCR4	TTD	2020.06.01	NULL	3.088686543276147	FLX475	drugbank:DB15570	FLX475	FALSE	FALSE	FALSE
EXTRACELLULAR SIGNAL-REGULATED KINASE 2	hgnc:6871	MAPK1	TTD	2020.06.01	NULL	0.08572681	LY3214996	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.1750255707856483	PCM-075	ncit:C143162	ONVANSERTIB	FALSE	FALSE	TRUE
CDC7-RELATED KINASE	hgnc:1745	CDC7	TTD	2020.06.01	NULL	4.039051633514961	TAK-931	ncit:C126641	SIMUROSERTIB	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9415	iuphar.ligand:9415	COMPOUND 11 [PMID: 15261275]	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:11695	iuphar.ligand:11695	HTL6641	FALSE	FALSE	FALSE
AMINOPEPTIDASE	hgnc:7032	MFAP1	TTD	2020.06.01	NULL	2.625383561784725	CHR-2797	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	0.6961244292611014	TPX-0005	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
JUN N TERMINAL KINASE	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	0.5147810905460245	BGP-15	chembl:CHEMBL4747845	BGP-15	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-21	hgnc:3678	FGF21	TTD	2020.06.01	NULL	17.50255707856483	BMS-986036	ncit:C174833	PEGBELFERMIN	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:11403	iuphar.ligand:11403	JH112	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	0.546954909	BI-505	chembl:CHEMBL2109482	BI-505	FALSE	FALSE	FALSE
DUAL SPECIFICITY PROTEIN KINASE TTK	hgnc:10416	RPS27	TTD	2020.06.01	NULL	2.500365296937833	BAY1161909	ncit:C116074	EMPESERTIB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.073954467	Altiratinib	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.4089382494991783	JNJ-42756493	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	DP-4088	chembl:CHEMBL30054	DPOC-4088	FALSE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	2.625383561784724	CARD-024	chembl:CHEMBL4297361	1.ALPHA.-HYDROXYVITAMIN D5	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:11448	iuphar.ligand:11448	DANAVOREXTON	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	2.333674277141977	ADL-5747	chembl:CHEMBL4297345	ADL-5747	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.596678082	Bicifadine	ncit:C79930	BICIFADINE	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	2.423430980108977	GSK933776	chembl:CHEMBL2109300	GSK933776	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	5.250767123569449	RO-4995819	chembl:CHEMBL3301593	DECOGLURANT	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8132	iuphar.ligand:8132	IL-94	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.2386712328895204	Nabumetone	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
ADENINE NUCLEOTIDE TRANSLOCATOR 1	hgnc:10990	SLC25A4	TTD	2020.06.01	NULL	0.502465753	Clodronate	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
DIHYDROTHYMINE DEHYDROGENASE	hgnc:3012	DPYD	TTD	2020.06.01	NULL	0.074927706	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1383601350084176	Droperidol	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:9541	iuphar.ligand:9541	5-BDBD	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.5357925636295356	Danaparoid	rxcui:78484	DANAPAROID	TRUE	FALSE	FALSE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	0.8334550989792776	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.2	hgnc:6256	KCNJ10	TTD	2020.06.01	NULL	7.501095891	Glisoxepide	ncit:C72801	GLISOXEPIDE	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	0.2302968036653267	Aldosterone	rxcui:1312358	ALDOSTERONE	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	1.479089330582943	Dezocine	rxcui:22713	DEZOCINE	TRUE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	3.000438356	GV1001	ncit:C62756	TERTOMOTIDE	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.048958202	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.3977853881492006	Pindolol	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.084689792	Ralfinamide	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	0.276356164	TKI258	ncit:C62435	DOVITINIB LACTATE	FALSE	FALSE	FALSE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	1.071585127259071	Ramatroban	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.005152357	Ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	1.129197231	Pegsunercept	ncit:C90875	PEGSUNERCEPT	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.4449802647092754	Pratosartan	ncit:C72935	PRATOSARTAN	FALSE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	3.889457128569962	MLN-2704	chembl:CHEMBL2109556	MLN-2704	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.4375639269641208	Pegamotecan	ncit:C174957	PEGAMOTECAN	FALSE	FALSE	FALSE
IMMUNOGLOBULIN GAMMA FC RECEPTOR IIA	hgnc:3616	FCGR2A	TTD	2020.06.01	NULL	2.917092846427472	SM-101	chembl:CHEMBL4298105	VALZIFLOCEPT	FALSE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR	hgnc:6008	IL2RA	TTD	2020.06.01	NULL	0.8579684842433742	Denileukin diftitox	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
ALKALINE PHOSPHATASE TISSUE-NONSPECIFIC	hgnc:438	ALPL	TTD	2020.06.01	NULL	0.2476776945079929	Levamisole	rxcui:6371	LEVAMISOLE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	1.640864726115453	ICARIIN	rxcui:1788871	ICARIIN	FALSE	FALSE	FALSE
PROTEIN KINASE C BETA	hgnc:9395	PRKCB	TTD	2020.06.01	NULL	0.6563458904461813	Sotrastaurin acetate	ncit:C80631	SOTRASTAURIN ACETATE	FALSE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.2128689374420047	Solifenacin	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	1.346350544504987	Clorgyline	drugbank:DB04017	CLORGILINE	FALSE	FALSE	FALSE
INTEGRIN ALPHA-L	hgnc:6148	ITGAL	TTD	2020.06.01	NULL	2.414145803939977	Efalizumab	rxcui:356988	EFALIZUMAB	TRUE	TRUE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	4.200613699	CTCE-9908	drugbank:DB05625	CTCE-9908	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.013836014	Phentolamine	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.5509279467829125	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	2.692701089009974	CX157	drugbank:DB05205	CX157	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	0.039778539	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
INTEGRIN ALPHA-V	hgnc:6150	ITGAV	TTD	2020.06.01	NULL	8.078103267029922	IMGN-388	chembl:CHEMBL2109633	IMGN-388	FALSE	FALSE	FALSE
AURORA KINASE C	hgnc:11391	AURKC	TTD	2020.06.01	NULL	0.8751278539282416	AMG 900	ncit:C82349	AURORA KINASE INHIBITOR AMG 900	FALSE	FALSE	FALSE
ONCOTROPHOBLAST GLYCOPROTEIN 5T4	hgnc:12004	TPBG	TTD	2020.06.01	NULL	10.50153424713889	TroVax	ncit:C49087	RECOMBINANT MODIFIED VACCINIA ANKARA-5T4 VACCINE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.064268875	Remimazolam	rxcui:2383941	REMIMAZOLAM	TRUE	FALSE	FALSE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	4.375639269641208	Emepepimut-S	ncit:C2195	EMEPEPIMUT-S	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.1704794520639431	TG02	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	SGN-CD33A	ncit:C111039	VADASTUXIMAB TALIRINE	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	1.029562181092049	RG7116	chembl:CHEMBL3707404	LUMRETUZUMAB	FALSE	FALSE	FALSE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	2.692701089009974	Topiroxostat	ncit:C96311	TOPIROXOSTAT	FALSE	FALSE	FALSE
PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9	hgnc:20001	PCSK9	TTD	2020.06.01	NULL	2.019525817	PF-04950615	iuphar.ligand:7730	BOCOCIZUMAB	FALSE	FALSE	FALSE
ONCOTROPHOBLAST GLYCOPROTEIN 5T4	hgnc:12004	TPBG	TTD	2020.06.01	NULL	21.00306849427779	Naptumomab estafenatox	ncit:C95789	NAPTUMOMAB ESTAFENATOX	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	2.423430980108977	Solanezumab	ncit:C88585	SOLANEZUMAB	FALSE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR ALPHA	hgnc:11765	TGFA	TTD	2020.06.01	NULL	6.563458904461812	LY3016859	chembl:CHEMBL4594573	FEPIXNEBART	FALSE	FALSE	FALSE
GALECTIN-3	hgnc:6563	LGALS3	TTD	2020.06.01	NULL	26.25383561784724	GR-MD-02	ncit:C115111	BELAPECTIN	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	2.625383561784724	GSK2245035	drugbank:DB16076	GSK2245035	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.6482428547616604	Dasotraline	ncit:C166750	DASOTRALINE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.3271505995993426	Dasotraline	ncit:C166750	DASOTRALINE	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.3977853881492006	Dasotraline	ncit:C166750	DASOTRALINE	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	2.493675356344019	PF-06463922	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
TRANSTHYRETIN	hgnc:12405	TTR	TTD	2020.06.01	NULL	8.751278539282415	Patisiran	rxcui:2053490	PATISIRAN	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2A	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.2616661357260523	MOXONIDINE	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Talipexole	ncit:C152496	TALIPEXOLE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	BRL 35135	iuphar.ligand:13194	BRL35135	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-5	hgnc:4079	GABRA5	TTD	2020.06.01	NULL	0.2983390411119005	RG-1662	ncit:C167009	BASMISANIL	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.3302369260106572	4SC-202	drugbank:DB13101	4SC-202	FALSE	FALSE	FALSE
CHOLESTERYL ESTER TRANSFER PROTEIN	hgnc:1869	CETP	TTD	2020.06.01	NULL	2.692701089009974	Dalcetrapib	ncit:C81529	DALCETRAPIB	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	Bb21217	ncit:C140310	AUTOLOGOUS ANTI-BCMA-CAR-4-1BB-CD3ZETA-EXPRESSING MEMORY T-LYMPHOCYTES BB21217	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 4	hgnc:1605	CCR4	TTD	2020.06.01	NULL	1.544343271638073	ATLCAR.CD30.CCR4 cells	ncit:C155293	AUTOLOGOUS CCR4-CD30CAR-CD28-CD3ZETA-EXPRESSING T-LYMPHOCYTES	FALSE	FALSE	FALSE
PANCREATIC ELASTASE 1	hgnc:3308	CELA1	TTD	2020.06.01	NULL	2.917092846427472	Erdosteine	rxcui:24305	ERDOSTEINE	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.4303907478335614	ONAPRISTONE	ncit:C170255	ONAPRISTONE	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV1.5	hgnc:6224	KCNA5	TTD	2020.06.01	NULL	3.500511415712966	BMS-394136	drugbank:DB12067	BMS-394136	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1389091831632129	Cipatinib	drugbank:DB16752	CIPATINIB	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.1260688385010672	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.061628722	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	0.078840347	Clotrimazole	rxcui:2623	CLOTRIMAZOLE	TRUE	FALSE	FALSE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	3.500511415712966	Alosetron	rxcui:85248	ALOSETRON	TRUE	FALSE	FALSE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	10.50153424713889	Almitrine	rxcui:528	ALMITRINE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.016927038	Aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	Argatroban	rxcui:15202	ARGATROBAN	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.064318974	Bicalutamide	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.1250182648468916	Buprenorphine	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	1.750255707856483	Cerivastatin	rxcui:596723	CERIVASTATIN	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	1.158257453728555	Edrophonium	rxcui:1546421	EDROPHONIUM CATION	TRUE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	13.12691780892362	Fendrix	wikidata:Q29005860	FENDRIX	FALSE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	0.084553416	Guggulsterone	iuphar.ligand:2745	GUGGULSTERONE	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.4243044140258141	Granisetron	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	0.7501095890813498	Repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
ARYL HYDROCARBON RECEPTOR	hgnc:348	AHR	TTD	2020.06.01	NULL	0.2187819634820604	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1A	hgnc:7463	MTNR1A	TTD	2020.06.01	NULL	7.501095891	Ramelteon	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	2.386712328895204	Tolvaptan	rxcui:358257	TOLVAPTAN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M4	hgnc:1953	CHRM4	TTD	2020.06.01	NULL	0.5303805175322677	Tropicamide	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	2.917092846427472	TOCOTRIENOL	rxcui:578285	TOCOTRIENOLS	FALSE	FALSE	FALSE
THYROTROPIN RECEPTOR	hgnc:12373	TSHR	TTD	2020.06.01	NULL	0.9309870786470656	Thyrotropin Alfa	rxcui:4952	THYROTROPIN ALFA	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.2218633995874415	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	1.312691780892362	NKTR-262	ncit:C148289	PEG-CONJUGATED TLR7/8 AGONIST NKTR-262	FALSE	FALSE	FALSE
INTERFERON RECEPTOR	hgnc:5447	IFNR	TTD	2020.06.01	NULL	52.50767123569449	Z-100	ncit:C118445	MYCOBACTERIUM TUBERCULOSIS ARABINOMANNAN Z-100	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1479089330582944	TAK-593	drugbank:DB13093	TAK-593	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	0.6250913242344582	BIIB074	iuphar.ligand:12645	VIXOTRIGINE	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	1.050153425	BGP-15	chembl:CHEMBL4747845	BGP-15	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.4518732464345482	MP470	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	0.49187514	MP470	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
GLYCINAMIDE RIBONUCLEOTIDE FORMYLTRANSFERASE	hgnc:4163	GART	TTD	2020.06.01	NULL	2.561349816375341	PELITREXOL	ncit:C2633	PELITREXOL	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR ALPHA	hgnc:9864	RARA	TTD	2020.06.01	NULL	0.8334550989792776	Tamibarotene	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
BETA-SECRETASE 1	hgnc:933	BACE1	TTD	2020.06.01	NULL	2.019525817	E-2609	iuphar.ligand:9818	ELENBECESTAT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.027505328	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.05751114	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:130	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1117184494376478	IUPHAR.LIGAND:60	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.065716735	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:73	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.079197091	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.037884323	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.034727296	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:62	iuphar.ligand:62	(+)-BUTACLAMOL	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:8424	iuphar.ligand:8424	BF-1	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:154	iuphar.ligand:154	(+)-LSD	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:160	iuphar.ligand:160	AL-37350A	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.012869527	IUPHAR.LIGAND:214	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:254	iuphar.ligand:254	RS 39604	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:101	ncit:C73303	TIOSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:259	iuphar.ligand:259	[3H]GR 113808	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:273	iuphar.ligand:273	ICI 169369	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:262	iuphar.ligand:262	[3H]5-CT	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.1023541349623674	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.053964719	IUPHAR.LIGAND:8170	iuphar.ligand:8170	COMPOUND 8H [PMID: 21561767]	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.025183535	IUPHAR.LIGAND:502	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.025183535	IUPHAR.LIGAND:502	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.094438258	IUPHAR.LIGAND:528	iuphar.ligand:526	RX821002	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.022220766	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:528	iuphar.ligand:526	RX821002	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.090530468	IUPHAR.LIGAND:6943	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:1198	hgnc:2071	CLK3	GuideToPharmacology	2024.1	NULL	17.50255707856483	IUPHAR.LIGAND:4624	iuphar.ligand:4624	[14C]METHYLAMINE	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:12709	iuphar.ligand:12709	JNJ-63576253	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6948	rxcui:4162	ETHYLESTRENOL	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:7865	drugbank:DB06973	BISPHENOL A	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:7930	iuphar.ligand:7930	APELIN RECEPTOR EARLY ENDOGENOUS LIGAND	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:3281	ncit:C96199	DERENOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:3284	iuphar.ligand:3284	PSB603	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1804387327687096	IUPHAR.LIGAND:5619	iuphar.ligand:5619	PSB-10	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:594	iuphar.ligand:3944	CGP42112	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:8159	iuphar.ligand:8159	COMPOUND 25 [PMID: 20855207]	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:589	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6910	iuphar.ligand:6910	LY303336	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:586	iuphar.ligand:586	EXP3174	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:6168	iuphar.ligand:6168	[LEU8]-PHYLLOLITORIN	FALSE	FALSE	FALSE
NCBIGENE:2792	hgnc:4411	GNGT1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:7733	iuphar.ligand:7733	GDC-0152	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:12093	iuphar.ligand:12093	ZANZALINTINIB	FALSE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:7729	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
NCBIGENE:1889	hgnc:3146	ECE1	GuideToPharmacology	2024.1	NULL	10.50153424713889	IUPHAR.LIGAND:5068	iuphar.ligand:5068	APRIL	FALSE	FALSE	FALSE
NCBIGENE:1889	hgnc:3146	ECE1	GuideToPharmacology	2024.1	NULL	3.500511415712966	IUPHAR.LIGAND:5069	iuphar.ligand:5069	BAFF	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.036062961	IUPHAR.LIGAND:551	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:567	iuphar.ligand:567	BRL 37344	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:7207	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:2948	ncit:C1626	ETALOCIB	FALSE	FALSE	FALSE
NCBIGENE:1941	hgnc:18041	BMP2K	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:7792	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
NCBIGENE:1789	hgnc:2979	DNMT3B	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8155	iuphar.ligand:8155	COMPOUND 13A [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:2722	ncbigene:2722	GLC1B	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8302	iuphar.ligand:8302	COMPOUND 1 [PMID: 25719566]	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:7514	iuphar.ligand:7514	GW841819X	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:7524	iuphar.ligand:7524	XD14	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:7524	iuphar.ligand:7524	XD14	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:6004	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4121	iuphar.ligand:4121	A804598	FALSE	FALSE	FALSE
NCBIGENE:2726	hgnc:14310	BRD7	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8572	iuphar.ligand:8572	LP99	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:11178	iuphar.ligand:11178	BIIB068	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1777	iuphar.ligand:1777	MRS2211	FALSE	FALSE	FALSE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:10545	iuphar.ligand:10545	DBRD9	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:12239	iuphar.ligand:12239	JNJ-64264681	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:10428	iuphar.ligand:10428	COMPOUND 25 [PMID: 31260299]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:9176	iuphar.ligand:9176	WZ4002	FALSE	FALSE	TRUE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10094	iuphar.ligand:10094	SOFNOBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3906	iuphar.ligand:3906	R-954	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:10254	iuphar.ligand:10254	NG29	FALSE	FALSE	FALSE
NCBIGENE:2471	hgnc:3881	FRA20A	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8994	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:6203	iuphar.ligand:6203	&ALPHA;.&BETA;-METHYLENE-2-THIO-UDP	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:653	iuphar.ligand:653	B-9430	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11276	iuphar.ligand:11276	ANI9	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.086361301	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1558	hgnc:2622	CYP2C8	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8158	iuphar.ligand:8158	COMPOUND 27 [PMID: 18337095]	FALSE	FALSE	FALSE
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	activator	1.166837138570988	IUPHAR.LIGAND:5242	iuphar.ligand:5242	PETCM	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:6079	iuphar.ligand:6079	CV-3988	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:836	iuphar.ligand:836	CXCL11	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:772	iuphar.ligand:772	CCL8	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:776	iuphar.ligand:776	CCL26	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:9680	iuphar.ligand:9680	GW766994	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:772	iuphar.ligand:772	CCL8	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	modulator	0.729273212	IUPHAR.LIGAND:10585	iuphar.ligand:10585	COMPOUND 39 [PMID: 31742400]	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:12147	iuphar.ligand:12147	TL12-186	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	1.458546423213736	IUPHAR.LIGAND:10545	iuphar.ligand:10545	DBRD9	FALSE	FALSE	FALSE
NCBIGENE:720	hgnc:1323	C4A	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:7821	iuphar.ligand:7821	AZD4619	FALSE	FALSE	FALSE
NCBIGENE:725	hgnc:1328	C4BPB	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:717	hgnc:1248	C2	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:3171	hgnc:5023	FOXA3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11540	iuphar.ligand:11540	SULFOPIN	FALSE	FALSE	FALSE
NCBIGENE:731	hgnc:1352	C8A	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:733	hgnc:1354	C8G	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:727	hgnc:1331	C5	GuideToPharmacology	2024.1	inhibitor	0.087512785	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:731	hgnc:1352	C8A	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:8534	iuphar.ligand:8534	CXCL12H25R (MONOMER)	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8948	iuphar.ligand:8948	AZD5069	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:3660	iuphar.ligand:3660	[125I]CXCL10 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:5662	iuphar.ligand:5662	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:8242	iuphar.ligand:8242	PI-3065	FALSE	FALSE	FALSE
NCBIGENE:1975	hgnc:3285	EIF4B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:5662	iuphar.ligand:5662	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:5974	drugbank:DB03444	6-BROMOINDIRUBIN-3'-OXIME	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.3621218705909966	IUPHAR.LIGAND:10063	iuphar.ligand:10063	CDK12 INHIBITOR 2	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.4412409347537352	IUPHAR.LIGAND:9626	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:8974	iuphar.ligand:8974	OMIPALISIB	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:10063	iuphar.ligand:10063	CDK12 INHIBITOR 2	FALSE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:5137	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.095295229	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.018385039	IUPHAR.LIGAND:5682	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
NCBIGENE:1325	hgnc:2257	CORT	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8777	iuphar.ligand:8777	COMPOUND 51 [CROSIGNANI ET AL., 2011]	FALSE	FALSE	FALSE
NCBIGENE:1325	hgnc:2257	CORT	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10559	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
NCBIGENE:1326	hgnc:6860	MAP3K8	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8777	iuphar.ligand:8777	COMPOUND 51 [CROSIGNANI ET AL., 2011]	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10581	iuphar.ligand:10581	COMPOUND 13E [PMID: 31811124]	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.046466966	IUPHAR.LIGAND:7221	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.4646696569530486	IUPHAR.LIGAND:10675	iuphar.ligand:10675	PN6047	FALSE	FALSE	FALSE
NCBIGENE:3244	ncbigene:3244	HPE1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12817	iuphar.ligand:12817	OICR-8268	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.051629962	IUPHAR.LIGAND:8866	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1610	iuphar.ligand:1610	ETHYLKETOCYCLAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.027333509	IUPHAR.LIGAND:1639	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1604	iuphar.ligand:1604	(-)-CYCLAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1161674142382621	IUPHAR.LIGAND:3828	iuphar.ligand:1640	NALTRIBEN	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	NULL	0.1161674142382621	IUPHAR.LIGAND:10482	iuphar.ligand:10482	COMPOUND 16 [PMID: 31498617]	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1548898856510162	IUPHAR.LIGAND:1633	ncit:C80570	QUADAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.006940869	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.088248187	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.038049037	IUPHAR.LIGAND:214	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:10598	iuphar.ligand:10598	COMPOUND 41 [PMID: 31855425]	FALSE	FALSE	FALSE
NCBIGENE:2834	hgnc:4464	PRLHR	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:8456	rxcui:2637535	MOLIDUSTAT	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:8011	iuphar.ligand:8011	KU-0060648	FALSE	FALSE	TRUE
NCBIGENE:3148	hgnc:5000	HMGB2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12707	iuphar.ligand:12707	PT2385	FALSE	FALSE	FALSE
NCBIGENE:3148	hgnc:5000	HMGB2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11251	iuphar.ligand:11251	BELZUTIFAN	FALSE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8603	iuphar.ligand:8603	COMPOUND 10L [PMID: 24556381]	FALSE	FALSE	FALSE
NCBIGENE:1823	hgnc:3035	DSC1	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8170	iuphar.ligand:8170	COMPOUND 8H [PMID: 21561767]	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9115	iuphar.ligand:9115	CPI-1205	FALSE	FALSE	FALSE
NCBIGENE:1827	hgnc:3040	RCAN1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8170	iuphar.ligand:8170	COMPOUND 8H [PMID: 21561767]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	antibody	0.2500365296937833	IUPHAR.LIGAND:10505	iuphar.ligand:10505	AMIVANTAMAB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:7644	ncit:C2713	PELITINIB	FALSE	FALSE	TRUE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:3141	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:9149	iuphar.ligand:9149	TUG-905	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:3367	iuphar.ligand:3367	COMPOUND B [PMID:18477808]	FALSE	FALSE	FALSE
NCBIGENE:2022	hgnc:3349	ENG	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
NCBIGENE:2985	hgnc:3621	FCGRT	GuideToPharmacology	2024.1	antibody	1.296485709523321	IUPHAR.LIGAND:9777	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.02271093	IUPHAR.LIGAND:5682	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
NCBIGENE:1111	hgnc:1925	CHEK1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:8810	iuphar.ligand:8810	COMPOUND 1L [PMID: 16644217]	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:6485	iuphar.ligand:6485	AMG-837	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	0.1315981735230438	IUPHAR.LIGAND:1049	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:7743	iuphar.ligand:7743	IZORLISIB	FALSE	FALSE	FALSE
NCBIGENE:2023	hgnc:3350	ENO1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:4339	iuphar.ligand:4339	URB597	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.013680998	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:2024	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.106290832	IUPHAR.LIGAND:7816	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1256164383629055	IUPHAR.LIGAND:9786	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
NCBIGENE:1299	hgnc:2219	COL9A3	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:7202	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:11545	iuphar.ligand:11545	FGF-19	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.039068208	IUPHAR.LIGAND:9428	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
NCBIGENE:2609	hgnc:4145	GAPDHP67	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:7974	ncit:C82294	ZOTAROLIMUS	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:8942	ncit:C101519	EDICOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:11565	iuphar.ligand:11565	COMPOUND 13AC [PMID: 33256400]	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	NULL	0.2500365296937833	IUPHAR.LIGAND:5089	iuphar.ligand:5089	VEGFE	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:8914	iuphar.ligand:8914	ONATASERTIB	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:3411	iuphar.ligand:3411	[3H]LXA4	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6241	iuphar.ligand:6241	CGEN-855A	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.3889457128569962	IUPHAR.LIGAND:1022	iuphar.ligand:1022	FMET-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:1041	iuphar.ligand:1041	ISOPROPYLUREIDO-FLFLF	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.105015342	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1023	iuphar.ligand:1023	FMET-MET-TYR-ALA-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:1047	iuphar.ligand:1047	HUMANIN	FALSE	FALSE	FALSE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:9865	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:1046	iuphar.ligand:1046	HP(2-20)	FALSE	FALSE	FALSE
NCBIGENE:232	hgnc:4042	FZD4	GuideToPharmacology	2024.1	modulator	26.25383561784724	IUPHAR.LIGAND:10321	iuphar.ligand:10321	FZM1.8	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6105	iuphar.ligand:6105	GAL-B2	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:5391	iuphar.ligand:5391	[125I][TYR26]GALANIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:3592	iuphar.ligand:3592	GALANIN	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:8784	iuphar.ligand:8784	SGI-1776	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:7978	drugbank:DB07426	[1-HYDROXY-2-(1,1':3',1''-TERPHENYL-3-YLOXY)ETHANE-1,1-DIYL]BIS(PHOSPHONIC ACID)	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.4688184931758437	IUPHAR.LIGAND:4251	iuphar.ligand:4251	LY503430	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:3515	iuphar.ligand:3515	NNC 92-1687	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.2442217266776488	IUPHAR.LIGAND:7062	rxcui:21245	CLOBETASOL PROPIONATE	TRUE	FALSE	FALSE
NCBIGENE:451	hgnc:769	ASS1P6	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:4246	iuphar.ligand:4246	LY339434	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:4240	iuphar.ligand:4240	L701324	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.1693795846312726	IUPHAR.LIGAND:4068	iuphar.ligand:4068	(RS)-(TETRAZOL-5-YL)GLYCINE	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:8126	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4619	iuphar.ligand:4619	[3H]NFPS	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:5584	iuphar.ligand:5584	IN-3	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:9066	ncit:C171663	CENDERITIDE	FALSE	FALSE	FALSE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4952	iuphar.ligand:4952	HS-142-1	FALSE	FALSE	FALSE
NCBIGENE:1720	hgnc:52354	DHFRP3	GuideToPharmacology	2024.1	agonist	0.8751278539282417	IUPHAR.LIGAND:4943	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	0.1630673019742065	IUPHAR.LIGAND:1594	rxcui:7393	NIACIN	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	modulator	2.282942227638891	IUPHAR.LIGAND:5794	iuphar.ligand:5794	COMPOUND 42 [PMID: 22420767]	FALSE	FALSE	FALSE
NCBIGENE:2032	ncbigene:2032	ENUR2	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:9664	iuphar.ligand:9664	BML-281	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:8156	iuphar.ligand:8156	COMPOUND 20 [PMID: 22136433]	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.049256727	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.1829535583125243	IUPHAR.LIGAND:7010	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.2134458180312784	IUPHAR.LIGAND:9664	iuphar.ligand:9664	BML-281	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.016311796	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.100589408	IUPHAR.LIGAND:10104	iuphar.ligand:10104	(S)-DIMETINDENE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:8981	iuphar.ligand:8981	CONESSINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:4024	iuphar.ligand:4024	IMMETHRIDINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:7318	rxcui:10847	TRIPELENNAMINE	TRUE	FALSE	FALSE
NCBIGENE:2945	ncbigene:2945	GSTM5P1	GuideToPharmacology	2024.1	activator	26.25383561784724	IUPHAR.LIGAND:9817	iuphar.ligand:9817	YODA1	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:7346	iuphar.ligand:7346	MK-0249	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:1218	iuphar.ligand:1218	ABT-239	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1261	iuphar.ligand:1261	GT2394	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:9872	iuphar.ligand:9872	COMPOUND 3A [PMID: 18606542]	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:1256	iuphar.ligand:1256	JNJ-5207852	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1264	iuphar.ligand:1264	[123I]IODOPROXYFAN	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:8981	iuphar.ligand:8981	CONESSINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:1226	iuphar.ligand:1226	IMPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:10232	iuphar.ligand:10232	SUVN-G3031	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2958	iuphar.ligand:2958	COMPOUND 9A [PATIL ET AL., 1989]	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.2143170254518142	IUPHAR.LIGAND:731	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:5545	iuphar.ligand:5545	2-ARACHIDONYL GLYCERYL ETHER	FALSE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1867	iuphar.ligand:1867	PROKINETICIN-2	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:10540	iuphar.ligand:10540	CHGB (511-532)	FALSE	FALSE	FALSE
NCBIGENE:2039	hgnc:3382	DMTN	GuideToPharmacology	2024.1	modulator	0.6819178082557728	IUPHAR.LIGAND:5669	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:5912	iuphar.ligand:5912	AG 1024	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:5852	iuphar.ligand:5852	MRE-269	FALSE	FALSE	FALSE
NCBIGENE:666	hgnc:1087	BOK	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:12609	iuphar.ligand:12609	COMPOUND 30 [PMID: 37057760]	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.082300425	IUPHAR.LIGAND:7792	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:10044	ncit:C147125	ABIVERTINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:8136	iuphar.ligand:8136	COMPOUND 2 [PMID: 15546730]	FALSE	FALSE	FALSE
NCBIGENE:2376	hgnc:3888	FRA2D	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10575	iuphar.ligand:10575	DKFZ‐251	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.069089041	IUPHAR.LIGAND:7221	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1618	iuphar.ligand:1618	DYNORPHIN-(1-11)	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.002054853	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0296486	IUPHAR.LIGAND:10476	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:10368	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.009809018	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12764	iuphar.ligand:12764	BI-2493	FALSE	FALSE	FALSE
NCBIGENE:515	hgnc:840	ATP5PB	GuideToPharmacology	2024.1	blocker	0.8751278539282418	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	blocker	0.1640864726115453	IUPHAR.LIGAND:2313	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NCBIGENE:386	hgnc:18866	KCNT2	GuideToPharmacology	2024.1	activator	0.2302968036653267	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.1262203635473425	IUPHAR.LIGAND:2604	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:7656	iuphar.ligand:7656	ICA-105574	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:11864	iuphar.ligand:11864	PF-04885614	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:2589	iuphar.ligand:2589	(3R,4S)-293B	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:2591	iuphar.ligand:2591	IKS124	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:7665	iuphar.ligand:7665	ML213	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:11566	iuphar.ligand:11566	EB-42486	FALSE	FALSE	FALSE
NCBIGENE:254	hgnc:6585	LHCGR	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1160	iuphar.ligand:1160	HCG	FALSE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9839	iuphar.ligand:9839	LIMKI3	FALSE	FALSE	FALSE
NCBIGENE:2055	hgnc:2079	CLN8	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9839	iuphar.ligand:9839	LIMKI3	FALSE	FALSE	FALSE
NCBIGENE:633	hgnc:1044	BGN	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:10484	iuphar.ligand:10484	RJW100	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:2751	iuphar.ligand:2751	24(S), 25-EPOXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:10587	iuphar.ligand:10587	UCM-05194	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:2753	iuphar.ligand:2753	ACETYL-PODOCARPIC DIMER	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:2754	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:2908	iuphar.ligand:2908	VPC32183	FALSE	FALSE	FALSE
NCBIGENE:2669	hgnc:4234	GEM	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8241	iuphar.ligand:8241	GSK-LSD1	FALSE	FALSE	FALSE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:7001	iuphar.ligand:7001	GARCINOL	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1300	iuphar.ligand:1300	P-GUANIDINOBENZOYL-MCH-(7-17)	FALSE	FALSE	FALSE
NCBIGENE:1217	hgnc:26439	SLC47A2	GuideToPharmacology	2024.1	NULL	0.4487835148349957	IUPHAR.LIGAND:4503	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1319	iuphar.ligand:1319	TETRALIN_UREA ANALOGUE (7O)	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:1327	iuphar.ligand:1327	ASIP [90-132 (L89Y)]	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:8293	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6211	iuphar.ligand:6211	A-794282	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:3346	iuphar.ligand:3346	LY456236	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:3347	iuphar.ligand:3347	LY456066	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1374	iuphar.ligand:1374	(S)-4C3HPG	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1406	iuphar.ligand:1406	(R,S)-4-PPG	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:5996	iuphar.ligand:5996	JNK INHIBITOR IX	FALSE	FALSE	FALSE
NCBIGENE:2393	hgnc:3905	FRA5A	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6545	iuphar.ligand:6545	COMPOUND 4 [PMID: 18163548]	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:290	iuphar.ligand:290	MCN-A-343	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:9228	iuphar.ligand:9228	PF-06767832	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:7449	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:10711	iuphar.ligand:10711	T‐495	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:316	rxcui:56092	METHSCOPOLAMINE BROMIDE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:7449	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:10104	iuphar.ligand:10104	(S)-DIMETINDENE	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:6043	drugbank:DB08009	SU-11652	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.054243462	IUPHAR.LIGAND:355	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:304	iuphar.ligand:304	PENTYLTHIO-TZTP	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:322	iuphar.ligand:322	HEXAHYDRODIFENIDOL	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:7449	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:10104	iuphar.ligand:10104	(S)-DIMETINDENE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.085239726	IUPHAR.LIGAND:329	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:327	iuphar.ligand:327	METHOCTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:11499	iuphar.ligand:11499	PCS1055	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:10104	iuphar.ligand:10104	(S)-DIMETINDENE	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.2027323213733378	IUPHAR.LIGAND:1363	iuphar.ligand:1363	LUZINDOLE	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.3547815624033412	IUPHAR.LIGAND:1356	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.064111931	IUPHAR.LIGAND:8866	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:6020	iuphar.ligand:6020	PDGF RECEPTOR TYROSINE KINASE INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1616	iuphar.ligand:1616	DIHYDROMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:9193	iuphar.ligand:9193	ZYKLOPHIN	FALSE	FALSE	FALSE
NCBIGENE:1552	hgnc:7590	MYLK	GuideToPharmacology	2024.1	activator	3.500511415712967	IUPHAR.LIGAND:2351	iuphar.ligand:2351	CALMODULIN	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:8645	iuphar.ligand:8645	GW853606	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:2617	ncit:C87421	ACONITINE	FALSE	FALSE	FALSE
NCBIGENE:585	hgnc:969	BBS4	GuideToPharmacology	2024.1	activator	1.500219178	IUPHAR.LIGAND:2619	iuphar.ligand:2619	BATRACHOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:11023	iuphar.ligand:11023	DS-1971A	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:11864	iuphar.ligand:11864	PF-04885614	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.040546464	IUPHAR.LIGAND:7547	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5759	ncit:C78006	BEFETUPITANT	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:2120	iuphar.ligand:2120	YM44778	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:2090	iuphar.ligand:2090	NEUROKININ B	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12172	iuphar.ligand:12172	EMLENOFLAST	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:10422	rxcui:2637134	FEZOLINETANT	TRUE	FALSE	FALSE
NCBIGENE:1408	hgnc:2385	CRY2	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8820	iuphar.ligand:8820	CCT129957	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:2133	iuphar.ligand:2133	SSR 146977	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:2110	ncit:C170264	OSANETANT	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1470	iuphar.ligand:1470	NEUROMEDIN U-25	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	0.1422972120208523	IUPHAR.LIGAND:8866	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
NCBIGENE:1762	hgnc:2936	DMWD	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8887	iuphar.ligand:8887	ML130	FALSE	FALSE	FALSE
NCBIGENE:3057	ncbigene:3057	HCL2	GuideToPharmacology	2024.1	activator	26.25383561784724	IUPHAR.LIGAND:7573	iuphar.ligand:7573	OMAVELOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:2964	hgnc:4654	GTF2F2P1	GuideToPharmacology	2024.1	blocker	10.50153424713889	IUPHAR.LIGAND:10042	iuphar.ligand:10042	CRAC CHANNEL INHIBITOR 5B [PMID: 26256403]	FALSE	FALSE	FALSE
NCBIGENE:1222	hgnc:13819	SLCO1C1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4547	iuphar.ligand:4546	[3H]TAUROCHOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1222	hgnc:13819	SLCO1C1	GuideToPharmacology	2024.1	inhibitor	0.5966780822238011	IUPHAR.LIGAND:4357	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10676	iuphar.ligand:10676	AZ1366	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.3182283105193605	IUPHAR.LIGAND:11169	ncit:C96858	CARBETOCIN	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.4773424657790409	IUPHAR.LIGAND:2179	iuphar.ligand:2179	[THR4,GLY7]OT	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:2194	iuphar.ligand:2194	L023103	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2254	iuphar.ligand:2254	[MPA1,D-TYR(ET)2,D-TIC7,D-TIC9]OT	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.1060761035064535	IUPHAR.LIGAND:2181	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:1730	iuphar.ligand:1730	4-THIO-UTP	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:6199	iuphar.ligand:6199	MRS2927	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:6201	iuphar.ligand:6201	2-AMINO-URIDINE-5'-MONOPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11452	iuphar.ligand:11452	TIM-38	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:12038	drugbank:DB14942	BMS-986141	FALSE	FALSE	FALSE
NCBIGENE:1256	hgnc:10894	PRMT5	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8288	iuphar.ligand:8288	CMP5 [PMID: 25742700]	FALSE	FALSE	FALSE
NCBIGENE:3179	hgnc:9257	PPID	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:1024	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:985	hgnc:10921	SLC15A2	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:11367	iuphar.ligand:11367	[18F]FEPPG	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:2671	iuphar.ligand:2671	DRF 2519	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:2675	ncit:C83791	IMIGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:2409	hgnc:3920	FRA7B	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10409	iuphar.ligand:10409	ZETOMIPZOMIB	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2697	iuphar.ligand:2697	SB-219994	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2701	iuphar.ligand:2701	AD5075	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2663	iuphar.ligand:2663	AD-5061	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:10702	iuphar.ligand:10702	COMPOUND 15A [PMID: 32069401]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:8917	iuphar.ligand:8917	AMG319	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.2949869170544634	IUPHAR.LIGAND:6024	iuphar.ligand:6024	PI 3-KG INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.036873365	IUPHAR.LIGAND:6004	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.035719504	IUPHAR.LIGAND:7955	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:8917	iuphar.ligand:8917	AMG319	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:9961	iuphar.ligand:9961	COMPOUND 20F [PMID: 28520415]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:11204	iuphar.ligand:11204	AZD8154	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:9961	iuphar.ligand:9961	COMPOUND 20F [PMID: 28520415]	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:8012	iuphar.ligand:8012	PIK-75	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:8969	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.015758605	IUPHAR.LIGAND:7950	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:8969	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
NCBIGENE:1310	hgnc:2196	COL19A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12323	iuphar.ligand:12323	MK-8189	FALSE	FALSE	FALSE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:7148	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.074797252	IUPHAR.LIGAND:2739	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:3453	iuphar.ligand:3453	ORG2058	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:2877	ncit:C66478	PROMEGESTONE	FALSE	FALSE	FALSE
NCBIGENE:2395	hgnc:3951	FXN	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:6565	iuphar.ligand:6565	S 17092	FALSE	FALSE	FALSE
NCBIGENE:1213	hgnc:2092	CLTC	GuideToPharmacology	2024.1	NULL	7.501095891	IUPHAR.LIGAND:6688	iuphar.ligand:6688	[3H]PEMETREXED	FALSE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:5973	iuphar.ligand:5973	G&OUML; 6976	FALSE	FALSE	FALSE
NCBIGENE:1161	hgnc:3439	ERCC8	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4709	iuphar.ligand:4709	INDOLE-3-PROPIONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1798	iuphar.ligand:1798	[ILE5,TRP23]PTHRP-(1-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1797	iuphar.ligand:1797	[ILE5,TRP23,TYR36]PTHRP-(1-36)-NH2 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:1819	iuphar.ligand:1819	[D-TRP12,TYR34]PTH-(7-34) (BOVINE)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:1820	iuphar.ligand:1820	[D-TRP12]PTH-(7-34) (BOVINE)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1809	iuphar.ligand:1809	[TRP23]PTHRP-(1-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1791	iuphar.ligand:1791	[125I][NLE8,21,TYR34]PTH-(1-34)-NH2 (RAT)	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9443	iuphar.ligand:9443	COMPOUND 25E [PMID: 25875054]	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:10387	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:10132	iuphar.ligand:10132	GSK963	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:5693	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11560	iuphar.ligand:11560	COMPOUND III [PMID: 29351497]	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.4039051633514961	IUPHAR.LIGAND:1992	iuphar.ligand:1992	RELAXIN	FALSE	FALSE	FALSE
NCBIGENE:1525	hgnc:2559	CXADR	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8036	iuphar.ligand:8036	PF-4708671	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:9320	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.5147810905460244	IUPHAR.LIGAND:9289	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:9331	rxcui:2668045	ETRASIMOD	TRUE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.5147810905460244	IUPHAR.LIGAND:9289	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.6177373086552295	IUPHAR.LIGAND:9320	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:9320	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:9331	rxcui:2668045	ETRASIMOD	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.034888818	IUPHAR.LIGAND:7547	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NCBIGENE:2223	hgnc:17209	STK36	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8203	iuphar.ligand:8203	RO-0505124	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1526385791735305	IUPHAR.LIGAND:7158	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
NCBIGENE:2400	hgnc:3911	FRA5G	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:7859	iuphar.ligand:7859	B3C	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:7551	rxcui:6465	LOFEPRAMINE	FALSE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:4588	iuphar.ligand:4588	REMOGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:10654	ncit:C150375	LICOGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9941	iuphar.ligand:9941	TAS05567	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:9815	iuphar.ligand:9815	CCT196969	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6046	iuphar.ligand:6046	SYK INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2048	iuphar.ligand:2048	L-363,377	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2005	iuphar.ligand:2005	CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.1244257612220248	IUPHAR.LIGAND:10343	iuphar.ligand:10343	GSK8612	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:10296	iuphar.ligand:10296	COMPOUND 31 [PMID: 29968758]	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.1244257612220248	IUPHAR.LIGAND:9579	iuphar.ligand:9579	COMPOUND II [PMID: 21329883]	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.049770304	IUPHAR.LIGAND:10597	iuphar.ligand:10597	BAY-985	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.027650169	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:10428	iuphar.ligand:10428	COMPOUND 25 [PMID: 31260299]	FALSE	FALSE	FALSE
NCBIGENE:2233	ncbigene:2233	FEB1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
NCBIGENE:1753	hgnc:11849	TLR3	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:5047	iuphar.ligand:5047	POLY(I:C)	FALSE	FALSE	FALSE
NCBIGENE:1758	hgnc:2932	DMP1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9795	iuphar.ligand:9795	CU-CPT8M	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:12568	iuphar.ligand:12568	GDC-0334	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:2438	iuphar.ligand:2438	BTP2	FALSE	FALSE	FALSE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	modulator	6.563458904461812	IUPHAR.LIGAND:12538	iuphar.ligand:12538	APV206690A	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:12542	iuphar.ligand:12542	ML-SA5	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	2.386712328895204	IUPHAR.LIGAND:12549	iuphar.ligand:12549	ISOCHLOROGENIC ACID B	FALSE	FALSE	FALSE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.079077818	IUPHAR.LIGAND:6809	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.5081387538938177	IUPHAR.LIGAND:10459	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:12318	iuphar.ligand:12318	GDC-0214	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2154	iuphar.ligand:2154	UROTENSIN-II	FALSE	FALSE	FALSE
NCBIGENE:1013	hgnc:1754	CDH15	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:4758	iuphar.ligand:4758	[3H]VESAMICOL	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:2766	iuphar.ligand:2766	3-KETO-LITHOCHOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2217	iuphar.ligand:2217	D(CH2)5[TYR(ET)2,VAL4,DES-GLY9]AVP	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:12704	iuphar.ligand:12704	TOLINAPANT	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1538	iuphar.ligand:1538	NPY-(20-36) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:3627	iuphar.ligand:3627	NEUROPEPTIDE Y-(3-36)	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.010685322	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	CIViC	10-Apr-24	NULL	0.7955707762984014	ANTI-CTLA-4 MONOCLONAL ANTIBODY	ncit:C128036	ANTI-CTLA-4 MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	CIViC	10-Apr-24	NULL	0.1071038678953482	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
WT1	hgnc:12796	WT1	CIViC	10-Apr-24	NULL	0.049864835	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
AREG	hgnc:651	AREG	CIViC	10-Apr-24	NULL	0.4039051633514962	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	CIViC	10-Apr-24	NULL	0.272767123	PEXIDARTINIB	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.2749092734853114	BRAF INHIBITOR	ncit:C155322	BRAF INHIBITOR	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.4605936073306534	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
MSH6	hgnc:7329	MSH6	CIViC	10-Apr-24	NULL	1.640864726115453	ANTI-PD-1 MONOCLONAL ANTIBODY MEDI0680	ncit:C113332	ANTI-PD-1 MONOCLONAL ANTIBODY MEDI0680	FALSE	FALSE	TRUE
TSC1	hgnc:12362	TSC1	CIViC	10-Apr-24	NULL	2.187819634820604	MTOR INHIBITOR	ncit:C2201	MTOR INHIBITOR	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.021878196	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.034363659	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
VHL	hgnc:12687	VHL	CIViC	10-Apr-24	NULL	0.1143957978991165	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
NTRK2	hgnc:8032	NTRK2	CIViC	10-Apr-24	NULL	0.042073455	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
ERCC1	hgnc:3433	ERCC1	CIViC	10-Apr-24	NULL	0.049723174	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	1.458546423213736	VE-821	iuphar.ligand:8042	VE-821	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	CIViC	10-Apr-24	NULL	0.1027547382303219	KU-0060648	iuphar.ligand:8011	KU-0060648	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.4167275494896388	NAQUOTINIB	ncit:C115110	NAQUOTINIB	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.014782565	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
EZH2	hgnc:3527	EZH2	CIViC	10-Apr-24	NULL	5.834185692854944	EPZ011989	iuphar.ligand:9273	EPZ011989	FALSE	FALSE	TRUE
PTPRD	hgnc:9668	PTPRD	CIViC	10-Apr-24	NULL	2.187819634820604	TEPROTUMUMAB	rxcui:2274802	TEPROTUMUMAB-TRBW	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	1.374546367426557	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	DoCM	10-Apr-24	NULL	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	2.493675356344019	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.021742307	Ixazomib	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	PF3644022	drugbank:DB07430	(10R)-10-METHYL-3-(6-METHYLPYRIDIN-3-YL)-9,10,11,12-TETRAHYDRO-8H-[1,4]DIAZEPINO[5',6':4,5]THIENO[3,2-F]QUINOLIN-8-ONE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.034363659	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	IMM-1-104	ncit:C192810	MEK INHIBITOR IMM-1-104	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.032342267	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	ASTX029	iuphar.ligand:11727	ASTX029	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.018327285	Voruciclib	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.041236391	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.5303805175322676	BAY1217389	iuphar.ligand:12705	BAY1217389	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.2273059360852575	Vantictumab	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	3.424413341458336	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.3271505995993426	3D185	ncit:C175460	FGFR/CSF-1R INHIBITOR 3D185	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1402073998282897	Vistusertib	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.4700175174550658	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.3642372228836055	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.2711239478607289	Pexidartinib	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.5903640284436551	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.1640864726115453	Blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.020257589	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.4167275494896388	DEL-22379	wikidata:Q21044462	DEL-22379	FALSE	FALSE	FALSE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.085378327	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.729273212	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.021902532	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.03849536	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.060492709	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.2047082699247349	Apitolisib	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	1.105424657593568	GSK126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.023151531	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	CC-115	drugbank:DB12740	CC-115	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.011575765	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	1.750255707856483	E7449	ncit:C102746	PARP/TANKYRASE INHIBITOR 2X-121	FALSE	FALSE	TRUE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	0.074797252	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	Torkinib	iuphar.ligand:5704	PP-242	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.007629711	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.064505739	GDC-0084	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.05913026	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.070956312	Uprosertib	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.019351722	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.2651902587661338	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CancerCommons	25-Jul-13	inhibitor	0.7143900848393808	BAY86-9766	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CancerCommons	25-Jul-13	inhibitor	0.5903640284436551	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.252440727	MESORIDAZINE BESYLATE	rxcui:203186	MESORIDAZINE BESYLATE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.022080602	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	ChEMBL	33	agonist	3.281729452230906	GONADOTROPIN, CHORIONIC	chembl:CHEMBL1201509	GONADOTROPIN, CHORIONIC	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	BAS-8770949	chembl:CHEMBL476025	CHEMBL:CHEMBL476025	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2773292494843019	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.5527123287967842	PI-88	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.009788902	dolutegravir	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.1535312024435511	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.8334550989792777	Ribociclib Succinate	rxcui:1873978	RIBOCICLIB SUCCINATE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	2.386712328895204	Fosfosal	ncit:C65760	FOSFOSAL	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4952	iuphar.ligand:4952	HS-142-1	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.2075402025126264	IUPHAR.LIGAND:10385	iuphar.ligand:10385	COMPOUND T.14	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	FLOPROPIONE	rxcui:25082	FLOPROPIONE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.02726255	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	NSC-748113	chembl:CHEMBL2063687	CHEMBL:CHEMBL2063687	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	2-AMINOFLURENE	chembl:CHEMBL84472	CHEMBL:CHEMBL84472	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00317843	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.9053046764774912	MAGNOLOL	rxcui:2562549	MAGNOLOL	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.300043836	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	chembl:CHEMBL284028	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	AFLOQUALONE	ncit:C83522	AFLOQUALONE	FALSE	FALSE	FALSE
GRM4	hgnc:4596	GRM4	DTC	9/2/20	NULL	2.500365296937833	N-(3-CHLOROPHENYL)PICOLINAMIDE	iuphar.ligand:6234	VU0364770	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	ZANOTERONE	ncit:C74123	ZANOTERONE	FALSE	FALSE	FALSE
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	0.6563458904461812	JNJ-26854165	ncit:C77904	SERDEMETAN	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	0.065634589	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:290	iuphar.ligand:290	MCN-A-343	FALSE	FALSE	FALSE
UNIPROT:P43088	hgnc:9600	PTGFR	TdgClinicalTrial	Jan-14	NULL	15.00219178	LATANOPROST	rxcui:43611	LATANOPROST	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.1043371509899543	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NDUFA4	hgnc:7687	NDUFA4	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
AVPR1B	hgnc:896	AVPR1B	ChEMBL	33	agonist	0.5770073762164232	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
HAVCR2	hgnc:18437	HAVCR2	ChEMBL	33	inhibitor	17.50255707856483	SABATOLIMAB	ncit:C124850	SABATOLIMAB	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004339477	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	8-(3-CHLOROSTYRYL)CAFFEINE	iuphar.ligand:5609	CSC	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	0.091636424	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P05091	hgnc:404	ALDH2	TEND	1-Aug-11	NULL	0.07963752	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.2333674277141978	IUPHAR.LIGAND:5820	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6248	iuphar.ligand:6248	V3 PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:12669	iuphar.ligand:12669	MMP13 TRACER  [18F]5J	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2272	iuphar.ligand:2272	PG 99-465	FALSE	FALSE	FALSE
NCBIGENE:1310	hgnc:2196	COL19A1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10400	iuphar.ligand:10400	PDE4 INHIBITOR 16	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:10489	iuphar.ligand:10489	COMPOUND 12B [PMID: 31465220]	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.015272737	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.2792961235941196	HYDROXYAMINE	chembl:CHEMBL1191361	HYDROXYAMINE	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1835932560688619	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.038722471	isradipine	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	FHND5071	ncit:C200562	RET INHIBITOR FHND5071	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	CIViC	10-Apr-24	NULL	0.093763699	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2717788366236775	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
EIF2AK4	hgnc:19687	EIF2AK4	DTC	9/2/20	inhibitor	0.2187819634820604	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.078136416	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.027767145	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P62937	hgnc:9253	PPIA	TdgClinicalTrial	Jan-14	NULL	3.750547945	SCY-635	drugbank:DB12451	SCY-635	FALSE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	OLESOXIME	ncit:C174604	OLESOXIME	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.0296486	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1724	iuphar.ligand:1724	MRS2500	FALSE	FALSE	FALSE
NCBIGENE:2412	hgnc:3923	FRA7E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8579	iuphar.ligand:8579	CID16197121	FALSE	FALSE	FALSE
NCBIGENE:1491	hgnc:2501	CTH	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:5192	iuphar.ligand:5192	G&OUML; 6983	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:12723	iuphar.ligand:12723	BMS-986202	FALSE	FALSE	FALSE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.038693936	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.039390601	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	ChEMBL	33	inhibitor	0.9546849315580819	MOLIDUSTAT	rxcui:2637535	MOLIDUSTAT	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.7458476027797514	BISOPROLOL	rxcui:19484	BISOPROLOL	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.046059361	IUPHAR.LIGAND:130	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.5000730593875666	IUPHAR.LIGAND:11311	drugbank:DB11987	GSK-2018682	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.4526523382387456	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
MTHFD1	hgnc:7432	MTHFD1	PharmGKB	4/5/24	NULL	0.1750255707856483	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:1489	hgnc:2499	CTF1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:5973	iuphar.ligand:5973	G&OUML; 6976	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.4167275494896388	VARLITINIB	ncit:C62530	VARLITINIB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	negative modulator	0.041672755	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	4.286340509036285	OLOKIZUMAB	ncit:C172654	OLOKIZUMAB	FALSE	FALSE	FALSE
KCNQ2	hgnc:6296	KCNQ2	ChEMBL	33	potentiator	3.000438356325399	EZOGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.022439176	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	1.591141552596802	DIETHYL-2-UNDECYLIDENEMALONATE	chembl:CHEMBL1797707	CHEMBL:CHEMBL1797707	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.013282993	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DICYCLOHEXYLCARBODIIMIDE	chembl:CHEMBL162598	DICYCLOHEXYLCARBODIIMIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	PIRETANIDE	rxcui:33770	PIRETANIDE	FALSE	FALSE	FALSE
NCBIGENE:3134	hgnc:4963	HLA-F	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:11104	iuphar.ligand:11104	SL-176	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	DTC	9/2/20	NULL	2.692701089009974	OBOVATAL	chembl:CHEMBL242530	OBOVATAL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	NU-2058	chembl:CHEMBL269881	CHEMBL:CHEMBL269881	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	0.103633562	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.3697723326457359	BUTORPHANOL TARTRATE	rxcui:203170	BUTORPHANOL TARTRATE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1835932560688619	VORTIOXETINE HYDROBROMIDE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	1.346350544504987	REVEXEPRIDE	ncit:C152202	REVEXEPRIDE	FALSE	FALSE	FALSE
NCBIGENE:1921	hgnc:19679	AAK1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984016	IUPHAR.LIGAND:7792	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.036463661	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.2035181055647073	Arbaclofen placarbil	ncit:C76088	ARBACLOFEN PLACARBIL	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1618	iuphar.ligand:1618	DYNORPHIN-(1-11)	FALSE	FALSE	FALSE
NCBIGENE:2182	hgnc:3571	ACSL4	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8186	iuphar.ligand:8186	COMPOUND 19A [PMID: 21855335]	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:1783	iuphar.ligand:1783	UDP-GLUCOSE	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.069638821	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	ChEMBL	33	agonist	8.751278539282417	DULANERMIN	ncit:C1685	DULANERMIN	FALSE	TRUE	TRUE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1944728564284981	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1472177698197042	OSPEMIFENE	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	0.4449802647092754	IRBESARTAN	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:9283	iuphar.ligand:9283	TG6-129	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2005	iuphar.ligand:2005	CGP 23996	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	1.265245090016735	AZD3229	iuphar.ligand:12703	AZD3229	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:9751	iuphar.ligand:9751	NECROSTATIN-1S	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	vaccine	1.389091831632129	RINDOPEPIMUT	ncit:C69076	RINDOPEPIMUT	FALSE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.023080295	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.4839416703750644	HMBA	ncit:C1125	HEXAMETHYLENE BISACETAMIDE	FALSE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	NCI	14-Sep-17	NULL	0.6177373086552295	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.5147810905460244	ITOPRIDE	ncit:C65991	ITOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:2812	iuphar.ligand:2812	METHOPRENE ACID	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:9992	iuphar.ligand:9992	COMPOUND 29 [MOSLIN ET AL., 2017]	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.8607814956671229	DYDROGESTERONE	rxcui:3706	DYDROGESTERONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.073089743	GALETERONE	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010122936	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1232574442152452	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1099637093941246	Milademetan	ncit:C141432	MILADEMETAN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.005127202	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.044878351	amprenavir	rxcui:228656	AMPRENAVIR	TRUE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4062	iuphar.ligand:4062	MM 11253	FALSE	FALSE	FALSE
COL6A6	hgnc:27023	COL6A6	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	DIMETACRINE	ncit:C81490	DIMETACRINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	ACRISORCIN	rxcui:89729	ACRISORCIN	TRUE	FALSE	FALSE
MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN 1	hgnc:51	ABCC1	TTD	2020.06.01	NULL	0.1844531776429549	Sulfinpyrazone	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
NCBIGENE:721	hgnc:1324	C4B	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.096167896	IUPHAR.LIGAND:7477	rxcui:787390	TAPENTADOL	TRUE	FALSE	FALSE
NCBIGENE:498	hgnc:823	ATP5F1A	GuideToPharmacology	2024.1	blocker	0.2625383561784725	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	QUERCETIN DIHYDRATE	ncit:C75768	QUERCETIN DIHYDRATE	FALSE	FALSE	FALSE
CYP27A1	hgnc:2605	CYP27A1	NCI	14-Sep-17	NULL	4.375639269641208	CHOLESTYRAMINE	rxcui:2447	CHOLESTYRAMINE RESIN	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.075496292	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:5614	ncit:C76394	PRELADENANT	FALSE	FALSE	FALSE
NCBIGENE:1758	hgnc:2932	DMP1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:10889	ncit:C170376	SELGANTOLIMOD	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.027538988	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.2778183663264258	AG-24322	drugbank:DB13035	AG-24322	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10424	iuphar.ligand:10424	HSD1590	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	RS-100329	iuphar.ligand:7381	RS-100329	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.036212187	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.1669560293662782	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:6161	iuphar.ligand:6161	CAY10583	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	positive modulator	0.3977853881492007	FARAMPATOR	ncit:C65620	FARAMPATOR	FALSE	FALSE	FALSE
RPL8	hgnc:10368	RPL8	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:7648	drugbank:DB14765	RIVOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:1324	hgnc:2615	CYP2B6	GuideToPharmacology	2024.1	inhibitor	0.1893305453210138	IUPHAR.LIGAND:7307	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2187	iuphar.ligand:2187	D[CHA4]AVP	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.1902451856365742	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	4.200613699	Risedronate	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10498	iuphar.ligand:10498	COMPOUND 8 [PMID: 25898023]	FALSE	FALSE	FALSE
TPH1	hgnc:12008	TPH1	ChEMBL	33	inhibitor	3.281729452230906	TELOTRISTAT	rxcui:1872382	TELOTRISTAT	TRUE	FALSE	FALSE
PRKAG3	hgnc:9387	PRKAG3	ChEMBL	33	activator	2.500365296937833	ACADESINE	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
IL2RG	hgnc:6010	IL2RG	ChEMBL	33	agonist	2.625383561784724	PEGENZILEUKIN	drugbank:DB17495	PEGENZILEUKIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.075010959	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	TCMDC-125587	chembl:CHEMBL532160	CHEMBL:CHEMBL532160	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.058602312	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	PHENELZINE SULFATE	rxcui:8124	PHENELZINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.019680536	IUPHAR.LIGAND:5717	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
S100A2	hgnc:10492	S100A2	NCI	14-Sep-17	NULL	1.591141552596803	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
SERPINA6	hgnc:1540	SERPINA6	PharmGKB	4/5/24	NULL	0.1442518440541057	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.011776541	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.027752469	IUPHAR.LIGAND:1225	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.2885036881082115	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:8464	iuphar.ligand:8464	DROXINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.048260727	IUPHAR.LIGAND:6004	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:11941	iuphar.ligand:11941	COMPOUND 17B [PMID: 35286086]	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2086	ncit:C80866	ELEDOISIN	FALSE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:9761	iuphar.ligand:9761	COMPOUND 9 [PMID: 26006010]	FALSE	FALSE	FALSE
NCBIGENE:3221	hgnc:5126	HOXC4	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:12409	iuphar.ligand:12409	AK-2292	FALSE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.3040984820600068	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.009098539	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.084553416	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	0.029590122	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NCBIGENE:2199	hgnc:3601	FBLN2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8049	iuphar.ligand:8049	HG-9-91-01	FALSE	FALSE	FALSE
NCBIGENE:435	hgnc:746	ASL	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:943	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	CIViC	10-Apr-24	NULL	0.025891357	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.036770078	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.1315981735230438	SODELGLITAZAR	ncit:C75193	SODELGLITAZAR	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.42006137	RIVOGLITAZONE	ncit:C72841	RIVOGLITAZONE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.069180068	ADOPRAZINE	ncit:C81482	ADOPRAZINE	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.4102161815288632	LY2780301	ncit:C95737	AKT INHIBITOR LY2780301	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.071439008	Plinabulin	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
NCBIGENE:1171	hgnc:14679	SLC38A4	GuideToPharmacology	2024.1	NULL	2.187819634820604	IUPHAR.LIGAND:4084	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
EPHRIN TYPE-A RECEPTOR 3	hgnc:3387	EPHA3	TTD	2020.06.01	NULL	11.66837138570988	Ifabotuzumab	ncit:C116629	IFABOTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:4289	iuphar.ligand:4289	PMBA	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1849	iuphar.ligand:1849	ABT-299	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:8447	iuphar.ligand:8447	2-CL-ADP(&ALPHA;-BH3)	FALSE	FALSE	FALSE
PSMC5	hgnc:9552	PSMC5	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
NCBIGENE:1169	hgnc:13447	SLC38A1	GuideToPharmacology	2024.1	NULL	10.50153425	IUPHAR.LIGAND:4542	rxcui:426	ALANINE	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1981421556063943	BRM	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.030670369	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	1.921012362281506	Oblimersen	ncit:C1870	OBLIMERSEN	FALSE	FALSE	TRUE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	1.500219178	GRNVAC1	ncit:C116888	HTERT-LAMP MRNA-LOADED AUTOLOGOUS DENDRITIC CELL VACCINE GRNVAC1	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:7518	iuphar.ligand:7518	I-BET151	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CGI	2/1/22	NULL	0.3642372228836055	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1131630845596864	IUPHAR.LIGAND:2020	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	PharmGKB	4/5/24	NULL	0.1591141552596803	cabazitaxel	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
IMMUNOGLOBULIN GAMMA FC RECEPTOR IIB	hgnc:3618	FCGR2B	TTD	2020.06.01	NULL	1.640864726115453	MGD010	chembl:CHEMBL4298039	MGD-010	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.053145416	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:5614	ncit:C76394	PRELADENANT	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.013673873	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.577007376	DALTEPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2208	hgnc:3612	FCER2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8188	iuphar.ligand:8188	COMPOUND 13 [PMID: 15925511]	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	BROMODIPHENHYDRAMINE HYDROCHLORIDE	rxcui:91065	BROMODIPHENHYDRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BCL2L1	hgnc:992	BCL2L1	ChEMBL	33	inhibitor	0.4688184931758437	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.038187397	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	DTC	9/2/20	NULL	0.4861821410712454	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	DESOXIMETASONE	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	THONZONIUM	rxcui:237058	THONZONIUM	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	PharmGKB	4/5/24	NULL	0.078428187	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2042	iuphar.ligand:2042	BOC-ATE	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.053361455	amifampridine phosphate	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.5585922471882393	CARBINOXAMINE	rxcui:20220	CARBINOXAMINE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	0.2573905452730122	8-AZAGUANINE	ncit:C28788	8-AZAGUANINE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1472177698197042	Ospemifene	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.062509132	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	CIViC	10-Apr-24	NULL	1.875273972703375	MONOMETHYL AURISTATIN E	ncit:C122637	MONOMETHYL AURISTATIN E	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.013631275	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.108040476	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2024	iuphar.ligand:2024	[125I]TYR10-CST14	FALSE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:3652	iuphar.ligand:3652	[125I]CCL17 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:5648	iuphar.ligand:5648	ANALOG 31 [PMID:18543899]	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:3552	iuphar.ligand:3552	CCK-58	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:3491	iuphar.ligand:3491	BAY27-9955	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.02804897	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	FRANGULIN B	chembl:CHEMBL496999	FRANGULIN B	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.300043836	IL-5	iuphar.ligand:4997	IL-5	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:2076	iuphar.ligand:2076	ACQ090	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:9903	iuphar.ligand:9903	SAMURACICLIB	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.030124883	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:2001	hgnc:3320	ELF5	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:8214	iuphar.ligand:8214	COMPOUND 14K [PMID: 21982499]	FALSE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9781	iuphar.ligand:9781	&ALPHA;-NETA	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.591141552596803	DEGARELIX	rxcui:475230	DEGARELIX	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	NCI	14-Sep-17	NULL	0.1944728564284981	INTERLEUKIN-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
GSTZ1	hgnc:4643	GSTZ1	PharmGKB	4/5/24	NULL	35.00511415712966	dichloroacetic acid	rxcui:155021	DICHLOROACETIC ACID	TRUE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.5645986154375752	CYT007-TNFQB	drugbank:DB05758	CYT007-TNFQB	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.1491695205559502	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	TESMILIFENE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.005636894	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008279355	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	TALC	12-May-16	inhibitor	0.4828291607879953	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
UNIPROT:P26358	hgnc:2976	DNMT1	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	MG98	ncit:C2530	DNMT1 MIXED-BACKBONE ANTISENSE OLIGONUCLEOTIDE MG 98	FALSE	FALSE	FALSE
DCK	hgnc:2704	DCK	PharmGKB	4/5/24	NULL	0.050174554	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.057955487	Dendritic cell vaccine	ncit:C28310	DENDRITIC CELL VACCINE	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.072125922	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.03292017	CDDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	NSC-45382	chembl:CHEMBL1214274	CHEMBL:CHEMBL1214274	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.2678962818147678	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	DTC	9/2/20	NULL	0.4579157375205915	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	MECLIZINE DIHCL	chembl:CHEMBL1085765	MECLIZINE DIHCL	FALSE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TEND	1-Aug-11	NULL	0.2187819634820604	AMLODIPINE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.044763573	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.006058344	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
MT-ND2	hgnc:7456	MT-ND2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.2869271652223742	ALLYLESTRENOL	rxcui:525	ALLYLESTRENOL	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	DOBUTAMINE HYDROCHLORIDE	rxcui:203121	DOBUTAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.6731752722524935	CALCIUM GLUCONATE	rxcui:1908	CALCIUM GLUCONATE	TRUE	FALSE	FALSE
UNIPROT:P02452	hgnc:2197	COL1A1	TEND	1-Aug-11	NULL	0.8036888454443035	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11233	iuphar.ligand:11233	NP-1815-PX	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	OX40 LIGAND	ncit:C1548	RECOMBINANT OX40 LIGAND	FALSE	FALSE	FALSE
GNMT	hgnc:4415	GNMT	PharmGKB	4/5/24	NULL	7.001022831425934	methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.068458502	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
NDUFC1	hgnc:7705	NDUFC1	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MMP9	hgnc:7176	MMP9	ChEMBL	33	inhibitor	4.200613699	ANDECALIXIMAB	ncit:C105803	ANDECALIXIMAB	FALSE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	blocker	0.112919723	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	agonist	2.187819634820604	SELICRELUMAB	ncit:C119740	SELICRELUMAB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.2318219480604613	ATRACTYLENOLIDE I	chembl:CHEMBL449520	ATRACTYLENOLIDE I	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9353	iuphar.ligand:9353	SAR405	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:5690	iuphar.ligand:5690	KI-20227	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TNFSF13	hgnc:11928	TNFSF13	ChEMBL	33	inhibitor	26.25383561784724	SIBEPRENLIMAB	ncit:C179120	SIBEPRENLIMAB	FALSE	FALSE	FALSE
NCBIGENE:2731	hgnc:4313	GLDC	GuideToPharmacology	2024.1	NULL	5.834185692854944	IUPHAR.LIGAND:8573	iuphar.ligand:8573	NI-57	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.3889457128569963	INFIGRATINIB	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.026830696	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.015434354	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.030996264	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-4798	chembl:CHEMBL584635	CHEMBL:CHEMBL584635	FALSE	FALSE	FALSE
BCL2L1	hgnc:992	BCL2L1	DTC	9/2/20	NULL	3.750547945	SANGIVAMYCIN	chembl:CHEMBL101892	SANGIVAMYCIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	NSC-600067	chembl:CHEMBL1491455	CHEMBL:CHEMBL1491455	FALSE	FALSE	FALSE
UNIPROT:P01589	hgnc:6008	IL2RA	TEND	1-Aug-11	NULL	0.8579684842433742	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	3.850562557284263	Plerixafor	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
MELATONIN RECEPTOR TYPE 1A	hgnc:7463	MTNR1A	TTD	2020.06.01	NULL	7.501095891	LY-156735	drugbank:DB16909	TIK-301	FALSE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:9761	iuphar.ligand:9761	COMPOUND 9 [PMID: 26006010]	FALSE	FALSE	FALSE
NCBIGENE:2025	hgnc:3352	ENO1P1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
SLC12A1	hgnc:10910	SLC12A1	ChEMBL	33	inhibitor	1.250182648468916	TORSEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
SLC6A9	hgnc:11056	SLC6A9	ChEMBL	33	inhibitor	1.944728564284981	BITOPERTIN	ncit:C174879	BITOPERTIN	FALSE	FALSE	FALSE
CCL3	hgnc:10627	CCL3	NCI	14-Sep-17	NULL	1.129197231	INFLIXIMAB	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.049349315	ANTI-CANCER AGENTS	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	0.1704794520639432	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.1256164383629055	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.030746697	APOMORPHINE HYDROCHLORIDE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.09741683	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.024814589	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.046549354	DIAMIDE	chembl:CHEMBL1255835	DIAMIDE	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.059397818	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
EPHB4	hgnc:3395	EPHB4	ChEMBL	33	inhibitor	0.2263261691193728	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.750109589	SOLABEGRON	ncit:C96754	SOLABEGRON	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	3.281729452230906	JNJ-10311795	iuphar.ligand:6563	JNJ-10311795	FALSE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	ChEMBL	33	inhibitor	0.5834185692854945	MUPARFOSTAT	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.057260274	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:3284	iuphar.ligand:3284	PSB603	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:4246	iuphar.ligand:4246	LY339434	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.021933029	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:8220	iuphar.ligand:8220	COMPOUND 15 [PMID: 24900237]	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	agonist	0.5000730593875667	IUPHAR.LIGAND:4131	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	2,4-DINITROPHENOL	drugbank:DB04528	2,4-DINITROPHENOL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.001975086	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE	chembl:CHEMBL460508	CHEMBL:CHEMBL460508	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	SJ000292689	chembl:CHEMBL602954	CHEMBL:CHEMBL602954	FALSE	FALSE	FALSE
DDX53	hgnc:20083	DDX53	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.133607306	ALDOSTERONE	rxcui:1312358	ALDOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.4375639269641209	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6171	iuphar.ligand:6171	5-OXO-12-HETE	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.8468979231563628	ACNU	ncit:C693	NIMUSTINE	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.029106248	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
MGAT4A	hgnc:7047	MGAT4A	PharmGKB	4/5/24	NULL	0.7292732116068681	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.1100789753368857	IUPHAR.LIGAND:488	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:310	hgnc:545	ANXA7	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1586	rxcui:28627	LEVOCABASTINE	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.3182283105193606	BRM	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	0.8008364246019593	ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:2341	hgnc:3784	FNTAP2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11754	ncit:C175138	MILVEXIAN	FALSE	FALSE	FALSE
NCBIGENE:1318	hgnc:11017	SLC31A2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8789	iuphar.ligand:8789	CHRYSIN	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0296486	IUPHAR.LIGAND:9428	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:12643	iuphar.ligand:12643	RELUTRIGINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	GNF-PF-4337	chembl:CHEMBL277148	CHEMBL:CHEMBL277148	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	agonist	0.033919684	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
TUBB8B	hgnc:24983	TUBB8B	ChEMBL	33	inhibitor	3.088686543276147	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3509871071904712	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
UNIPROT:P01589	hgnc:6008	IL2RA	TdgClinicalTrial	Jan-14	NULL	1.715936968486748	BASILIXIMAB	rxcui:196102	BASILIXIMAB	TRUE	TRUE	FALSE
UNIPROT:Q09428	hgnc:59	ABCC8	TdgClinicalTrial	Jan-14	NULL	0.7501095890813498	REPAGLINIDE	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.037884323	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:8731	iuphar.ligand:8731	COMPOUND 10B [PMID: 26222319]	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.054981855	Uprosertib	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	SAPPANONE A TRIMETHYL ETHER	chembl:CHEMBL1606022	SAPPANONE A TRIMETHYL ETHER	FALSE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.025588534	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SLCO1B3	hgnc:10961	SLCO1B3	PharmGKB	4/5/24	NULL	0.3500511415712966	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00667527	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.066241806	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.5048814541893701	Benzthiazide	rxcui:19008	BENZTHIAZIDE	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	4.200613699	TAG-72	ncit:C1269	TAG-72 ANTIGEN	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.015088411	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.1595977849109255	IUPHAR.LIGAND:2031	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	CancerCommons	25-Jul-13	inhibitor	0.021138354	PF00562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.068847471	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.067317527	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4688184931758437	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1544343271638073	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.020117882	IUPHAR.LIGAND:214	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:1484	ncbigene:1484	CTAA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524936	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TEND	1-Aug-11	NULL	1.944728564284981	CHLORZOXAZONE	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	IDEBENONE	rxcui:51296	IDEBENONE	TRUE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	DTC	9/2/20	NULL	1.591141552596803	EPIBATIDINE	drugbank:DB07720	EPIBATIDINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
ACTB	hgnc:132	ACTB	NCI	14-Sep-17	NULL	0.036590712	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.2858856873086814	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
AK2	hgnc:362	AK2	PharmGKB	4/5/24	NULL	2.917092846427472	adefovir dipivoxil	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.2243917574174978	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
NDUFA7	hgnc:7691	NDUFA7	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	ChEMBL	33	agonist	0.043756393	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.01858569	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:10433	iuphar.ligand:10433	COMPOUND 5A [PMID: 31287314]	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	OBTUSAQUINONE	chembl:CHEMBL1333653	OBTUSAQUINONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB]	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002552882	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6236	iuphar.ligand:6236	COMPOUND 1 [PMID: 22465637]	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
UNIPROT:P53609	hgnc:8895	PGGT1B	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	GGTI-2418	chembl:CHEMBL3218390	GGTI-2418	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.032003863	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	1.413668071730236	AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:84	rxcui:21877	CYAMEMAZINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:1216	iuphar.ligand:1216	A-317920	FALSE	FALSE	FALSE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:8939	iuphar.ligand:8939	FRAX597	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2677	iuphar.ligand:2677	MK-0767	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.5707355569097228	IUPHAR.LIGAND:2476	iuphar.ligand:2476	NI2+	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2236	iuphar.ligand:2236	D(CH2)5[D-ILE2,ILE4]AVP	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.2573905452730122	BIIB068	iuphar.ligand:11178	BIIB068	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.006375385	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TEND	1-Aug-11	NULL	1.207072901969988	MITIGLINIDE	ncit:C81699	MITIGLINIDE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.034184682	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.028199609	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	0.1544343271638073	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.169927739	RO-0282750	chembl:CHEMBL1397270	CHEMBL:CHEMBL1397270	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	TRIMEPRAZINE	rxcui:10825	TRIMEPRAZINE	TRUE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:3426	iuphar.ligand:3426	L659989	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.085239726	SJ000071854	chembl:CHEMBL602127	CHEMBL:CHEMBL602127	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	LYNGBYABELLIN A	chembl:CHEMBL453207	LYNGBYABELLIN A	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
UNIPROT:P49721	hgnc:9539	PSMB2	TdgClinicalTrial	Jan-14	NULL	0.4579157375205915	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	TCMDC-124422	chembl:CHEMBL527620	CHEMBL:CHEMBL527620	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	0.6731752722524935	CP-101,606	ncit:C87769	TRAXOPRODIL	FALSE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:11397	iuphar.ligand:11397	COMPOUND 40 [PMID: 33470814]	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.036847489	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.6563458904461812	Karenitecin	chembl:CHEMBL1743260	KARENITECIN	FALSE	FALSE	FALSE
NDUFS7	hgnc:7714	NDUFS7	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.1396480617970598	IUPHAR.LIGAND:2020	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
PRKCI	hgnc:9404	PRKCI	ChEMBL	33	inhibitor	0.3088686543276147	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.064111931	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1223955040459079	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:8376	rxcui:1992672	ERTUGLIFLOZIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ISOKOBUSONE	chembl:CHEMBL1522104	ISOKOBUSONE	FALSE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	3.182283105193605	Acarbose	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:11555	iuphar.ligand:11555	DIABZI-4	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1060761035064535	granisetron	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.1715936968486748	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
CYP11B2	hgnc:2592	CYP11B2	PharmGKB	4/5/24	NULL	0.9723642821424908	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1902451856365742	CUMENE HYDROPEROXIDE	chembl:CHEMBL1518369	CUMENE HYDROPEROXIDE	FALSE	FALSE	FALSE
ERRFI1	hgnc:18185	ERRFI1	CIViC	10-Apr-24	NULL	0.4449802647092754	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
KCNC4	hgnc:6236	KCNC4	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.1223955040459079	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1182605208011137	SOFPIRONIUM BROMIDE	ncit:C152384	SOFPIRONIUM BROMIDE	FALSE	FALSE	FALSE
ARAF	hgnc:646	ARAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3818739726232327	1096708-71-2	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.036531311	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	agonist	0.036463661	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:6071	iuphar.ligand:6071	AGN 191976	FALSE	FALSE	FALSE
IL15RA	hgnc:5978	IL15RA	ChEMBL	33	agonist	4.375639269641208	RECOMBINANT HUMAN INTERLEUKIN-15	ncit:C1545	RECOMBINANT HUMAN INTERLEUKIN-15	FALSE	FALSE	FALSE
UNIPROT:P10276	hgnc:9864	RARA	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	TAMIBAROTENE	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
THROMBOXANE-A SYNTHASE	hgnc:11609	TBXAS1	TTD	2020.06.01	NULL	6.563458904461812	PYRIDINE	chembl:CHEMBL266158	PYRIDINE	FALSE	FALSE	FALSE
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	1.750255707856483	RG7388	ncit:C99131	IDASANUTLIN	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.024286619	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:2421	hgnc:3931	FRA8C	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8670	iuphar.ligand:8670	COMPOUND 5 [PMID: 21741839]	FALSE	FALSE	FALSE
NDUFB10	hgnc:7696	NDUFB10	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.038159645	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	TD-2749	drugbank:DB05905	TD-2749	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:237	iuphar.ligand:237	RS 67333	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.3889457128569963	IUPHAR.LIGAND:11888	ncit:C175551	ZILURGISERTIB	FALSE	FALSE	FALSE
NCBIGENE:2903	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	antibody	0.3804903712731485	IUPHAR.LIGAND:12229	iuphar.ligand:12229	ZWB67	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6042	iuphar.ligand:6042	SRC KINASE INHIBITOR I	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.2778183663264259	AV-412	drugbank:DB06021	AV-412	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SB-269970	drugbank:DB13988	SB-269970	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	CHLORDANE	iuphar.ligand:2831	CHLORDANE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.002232754	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,7-BIS[3-(PIPERIDINO)PROPIONAMIDO]ANTHRAQUINONE	chembl:CHEMBL89250	CHEMBL:CHEMBL89250	FALSE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	0.7955707762984013	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1795	hgnc:2989	DOCK3	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8075	iuphar.ligand:8075	LY2109761	FALSE	FALSE	FALSE
TSC22D3	hgnc:3051	TSC22D3	NCI	14-Sep-17	NULL	0.4268916360625569	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	0.5000730593875666	9-CRA	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.4565884455277783	IUPHAR.LIGAND:7091	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
VAMP2	hgnc:12643	VAMP2	ChEMBL	33	inhibitor	17.50255707856483	BOTULINUM TOXIN TYPE B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.062509132	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	blocker	0.1881995384791917	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	2.763561643983921	IUPHAR.LIGAND:6333	iuphar.ligand:6333	OAADPR	FALSE	FALSE	FALSE
NCBIGENE:2839	hgnc:584	APCS	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:8255	iuphar.ligand:8255	DEZAMIZUMAB	FALSE	FALSE	FALSE
DOT1L	hgnc:24948	DOT1L	PharmGKB	4/5/24	NULL	7.001022831425933	candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.050294704	HEMATOXYLIN	drugbank:DB16871	HEMATOXYLIN	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.1256164383629055	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	CHRYSOPHANOL	chembl:CHEMBL41092	CHRYSOPHANOL	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.009905239	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	0.6250913242344582	MF-101	wikidata:Q6816906	MENERBA	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.05073205	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	ENTACAPONE	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12555	iuphar.ligand:12555	CIMIFUGIN	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	BUCLIZINE	rxcui:59636	BUCLIZINE	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	ChEMBL	33	inhibitor	0.050294704	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.096167896	DELUCEMINE	ncit:C76776	DELUCEMINE	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:1028	iuphar.ligand:1028	I-BOC-MET-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.2651902587661338	IUPHAR.LIGAND:12737	ncit:C166556	LANIFIBRANOR	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6418	iuphar.ligand:6418	TETRAHYDROCANNABIVARIN	FALSE	FALSE	FALSE
NCBIGENE:2142	hgnc:8810	PDK2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:9350	iuphar.ligand:9350	VER-246608	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.044161204	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.075010959	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.032134438	IUPHAR.LIGAND:2398	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NDUFA12	hgnc:23987	NDUFA12	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PAK4	hgnc:16059	PAK4	ChEMBL	33	inhibitor	2.187819634820604	PF-03758309	drugbank:DB11775	PF-03758309	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12562	drugbank:DB15366	SOR-C13	FALSE	FALSE	FALSE
HTR3C	hgnc:24003	HTR3C	ChEMBL	33	agonist	0.2206204673768676	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.075442056	IUPHAR.LIGAND:380	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:7355	rxcui:1441386	BAZEDOXIFENE	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	LY2780301	ncit:C95737	AKT INHIBITOR LY2780301	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.2785552850699974	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001682938	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	4.039051633514961	GS-5829	ncit:C126640	ALOBRESIB	FALSE	FALSE	FALSE
ERAP1	hgnc:18173	ERAP1	DTC	9/2/20	NULL	1.458546423213736	SCOPOLETIN	chembl:CHEMBL71851	SCOPOLETIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001420662	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:10631	iuphar.ligand:10631	LORPUCITINIB	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	ChEMBL	33	inhibitor	0.075768645	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:328	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2695	iuphar.ligand:2695	GW0072	FALSE	FALSE	FALSE
NCBIGENE:3229	hgnc:5125	HOXC13	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:12637	iuphar.ligand:12637	EN67	FALSE	FALSE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TEND	1-Aug-11	NULL	3.454452054979901	EPLERENONE	rxcui:298869	EPLERENONE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.2263261691193728	KBP5209	chembl:CHEMBL4650289	KBP5209	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.042140988	IUPHAR.LIGAND:8918	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	CARBARIL	ncit:C76389	CARBARIL	TRUE	FALSE	FALSE
NCBIGENE:3228	hgnc:5124	HOXC12	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:12636	iuphar.ligand:12636	EN450	FALSE	FALSE	FALSE
CYP46A1	hgnc:2641	CYP46A1	ChEMBL	33	inhibitor	52.50767123569449	SOTICLESTAT	ncit:C166470	SOTICLESTAT	FALSE	FALSE	FALSE
UNIPROT:P06239	hgnc:6524	LCK	TdgClinicalTrial	Jan-14	NULL	0.033211683	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.030211548	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7487	rxcui:535	ALPHA 1-ANTITRYPSIN	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	TCMDC-125653	chembl:CHEMBL580918	CHEMBL:CHEMBL580918	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.013008218	erythromycin	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.105015342	gliclazide	rxcui:4816	GLICLAZIDE	TRUE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	0.3017682254924971	CAMBINOL	drugbank:DB15493	CAMBINOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	ETHACRIDINE LACTATE	rxcui:4107	ETHACRIDINE LACTATE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.5509279467829125	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	KETOTIFEN FUMARATE	rxcui:11404	KETOTIFEN FUMARATE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
MAG	hgnc:6783	MAG	ChEMBL	33	inhibitor	17.50255707856483	GSK-249320	chembl:CHEMBL2109573	GSK-249320	FALSE	FALSE	FALSE
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	0.3977853881492008	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
NCBIGENE:2645	hgnc:4195	GCK	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:6839	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	modulator	1.591141552596803	IUPHAR.LIGAND:10586	iuphar.ligand:10586	JNJ-27141491	FALSE	FALSE	FALSE
NCBIGENE:2451	hgnc:3848	FRA12D	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9719	iuphar.ligand:9719	BI-1950	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.1562728310586145	IUPHAR.LIGAND:2616	iuphar.ligand:2616	TETRODOTOXIN	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	4.699760697022038	SELPERCATINIB	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
ADD1	hgnc:243	ADD1	PharmGKB	4/5/24	NULL	2.187819634820604	torasemide	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	2.100306849	MT203	ncit:C97943	NAMILUMAB	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	TCMDC-123653	chembl:CHEMBL548540	CHEMBL:CHEMBL548540	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.084963869	DNDI1417447	chembl:CHEMBL1307453	CHEMBL:CHEMBL1307453	FALSE	FALSE	FALSE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	0.032134438	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:717	hgnc:1248	C2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.032055965	IUPHAR.LIGAND:2176	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.091636424	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.3947945205691315	VECURONIUM BROMIDE	rxcui:11153	VECURONIUM BROMIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.014883127	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
OXYTOCIN RECEPTOR	hgnc:8529	OXTR	TTD	2020.06.01	NULL	3.088686543276147	GSK221149	ncit:C76681	RETOSIBAN	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:7518	iuphar.ligand:7518	I-BET151	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:6127	iuphar.ligand:6127	GALR3ANT	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2778183663264258	IUPHAR.LIGAND:2183	iuphar.ligand:2183	DVDAVP	FALSE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1868	iuphar.ligand:1868	PROKINETICIN-2&BETA;	FALSE	FALSE	FALSE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.064268875	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
KCNQ4	hgnc:6298	KCNQ4	ChEMBL	33	potentiator	1.500219178162699	EZOGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	1.071585127259071	Rocuronium	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2222	iuphar.ligand:2222	D(CH2)5[TYR(ME)2,THR4]OVT	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.027010119	AT-9283	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.050488145	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1835932560688619	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.3226277802500429	CERTOLIZUMAB PEGOL	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.097236428	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.025147352	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.151537291	IUPHAR.LIGAND:7938	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2210	iuphar.ligand:2210	[PHAA1,D-TYR(ME)2,ARG6,TYR-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5630	iuphar.ligand:5630	[125I][TYR3,THR8]OCTREOTIDE	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	4.773424657790408	IUPHAR.LIGAND:10303	iuphar.ligand:10303	FORSYTHOSIDE B	FALSE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	3.462044257298538	Dostarlimab-gxly	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2209	iuphar.ligand:2209	[PHAA1,D-TYR(ET)2,VAL4,LYS6,TYR-NH28,DES-GLY9]AVP	FALSE	FALSE	FALSE
ITGB1	hgnc:6153	ITGB1	TALC	12-May-16	antibody	1.093909817410302	VITAXIN	ncit:C1800	ETARACIZUMAB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DICHLOFLUANID	chembl:CHEMBL1269177	DICHLOFLUANID	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.061041236	PERGOLIDE	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.011741429	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.036237178	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.2035181055647073	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	MELENGESTROL ACETATE	rxcui:1537798	MELENGESTROL ACETATE	TRUE	FALSE	FALSE
RARB	hgnc:9865	RARB	NCI	14-Sep-17	NULL	0.1018248310970158	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2212	iuphar.ligand:2212	[TBAA1,D-TYR(ET)2,VAL4,LYS6,ARG-NH28,DES-GLY9]AVP	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.047734247	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.2651902587661338	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.053579256	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.1875273972703375	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.051655358	DEXTROAMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2205	iuphar.ligand:2205	YM 471	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	other/unknown	2.187819634820604	AR-20.5	chembl:CHEMBL2109364	AR-20.5	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.014630168	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:1794	hgnc:2988	DOCK2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10432	rxcui:2612087	DEUCRAVACITINIB	TRUE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:9696	iuphar.ligand:9696	OCLACITINIB	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.018942161	CPT-11	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	FENBENDAZOLE	rxcui:4325	FENBENDAZOLE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
NCBIGENE:2093	ncbigene:2093	ERVT3	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9406	iuphar.ligand:9406	XMD17-109	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2211	iuphar.ligand:2211	[PHAA1,D-TYR2,VAL4,ARG6,ARG-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:6048	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.07631929	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CA10	hgnc:1369	CA10	PharmGKB	4/5/24	NULL	2.386712328895204	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2209	iuphar.ligand:2209	[PHAA1,D-TYR(ET)2,VAL4,LYS6,TYR-NH28,DES-GLY9]AVP	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 2	hgnc:11848	TLR2	TTD	2020.06.01	NULL	1.875273972703375	OM-174	ncit:C169880	DEFOSLIMOD	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.085239726	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.1396480617970598	DERAZANTINIB	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2205	iuphar.ligand:2205	YM 471	FALSE	FALSE	FALSE
HTR6	hgnc:5301	HTR6	ChEMBL	33	inhibitor	3.500511415712966	CERLAPIRDINE	ncit:C169839	CERLAPIRDINE	FALSE	FALSE	FALSE
C5AR1	hgnc:1338	C5AR1	ChEMBL	33	inhibitor	6.563458904461812	AVACOPAN	rxcui:2572100	AVACOPAN	TRUE	FALSE	FALSE
NCBIGENE:75	hgnc:148	ACTG1P3	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:3647	iuphar.ligand:3647	XCL1	FALSE	FALSE	FALSE
NCBIGENE:722	hgnc:1325	C4BPA	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.6141248097742047	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001914661	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.049864835	terfenadine	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6915	iuphar.ligand:6915	[SAR1,ALA8]ANG-II	FALSE	FALSE	FALSE
NCBIGENE:2789	hgnc:4409	GNG5P1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10052	ncit:C152861	VERDIPERSTAT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	5-CARBOXAMIDOTRYPTAMINE	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.276356164	(S)-NOMIFENSINE	chembl:CHEMBL51697	CHEMBL:CHEMBL51697	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.009098539	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.01609924	granisetron	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.2	hgnc:6256	KCNJ10	TTD	2020.06.01	NULL	1.071585127259071	Tolazamide	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.005955952	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:75	hgnc:148	ACTG1P3	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:857	iuphar.ligand:857	[125I]XCL1 (HUMAN)	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.010082118	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	SB-200646	chembl:CHEMBL85194	CHEMBL:CHEMBL85194	FALSE	FALSE	FALSE
MBP	hgnc:6925	MBP	NCI	14-Sep-17	NULL	0.1724389859957126	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
MAPK1	hgnc:6871	MAPK1	PharmGKB	4/5/24	NULL	0.005263927	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PRKAA2	hgnc:9377	PRKAA2	PharmGKB	4/5/24	NULL	0.1256164383629055	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	DTC	9/2/20	NULL	1.166837138570988	SB-0304	chembl:CHEMBL409225	CHEMBL:CHEMBL409225	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	NCI	14-Sep-17	NULL	0.1653584607713247	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	SJ000260158	chembl:CHEMBL601918	CHEMBL:CHEMBL601918	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	BIFENAZATE	chembl:CHEMBL1872845	BIFENAZATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.097308509	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.029366707	MACROLIDES	ncit:C261	MACROLIDE ANTIBIOTIC	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:790	iuphar.ligand:790	RO116-9132/238	FALSE	FALSE	FALSE
NCBIGENE:1528	hgnc:2570	CYB5A	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:2162	iuphar.ligand:2162	BIM 23127	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	PharmGKB	4/5/24	NULL	0.023620185	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
SULT2B1	hgnc:11459	SULT2B1	PharmGKB	4/5/24	NULL	0.7721716358190368	fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.040893825	leflunomide	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
TTR	hgnc:12405	TTR	PharmGKB	4/5/24	NULL	17.50255707856483	tafamidis	rxcui:1545063	TAFAMIDIS	TRUE	FALSE	FALSE
DYSTROPHIN	hgnc:2928	DMD	TTD	2020.06.01	NULL	7.501095891	WVE-210201	chembl:CHEMBL4298192	SUVODIRSEN	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.01858569	Risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.004842988	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
NDUFV2	hgnc:7717	NDUFV2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
RPS25	hgnc:10413	RPS25	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	0.4375639269641208	flupirtine	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
SLC10A2	hgnc:10906	SLC10A2	PharmGKB	4/5/24	NULL	0.097326545	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.05293112	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	blocker	0.3125456621172291	IUPHAR.LIGAND:4138	iuphar.ligand:4138	ARGIOTOXIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.017715139	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.06375385	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007813642	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	NSC-125034	chembl:CHEMBL239439	CHEMBL:CHEMBL239439	FALSE	FALSE	FALSE
NDUFA10	hgnc:7684	NDUFA10	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.4167275494896388	PKI-166	iuphar.ligand:7642	PKI166	FALSE	FALSE	FALSE
SRD5A3	hgnc:25812	SRD5A3	ChEMBL	33	inhibitor	2.187819634820604	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2004109589148645	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:5662	iuphar.ligand:5662	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:2832	hgnc:4530	NPBWR2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12285	ncit:C169887	DESIDUSTAT	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.072424374	CICLOPIROX OLAMINE	rxcui:52172	CICLOPIROX OLAMINE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1325951293830669	STROPHANTHIDIN	chembl:CHEMBL111743	STROPHANTHIDIN	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.1988926940746003	VIOXX	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	NCI	14-Sep-17	NULL	0.051731696	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	0.546954909	DS-6051	chembl:CHEMBL4650989	TALETRECTINIB	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.008479921	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.003936107	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CDC37	hgnc:1735	CDC37	DTC	9/2/20	NULL	3.750547945406749	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	2.187819634820604	isoniazid / pyrazinamide / rifampin	wikidata:Q48566689	ISONIAZID / PYRAZINAMIDE / RIFAMPIN	FALSE	FALSE	FALSE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TEND	1-Aug-11	NULL	0.2792961235941196	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	JCARH125	ncit:C147523	ORVACABTAGENE AUTOLEUCEL	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:155	ncit:C80757	BROLAMFETAMINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	CARBETAPENTANE	rxcui:20217	CARBETAPENTANE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	PharmGKB	4/5/24	NULL	0.5181678082469852	levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:10030	iuphar.ligand:10030	VCE-004.3	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2035181055647073	NAVAFENTEROL	ncit:C174920	NAVAFENTEROL	FALSE	FALSE	FALSE
HOXD1	hgnc:5132	HOXD1	NCI	14-Sep-17	NULL	0.5770073762164231	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	3.750547945	Ridogrel	ncit:C96931	RIDOGREL	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 1	hgnc:4584	GRIN1	TTD	2020.06.01	NULL	0.06697407	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	0.1988926940746003	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TdgClinicalTrial	Jan-14	NULL	0.7693431682885642	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.1930429089547591	EPLIVANSERINE	ncit:C65517	EPLIVANSERIN	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.3472729579080324	CO-1686	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
SLC13A3	hgnc:14430	SLC13A3	PharmGKB	4/5/24	NULL	0.3500511415712966	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.1013661606866689	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	CancerCommons	25-Jul-13	inhibitor	0.3889457128569963	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
AKT3	hgnc:393	AKT3	CGI	2/1/22	NULL	0.4688184931758437	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	1.374546367426557	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
DPYD	hgnc:3012	DPYD	CGI	2/1/22	NULL	0.091732479	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CGI	2/1/22	NULL	0.053217234	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
NOTCH1	hgnc:7881	NOTCH1	CGI	2/1/22	NULL	3.938075342677087	Ro4929097	iuphar.ligand:7338	RO4929097	FALSE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	CGI	2/1/22	NULL	0.1060761035064535	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CGI	2/1/22	NULL	0.032412143	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CGI	2/1/22	NULL	0.1043371509899543	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	agonist	0.729273212	METHYLERGONOVINE MALEATE	rxcui:84158	METHYLERGONOVINE MALEATE	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	1.887530665335423	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1396480617970598	ATROPINE SULFATE	rxcui:153971	ATROPINE SULFATE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.105015342	BALSALAZIDE DISODIUM	rxcui:153718	BALSALAZIDE DISODIUM	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	ChEMBL	33	inhibitor	0.7249579855026854	FEBUXOSTAT	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	0.8334550989792776	DALTEPARIN SODIUM	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.09972967	SOTALOL HYDROCHLORIDE	rxcui:7008	SOTALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.047561296	DEXTROMETHORPHAN POLISTIREX	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP PURIFIED PORK	chembl:CHEMBL1201653	INSULIN ZINC SUSP PURIFIED PORK	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN SUSP ISOPHANE SEMISYNTHETIC PURIFIED HUMAN	chembl:CHEMBL1201627	INSULIN SUSP ISOPHANE SEMISYNTHETIC PURIFIED HUMAN	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.063110182	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	15.00219178	LATANOPROST	rxcui:43611	LATANOPROST	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.3125456621172291	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	0.7721716358190367	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1715936968486748	BUPROPION HYDROCHLORIDE	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	PROPOXYPHENE NAPSYLATE	rxcui:8786	PROPOXYPHENE NAPSYLATE	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.016764901	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GHRHR	hgnc:4266	GHRHR	ChEMBL	33	agonist	13.12691780892362	SERMORELIN ACETATE	rxcui:58932	SERMORELIN ACETATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.133607306	DIFLORASONE DIACETATE	rxcui:23033	DIFLORASONE DIACETATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2004109589148645	ALCLOMETASONE DIPROPIONATE	rxcui:108088	ALCLOMETASONE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	BETAMETHASONE ACETATE	rxcui:1516	BETAMETHASONE ACETATE	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	ChEMBL	33	inhibitor	0.4167275494896388	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.2453629496995069	ESTRADIOL CYPIONATE	rxcui:1000146	ESTRADIOL CYPIONATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.051655358	DEXTROAMPHETAMINE SULFATE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.1296485709523321	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.046303061	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.05068308	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.3125456621172291	ESTROGENS, CONJUGATED SYNTHETIC A	chembl:CHEMBL1201466	ESTROGENS, CONJUGATED SYNTHETIC A	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.06466462	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	HYDROCODONE BITARTRATE	rxcui:142439	HYDROCODONE BITARTRATE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	HYDROCODONE POLISTIREX	rxcui:221107	HYDROCODONE POLISTIREX	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.212152207	OXYMORPHONE HYDROCHLORIDE	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	agonist	0.8751278539282416	BECAPLERMIN	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.079557078	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.067231333	DEXMEDETOMIDINE HYDROCHLORIDE	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1363835616511545	MECLOFENAMATE SODIUM	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	FLURBIPROFEN SODIUM	rxcui:91351	FLURBIPROFEN SODIUM	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.068191781	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.093763699	MECLOFENAMATE SODIUM	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
IMPDH2	hgnc:6053	IMPDH2	ChEMBL	33	inhibitor	2.625383561784724	MYCOPHENOLATE MOFETIL HYDROCHLORIDE	rxcui:237112	MYCOPHENOLATE MOFETIL HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.2263261691193728	TOLBUTAMIDE	rxcui:10635	TOLBUTAMIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.073954467	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.283060222	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.06375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.2083637747448194	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.1389091831632129	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.1241316104862754	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
THRA	hgnc:11796	THRA	ChEMBL	33	agonist	7.501095891	DEXTROTHYROXINE SODIUM	rxcui:40070	DEXTROTHYROXINE SODIUM	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	1.479089330582943	DEZOCINE	rxcui:22713	DEZOCINE	TRUE	FALSE	FALSE
THRA	hgnc:11796	THRA	ChEMBL	33	agonist	1.875273972703375	LEVOTHYROXINE SODIUM	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2035181055647073	PROTOKYLOL HYDROCHLORIDE	ncit:C66496	PROTOKYLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NPC1L1	hgnc:7898	NPC1L1	ChEMBL	33	inhibitor	26.25383561784724	EZETIMIBE	rxcui:341248	EZETIMIBE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.1356787370431382	SOTALOL HYDROCHLORIDE	rxcui:7008	SOTALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.4070362111294147	LEVOBUNOLOL HYDROCHLORIDE	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
GH	hgnc:4261	GH1	ChEMBL	33	inhibitor	1.093909817410302	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
COL4A3	hgnc:2204	COL4A3	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL24A1	hgnc:20821	COL24A1	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL1A2	hgnc:2198	COL1A2	ChEMBL	33	cleavage	0.6250913242344583	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	ChEMBL	33	inhibitor	0.4273880216858854	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA3	hgnc:9532	PSMA3	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA6	hgnc:9535	PSMA6	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.3968833804663227	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.4167275494896388	PANCURONIUM BROMIDE	rxcui:7884	PANCURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.4605936073306534	PANCURONIUM BROMIDE	rxcui:7884	PANCURONIUM BROMIDE	TRUE	FALSE	FALSE
MT-ND5	hgnc:7461	MT-ND5	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFA2	hgnc:7685	NDUFA2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFA11	hgnc:20371	NDUFA11	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFA8	hgnc:7692	NDUFA8	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	ChEMBL	33	agonist	0.2333674277141977	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	0.1930429089547591	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	0.1018248310970158	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
RXRB	hgnc:10478	RXRB	ChEMBL	33	agonist	0.8334550989792776	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.1795134059339983	VORTIOXETINE HYDROBROMIDE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.054695491	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.040703621	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.080781033	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.2841324201065719	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.2651902587661338	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	1.419126249613364	ROLAPITANT HYDROCHLORIDE	rxcui:1673367	ROLAPITANT HYDROCHLORIDE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	0.760980743	PX-102	drugbank:DB15416	PX-102	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	ALLITINIB	ncit:C179280	ALLITINIB	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.2397610558707511	AZD-6918	chembl:CHEMBL3545298	AZD-6918	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.4070362111294147	AZD-6918	chembl:CHEMBL3545298	AZD-6918	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.364636606	AZD-6918	chembl:CHEMBL3545298	AZD-6918	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	ChEMBL	33	inhibitor	0.6908904109959803	AZD-7762	drugbank:DB12242	AZD-7762	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.074443768	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.2287915957982331	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.059532507	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
MT-ND1	hgnc:7455	MT-ND1	ChEMBL	33	inhibitor	0.105015342	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFV3	hgnc:7719	NDUFV3	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA2	hgnc:7685	NDUFA2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFB9	hgnc:7704	NDUFB9	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFAF4	hgnc:21034	NDUFAF4	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	2.282942227638891	RO-3201195	chembl:CHEMBL203567	RO-3201195	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.1715936968486748	ZOTIRACICLIB	ncit:C171725	ZOTIRACICLIB	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1530835896084387	DELUCEMINE	ncit:C76776	DELUCEMINE	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.1356787370431382	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	ChEMBL	33	inhibitor	4.375639269641208	CB-189625	chembl:CHEMBL3707378	CB-189625	FALSE	FALSE	FALSE
RXRB	hgnc:10478	RXRB	ChEMBL	33	agonist	1.944728564284981	IRX-4204	chembl:CHEMBL75133	IRX-4204	FALSE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	ChEMBL	33	inhibitor	3.750547945	GALETERONE	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.116943588	MK-0773	drugbank:DB16244	MK-0773	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	1.019566431761058	MB07811	drugbank:DB05192	MB07811	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.2711239478607289	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.031479419	AT-9283	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	0.2941606231691568	SAPITINIB	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	INSM-18	chembl:CHEMBL3545025	INSM-18	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.7778914257139926	TIRBANIBULIN	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:1528	iuphar.ligand:1528	BIBO3304	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1406455479527531	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.047518255	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1715936968486748	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.073540156	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1442518440541057	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.062139256	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.6482428547616604	TRICIRIBINE PHOSPHATE	ncit:C1262	TRICIRIBINE PHOSPHATE	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	1.093909817410302	TRICIRIBINE PHOSPHATE	ncit:C1262	TRICIRIBINE PHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.3889457128569963	IUPHAR.LIGAND:1514	iuphar.ligand:1514	PEPTIDE YY	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	GSK239512	chembl:CHEMBL3092650	GSK239512	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.5585922471882393	CP-601927	drugbank:DB12244	CP-601927	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.5585922471882393	ALTINICLINE	ncit:C77841	ALTINICLINE	FALSE	FALSE	FALSE
NCBIGENE:1579	hgnc:2642	CYP4A11	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8632	iuphar.ligand:8632	COMPOUND 6 [PMID: 10395480]	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	ChEMBL	33	inhibitor	0.7955707762984013	LOSMAPIMOD	ncit:C96532	LOSMAPIMOD	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.6159257622955366	BARICITINIB	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.2465148884304905	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.525076712	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
FNTA	hgnc:3782	FNTA	ChEMBL	33	inhibitor	2.917092846427472	TIPIFARNIB	ncit:C1703	TIPIFARNIB	FALSE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.3889457128569963	IUPHAR.LIGAND:1504	iuphar.ligand:1504	NEUROPEPTIDE Y	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1591141552596802	NAPROXCINOD	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
METAP2	hgnc:16672	METAP2	ChEMBL	33	inhibitor	0.3281729452230906	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PSMD4	hgnc:9561	PSMD4	ChEMBL	33	inhibitor	0.192335792	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	ChEMBL	33	inhibitor	0.3365876361262467	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB8	hgnc:9545	PSMB8	ChEMBL	33	inhibitor	0.1223955040459079	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMA6	hgnc:9535	PSMA6	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMC1	hgnc:9547	PSMC1	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB4	hgnc:9541	PSMB4	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.035719504	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
PLA2G7	hgnc:9040	PLA2G7	ChEMBL	33	inhibitor	6.563458904461812	RILAPLADIB	ncit:C76401	RILAPLADIB	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.038894571	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1518	iuphar.ligand:1518	[125I]NPY (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.3040984820600068	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.041672755	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	blocker	0.091476779	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNS3	hgnc:6302	KCNS3	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNB2	hgnc:6232	KCNB2	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNH5	hgnc:6254	KCNH5	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCND1	hgnc:6237	KCND1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.013589562	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1620607136904151	GILTERITINIB FUMARATE	rxcui:2105823	GILTERITINIB FUMARATE	TRUE	FALSE	FALSE
KCNV2	hgnc:19698	KCNV2	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNH4	hgnc:6253	KCNH4	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNF1	hgnc:6246	KCNF1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNS2	hgnc:6301	KCNS2	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	agonist	1.944728564284981	SIPONIMOD FUMARATE	ncit:C170378	SIPONIMOD FUMARATE	TRUE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	ChEMBL	33	inhibitor	0.3977853881492006	MOLIBRESIB	ncit:C101538	MOLIBRESIB	FALSE	FALSE	FALSE
BRDT	hgnc:1105	BRDT	ChEMBL	33	inhibitor	0.5357925636295356	BIRABRESIB	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	3.500511415712966	RIMEGEPANT SULFATE	rxcui:2282322	RIMEGEPANT SULFATE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.2365210416022274	ADOPRAZINE	ncit:C81482	ADOPRAZINE	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.8334550989792776	TAMIBAROTENE	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
FDPS	hgnc:3631	FDPS	ChEMBL	33	inhibitor	3.500511415712966	MINODRONIC ACID	ncit:C81673	MINODRONIC ACID	FALSE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	FOSTEMSAVIR TROMETHAMINE	rxcui:2380374	FOSTEMSAVIR TROMETHAMINE	TRUE	FALSE	FALSE
PRPS1	hgnc:9462	PRPS1	CIViC	10-Apr-24	NULL	0.3889457128569962	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	4.699760697022038	SELPERCATINIB	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
TTR	hgnc:12405	TTR	ChEMBL	33	inhibitor	17.50255707856483	INOTERSEN	rxcui:2099289	INOTERSEN	TRUE	FALSE	FALSE
KLKB1	hgnc:6371	KLKB1	ChEMBL	33	inhibitor	1.875273972703375	HUMAN C1-ESTERASE INHIBITOR	ncit:C87730	HUMAN C1-ESTERASE INHIBITOR	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	BARNIDIPINE	rxcui:39879	MEPIRODIPINE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.3454452054979901	TRASTUZUMAB DERUXTECAN	rxcui:2267574	FAM-TRASTUZUMAB DERUXTECAN-NXKI	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.03151721	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	2.187819634820604	MAGNESIUM OXYBATE	rxcui:2387308	MAGNESIUM OXYBATE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.4167275494896388	NAQUOTINIB	ncit:C115110	NAQUOTINIB	FALSE	FALSE	TRUE
IL23A	hgnc:15488	IL23A	ChEMBL	33	inhibitor	2.187819634820604	MIRIKIZUMAB	rxcui:2668384	MIRIKIZUMAB	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
PPP2CA	hgnc:9299	PPP2CA	ChEMBL	33	inhibitor	21.00306849	LB-100	drugbank:DB15412	LB-100	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	CIViC	10-Apr-24	NULL	0.3365876361262467	B-RAF/VEGFR-2 INHIBITOR RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
PDE4	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	1.193356164447602	UK-500001	drugbank:DB12837	UK-500001	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	agonist	0.042619863	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.2778183663264258	PERZINFOTEL	ncit:C72122	PERZINFOTEL	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.1209854175937661	PERZINFOTEL	ncit:C72122	PERZINFOTEL	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.2586584789935689	PERZINFOTEL	ncit:C72122	PERZINFOTEL	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	agonist	0.039068208	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.1029562181092049	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
CXCL12	hgnc:10672	CXCL12	ChEMBL	33	inhibitor	13.12691780892362	OLAPTESED PEGOL	ncit:C99379	OLAPTESED PEGOL	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.057574201	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
CTAG1A	hgnc:24198	CTAG1A	ChEMBL	33	vaccine	17.50255707856483	RASDEGAFUSP ALFA	ncit:C170362	RASDEGAFUSP ALFA	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	2.187819634820604	SENAPARIB	ncit:C168601	SENAPARIB	FALSE	FALSE	FALSE
PDGFB	hgnc:8800	PDGFB	CIViC	10-Apr-24	NULL	0.3500511415712966	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	LACIDIPINE	rxcui:28382	LACIDIPINE	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.036770078	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
CFLAR	hgnc:1876	CFLAR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2983390411119005	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
DHFR	hgnc:2861	DHFR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	2.734774543525755	PRALATREXATE	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
APH1B	hgnc:24080	APH1B	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.009762908	UNII-DRL23N424R	ncit:C116872	OSUGACESTAT	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PARP2	hgnc:272	PARP2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	2.187819634820604	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2083637747448194	PKI-590	ncit:C84837	PI3K/MTOR KINASE INHIBITOR PF-04691502	FALSE	FALSE	TRUE
PARP2	hgnc:272	PARP2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3241214273808302	1207456-01-6	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
PARP2	hgnc:272	PARP2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.250182648468916	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.073540156	GDC-0944	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
TNFSF11	hgnc:11926	TNFSF11	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	43.75639269641208	DENOSUMAB	rxcui:993449	DENOSUMAB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	1.090323227845022	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.1141471113819445	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	5-METHOXYTRYPTAMINE	rxcui:1426888	5-METHOXYTRYPTAMINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00224853	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TDR78277	chembl:CHEMBL1308346	CHEMBL:CHEMBL1308346	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	CIViC	10-Apr-24	NULL	0.008230043	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CD28	hgnc:1653	CD28	DTC	9/2/20	NULL	1.166837138570988	3-HYDROXYANTHRANILIC ACID	drugbank:DB03644	3-HYDROXYANTHRANILIC ACID	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	NILE RED	chembl:CHEMBL144472	NILE RED	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.007717177	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	HYDROXYSTILBAMIDINE ISETHIONATE	ncit:C65871	HYDROXYSTILBAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	3-METHYLCHOLANTHRENE	chembl:CHEMBL40583	3-METHYLCHOLANTHRENE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.169927739	QUINALDINE BLUE	chembl:CHEMBL1433292	QUINALDINE BLUE	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.090064616	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.025865848	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	DTC	9/2/20	NULL	1.458546423213736	BENZYL ISOTHIOCYANATE	drugbank:DB16860	BENZYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.2917092846427472	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	TDR77135	chembl:CHEMBL1529479	CHEMBL:CHEMBL1529479	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.4700175174550658	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1861974157294131	ILEPCIMIDE	ncit:C72810	ILEPCIMIDE	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	CIViC	10-Apr-24	NULL	0.5173169579871378	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	OCTYL_GALLATE	chembl:CHEMBL277346	OCTYL_GALLATE	FALSE	FALSE	FALSE
RNASE1	hgnc:10044	RNASE1	DTC	9/2/20	NULL	105.0153424713889	CYTIDINE 3'-PHOSPHATE	drugbank:DB01961	CYTIDINE 3'-MONOPHOSPHATE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006233104	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.016156207	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.011472071	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	ETHACRIDINE LACTATE	rxcui:4107	ETHACRIDINE LACTATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	GNF-PF-4967	chembl:CHEMBL585827	CHEMBL:CHEMBL585827	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	CIViC	10-Apr-24	NULL	1.467605717767858	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	1.230648544586589	ELACRIDAR	ncit:C73318	ELACRIDAR	FALSE	FALSE	FALSE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	0.9376369863516874	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
HRH4	hgnc:17383	HRH4	DTC	9/2/20	NULL	1.101559536413171	HISTAMINE	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1426838892274307	DINITRO CRESOL	chembl:CHEMBL419564	DINITRO CRESOL	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.043866058	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1136529680426287	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	MERCAPTOPURINE HYDRATE	chembl:CHEMBL1200751	MERCAPTOPURINE	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.076098074	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
CLK1	hgnc:2068	CLK1	DTC	9/2/20	inhibitor	0.2625383561784725	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	ARSANILIC ACID	ncit:C29883	ARSANILIC ACID	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.045265234	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.5303805175322676	PIRINIXIC ACID	iuphar.ligand:2666	PIRINIXIC ACID	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.084770219	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.1682938180631234	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	MELITRACEN	rxcui:446248	MELITRACEN	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	2.187819634820604	REDIOCIDE A	chembl:CHEMBL454246	REDIOCIDE A	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.048394167	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.3922986931402463	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.019107595	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	inhibitor	0.062509132	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	1.458546423213736	DICARBONODITHIOIMIDIC DIAMIDE	chembl:CHEMBL501562	DICARBONODITHIOIMIDIC DIAMIDE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.090530468	DIOXYBENZONE	rxcui:23350	DIOXYBENZONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	GNF-PF-3546	chembl:CHEMBL598680	CHEMBL:CHEMBL598680	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011738804	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CHLOROGENIC ACID	rxcui:1311387	CHLOROGENIC ACID	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.050879526	NSC-36398	chembl:CHEMBL483206	CHEMBL:CHEMBL483206	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.1715936968486748	JNK INHIBITOR VIII	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.018031481	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	GNF-PF-806	chembl:CHEMBL547101	CHEMBL:CHEMBL547101	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.005879918	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	TCMDC-124317	chembl:CHEMBL586937	CHEMBL:CHEMBL586937	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.050488145	FALNIDAMOL	ncit:C80868	FALNIDAMOL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007813642	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00445925	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.1346350544504987	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	KETANSERIN TARTRATE	ncit:C2036	KETANSERIN TARTRATE	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.010344301	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.058602312	TDR77585	chembl:CHEMBL1333386	CHEMBL:CHEMBL1333386	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-710	chembl:CHEMBL596839	CHEMBL:CHEMBL596839	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	SJ000117451	chembl:CHEMBL592123	CHEMBL:CHEMBL592123	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	S(+)-ISOPROTERENOL-BITARTRATE	chembl:CHEMBL1257092	CHEMBL:CHEMBL1257092	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.018071819	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	PIFEXOLE	ncit:C76774	PIFEXOLE	FALSE	FALSE	FALSE
PTPN5	hgnc:9657	PTPN5	DTC	9/2/20	NULL	7.501095890813499	MESO-2,3-DIMERCAPTOSUCCINIC ACID	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	Z-PRO-PROLINAL	drugbank:DB03535	Z-PRO-PROLINAL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	NSC-47924	chembl:CHEMBL1269845	CHEMBL:CHEMBL1269845	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	1.479089330582943	12-EPI-SALVINORIN B ETHOXYMETHYL ETHER	chembl:CHEMBL1941031	CHEMBL:CHEMBL1941031	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	0.4339476961627644	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.082950507	CLINAFLOXACIN	ncit:C74372	CLINAFLOXACIN	FALSE	FALSE	FALSE
AKR1C1	hgnc:384	AKR1C1	DTC	9/2/20	NULL	17.50255707856483	3,5-DICHLOROSALICYLIC ACID	chembl:CHEMBL449129	CHEMBL:CHEMBL449129	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.061773731	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	BENZETHONIUM	rxcui:1390	BENZETHONIUM	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	MECLIZINE	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	IODOFORM	rxcui:27748	IODOFORM	FALSE	FALSE	FALSE
PAK3	hgnc:8592	PAK3	DTC	9/2/20	inhibitor	1.312691780892362	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	TCMDC-125620	chembl:CHEMBL530291	CHEMBL:CHEMBL530291	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.012004497	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00575742	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001581175	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003604068	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.02617531	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	1.981421556063943	CYNAROPICRIN	chembl:CHEMBL374146	CYNAROPICRIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.010742159	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	DTC	9/2/20	NULL	4.039051633514961	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	SJ000120081	chembl:CHEMBL606532	CHEMBL:CHEMBL606532	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.2638576444004749	PERSEITOL	chembl:CHEMBL1597273	PERSEITOL	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.070010228	2,3,7,8-TETRACHLORODIBENZO-P-DIOXIN	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.024896952	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW682841X	chembl:CHEMBL206544	GW682841X	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	OLVANIL	ncit:C166774	OLVANIL	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	inhibitor	0.011414711	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
SIRT3	hgnc:14931	SIRT3	DTC	9/2/20	NULL	8.751278539282415	NIACINAMIDE	rxcui:7405	NIACINAMIDE	TRUE	FALSE	FALSE
PRMT1	hgnc:5187	PRMT1	DTC	9/2/20	NULL	4.375639269641208	EOSIN	drugbank:DB13706	EOSIN	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.078136416	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	GETIACAULEIN	chembl:CHEMBL467590	GETIACAULEIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TCMDC-125472	chembl:CHEMBL587389	CHEMBL:CHEMBL587389	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.026045472	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.015959778	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	FORMESTANE	rxcui:15070	FORMESTANE	FALSE	FALSE	FALSE
CSNK1E	hgnc:2453	CSNK1E	DTC	9/2/20	NULL	0.7292732116068681	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	DTC	9/2/20	NULL	0.2403097081725148	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009170044	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
GABRB2	hgnc:4082	GABRB2	DTC	9/2/20	NULL	0.07631929	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	DTC	9/2/20	NULL	0.072125922	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00389812	AMLODIPINE BESYLATE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	CYCLOVALONE	ncit:C81040	CYCLOVALONE	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	DTC	9/2/20	NULL	0.088695391	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	TRIPARANOL	ncit:C152752	TRIPARANOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	ICOSAPENT	rxcui:90	EICOSAPENTAENOIC ACID	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	OCTRIZOLE	ncit:C80799	OCTRIZOLE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00747866	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.061412481	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	Z-PRO-PROLINAL	drugbank:DB03535	Z-PRO-PROLINAL	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.2792961235941196	ISOXANTHOPTERIN	chembl:CHEMBL464251	ISOXANTHOPTERIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	SPERMIDINE	rxcui:1483262	SPERMIDINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TETRACONAZOLE	chembl:CHEMBL2137654	TETRACONAZOLE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	PHTHALYLSULFATHIAZOLE	rxcui:33632	PHTHALYLSULFATHIAZOLE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.068369364	PALMITOYL-CARNITINE	chembl:CHEMBL301722	PALMITOYL-CARNITINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.046673486	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.008728004	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.069089041	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1238388472539964	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1773907812016706	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.4861821410712454	SKF-38393	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.2651902587661338	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-4967	chembl:CHEMBL585827	CHEMBL:CHEMBL585827	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.029465584	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	DEFERIPRONE	rxcui:11645	DEFERIPRONE	TRUE	FALSE	FALSE
NPY1R	hgnc:7956	NPY1R	DTC	9/2/20	NULL	5.250767123569449	BMS-193885	chembl:CHEMBL324554	CHEMBL:CHEMBL324554	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.00731101	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	NELFINAVIR MESYLATE	rxcui:266565	NELFINAVIR MESYLATE	TRUE	FALSE	FALSE
PDK1	hgnc:8809	PDK1	DTC	9/2/20	NULL	2.500365296937833	3-HYDROXYANTHRANILIC ACID	drugbank:DB03644	3-HYDROXYANTHRANILIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BROMEBRIC ACID	ncit:C72089	BROMEBRIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.016602341	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	4,4'-DITHIODIPYRIDINE	chembl:CHEMBL1232076	CHEMBL:CHEMBL1232076	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.013505059	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	6ALPHA-METHYLPREDNISOLONE ACETATE	chembl:CHEMBL1364144	METHYLPREDNISOLONE ACETATE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	AZARIBINE	ncit:C1008	AZARIBINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
PLK3	hgnc:2154	PLK3	DTC	9/2/20	NULL	0.04321619	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.013229446	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.000743461	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006381584	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	DNDI1417607	chembl:CHEMBL1588679	CHEMBL:CHEMBL1588679	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	LIDOFLAZINE	rxcui:6390	LIDOFLAZINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.008475815	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.008799677	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.056097939	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.019724895	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
PPP1CA	hgnc:9281	PPP1CA	DTC	9/2/20	NULL	1.166837138570989	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.032899543	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	KARANJIN	chembl:CHEMBL208484	KARANJIN	FALSE	FALSE	FALSE
TRPC5	hgnc:12337	TRPC5	DTC	9/2/20	NULL	4.200613698855561	3-MORPHOLINOSYDNONIMINE HCL	chembl:CHEMBL538104	CHEMBL:CHEMBL538104	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	IODOPHTHALEIN	chembl:CHEMBL1160008	IODOPHTHALEIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	COUMAPHOS	ncit:C76867	COUMAPHOS	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	PHENSERINE	drugbank:DB04892	PHENSERINE	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.9907107780319716	MORUSINOL	chembl:CHEMBL1719948	MORUSINOL	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
RCE1	hgnc:13721	RCE1	DTC	9/2/20	NULL	1.500219178	FLUNARIZINE DIHYDROCHLORIDE	chembl:CHEMBL539027	FLUNARIZINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.038981196	ACETOPHENAZINE	rxcui:16735	ACETOPHENAZINE	TRUE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.2500365296937833	GNF-PF-1399	chembl:CHEMBL578504	CHEMBL:CHEMBL578504	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DAZOMET	chembl:CHEMBL1407826	DAZOMET	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	GNF-PF-3149	chembl:CHEMBL582507	CHEMBL:CHEMBL582507	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.027929612	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.040235763	DIACEREIN	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
IL6R	hgnc:6019	IL6R	DTC	9/2/20	NULL	0.1615620653405984	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	TCMDC-123762	chembl:CHEMBL547483	CHEMBL:CHEMBL547483	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	CYCLOVALONE	ncit:C81040	CYCLOVALONE	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.1250182648468916	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.2117244807890907	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	AZARIBINE	ncit:C1008	AZARIBINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	TCMDC-125620	chembl:CHEMBL530291	CHEMBL:CHEMBL530291	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.023151531	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	GNF-PF-1731	chembl:CHEMBL581251	CHEMBL:CHEMBL581251	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.6105543166941221	TCMDC-124321	chembl:CHEMBL526952	CHEMBL:CHEMBL526952	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	DNDI1417336	chembl:CHEMBL1472891	CHEMBL:CHEMBL1472891	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	GW305074X	chembl:CHEMBL1880739	GW305074X	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	GNF-PF-3201	chembl:CHEMBL581872	CHEMBL:CHEMBL581872	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.016429184	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	TCMDC-125556	chembl:CHEMBL587092	CHEMBL:CHEMBL587092	FALSE	FALSE	FALSE
S1PR4	hgnc:3170	S1PR4	DTC	9/2/20	NULL	0.5834185692854945	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
PLD1	hgnc:9067	PLD1	DTC	9/2/20	NULL	0.5385402178019949	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	DEGUELIN	ncit:C63666	DEGUELIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.058602312	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.010287553	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.4861821410712453	NSC-67746	chembl:CHEMBL333177	CHEMBL:CHEMBL333177	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.024513385	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.2778183663264259	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.303074581	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.6908904109959803	CCT244747	iuphar.ligand:8215	CCT244747	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	SJ000044417	chembl:CHEMBL609438	CHEMBL:CHEMBL609438	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004427291	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	SJ000032151	chembl:CHEMBL592600	CHEMBL:CHEMBL592600	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.1495945049449986	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV666093	chembl:CHEMBL585686	CHEMBL:CHEMBL585686	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003291811	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.006286838	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.075010959	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	GNF-PF-1509	chembl:CHEMBL576412	CHEMBL:CHEMBL576412	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.072125922	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	PIPERIDOLATE	rxcui:59064	PIPERIDOLATE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	TCMDC-123920	chembl:CHEMBL1606	CHEMBL:CHEMBL1606	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006054153	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.024275391	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.006359941	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.093098708	N-(4-NITROPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1574420	CHEMBL:CHEMBL1574420	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00731101	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.051478109	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DAMNACANTHAL	ncit:C1480	DAMNACANTHAL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	N,N-HEXAMETHYLENEAMILORIDE	iuphar.ligand:1192	5-(N,N-HEXAMETHYLENE)-AMILORIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.01036063	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.020936073	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	BENZO[B]FLUORANTHENE	chembl:CHEMBL1337502	BENZO[B]FLUORANTHENE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	SJ000032152	chembl:CHEMBL590665	CHEMBL:CHEMBL590665	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	MINAPRINE HYDROCHLORIDE	rxcui:236400	MINAPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	TCMDC-124317	chembl:CHEMBL586937	CHEMBL:CHEMBL586937	FALSE	FALSE	FALSE
UBA2	hgnc:30661	UBA2	DTC	9/2/20	NULL	1.312691780892362	PEVONEDISTAT	ncit:C77906	PEVONEDISTAT	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.801643836	6-HYDROXYFLAVONOL	chembl:CHEMBL210411	CHEMBL:CHEMBL210411	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.025489161	OXIDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.007946076	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.045579576	2-MESATP	iuphar.ligand:1711	2MESATP	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004579424	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	PROSULTIAMINE	ncit:C82256	PROSULTIAMINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002542744	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.039479452	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	DNDI1417215	chembl:CHEMBL1390650	CHEMBL:CHEMBL1390650	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2035181055647073	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	NSC-659162	chembl:CHEMBL471005	CHEMBL:CHEMBL471005	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002269228	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2134458180312784	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	DTC	9/2/20	NULL	0.8975670296699914	SB-207710	iuphar.ligand:257	SB 207710	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.031784305	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.00502947	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	CINOBUFOTALIN	ncit:C151929	CINOBUFOTALIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	BROMOCICLEN	ncit:C74161	BROMOCICLEN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE	chembl:CHEMBL1599728	2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008681824	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	2-METHOXYPHENAZINE	chembl:CHEMBL1420181	CHEMBL:CHEMBL1420181	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.4861821410712453	GNF-PF-4746	chembl:CHEMBL584868	CHEMBL:CHEMBL584868	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	NSC-36398	chembl:CHEMBL483206	CHEMBL:CHEMBL483206	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.04321619	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	TESMILIFENE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW795493X	chembl:CHEMBL273564	GW795493X	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.034229251	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	IPCONAZOLE	chembl:CHEMBL3185422	IPCONAZOLE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.007196775	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.003739863	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	0.1041818873724097	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	ETHACRIDINE LACTATE	rxcui:4107	ETHACRIDINE LACTATE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005085489	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1000146118775133	MUNDULONE ACETATE	chembl:CHEMBL1372368	MUNDULONE ACETATE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	GNF-PF-2947	chembl:CHEMBL581677	CHEMBL:CHEMBL581677	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	STROPHANTHIDIN	chembl:CHEMBL111743	STROPHANTHIDIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.040766825	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-806	chembl:CHEMBL547101	CHEMBL:CHEMBL547101	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1131630845596864	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.05309168	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.002355872	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	AROMATICIN	chembl:CHEMBL494255	AROMATICIN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.040328473	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.010626932	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	GNF-PF-2335	chembl:CHEMBL601146	CHEMBL:CHEMBL601146	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014993624	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	CALANOLIDE A	drugbank:DB04886	CALANOLIDE A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	GNF-PF-4746	chembl:CHEMBL584868	CHEMBL:CHEMBL584868	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.034118045	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	7-METHOXY-BAPTIGENIN	chembl:CHEMBL583578	CHEMBL:CHEMBL583578	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.023420014	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.019889269	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.007244436	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.020391329	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.074797252	2'-HYDROXYCHALCONE	chembl:CHEMBL32147	2'-HYDROXYCHALCONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.034590034	QUETIAPINE	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.1666910197958555	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.029399592	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	DTC	9/2/20	NULL	0.1052961321571413	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.020268015	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.009237803	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	SB-222200	iuphar.ligand:2131	SB 222200	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	LOXAPINE SUCCINATE	rxcui:6476	LOXAPINE SUCCINATE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV667492	chembl:CHEMBL2028068	CHEMBL:CHEMBL2028068	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	4-PHENYLPHENOL	chembl:CHEMBL73380	CHEMBL:CHEMBL73380	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.023110771	DEQUALINIUM	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1296485709523321	SKF-38393	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	CUPRIC CHLORIDE	rxcui:150596	COPPER CHLORIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	ZARDAVERINE	ncit:C66686	ZARDAVERINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001976425	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	SK&F-82958	iuphar.ligand:10742	SKF-82958	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	MG-132	iuphar.ligand:8616	MG-132	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.017709164	Amoxapine	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	1-NITROPYRENE	chembl:CHEMBL167395	1-NITROPYRENE	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.071341945	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.1166837138570988	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	FDA	10-Apr-24	NULL	0.09869863	Azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.022136455	Darifenacin	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.027635616	Eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1415301111474245	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1415301111474245	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.9460841664089098	UFT	ncit:C9506	TEGAFUR-URACIL	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.1182605208011137	ICI 182,780	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.070956312	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
GABPA	hgnc:4071	GABPA	NCI	14-Sep-17	NULL	0.201178817	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.045658845	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.042006137	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
GATA4	hgnc:4173	GATA4	NCI	14-Sep-17	NULL	1.458546423213736	ANTHRACYCLINES	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	0.2243917574174978	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.072125922	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.1143957978991165	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1190650141398968	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
HCK	hgnc:4840	HCK	NCI	14-Sep-17	NULL	0.066676408	STI571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
HAS3	hgnc:4820	HAS3	NCI	14-Sep-17	NULL	0.5770073762164231	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.1051204629343233	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.1973972602845657	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.016647962	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.086361301	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.028397875	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	2.442217266776488	DON	ncit:C427	DIAZOOXONORLEUCINE	FALSE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.09972967	VCR	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
HSPA8	hgnc:5241	HSPA8	NCI	14-Sep-17	NULL	0.3860858179095184	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	NCI	14-Sep-17	NULL	0.1262203635473425	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
HSPA9	hgnc:5244	HSPA9	NCI	14-Sep-17	NULL	157.5230137070835	MKT-077	ncit:C2731	RHODACYANINE ANALOG MKT-077	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	1.250182648468916	MONOCLONAL ANTIBODY 17-1A	rxcui:80726	EDRECOLOMAB	FALSE	FALSE	FALSE
IGFBP1	hgnc:5469	IGFBP1	NCI	14-Sep-17	NULL	0.6731752722524935	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.2019525816757481	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.9376369863516875	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.061737415	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.1143957978991165	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.1973972602845657	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
LPAR2	hgnc:3168	LPAR2	NCI	14-Sep-17	NULL	0.760980743	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.167488584	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
LOH19CR1	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.2885036881082115	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
LIPE	hgnc:6621	LIPE	NCI	14-Sep-17	NULL	0.8204323630577265	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
LTB4R	hgnc:6713	LTB4R	NCI	14-Sep-17	NULL	0.2524407270946851	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1630673019742065	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.5357925636295356	RECOMBINANT INTERLEUKIN	ncit:C593	RECOMBINANT INTERLEUKIN	FALSE	FALSE	FALSE
LPO	hgnc:6678	LPO	NCI	14-Sep-17	NULL	0.8078103267029924	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.1342907192728759	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
MDK	hgnc:6972	MDK	NCI	14-Sep-17	NULL	1.154014752432846	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	1.312691780892362	INTERFERON BETA	chembl:CHEMBL2108510	INTERFERON BETA	TRUE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	5.834185692854944	INCOMPLETE FREUND&APOS;S ADJUVANT	ncit:C1573	INCOMPLETE FREUND'S ADJUVANT	FALSE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.2282942227638891	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.3500511415712967	RHIL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
MT-CO1	hgnc:7419	MT-CO1	NCI	14-Sep-17	NULL	3.182283105193606	MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.1355619739303644	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	0.300043836	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.7292732116068681	GOSERELIN	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.2243917574174979	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.1767935058440892	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.016253729	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.7778914257139926	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.07767407	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.055329474	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.1027547382303219	ANTI-CANCER AGENTS	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.7192831676122533	EO9	ncit:C1087	APAZIQUONE	FALSE	FALSE	FALSE
OCLN	hgnc:8104	OCLN	NCI	14-Sep-17	NULL	1.154014752432846	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PI3	hgnc:8947	PI3	NCI	14-Sep-17	NULL	1.779921058837101	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.023151531	CPT-11	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.046303061	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
PLAT	hgnc:9051	PLAT	NCI	14-Sep-17	NULL	0.1909369863116163	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.042898424	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.016027983	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PTGER4	hgnc:9596	PTGER4	NCI	14-Sep-17	NULL	0.6177373086552295	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
PTCH1	hgnc:9585	PTCH1	NCI	14-Sep-17	NULL	0.2885036881082115	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
LEP	hgnc:6553	LEP	PharmGKB	4/5/24	NULL	0.1562728310586145	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
HMGCS2	hgnc:5008	HMGCS2	PharmGKB	4/5/24	NULL	1.141471113819445	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	PharmGKB	4/5/24	NULL	0.02302968	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	PharmGKB	4/5/24	NULL	0.06525008	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.3977853881492007	amodiaquine	rxcui:720	AMODIAQUINE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.2625383561784725	amodiaquine	rxcui:720	AMODIAQUINE	FALSE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	0.4640829528407342	halothane	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
ALDH1L1	hgnc:3978	ALDH1L1	PharmGKB	4/5/24	NULL	10.50153425	methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.008854582	tiotropium	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.445925021	calcium	rxcui:1895	CALCIUM	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.1842374429322613	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.016780975	brexpiprazole	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00202529	vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.023493365	ropivacaine	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.009788902	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006525935	terfenadine	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.091636424	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.9723642821424908	sibutramine	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.525076712	carbasalate calcium	hemonc:116701	CARBASALATE CALCIUM	FALSE	FALSE	FALSE
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.3106962795011509	troglitazone	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.1302273592155121	fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.097236428	dolutegravir	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
ARAF	hgnc:646	ARAF	PharmGKB	4/5/24	NULL	0.075369863	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	PharmGKB	4/5/24	NULL	0.032899543	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	PharmGKB	4/5/24	NULL	0.015019357	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ADAMTS18	hgnc:17110	ADAMTS18	PharmGKB	4/5/24	NULL	0.9211872146613069	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.3571950424196904	rasagiline	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.041872146	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPK9	hgnc:6886	MAPK9	PharmGKB	4/5/24	NULL	0.0287871	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	PharmGKB	4/5/24	NULL	0.017380891	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
LTA4H	hgnc:6710	LTA4H	PharmGKB	4/5/24	NULL	0.5303805175322677	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.063110182	hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.182318303	isoniazid	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.078252863	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.038693936	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
CDX2	hgnc:1806	CDX2	PharmGKB	4/5/24	NULL	0.6482428547616604	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
CCDC70	hgnc:25303	CCDC70	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
DMD	hgnc:2928	DMD	PharmGKB	4/5/24	NULL	15.00219178	golodirsen	rxcui:2267207	GOLODIRSEN	TRUE	FALSE	FALSE
DMD	hgnc:2928	DMD	PharmGKB	4/5/24	NULL	7.501095891	casimersen	rxcui:2480096	CASIMERSEN	TRUE	FALSE	FALSE
SSU72	hgnc:25016	SSU72	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.018019105	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
DLG5	hgnc:2904	DLG5	PharmGKB	4/5/24	NULL	0.9723642821424907	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1193356164447602	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1193356164447602	propylthiouracil	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1491695205559502	flupirtine	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
CDC5L	hgnc:1743	CDC5L	PharmGKB	4/5/24	NULL	0.2822993077187876	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.2785552850699973	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.6819178082557728	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	0.05751114	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.1835932560688619	vortioxetine	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
ETS2	hgnc:3489	ETS2	PharmGKB	4/5/24	NULL	0.2258394461750301	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.019629036	eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	inhibitor	0.3889457128569963	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.1041818873724097	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	TALC	12-May-16	inhibitor	0.2917092846427472	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.1902451856365742	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.29374921	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.2545826484154885	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	1.000146118775133	PF-4217903	chembl:CHEMBL2001019	PF-04217903	FALSE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	TALC	12-May-16	NULL	0.066297565	ILOPROST	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	TALC	12-May-16	agonist	8.751278539282417	DULANERMIN	ncit:C1685	DULANERMIN	FALSE	TRUE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	TALC	12-May-16	agonist	5.834185692854944	CONATUMUMAB	ncit:C71015	CONATUMUMAB	FALSE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
UNIPROT:Q9NYA1	hgnc:11240	SPHK1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	ABC294640	ncit:C98278	OPAGANIB	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	ADL5747	iuphar.ligand:9003	ADL5747	TRUE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	3.889457128569962	AFUTUZUMAB	rxcui:974779	OBINUTUZUMAB	TRUE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	0.192335792	AZD-6765	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.5173169579871378	AZD-6765	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
UNIPROT:P19838	hgnc:7794	NFKB1	TdgClinicalTrial	Jan-14	NULL	0.1842374429322613	BARDOXOLONE	ncit:C48382	BARDOXOLONE	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.016131389	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.020084536	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.026519026	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	0.086361301	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.2218633995874415	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1025540453822158	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P15509	hgnc:2435	CSF2RA	TdgClinicalTrial	Jan-14	NULL	11.66837138570988	RECOMBINANT GM-CSF	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
UNIPROT:O15123	hgnc:485	ANGPT2	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	REGN910	chembl:CHEMBL2108678	NESVACUMAB	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.050879526	GLYCOPYRRONIUM BROMIDE	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.085378327	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P31751	hgnc:392	AKT2	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	RX-0201	ncit:C88335	ARCHEXIN	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	RUBITECAN	ncit:C1485	RUBITECAN	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.036531311	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	2.423430980108977	SOLANEZUMAB	ncit:C88585	SOLANEZUMAB	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	TAS-108	drugbank:DB05966	TAS-108	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.7955707762984014	TALAMPANEL	ncit:C38139	TALAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P48058	hgnc:4574	GRIA4	TdgClinicalTrial	Jan-14	NULL	0.596678082	TALAMPANEL	ncit:C38139	TALAMPANEL	FALSE	FALSE	FALSE
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.652269208	TG101348	rxcui:2197490	FEDRATINIB	TRUE	FALSE	TRUE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.1530835896084387	TINZAPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	TINZAPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.400821918	HE3286	drugbank:DB05212	HE3286	FALSE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	TRIPTORELIN PAMOATE	rxcui:338529	TRIPTORELIN PAMOATE	TRUE	FALSE	FALSE
UNIPROT:Q08431	hgnc:7036	MFGE8	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	TRIAB	ncit:C2606	MONOCLONAL ANTIBODY 11D10 ANTI-IDIOTYPE VACCINE	FALSE	FALSE	FALSE
UNIPROT:P52564	hgnc:6846	MAP2K6	TdgClinicalTrial	Jan-14	NULL	0.7501095890813498	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
UNIPROT:P16109	hgnc:10721	SELP	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	YSPSL	drugbank:DB06256	RPSGL-IG	FALSE	FALSE	FALSE
UNIPROT:P09917	hgnc:435	ALOX5	TdgClinicalTrial	Jan-14	NULL	1.887530665335423	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
UNIPROT:P28702	hgnc:10478	RXRB	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
UNIPROT:P42081	hgnc:1705	CD86	TdgClinicalTrial	Jan-14	NULL	0.5303805175322677	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
UNIPROT:P01730	hgnc:1678	CD4	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
UNIPROT:Q95460	hgnc:4975	MR1	TdgClinicalTrial	Jan-14	NULL	4.773424657790409	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.038765353	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.055563673	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.06757744	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.059297201	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1070492787679806	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.1193356164447602	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P06241	hgnc:4037	FYN	TEND	1-Aug-11	NULL	0.075768645	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.068847471	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.09741683	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	CARBINOXAMINE	rxcui:20220	CARBINOXAMINE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.1013661606866689	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.089501712	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.100976291	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P02461	hgnc:2201	COL3A1	TEND	1-Aug-11	NULL	2.812910959055062	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P08123	hgnc:2198	COL1A2	TEND	1-Aug-11	NULL	0.6250913242344583	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.076934317	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.091583148	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.021715331	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TEND	1-Aug-11	NULL	3.500511415712966	ALOSETRON	rxcui:85248	ALOSETRON	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.7721716358190367	ALMOTRIPTAN	rxcui:279645	ALMOTRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	1.479089330582943	DEZOCINE	rxcui:22713	DEZOCINE	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.028078969	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:P31785	hgnc:6010	IL2RG	TEND	1-Aug-11	NULL	0.5250767123569451	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
UNIPROT:Q9NPF7	hgnc:15488	IL23A	TEND	1-Aug-11	NULL	1.640864726115453	USTEKINUMAB	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	CIViC	10-Apr-24	NULL	0.2486158675932504	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.6105543166941221	DIPIVEFRIN	rxcui:23410	DIPIVEFRIN	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.1665148136438514	GUANFACINE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	CIViC	10-Apr-24	NULL	0.069454592	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TEND	1-Aug-11	NULL	0.2812910959055062	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TEND	1-Aug-11	NULL	0.8468979231563629	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P15559	hgnc:2874	NQO1	TEND	1-Aug-11	NULL	0.069638821	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.150021918	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.073266518	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TEND	1-Aug-11	NULL	0.3621218705909965	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
DKK1	hgnc:2891	DKK1	CIViC	10-Apr-24	NULL	5.834185692854944	LEVOLEUCOVORIN	rxcui:877015	LEVOLEUCOVORIN	TRUE	FALSE	TRUE
UNIPROT:Q9Y478	hgnc:9378	PRKAB1	TEND	1-Aug-11	NULL	1.009762908	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
UNIPROT:P00734	hgnc:3535	F2	TEND	1-Aug-11	NULL	0.047647615	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P38435	hgnc:4247	GGCX	TEND	1-Aug-11	NULL	0.7242437411819931	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.3351553483129436	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.067839369	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.032154116	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	CIViC	10-Apr-24	NULL	0.9723642821424906	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:O60894	hgnc:9843	RAMP1	TEND	1-Aug-11	NULL	3.750547945406749	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TEND	1-Aug-11	NULL	0.1396480617970598	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	1.029562181092048	NEOSTIGMINE	rxcui:7315	NEOSTIGMINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.837888371	OXYPHENONIUM	rxcui:7818	OXYPHENONIUM	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.064347636	PERGOLIDE	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	1.790034246671403	PRACTOLOL	rxcui:8620	PRACTOLOL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.009659248	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	7.501095891	PIPECURONIUM	rxcui:33742	PIPECURONIUM	TRUE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.33338204	Rocilinostat	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	0.5527123287967842	CF502	iuphar.ligand:5601	MRS3558	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.500219178	SGX523	ncit:C74062	MET TYROSINE KINASE INHIBITOR SGX523	FALSE	FALSE	TRUE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.2112984757975633	GSK2110183	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	CIViC	10-Apr-24	NULL	0.3704244884352345	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
APOPTOSIS INHIBITOR SURVIVIN	hgnc:593	BIRC5	TTD	2020.06.01	NULL	0.596678082	DPX-Survivac	ncit:C97951	MAVEROPEPIMUT-S	FALSE	FALSE	FALSE
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	1.750255707856483	Interferon alfa-n3	rxcui:612937	INTERFERON ALFA-N3	TRUE	TRUE	TRUE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.8204323630577265	Human interleukin-2	drugbank:DB14865	HUMAN INTERLEUKIN-2	FALSE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	1.346350544504987	DA-6886	drugbank:DB12853	DA-6886	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.1900426678745596	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
MYOSTATIN	hgnc:4223	MSTN	TTD	2020.06.01	NULL	4.375639269641208	AAV1-FS344	drugbank:DB17855	AAV1-FS344	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.2226788432387383	LAS-41002	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
FGF19	hgnc:3675	FGF19	CIViC	10-Apr-24	NULL	13.12691780892362	FISOGATINIB	ncit:C123826	FISOGATINIB	FALSE	FALSE	TRUE
METALLOREDUCTASE STEAP1	hgnc:11378	STEAP1	TTD	2020.06.01	NULL	9.845188356692718	RG7450	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	10.50153424713889	SUVN-502	drugbank:DB06140	SUVN-502	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	2.019525817	E-2609	iuphar.ligand:9818	ELENBECESTAT	FALSE	FALSE	FALSE
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A	hgnc:7943	NPR1	TTD	2020.06.01	NULL	16.15620653405984	PL-3994	drugbank:DB15355	PL-3994	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	Fludrocortisone	rxcui:4452	FLUDROCORTISONE	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.3251536612259921	Calcitriol	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2A	hgnc:4585	GRIN2A	TTD	2020.06.01	NULL	0.047561296	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
MONOCYTE DIFFERENTIATION ANTIGEN CD14	hgnc:1628	CD14	TTD	2020.06.01	NULL	14.32027397337122	IC14	chembl:CHEMBL2109330	IC14	FALSE	FALSE	FALSE
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	1.166837138570989	Hesperetin	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.021697385	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.2983390411119005	Piclamilast	ncit:C96718	PICLAMILAST	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.5479061346333338	TAE684	ncit:C171615	ALK INHIBITOR TAE684	FALSE	FALSE	TRUE
LIPID PEROXIDATION	hgnc:6678	LPO	TTD	2020.06.01	NULL	10.50153424713889	RAXOFELAST	ncit:C74328	RAXOFELAST	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.7395446652914718	Apadoline	ncit:C72136	APADOLINE	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.062262061	Mesoridazine	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.073954467	GNTI	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.6087845940370376	TQ-B3139	ncit:C148513	ALK/C-MET INHIBITOR TQ-B3139	FALSE	FALSE	FALSE
REACTIVE OXYGEN SPECIES	hgnc:10261	ROS1	TTD	2020.06.01	NULL	1.093909817410302	Sodium pyruvate	rxcui:1358847	SODIUM PYRUVATE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.2573905452730122	Trospium	rxcui:236778	TROSPIUM	TRUE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.8514757497680189	BIIB014	ncit:C152892	VIPADENANT	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	0.9845188356692718	Alseroxylon	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.4795221117415022	Bendamustine	rxcui:134547	BENDAMUSTINE	TRUE	FALSE	TRUE
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	8.751278539282415	Penciclovir	rxcui:59839	PENCICLOVIR	TRUE	FALSE	FALSE
LEUTINIZING-HORMONE-RELEASING HORMONE	hgnc:4419	GNRH1	TTD	2020.06.01	NULL	2.763561643983921	NAL-GLU	chembl:CHEMBL208519	CHEMBL:CHEMBL208519	FALSE	FALSE	FALSE
PROLYL ENDOPEPTIDASE FAP	hgnc:3590	FAP	TTD	2020.06.01	NULL	0.8078103267029924	Talabostat	ncit:C48264	TALABOSTAT	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.4546118721705151	Pamiparib	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
ALPHA-FETOPROTEIN	hgnc:317	AFP	TTD	2020.06.01	NULL	2.019525817	MM-093	drugbank:DB05512	MM-093	FALSE	FALSE	FALSE
SUBSTANCE-K RECEPTOR	hgnc:11527	TACR2	TTD	2020.06.01	NULL	10.50153424713889	Nepadutant	ncit:C84001	NEPADUTANT	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.090922374	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
CDC-LIKE KINASE 1	hgnc:2068	CLK1	TTD	2020.06.01	NULL	3.500511415712966	TG003	iuphar.ligand:5942	CDC2-LIKE KINASE INHIBITOR	FALSE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	1.458546423213736	Capadenoson	ncit:C87279	CAPADENOSON	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.083016081	Chlorprothixene	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.801643836	ORG-34517	drugbank:DB05423	ORG-34517	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.3923362732430473	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
DIHYDROPYRIMIDINASE RELATED PROTEIN 2	hgnc:3014	DPYSL2	TTD	2020.06.01	NULL	0.2125816649218401	Lacosamide	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.065799087	Chlordiazepoxide	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	3.281729452230906	Etelcalcetide	rxcui:1876119	ETELCALCETIDE	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.2404931506978374	Fluocinolone Acetonide	rxcui:4461	FLUOCINOLONE ACETONIDE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.047127304	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	1.211715490054488	Frovatriptan	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.1495945049449986	Diazoxide	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	6.563458904461812	Guanadrel Sulfate	rxcui:91239	GUANADREL SULFATE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.097236428	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
LUTEINIZING HORMONE RECEPTOR	hgnc:6585	LHCGR	TTD	2020.06.01	NULL	3.281729452230906	Gonadotropin, Chorionic	chembl:CHEMBL1201509	GONADOTROPIN, CHORIONIC	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.4398548375764984	Tovorafenib	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	2.917092846427472	Ribociclib Succinate	rxcui:1873978	RIBOCICLIB SUCCINATE	TRUE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	2.282942227638891	GI-6207	drugbank:DB17532	GI-6207	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.235474617310458	SL-279252	ncit:C161803	ARC FUSION PROTEIN SL-279252	FALSE	FALSE	FALSE
E3 UBIQUITIN-PROTEIN LIGASE COP1	hgnc:17440	COP1	TTD	2020.06.01	NULL	5.250767123569449	Tocainide	rxcui:42359	TOCAINIDE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	MCLA-145	ncit:C160772	ANTI-PD-L1/CD137 BISPECIFIC ANTIBODY MCLA-145	FALSE	FALSE	FALSE
TRANSFERRIN	hgnc:11740	TF	TTD	2020.06.01	NULL	6.563458904461812	CALAA-01	ncit:C78450	TRANSFERRIN RECEPTOR-TARGETED ANTI-RRM2 SIRNA CALAA-01	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Mazapertine succinate	ncit:C174754	MAZAPERTINE SUCCINATE	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	Mazapertine succinate	ncit:C174754	MAZAPERTINE SUCCINATE	FALSE	FALSE	FALSE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	0.044347695	Leucovorin Calcium	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	GB226	chembl:CHEMBL4594355	APL-501	FALSE	FALSE	FALSE
INTERLEUKIN 13 RECEPTOR ALPHA-2	hgnc:5975	IL13RA2	TTD	2020.06.01	NULL	6.563458904461812	Tralokinumab	rxcui:2589225	TRALOKINUMAB	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.6908904109959803	MM-111	drugbank:DB17983	MM-111	FALSE	TRUE	TRUE
T-CELL SURFACE GLYCOPROTEIN CD3 GAMMA	hgnc:1675	CD3G	TTD	2020.06.01	NULL	1.050153425	AFM-11	chembl:CHEMBL4297874	AFM-11	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.020084536	Bromocriptine	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	2.763561643983921	Fludrocortisone	rxcui:4452	FLUDROCORTISONE	TRUE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	2.423430980108977	Gemtuzumab ozogamicin	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	0.3017682254924971	Lisdexamfetamine	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.1154014752432846	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ALDEHYDE OXIDASE	hgnc:553	AOX1	TTD	2020.06.01	NULL	0.3621218705909965	Menadione	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.760980743	PF-07284892	ncit:C178469	SHP2 INHIBITOR PF-07284892	FALSE	FALSE	FALSE
HYDROXYPHENYLPYRUVATE DIOXYGENASE	hgnc:5147	HPD	TTD	2020.06.01	NULL	70.01022831425932	Nitisinone	rxcui:61805	NITISINONE	TRUE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	4.861821410712453	Ofatumumab	rxcui:712566	OFATUMUMAB	TRUE	TRUE	TRUE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.081407242	Pentobarbital	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-2	hgnc:3676	FGF2	TTD	2020.06.01	NULL	0.4730420832044549	Sucralfate	rxcui:10156	SUCRALFATE	TRUE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	1.29648571	Pinometostat	ncit:C103179	PINOMETOSTAT	FALSE	FALSE	TRUE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	1.458546423213736	ALX-5407	iuphar.ligand:4618	(R)-NFPS	FALSE	FALSE	FALSE
ENDOTHELIAL PLASMINOGEN ACTIVATOR INHIBITOR	hgnc:8583	SERPINE1	TTD	2020.06.01	NULL	1.544343271638073	DIAPLASININ	ncit:C72739	DIAPLASININ	FALSE	FALSE	FALSE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	8.751278539282415	LEQ-506	chembl:CHEMBL3133037	LEQ506	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR ALPHA	hgnc:9864	RARA	TTD	2020.06.01	NULL	1.250182648468916	IRX-5183	drugbank:DB05653	IRX-5183	FALSE	FALSE	FALSE
SLAM FAMILY MEMBER 7 SLAMF7	hgnc:21394	SLAMF7	TTD	2020.06.01	NULL	17.50255707856483	PVX-410	ncit:C103823	XBP1-US/XBP1-SP/CD138/CS1 MULTIPEPTIDE VACCINE PVX-410	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	AGEN2034	ncit:C136465	BALSTILIMAB	FALSE	FALSE	FALSE
ADVANCED GLYCOSYLATION END PRODUCT RECEPTOR	hgnc:320	AGER	TTD	2020.06.01	NULL	10.50153424713889	Pyridoxamine	drugbank:DB11673	PYRIDOXAMINE	FALSE	FALSE	FALSE
NCBIGENE:2464	hgnc:3861	FRA16E	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8841	iuphar.ligand:8841	4-ACRYLOYLPHENOL	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.040051618	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:55	ncit:C87208	TANDOSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:9236	iuphar.ligand:9236	COMPOUND 4G [PMID: 22220592]	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:9530	iuphar.ligand:9530	DU172	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:5608	rxcui:2199015	ISTRADEFYLLINE	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.069180068	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:412	iuphar.ligand:412	SAKURANETIN	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:456	iuphar.ligand:456	ALLOXAZINE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5608	rxcui:2199015	ISTRADEFYLLINE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:450	iuphar.ligand:450	OSIP339391	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:3281	ncit:C96199	DERENOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:11943	iuphar.ligand:11943	TRV023	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	0.9723642821424907	IUPHAR.LIGAND:8003	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:12249	iuphar.ligand:12249	COMPOUND 6LI [CHAN ET AL., 2022]	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:620	iuphar.ligand:620	PD 165929	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3840	iuphar.ligand:3840	[D-PHE6, LEU13, CPA14,&PSI;13-14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6182	iuphar.ligand:6182	[D-PHE6]BOMBESIN(6-13)PROPYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:625	iuphar.ligand:625	AC-GRP-(20-26)-METHYLESTER	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:545	iuphar.ligand:545	NIHP	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:544	iuphar.ligand:544	LK 204-545	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:10428	iuphar.ligand:10428	COMPOUND 25 [PMID: 31260299]	FALSE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:3368	iuphar.ligand:3368	CP105696	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:7246	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:932	hgnc:7317	MS4A3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:6512	iuphar.ligand:6512	(R)-EF-1520	FALSE	FALSE	FALSE
NCBIGENE:1794	hgnc:2988	DOCK2	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:8155	iuphar.ligand:8155	COMPOUND 13A [PMID: 23639540]	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.760980743	TQ-B3139	ncit:C148513	ALK/C-MET INHIBITOR TQ-B3139	FALSE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:3404	iuphar.ligand:3404	12S-HETE	FALSE	FALSE	FALSE
NCBIGENE:2730	hgnc:4312	GCLM	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:7811	iuphar.ligand:7811	COMPOUND 3 [PMID: 25408830]	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	agonist	0.050488145	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11701	iuphar.ligand:11701	UAWJ9-36-3	FALSE	FALSE	FALSE
NCBIGENE:390	hgnc:671	RND3	GuideToPharmacology	2024.1	activator	0.4375639269641209	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.8325740682192574	Futibatinib	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1695984213039228	Lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
NCBIGENE:3234	hgnc:5139	HOXD8	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12694	iuphar.ligand:12694	C7683	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:9705	iuphar.ligand:9705	AM2201	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:9799	iuphar.ligand:9799	SCH.336	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	1.628144844517658	Pemigatinib	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:9071	iuphar.ligand:9071	NABILONE	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:9607	iuphar.ligand:9607	BMS-202	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:8411	iuphar.ligand:8411	GASTRIN-14	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.006210251	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.019665794	IUPHAR.LIGAND:966	ncit:C65572	ETICLOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.003189048	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.055504938	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.008428198	IUPHAR.LIGAND:960	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.060077427	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.015019357	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:10687	iuphar.ligand:10687	GNF2133	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:10044	ncit:C147125	ABIVERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:5675	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.049841169	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:1913	iuphar.ligand:1913	MB-28767	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.097236428	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:1937	iuphar.ligand:1937	GR 63799	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:4041	iuphar.ligand:4041	MK-2894	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.3977853881492007	IUPHAR.LIGAND:4159	rxcui:2596	CLOMIPHENE	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:989	iuphar.ligand:989	ENDOTHELIN-1	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.092118721	Ipatasertib	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:990	iuphar.ligand:990	ENDOTHELIN-2	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:3951	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:13015	ncit:C76587	EDONENTAN ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:1718	hgnc:2859	DHCR24	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:9677	ncit:C171683	CIBINETIDE	FALSE	FALSE	FALSE
NCBIGENE:870	hgnc:10939	SLC1A1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:4625	iuphar.ligand:4625	L-&BETA;-BA	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1228249619548409	RO5126766	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.3454452054979901	IUPHAR.LIGAND:4179	iuphar.ligand:4179	DMCM	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.065799087	IUPHAR.LIGAND:4108	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	blocker	0.2134458180312784	IUPHAR.LIGAND:4369	iuphar.ligand:4369	[35S]TBPS	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:4238	iuphar.ligand:4238	L655708	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	1.810609352954982	IUPHAR.LIGAND:12403	iuphar.ligand:12403	PZ-II-029	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:4107	iuphar.ligand:4107	5-ME-IAA	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.042741287	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:3592	iuphar.ligand:3592	GALANIN	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:5869	iuphar.ligand:5869	WFW-ISN-NH2	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.2476776945079929	IUPHAR.LIGAND:11429	rxcui:2601723	TIRZEPATIDE	TRUE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:9060	iuphar.ligand:9060	PF-05190457	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:4166	iuphar.ligand:4166	CX546	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.108040476	Dubermatinib	ncit:C127116	DUBERMATINIB	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4209	iuphar.ligand:4209	GYKI53655	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:4131	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:1133	rxcui:475968	LIRAGLUTIDE	TRUE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.6563458904461812	IUPHAR.LIGAND:4251	iuphar.ligand:4251	LY503430	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.6563458904461812	IUPHAR.LIGAND:4166	iuphar.ligand:4166	CX546	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:4166	iuphar.ligand:4166	CX546	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:3785	iuphar.ligand:3785	[125I]GLUCAGON (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:11310	iuphar.ligand:11310	ORG 214007-0	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1521961485092594	IUPHAR.LIGAND:4086	iuphar.ligand:4086	[3H]L689560	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:4240	iuphar.ligand:4240	L701324	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.3387591692625452	IUPHAR.LIGAND:4068	iuphar.ligand:4068	(RS)-(TETRAZOL-5-YL)GLYCINE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.8468979231563628	IUPHAR.LIGAND:9052	iuphar.ligand:9052	DEXTRORPHAN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	Entospletinib	ncit:C105402	ENTOSPLETINIB	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:2366	iuphar.ligand:2366	BILOBALIDE	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	blocker	0.4234489615781814	IUPHAR.LIGAND:4282	ncit:C738	PHENCYCLIDINE	FALSE	FALSE	FALSE
NCBIGENE:1273	hgnc:4093	GAD2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:5267	iuphar.ligand:5267	S-ALLYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	modulator	0.8078103267029924	IUPHAR.LIGAND:4164	iuphar.ligand:4164	CU2+	FALSE	FALSE	FALSE
NCBIGENE:2959	hgnc:4648	GTF2B	GuideToPharmacology	2024.1	antibody	6.563458904461812	IUPHAR.LIGAND:8406	iuphar.ligand:8406	CODRITUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.046840028	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:311	hgnc:535	ANXA11	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:5783	iuphar.ligand:5783	3,5-DIHYDROXYBENZOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:1248	iuphar.ligand:1248	DIMAPRIT	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:7346	iuphar.ligand:7346	MK-0249	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1239	iuphar.ligand:1239	N-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:8982	iuphar.ligand:8982	INCB-38579	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:1238	iuphar.ligand:1238	(S)-&ALPHA;-METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:1266	iuphar.ligand:1266	IODOPHENPROPIT	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3029	iuphar.ligand:3029	COMPOUND 29 [PMID: 1527791]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5724	iuphar.ligand:5724	COMPOUND 3 [PMID: 21310611]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5721	iuphar.ligand:5721	(S)-N-OLEOYLTYROSINOL	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5722	iuphar.ligand:5722	AS1535907	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5756	iuphar.ligand:5756	1-OLEOYL GLYCEROL	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5519	iuphar.ligand:5519	ASN04450772	FALSE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:11685	iuphar.ligand:11685	ZELATRIAZIN (TAK-041)	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:5558	iuphar.ligand:5558	JWH015	FALSE	FALSE	FALSE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9741	iuphar.ligand:9741	CID2745687	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:11213	iuphar.ligand:11213	DL-175	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5850	iuphar.ligand:5850	3-HYDROXYLAURIC ACID	FALSE	FALSE	FALSE
NCBIGENE:150	hgnc:281	ADRA2A	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7043	iuphar.ligand:7043	AR305352	FALSE	FALSE	FALSE
NCBIGENE:2829	hgnc:1625	XCR1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:9019	iuphar.ligand:9019	NAVOXIMOD	FALSE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	0.4730420832044549	IUPHAR.LIGAND:8759	iuphar.ligand:8759	L-NNA	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.5770073762164231	IUPHAR.LIGAND:1674	iuphar.ligand:1674	CTOP	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.082429625	IUPHAR.LIGAND:1606	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
NCBIGENE:629	hgnc:1037	CFB	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:12997	iuphar.ligand:12997	COMPOUND 111 [PMID: 37918435]	FALSE	FALSE	FALSE
NCBIGENE:463	hgnc:777	ZFHX3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:3963	ncit:C75979	HEXAMETHONIUM	FALSE	FALSE	FALSE
NCBIGENE:470	ncbigene:470	ATHS	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:463	hgnc:777	ZFHX3	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:9056	iuphar.ligand:9056	CP-601927	FALSE	FALSE	FALSE
NCBIGENE:465	ncbigene:465	ATD	GuideToPharmacology	2024.1	modulator	3.750547945	IUPHAR.LIGAND:3993	iuphar.ligand:3993	NS9283	FALSE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:3972	iuphar.ligand:3972	[125I]&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3972	iuphar.ligand:3972	[125I]&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:3972	iuphar.ligand:3972	[125I]&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:2086	ncit:C80866	ELEDOISIN	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:3805	iuphar.ligand:3805	[125I]SP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:2122	iuphar.ligand:2122	YM49598	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3880	iuphar.ligand:3880	GR100679	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:3471	iuphar.ligand:3471	[125I]L703,606	FALSE	FALSE	FALSE
NCBIGENE:303	hgnc:538	ANXA2P1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:1495	iuphar.ligand:1495	NEUROPEPTIDE W-23	FALSE	FALSE	FALSE
NCBIGENE:2629	hgnc:4177	GBA1	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:6816	rxcui:341248	EZETIMIBE	TRUE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:1568	iuphar.ligand:1568	JMV2004	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1697	iuphar.ligand:1697	OREXIN-A	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:3778	iuphar.ligand:3778	[125I]D(CH2)5[TYR(ME)2,THR4,ORN8,TYR-NH29]OVT	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:11447	iuphar.ligand:11447	COMPOUND 1 [PMID: 33547286]	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.1060761035064535	IUPHAR.LIGAND:2200	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:11449	iuphar.ligand:11449	[3H]T-516	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9121	iuphar.ligand:9121	LSN2424100	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2890	rxcui:1547099	SUVOREXANT	TRUE	FALSE	FALSE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9454	iuphar.ligand:9454	PQA-18	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:9540	ncit:C166945	GEFAPIXANT	FALSE	FALSE	FALSE
NCBIGENE:479	hgnc:13816	ATP12A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9546	iuphar.ligand:9546	NF778	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4225	iuphar.ligand:4225	IP5I	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:12566	iuphar.ligand:12566	PSB-12054	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	modulator	0.145450613	IUPHAR.LIGAND:2523	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	modulator	1.093909817410302	IUPHAR.LIGAND:10504	iuphar.ligand:10504	GSK1482160	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:10504	iuphar.ligand:10504	GSK1482160	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7538	iuphar.ligand:7538	JNJ-47965567	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1778	iuphar.ligand:1778	MRS2603	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3398	iuphar.ligand:3398	2-THIOUTP	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1831	drugbank:DB02261	PLATELET ACTIVATING FACTOR	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1152	iuphar.ligand:1152	VIP	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1834	iuphar.ligand:1834	ENANTIO PAF C-16	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:3914	iuphar.ligand:3914	TRANS-CINNAMOYL-LIGRLO [N-[3H]PROPIONYL]-NH2	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:3754	iuphar.ligand:3754	(DES 1-8) A-CHAIN INSL3 ANALOGUE	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:8350	iuphar.ligand:8350	INSL5 AMIDE (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:12777	iuphar.ligand:12777	EST73502	FALSE	FALSE	FALSE
NCBIGENE:959	hgnc:11935	CD40LG	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:63	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1041	hgnc:1802	CDSN	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:4285	drugbank:DB07810	PHLORETIN	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9764	iuphar.ligand:9764	LANRAPLENIB	FALSE	FALSE	FALSE
NCBIGENE:1416	hgnc:2399	CRYBB2P1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8764	iuphar.ligand:8764	COMPOUND 28XVII [PMID: 8809154]	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2005	iuphar.ligand:2005	CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:2017	iuphar.ligand:2017	NC 4-28B	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5640	iuphar.ligand:5640	GA-KE88	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2057	iuphar.ligand:2057	[111IN,90Y]DOTA-NOC	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:2067	iuphar.ligand:2067	PRL-2970	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:2028	iuphar.ligand:2028	[D-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:12011	iuphar.ligand:12011	SNX281	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.024932417	CUDC-907	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:12611	ncit:C174060	BASROPARIB	FALSE	FALSE	FALSE
NCBIGENE:2231	hgnc:3640	FDX1P1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9524	iuphar.ligand:9524	BAY-299	FALSE	FALSE	FALSE
NCBIGENE:2642	hgnc:4192	GCGR	GuideToPharmacology	2024.1	inhibitor	0.048618214	IUPHAR.LIGAND:6799	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:5018	ncit:C1470	LOXORIBINE	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1970	iuphar.ligand:1970	CARBOCYCLIC THROMBOXANE A2	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1898	iuphar.ligand:1898	S-5751	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1938	iuphar.ligand:1938	I-BOP	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1913	iuphar.ligand:1913	MB-28767	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.092606122	Tazemetostat	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11856	iuphar.ligand:11856	SG-094	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4158	iuphar.ligand:4158	CHLOROBENZYLIDENE MALONONITRILE	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:10290	iuphar.ligand:10290	AC1903	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.5147810905460244	IUPHAR.LIGAND:4232	iuphar.ligand:4232	KB-R7943	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.072725306	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.5147810905460244	IUPHAR.LIGAND:10283	iuphar.ligand:10283	SAR7334	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	2.763561643983921	IUPHAR.LIGAND:4200	iuphar.ligand:4200	GEA 3162	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.054020238	Ipatasertib	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:10295	iuphar.ligand:10295	LARIXYL ACETATE	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.085796848	IUPHAR.LIGAND:2694	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	1.875273972703375	IUPHAR.LIGAND:10039	iuphar.ligand:10039	COMPOUND 6 [PMID: 29579323]	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10039	iuphar.ligand:10039	COMPOUND 6 [PMID: 29579323]	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2438	iuphar.ligand:2438	BTP2	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:4145	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	0.1151484018326633	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.1973972602845657	E6201	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:6402	iuphar.ligand:6402	SN-2	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	activator	0.1093909817410302	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:9145	iuphar.ligand:9145	COMPOUND 74A [PMID: 27077528]	FALSE	FALSE	FALSE
NCBIGENE:511	hgnc:3145	TRPV5	GuideToPharmacology	2024.1	inhibitor	0.326134604	IUPHAR.LIGAND:2427	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12558	iuphar.ligand:12558	GSK-BZ DERIVATIVE 2B	FALSE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.028529025	Berzosertib	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:11613	ncit:C180657	ROPSACITINIB	FALSE	FALSE	FALSE
NCBIGENE:1841	hgnc:3061	DTYMK	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:12249	iuphar.ligand:12249	COMPOUND 6LI [CHAN ET AL., 2022]	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:8872	iuphar.ligand:8872	COMPOUND 1A [PMID: 18573659]	FALSE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:4834	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.014617949	IUPHAR.LIGAND:2187	iuphar.ligand:2187	D[CHA4]AVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.002248915	IUPHAR.LIGAND:2174	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:2219	iuphar.ligand:2219	D(CH2)5[TYR(ME)2,THR4,PHE(3I,4N3)-NH29]OVT	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2170	iuphar.ligand:2170	DAVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:3537	iuphar.ligand:3537	VNA932	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.033658764	IUPHAR.LIGAND:2174	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2217	iuphar.ligand:2217	D(CH2)5[TYR(ET)2,VAL4,DES-GLY9]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2190	iuphar.ligand:2190	D[LEU4]AVP	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:7729	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:2200	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.004504583	Valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
NCBIGENE:2831	hgnc:4522	NPBWR1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8231	iuphar.ligand:8231	OICR-9429	FALSE	FALSE	TRUE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:1529	iuphar.ligand:1529	GR231118	FALSE	FALSE	FALSE
NCBIGENE:2289	hgnc:3721	FKBP5	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:12845	iuphar.ligand:12845	KC-130	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	CIViC	10-Apr-24	NULL	0.1151484018326633	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.1715936968486748	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	CIViC	10-Apr-24	NULL	0.049723174	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.002821552	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	0.3642372228836055	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PTPN12	hgnc:9645	PTPN12	CIViC	10-Apr-24	NULL	0.6731752722524936	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.017549355	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.1151484018326633	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.012695278	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.004120188	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.010884675	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.1043371509899543	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
CSF1	hgnc:2432	CSF1	CIViC	10-Apr-24	NULL	0.5357925636295356	PEXIDARTINIB	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.5233322714521047	ROGARATINIB	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	CIViC	10-Apr-24	NULL	0.01893533	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	4.109296009750004	Ensartinib	ncit:C102754	ENSARTINIB	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.3977853881492007	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.091796628	Vinorelbine	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	1.060761035064535	VE-821	iuphar.ligand:8042	VE-821	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.026640117	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.024802868	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	0.6563458904461813	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	IMIPRAMINE PAMOATE	rxcui:91118	IMIPRAMINE PAMOATE	TRUE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1154014752432846	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.2419708351875322	ETHOPROPAZINE HYDROCHLORIDE	rxcui:6541	ETHOPROPAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	MAPROTILINE HYDROCHLORIDE	rxcui:203126	MAPROTILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.020470827	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.024275391	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	NCI	14-Sep-17	NULL	0.4412409347537353	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1215455352678113	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	PharmGKB	4/5/24	NULL	0.9376369863516875	lisinopril	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1	hgnc:2432	CSF1	TTD	2020.06.01	NULL	3.750547945	RG7155	ncit:C125548	EMACTUZUMAB	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.088945801	OPC-34712	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	modulator	0.3365876361262467	IUPHAR.LIGAND:12050	iuphar.ligand:12050	SAGE-718	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6102	iuphar.ligand:6102	M1151	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6209	iuphar.ligand:6209	COMPOUND 24 [PMID: 20346665]	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.729273212	Ceralasertib	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.062808219	IUPHAR.LIGAND:7519	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1512	iuphar.ligand:1512	PANCREATIC POLYPEPTIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.002253065	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	TALIPEXOLE HYDROCHLORIDE	chembl:CHEMBL1504869	TALIPEXOLE HYDROCHLORIDE	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.002546567	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.1305078821102597	NALOXONE HYDROCHLORIDE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	SAPPANONE A TRIMETHYL ETHER	chembl:CHEMBL1606022	SAPPANONE A TRIMETHYL ETHER	FALSE	FALSE	FALSE
KCNA4	hgnc:6222	KCNA4	ChEMBL	33	blocker	0.1829535583125243	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	PharmGKB	4/5/24	NULL	0.03140411	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P22455	hgnc:3691	FGFR4	TEND	1-Aug-11	NULL	0.2792961235941196	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.8899605294185507	MK-5108	drugbank:DB12556	MK-5108	FALSE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR	hgnc:2436	CSF2RB	TTD	2020.06.01	NULL	2.917092846427472	SL-401	rxcui:2109054	TAGRAXOFUSP-ERZS	TRUE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	2.282942227638891	Anti-CEA CAR-T cells	ncit:C188356	ANTI-CEA CAR T CELLS	FALSE	FALSE	FALSE
C6ORF15	hgnc:13927	C6orf15	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8329	iuphar.ligand:8329	A(9-26)INSL3	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	DoCM	10-Apr-24	NULL	0.1088116604009326	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.092606122	IUPHAR.LIGAND:2181	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.093763699	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.054695491	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
TSG101	hgnc:15971	TSG101	DTC	9/2/20	NULL	0.5048814541893701	FLUORANTHEN-3-YLAMINE	chembl:CHEMBL103583	CHEMBL:CHEMBL103583	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.025421288	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.015312823	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	MADOLIN T	chembl:CHEMBL2333550	MADOLIN T	FALSE	FALSE	FALSE
UNIPROT:P04049	hgnc:9829	RAF1	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	XL281	drugbank:DB05190	XL281	FALSE	FALSE	TRUE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	DAPIPRAZOLE	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1037701012563132	REMOXIPRIDE	rxcui:35350	REMOXIPRIDE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.09969811	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6138	iuphar.ligand:6138	GALANIN(3-30) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:9457	iuphar.ligand:9457	AC-98170	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:10466	iuphar.ligand:10466	LINPERLISIB	FALSE	FALSE	FALSE
NCBIGENE:2214	hgnc:3619	FCGR3A	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:10597	iuphar.ligand:10597	BAY-985	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.06109095	Tivozanib	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2208	iuphar.ligand:2208	[PHAA1,D-TYR(ET)2,LYS6,DES-GLY9]AVP	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.004668386	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.4817217544559128	METHYLSAMIDORPHAN	ncit:C175135	METHYLSAMIDORPHAN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	RS-17053	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	(S)-FELODIPINE	chembl:CHEMBL428768	(S)-FELODIPINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:4606	iuphar.ligand:4605	[3H]WIN35428	FALSE	FALSE	FALSE
UNIPROT:P01589	hgnc:6008	IL2RA	TdgClinicalTrial	Jan-14	NULL	0.3431873936973496	INTERLEUKIN 2	chembl:CHEMBL1201438	ALDESLEUKIN	FALSE	FALSE	FALSE
TGFA	hgnc:11765	TGFA	PharmGKB	4/5/24	NULL	0.364636606	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.561579372	telmisartan	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.027433475	IUPHAR.LIGAND:7282	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	blocker	4.773424657790408	IUPHAR.LIGAND:4218	iuphar.ligand:4218	IBERIOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:10549	iuphar.ligand:10549	COMPOUND 18E [PMID: 31670517]	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.008382451	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.018206543	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.078682824	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	1.750255707856483	BMS-820132	iuphar.ligand:11932	BMS-820132	FALSE	FALSE	FALSE
NCBIGENE:1016	hgnc:1757	CDH18	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:4628	rxcui:10454	THIAMINE	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:11239	iuphar.ligand:11239	NSC212069	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	CGI	2/1/22	NULL	0.1944728564284981	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1840222122746302	DESVENLAFAXINE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	2.386712328895204	Asasantin	wikidata:Q4803642	ACETYLSALICYLIC ACID/DIPYRIDAMOLE	FALSE	FALSE	FALSE
NCBIGENE:1723	hgnc:2867	DHODH	GuideToPharmacology	2024.1	agonist	0.086361301	IUPHAR.LIGAND:7462	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
NCBIGENE:1823	hgnc:3035	DSC1	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:8925	iuphar.ligand:8925	FIBATUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.002357564	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.2592971419046642	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.4375639269641208	amodiaquine	rxcui:720	AMODIAQUINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.036770078	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	ALBENDAZOLE	rxcui:430	ALBENDAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	GNF-PF-840	chembl:CHEMBL601605	CHEMBL:CHEMBL601605	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	AMINOPURVALANOL	iuphar.ligand:5927	AMINOPURVALANOL A	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:11204	iuphar.ligand:11204	AZD8154	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:2650	iuphar.ligand:2650	BMS753	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10425	iuphar.ligand:10425	ROCK INHIBITOR 3	FALSE	FALSE	FALSE
CCNE1	hgnc:1589	CCNE1	CIViC	10-Apr-24	NULL	1.312691780892362	FADRACICLIB	ncit:C123902	FADRACICLIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	AZD8835	iuphar.ligand:8915	AZD8835	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.1372749574789398	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:5357	iuphar.ligand:5357	GALANIN(2-11)	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.175415383	APC-100	chembl:CHEMBL37676	APC-100	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.2778183663264258	ZANDELISIB	ncit:C123925	ZANDELISIB	FALSE	FALSE	FALSE
UNIPROT:P51681	hgnc:1606	CCR5	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	TBR-652	ncit:C169838	CENICRIVIROC MESYLATE	FALSE	FALSE	FALSE
UNIPROT:P39086	hgnc:4579	GRIK1	TEND	1-Aug-11	NULL	1.432027397337122	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:Q9P0X4	hgnc:1396	CACNA1I	TEND	1-Aug-11	NULL	0.055563673	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.9546849315580818	Liraglutide	rxcui:475968	LIRAGLUTIDE	TRUE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.3739862623624964	Cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
NCBIGENE:2721	ncbigene:2721	GLC#	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8571	iuphar.ligand:8571	BAZ2-ICR	FALSE	FALSE	FALSE
NCBIGENE:726	hgnc:1482	CAPN5	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2074	hgnc:3438	ERCC6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11595	iuphar.ligand:11595	COMPOUND 18 [PMID: 34212719]	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.3113103037689397	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.065634589	Mepivacaine	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2904	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:9211	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:9543	iuphar.ligand:9543	BX-430	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:9636	iuphar.ligand:9636	INAVOLISIB	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.1151484018326633	DARIFENACIN HYDROBROMIDE	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.1666910197958555	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.011710007	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.065226921	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.066423367	TZT-1027	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	PharmGKB	4/5/24	NULL	0.084214389	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:8145	iuphar.ligand:8145	COMPOUND 38 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	activator	0.8751278539282418	IUPHAR.LIGAND:2619	iuphar.ligand:2619	BATRACHOTOXIN	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.1544343271638073	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
PTK2B	hgnc:9612	PTK2B	ChEMBL	33	inhibitor	0.2853677784548614	CONTELTINIB	ncit:C169863	CONTELTINIB	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.047647615	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	NSC-8186	chembl:CHEMBL122355	CHEMBL:CHEMBL122355	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:1857	ncit:C65987	ISRAPAFANT	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.175610941	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	3.281729452230906	Iclaprim	ncit:C65877	ICLAPRIM	FALSE	FALSE	FALSE
NCBIGENE:128	hgnc:253	ADH5	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:11337	iuphar.ligand:11337	ONC212	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.1097339001790898	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.1912847768149162	goserelin	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
IL6R	hgnc:6019	IL6R	ChEMBL	33	inhibitor	4.039051633514961	TOCILIZUMAB	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	DNDI1417300	chembl:CHEMBL1401091	CHEMBL:CHEMBL1401091	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.6674703970639131	DESERPIDINE	rxcui:62174	DESERPIDINE	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.042174836	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.085032666	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1035654265003836	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	DIHYDROERGOCRISTINE MESYLATE	ncit:C75939	DIHYDROERGOCRISTINE MESYLATE	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.6775183385250904	Decernotinib	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:9361	iuphar.ligand:9361	WYE-354	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.1305078821102597	NALOXONE HYDROCHLORIDE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.041872146	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	1.093909817410302	HMPL-306	ncit:C175602	IDH1/IDH2 DUAL INHIBITOR HMPL-306	FALSE	FALSE	FALSE
PTCH1	hgnc:9585	PTCH1	MyCancerGenome	20-Jun-17	other/unknown	19.69037671338543	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.1339481409073839	Vindesine	rxcui:11204	VINDESINE	FALSE	FALSE	TRUE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1253	iuphar.ligand:1253	IODOPROXYFAN	FALSE	FALSE	FALSE
HTR1F	hgnc:5292	HTR1F	ChEMBL	33	agonist	0.280789686	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O14965	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.1435420208739598	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	3.842024724563012	MDX-1342	chembl:CHEMBL2109337	MDX-1342	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.1056492378987816	MOXONIDINE	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.2983390411119005	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.047049885	Lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.099446347	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.070574827	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	8.751278539282415	HQK-1004	ncit:C2570	ARGININE BUTYRATE	FALSE	FALSE	FALSE
THIOREDOXIN	hgnc:12435	TXN	TTD	2020.06.01	NULL	39.38075342677087	PX-12	drugbank:DB05448	PX-12	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.02887152	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1406	iuphar.ligand:1406	(R,S)-4-PPG	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	DTC	9/2/20	NULL	2.143170254518142	MANGIFERIN HEPTASULFATE	chembl:CHEMBL2158201	MANGIFERIN HEPTASULFATE	FALSE	FALSE	FALSE
UNIPROT:P25103	hgnc:11526	TACR1	TEND	1-Aug-11	NULL	0.2027323213733378	VAPREOTIDE	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.06638138	IUPHAR.LIGAND:1606	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	blocker	0.1902451856365742	IUPHAR.LIGAND:4282	ncit:C738	PHENCYCLIDINE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	9-PHENYLIMIDAZO[1,2-H][1,7]NAPHTHYRIDINE	chembl:CHEMBL455004	CHEMBL:CHEMBL455004	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002059205	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.017243899	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2138	hgnc:3519	EYA1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.062212881	IUPHAR.LIGAND:8196	iuphar.ligand:8196	COMPOUND 17D [PMID: 23099093]	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.046549354	DIZOCILPINE	ncit:C65450	DIZOCILPINE	FALSE	FALSE	FALSE
MC1R	hgnc:6929	MC1R	ChEMBL	33	agonist	3.750547945	MODIMELANOTIDE	ncit:C175147	MODIMELANOTIDE	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	MK-8353	iuphar.ligand:9974	MK-8353	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	FF-10101	chembl:CHEMBL4650283	FF-10101	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	0.4268916360625568	BENZYL ISOTHIOCYANATE	drugbank:DB16860	BENZYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	NCI	14-Sep-17	NULL	0.3684748858645228	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.060772768	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:653	iuphar.ligand:653	B-9430	FALSE	FALSE	FALSE
NDUFB10	hgnc:7696	NDUFB10	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1190650141398968	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.066297565	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	GSK2334470	iuphar.ligand:8008	GSK2334470	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.013546871	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.056826484	IUPHAR.LIGAND:4108	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2187	iuphar.ligand:2187	D[CHA4]AVP	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:11304	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
NCBIGENE:1889	hgnc:3146	ECE1	GuideToPharmacology	2024.1	antibody	0.6177373086552295	IUPHAR.LIGAND:11117	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.00854061	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.1440539677248134	Lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.009053047	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.2660861718025059	AZD8186	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.201178817	PENICILLIOL B	chembl:CHEMBL513800	PENICILLIOL B	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.1750255707856483	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.1435420208739598	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	0.2243917574174978	IUPHAR.LIGAND:2597	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
NCBIGENE:2199	hgnc:3601	FBLN2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9581	iuphar.ligand:9581	ARN-3236	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.019739726	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.5000730593875667	Revamilast	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.9376369863516876	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:10727	iuphar.ligand:10727	4F-MT-45	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.5303805175322677	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.138178082	Ulixertinib	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005130207	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.054695491	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.1440539677248134	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	1.080404757936101	RXDX-105	ncit:C107245	AGERAFENIB	FALSE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	TALC	12-May-16	inhibitor	1.086365611772989	PX-478	drugbank:DB06082	PX-478	FALSE	FALSE	TRUE
UNIPROT:P54284	hgnc:1403	CACNB3	TEND	1-Aug-11	NULL	0.1795134059339982	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.074084898	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:776	iuphar.ligand:776	CCL26	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:913	iuphar.ligand:913	CORTICOTROPIN-RELEASING FACTOR	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.375054795	BINIMETINIB	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MACROPHAGE COLONY-STIMULATING FACTOR 1	hgnc:2432	CSF1	TTD	2020.06.01	NULL	3.750547945	Emactuzumab	ncit:C125548	EMACTUZUMAB	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.2263261691193728	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1591141552596803	Trazodone	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:399	iuphar.ligand:399	MRS1093	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:1739	iuphar.ligand:1739	REACTIVE BLUE-2	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.066297565	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.022439176	nitrendipine	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	inhibitor	0.027347745	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000756409	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.09972967	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.6886251965336985	NORGESTIMATE	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.5556367326528517	AZD-6765	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.2011788169949981	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
UNIPROT:P21796	hgnc:12669	VDAC1	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	OLESOXIME	ncit:C174604	OLESOXIME	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	modulator	1.810609352954982	IUPHAR.LIGAND:12213	iuphar.ligand:12213	D5261	FALSE	FALSE	FALSE
UNIPROT:P51172	hgnc:10601	SCNN1D	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.2368767123414789	Anlotinib	ncit:C138997	ANLOTINIB	FALSE	FALSE	FALSE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.1988926940746004	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	PIFEXOLE	ncit:C76774	PIFEXOLE	FALSE	FALSE	FALSE
FES	hgnc:3657	FES	DTC	9/2/20	NULL	0.1704794520639432	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.044161204	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.041396776	Seliciclib	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
UNIPROT:P11166	hgnc:11005	SLC2A1	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.010209541	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	NSC-659162	chembl:CHEMBL471005	CHEMBL:CHEMBL471005	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	DTC	9/2/20	NULL	0.2983390411119005	PYRIMETHAMINE	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9903	iuphar.ligand:9903	SAMURACICLIB	FALSE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:10597	iuphar.ligand:10597	BAY-985	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.04636439	Selinexor	rxcui:2178390	SELINEXOR	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	SJ000067611	chembl:CHEMBL602126	CHEMBL:CHEMBL602126	FALSE	FALSE	FALSE
CDC-LIKE KINASE 2	hgnc:2069	CLK2	TTD	2020.06.01	NULL	0.729273212	TG003	iuphar.ligand:5942	CDC2-LIKE KINASE INHIBITOR	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	KINETIN RIBOSIDE	chembl:CHEMBL411066	KINETIN RIBOSIDE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.007792334	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.3281729452230906	TRICHOSTATIN A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
UNIPROT:Q01718	hgnc:6930	MC2R	TEND	1-Aug-11	NULL	13.12691780892362	COSYNTROPIN	rxcui:2890	COSYNTROPIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	1-BENZYLMALEIMIDE	chembl:CHEMBL388979	CHEMBL:CHEMBL388979	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	0.088770366	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	1.721562991334245	Telapristone	ncit:C104057	TELAPRISTONE	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.2333674277141978	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
ABCC5	hgnc:56	ABCC5	DTC	9/2/20	NULL	0.7501095890813498	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
NCBIGENE:1276	hgnc:8109	ODC1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:5139	iuphar.ligand:5139	APA	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	ChEMBL	33	inhibitor	0.5000730593875666	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
KCNA10	hgnc:6219	KCNA10	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
STK11	hgnc:11389	STK11	DoCM	10-Apr-24	NULL	0.4138535663897103	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.015791781	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	ChEMBL	33	inhibitor	0.1141471113819445	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:10030	iuphar.ligand:10030	VCE-004.3	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	CRIDANIMOD	ncit:C77948	CRIDANIMOD	FALSE	FALSE	FALSE
GD	hgnc:8573	PAEP	ChEMBL	33	inhibitor	2.187819634820604	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.052090944	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	LERSIVIRINE	ncit:C83872	LERSIVIRINE	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	FDA	10-Apr-24	NULL	5.469549087051511	Enasidenib	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	FENPYROXYMATE	chembl:CHEMBL365100	FENPYROXYMATE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.061628722	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.029918901	nitrendipine	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	PharmGKB	4/5/24	NULL	0.5933070196123671	perindopril	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
NCBIGENE:1443	hgnc:2441	CSH2	GuideToPharmacology	2024.1	inhibitor	3.750547945406749	IUPHAR.LIGAND:5150	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.051478109	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.010750956	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.1136529680426287	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
AXL	hgnc:905	AXL	ChEMBL	33	inhibitor	0.546954909	GILTERITINIB FUMARATE	rxcui:2105823	GILTERITINIB FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	JCAR014	drugbank:DB17232	JCAR014	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	ChEMBL	33	positive modulator	1.381780822	NONACOG ALFA	rxcui:1300488	NONACOG ALFA	TRUE	FALSE	FALSE
ULK3	hgnc:19703	ULK3	DTC	9/2/20	inhibitor	0.6563458904461813	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.009882867	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.043976274	6-HYDROXYMELATONIN	iuphar.ligand:1347	6-HYDROXYMELATONIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	PHENAZINE	chembl:CHEMBL119870	PHENAZINE	FALSE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.4375639269641208	danazol	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.2461297089173179	meperidine	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CLEC16A	hgnc:29013	CLEC16A	PharmGKB	4/5/24	NULL	15.00219178162699	glatiramer acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	GF-109203	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TEND	1-Aug-11	NULL	0.31919557	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA 3	hgnc:11769	TGFB3	TTD	2020.06.01	NULL	13.12691780892362	Avotermin	rxcui:1427086	AVOTERMIN	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	1.141471113819445	LGH447	ncit:C106259	PIM KINASE INHIBITOR LGH447	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002258977	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:5776	iuphar.ligand:5776	YSFKPMPLAR	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.09814518	ETONOGESTREL	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	ETHOPROPAZINE HYDROCHLORIDE	rxcui:6541	ETHOPROPAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IGF2BP2	hgnc:28867	IGF2BP2	PharmGKB	4/5/24	NULL	0.6403374540938354	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.6000876712650799	MAPK INHIBITORS	ncit:C2149	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:967	hgnc:1692	CD63	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8814	iuphar.ligand:8814	COMPOUND 6B [PMID: 22749870]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12983	iuphar.ligand:12983	TQB3804	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:3825	iuphar.ligand:3825	[3H]LYS-[DES-ARG9]BK	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.049723174	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
KIDNEY-TYPE ARGINASE	hgnc:664	ARG2	TTD	2020.06.01	NULL	0.5000730593875667	Difluoromethylornithine	ncit:C226	EFLORNITHINE	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.400821918	Meprednisone	rxcui:29523	MEPREDNISONE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	1.060761035064535	IUPHAR.LIGAND:1190	rxcui:68147	CETRORELIX	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.1389091831632129	MM121	chembl:CHEMBL3545071	SERIBANTUMAB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.375054795	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:1879	hgnc:3126	EBF1	GuideToPharmacology	2024.1	NULL	1.750255707856483	IUPHAR.LIGAND:5065	iuphar.ligand:5065	TRAIL	FALSE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	0.033148782	IUPHAR.LIGAND:2801	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:4297	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TdgClinicalTrial	Jan-14	NULL	11.66837138570988	POLYTHIAZIDE	rxcui:8565	POLYTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:10104	iuphar.ligand:10104	(S)-DIMETINDENE	FALSE	FALSE	FALSE
UNIPROT:Q14416	hgnc:4594	GRM2	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	LY2140023	drugbank:DB05096	LY2140023	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	FLAVOXATE	rxcui:4440	FLAVOXATE	TRUE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:10149	iuphar.ligand:10149	SLC-0111	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.1190650141398968	IUPHAR.LIGAND:10357	iuphar.ligand:10357	CDK INHIBITOR 4.35	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	agonist	0.4167275494896389	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1282238613814273	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	CGI	2/1/22	NULL	0.458240639	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.038608582	IUPHAR.LIGAND:7227	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:1366	hgnc:2049	CLDN7	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8790	iuphar.ligand:8790	COMPOUND 5 [PMID: 21838328]	FALSE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	NCI	14-Sep-17	NULL	0.4412409347537353	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BRUCINE	rxcui:2181419	BRUCINE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.3302369260106572	N-(3-OXODODECANOYL)HOMOSERINELACTONE	chembl:CHEMBL8483	CHEMBL:CHEMBL8483	FALSE	FALSE	FALSE
UNIPROT:P30273	hgnc:3611	FCER1G	TEND	1-Aug-11	NULL	17.50255707856483	BENZYLPENICILLOYL POLYLYSINE	rxcui:19079	BENZYLPENICILLOYL POLYLYSINE	TRUE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.044498026	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.3684748858645228	METIXENE	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.3281729452230906	DELAVIRDINE	rxcui:83816	DELAVIRDINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PREGNENOLONE CARBONITRILE	iuphar.ligand:2762	PREGNENOLONE-16&ALPHA;-CARBONITRILE	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	NCI	14-Sep-17	NULL	0.3079628811477683	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.075010959	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	DIACEREIN	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	A-1331852	iuphar.ligand:11102	A-1331852	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.043611023	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.2287915957982331	ZIDOVUDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:649	iuphar.ligand:649	BRADYKININ	FALSE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TdgClinicalTrial	Jan-14	NULL	0.7001022831425934	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TdgClinicalTrial	Jan-14	NULL	18.37768493249307	MENOTROPINS	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.026319635	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
SOLUBLE GUANYLYL CYCLASE	hgnc:4689	GUCY2D	TTD	2020.06.01	NULL	17.50255707856483	BAY 1021189	chembl:CHEMBL4066936	VERICIGUAT	FALSE	FALSE	FALSE
NCBIGENE:1620	hgnc:2687	BRINP1	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:8654	iuphar.ligand:8654	M826	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.085239726	IUPHAR.LIGAND:329	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.222962511	ELOCALCITOL	drugbank:DB06194	ELOCALCITOL	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.1110098757625676	IUPHAR.LIGAND:7076	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
CD14	hgnc:1628	CD14	PharmGKB	4/5/24	NULL	0.502465753	fluticasone propionate	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
WT1	hgnc:12796	WT1	ChEMBL	33	vaccine	4.039051633514961	GALINPEPIMUT-S	ncit:C161778	GALINPEPIMUT-S	FALSE	FALSE	FALSE
MTRR	hgnc:7473	MTRR	PharmGKB	4/5/24	NULL	0.5676504998453459	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.008310806	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.07631929	DIOSMIN	rxcui:3489	DIOSMIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	SKF-38393	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.1154014752432846	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.1136529680426287	BI847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.064347636	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	0.1944728564284981	IUPHAR.LIGAND:2661	iuphar.ligand:2661	N-OLEOYLETHANOLAMIDE	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.05853698	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.021997349	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
GLRB	hgnc:4329	GLRB	ChEMBL	33	positive modulator	0.1693795846312726	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
NCBIGENE:1990	hgnc:3308	CELA1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:8161	iuphar.ligand:8161	COMPOUND 17 [PMID: 23642479]	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	ChEMBL	33	inhibitor	0.013113804	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.061737415	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.09972967	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	0.6482428547616605	IUPHAR.LIGAND:8003	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.053145416	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.042793538	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.031631127	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6095	iuphar.ligand:6095	GALANIN(D-TRP2) (PIG)	FALSE	FALSE	FALSE
LOW-AFFINITY NERVE GROWTH FACTOR RECEPTOR	hgnc:7809	NGFR	TTD	2020.06.01	NULL	8.751278539282415	Fulranumab	ncit:C84838	FULRANUMAB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.079376676	TYRPHOSTIN AG-1478	iuphar.ligand:4862	AG1478	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.1215455352678113	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.020117882	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.03233231	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.029074015	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NCOA7	hgnc:21081	NCOA7	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.019447286	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1344626664166312	BSO	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.5000730593875666	GNF-PF-2671	chembl:CHEMBL578878	CHEMBL:CHEMBL578878	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.729273212	L-GLUTAMINE	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	AZQ	ncit:C1363	DIAZIQUONE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	0.4734548598913698	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
PPP1R18	hgnc:29413	PPP1R18	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.091159151	lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
PRB2	hgnc:9338	PRB2	PharmGKB	4/5/24	NULL	0.1613138901250215	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CD3D	hgnc:1673	CD3D	ChEMBL	33	modulator	0.4102161815288632	IMC-GP100	chembl:CHEMBL2109434	IMC-GP100	FALSE	FALSE	FALSE
FUT2	hgnc:4013	FUT2	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.150021918	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.035358701	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
TNNT2	hgnc:11949	TNNT2	DTC	9/2/20	NULL	0.5707355569097228	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	KARANJIN	chembl:CHEMBL208484	KARANJIN	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.065389379	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.050879526	Ethchlorvynol	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.030868707	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
PSMD7	hgnc:9565	PSMD7	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.005905046	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.4526523382387456	AMRUBICIN	ncit:C80089	AMRUBICIN	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.018540844	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	1.969037671338543	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:223	iuphar.ligand:223	[3H]RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3333	iuphar.ligand:3333	RESOLVIN E1	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:11439	iuphar.ligand:11439	RCI-0879	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.078958904	TYRPHOSTIN AG-1478	iuphar.ligand:4862	AG1478	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.1193356164447602	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
APP	hgnc:620	APP	DTC	9/2/20	NULL	1.615620653405984	REL-3,5-DICAFFEOYLQUINIC ACID	chembl:CHEMBL249447	3,5-DICAFFEOYLQUINIC ACID	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.4773424657790409	Tolmetin	rxcui:10636	TOLMETIN	TRUE	FALSE	FALSE
NCBIGENE:2605	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8891	iuphar.ligand:8891	SGI-1027	FALSE	FALSE	FALSE
NCBIGENE:2757	hgnc:23177	KEAP1	GuideToPharmacology	2024.1	NULL	2.100306849	IUPHAR.LIGAND:10071	iuphar.ligand:10071	ISOQUINOLINE 17 [PMID: 30122040]	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:2929	iuphar.ligand:2929	COMPOUND 26 [PMID: 16190743]	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	TAXOL C	chembl:CHEMBL306601	TAXOL C	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.6168664383892681	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
ALDEHYDE OXIDASE	hgnc:553	AOX1	TTD	2020.06.01	NULL	10.50153424713889	Isovanillin	chembl:CHEMBL275563	ISOVANILLIN	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.5834185692854944	TAK-960	chembl:CHEMBL2392545	TAK-960	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.1402073998282897	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.070448575	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.081281225	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	7.501095891	BMS-986205	ncit:C141135	LINRODOSTAT	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	Levopropoxyphene Napsylate Anhydrous	ncit:C90775	LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.090530468	NSC-327705	chembl:CHEMBL1317986	CHEMBL:CHEMBL1317986	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2083637747448194	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1750255707856483	BROMOXYNIL	chembl:CHEMBL453905	BROMOXYNIL	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.092988792	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	modulator	0.7955707762984014	IUPHAR.LIGAND:10585	iuphar.ligand:10585	COMPOUND 39 [PMID: 31742400]	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1930429089547591	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.01060761	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	4.039051633514961	2,5-DINITRO-PHENOL	chembl:CHEMBL107513	CHEMBL:CHEMBL107513	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2075402025126264	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
LEUKOTRIENE B4 RECEPTOR 2	hgnc:19260	LTB4R2	TTD	2020.06.01	NULL	3.281729452230906	LTB4	iuphar.ligand:2487	LTB4	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.096167896	domperidone	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.4134462302023188	SIMAZINE	chembl:CHEMBL1605837	SIMAZINE	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	3.000438356	TAK-659	ncit:C188286	MIVAVOTINIB CITRATE	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1041818873724097	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
CD33	hgnc:1659	CD33	ChEMBL	33	binder	4.039051633514961	GEMTUZUMAB	ncit:C171025	GEMTUZUMAB	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	1,5-NAPHTHALENEDIAMINE	chembl:CHEMBL538965	CHEMBL:CHEMBL538965	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	GALUTEOLIN	chembl:CHEMBL233929	GALUTEOLIN	FALSE	FALSE	FALSE
TERC	hgnc:11727	TERC	NCI	14-Sep-17	NULL	1.875273972703374	IFO	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
NRG2	hgnc:7998	NRG2	PharmGKB	4/5/24	NULL	0.7292732116068681	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	RO-318220	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
YES TYROSINE KINASE	hgnc:12841	YES1	TTD	2020.06.01	NULL	0.056097939	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.030996264	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	0.064824285	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6156	iuphar.ligand:6156	SC-41930	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	inhibitor	0.3431873936973497	NALOXONE HYDROCHLORIDE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRM1	hgnc:15759	ADRM1	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
KCNC1	hgnc:6233	KCNC1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
UNIPROT:P19838	hgnc:7794	NFKB1	TdgClinicalTrial	Jan-14	NULL	0.029876342	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.074478966	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.085239726	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:160	iuphar.ligand:160	AL-37350A	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.3170753093942904	DOXAZOSIN	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.3314878234576672	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
MT-CO2	hgnc:7421	MT-CO2	DTC	9/2/20	NULL	1.567393171214761	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
UNIPROT:Q08493	hgnc:8782	PDE4C	TEND	1-Aug-11	NULL	0.7759754369807069	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	DEQUALINIUM	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.049349315	IUPHAR.LIGAND:5677	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
KAT5	hgnc:5275	KAT5	DTC	9/2/20	NULL	7.501095890813499	ANACARDIC ACID	iuphar.ligand:6999	ANACARDIC ACID	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	2.187819634820604	FIBRIN SEALANT	ncit:C2664	FIBRIN SEALANT	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 1	hgnc:1602	CCR1	TTD	2020.06.01	NULL	5.834185692854944	CCX-354	drugbank:DB12963	CCX-354	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:12119	iuphar.ligand:12119	NVP-CLR457	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS	ncit:C90775	LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.057385433	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
STK33	hgnc:14568	STK33	DTC	9/2/20	inhibitor	1.312691780892362	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.1023541349623674	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.4167275494896388	RANTES	ncit:C1211	RECOMBINANT RANTES	FALSE	FALSE	FALSE
SODIUM/BILE ACID COTRANSPORTER	hgnc:10905	SLC10A1	TTD	2020.06.01	NULL	2.917092846427472	LUM001	iuphar.ligand:11708	MARALIXIBAT	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.2430910705356226	IUPHAR.LIGAND:1935	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
GRM1	hgnc:4593	GRM1	NCI	14-Sep-17	NULL	0.2853677784548614	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
TRPC5	hgnc:12337	TRPC5	DTC	9/2/20	NULL	21.00306849427779	2-AMINOETHYLMETHANETHIOSULPHONATE HYDROBROMIDE	chembl:CHEMBL271256	CHEMBL:CHEMBL271256	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.076934317	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	DTC	9/2/20	NULL	3.500511415712966	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
TNFRSF1B	hgnc:11917	TNFRSF1B	NCI	14-Sep-17	NULL	0.2143170254518142	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.026412309	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002629854	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	1.666910197958555	raltitrexed	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.00897567	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ARF1	hgnc:652	ARF1	PharmGKB	4/5/24	NULL	0.5933070196123672	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.050488145	vilazodone	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.305277158	ABEDITEROL	ncit:C132738	ABEDITEROL	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10549	iuphar.ligand:10549	COMPOUND 18E [PMID: 31670517]	FALSE	FALSE	FALSE
CYP11B1	hgnc:2591	CYP11B1	ChEMBL	33	inhibitor	8.751278539282415	OSILODROSTAT PHOSPHATE	rxcui:2286253	OSILODROSTAT PHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:636	hgnc:1049	BICD1	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:8838	iuphar.ligand:8838	COMPOUND 10 [PMID: 18759424]	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6290	iuphar.ligand:6290	METHYL ISOCYANATE	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.1419126249613365	Trazodone	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	PALMITOYL-CARNITINE	chembl:CHEMBL301722	PALMITOYL-CARNITINE	FALSE	FALSE	FALSE
AQP4	hgnc:637	AQP4	PharmGKB	4/5/24	NULL	0.4605936073306534	satralizumab	rxcui:2391541	SATRALIZUMAB	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	inhibitor	0.01875274	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.1041818873724097	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.033338204	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
GAA	hgnc:4065	GAA	ChEMBL	33	inhibitor	0.5469549087051511	MIGLITOL	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	3,4-METHYLENEDIOXYB-NITROSTYRENE	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.9546849315580819	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	OncoKB	23-Jul-20	NULL	0.096264064	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	DOXYLAMINE SUCCINATE	rxcui:23665	DOXYLAMINE SUCCINATE	TRUE	FALSE	FALSE
NCBIGENE:2832	hgnc:4530	NPBWR2	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:11831	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.4375639269641208	PANCURONIUM BROMIDE	rxcui:7884	PANCURONIUM BROMIDE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.096050618	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.014099804	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inverse agonist	0.1544343271638073	HALOPERIDOL LACTATE	rxcui:217483	HALOPERIDOL LACTATE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.118072806	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:1447	hgnc:2447	CSN2	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9548	iuphar.ligand:9548	GNF362	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:7158	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
NCBIGENE:3015	hgnc:4741	H2AZ1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12802	iuphar.ligand:12802	ZED1227	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.021501913	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	H-89 CHLORIDE	chembl:CHEMBL1315166	CHEMBL:CHEMBL1315166	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	4,4'-DITHIODIPYRIDINE	chembl:CHEMBL1232076	CHEMBL:CHEMBL1232076	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.012020987	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1752592497853621	DIENESTROL	rxcui:3368	DIENESTROL	TRUE	FALSE	FALSE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	0.7721716358190367	ADAPALENE	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
NCBIGENE:659	hgnc:1078	BMPR2	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:12422	iuphar.ligand:12422	COHUMULONE	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.056142926	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.074163377	AT-9283	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7568	iuphar.ligand:7568	CANGITOXIN II	FALSE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	0.1440539677248134	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.2453629496995069	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.007841647	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-239272	chembl:CHEMBL275798	CHEMBL:CHEMBL275798	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	NSC-327705	chembl:CHEMBL1317986	CHEMBL:CHEMBL1317986	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	ZAPA	chembl:CHEMBL20562	ZAPA	FALSE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TEND	1-Aug-11	NULL	0.8078103267029924	ISOSORBIDE-5-MONONITRATE	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.075732218	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	ChEMBL	33	inhibitor	0.3409589041278863	BIRABRESIB	ncit:C103298	BIRABRESIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	FLUMETHASONE PIVALATE	rxcui:25113	FLUMETHASONE PIVALATE	TRUE	FALSE	FALSE
ABCA1	hgnc:29	ABCA1	PharmGKB	4/5/24	NULL	0.011096296	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	TELENZEPINE	ncit:C75285	TELENZEPINE	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.046549354	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.062645859	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.3281729452230906	artemether	rxcui:18343	ARTEMETHER	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	PharmGKB	4/5/24	NULL	0.4773424657790409	temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.2397610558707511	NSC-407228	chembl:CHEMBL74852	CHEMBL:CHEMBL74852	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.03409589	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	blocker	0.1058622403945453	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPS12	hgnc:10385	RPS12	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	inhibitor	5.250767123569449	VOLAGIDEMAB	ncit:C167005	VOLAGIDEMAB	FALSE	FALSE	FALSE
NCBIGENE:1244	hgnc:53	ABCC2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:9017	iuphar.ligand:9017	COMPOUND 9 [PMID: 23472952]	FALSE	FALSE	FALSE
NCBIGENE:1617	hgnc:2682	DAZ1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9034	iuphar.ligand:9034	VRT-043198	FALSE	FALSE	FALSE
NCBIGENE:2821	hgnc:4458	GPI	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7827	iuphar.ligand:7827	AZD7687	FALSE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:3945	drugbank:DB12480	BETULINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:8959	iuphar.ligand:8959	ENSARTINIB	FALSE	FALSE	FALSE
KMT2D	hgnc:7133	KMT2D	CIViC	10-Apr-24	NULL	13.12691780892362	HDAC INHIBITOR REC-2282	ncit:C116850	HDAC INHIBITOR REC-2282	FALSE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.061412481	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.018193926	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
GYPA	hgnc:4702	GYPA	NCI	14-Sep-17	NULL	3.750547945	IL-8	ncit:C1289	RECOMBINANT INTERLEUKIN-8	FALSE	FALSE	FALSE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	1.250182648468916	RADOTINIB	ncit:C98110	RADOTINIB	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	1.050153425	SENAPARIB	ncit:C168601	SENAPARIB	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.079557078	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	3.500511415712966	NERIDRONIC ACID	ncit:C66230	NERIDRONIC ACID	FALSE	FALSE	FALSE
CYR61	hgnc:2654	CCN1	NCI	14-Sep-17	NULL	4.375639269641208	HYPOTENSIVE AGENTS	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	SEROTONIN	rxcui:1311214	SEROTONIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.008475815	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.012805187	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.02875557	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.017691264	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.098328972	IUPHAR.LIGAND:8969	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1715936968486748	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	5.834185692854944	IUPHAR.LIGAND:10522	ncit:C160786	AVADOMIDE	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.05814803	IUPHAR.LIGAND:4108	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	1.166837138570988	2,4-DIHYDROXY BENZOIC ACID HYDRAZIDE	chembl:CHEMBL1339206	CHEMBL:CHEMBL1339206	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.2548916079402645	SCANDENIN	chembl:CHEMBL1603825	SCANDENIN	FALSE	FALSE	FALSE
MT-ND1	hgnc:7455	MT-ND1	ChEMBL	33	inhibitor	0.1029562181092049	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.020218587	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.1400204566285186	MITOGLITAZONE	drugbank:DB11721	MITOGLITAZONE	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.2386712328895204	2-PICOLINIC ACID	chembl:CHEMBL72628	2-PICOLINIC ACID	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.050488145	CCT018159	chembl:CHEMBL399530	CHEMBL:CHEMBL399530	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.014206621	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.577007376	GNF-PF-4085	chembl:CHEMBL528181	CHEMBL:CHEMBL528181	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000547046	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.087537101	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.8468979231563628	PHENINDAMINE	rxcui:33283	PHENINDAMINE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.346350544504987	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.008458066	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1459	iuphar.ligand:1459	MOTILIN	FALSE	FALSE	FALSE
MAT1A	hgnc:6903	MAT1A	NCI	14-Sep-17	NULL	3.182283105193606	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.026599631	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:11224	iuphar.ligand:11224	BAY-545	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	5-NITROACENAPHTHENE	chembl:CHEMBL423081	CHEMBL:CHEMBL423081	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.7955707762984014	FORMESTANE	rxcui:15070	FORMESTANE	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.06886252	eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
FGF22	hgnc:3679	FGF22	DTC	9/2/20	NULL	0.7501095890813501	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
FDPS	hgnc:3631	FDPS	ChEMBL	33	inhibitor	3.500511415712966	IBANDRONATE SODIUM	rxcui:236916	IBANDRONATE SODIUM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.040021091	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1546	iuphar.ligand:1546	[PRO34]PYY (HUMAN)	FALSE	FALSE	FALSE
E2F5	hgnc:3119	E2F5	ChEMBL	33	inhibitor	2.187819634820604	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.1392776425349987	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.01893533	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW829906X	chembl:CHEMBL434729	GW829906X	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.2160809515872201	ALECTINIB HYDROCHLORIDE	rxcui:1727454	ALECTINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.150021918	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.9479406894984094	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.1137761023525341	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.062065805	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	FDA	10-Apr-24	NULL	0.03849536	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.03261346	Morphine	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1166837138570989	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.2344092465879218	GUANABENZ ACETATE	rxcui:227225	GUANABENZ ACETATE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	AG-13958	chembl:CHEMBL3545335	AG-13958	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.048935388	IUPHAR.LIGAND:1357	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
PPT1	hgnc:9325	PPT1	NCI	14-Sep-17	NULL	2.386712328895204	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	NCI	14-Sep-17	NULL	0.9723642821424906	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	CIRAZOLINE	ncit:C77294	CIRAZOLINE	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.1919140030544389	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	NULL	10.74020548002842	IUPHAR.LIGAND:10199	rxcui:1999382	TEZACAFTOR	TRUE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	blocker	0.3017682254924971	IUPHAR.LIGAND:4369	iuphar.ligand:4369	[35S]TBPS	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.1162960603226899	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.070574827	TERFENADINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	3-HYDROXYBENZYLHYDRAZINE DIHYDROCHLORIDE	iuphar.ligand:5116	3-HYDROXYBENZYLHYDRAZINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.005085489	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	1.848379561100067	Captopril	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	0.021501913	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.080905503	BI847325	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
PRKAG2	hgnc:9386	PRKAG2	PharmGKB	4/5/24	NULL	0.5707355569097228	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
PRSS3	hgnc:9486	PRSS3	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	1.250182648468916	Savolitinib	ncit:C104732	SAVOLITINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	EMETINE DIHYDROCHLORIDE	chembl:CHEMBL493439	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.018031481	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
B2M	hgnc:914	B2M	NCI	14-Sep-17	NULL	1.875273972703374	AMIKACIN	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.041872146	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	1.779921058837101	TASOSARTAN	ncit:C152517	TASOSARTAN	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.182318303	TEPROTUMUMAB	rxcui:2274802	TEPROTUMUMAB-TRBW	TRUE	FALSE	TRUE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.049723174	IUPHAR.LIGAND:360	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
SDHB	hgnc:10681	SDHB	NCI	14-Sep-17	NULL	1.544343271638073	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
P2Y PURINOCEPTOR 12	hgnc:18124	P2RY12	TTD	2020.06.01	NULL	9.845188356692718	Elinogrel	ncit:C96896	ELINOGREL	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.2678962818147679	Fruquintinib	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.05814803	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.4948366922735607	binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	2-METHOXYPHENAZINE	chembl:CHEMBL1420181	CHEMBL:CHEMBL1420181	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TCMDC-125539	chembl:CHEMBL533388	CHEMBL:CHEMBL533388	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	inhibitor	0.008103036	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	NCI	14-Sep-17	NULL	0.010672291	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
THRA	hgnc:11796	THRA	ChEMBL	33	agonist	0.9092237443410304	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
LRP1B	hgnc:6693	LRP1B	CIViC	10-Apr-24	NULL	0.1166837138570988	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
DNPEP	hgnc:2981	DNPEP	ChEMBL	33	inhibitor	1.312691780892362	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	4.039051633514961	RG-7652	chembl:CHEMBL2109539	RG-7652	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.060772768	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001573971	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
UNIPROT:P43116	hgnc:9594	PTGER2	TEND	1-Aug-11	NULL	0.5707355569097228	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	RO-0282750	chembl:CHEMBL1397270	CHEMBL:CHEMBL1397270	FALSE	FALSE	FALSE
NADH DEHYDROGENASE	hgnc:7458	MT-ND3	TTD	2020.06.01	NULL	13.12691780892362	NADH	rxcui:7222	NADH	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.052507671	quinacrine	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	modulator	0.1312691780892362	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CXCR1	hgnc:6026	CXCR1	ChEMBL	33	inhibitor	3.750547945	SX-682	chembl:CHEMBL4297480	SX-682	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	E-10030	chembl:CHEMBL3301576	PEGPLERANIB SODIUM	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	1.129197231	AVX-470	drugbank:DB18455	AVX-470	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.05814803	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.1881995384791917	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:706	hgnc:1158	TSPO	GuideToPharmacology	2024.1	blocker	0.2763561643983921	IUPHAR.LIGAND:4177	iuphar.ligand:4177	DIDS	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:13009	iuphar.ligand:13009	NDT-19795	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 5	hgnc:1606	CCR5	TTD	2020.06.01	NULL	2.625383561784724	INCB9471	chembl:CHEMBL1688243	INCB-9471	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	NCI	14-Sep-17	NULL	0.217423069	9-CRA	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	1.334940794127826	Azilsartan	rxcui:1091642	AZILSARTAN MEDOXOMIL	TRUE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	negative modulator	0.1187956362798518	KETAMINE HYDROCHLORIDE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1060761035064535	SAQUINAVIR	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.5000730593875667	MIVACURIUM CHLORIDE	rxcui:52796	MIVACURIUM CHLORIDE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.1209854175937661	DELUCEMINE	ncit:C76776	DELUCEMINE	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1154014752432846	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.058997383	IUPHAR.LIGAND:957	iuphar.ligand:957	(+)-UH232	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.2160809515872201	IUPHAR.LIGAND:5820	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	1,2-DIPHENYLDISULFANE	chembl:CHEMBL462861	CHEMBL:CHEMBL462861	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.3977853881492007	LYNGBYABELLIN A	chembl:CHEMBL453207	LYNGBYABELLIN A	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
PSMB6	hgnc:9543	PSMB6	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	NCI	14-Sep-17	NULL	0.019093699	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CTSK	hgnc:2536	CTSK	TALC	12-May-16	inhibitor	11.66837138570988	BALICATIB	ncit:C79521	BALICATIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.011316308	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DAZOMET	chembl:CHEMBL1407826	DAZOMET	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
RPS2	hgnc:10404	RPS2	NCI	14-Sep-17	NULL	17.50255707856483	FGF3	ncit:C1466	RECOMBINANT FIBROBLAST GROWTH FACTOR 3	FALSE	FALSE	FALSE
UNIPROT:P49190	hgnc:9609	PTH2R	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	ALX1-11	chembl:CHEMBL2108078	PARATHYROID HORMONE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.8178764989983567	INCB54828	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.052718545	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.045898314	IUPHAR.LIGAND:5617	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8537	iuphar.ligand:8537	ONO-AE3-237	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.057700738	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.022632617	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	GNF-PF-4337	chembl:CHEMBL277148	CHEMBL:CHEMBL277148	FALSE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.3804903712731485	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.03378872	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	NIALAMIDE	rxcui:7394	NIALAMIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
VASOACTIVE INTESTINAL POLYPEPTIDE RECEPTOR 1	hgnc:12694	VIPR1	TTD	2020.06.01	NULL	6.563458904461812	Vasoactive intestinal peptide	rxcui:1942960	VASOACTIVE INTESTINAL PEPTIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00607587	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.054355767	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.021422958	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.090922374	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
ENOSF1	hgnc:30365	ENOSF1	NCI	14-Sep-17	NULL	0.8751278539282416	3TC	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.015613343	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.2071308530007672	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	CancerCommons	25-Jul-13	inhibitor	0.1103102336884338	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	CancerCommons	25-Jul-13	inhibitor	0.2083637747448194	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	CancerCommons	25-Jul-13	inhibitor	1.826353782111112	X-396	drugbank:DB13104	X-396	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.051511777	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.0545251	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.035122188	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
HGF	hgnc:4893	HGF	CGI	2/1/22	NULL	0.04321619	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	LEVOCABASTINE HYDROCHLORIDE	rxcui:1294532	LEVOCABASTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.8468979231563628	ACRIVASTINE	rxcui:19959	ACRIVASTINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1383601350084176	MOLINDONE HYDROCHLORIDE	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	ACETOPHENAZINE MALEATE	rxcui:91127	ACETOPHENAZINE MALEATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.034590034	TRIFLUPROMAZINE HYDROCHLORIDE	rxcui:91125	TRIFLUPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
INHA	hgnc:6065	INHA	ChEMBL	33	inhibitor	17.50255707856483	ETHIONAMIDE	rxcui:4127	ETHIONAMIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.546954909	SILODOSIN	rxcui:720825	SILODOSIN	TRUE	FALSE	FALSE
CALCR	hgnc:1440	CALCR	ChEMBL	33	agonist	6.563458904461812	CALCITONIN HUMAN	rxcui:235481	HUMAN CALCITONIN	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	0.2206204673768676	MECLOFENAMATE SODIUM	rxcui:6677	MECLOFENAMATE SODIUM	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2792961235941196	BENZTROPINE MESYLATE	rxcui:18927	BENZTROPINE MESYLATE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	CYCRIMINE HYDROCHLORIDE	rxcui:235421	CYCRIMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TXNRD1	hgnc:12437	TXNRD1	ChEMBL	33	inhibitor	1.009762908	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1591141552596803	TRAZODONE HYDROCHLORIDE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.1193356164447602	DIBUCAINE HYDROCHLORIDE	rxcui:235402	DIBUCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.1486416737033106	PARICALCITOL	rxcui:73710	PARICALCITOL	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.084146909	MOLINDONE HYDROCHLORIDE	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.077217164	TRAZODONE HYDROCHLORIDE	rxcui:10737	TRAZODONE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1262203635473425	HALOPERIDOL LACTATE	rxcui:217483	HALOPERIDOL LACTATE	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	15.00219178	TRAVOPROST	rxcui:283809	TRAVOPROST	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1204304386139782	SUFENTANIL CITRATE	rxcui:58964	SUFENTANIL CITRATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.060215219	TRAMADOL HYDROCHLORIDE	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	LEVORPHANOL TARTRATE	rxcui:153973	LEVORPHANOL TARTRATE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	DONEPEZIL HYDROCHLORIDE	rxcui:236559	DONEPEZIL HYDROCHLORIDE	TRUE	FALSE	FALSE
GHRHR	hgnc:4266	GHRHR	ChEMBL	33	agonist	13.12691780892362	TESAMORELIN ACETATE	rxcui:1044583	TESAMORELIN ACETATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.2408608772279564	BUTORPHANOL TARTRATE	rxcui:203170	BUTORPHANOL TARTRATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.133607306	PREDNISOLONE ACETATE	rxcui:34372	PREDNISOLONE ACETATE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	0.047561296	URSODIOL	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.062645859	ESTRADIOL ACETATE	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.7095631248066824	SELEGILINE HYDROCHLORIDE	rxcui:203137	SELEGILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.1182605208011137	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	agonist	0.8607814956671229	BECAPLERMIN	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	negative modulator	0.1891032577516008	KETAMINE HYDROCHLORIDE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.062139256	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.3241214273808303	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.1620607136904151	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	potentiator	0.1508841127462485	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.080781033	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.043866058	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	0.5048814541893702	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.019949723	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3125456621172291	AMLODIPINE MALEATE	ncit:C65230	AMLODIPINE MALEATE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.2476776945079929	AMLODIPINE MALEATE	ncit:C65230	AMLODIPINE MALEATE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.305277158	AMLODIPINE MALEATE	ncit:C65230	AMLODIPINE MALEATE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.04464938	NIFEDIPINE	rxcui:7417	NIFEDIPINE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	0.5097832158805291	DEXTROTHYROXINE SODIUM	rxcui:40070	DEXTROTHYROXINE SODIUM	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	ChEMBL	33	agonist	0.1593072549626653	LEVOTHYROXINE SODIUM	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	ChEMBL	33	inhibitor	0.6863747873946993	RILONACEPT	rxcui:763450	RILONACEPT	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	INDACATEROL MALEATE	rxcui:1114325	INDACATEROL MALEATE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	0.7095631248066824	FOSAPREPITANT DIMEGLUMINE	rxcui:1731071	FOSAPREPITANT	TRUE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:3875	iuphar.ligand:3875	EUROPIUM-LABELLED INSL3	FALSE	FALSE	FALSE
GE	hgnc:4704	GYPC	ChEMBL	33	inhibitor	2.187819634820604	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
GL	hgnc:14942	PPP1R3B	ChEMBL	33	inhibitor	6.563458904461812	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
COL6A2	hgnc:2212	COL6A2	ChEMBL	33	cleavage	0.6250913242344582	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL6A5	hgnc:26674	COL6A5	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	ChEMBL	33	cleavage	0.1339481409073839	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL15A1	hgnc:2192	COL15A1	ChEMBL	33	cleavage	0.3750547945406749	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL5A2	hgnc:2210	COL5A2	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.100976291	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
PSMB6	hgnc:9543	PSMB6	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD14	hgnc:16889	PSMD14	ChEMBL	33	inhibitor	0.1878628666751144	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD8	hgnc:9566	PSMD8	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD4	hgnc:9561	PSMD4	ChEMBL	33	inhibitor	0.3488881809680698	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV006787	chembl:CHEMBL584235	CHEMBL:CHEMBL584235	FALSE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	agonist	3.938075342677087	IMIQUIMOD	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.3281729452230906	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.5527123287967842	MIVACURIUM CHLORIDE	rxcui:52796	MIVACURIUM CHLORIDE	TRUE	FALSE	FALSE
NDUFB6	hgnc:7701	NDUFB6	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MT-ND4L	hgnc:7460	MT-ND4L	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MT-ND3	hgnc:7458	MT-ND3	ChEMBL	33	inhibitor	0.2344092465879218	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PROPARGITE	chembl:CHEMBL1416084	PROPARGITE	FALSE	FALSE	FALSE
NDUFA6	hgnc:7690	NDUFA6	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFAB1	hgnc:7694	NDUFAB1	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	ChEMBL	33	agonist	0.4667348554283955	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	0.4412409347537352	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
RXRB	hgnc:10478	RXRB	ChEMBL	33	agonist	0.364636606	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
ATP1A3	hgnc:801	ATP1A3	ChEMBL	33	inhibitor	0.364636606	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	METHYLBENZETHONIUM CHLORIDE	rxcui:1796444	METHYLBENZETHONIUM CHLORIDE	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.026227608	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.070543222	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.077789143	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.053854022	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.088945801	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.075261832	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.081533651	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.027840759	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.076098074	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.07963752	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1346350544504987	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	TIGECYCLINE	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	ChEMBL	33	agonist	0.091159151	PEGINTERFERON ALFA-2B	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	potentiator	0.073885091	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
FSHR	hgnc:3969	FSHR	ChEMBL	33	agonist	18.37768493249307	MENOTROPINS	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	ChEMBL	33	inhibitor	0.151464436	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.6250913242344582	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.076098074	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.2251615404618117	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.3113103037689397	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.3314878234576672	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NR1H2	hgnc:7965	NR1H2	ChEMBL	33	agonist	4.039051633514961	BMS-779788	chembl:CHEMBL3545418	BMS-779788	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.111481255	ILX23-7553	chembl:CHEMBL284121	ILX23-7553	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	1.579178082276526	CER-002	chembl:CHEMBL3544958	CER-002	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.098605955	ESTROGEN ANTAGONIST	ncit:C481	ANTIESTROGEN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.3947945205691315	DB959	chembl:CHEMBL3545176	DB959	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.2273059360852575	AG-24322	drugbank:DB13035	AG-24322	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.276356164	DERAZANTINIB	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.3680444245492605	DERAZANTINIB	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.035216413	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
CO-STIMULATORY MOLECULE 4-1BB	hgnc:11924	TNFRSF9	TTD	2020.06.01	NULL	52.50767123569449	PF-05082566	ncit:C116619	UTOMILUMAB	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	ChEMBL	33	inhibitor	3.889457128569962	BI-853520	chembl:CHEMBL3544961	BI-853520	FALSE	FALSE	FALSE
NDUFB6	hgnc:7701	NDUFB6	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA6	hgnc:7690	NDUFA6	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
MT-ND6	hgnc:7462	MT-ND6	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFB7	hgnc:7702	NDUFB7	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA7	hgnc:7691	NDUFA7	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.6667640791834221	PF-04217903	drugbank:DB12848	PF-04217903	FALSE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.095122593	PF-03715455	drugbank:DB12138	PF-03715455	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	2.019525817	LY-2811376	drugbank:DB13065	LY-2811376	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	TA-5493	chembl:CHEMBL3545201	TA-5493	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.097236428	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.2778183663264258	DELUCEMINE	ncit:C76776	DELUCEMINE	FALSE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.182318303	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	ChEMBL	33	modulator	0.7001022831425933	SDX-101	chembl:CHEMBL1716091	SDX-101	FALSE	FALSE	FALSE
NCBIGENE:2798	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	activator	0.3977853881492007	IUPHAR.LIGAND:11932	iuphar.ligand:11932	BMS-820132	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	1.591141552596803	LY-518674	drugbank:DB12988	LY-518674	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.075768645	BRIGATINIB	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2083637747448194	AG-13958	chembl:CHEMBL3545335	AG-13958	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.4688184931758437	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	1.250182648468916	SAVOLITINIB	ncit:C104732	SAVOLITINIB	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	0.750109589	ENTOSPLETINIB	ncit:C105402	ENTOSPLETINIB	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.2734774543525755	MIRDAMETINIB	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.5000730593875666	RIVICICLIB	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1355619739303644	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.095500063	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.09869863	IUPHAR.LIGAND:9619	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.192335792	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.6141248097742047	ABEMACICLIB	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1035654265003836	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.375054795	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1875273972703375	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.082754407	INFIGRATINIB	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.6783936852156912	INFIGRATINIB	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	inhibitor	0.5048814541893701	GSK163090	chembl:CHEMBL1631540	GSK163090	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	1.009762908	PRUVANSERIN	ncit:C72834	PRUVANSERIN	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1491695205559502	GSK163090	chembl:CHEMBL1631540	GSK163090	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	inhibitor	0.1773907812016706	GSK163090	chembl:CHEMBL1631540	GSK163090	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	1.346350544504987	NARONAPRIDE	ncit:C175157	NARONAPRIDE	FALSE	FALSE	FALSE
CXCR2	hgnc:6027	CXCR2	ChEMBL	33	inhibitor	2.917092846427472	DANIRIXIN	ncit:C169874	DANIRIXIN	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	PF-03654746	drugbank:DB12201	PF-03654746	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	2.917092846427472	SELODENOSON	ncit:C75135	SELODENOSON	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	CYH33	ncit:C178401	RISOVALISIB	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.4150804050252529	APLINDORE FUMARATE	ncit:C76649	APLINDORE FUMARATE	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	2.763561643983921	ADC3680	chembl:CHEMBL3545343	ADC3680	FALSE	FALSE	FALSE
CXCR1	hgnc:6026	CXCR1	ChEMBL	33	modulator	3.750547945	LADARIXIN	ncit:C170087	LADARIXIN	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	agonist	0.042619863	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	agonist	0.038159645	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	agonist	0.025439763	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	agonist	0.039068208	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	agonist	0.040515178	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	agonist	0.036062961	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	agonist	0.042073455	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	agonist	0.041540879	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	agonist	0.044347695	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.2917092846427472	LYCOBETAINE	chembl:CHEMBL253553	LYCOBETAINE	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	agonist	0.072927321	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.4167275494896388	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.037213091	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	8.078103267029922	BOCOCIZUMAB	ncit:C166723	BOCOCIZUMAB	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.038894571	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.042174836	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	SJ000147784	chembl:CHEMBL590186	CHEMBL:CHEMBL590186	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.035719504	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1029562181092049	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
LNPEP	hgnc:6656	LNPEP	ChEMBL	33	inhibitor	0.8751278539282418	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.091796628	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
LAP3	hgnc:18449	LAP3	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PSMA3	hgnc:9532	PSMA3	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB9	hgnc:9546	PSMB9	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMD13	hgnc:9558	PSMD13	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	ChEMBL	33	inhibitor	0.192335792	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMA8	hgnc:22985	PSMA8	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-23	hgnc:3680	FGF23	TTD	2020.06.01	NULL	105.0153424713889	Burosumab	rxcui:2043854	BUROSUMAB-TWZA	TRUE	FALSE	FALSE
PSMC6	hgnc:9553	PSMC6	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.042174836	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.2122951667211368	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	1.458546423213736	ARBACLOFEN PLACARBIL	ncit:C76088	ARBACLOFEN PLACARBIL	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	negative modulator	0.042174836	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
NCBIGENE:122	ncbigene:122	ADFN	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:2916	iuphar.ligand:2916	DIOCTANOYLGLYCEROL PYROPHOSPHATE	FALSE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	ChEMBL	33	inhibitor	0.596678082	BEGACESTAT	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
EGLN2	hgnc:14660	EGLN2	ChEMBL	33	inhibitor	2.100306849	DAPRODUSTAT	rxcui:2628210	DAPRODUSTAT	TRUE	FALSE	FALSE
P4HTM	hgnc:28858	P4HTM	ChEMBL	33	inhibitor	5.250767124	DAPRODUSTAT	rxcui:2628210	DAPRODUSTAT	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.094099769	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
BCL2L2	hgnc:995	BCL2L2	ChEMBL	33	inhibitor	0.8204323630577265	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
GAA	hgnc:4065	GAA	ChEMBL	33	inhibitor	0.182318303	VOGLIBOSE	ncit:C95221	VOGLIBOSE	TRUE	FALSE	FALSE
CRBN	hgnc:30185	CRBN	ChEMBL	33	inhibitor	2.917092846427472	POMALIDOMIDE	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
SI	hgnc:10856	SI	ChEMBL	33	inhibitor	1.640864726115453	VOGLIBOSE	ncit:C95221	VOGLIBOSE	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	ChEMBL	33	inhibitor	8.290684931951763	CAPLACIZUMAB	rxcui:2110604	CAPLACIZUMAB-YHDP	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.3697723326457359	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
VEGFB	hgnc:12681	VEGFB	ChEMBL	33	inhibitor	1.750255707856483	CONBERCEPT	ncit:C162879	CONBERCEPT	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	other/unknown	0.7059854956059763	AVELUMAB	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
F10	hgnc:3528	F10	ChEMBL	33	other/unknown	0.5357925636295356	EMICIZUMAB	rxcui:1989794	EMICIZUMAB	TRUE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	other/unknown	4.375639269641208	SONTUZUMAB	ncit:C38697	SONTUZUMAB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	HEXYLRESORCINOL	rxcui:5321	HEXYLRESORCINOL	TRUE	FALSE	FALSE
PTHLH	hgnc:9607	PTHLH	ChEMBL	33	inhibitor	8.751278539282415	CAL	chembl:CHEMBL2109562	CAL	FALSE	FALSE	FALSE
TRAV29DV5	hgnc:12127	TRAV29DV5	ChEMBL	33	inhibitor	3.500511415712967	TOL-101	drugbank:DB16980	TOL-101	FALSE	FALSE	FALSE
PARP3	hgnc:273	PARP3	ChEMBL	33	inhibitor	2.917092846427472	RUCAPARIB CAMSYLATE	rxcui:1862578	RUCAPARIB CAMSYLATE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.5645986154375752	AZ9773	chembl:CHEMBL2109587	AZ9773	FALSE	FALSE	FALSE
HTR3D	hgnc:24004	HTR3D	ChEMBL	33	agonist	0.2206204673768676	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1E	hgnc:5291	HTR1E	ChEMBL	33	agonist	0.6177373086552295	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MUC5AC	hgnc:7515	MUC5AC	ChEMBL	33	binder	13.12691780892362	CLIVATUZUMAB TETRAXETAN	ncit:C166491	CLIVATUZUMAB TETRAXETAN	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	1.750255707856483	VANUCIZUMAB	ncit:C118578	VANUCIZUMAB	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	4.449802647092754	CILAZAPRIL	rxcui:21102	CILAZAPRIL	TRUE	FALSE	FALSE
FSHR	hgnc:3969	FSHR	ChEMBL	33	agonist	21.00306849427779	CORIFOLLITROPIN ALFA	ncit:C169865	CORIFOLLITROPIN ALFA	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.09969811	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.096050618	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2237542808339254	CELIPROLOL	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.1229687850953032	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	2.625383561784724	DUTETRABENAZINE	chembl:CHEMBL3137326	DUTETRABENAZINE	TRUE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	2.917092846427472	IMMURAIT-LL2	chembl:CHEMBL2109508	IMMURAIT-LL2	FALSE	FALSE	FALSE
FAP	hgnc:3590	FAP	ChEMBL	33	binder	4.039051633514961	SIBROTUZUMAB	ncit:C156438	SIBROTUZUMAB	FALSE	FALSE	FALSE
CDH3	hgnc:1762	CDH3	ChEMBL	33	inhibitor	26.25383561784724	PF-03732010	chembl:CHEMBL2109534	PF-03732010	FALSE	FALSE	FALSE
CD276	hgnc:19137	CD276	ChEMBL	33	modulator	31.50460274141669	ENOBLITUZUMAB	ncit:C97510	ENOBLITUZUMAB	FALSE	FALSE	FALSE
KCNS1	hgnc:6300	KCNS1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	ERAVACYCLINE DIHYDROCHLORIDE	rxcui:2055907	ERAVACYCLINE DIHYDROCHLORIDE	TRUE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	ChEMBL	33	inhibitor	0.6731752722524935	BMS-986158	drugbank:DB15435	BMS-986158	FALSE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	ChEMBL	33	inhibitor	0.4605936073306534	CD24FC	chembl:CHEMBL4297717	CD24FC	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	ChEMBL	33	positive modulator	0.2051080907644316	ONASEMNOGENE ABEPARVOVEC	rxcui:2170225	ONASEMNOGENE ABEPARVOVEC-XIOI	TRUE	FALSE	FALSE
EZH2	hgnc:3527	EZH2	ChEMBL	33	inhibitor	2.917092846427472	TAZEMETOSTAT HYDROBROMIDE	rxcui:2274379	TAZEMETOSTAT HYDROBROMIDE	TRUE	FALSE	FALSE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	2.561349816375341	AXICABTAGENE CILOLEUCEL	rxcui:1987398	AXICABTAGENE CILOLEUCEL	TRUE	FALSE	FALSE
HSPA1A	hgnc:5232	HSPA1A	ChEMBL	33	inhibitor	2.187819634820604	CD24FC	chembl:CHEMBL4297717	CD24FC	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2234368988752957	PIRENZEPINE	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.5125748858722557	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.1193356164447602	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
CETP	hgnc:1869	CETP	ChEMBL	33	inhibitor	8.078103267029922	TORCETRAPIB	ncit:C91058	TORCETRAPIB	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	BENZHYDROCODONE HYDROCHLORIDE	rxcui:2122776	BENZHYDROCODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3125456621172291	LEVAMLODIPINE MALEATE	rxcui:2377031	LEVAMLODIPINE MALEATE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
KIF5B	hgnc:6324	KIF5B	ChEMBL	33	inhibitor	6.563458904461812	SELPERCATINIB	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.8178764989983567	PEMIGATINIB	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.2476776945079929	BARNIDIPINE	rxcui:39879	MEPIRODIPINE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	1.250182648468916	AMEDIPLASE	ncit:C169777	AMEDIPLASE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.8334550989792777	DEPATUXIZUMAB	ncit:C95206	DEPATUXIZUMAB	FALSE	TRUE	TRUE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	SASANLIMAB	ncit:C124058	SASANLIMAB	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.6403374540938354	RETIFANLIMAB	rxcui:2632981	RETIFANLIMAB	TRUE	FALSE	FALSE
RBX1	hgnc:9928	RBX1	ChEMBL	33	modulator	1.875273972703375	IBERDOMIDE	ncit:C129048	IBERDOMIDE	FALSE	FALSE	FALSE
FCGRT	hgnc:3621	FCGRT	ChEMBL	33	inhibitor	0.5834185692854945	ROZANOLIXIZUMAB	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.7395446652914718	PEGDINETANIB	ncit:C62791	PEGDINETANIB	FALSE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	agonist	0.036062961	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	agonist	0.03729238	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
TXN	hgnc:12435	TXN	ChEMBL	33	inhibitor	39.38075342677087	PX-12	drugbank:DB05448	PX-12	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	negative modulator	0.1479089330582944	TAS-117	drugbank:DB15054	TAS-117	FALSE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	ChEMBL	33	inhibitor	2.019525817	BIMEKIZUMAB	rxcui:2668041	BIMEKIZUMAB	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.096167896	PERZINFOTEL	ncit:C72122	PERZINFOTEL	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1530835896084387	PERZINFOTEL	ncit:C72122	PERZINFOTEL	FALSE	FALSE	FALSE
RPS8	hgnc:10441	RPS8	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS15	hgnc:10388	RPS15	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS5	hgnc:10426	RPS5	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS4X	hgnc:10424	RPS4X	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS18	hgnc:10401	RPS18	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS7	hgnc:10440	RPS7	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS23	hgnc:10410	RPS23	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL30	hgnc:10333	RPL30	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPLP1	hgnc:10372	RPLP1	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL41	hgnc:10354	RPL41	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL36A	hgnc:10359	RPL36A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL34	hgnc:10340	RPL34	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
PPP5C	hgnc:9322	PPP5C	ChEMBL	33	inhibitor	10.50153425	LB-100	drugbank:DB15412	LB-100	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.1325951293830669	LANIFIBRANOR	ncit:C166556	LANIFIBRANOR	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	SUTEZOLID	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.039068208	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.038894571	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.6403374540938354	APL-501	chembl:CHEMBL4594355	APL-501	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.042174836	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	ISLATRAVIR	ncit:C174896	ISLATRAVIR	FALSE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	inhibitor	1.009762908	ATN-161	drugbank:DB05491	ATN-161	FALSE	FALSE	FALSE
CTSS	hgnc:2545	CTSS	ChEMBL	33	inhibitor	7.001022831425932	PETESICATIB	ncit:C174598	PETESICATIB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
RPS6KA1	hgnc:10430	RPS6KA1	ChEMBL	33	inhibitor	0.8751278539282418	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
OSMR	hgnc:8507	OSMR	ChEMBL	33	inhibitor	52.50767123569449	VIXARELIMAB	ncit:C174929	VIXARELIMAB	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.0701037	E-7090	iuphar.ligand:11414	TASURGRATINIB	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	ChEMBL	33	inhibitor	0.150021918	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
LRP1	hgnc:6692	LRP1	ChEMBL	33	binder	1.029562181092049	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.2476776945079929	CONTELTINIB	ncit:C169863	CONTELTINIB	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	ChEMBL	33	inhibitor	0.6419030713410085	BAY1436032	chembl:CHEMBL4206033	BAY1436032	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	ChEMBL	33	inhibitor	0.01305187	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.086361301	KBP5209	chembl:CHEMBL4650289	KBP5209	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	ChEMBL	33	inhibitor	2.092697042002317	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
RELA	hgnc:9955	RELA	ChEMBL	33	inhibitor	0.3302369260106572	EDASALONEXENT	ncit:C171665	EDASALONEXENT	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	ChEMBL	33	inhibitor	0.043592919	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	cleavage	0.2453629496995069	AMCENESTRANT	ncit:C174915	AMCENESTRANT	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	1.071585127259071	DAREXABAN	ncit:C90973	TANEXABAN	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	0.4861821410712453	EPCORITAMAB	rxcui:2637392	EPCORITAMAB	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.4930297768609811	FIPAMEZOLE	ncit:C65684	FIPAMEZOLE	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	EPCORITAMAB	rxcui:2637392	EPCORITAMAB	TRUE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	EPCORITAMAB	rxcui:2637392	EPCORITAMAB	TRUE	FALSE	FALSE
STING1	hgnc:27962	STING1	ChEMBL	33	agonist	52.50767123569449	ADU-S100	drugbank:DB14722	ADU-S100	FALSE	FALSE	FALSE
CD14	hgnc:1628	CD14	ChEMBL	33	inhibitor	1.193356164447602	VB-201	drugbank:DB15259	VB-201	FALSE	FALSE	FALSE
KCNQ3	hgnc:6297	KCNQ3	ChEMBL	33	potentiator	2.678962818147678	EZOGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.084621549	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
EGR1	hgnc:3238	EGR1	ChEMBL	33	inhibitor	26.25383561784724	BRIVOLIGIDE	ncit:C174783	BRIVOLIGIDE	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.021590325	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
GAS6	hgnc:4168	GAS6	ChEMBL	33	inhibitor	8.751278539282415	BATIRAXCEPT	ncit:C156017	BATIRAXCEPT	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.1221108633388244	TALETRECTINIB	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.037213091	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
NCBIGENE:1014	hgnc:1755	CDH16	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:4815	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
APH1A	hgnc:29509	APH1A	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.9376369863516875	UNII-DRL23N424R	ncit:C116872	OSUGACESTAT	FALSE	FALSE	TRUE
MEK2	hgnc:6842	MAP2K2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1808115400678185	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PARP1	hgnc:270	PARP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.225178995499538	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	COSMIC	4-Sep-20	NULL	1.029066006546944	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.01439355	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1842374429322613	ICP-192	ncit:C178318	GUNAGRATINIB	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.005135727	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	ACTINONIN	drugbank:DB04310	2-[(FORMYL-HYDROXY-AMINO)-METHYL]-HEPTANOIC ACID [1-(2-HYDROXYMETHYL-PYRROLIDINE-1-CARBONYL)-2-METHYL-PROPYL]-AMIDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	NSC-3323	chembl:CHEMBL1270169	CHEMBL:CHEMBL1270169	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1250182648468916	CHLOROTRIANISENE	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.006043701	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	NSC-42384	chembl:CHEMBL1270168	CHEMBL:CHEMBL1270168	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.091159151	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	ALTISSIMACOUMARIN F	chembl:CHEMBL2071528	ALTISSIMACOUMARIN F	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	2.386712328895204	COCHINCHINENIN C	chembl:CHEMBL254649	COCHINCHINENIN C	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.062645859	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.012993732	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.050488145	Rigosertib	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	MEDRYSONE	rxcui:29439	MEDRYSONE	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	1.458546423213736	4,6-DICHLORORESORCINOL	chembl:CHEMBL2332783	CHEMBL:CHEMBL2332783	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	L-750667	iuphar.ligand:978	L-750,667	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004139678	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	GNF-PF-710	chembl:CHEMBL596839	CHEMBL:CHEMBL596839	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	SKF-38393	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.071004288	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.025588534	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PROPANIL	chembl:CHEMBL1222498	PROPANIL	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	7,4'-DIMETHOXYISOFLAVONE	chembl:CHEMBL12658	CHEMBL:CHEMBL12658	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.056622219	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	3-HYDROXYANTHRANILIC ACID	drugbank:DB03644	3-HYDROXYANTHRANILIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	GNF-PF-4798	chembl:CHEMBL584635	CHEMBL:CHEMBL584635	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.1422972120208522	IUPHAR.LIGAND:9812	iuphar.ligand:9812	AZD9567	FALSE	FALSE	FALSE
NCOR2	hgnc:7673	NCOR2	DTC	9/2/20	NULL	0.6731752722524936	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.054020238	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE	iuphar.ligand:5445	N-DOCOSATETRA-7,10,13,16-ENOYLETHANOLAMINE	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.1342907192728759	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	CAULIBUGULONE D	chembl:CHEMBL447876	CAULIBUGULONE D	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CHLOROACETIC ACID	rxcui:2374	CHLOROACETIC ACID	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.2612321952024601	EUPATORIN	chembl:CHEMBL487402	EUPATORIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	1.009762908	LORLATINIB	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	TCMDC-123920	chembl:CHEMBL1606	CHEMBL:CHEMBL1606	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.007979889	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	SNC-80	iuphar.ligand:1611	SNC80	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.1450488155682168	GNF-PF-3467	chembl:CHEMBL601774	CHEMBL:CHEMBL601774	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	ERGOCORNINE	chembl:CHEMBL1385840	ERGOCORNINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	NSC-102042	chembl:CHEMBL273103	CHEMBL:CHEMBL273103	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	QUINOXALINE-2-CARBOXYLIC ACID	chembl:CHEMBL151797	CHEMBL:CHEMBL151797	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.018687904	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.015268296	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	NSC-47924	chembl:CHEMBL1269845	CHEMBL:CHEMBL1269845	FALSE	FALSE	FALSE
BAK1	hgnc:949	BAK1	DTC	9/2/20	NULL	1.250182648468916	KERACYANIN	rxcui:28165	KERACYANIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.043180651	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
HSF1	hgnc:5224	HSF1	DTC	9/2/20	NULL	0.3323270331373069	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.037925367	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PROPANIL	chembl:CHEMBL1222498	PROPANIL	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	4.773424657790408	DIETHYL-2-TETRADECYLMALONATE	chembl:CHEMBL1797712	CHEMBL:CHEMBL1797712	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	TRACAZOLATE	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	CHALCONE	rxcui:2592960	CHALCONE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	GNF-PF-4157	chembl:CHEMBL584905	CHEMBL:CHEMBL584905	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.004486301	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	RS-17053	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.039068208	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	ICI-162846	chembl:CHEMBL1593717	CHEMBL:CHEMBL1593717	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.010620484	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	TCMDC-124059	chembl:CHEMBL530733	CHEMBL:CHEMBL530733	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-125587	chembl:CHEMBL532160	CHEMBL:CHEMBL532160	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	TCMDC-123920	chembl:CHEMBL1606	CHEMBL:CHEMBL1606	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	CANTHARIDIC_ACID	chembl:CHEMBL275516	CANTHARIDIC_ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	METHYLMALONIC ACID	drugbank:DB04183	METHYLMALONIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	STANOZOLOL	rxcui:10032	STANOZOLOL	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.023080295	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	SULFADOXINE	rxcui:10173	SULFADOXINE	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.3571950424196904	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	COUMAPHOS	ncit:C76867	COUMAPHOS	FALSE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.3977853881492006	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	BTCP	chembl:CHEMBL279556	CHEMBL:CHEMBL279556	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.01555322	DEQUALINIUM	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002784371	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.2811655755592744	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665812	chembl:CHEMBL589922	CHEMBL:CHEMBL589922	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.056097939	TANGERETIN	chembl:CHEMBL73930	TANGERETIN	FALSE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.064824285	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	RESACTIN A	chembl:CHEMBL509617	RESACTIN A	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.03233231	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011762471	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.098513454	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW827106X	chembl:CHEMBL188257	GW827106X	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	2-AMINOETHOXYDIPHENYL BORATE	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	DTC	9/2/20	NULL	2.234368988752957	THYMIDINE MONOPHOSPHATE	drugbank:DB01643	THYMIDINE MONOPHOSPHATE	FALSE	FALSE	FALSE
BMX	hgnc:1079	BMX	DTC	9/2/20	NULL	3.000438356325399	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.005722283	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	0.091159151	NAFTOPIDIL	ncit:C72927	NAFTOPIDIL	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	HARMALOL	chembl:CHEMBL129177	HARMALOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	FENAMIC ACID	iuphar.ligand:4182	DIPHENYLAMINE-2-CARBOXYLIC ACID	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.015062442	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.1383601350084176	STEPHOLIDINE	iuphar.ligand:8370	(-)-STEPHOLIDINE	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.022632617	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	1-[2-(TRIFLUOROMETHYL)PHENYL]IMIDAZOLE	iuphar.ligand:4331	TRIM	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.017775109	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	1.500219178	1,3-BIS(3-CHLOROPHENYL)UREA	chembl:CHEMBL1417470	CHEMBL:CHEMBL1417470	FALSE	FALSE	FALSE
NCBIGENE:2741	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	antibody	1.591141552596803	IUPHAR.LIGAND:8998	iuphar.ligand:8998	QUILIZUMAB	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	FEBUXOSTAT	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.0287871	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.002787031	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.001146255	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.2561349816375342	TCMDC-125221	chembl:CHEMBL546649	CHEMBL:CHEMBL546649	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	GNF-PF-3403	chembl:CHEMBL602209	CHEMBL:CHEMBL602209	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.070574827	QUINPIROLE	ncit:C152128	QUINPIROLE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	5-NITROQUINOLINE	chembl:CHEMBL164449	CHEMBL:CHEMBL164449	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	4-METHYLBENZOIC ACID METHYL ESTER	chembl:CHEMBL1480173	4-METHYLBENZOIC ACID METHYL ESTER	FALSE	FALSE	FALSE
DDO	hgnc:2727	DDO	DTC	9/2/20	NULL	17.50255707856483	MALONIC ACID	drugbank:DB02175	MALONIC ACID	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	CCG-63802	iuphar.ligand:8724	CCG-63802	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002059205	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	GNF-PF-3012	chembl:CHEMBL582715	CHEMBL:CHEMBL582715	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1892	iuphar.ligand:1892	BUTAPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008345148	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.040893825	METHYLTESTOSTERONE	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	SCOPOLETIN	chembl:CHEMBL71851	SCOPOLETIN	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1591141552596803	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1041818873724097	ERGOCORNINE	chembl:CHEMBL1385840	ERGOCORNINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006324701	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005574063	OXIDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.033338204	AMITRIPTYLINE HYDROCHLORIDE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
P2RY2	hgnc:8541	P2RY2	ChEMBL	33	agonist	1.312691780892362	DIQUAFOSOL TETRASODIUM	ncit:C65437	DIQUAFOSOL TETRASODIUM	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	SJ000117451	chembl:CHEMBL592123	CHEMBL:CHEMBL592123	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	(+)-TETRAHYDROBERBERINE	chembl:CHEMBL476501	CHEMBL:CHEMBL476501	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.002567612	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.1166837138570989	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	12-METHYL TETRADECANOIC ACID	chembl:CHEMBL495852	CHEMBL:CHEMBL495852	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.099071078	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.1875273972703374	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	DTC	9/2/20	NULL	1.193356164447602	4-METHYLTHIOAMPHETAMINE	chembl:CHEMBL6467	4-METHYLTHIOAMPHETAMINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.1159109740302306	ACEQUINOCYL	chembl:CHEMBL1869353	ACEQUINOCYL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	TCMDC-125221	chembl:CHEMBL546649	CHEMBL:CHEMBL546649	FALSE	FALSE	FALSE
GLA	hgnc:4296	GLA	DTC	9/2/20	NULL	0.2375912725597036	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.057260274	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009081623	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.3302369260106572	NU-2058	chembl:CHEMBL269881	CHEMBL:CHEMBL269881	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.020688602	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.041972559	DIMETHYL FUMARATE	rxcui:1373478	DIMETHYL FUMARATE	TRUE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	0.6250913242344582	SJ000047240	chembl:CHEMBL590706	CHEMBL:CHEMBL590706	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.6482428547616604	CNQX DISODIUM	chembl:CHEMBL1255647	CHEMBL:CHEMBL1255647	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	(S)-PINACIDIL	chembl:CHEMBL251647	(S)-PINACIDIL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	FRAXETIN	chembl:CHEMBL54909	FRAXETIN	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	ACRIDONE	chembl:CHEMBL436589	ACRIDONE	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.074163377	DIAMIDE	chembl:CHEMBL1255835	DIAMIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	DAMNACANTHAL	ncit:C1480	DAMNACANTHAL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	LORECLEZOLE	ncit:C66036	LORECLEZOLE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	CLOBENPROPIT	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.019483366	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	6,7-ADTN HYDROBROMIDE	chembl:CHEMBL1255656	CHEMBL:CHEMBL1255656	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	1.000146118775133	BAS-8770949	chembl:CHEMBL476025	CHEMBL:CHEMBL476025	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.013313304	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	CONICASTEROL B	chembl:CHEMBL1782604	CONICASTEROL B	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	GR-103691	chembl:CHEMBL294747	CHEMBL:CHEMBL294747	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	CAULIBUGULONE B	chembl:CHEMBL508779	CAULIBUGULONE B	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.01214331	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.1643432589536604	M2698	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	PT-101	chembl:CHEMBL316796	CHEMBL:CHEMBL316796	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004128935	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	ALBENDAZOLE	rxcui:430	ALBENDAZOLE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	ANAZOLENE	chembl:CHEMBL1555467	ANAZOLENE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.016161179	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	ARBACLOFEN	ncit:C90890	ARBACLOFEN	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.061340737	13-CIS-RETINAL	iuphar.ligand:6671	13-CIS-RETINAL	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00402481	E-DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	FANCHININ	drugbank:DB14066	TETRANDRINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	UNC0224	chembl:CHEMBL576781	CHEMBL:CHEMBL576781	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	4.375639269641208	6-METHOXYCOMAPARVIN	chembl:CHEMBL401565	CHEMBL:CHEMBL401565	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2180551131050435	ROMIDEPSIN	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.06697407	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	6-DESOXYCODEINE	chembl:CHEMBL408422	CHEMBL:CHEMBL408422	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	GNF-PF-2413	chembl:CHEMBL578515	CHEMBL:CHEMBL578515	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	NSC-98938	chembl:CHEMBL1939691	CHEMBL:CHEMBL1939691	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	DNDI1417264	chembl:CHEMBL1467200	CHEMBL:CHEMBL1467200	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.011188509	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005483257	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003050289	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.1041818873724097	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.040051618	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	5.527123287967842	SULFURIC ACID	rxcui:10231	SULFURIC ACID	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	MERCAPTOPURINE HYDRATE	chembl:CHEMBL1200751	MERCAPTOPURINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	NSC-37642	chembl:CHEMBL1707907	CHEMBL:CHEMBL1707907	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	CITROPTEN	chembl:CHEMBL481049	CITROPTEN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.039479452	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	NCI	14-Sep-17	NULL	0.3281729452230906	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.015344147	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.024932417	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	METHANDROSTENOLONE	rxcui:6818	METHANDROSTENOLONE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.085239726	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.1000146118775133	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	DTC	9/2/20	NULL	6.177373086552294	TORMENTIC ACID METHYL ESTER	chembl:CHEMBL600614	TORMENTIC ACID METHYL ESTER	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	0.2800409132570373	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.3125456621172291	3-HYDROXYANTHRANILIC ACID	drugbank:DB03644	3-HYDROXYANTHRANILIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	ZM-336372	iuphar.ligand:9130	ZM336372	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	inhibitor	0.025739055	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	DIENOCHLOR	chembl:CHEMBL1355965	DIENOCHLOR	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.173866461	MECETRONIUM	ncit:C87264	MECETRONIUM	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	CILOSTAZOL	rxcui:21107	CILOSTAZOL	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.061628722	GW305074X	chembl:CHEMBL1880739	GW305074X	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	BENZYLACETONE	chembl:CHEMBL1490851	BENZYLACETONE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	LINOPIRDINE	ncit:C82306	LINOPIRDINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	DTC	9/2/20	NULL	0.078136416	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.3182283105193605	TH0318	drugbank:DB05145	TH0318	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	GNF-PF-3201	chembl:CHEMBL581872	CHEMBL:CHEMBL581872	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	DTC	9/2/20	NULL	0.080042182	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	RETINYLRETINOATE	chembl:CHEMBL451039	RETINYLRETINOATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.001146255	TCMDC-125488	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	A-77636	iuphar.ligand:9637	A77636	FALSE	FALSE	FALSE
PAK1	hgnc:8590	PAK1	DTC	9/2/20	NULL	0.055859225	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	INDOXACARB	chembl:CHEMBL197676	INDOXACARB	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.027177884	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	ROXINDOLE	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV1.3	hgnc:6221	KCNA3	TTD	2020.06.01	NULL	7.501095891	Dalazatide	ncit:C166962	DALAZATIDE	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.004230396	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002784371	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	DNDI1416982	chembl:CHEMBL1479114	CHEMBL:CHEMBL1479114	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BMS-564929	drugbank:DB07286	BMS-564929	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	MAPROTILINE HYDROCHLORIDE	rxcui:203126	MAPROTILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	METHYLEUGENOL	rxcui:1368373	METHYLEUGENOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003541833	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	SARPOGRELATE	ncit:C73158	SARPOGRELATE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1041818873724097	(E)-2-STYRYLCHROMONE	chembl:CHEMBL388823	CHEMBL:CHEMBL388823	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.006221288	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.1902451856365742	XANTHOHUMOL	ncit:C121950	XANTHOHUMOL	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.6482428547616604	XANTHOHUMOL	ncit:C121950	XANTHOHUMOL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009433646	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002499294	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	2.128689374420047	VESTIPITANT	ncit:C95194	VESTIPITANT	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.008651783	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	0.9376369863516875	NSC-50688	chembl:CHEMBL1456848	CHEMBL:CHEMBL1456848	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.014145386	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.009031247	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	REVERSETRIIODOTHYRONINE	iuphar.ligand:2636	RT3	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2083637747448194	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.1944728564284981	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2187819634820604	3-METHYLCHOLANTHRENE	chembl:CHEMBL40583	3-METHYLCHOLANTHRENE	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR	hgnc:2438	CSF3	TTD	2020.06.01	NULL	8.751278539282415	F-627	rxcui:2670630	EFBEMALENOGRASTIM ALFA	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	GNF-PF-1678	chembl:CHEMBL580340	CHEMBL:CHEMBL580340	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.010418189	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	6,7-ADTN HYDROBROMIDE	chembl:CHEMBL1255656	CHEMBL:CHEMBL1255656	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.035550217	SJ000071854	chembl:CHEMBL602127	CHEMBL:CHEMBL602127	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	DNDI1417607	chembl:CHEMBL1588679	CHEMBL:CHEMBL1588679	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.018962684	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	GNF-PF-4798	chembl:CHEMBL584635	CHEMBL:CHEMBL584635	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	DTC	9/2/20	NULL	0.1411496538593938	5,7-DIHYDROXY-4-METHYLCOUMARIN	chembl:CHEMBL12252	5,7-DIHYDROXY-4-METHYLCOUMARIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	SALICYLALDEHYDE THIOSEMICARBAZONE	chembl:CHEMBL242112	SALICYLALDEHYDE THIOSEMICARBAZONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1146455703836124	1,7-O-DIACETYLGEOPYXIN A	chembl:CHEMBL1873045	CHEMBL:CHEMBL1873045	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	ROBUSTIC ACID	chembl:CHEMBL400777	ROBUSTIC ACID	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.019142425	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.2419708351875322	NSC-119889	chembl:CHEMBL516616	CHEMBL:CHEMBL516616	FALSE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.045265234	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1902451856365742	TRICLOFENOL	chembl:CHEMBL109095	TRICLOFENOL	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:7110	rxcui:279645	ALMOTRIPTAN	TRUE	FALSE	FALSE
SHH	hgnc:10848	SHH	DTC	9/2/20	NULL	26.25383561784724	ROBOTNIKININ	chembl:CHEMBL473392	ROBOTNIKININ	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	IODOFORM	rxcui:27748	IODOFORM	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007592202	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	TDR77585	chembl:CHEMBL1333386	CHEMBL:CHEMBL1333386	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.375054795	NSC-50688	chembl:CHEMBL1456848	CHEMBL:CHEMBL1456848	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	NSC-659162	chembl:CHEMBL471005	CHEMBL:CHEMBL471005	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:3773	iuphar.ligand:3773	[125I]C3A (HUMAN)	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.021258166	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	DTC	9/2/20	NULL	2.625383561784724	REDIOCIDE A	chembl:CHEMBL454246	REDIOCIDE A	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	DTC	9/2/20	NULL	0.1457197166578015	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	SJ000201681	chembl:CHEMBL602135	CHEMBL:CHEMBL602135	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIDECYLDIMETHYLAMMONIUM CHLORIDE	rxcui:1011450	DIDECYLDIMETHYLAMMONIUM CHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	FTI-276	iuphar.ligand:6531	FTI 276	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	FELBAMATE	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
NCBIGENE:1992	hgnc:3311	SERPINB1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8055	drugbank:DB08691	ETHYL 3-[(E)-2-AMINO-1-CYANOETHENYL]-6,7-DICHLORO-1-METHYL-1H-INDOLE-2-CARBOXYLATE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	FRAXIDIN METHYL ETHER	chembl:CHEMBL253551	FRAXIDIN METHYL ETHER	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	ZM-336372	iuphar.ligand:9130	ZM336372	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016018204	LOSARTAN	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.02321294	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.031784305	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.01816246	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	0.5676505	NAPHTHOQUINONE	chembl:CHEMBL55934	NAPHTHOQUINONE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	NSC-119889	chembl:CHEMBL516616	CHEMBL:CHEMBL516616	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	0.6563458904461813	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.5738543304447485	SCUTELLARIN	iuphar.ligand:13075	SCUTELLARIN	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.014103592	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	CHLOROPHENYLPIPERAZINE	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GNF-PF-3257	chembl:CHEMBL601768	CHEMBL:CHEMBL601768	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ISOFENPHOS	ncit:C163668	ISOFENPHOS	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	SIB-1757	iuphar.ligand:1431	SIB-1757	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.017059022	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.065799087	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.086789539	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.1548898856510162	CALANOLIDE A	drugbank:DB04886	CALANOLIDE A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	STIROFOS	chembl:CHEMBL1452359	STIROFOS	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.060353645	HARMALINE	drugbank:DB13875	HARMALINE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.016005996	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.055711057	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.055563673	DNDI1417025	chembl:CHEMBL1320453	CHEMBL:CHEMBL1320453	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	BAS-8770949	chembl:CHEMBL476025	CHEMBL:CHEMBL476025	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.1029562181092049	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	PIRINIXIC ACID	iuphar.ligand:2666	PIRINIXIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	GNF-PF-1731	chembl:CHEMBL581251	CHEMBL:CHEMBL581251	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	ARACHIDONYL TRIFLUOROMETHYLKETONE	iuphar.ligand:5142	ARACHIDONYL TRIFLUOROMETHYL KETONE	FALSE	FALSE	FALSE
NCBIGENE:2444	hgnc:3955	FRK	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:10236	iuphar.ligand:10236	VOLOCIXIMAB	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.05853698	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1274458039701322	DIENOCHLOR	chembl:CHEMBL1355965	DIENOCHLOR	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	NSC-343227	chembl:CHEMBL1329326	CHEMBL:CHEMBL1329326	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.033985548	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	GNF-PF-3501	chembl:CHEMBL581910	CHEMBL:CHEMBL581910	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.015184405	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	1-ETHYLPYRIDINIUM IODIDE	chembl:CHEMBL539954	CHEMBL:CHEMBL539954	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	NSC-8186	chembl:CHEMBL122355	CHEMBL:CHEMBL122355	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.038382801	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	2.763561643983921	APRAMIDE A	chembl:CHEMBL508600	APRAMIDE A	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	PESUDOGINSENOSIDE RP1 METHYL ESTER	chembl:CHEMBL1288831	PESUDOGINSENOSIDE RP1 METHYL ESTER	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.030202859	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	3,4-DIMETHOXYDALBERGIONE	chembl:CHEMBL1591258	3,4-DIMETHOXYDALBERGIONE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.005818669	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003981473	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	GBR-12935	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.021933029	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.027781837	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.016621612	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	PSORALEN	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.016764901	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.100589408	2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE	chembl:CHEMBL1599728	2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.013638356	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P41743	hgnc:9404	PRKCI	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
POLL	hgnc:9184	POLL	DTC	9/2/20	NULL	13.12691780892362	HYMENOIC ACID	chembl:CHEMBL494213	HYMENOIC ACID	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	PIFEXOLE	ncit:C76774	PIFEXOLE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.031032903	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
STK16	hgnc:11394	STK16	DTC	9/2/20	inhibitor	1.312691780892362	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.030004384	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	0.3201687270469177	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2713574740862764	MEPINDOLOL	rxcui:29518	MEPINDOLOL	FALSE	FALSE	FALSE
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 2	hgnc:3093	DYRK2	TTD	2020.06.01	NULL	5.250767124	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	GNF-PF-1399	chembl:CHEMBL578504	CHEMBL:CHEMBL578504	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.9376369863516875	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.1268301237577161	DIACEREIN	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	SJ000201681	chembl:CHEMBL602135	CHEMBL:CHEMBL602135	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	OBTUSAQUINONE	chembl:CHEMBL1333653	OBTUSAQUINONE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.157680694	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	SJ000089001	chembl:CHEMBL591618	CHEMBL:CHEMBL591618	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.042863405	TYRPHOSTIN AG-1478	iuphar.ligand:4862	AG1478	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.04724037	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	INDIGO	rxcui:1426889	INDIGO	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	DICYCLOMINE HYDROCHLORIDE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.001225069	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	S(+)-ISOPROTERENOL-BITARTRATE	chembl:CHEMBL1257092	CHEMBL:CHEMBL1257092	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1060761035064535	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	LAPACHOL	chembl:CHEMBL15193	LAPACHOL	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	LAPACHOL	chembl:CHEMBL15193	LAPACHOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00747866	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	SEW-03621	chembl:CHEMBL1271059	CHEMBL:CHEMBL1271059	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.051731696	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	1.666910197958555	ANACARDIC ACID	iuphar.ligand:6999	ANACARDIC ACID	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.043866058	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	BENANSERIN HYDROCHLORIDE	ncit:C79720	BENANSERIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.061992528	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	NSC-270156	chembl:CHEMBL471226	CHEMBL:CHEMBL471226	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.002394986	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	1.050153425	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.013505059	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	GALUTEOLIN	chembl:CHEMBL233929	GALUTEOLIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004139678	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004427291	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	GNF-PF-5233	chembl:CHEMBL528316	CHEMBL:CHEMBL528316	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	SPIRADOLINE	ncit:C152417	SPIRADOLINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	PAPAVERINE HYDROCHLORIDE	rxcui:203132	PAPAVERINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.1244257612220248	UNC0224	chembl:CHEMBL576781	CHEMBL:CHEMBL576781	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	(-)-PROPANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.007596596	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.006071655	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	SAPPANONE A DIMETHYL ETHER	chembl:CHEMBL1489223	SAPPANONE A DIMETHYL ETHER	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	DTC	9/2/20	NULL	5.250767123569449	PF-04862853	chembl:CHEMBL1915783	CHEMBL:CHEMBL1915783	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.063110182	GW305074X	chembl:CHEMBL1880739	GW305074X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	OXYQUINOLINE SULFATE	rxcui:42836	OXYQUINOLINE SULFATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.042481935	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.028184472	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.2476776945079929	DIHYDRODAPHNODORIN B	chembl:CHEMBL1532097	DIHYDRODAPHNODORIN B	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	BISINDOLYLMALEIMIDE IX	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	PT-101	chembl:CHEMBL316796	CHEMBL:CHEMBL316796	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	TANSHINONE IIA SULFONATE	chembl:CHEMBL1473252	TANSHINONE IIA SULFONATE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.046059361	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CYCLANDELATE	rxcui:2970	CYCLANDELATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	GNF-PF-1399	chembl:CHEMBL578504	CHEMBL:CHEMBL578504	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	DTC	9/2/20	NULL	0.3804903712731485	DIZOCILPINE	ncit:C65450	DIZOCILPINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	NSC-125034	chembl:CHEMBL239439	CHEMBL:CHEMBL239439	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.021370644	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.009905239	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	PIRINIXIC ACID	iuphar.ligand:2666	PIRINIXIC ACID	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	GNF-PF-4325	chembl:CHEMBL598263	CHEMBL:CHEMBL598263	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.4526523382387456	TCMDC-124354	chembl:CHEMBL546344	CHEMBL:CHEMBL546344	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	ALAZANINE	chembl:CHEMBL578063	ALAZANINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	METHYSERGIDE MALEATE	rxcui:203190	METHYSERGIDE MALEATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004252322	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	NSC-125034	chembl:CHEMBL239439	CHEMBL:CHEMBL239439	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	OXOPURPUREINE	chembl:CHEMBL456295	OXOPURPUREINE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	DNDI1417331	chembl:CHEMBL1092508	CHEMBL:CHEMBL1092508	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.1640864726115453	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.015123177	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	TCMDC-124166	chembl:CHEMBL528712	CHEMBL:CHEMBL528712	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	VINCAMINE	rxcui:11201	VINCAMINE	TRUE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	DTC	9/2/20	NULL	3.750547945	BERKELEYACETAL B	chembl:CHEMBL252921	BERKELEYACETAL B	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	CCT018159	chembl:CHEMBL399530	CHEMBL:CHEMBL399530	FALSE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.032858367	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	OLVANIL	ncit:C166774	OLVANIL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	NEPAPRAZOLE	ncit:C84002	NEPAPRAZOLE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	13-CIS-RETINAL	iuphar.ligand:6671	13-CIS-RETINAL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CARBOQUONE	ncit:C342	CARBOQUONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	GNF-PF-1678	chembl:CHEMBL580340	CHEMBL:CHEMBL580340	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	ELIPRODIL	ncit:C80994	ELIPRODIL	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.045579576	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.044198376	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.007867496	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	TRIFLUPROMAZINE HYDROCHLORIDE	rxcui:91125	TRIFLUPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.009087517	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	ZK-159222	iuphar.ligand:2789	ZK159222	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.3671865121377238	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	4.773424657790408	CYCLIC CRYPEVEIC	chembl:CHEMBL1784538	CYCLIC CRYPEVEIC	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0191914	TRYPTOPHAN	rxcui:10898	TRYPTOPHAN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NITRALIN	chembl:CHEMBL1256763	NITRALIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.05664258	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	GBR-12935	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.014601688	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.014634245	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.013299815	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.1325951293830669	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002529881	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.525076712	GNF-PF-3467	chembl:CHEMBL601774	CHEMBL:CHEMBL601774	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.210030685	BENSULIDE	chembl:CHEMBL1895252	BENSULIDE	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.011906501	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.055563673	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ISOBERGAPTENE	chembl:CHEMBL141690	ISOBERGAPTENE	FALSE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	DTC	9/2/20	NULL	2.386712328895204	LY-411575	chembl:CHEMBL392068	CHEMBL:CHEMBL392068	FALSE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	DTC	9/2/20	NULL	1.875273972703375	LY-411575	chembl:CHEMBL392068	CHEMBL:CHEMBL392068	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.025147352	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.2917092846427472	SJ000032159	chembl:CHEMBL591361	CHEMBL:CHEMBL591361	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	inhibitor	0.087512785	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	AZETIDINE-2,4-DICARBOXYLIC ACID	chembl:CHEMBL41680	CHEMBL:CHEMBL41680	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	TRIBROMSALAN	ncit:C47768	TRIBROMSALAN	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	SJ000260177	chembl:CHEMBL592118	CHEMBL:CHEMBL592118	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.06697407	DNDI1417025	chembl:CHEMBL1320453	CHEMBL:CHEMBL1320453	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016780975	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.2051080907644316	7,2'-DIHYDROXYFLAVONE	chembl:CHEMBL475908	CHEMBL:CHEMBL475908	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TCMDC-125756	chembl:CHEMBL536599	CHEMBL:CHEMBL536599	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.007773732	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	3-HYDROXYANTHRANILIC ACID	drugbank:DB03644	3-HYDROXYANTHRANILIC ACID	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.023151531	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	SJ000089001	chembl:CHEMBL591618	CHEMBL:CHEMBL591618	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	DESOXIMETASONE	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	inhibitor	0.021172448	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	N-(4-NITROPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1574420	CHEMBL:CHEMBL1574420	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.040515178	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	MMV007764	chembl:CHEMBL609628	CHEMBL:CHEMBL609628	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	TCMDC-125185	chembl:CHEMBL580819	CHEMBL:CHEMBL580819	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	ALAZANINE	chembl:CHEMBL578063	ALAZANINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	AZETIDINE-2,4-DICARBOXYLIC ACID	chembl:CHEMBL41680	CHEMBL:CHEMBL41680	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	TRIBROMSALAN	ncit:C47768	TRIBROMSALAN	TRUE	FALSE	FALSE
TXN	hgnc:12435	TXN	DTC	9/2/20	NULL	13.12691780892362	GAMBOGENIC ACID	chembl:CHEMBL2205166	GAMBOGENIC ACID	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	IDEBENONE	rxcui:51296	IDEBENONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DIBENZOYLMETHANE	chembl:CHEMBL371523	DIBENZOYLMETHANE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DIHYDREXIDINE HYDROCHLORIDE	chembl:CHEMBL1256832	DIHYDREXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.061701141	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.079798892	SB-222200	iuphar.ligand:2131	SB 222200	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.048708415	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	CIS(Z)-FLUPENTIXOL DIHYDROCHLORIDE	chembl:CHEMBL1496351	CHEMBL:CHEMBL1496351	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003001553	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.029074015	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	DEMETHYL-CANTHARIDIN	chembl:CHEMBL8327	DEMETHYL-CANTHARIDIN	FALSE	FALSE	FALSE
RASGRP1	hgnc:9878	RASGRP1	DTC	9/2/20	NULL	35.00511415712966	BYROSTATIN 1	chembl:CHEMBL223661	BYROSTATIN 1	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.012794267	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	CLOFLUCARBAN	ncit:C47457	CLOFLUCARBAN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	NSC-125034	chembl:CHEMBL239439	CHEMBL:CHEMBL239439	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE	chembl:CHEMBL152028	N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.5966780822238011	CIPROFIBRATE	rxcui:21149	CIPROFIBRATE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.042619863	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	SULFADOXINE	rxcui:10173	SULFADOXINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.2251615404618117	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2775246894064191	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	HALOFANTRINE HYDROCHLORIDE	rxcui:58130	HALOFANTRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	1.050153425	ANETHOLTRITHION	rxcui:820	ANETHOLE TRITHIONE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.5546584989686039	AZD-8055	drugbank:DB12774	AZD-8055	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	METHYSERGIDE MALEATE	rxcui:203190	METHYSERGIDE MALEATE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	VOLVALERENAL D	chembl:CHEMBL1224789	VOLVALERENAL D	FALSE	FALSE	FALSE
MMP12	hgnc:7158	MMP12	DTC	9/2/20	NULL	0.6863747873946994	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.018799739	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GNF-PF-3876	chembl:CHEMBL596631	CHEMBL:CHEMBL596631	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	IPSAPIRONE	ncit:C74391	IPSAPIRONE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.01715937	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.04464938	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.010594768	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	NAFTOPIDIL	ncit:C72927	NAFTOPIDIL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.001373252	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1033615575505797	(S)-THIORPHAN	drugbank:DB08626	THIORPHAN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	ETHACRIDINE LACTATE	rxcui:4107	ETHACRIDINE LACTATE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	GNF-PF-3149	chembl:CHEMBL582507	CHEMBL:CHEMBL582507	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	DIHYDREXIDINE HYDROCHLORIDE	chembl:CHEMBL1256832	DIHYDREXIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.012360563	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CINOBUFOTALIN	ncit:C151929	CINOBUFOTALIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.033985548	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010569177	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	(R)-DIHYDRONIPHATENONE B	chembl:CHEMBL1946449	CHEMBL:CHEMBL1946449	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.020383413	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CARBETAPENTANE	rxcui:20217	CARBETAPENTANE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.01823183	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.021933029	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.055563673	PIFEXOLE	ncit:C76774	PIFEXOLE	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	DTC	9/2/20	NULL	0.1891032577516008	KETAMINE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.007184958	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-125236	chembl:CHEMBL548469	CHEMBL:CHEMBL548469	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2365210416022274	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	TCMDC-124317	chembl:CHEMBL586937	CHEMBL:CHEMBL586937	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	TCMDC-123653	chembl:CHEMBL548540	CHEMBL:CHEMBL548540	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	DNDI1417413	chembl:CHEMBL1343568	CHEMBL:CHEMBL1343568	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.9546849315580818	(R)-IBUPROPHEN	chembl:CHEMBL427526	(R)-IBUPROPHEN	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	DTC	9/2/20	NULL	0.1470803115845784	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	DTC	9/2/20	NULL	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006193403	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	SB-200646	chembl:CHEMBL85194	CHEMBL:CHEMBL85194	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	CONICASTEROL B	chembl:CHEMBL1782604	CONICASTEROL B	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01823183	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	METRAZOLINE OXALATE	chembl:CHEMBL1255866	METRAZOLINE OXALATE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	2-PHENYL-1H-INDOLE	chembl:CHEMBL75756	2-PHENYL-1H-INDOLE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	5-FLUOROURIDINE	drugbank:DB01629	5-FLUOROURIDINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	NELFINAVIR MESYLATE	rxcui:266565	NELFINAVIR MESYLATE	TRUE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.7955707762984014	8-BROMO-CAMP SODIUM	chembl:CHEMBL1256796	CHEMBL:CHEMBL1256796	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	2-ETHYLANTHRAQUINONE	chembl:CHEMBL42355	CHEMBL:CHEMBL42355	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.041672755	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.7721716358190367	DNDI1417629	chembl:CHEMBL1731432	CHEMBL:CHEMBL1731432	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	NSC-102042	chembl:CHEMBL273103	CHEMBL:CHEMBL273103	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	7-HYDROXY ISOFLAVONE	chembl:CHEMBL491981	7-HYDROXY ISOFLAVONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002018051	IRINOTECAN HYDROCHLORIDE	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.012710644	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01150727	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.050007306	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	SAPPANONE A DIMETHYL ETHER	chembl:CHEMBL1489223	SAPPANONE A DIMETHYL ETHER	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001990963	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.019339842	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1396480617970598	HARMALOL	chembl:CHEMBL129177	HARMALOL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.041672755	NSC-8186	chembl:CHEMBL122355	CHEMBL:CHEMBL122355	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002356506	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	inhibitor	0.013817808	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.008230043	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.2344092465879218	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.019687916	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
ENPP2	hgnc:3357	ENPP2	DTC	9/2/20	NULL	8.751278539282415	(S)-CARBA CYCLIC-PHOSPHATIDIC ACID	chembl:CHEMBL1630084	CHEMBL:CHEMBL1630084	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.056157937	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	VER-3323	iuphar.ligand:168	VER-3323	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.008401227	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005208578	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	MONOBENZONE	rxcui:17145	MONOBENZONE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.002801007	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	AMPEROZIDE HYDROCHLORIDE	ncit:C77259	AMPEROZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.039068208	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000759374	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.031032903	3,4-METHYLENEDIOXYB-NITROSTYRENE	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	A-70108	iuphar.ligand:6077	A68930	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.2917092846427472	TANGERETIN	chembl:CHEMBL73930	TANGERETIN	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.210030685	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	7-METHOXY-BAPTIGENIN	chembl:CHEMBL583578	CHEMBL:CHEMBL583578	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.375054795	4,4'-THIODIANILINE	chembl:CHEMBL348856	4,4'-THIODIANILINE	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.0095957	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.2465148884304905	NALMEFENE	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ISOFLUPREDONE ACETATE	rxcui:1364586	ISOFLUPREDONE ACETATE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.023524942	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	DTC	9/2/20	NULL	0.1187956362798518	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	DTC	9/2/20	NULL	0.1103102336884338	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	BENZPIPERYLON	ncit:C83547	BENZPIPERYLON	FALSE	FALSE	FALSE
MATK	hgnc:6906	MATK	DTC	9/2/20	NULL	0.06466462	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.1029562181092049	TCMDC-124022	chembl:CHEMBL548017	CHEMBL:CHEMBL548017	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	BEMESETRON	ncit:C80766	BEMESETRON	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	DTC	9/2/20	NULL	0.087537101	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	O-NITROANISOLE	chembl:CHEMBL166415	2-NITROANISOLE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001120833	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.8751278539282416	BENZO[DEF]CHRYSENE	chembl:CHEMBL31184	BENZO[DEF]CHRYSENE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002681699	E-DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.007329379	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	TRICLOFENOL	chembl:CHEMBL109095	TRICLOFENOL	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.2237542808339254	CELIPROLOL	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	DTC	9/2/20	NULL	2.917092846427472	PD-117915	chembl:CHEMBL303124	CHEMBL:CHEMBL303124	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	2.838252499226729	[18F]FLUORORASAGILINE	chembl:CHEMBL2023193	[18F]FLUORORASAGILINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PROADIFEN	ncit:C84107	PROADIFEN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	MAPROTILINE HYDROCHLORIDE	rxcui:203126	MAPROTILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	DEXPROPRANOLOL	ncit:C77944	DEXPROPRANOLOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.018641225	Amphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	3-MORPHOLINOSYDNONIMINE HCL	chembl:CHEMBL538104	CHEMBL:CHEMBL538104	FALSE	FALSE	FALSE
NUDT15	hgnc:23063	NUDT15	FDA	10-Apr-24	NULL	0.6908904109959803	Azathioprine	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	2.080014029626545	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	1.050153425	Sodium Ascorbate	rxcui:267366	SODIUM ASCORBATE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.095468493	Ceftriaxone	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.04427291	Donepezil	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	FDA	10-Apr-24	NULL	1.346350544504987	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.018081154	Esomeprazole	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
F5	hgnc:3542	F5	FDA	10-Apr-24	NULL	0.1474934585272317	Eltrombopag	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.06886252	Eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.006811217	Fluvoxamine	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	2.100306849	Pegloticase	rxcui:1011650	PEGLOTICASE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	0.065634589	Peginterferon Alfa-2b	rxcui:253453	PEGINTERFERON ALFA-2B	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.011068227	Propranolol	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.081030357	Siponimod	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.003689409	Tramadol	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	MyCancerGenome	20-Jun-17	inhibitor	0.4565884455277782	TSR-011	ncit:C114287	ALK/TRK INHIBITOR TSR-011	FALSE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	MyCancerGenome	20-Jun-17	inhibitor	0.2500365296937833	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.3454452054979901	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.2778183663264259	MEHD7945A	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1848861663228679	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
CTLA4	hgnc:2505	CTLA4	MyCancerGenome	20-Jun-17	immunotherapy	0.9723642821424907	TREMELIMUMAB	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
CTLA4	hgnc:2505	CTLA4	MyCancerGenome	20-Jun-17	antibody	0.9723642821424907	TREMELIMUMAB	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MS4A1	hgnc:7315	MS4A1	MyCancerGenome	20-Jun-17	antibody	0.3025133322221082	RITUXIMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
PIGF	hgnc:8962	PIGF	MyCancerGenome	20-Jun-17	antibody	21.00306849	ZIV-AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
HGF	hgnc:4893	HGF	MyCancerGenome	20-Jun-17	antibody	9.723642821424907	FICLATUZUMAB	ncit:C78844	FICLATUZUMAB	FALSE	TRUE	TRUE
VEGFB	hgnc:12681	VEGFB	MyCancerGenome	20-Jun-17	antibody	7.001022831425934	ZIV-AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
HSP90AA2	hgnc:5256	HSP90AA2P	MyCancerGenome	20-Jun-17	other/unknown	0.8751278539282416	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	MyCancerGenome	20-Jun-17	other/unknown	0.3319450480417468	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	2.080014029626545	1032900-25-6	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.043866058	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.003768854	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.020257589	IDARUBICINE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.030202859	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.047626006	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.08572681	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1565057264849314	BUTHIONINE SULFOXIMINE	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.027326397	CPT-11	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.032817295	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ADM	hgnc:259	ADM	NCI	14-Sep-17	NULL	0.3281729452230906	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
ADK	hgnc:257	ADK	NCI	14-Sep-17	NULL	0.6563458904461812	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
ALPL	hgnc:438	ALPL	NCI	14-Sep-17	NULL	0.021773863	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	4.565884455277782	GENERIC	ncit:C1312	GENERIC DRUG	FALSE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.3804903712731485	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.6731752722524935	CHOLESTYRAMINE	rxcui:2447	CHOLESTYRAMINE RESIN	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.4667348554283955	FLT3 LIGAND	ncit:C1714	RECOMBINANT FLT3 LIGAND	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.2800409132570373	PROCARBAZINE	rxcui:8702	PROCARBAZINE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1555782851427985	VIOXX	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.2000292237550266	SULFORAPHANE	ncit:C1424	SULFORAPHANE	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.3842024724563012	HYPERBARIC OXYGEN	ncit:C2351	HYPERBARIC OXYGEN	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	1.280674908	EPISIALIN	ncit:C2407	MUC-1 ANTIGEN	FALSE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.4375639269641208	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.2059124362184098	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.1041818873724097	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
CCL7	hgnc:10634	CCL7	NCI	14-Sep-17	NULL	0.8537832721251138	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	0.5000730593875666	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	0.2573905452730122	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
CD44	hgnc:1681	CD44	NCI	14-Sep-17	NULL	0.2403097081725148	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	4.375639269641208	SGN-14	ncit:C2005	MONOCLONAL ANTIBODY SGN-14	FALSE	FALSE	FALSE
CDA	hgnc:1712	CDA	NCI	14-Sep-17	NULL	11.25164383622025	TETRAHYDROURIDINE	ncit:C868	TETRAHYDROURIDINE	FALSE	FALSE	FALSE
CD86	hgnc:1705	CD86	NCI	14-Sep-17	NULL	0.6482428547616605	ANTIHISTAMINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.075768645	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.8468979231563628	SODIUM SALICYLATE	rxcui:9907	SODIUM SALICYLATE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.043756393	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.3500511415712966	SODIUM SALICYLATE	rxcui:9907	SODIUM SALICYLATE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.053854022	NAVELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.098513454	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.4039051633514962	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.1666910197958555	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.3633748874442526	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
CTSC	hgnc:2528	CTSC	NCI	14-Sep-17	NULL	0.2542744369767288	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.003001553	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.1230648544586589	EFAVIRENZ	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	0.4487835148349957	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.042107194	PS-341	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
EIF2AK2	hgnc:9437	EIF2AK2	NCI	14-Sep-17	NULL	2.187819634820604	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.2302968036653267	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.2201579506737715	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.079557078	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	NCI	14-Sep-17	NULL	0.0701037	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.1669560293662782	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
FGR	hgnc:3697	FGR	NCI	14-Sep-17	NULL	0.192335792	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.4054646427466756	LYMPHOKINES	ncit:C621	RECOMBINANT LYMPHOKINE	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.069225671	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.069454592	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	NCI	14-Sep-17	NULL	0.7778914257139926	DIHYDROTESTOSTERONE	ncit:C29619	DIHYDROTESTOSTERONE	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	NCI	14-Sep-17	NULL	0.094864808	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.2210849315187136	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.037505479	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.1553481397505754	OXYTOCIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
GDF15	hgnc:30142	GDF15	NCI	14-Sep-17	NULL	0.4412409347537353	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	3.889457128569962	4-IPOMEANOL	ncit:C976	IPOMEANOL	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.078136416	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.042379073	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
GYPA	hgnc:4702	GYPA	NCI	14-Sep-17	NULL	1.250182648468916	ANTHRACYCLINES	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
GYPA	hgnc:4702	GYPA	NCI	14-Sep-17	NULL	2.500365296937833	ETHER	ncit:C29819	ETHER	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	NCI	14-Sep-17	NULL	0.1448487482363986	HYPERBARIC OXYGEN	ncit:C2351	HYPERBARIC OXYGEN	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.1389091831632129	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	NCI	14-Sep-17	NULL	0.2302968036653267	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
HMOX2	hgnc:5014	HMOX2	NCI	14-Sep-17	NULL	1.000146118775133	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.1151484018326633	ANTHRACYCLINES	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
HP	hgnc:5141	HP	NCI	14-Sep-17	NULL	7.501095891	HEPATITIS B VACCINE	ncit:C29091	HEPATITIS B VACCINE	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.6105543166941221	SODIUM SALICYLATE	rxcui:9907	SODIUM SALICYLATE	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.04573839	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	NCI	14-Sep-17	NULL	0.1508841127462485	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.9376369863516875	5&APOS;-DEOXY-5-FLUOROURIDINE	ncit:C978	DOXIFLURIDINE	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	NCI	14-Sep-17	NULL	0.039628431	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	0.2155487324946408	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.2386712328895204	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.7721716358190367	ACNU	ncit:C693	NIMUSTINE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.034900413	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.024932417	ANTIDEPRESSANTS	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.049864835	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
LPO	hgnc:6678	LPO	NCI	14-Sep-17	NULL	2.625383561784724	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.1715936968486748	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.079197091	OXYTOCIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.7955707762984014	ACNU	ncit:C693	NIMUSTINE	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.151537291	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	3.500511415712966	CANCER VACCINES	ncit:C1663	ANTINEOPLASTIC VACCINE	FALSE	FALSE	FALSE
MST1	hgnc:7380	MST1	NCI	14-Sep-17	NULL	1.154014752432846	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1842374429322614	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.2692701089009974	PYRAZINAMIDE	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
MYO9B	hgnc:7609	MYO9B	NCI	14-Sep-17	NULL	0.3125456621172291	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.004842988	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
NME2	hgnc:7850	NME2	NCI	14-Sep-17	NULL	0.3559842117674203	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.056888051	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1232574442152452	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.4861821410712453	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2958178661165888	GINKGO BILOBA	rxcui:236809	GINKGO BILOBA EXTRACT	TRUE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.315361389	CONJUGATED ESTROGENS	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.1271372184883644	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NR4A3	hgnc:7982	NR4A3	NCI	14-Sep-17	NULL	3.182283105193606	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.049256727	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
PDYN	hgnc:8820	PDYN	NCI	14-Sep-17	NULL	1.141471113819445	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
PHEX	hgnc:8918	PHEX	NCI	14-Sep-17	NULL	2.333674277141977	RECOMBINANT HUMAN GROWTH HORMONE	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.092606122	CHEMOPREVENTIVE	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.073540156	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.044878351	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.2083637747448194	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1458546423213736	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.091159151	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1620607136904151	SELECTIVE ESTROGEN RECEPTOR MODULATOR	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
PTPRZ1	hgnc:9685	PTPRZ1	NCI	14-Sep-17	NULL	0.384671584	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SCG5	hgnc:10816	SCG5	NCI	14-Sep-17	NULL	3.889457128569963	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	NCI	14-Sep-17	NULL	2.625383561784724	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.057700738	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SLC29A1	hgnc:11003	SLC29A1	NCI	14-Sep-17	NULL	0.2224901323546377	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.2130128650535274	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.2011788169949981	FUROSEMIDE	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	NCI	14-Sep-17	NULL	0.1091635576625665	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
TBP	hgnc:11588	TBP	NCI	14-Sep-17	NULL	0.384671584	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.2302968036653267	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1112450661773188	13-CIS-RETINOIC ACID	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.053937002	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.4449802647092754	KEYHOLE LIMPET HEMOCYANIN	ncit:C1139	KEYHOLE LIMPET HEMOCYANIN	FALSE	FALSE	FALSE
THRSP	hgnc:11800	THRSP	NCI	14-Sep-17	NULL	1.250182648468916	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.2822993077187876	LACTULOSE	rxcui:6218	LACTULOSE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.053253216	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
TNFRSF1A	hgnc:11916	TNFRSF1A	NCI	14-Sep-17	NULL	0.4268916360625569	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	0.1779921058837101	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	5.250767123569449	EO9	ncit:C1087	APAZIQUONE	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.7447896629176524	ANTIFOLATES	ncit:C511	FOLATE ANTAGONIST	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.1105424657593568	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.010617262	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.055740628	PSC-833	ncit:C1405	VALSPODAR	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	NCI	14-Sep-17	NULL	0.1495945049449986	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.5048814541893701	CC-1088	ncit:C2210	SELECTIVE CYTOKINE INHIBITORY DRUG CC-1088	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	6.058577450272442	benzene	rxcui:1311295	BENZENE	FALSE	FALSE	FALSE
CDA	hgnc:1712	CDA	PharmGKB	4/5/24	NULL	0.1648592503475494	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NCAM1	hgnc:7656	NCAM1	PharmGKB	4/5/24	NULL	1.009762908	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
REN	hgnc:9958	REN	PharmGKB	4/5/24	NULL	0.2282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.6168664383892681	neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.011710007	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	1.505278939303214	sparteine	ncit:C152414	SPARTEINE	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.182318303	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	PharmGKB	4/5/24	NULL	0.039479452	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.364636606	trabectedin	rxcui:1716278	TRABECTEDIN	TRUE	FALSE	TRUE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	0.1474934585272317	eltrombopag	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.019577804	felbamate	rxcui:24812	FELBAMATE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.3281729452230906	eltrombopag	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.1881995384791917	adefovir dipivoxil	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.022583945	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.06638138	cyproterone	rxcui:3014	CYPROTERONE	TRUE	FALSE	FALSE
LEPR	hgnc:6554	LEPR	PharmGKB	4/5/24	NULL	0.3070624048871023	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.011196859	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.016023092	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.006195595	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.051629962	artemisinin	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1858678627812194	etonogestrel	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.01787191	troglitazone	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.009349657	hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.006945459	primidone	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.07596596	flurbiprofen	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
MT1A	hgnc:7393	MT1A	PharmGKB	4/5/24	NULL	2.019525816757481	arsenic trioxide	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.009349657	mitomycin	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.2051080907644316	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
RYR2	hgnc:10484	RYR2	PharmGKB	4/5/24	NULL	1.909369863116163	cerivastatin	rxcui:596723	CERIVASTATIN	FALSE	FALSE	FALSE
TEX10	hgnc:25988	TEX10	PharmGKB	4/5/24	NULL	4.039051633514962	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
INVS	hgnc:17870	INVS	PharmGKB	4/5/24	NULL	4.039051633514962	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KMT2E	hgnc:18541	KMT2E	PharmGKB	4/5/24	NULL	4.039051633514962	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.6087845940370378	cerivastatin	rxcui:596723	CERIVASTATIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.01036472	clarithromycin	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.069454592	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MIR1264	hgnc:35246	MIR1264	PharmGKB	4/5/24	NULL	0.3454452054979901	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.002669701	cabazitaxel	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.068637479	clarithromycin	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.9376369863516874	rasagiline	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	PharmGKB	4/5/24	NULL	0.060772768	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
RUNX1	hgnc:10471	RUNX1	PharmGKB	4/5/24	NULL	0.5000730593875666	methacholine chloride	rxcui:40165	METHACHOLINE CHLORIDE	TRUE	FALSE	FALSE
AOC1	hgnc:80	AOC1	PharmGKB	4/5/24	NULL	0.2651902587661338	cannabidiol	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.059297201	rasagiline	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.02550154	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CSK	hgnc:2444	CSK	PharmGKB	4/5/24	NULL	0.760980743	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	PharmGKB	4/5/24	NULL	0.3509871071904712	rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
CCR5	hgnc:1606	CCR5	PharmGKB	4/5/24	NULL	3.938075342677087	maraviroc	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.2625383561784725	sulfisoxazole	rxcui:10207	SULFISOXAZOLE	TRUE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.2692701089009974	chloroprocaine	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.008481291	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.068115956	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	PharmGKB	4/5/24	NULL	0.030688294	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	PharmGKB	4/5/24	NULL	0.033903258	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.003001553	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.001990963	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	0.1977690065374557	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.019776901	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NUP62	hgnc:8066	NUP62	PharmGKB	4/5/24	NULL	0.5933070196123672	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.1483267549030917	torasemide	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	0.4773424657790409	cysteamine	rxcui:1426886	CYSTEAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:O43653	hgnc:9500	PSCA	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	AGS-PSCA	chembl:CHEMBL2109548	MK-4721	FALSE	FALSE	FALSE
SULT1C3	hgnc:33543	SULT1C3	PharmGKB	4/5/24	NULL	7.001022831425933	candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
ANKK1	hgnc:21027	ANKK1	PharmGKB	4/5/24	NULL	0.2631963470460877	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
SLC29A2	hgnc:11004	SLC29A2	PharmGKB	4/5/24	NULL	0.2258394461750301	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	13.43946347104085	halothane	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
NOX3	hgnc:7890	NOX3	PharmGKB	4/5/24	NULL	2.187819634820604	levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
GSTA2	hgnc:4627	GSTA2	PharmGKB	4/5/24	NULL	0.2333674277141977	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCB11	hgnc:42	ABCB11	PharmGKB	4/5/24	NULL	0.063645662	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.105015342	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GPR83	hgnc:4523	GPR83	PharmGKB	4/5/24	NULL	1.141471113819445	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	0.081597003	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	1.419126249613364	MRE-0094	chembl:CHEMBL1950553	SONEDENOSON	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	PharmGKB	4/5/24	NULL	0.092118721	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.138178082	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011746683	pitavastatin	rxcui:861634	PITAVASTATIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011746683	artemether	rxcui:18343	ARTEMETHER	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004195244	mifepristone	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004517955	hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.002258977	oxazepam	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003174779	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
C18ORF56	hgnc:29553	TYMSOS	PharmGKB	4/5/24	NULL	0.1628144844517658	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.001030411	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	4.375639269641208	hydralazine / isosorbide dinitrate	wikidata:Q48566743	HYDRALAZINE / ISOSORBIDE DINITRATE	FALSE	FALSE	FALSE
EHF	hgnc:3246	EHF	PharmGKB	4/5/24	NULL	3.387591692625451	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.2044691247495891	fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
EPM2AIP1	hgnc:19735	EPM2AIP1	PharmGKB	4/5/24	NULL	10.50153425	procarbazine	rxcui:8702	PROCARBAZINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.525076712	lidocaine and tetracaine	drugsatfda.nda:021717	DRUGSATFDA.NDA:021717	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	PharmGKB	4/5/24	NULL	0.043866058	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPK12	hgnc:6874	MAPK12	PharmGKB	4/5/24	NULL	0.034118045	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	1.117184494376478	raltitrexed	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.2453629496995069	BMS-695735	chembl:CHEMBL459729	CHEMBL:CHEMBL459729	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	PharmGKB	4/5/24	NULL	0.018062494	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GALNS	hgnc:4122	GALNS	PharmGKB	4/5/24	NULL	105.0153424713889	elosulfase alfa	rxcui:1489914	ELOSULFASE ALFA	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.9211872146613068	penicillin g	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
MAPK6	hgnc:6879	MAPK6	PharmGKB	4/5/24	NULL	0.9211872146613069	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.053145416	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
LTC4S	hgnc:6719	LTC4S	PharmGKB	4/5/24	NULL	0.7955707762984016	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.053038052	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.1268301237577161	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
ADGRG7	hgnc:19241	ADGRG7	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	CIViC	10-Apr-24	NULL	0.4930297768609811	ARQ092	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
ZMIZ1	hgnc:16493	ZMIZ1	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
MAN1A1	hgnc:6821	MAN1A1	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	PharmGKB	4/5/24	NULL	0.014622019	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.020257589	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.041888848	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
CDSN	hgnc:1802	CDSN	PharmGKB	4/5/24	NULL	0.2822993077187876	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1988926940746003	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	PharmGKB	4/5/24	NULL	0.070322774	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.1442518440541057	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.1372749574789398	tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
CXCL8	hgnc:6025	CXCL8	PharmGKB	4/5/24	NULL	0.4321619031744402	ranibizumab	rxcui:595060	RANIBIZUMAB	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	3.500511415712966	deleobuvir	ncit:C166826	DELEOBUVIR	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	PharmGKB	4/5/24	NULL	0.058602312	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
ZSCAN25	hgnc:21961	ZSCAN25	PharmGKB	4/5/24	NULL	2.812910959055062	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
ABI1	hgnc:11320	ABI1	PharmGKB	4/5/24	NULL	0.525076712	ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.051327147	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.7032277397637656	Antihypertensives	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
BRINP3	hgnc:22393	BRINP3	PharmGKB	4/5/24	NULL	35.00511415712966	uric acid	rxcui:1427088	URIC ACID	FALSE	FALSE	FALSE
PTPRD	hgnc:9668	PTPRD	PharmGKB	4/5/24	NULL	1.640864726115453	Antihypertensives	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.007001023	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TBC1D1	hgnc:11578	TBC1D1	PharmGKB	4/5/24	NULL	0.6908904109959803	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	PharmGKB	4/5/24	NULL	0.09869863	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.3182283105193606	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
TMEM8A	hgnc:17205	PGAP6	PharmGKB	4/5/24	NULL	8.751278539282415	remifentanil	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.1201548540862574	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
LUC7L2	hgnc:21608	LUC7L2	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
ALR	hgnc:380	AKR1A1	ChEMBL	33	inhibitor	6.563458904461812	CYCLOSERINE	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
UBASH3B	hgnc:29884	UBASH3B	PharmGKB	4/5/24	NULL	1.129197231	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SLC22A7	hgnc:10971	SLC22A7	PharmGKB	4/5/24	NULL	0.192335792	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.3182283105193606	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
AKR1C3	hgnc:386	AKR1C3	PharmGKB	4/5/24	NULL	1.750255707856483	Antiandrogens	ncit:C242	ANTI-ANDROGEN	FALSE	FALSE	FALSE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.192335792	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.043109746	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.096167896	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	PharmGKB	4/5/24	NULL	0.020575106	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CCT3	hgnc:1616	CCT3	PharmGKB	4/5/24	NULL	17.50255707856483	ranibizumab	rxcui:595060	RANIBIZUMAB	TRUE	FALSE	FALSE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.077789143	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CBR1	hgnc:1548	CBR1	PharmGKB	4/5/24	NULL	0.2917092846427472	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PPP1R13L	hgnc:18838	PPP1R13L	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.7343730242754476	granisetron	rxcui:26237	GRANISETRON	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.079557078	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1312691780892362	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	PharmGKB	4/5/24	NULL	0.1919140030544389	entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
FTO	hgnc:24678	FTO	PharmGKB	4/5/24	NULL	0.9376369863516874	interferon alfa-2b, recombinant	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
P2RY12	hgnc:18124	P2RY12	PharmGKB	4/5/24	NULL	4.375639269641208	cangrelor	rxcui:1656052	CANGRELOR	TRUE	FALSE	FALSE
SNORD68	hgnc:32729	SNORD68	PharmGKB	4/5/24	NULL	0.6326225450083675	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
POMT2	hgnc:19743	POMT2	PharmGKB	4/5/24	NULL	35.00511415712966	dichloroacetic acid	rxcui:155021	DICHLOROACETIC ACID	TRUE	FALSE	FALSE
SULT1C4	hgnc:11457	SULT1C4	PharmGKB	4/5/24	NULL	0.6326225450083675	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	PharmGKB	4/5/24	NULL	0.024808727	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	TALC	12-May-16	inhibitor	2.080014029626545	LDK378	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.6783936852156912	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.4167275494896388	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
ANPEP	hgnc:500	ANPEP	TALC	12-May-16	inhibitor	0.077217164	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.3571950424196904	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.157680694	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.2128689374420047	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	TALC	12-May-16	inhibitor	0.2263261691193728	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	0.5000730593875666	MK2461	ncit:C90591	C-MET INHIBITOR MK2461	FALSE	FALSE	TRUE
MMP9	hgnc:7176	MMP9	TALC	12-May-16	vaccine	1.050153425	S-3304	drugbank:DB12149	S-3304	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	TALC	12-May-16	inhibitor	0.1848861663228679	NVP-BGT226	ncit:C74073	PI3K INHIBITOR BGT226	FALSE	FALSE	TRUE
RPTOR	hgnc:30287	RPTOR	TALC	12-May-16	inhibitor	0.057574201	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TGFB2	hgnc:11768	TGFB2	TALC	12-May-16	vaccine	15.00219178	BELAGENPUMATUCEL-L	ncit:C73438	BELAGENPUMATUCEL-L	FALSE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	TALC	12-May-16	NULL	0.4667348554283955	BEXAROTENE	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	HALETHAZOLE	ncit:C65837	HALETHAZOLE	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	TALC	12-May-16	antibody	7.501095891	CVX-045	ncit:C82384	TSP-1 MIMETIC FUSION PROTEIN CVX-045	FALSE	FALSE	TRUE
ACVR2A	hgnc:173	ACVR2A	TALC	12-May-16	NULL	17.50255707856483	SOTATERCEPT	ncit:C80038	SOTATERCEPT	FALSE	FALSE	TRUE
UNIPROT:Q9NRA0	hgnc:18859	SPHK2	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	ABC294640	ncit:C98278	OPAGANIB	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.375054795	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.081030357	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:Q96KS0	hgnc:14660	EGLN2	TdgClinicalTrial	Jan-14	NULL	4.200613698855561	AKB-6548	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.09814518	BAZEDOXIFENE	rxcui:1441386	BAZEDOXIFENE	TRUE	FALSE	FALSE
UNIPROT:P25942	hgnc:11919	CD40	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	BPX-101	ncit:C82361	AUTOLOGOUS PROSTATE CANCER ANTIGEN-EXPRESSING DENDRITIC CELL VACCINE BPX-101	FALSE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	CANGRELOR	rxcui:1656052	CANGRELOR	TRUE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TdgClinicalTrial	Jan-14	NULL	0.1182605208011137	OMEPRAZOL	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	CHF 4227	drugbank:DB05882	CHF 4227	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	CHF 4227	drugbank:DB05882	CHF 4227	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.043502627	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q9HBE5	hgnc:6006	IL21R	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	DENENICOKIN	ncit:C62492	DENENICOKIN	FALSE	FALSE	FALSE
UNIPROT:P08238	hgnc:5258	HSP90AB1	TdgClinicalTrial	Jan-14	NULL	0.5707355569097228	DEBIO 0932	ncit:C92572	HSP90 INHIBITOR DEBIO 0932	FALSE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.1691068316769549	METHYLPHENIDATE	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:Q12879	hgnc:4585	GRIN2A	TdgClinicalTrial	Jan-14	NULL	0.1268301237577161	DEXANABINOL	ncit:C99381	DEXANABINOL	FALSE	FALSE	FALSE
UNIPROT:P32238	hgnc:1570	CCKAR	TdgClinicalTrial	Jan-14	NULL	7.876150685354174	DEXLOXIGLUMIDE	ncit:C96871	DEXLOXIGLUMIDE	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.1411496538593938	DERSALAZINE	ncit:C77949	DERSALAZINE	FALSE	FALSE	FALSE
UNIPROT:P15509	hgnc:2435	CSF2RA	TdgClinicalTrial	Jan-14	NULL	0.729273212	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.08178765	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.036463661	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.082171629	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.072927321	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.07458476	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:Q9NQ25	hgnc:21394	SLAMF7	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	ELOTUZUMAB	rxcui:1726104	ELOTUZUMAB	TRUE	FALSE	FALSE
UNIPROT:Q08493	hgnc:8782	PDE4C	TdgClinicalTrial	Jan-14	NULL	0.1131630845596864	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.040814358	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.317586721	EPINASTINE	rxcui:39684	EPINASTINE	TRUE	FALSE	FALSE
UNIPROT:P08514	hgnc:6138	ITGA2B	TdgClinicalTrial	Jan-14	NULL	3.500511415712967	EPTIFIBATIDE	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.04182212	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P22732	hgnc:11010	SLC2A5	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:P01148	hgnc:4419	GNRH1	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	GNRH PHARMACCINE	drugbank:DB05815	GNRH PHARMACCINE	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.06697407	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
UNIPROT:Q96BI3	hgnc:29509	APH1A	TdgClinicalTrial	Jan-14	NULL	0.5357925636295356	GSI-136	drugbank:DB12819	GSI-136	FALSE	FALSE	FALSE
UNIPROT:P49810	hgnc:9509	PSEN2	TdgClinicalTrial	Jan-14	NULL	0.6819178082557726	GSI-136	drugbank:DB12819	GSI-136	FALSE	FALSE	FALSE
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	HUMANIZED SMART ANTI-IL-12 ANTIBODY	drugbank:DB05848	HUMANIZED SMART ANTI-IL-12 ANTIBODY	FALSE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.1491695205559502	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TdgClinicalTrial	Jan-14	NULL	0.4318065068724876	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
UNIPROT:O43525	hgnc:6297	KCNQ3	TdgClinicalTrial	Jan-14	NULL	1.500219178	ICA-105665	drugbank:DB06089	ICA-105665	FALSE	FALSE	FALSE
UNIPROT:P20273	hgnc:1643	CD22	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	INOTUZUMAB OZOGAMICIN	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
UNIPROT:P41597	hgnc:1603	CCR2	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	INCB3284	drugbank:DB05130	INCB3284	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.015921065	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	1.050153425	KRP-104	chembl:CHEMBL4297624	BISEGLIPTIN	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.004191225	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	ENOXAPARIN	rxcui:221095	ENOXAPARIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.1544343271638073	ZICRONAPINE	ncit:C152950	ZICRONAPINE	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	LUMIRACOXIB	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.030598876	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.037003292	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.027752469	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.027752469	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.375054795	OSPEMIFENE	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.7143900848393808	OTAMIXABAN	ncit:C90704	OTAMIXABAN	FALSE	FALSE	FALSE
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.094608417	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.4412409347537352	RIVASTIGMINE	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
UNIPROT:P17752	hgnc:12008	TPH1	TdgClinicalTrial	Jan-14	NULL	2.625383561784725	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:P00439	hgnc:8582	PAH	TdgClinicalTrial	Jan-14	NULL	3.500511415712967	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:P11309	hgnc:8986	PIM1	TdgClinicalTrial	Jan-14	NULL	0.5000730593875666	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TdgClinicalTrial	Jan-14	NULL	2.059124362184097	TAMIBAROTENE	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1469979597863787	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P30559	hgnc:8529	OXTR	TdgClinicalTrial	Jan-14	NULL	0.3563869088395554	OXYTOCIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.012901148	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:P14780	hgnc:7176	MMP9	TdgClinicalTrial	Jan-14	NULL	1.050153425	TST10088	drugbank:DB05151	TST10088	FALSE	FALSE	FALSE
UNIPROT:P46734	hgnc:6843	MAP2K3	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
UNIPROT:P00749	hgnc:9052	PLAU	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	WX-UK1	drugbank:DB05476	WX-UK1	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.092443083	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
UNIPROT:P08581	hgnc:7029	MET	TdgClinicalTrial	Jan-14	NULL	0.1842374429322613	XL880	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	YKP-10A	chembl:CHEMBL4297620	SOLRIAMFETOL	FALSE	FALSE	FALSE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TdgClinicalTrial	Jan-14	NULL	0.1215455352678113	XP13512	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
UNIPROT:P31994	hgnc:3618	FCGR2B	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.05814803	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.064111931	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.192335792	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.059532507	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.096050618	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.063072278	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.1141471113819445	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	4.449802647092754	CILAZAPRIL	rxcui:21102	CILAZAPRIL	TRUE	FALSE	FALSE
UNIPROT:Q13639	hgnc:5299	HTR4	TdgClinicalTrial	Jan-14	NULL	1.923357921	CISAPRIDE	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TdgClinicalTrial	Jan-14	NULL	0.8751278539282417	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1215455352678113	DRONEDARONE	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.1325951293830669	DRONEDARONE	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.081872668	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.1201548540862574	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.08914715	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.083744292	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.078682824	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.055504938	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.083257407	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.3697723326457359	PROPOXYPHENE	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.090739063	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.056622219	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.081365193	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.093763699	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
UNIPROT:O43497	hgnc:1394	CACNA1G	TEND	1-Aug-11	NULL	1.750255707856483	ETHOSUXIMIDE	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
UNIPROT:P13631	hgnc:9866	RARG	TEND	1-Aug-11	NULL	0.4412409347537352	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
UNIPROT:Q02641	hgnc:1401	CACNB1	TEND	1-Aug-11	NULL	1.071585127259071	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
UNIPROT:P51681	hgnc:1606	CCR5	TEND	1-Aug-11	NULL	3.938075342677087	MARAVIROC	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
UNIPROT:P34972	hgnc:2160	CNR2	TEND	1-Aug-11	NULL	1.514644363	NABILONE	rxcui:31447	NABILONE	TRUE	FALSE	FALSE
UNIPROT:P12259	hgnc:3542	F5	TEND	1-Aug-11	NULL	1.179947668217853	DROTRECOGIN ALFA	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
UNIPROT:P00451	hgnc:3546	F8	TEND	1-Aug-11	NULL	4.118248724368195	DROTRECOGIN ALFA	rxcui:352374	DROTRECOGIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P12319	hgnc:3609	FCER1A	TEND	1-Aug-11	NULL	3.750547945	BENZYLPENICILLOYL POLYLYSINE	rxcui:19079	BENZYLPENICILLOYL POLYLYSINE	TRUE	FALSE	FALSE
UNIPROT:P05230	hgnc:3665	FGF1	TEND	1-Aug-11	NULL	2.333674277141978	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.059532507	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	CRA-024781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.192335792	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.064111931	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TEND	1-Aug-11	NULL	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TEND	1-Aug-11	NULL	0.043866058	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P08620	hgnc:3682	FGF4	TEND	1-Aug-11	NULL	6.300920548283339	PENTOSAN POLYSULFATE	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.1166837138570989	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TEND	1-Aug-11	NULL	1.060761035064535	CETRORELIX	rxcui:68147	CETRORELIX	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.091476779	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.096167896	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.087222045	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.087512785	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.106290832	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.1022876712383659	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.1376949420516464	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.1132444383228493	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	1.514644363	ALMOTRIPTAN	rxcui:279645	ALMOTRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.045898314	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.3977853881492006	DEXFENFLURAMINE	rxcui:3268	DEXFENFLURAMINE	TRUE	FALSE	FALSE
UNIPROT:P26358	hgnc:2976	DNMT1	TEND	1-Aug-11	NULL	0.1909369863116163	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
UNIPROT:Q13639	hgnc:5299	HTR4	TEND	1-Aug-11	NULL	1.923357921	CISAPRIDE	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.028645756	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.070543222	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P01589	hgnc:6008	IL2RA	TEND	1-Aug-11	NULL	0.1715936968486748	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
UNIPROT:O14920	hgnc:5960	IKBKB	TEND	1-Aug-11	NULL	2.500365296937833	AURANOFIN	rxcui:1227	AURANOFIN	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.033458584	DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TEND	1-Aug-11	NULL	0.021087418	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.4817217544559128	DIPHENOXYLATE	rxcui:3500	DIPHENOXYLATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	GLYCOPYRROLATE	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TEND	1-Aug-11	NULL	0.3059887601147698	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1241316104862754	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TEND	1-Aug-11	NULL	0.2778183663264259	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.076840494	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.3580068493342807	MELOXICAM	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
UNIPROT:P22891	hgnc:9460	PROZ	TEND	1-Aug-11	NULL	1.810609352954982	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.2853677784548614	MIDODRINE	rxcui:6963	MIDODRINE	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TEND	1-Aug-11	NULL	0.3454452054979901	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
UNIPROT:Q16647	hgnc:9603	PTGIS	TEND	1-Aug-11	NULL	7.501095890813499	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.5707355569097228	PHENDIMETRAZINE	rxcui:33272	PHENDIMETRAZINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.172722603	elacestrant	rxcui:2628469	ELACESTRANT	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.031555091	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	0.3088686543276147	PHYSOSTIGMINE	rxcui:8299	PHYSOSTIGMINE	TRUE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TEND	1-Aug-11	NULL	3.828684360936057	PRASUGREL	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.056581542	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
UNIPROT:P04818	hgnc:12441	TYMS	TEND	1-Aug-11	NULL	1.117184494376478	RALTITREXED	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
UNIPROT:P04035	hgnc:5006	HMGCR	TEND	1-Aug-11	NULL	0.729273212	ROSUVASTATIN	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.1666910197958555	ROPINIROLE	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	1.154014752432846	RIZATRIPTAN	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.1154014752432845	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TEND	1-Aug-11	NULL	0.1124502911321247	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.4070362111294147	TERBUTALINE	rxcui:10368	TERBUTALINE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.1136529680426287	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.1084869240406911	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TEND	1-Aug-11	NULL	0.05593857	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TEND	1-Aug-11	NULL	0.31919557	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
UNIPROT:P23945	hgnc:3969	FSHR	TEND	1-Aug-11	NULL	18.37768493249307	UROFOLLITROPIN	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:Q9NYX4	hgnc:17938	CALY	TEND	1-Aug-11	NULL	1.750255707856483	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TEND	1-Aug-11	NULL	0.074478966	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P07947	hgnc:12841	YES1	TEND	1-Aug-11	NULL	0.013113804	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TEND	1-Aug-11	NULL	0.2917092846427472	VINDESINE	rxcui:11204	VINDESINE	FALSE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.4070362111294147	ZALEPLON	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.4907258993990139	AM-001	ncit:C151946	TOPICAL POTASSIUM DOBESILATE	FALSE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	6.563458904461812	ASP7991	chembl:CHEMBL3545100	ASP7991	FALSE	FALSE	FALSE
ATRIAL NATRIURETIC PEPTIDE RECEPTOR A	hgnc:7943	NPR1	TTD	2020.06.01	NULL	0.8078103267029924	Ataciguat	ncit:C79587	ATACIGUAT	FALSE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.1875273972703375	everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
SERINE/THREONINE-PROTEIN KINASE RAF	hgnc:18513	ZHX2	TTD	2020.06.01	NULL	2.100306849	MLN2480	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	0.1426838892274307	TD-1473	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	2.100306849	GSK3196165	ncit:C170271	OTILIMAB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	0.2282942227638891	ABT-494	iuphar.ligand:9246	UPADACITINIB	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	BGB-A317	rxcui:2677426	TISLELIZUMAB	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	0.1426838892274307	ASP-015K	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	1.400204566285186	Lenzilumab	ncit:C125081	LENZILUMAB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	3.000438356	Fostamatinib disodium	rxcui:2055929	FOSTAMATINIB DISODIUM	TRUE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.2187819634820604	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.061737415	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1232574442152452	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE LYN	hgnc:6735	LYN	TTD	2020.06.01	NULL	0.2917092846427472	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	1.750255707856483	Golotimod	rxcui:2367440	GOLOTIMOD	FALSE	FALSE	FALSE
LCK TYROSINE PROTEIN KINASE	hgnc:6524	LCK	TTD	2020.06.01	NULL	0.2287915957982331	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
INTERLEUKIN-21	hgnc:6005	IL21	TTD	2020.06.01	NULL	17.50255707856483	IL-21	iuphar.ligand:4987	IL-21	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	0.1103102336884338	BAY 10-00394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	0.2083637747448194	BAY 10-00394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
FOLLICLE STIMULATING HORMONE	hgnc:3964	FSHB	TTD	2020.06.01	NULL	13.12691780892362	Follicle stimulating hormone	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
CELL DIFFERENTIATION	hgnc:2505	CTLA4	TTD	2020.06.01	NULL	1.750255707856483	FF-10501	ncit:C122835	INOSINE 5'-MONOPHOSPHATE DEHYDROGENASE INHIBITOR FF-10501-01	FALSE	FALSE	FALSE
GABA TRANSPORTER GAT-1	hgnc:11042	SLC6A1	TTD	2020.06.01	NULL	14.00204566285186	Tiagabine	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA 1	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	1.779921058837101	Disitertide	ncit:C166687	DISITERTIDE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.3561566847382379	Brimonidine	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC KAINATE 1	hgnc:4579	GRIK1	TTD	2020.06.01	NULL	0.6563458904461812	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
GERANYLTRANSTRANSFERASE	hgnc:3631	FDPS	TTD	2020.06.01	NULL	1.750255707856483	Incadronate	ncit:C65906	INCADRONIC ACID	FALSE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	1.514644363	Almogran	rxcui:279645	ALMOTRIPTAN	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	1.346350544504987	Metastat	chembl:CHEMBL2104970	INCYCLINIDE	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.7721716358190367	Isoflurophate	rxcui:6027	ISOFLUROPHATE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4B	hgnc:8781	PDE4B	TTD	2020.06.01	NULL	0.2917092846427472	Piclamilast	ncit:C96718	PICLAMILAST	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.150021918	GNTI	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.2966535098061835	Gallopamil	rxcui:4648	GALLOPAMIL	FALSE	FALSE	FALSE
TUBULIN BETA-2 CHAIN	hgnc:12412	TUBB2A	TTD	2020.06.01	NULL	0.078136416	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA-2/DELTA-1	hgnc:1399	CACNA2D1	TTD	2020.06.01	NULL	0.192335792	Pregabalin	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	0.1093909817410302	Acitretin	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA 1	hgnc:4571	GRIA1	TTD	2020.06.01	NULL	0.1058622403945453	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.090739063	Propiomazine	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD1A	hgnc:1634	CD1A	TTD	2020.06.01	NULL	4.773424657790409	Antithymocyte globulin	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.138178082	CI-1033	ncit:C1880	CANERTINIB DIHYDROCHLORIDE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1017590527823536	Methyprylon	rxcui:6910	METHYPRYLON	TRUE	FALSE	FALSE
ENDOTHELIAL LIPASE	hgnc:6623	LIPG	TTD	2020.06.01	NULL	26.25383561784724	GSK-264220A	iuphar.ligand:6697	GSK-264220A	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	0.9845188356692718	Glimepiride	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	2.019525817	GUAIACOL	rxcui:5031	GUAIACOL	TRUE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	15.00219178	Travoprost	rxcui:283809	TRAVOPROST	TRUE	FALSE	FALSE
SERINE PROTEASE UNSPECIFIC	hgnc:11756	TFF2	TTD	2020.06.01	NULL	4.375639269641208	Gabexate	ncit:C76960	GABEXATE	FALSE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 2	hgnc:11331	SSTR2	TTD	2020.06.01	NULL	0.9723642821424906	Octreotide	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.011474579	Acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.2108741816694558	Pazopanib HCl	chembl:CHEMBL1201733	PAZOPANIB HYDROCHLORIDE	FALSE	FALSE	FALSE
INTERLEUKIN 6 RECEPTOR	hgnc:6019	IL6R	TTD	2020.06.01	NULL	4.039051633514961	Tocilizumab	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
RETINAL PIGMENT EPITHELIUM PROTEIN	hgnc:10294	RPE65	TTD	2020.06.01	NULL	15.00219178	AAV2-hRPE65v2	rxcui:1995537	VORETIGENE NEPARVOVEC	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	KW-2478	chembl:CHEMBL4297298	KW-2478	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	13.12691780892362	ND7001	drugbank:DB05142	ND7001	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Nemorubicin	ncit:C83999	NEMORUBICIN	FALSE	FALSE	FALSE
INTERCELLULAR ADHESION MOLECULE ICAM-1	hgnc:5344	ICAM1	TTD	2020.06.01	NULL	13.12691780892362	BI-505	chembl:CHEMBL2109482	BI-505	FALSE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	2.333674277141977	BMS-927711	rxcui:2282307	RIMEGEPANT	TRUE	FALSE	FALSE
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.9546849315580818	RG7155	ncit:C125548	EMACTUZUMAB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.2678962818147679	Fruquintinib	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	2.059124362184098	AV-203	chembl:CHEMBL2109401	AV-203	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.3081436105381133	Ramucirumab	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.069089041	Clotiazepam	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	1.193356164447602	SGI110	hemonc:252	GUADECITABINE	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	1.029562181092049	ABT-981	ncit:C166465	LUTIKIZUMAB	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	0.6731752722524935	CERC-301	ncit:C152228	RISLENEMDAZ	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.3659071166250487	TSR-042	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	AUNP-12	drugbank:DB15771	AUNP-12	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.042845917	EVT-201	chembl:CHEMBL5095096	DIMDAZENIL	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.097236428	Loperamide	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	0.5048814541893701	Clobetasol	rxcui:2590	CLOBETASOL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2B	hgnc:282	ADRA2B	TTD	2020.06.01	NULL	0.1339481409073839	MOXONIDINE	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE BETA	hgnc:5960	IKBKB	TTD	2020.06.01	NULL	0.089298761	Staurosporine	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
NOTCH-3 RECEPTOR	hgnc:7883	NOTCH3	TTD	2020.06.01	NULL	21.00306849427779	Tarextumab	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.2419708351875322	AC-170	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	2.282942227638891	ABT-126	chembl:CHEMBL3545231	ABT-126	FALSE	FALSE	FALSE
CHOLINE TRANSPORTER-LIKE PROTEIN 4	hgnc:13941	SLC44A4	TTD	2020.06.01	NULL	6.563458904461812	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
SUCCINATE-SEMIALDEHYDE DEHYDROGENASE	hgnc:408	ALDH5A1	TTD	2020.06.01	NULL	3.750547945	Chlormerodrin	ncit:C65315	CHLORMERODRIN	TRUE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.2778183663264258	Ibutilide	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	1.875273972703375	Potassium Chloride	rxcui:8591	POTASSIUM CHLORIDE	TRUE	FALSE	FALSE
E3 UBIQUITIN-PROTEIN LIGASE COP1	hgnc:17440	COP1	TTD	2020.06.01	NULL	2.625383561784724	Procainamide	rxcui:8700	PROCAINAMIDE	TRUE	FALSE	FALSE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	1.458546423213736	Vidarabine	rxcui:11194	VIDARABINE	TRUE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	2.625383561784724	NN-414	chembl:CHEMBL135191	TIFENAZOXIDE	FALSE	FALSE	FALSE
FACILITATES CHROMATIN TRANSCRIPTION COMPLEX	hgnc:11465	SUPT16H	TTD	2020.06.01	NULL	26.25383561784724	CBL0137	ncit:C107239	FACT COMPLEX-TARGETING CURAXIN CBL0137	FALSE	FALSE	TRUE
PI3-KINASE BETA	hgnc:8976	PIK3CB	TTD	2020.06.01	NULL	0.4167275494896388	BAY 1082439	chembl:CHEMBL3545245	BAY-1082439	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1389091831632129	LY3164530	ncit:C118281	ANTI-MET/EGFR MONOCLONAL ANTIBODY LY3164530	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Butylscopolamine	rxcui:1085787	BUTYLSCOPOLAMINE	TRUE	FALSE	FALSE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	3.750547945	Dinoprost Tromethamine	rxcui:23321	DINOPROST TROMETHAMINE	TRUE	FALSE	FALSE
IDURONATE 2-SULFATASE	hgnc:5389	IDS	TTD	2020.06.01	NULL	26.25383561784724	Idursulfase	rxcui:644101	IDURSULFASE	TRUE	FALSE	FALSE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	1.406455479527531	Misoprostol	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
ALPHA-N-ACETYLGLUCOSAMINIDASE	hgnc:7632	NAGLU	TTD	2020.06.01	NULL	52.50767123569449	N-Acetyl-D-glucosamine	rxcui:1362871	ACETYLGLUCOSAMINE	TRUE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	0.3025133322221082	Rituximab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	Alvespimycin hydrochloride	ncit:C76665	ALVESPIMYCIN HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TdgClinicalTrial	Jan-14	NULL	0.2344092465879218	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	1.810609352954982	CP-870893	chembl:CHEMBL2109477	SELICRELUMAB	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE PIM-2	hgnc:8987	PIM2	TTD	2020.06.01	NULL	1.312691780892362	AZD1208	iuphar.ligand:7698	AZD1208	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	1.544343271638073	CMP-001	ncit:C175875	VIDUTOLIMOD	FALSE	FALSE	FALSE
SOLUBLE EPOXIDE HYDROLASE	hgnc:3402	EPHX2	TTD	2020.06.01	NULL	1.500219178	GSK2256294	iuphar.ligand:9718	GSK2256294	FALSE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	1.810609352954982	MEDI4920	chembl:CHEMBL4594331	DAZODALIBEP	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	GSK1521498	iuphar.ligand:9287	GSK1521498	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:3288	iuphar.ligand:3288	GR79236	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.8255923150266431	AMG 479	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
APOPTOSIS REGULATOR BCL-W	hgnc:995	BCL2L2	TTD	2020.06.01	NULL	0.8204323630577265	ABT-263	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
SPHINGOSINE KINASE 2	hgnc:18859	SPHK2	TTD	2020.06.01	NULL	13.12691780892362	ABC294640	ncit:C98278	OPAGANIB	FALSE	FALSE	FALSE
NCBIGENE:1949	hgnc:3228	EFNB3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9126	iuphar.ligand:9126	BAY-320	FALSE	FALSE	FALSE
NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE	hgnc:30092	NAMPT	TTD	2020.06.01	NULL	10.50153424713889	CHS-828	drugbank:DB12980	CHS-828	FALSE	FALSE	FALSE
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	0.2853677784548614	GSK2981278	iuphar.ligand:9661	GSK2981278	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR BETA	hgnc:9865	RARB	TTD	2020.06.01	NULL	2.059124362184097	Tamibarotene	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	Hirudin	rxcui:1546205	HIRUDIN	FALSE	FALSE	FALSE
NCBIGENE:1519	hgnc:2542	CTSO	GuideToPharmacology	2024.1	inhibitor	0.8334550989792778	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
NCBIGENE:1389	hgnc:2350	CREBL2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10264	iuphar.ligand:10264	MLS000536924	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.041150213	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:69	iuphar.ligand:69	GR 125,743	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	modulator	0.4526523382387456	IUPHAR.LIGAND:104	iuphar.ligand:104	RS-30199	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.012233847	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	HARMINE HYDROCHLORIDE	chembl:CHEMBL1593867	HARMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.026626608	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.090530468	IUPHAR.LIGAND:92	rxcui:33739	PIPAMPERONE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.021554873	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.6326225450083675	IUPHAR.LIGAND:3219	iuphar.ligand:3219	[3H]N-METHYL-AZ10419369	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	0.3500511415712967	IUPHAR.LIGAND:608	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.037213091	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:141	drugbank:DB01488	DIMETHYLTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:262	iuphar.ligand:262	[3H]5-CT	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.056826484	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.056826484	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1396480617970598	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.011262907	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.012256693	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.276356164	IUPHAR.LIGAND:216	iuphar.ligand:216	(+)-NORFENFLURAMINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:8424	iuphar.ligand:8424	BF-1	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:230	iuphar.ligand:230	YM348	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.077217164	IUPHAR.LIGAND:167	iuphar.ligand:167	S 16924	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.020320306	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.040452751	IUPHAR.LIGAND:204	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.046840028	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:84	rxcui:21877	CYAMEMAZINE	FALSE	FALSE	FALSE
NCBIGENE:1263	hgnc:2154	PLK3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:12242	ncit:C177068	CLESACOSTAT	FALSE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	DTC	9/2/20	NULL	1.093909817410302	SRIF-28	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:8994	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1259176768242074	IUPHAR.LIGAND:9913	iuphar.ligand:9913	FLUMBATINIB	FALSE	FALSE	FALSE
NCBIGENE:1662	hgnc:2735	DDX10	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8680	iuphar.ligand:8680	IK-862	FALSE	FALSE	FALSE
NCBIGENE:1231	hgnc:1603	CCR2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:5131	iuphar.ligand:5131	ABT702	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.3017682254924971	THIOINOSINE	ncit:C877	THIOINOSINE	FALSE	FALSE	FALSE
NCBIGENE:3068	hgnc:4856	HDGF	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10023	iuphar.ligand:10023	LRE1	FALSE	FALSE	FALSE
NCBIGENE:1674	hgnc:2770	DES	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8663	iuphar.ligand:8663	COMPOUND 12C [PMID: 16516466]	FALSE	FALSE	FALSE
NOTCH1	hgnc:7881	NOTCH1	MyCancerGenome	20-Jun-17	other/unknown	0.6563458904461813	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:12216	iuphar.ligand:12216	MS15	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:490	iuphar.ligand:490	A-119637	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:489	iuphar.ligand:489	5-METHYLURAPIDIL	FALSE	FALSE	FALSE
NCBIGENE:1921	hgnc:19679	AAK1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:11957	iuphar.ligand:11957	PILAVAPADIN	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:6456	rxcui:50166	FOSINOPRIL	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:6377	rxcui:60245	IMIDAPRIL	TRUE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.08334551	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	0.3454452054979901	IUPHAR.LIGAND:4145	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
NCBIGENE:684	hgnc:1119	BST2	GuideToPharmacology	2024.1	blocker	1.381780822	IUPHAR.LIGAND:11474	iuphar.ligand:11474	NS383	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:432	iuphar.ligand:404	XANTHINE AMINE CONGENER	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:5619	iuphar.ligand:5619	PSB-10	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5606	iuphar.ligand:5606	FK-453	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.085239726	IUPHAR.LIGAND:380	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:3284	iuphar.ligand:3284	PSB603	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.067664525	IUPHAR.LIGAND:380	iuphar.ligand:380	CYCLOPENTYLADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.5413161983061289	IUPHAR.LIGAND:436	iuphar.ligand:436	[125I]AB-MECA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:5608	rxcui:2199015	ISTRADEFYLLINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:459	iuphar.ligand:459	MRE 3008F20	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1353290495765322	IUPHAR.LIGAND:459	iuphar.ligand:459	MRE 3008F20	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	0.1881995384791917	IUPHAR.LIGAND:3936	iuphar.ligand:3936	L-162,313	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:585	iuphar.ligand:585	ANGIOTENSIN III	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9390	iuphar.ligand:9390	CERALASERTIB	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:8358	iuphar.ligand:8358	GSK1070916	FALSE	FALSE	TRUE
PROTEIN-TYROSINE PHOSPHATASE 1B	hgnc:9642	PTPN1	TTD	2020.06.01	NULL	2.100306849	Trodusquemine	ncit:C123882	TRODUSQUEMINE	FALSE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.039960176	IUPHAR.LIGAND:5718	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:6475	iuphar.ligand:6475	LY2886721	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.252440727	IUPHAR.LIGAND:9512	ncit:C96754	SOLABEGRON	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:555	rxcui:8620	PRACTOLOL	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:3462	iuphar.ligand:3462	CL316243	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:545	iuphar.ligand:545	NIHP	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:7246	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:8136	iuphar.ligand:8136	COMPOUND 2 [PMID: 15546730]	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	Zalospirone	ncit:C152944	ZALOSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:2722	ncbigene:2722	GLC1B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8233	iuphar.ligand:8233	GSK2801	FALSE	FALSE	FALSE
NCBIGENE:1624	hgnc:2692	DBIP1	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:6508	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:719	iuphar.ligand:719	CALINDOL	FALSE	FALSE	FALSE
NCBIGENE:2344	hgnc:2528	CTSC	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:9412	iuphar.ligand:9412	BRENSOCATIB	FALSE	FALSE	FALSE
NCBIGENE:2352	hgnc:3795	FOLR3	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8561	iuphar.ligand:8561	CITIBRASINE	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:746	ncit:C184881	ONTERNABEZ	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.1442518440541057	IUPHAR.LIGAND:731	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:3503	iuphar.ligand:3503	GV150013	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.3163112725041837	IUPHAR.LIGAND:119	iuphar.ligand:119	[3H]SUMATRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:750	iuphar.ligand:750	AM-630	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:760	iuphar.ligand:760	FLU-CCL3	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	6.177373086552294	IUPHAR.LIGAND:9679	iuphar.ligand:9679	AZD1678	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:757	iuphar.ligand:757	CCL4	FALSE	FALSE	FALSE
NCBIGENE:1318	hgnc:11017	SLC31A2	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:11350	iuphar.ligand:11350	65PF	FALSE	FALSE	FALSE
NCBIGENE:2997	hgnc:4706	GYS1	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:9899	iuphar.ligand:9899	AH10-7	FALSE	FALSE	FALSE
NCBIGENE:1876	hgnc:3120	E2F6	GuideToPharmacology	2024.1	NULL	17.50255707856483	IUPHAR.LIGAND:5079	iuphar.ligand:5079	CD70	FALSE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:11442	iuphar.ligand:11442	EPCORITAMAB	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:11442	iuphar.ligand:11442	EPCORITAMAB	FALSE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:12975	iuphar.ligand:12975	MW05	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	agonist	0.007866318	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:1507	hgnc:1737	CDC42BPA	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8197	iuphar.ligand:8197	COMPOUND 11D [DOI: 10.1039/C0MD00194E]	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.095295229	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:2836	hgnc:1817	CEACAM5	GuideToPharmacology	2024.1	antibody	2.282942227638891	IUPHAR.LIGAND:8252	iuphar.ligand:8252	LABETUZUMAB GOVITECAN	FALSE	FALSE	FALSE
NCBIGENE:706	hgnc:1158	TSPO	GuideToPharmacology	2024.1	blocker	0.172722603	IUPHAR.LIGAND:4270	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
NCBIGENE:2903	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	antibody	0.760980743	IUPHAR.LIGAND:9209	iuphar.ligand:9209	ZOLBETUXIMAB	FALSE	FALSE	FALSE
NCBIGENE:705	hgnc:1157	BYSL	GuideToPharmacology	2024.1	blocker	10.50153425	IUPHAR.LIGAND:4177	iuphar.ligand:4177	DIDS	FALSE	FALSE	FALSE
NCBIGENE:3201	hgnc:5105	HOXA4	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12035	iuphar.ligand:12035	ELAFIN	FALSE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:3996	iuphar.ligand:3996	MUSCARINE	FALSE	FALSE	FALSE
NCBIGENE:396	hgnc:678	ARHGDIA	GuideToPharmacology	2024.1	activator	5.834185692854944	IUPHAR.LIGAND:2352	drugbank:DB02527	CYCLIC ADENOSINE MONOPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	antibody	1.312691780892362	IUPHAR.LIGAND:9744	rxcui:1989794	EMICIZUMAB	TRUE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10099	iuphar.ligand:10099	ZIFAXABAN	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:8914	iuphar.ligand:8914	ONATASERTIB	FALSE	FALSE	FALSE
NCBIGENE:2842	hgnc:4473	GPR19	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11988	ncit:C148181	DANICOPAN	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9850	iuphar.ligand:9850	GW406381	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9253	iuphar.ligand:9253	PEPTIDE 30 [PMID: 27019010]	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.03357268	IUPHAR.LIGAND:2714	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:913	iuphar.ligand:913	CORTICOTROPIN-RELEASING FACTOR	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:923	iuphar.ligand:923	&ALPHA;-HELICAL CRF	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:3512	iuphar.ligand:3512	NBI27914	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:684	iuphar.ligand:684	ADRENOMEDULLIN 2/INTERMEDIN	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:690	iuphar.ligand:690	CT-(8-32) (SALMON)	FALSE	FALSE	FALSE
NCBIGENE:718	hgnc:1318	C3	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:719	hgnc:1319	C3AR1	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1432	hgnc:6876	MAPK14	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:10062	iuphar.ligand:10062	ABX-1431	FALSE	FALSE	FALSE
NCBIGENE:723	hgnc:4283	GJB1	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:728	hgnc:1338	C5AR1	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:728	hgnc:1338	C5AR1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:731	hgnc:1352	C8A	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	LY3009120	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
NCBIGENE:734	hgnc:1355	OSGIN2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9170	iuphar.ligand:9170	COMPOUND 51 [MALLINGER ET AL., 2016]	FALSE	FALSE	FALSE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8913	iuphar.ligand:8913	AMG-337	FALSE	FALSE	FALSE
TDO2	hgnc:11708	TDO2	NCI	14-Sep-17	NULL	0.84012274	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
NCBIGENE:1356	hgnc:2295	CP	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:5281	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
NCBIGENE:1354	hgnc:2651	CYP7A1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8871	iuphar.ligand:8871	(2S,4S)-KETOCONAZOLE	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:3352	iuphar.ligand:3352	LTE4	FALSE	FALSE	FALSE
NCBIGENE:642	hgnc:1059	BLMH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:3207	iuphar.ligand:3207	P'-GERANYL 2-FLUOROMEVALONATE 5-DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10481	iuphar.ligand:10481	COMPOUND 1 [PMID: 31477924]	FALSE	FALSE	FALSE
NCBIGENE:3230	hgnc:5131	HOXD@	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:12657	iuphar.ligand:12657	ART558	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.5000730593875666	AMG 337	ncit:C95203	C-MET INHIBITOR AMG 337	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:1900	iuphar.ligand:1900	13,14-DIHYDRO-15-KETO-PGD2	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:1890	iuphar.ligand:1890	ZK118182	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:3304	ncit:C87494	ECOPIPAM HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.089756703	IUPHAR.LIGAND:948	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.079197091	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:7680	iuphar.ligand:7680	AZD1981	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.017715139	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:7227	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.018921683	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:950	iuphar.ligand:3296	[3H]7-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.070010228	IUPHAR.LIGAND:7227	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.070010228	IUPHAR.LIGAND:11976	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.009211872	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:3301	iuphar.ligand:3301	A412997	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.06714536	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	antibody	0.025003653	IUPHAR.LIGAND:6883	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.105015342	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	modulator	1.944728564284981	IUPHAR.LIGAND:5819	iuphar.ligand:5819	COMPOUND 1 [PMID: 20080612]	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.6482428547616604	IUPHAR.LIGAND:5852	iuphar.ligand:5852	MRE-269	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:5859	iuphar.ligand:5859	TCS 2510	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.045461187	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:4039	iuphar.ligand:4039	CP734432	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:12521	iuphar.ligand:12521	KMN-159	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1946	iuphar.ligand:1946	13,14-DIHYDRO-PGE1	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:1941	iuphar.ligand:1941	L-798,106	FALSE	FALSE	FALSE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:4511	iuphar.ligand:4511	[3H]NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE	FALSE	FALSE	FALSE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:4590	ncit:C76030	DRAFLAZINE	FALSE	FALSE	FALSE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:4512	iuphar.ligand:4512	NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE	FALSE	FALSE	FALSE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:4734	iuphar.ligand:4734	KF24345	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:5856	iuphar.ligand:5856	MF 498	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1953	iuphar.ligand:1953	GW 627368	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.048216411	IUPHAR.LIGAND:2801	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:9761	iuphar.ligand:9761	COMPOUND 9 [PMID: 26006010]	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:7717	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
ANGPT1	hgnc:484	ANGPT1	ChEMBL	33	inhibitor	1.312691780892362	AMG-780	chembl:CHEMBL2109586	AMG-780	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:7355	rxcui:1441386	BAZEDOXIFENE	TRUE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.2734774543525755	IUPHAR.LIGAND:2828	iuphar.ligand:2828	DAIDZEIN	FALSE	FALSE	FALSE
NCBIGENE:624	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2817	drugbank:DB04468	AFIMOXIFENE	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:7349	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
NCBIGENE:623	hgnc:1029	BDKRB1	GuideToPharmacology	2024.1	inhibitor	0.1767935058440892	IUPHAR.LIGAND:2801	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:13016	iuphar.ligand:13016	BMS-193884	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:3494	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:1005	iuphar.ligand:1005	[125I]BQ3020	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:1009	iuphar.ligand:1009	A192621	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:13016	iuphar.ligand:13016	BMS-193884	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	1.009762908	WR-243246	chembl:CHEMBL117217	CHEMBL:CHEMBL117217	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:3951	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
NCBIGENE:2018	hgnc:3341	EMX2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12236	iuphar.ligand:12236	COMPOUND 39 [PMID: 36127295]	FALSE	FALSE	FALSE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:5206	iuphar.ligand:5206	JNJ1661010	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3154	iuphar.ligand:3154	NE58027	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:4346	iuphar.ligand:4346	ZK93423	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	blocker	0.1988926940746003	IUPHAR.LIGAND:4369	iuphar.ligand:4369	[35S]TBPS	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:4363	iuphar.ligand:4363	[3H]L655708	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:4107	iuphar.ligand:4107	5-ME-IAA	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.072424374	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6110	iuphar.ligand:6110	GAL-(K)4	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6102	iuphar.ligand:6102	M1151	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6112	iuphar.ligand:6112	GAL-B2-C10	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6141	iuphar.ligand:6141	GALANIN(1-12)	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:7976	drugbank:DB07410	[2-(3-DIBENZOFURAN-4-YL-PHENYL)-1-HYDROXY-1-PHOSPHONO-ETHYL]-PHOSPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:247	hgnc:434	ALOX15B	GuideToPharmacology	2024.1	agonist	0.3804903712731485	IUPHAR.LIGAND:6998	rxcui:56188	SERMORELIN	TRUE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:10740	iuphar.ligand:10740	HM01	FALSE	FALSE	FALSE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:11429	rxcui:2601723	TIRZEPATIDE	TRUE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:3544	iuphar.ligand:3544	GLUCAGON-LIKE PEPTIDE 1-(7-37)	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	modulator	0.9907107780319716	IUPHAR.LIGAND:7585	iuphar.ligand:7585	BETP	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:4249	iuphar.ligand:4249	LY404187	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	LONIDAMINE	ncit:C1146	LONIDAMINE	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	modulator	0.4688184931758437	IUPHAR.LIGAND:4249	iuphar.ligand:4249	LY404187	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:3448	iuphar.ligand:3448	ZK112993	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.010650643	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1268301237577161	IUPHAR.LIGAND:4240	iuphar.ligand:4240	L701324	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4155	ncit:C152322	SELFOTEL	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	blocker	0.09963505	IUPHAR.LIGAND:4233	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:746	ncit:C184881	ONTERNABEZ	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	positive modulator	0.4234489615781814	CX1739	chembl:CHEMBL3707399	CX1739	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:2360	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:746	ncit:C184881	ONTERNABEZ	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:2360	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:2366	iuphar.ligand:2366	BILOBALIDE	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.017114626	IUPHAR.LIGAND:5925	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.068458502	IUPHAR.LIGAND:8018	iuphar.ligand:8018	1-AZAKENPAULLONE	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10064	iuphar.ligand:10064	GLYT1 INHIBITOR 27A	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:9664	iuphar.ligand:9664	BML-281	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:7010	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	ChEMBL	33	inhibitor	12.11715490054488	BMS-863233	drugbank:DB12357	BMS-863233	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.07767407	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:1229	iuphar.ligand:1229	BURIMAMIDE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.4487835148349957	IUPHAR.LIGAND:1242	iuphar.ligand:1241	N-[3H]METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:1267	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
NCBIGENE:128	hgnc:253	ADH5	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:5567	iuphar.ligand:5567	9-HYDROXYOCTADECADIENOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	1.591141552596802	IUPHAR.LIGAND:3353	iuphar.ligand:3353	LTD4	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	1.591141552596802	IUPHAR.LIGAND:1749	drugbank:DB03435	URIDINE-5'-DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:87	hgnc:163	ACTN1	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:10567	iuphar.ligand:10567	GPR15L	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5520	iuphar.ligand:5520	ASN04885796	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:9967	iuphar.ligand:9967	ML193	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	agonist	0.03729238	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	0.577007376	IUPHAR.LIGAND:9176	iuphar.ligand:9176	WZ4002	FALSE	FALSE	TRUE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:5531	iuphar.ligand:5531	COMPOUND 48/80	FALSE	FALSE	FALSE
NCBIGENE:1398	hgnc:2362	CRK	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11054	iuphar.ligand:11054	LEI-401	FALSE	FALSE	FALSE
NCBIGENE:2453	hgnc:3850	FRA13A	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9689	iuphar.ligand:9689	MK-0429	FALSE	FALSE	FALSE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8220	iuphar.ligand:8220	COMPOUND 15 [PMID: 24900237]	FALSE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10152	drugbank:DB18060	EMAVUSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1723	hgnc:2867	DHODH	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:4967	iuphar.ligand:4967	IFN-&BETA;	FALSE	FALSE	FALSE
NCBIGENE:1736	hgnc:2890	DKC1	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:12169	iuphar.ligand:12169	SPESOLIMAB	FALSE	FALSE	FALSE
NCBIGENE:1706	ncbigene:1706	DFNB14	GuideToPharmacology	2024.1	agonist	5.250767124	IUPHAR.LIGAND:4997	iuphar.ligand:4997	IL-5	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	activator	0.1458546423213736	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:666	hgnc:1087	BOK	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:12433	iuphar.ligand:12433	DENATONIUM	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:12465	iuphar.ligand:12465	THEAFLAVIN-3′-O-GALLATE	FALSE	FALSE	FALSE
NCBIGENE:674	ncbigene:674	BRAFPS1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:12438	iuphar.ligand:12438	ARISTOLOCHIC ACID	FALSE	FALSE	FALSE
CLCN6	hgnc:2024	CLCN6	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:669	hgnc:1093	BPGM	GuideToPharmacology	2024.1	inhibitor	0.6819178082557728	IUPHAR.LIGAND:4357	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10156	iuphar.ligand:10156	JAK3 INHIBITOR 32	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:6977	iuphar.ligand:6977	COMPOUND 19A [PMID: 24359159]	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:12318	iuphar.ligand:12318	GDC-0214	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:7954	iuphar.ligand:7954	BMS-911543	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:9696	iuphar.ligand:9696	OCLACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:11178	iuphar.ligand:11178	BIIB068	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:11565	iuphar.ligand:11565	COMPOUND 13AC [PMID: 33256400]	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:9862	ncit:C141273	POSELTINIB	FALSE	FALSE	FALSE
NCBIGENE:2379	hgnc:3891	FRA2G	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11947	ncit:C184930	SEBETRALSTAT	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.076765601	IUPHAR.LIGAND:8866	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.064111931	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	NULL	0.172722603	IUPHAR.LIGAND:10482	iuphar.ligand:10482	COMPOUND 16 [PMID: 31498617]	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.015964631	IUPHAR.LIGAND:7816	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.1037701012563132	IUPHAR.LIGAND:12381	iuphar.ligand:12381	RESENCATINIB	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:10223	iuphar.ligand:10223	[D-TYR-14C]TAK-448	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:4014	iuphar.ligand:4014	4-FLUOROBENZOYL-FGLRW-NH2	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:9930	iuphar.ligand:9930	HENATINIB	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1282	iuphar.ligand:1282	[125I]KISSPEPTIN-54 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	blocker	0.9546849315580819	IUPHAR.LIGAND:2328	iuphar.ligand:2328	CHARYBDOTOXIN	FALSE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	0.3804903712731485	Mozavaptan	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:516	hgnc:841	ATP5MC1	GuideToPharmacology	2024.1	activator	2.625383561784725	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	activator	0.082043236	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:441	hgnc:6269	KCNJ8	GuideToPharmacology	2024.1	activator	0.546954909	IUPHAR.LIGAND:4254	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	4.773424657790408	IUPHAR.LIGAND:2607	iuphar.ligand:2607	MK-499	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:10494	iuphar.ligand:10494	SWE101	FALSE	FALSE	FALSE
NCBIGENE:546	hgnc:886	ATRX	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:7760	iuphar.ligand:7760	GXTX-1E	FALSE	FALSE	FALSE
NCBIGENE:545	hgnc:882	ATR	GuideToPharmacology	2024.1	blocker	0.051478109	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:2908	iuphar.ligand:2908	VPC32183	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1290	iuphar.ligand:1290	AC-HMCH-(6-16)-NH2	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1302	iuphar.ligand:1302	VARIANT MCH	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:10702	iuphar.ligand:10702	COMPOUND 15A [PMID: 32069401]	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:8914	iuphar.ligand:8914	ONATASERTIB	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7973	iuphar.ligand:7973	XL388	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:12614	iuphar.ligand:12614	METATINIB	FALSE	FALSE	FALSE
NCBIGENE:2386	hgnc:3898	FRA3C	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:6564	iuphar.ligand:6564	PHENYLACETYL-ARG-VAL-ARG-4-AMIDINOBENZYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	antibody	0.3088686543276147	IUPHAR.LIGAND:10505	iuphar.ligand:10505	AMIVANTAMAB	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.3088686543276147	IUPHAR.LIGAND:8913	iuphar.ligand:8913	AMG-337	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:11623	iuphar.ligand:11623	GUMARONTINIB	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.1235474617310458	IUPHAR.LIGAND:5700	iuphar.ligand:5700	PHA-665752	FALSE	FALSE	TRUE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1410	iuphar.ligand:1410	L-AP4	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:10135	iuphar.ligand:10135	VU2957	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6442	iuphar.ligand:6442	COMPOUND 18 [PMID: 21927650]	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:9622	iuphar.ligand:9622	FOLIGLURAX	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1410	iuphar.ligand:1410	L-AP4	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1393	iuphar.ligand:1393	EGLUMEGAD	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1410	iuphar.ligand:1410	L-AP4	FALSE	FALSE	FALSE
NCBIGENE:2072	hgnc:3436	ERCC4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9988	iuphar.ligand:9988	COMPOUND 16D [TAO ET AL., 2009]	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:1443	iuphar.ligand:1443	D-AP4	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1411	ncit:C169894	DEXFOSFOSERINE	FALSE	FALSE	FALSE
NCBIGENE:2093	ncbigene:2093	ERVT3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9380	iuphar.ligand:9380	BIX02189	FALSE	FALSE	FALSE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9699	iuphar.ligand:9699	COMPOUND 5 [PMID: 28038940]	FALSE	FALSE	FALSE
NCBIGENE:2076	ncbigene:2076	ERCM1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11178	iuphar.ligand:11178	BIIB068	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NCBIGENE:2088	ncbigene:2088	ERVK3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8134	iuphar.ligand:8134	COMPOUND 26 [PMID: 24673130]	FALSE	FALSE	FALSE
NCBIGENE:1631	hgnc:7174	MMP7	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:8567	iuphar.ligand:8567	RS 39066	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10887	iuphar.ligand:10887	(R)-ND-336	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:12123	iuphar.ligand:12123	MAGLI 432	FALSE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:7844	iuphar.ligand:7844	AZD1236	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:5281	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1455	iuphar.ligand:1455	[NLEU13,GLU14]MOTILIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.042073455	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.078958904	IUPHAR.LIGAND:329	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:327	iuphar.ligand:327	METHOCTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:8591	iuphar.ligand:8591	ML381	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:326	iuphar.ligand:326	LITHOCHOLYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:1363	iuphar.ligand:1363	LUZINDOLE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.1154014752432846	IUPHAR.LIGAND:7471	rxcui:1516803	ALVIMOPAN ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:8870	iuphar.ligand:8870	AT-076	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.030850571	IUPHAR.LIGAND:7236	rxcui:203188	METHYLPHENIDATE HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.037345428	IUPHAR.LIGAND:2398	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:2998	hgnc:4707	GYS2	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:9904	iuphar.ligand:9904	EG01377	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:10257	iuphar.ligand:10257	GR-389988	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1468	iuphar.ligand:1468	NEUROMEDIN S-33	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1474	iuphar.ligand:1474	[125I]NEUROMEDIN U-25 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:304	hgnc:539	ANXA2P2	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:1495	iuphar.ligand:1495	NEUROPEPTIDE W-23	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11707	iuphar.ligand:11707	SHA 68R	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:10280	iuphar.ligand:10280	CP-1	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1700	iuphar.ligand:1700	[ALA11, D-LEU15]OREXIN-B	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1697	iuphar.ligand:1697	OREXIN-A	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1699	iuphar.ligand:1699	OREXIN-B	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1701	iuphar.ligand:1701	JNJ-10397049	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:9305	iuphar.ligand:9305	NAG 26	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8939	iuphar.ligand:8939	FRAX597	FALSE	FALSE	FALSE
NCBIGENE:2137	hgnc:3518	EXTL3	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:9542	iuphar.ligand:9542	PSB-12062	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.029317516	IUPHAR.LIGAND:1765	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:3384	iuphar.ligand:3384	ARL66096	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5809	iuphar.ligand:5809	MRS2950	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:1779	iuphar.ligand:1779	UDP N-ACETYL-GLUCOSAMINE	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1750	iuphar.ligand:1750	UDP-&BETA;-S	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:10365	iuphar.ligand:10365	COMPOUND 2Q [PMID: 30986068]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:9571	iuphar.ligand:9571	ECF309	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.029698909	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.055155117	IUPHAR.LIGAND:8918	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:9425	ncit:C174798	NEMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:1295	hgnc:2215	COL8A1	GuideToPharmacology	2024.1	activator	3.500511415712967	IUPHAR.LIGAND:2351	iuphar.ligand:2351	CALMODULIN	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12114	iuphar.ligand:12114	EXAMPLE 2 [WO2013026797A1]	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:10626	ncit:C124226	UZANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:8167	iuphar.ligand:8167	LEUCETTINE L41	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:10626	ncit:C124226	UZANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6433	iuphar.ligand:6433	TRIAZINE COMPOUND PC10	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:11619	ncit:C80870	TOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:1433	hgnc:9067	PLD1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8782	iuphar.ligand:8782	COMPOUND 69 [PMID: 19136975]	FALSE	FALSE	FALSE
NCBIGENE:2386	hgnc:3898	FRA3C	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8648	iuphar.ligand:8648	MULTI-LEU (ML)-PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:7420	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1254	ncbigene:1254	CMTX3	GuideToPharmacology	2024.1	modulator	17.50255707856483	IUPHAR.LIGAND:8552	iuphar.ligand:8552	SGC707	FALSE	FALSE	FALSE
NCBIGENE:1544	hgnc:2596	CYP1A2	GuideToPharmacology	2024.1	modulator	0.04427291	IUPHAR.LIGAND:8821	iuphar.ligand:8821	MT47-100	FALSE	FALSE	FALSE
NCBIGENE:1486	hgnc:2496	CTBS	GuideToPharmacology	2024.1	inhibitor	0.5770073762164232	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.2524407270946851	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12319	iuphar.ligand:12319	LARTESERTIB	FALSE	FALSE	FALSE
NCBIGENE:1489	hgnc:2499	CTF1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9964	iuphar.ligand:9964	NIK SMI1	FALSE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:12311	iuphar.ligand:12311	SZM679	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9688	iuphar.ligand:9688	RIPK2 INHIBITOR 8	FALSE	FALSE	FALSE
NCBIGENE:2811	hgnc:4439	GP1BA	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:8721	iuphar.ligand:8721	CCG-4986	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:2647	iuphar.ligand:2647	RO 40-6055	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2647	iuphar.ligand:2647	RO 40-6055	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9322	rxcui:1992864	NETARSUDIL	TRUE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:8326	iuphar.ligand:8326	MINIMISED RELAXIN-3 ANALOGUE 3	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:11911	iuphar.ligand:11911	R3/I5- SMBIT	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	activator	0.1419126249613364	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:2929	iuphar.ligand:2929	COMPOUND 26 [PMID: 16190743]	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:9289	rxcui:2121085	SIPONIMOD	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:2927	iuphar.ligand:2927	CYM5181	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:12125	iuphar.ligand:12125	BD-1063	FALSE	FALSE	FALSE
NCBIGENE:2707	hgnc:4285	GJB3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8100	ncit:C152325	SELISISTAT	FALSE	FALSE	FALSE
NCBIGENE:2707	hgnc:4285	GJB3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8778	iuphar.ligand:8778	COMPOUND 17 [PMID: 23570514]	FALSE	FALSE	FALSE
NCBIGENE:959	hgnc:11935	CD40LG	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:589	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11146	iuphar.ligand:11146	COMPOUND 59 [PMID: 30889352]	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9611	iuphar.ligand:9611	ER-27319	FALSE	FALSE	FALSE
NCBIGENE:1417	hgnc:2400	CRYBB3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9657	ncit:C152832	VARESPLADIB	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:7731	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2014	iuphar.ligand:2014	L-362,855	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:10004	iuphar.ligand:10004	KX2-361	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:2028	iuphar.ligand:2028	[D-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:5647	iuphar.ligand:5647	ANALOG 30 [PMID:18543899]	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.210030685	IUPHAR.LIGAND:2014	iuphar.ligand:2014	L-362,855	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.1973972602845657	IUPHAR.LIGAND:8487	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2058	iuphar.ligand:2058	[111IN,90Y]DOTA-OC	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2017	iuphar.ligand:2017	NC 4-28B	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2014	iuphar.ligand:2014	L-362,855	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:2037	iuphar.ligand:2037	BIM 23059	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2034	iuphar.ligand:2034	BIM 23030	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	0.5585922471882393	IUPHAR.LIGAND:2067	iuphar.ligand:2067	PRL-2970	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	0.2234368988752957	IUPHAR.LIGAND:2028	iuphar.ligand:2028	[D-TYR8]CYN 154806	FALSE	FALSE	FALSE
NCBIGENE:1462	hgnc:2464	VCAN	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12667	iuphar.ligand:12667	EXAMPLE 15 [WO2015079413]	FALSE	FALSE	FALSE
NCBIGENE:1015	hgnc:1756	CDH17	GuideToPharmacology	2024.1	NULL	4.375639269641208	IUPHAR.LIGAND:4628	rxcui:10454	THIAMINE	TRUE	FALSE	FALSE
NCBIGENE:1754	hgnc:11850	TLR4	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:10091	iuphar.ligand:10091	CRX-555	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3332	iuphar.ligand:3332	I-SAP	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	activator	0.3977853881492008	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	0.3977853881492008	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.7721716358190367	IUPHAR.LIGAND:10295	iuphar.ligand:10295	LARIXYL ACETATE	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	2.763561643983921	IUPHAR.LIGAND:2445	iuphar.ligand:2445	CADPR	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	0.2083637747448194	IUPHAR.LIGAND:710	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11862	iuphar.ligand:11862	PRU-12	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:12543	iuphar.ligand:12543	EVP-21	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	0.3977853881492008	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	6.563458904461812	IUPHAR.LIGAND:6404	iuphar.ligand:6404	SF-11	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4110	iuphar.ligand:4110	6-IODO-NORDIHYDROCAPSAICIN	FALSE	FALSE	FALSE
NCBIGENE:2424	ncbigene:2424	FRA8F	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9333	iuphar.ligand:9333	RWJ-56423	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	1.117184494376478	IUPHAR.LIGAND:9400	iuphar.ligand:9400	AZ3146	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:4294	iuphar.ligand:4294	RN1734	FALSE	FALSE	FALSE
NCBIGENE:1884	ncbigene:1884	EBR3	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:5067	iuphar.ligand:5067	TWEAK	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:11565	iuphar.ligand:11565	COMPOUND 13AC [PMID: 33256400]	FALSE	FALSE	FALSE
NCBIGENE:2427	hgnc:3937	FRA9C	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8660	iuphar.ligand:8660	COMPOUND 6 [PMID: 17948018]	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:1155	iuphar.ligand:1155	SECRETIN	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:1152	iuphar.ligand:1152	VIP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:10615	ncit:C169802	BALOVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:2213	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.092606122	IUPHAR.LIGAND:2200	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.007308974	IUPHAR.LIGAND:2213	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.058471794	IUPHAR.LIGAND:3483	iuphar.ligand:3483	[3H]NELIVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2225	iuphar.ligand:2225	D[PEN1,TYR(ME)2]AVP	FALSE	FALSE	FALSE
NCBIGENE:2278	ncbigene:2278	FIM1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:7702	iuphar.ligand:7702	ADAVOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1505	iuphar.ligand:1505	NPY	FALSE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	0.5048814541893702	IUPHAR.LIGAND:7731	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.009220191	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.010160153	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	1.500219178	CAPMATINIB	rxcui:2362165	CAPMATINIB	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	CIViC	10-Apr-24	NULL	0.2681242786503549	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	1.346350544504987	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	CIViC	10-Apr-24	NULL	0.027276712	ERIBULIN	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	CIViC	10-Apr-24	NULL	0.2187819634820604	AZD3463	iuphar.ligand:7706	AZD3463	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.3241214273808302	TYRPHOSTIN AG 1296	ncit:C1731	TYRPHOSTIN AG 1296	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.2546668357992238	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.1852122442176172	MULTIKINASE INHIBITOR AEE788	ncit:C48369	MULTIKINASE INHIBITOR AEE788	FALSE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	CIViC	10-Apr-24	NULL	0.3302369260106572	TEGAFUR	rxcui:10995	URACIL	TRUE	FALSE	TRUE
RIT1	hgnc:10023	RIT1	CIViC	10-Apr-24	NULL	0.7721716358190368	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
GNA11	hgnc:4379	GNA11	CIViC	10-Apr-24	NULL	1.050153425	SOTRASTAURIN ACETATE	ncit:C80631	SOTRASTAURIN ACETATE	FALSE	FALSE	TRUE
NOTCH3	hgnc:7883	NOTCH3	CIViC	10-Apr-24	NULL	21.00306849427779	TAREXTUMAB	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	CIViC	10-Apr-24	NULL	0.022122465	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SRSF2	hgnc:10783	SRSF2	CIViC	10-Apr-24	NULL	26.25383561784724	CTX-712	ncit:C199490	CLK INHIBITOR CTX-712	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.03043923	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.034244133	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.041150213	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1026542937159227	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1193356164447602	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.1598407039138341	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.071928317	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	1.237091730683901	Lifirafenib	ncit:C124995	LIFIRAFENIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.4948366922735607	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.074975256	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.026181836	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.056157937	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.061773731	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.1372749574789398	Tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
CDK12	hgnc:24224	CDK12	JAX-CKB	10-Apr-24	NULL	0.2592971419046642	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.760980743	THZ1	iuphar.ligand:8052	THZ1	FALSE	FALSE	FALSE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	0.5556367326528517	I-BET151	iuphar.ligand:7518	I-BET151	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.050764748	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1962903597596056	RO4987655	ncit:C82696	MEK INHIBITOR RO4987655	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	1.658136986390352	Vofatamab	ncit:C116863	VOFATAMAB	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.033497717	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.3684748858645227	3D185	ncit:C175460	FGFR/CSF-1R INHIBITOR 3D185	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1944728564284981	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.04182212	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.020257589	Idarubicin	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.4605936073306534	ERAS-007	ncit:C150248	ERK1/2 INHIBITOR ERAS-007	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.172722603	PD173074	iuphar.ligand:5037	PD173074	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.6419030713410085	BAY1436032	chembl:CHEMBL4206033	BAY1436032	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.032095154	CG-806	ncit:C162573	LUXEPTINIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.039688338	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.024759276	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.024309107	Uprosertib	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.097236428	GSK126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.005653281	Bortezomib	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.033529803	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.1919140030544389	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.011591097	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.028977744	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001750547	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.033117421	PD0166285	iuphar.ligand:8183	PD166285	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.013636585	Acalabrutinib	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.2318219480604613	Napabucasin	ncit:C96429	NAPABUCASIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.00473106	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	negative modulator	0.2778183663264258	ESKETAMINE HYDROCHLORIDE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3125456621172291	BARNIDIPINE	rxcui:39879	MEPIRODIPINE	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
SLC28A1	hgnc:11001	SLC28A1	DTC	9/2/20	NULL	1.400204566285186	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	7-OXOCALLITRISIC ACID, METHYL ESTER	chembl:CHEMBL1568605	7-OXOCALLITRISIC ACID, METHYL ESTER	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	ISOCYANATO-CYCLOHEXANE	chembl:CHEMBL26886	CHEMBL:CHEMBL26886	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	L-687384	chembl:CHEMBL1256916	CHEMBL:CHEMBL1256916	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.100589408	ROBINETIN	chembl:CHEMBL170405	ROBINETIN	FALSE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	4.039051633514961	KUSHENOL A	chembl:CHEMBL455679	KUSHENOL A	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.071439008	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
IL1A	hgnc:5991	IL1A	NCI	14-Sep-17	NULL	0.4375639269641208	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
CHUK	hgnc:1974	CHUK	DTC	9/2/20	NULL	1.250182648468916	N-(3-OXODODECANOYL)HOMOSERINELACTONE	chembl:CHEMBL8483	CHEMBL:CHEMBL8483	FALSE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.012573676	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:2729	hgnc:4311	GCLC	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:7524	iuphar.ligand:7524	XD14	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.067059606	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.047626006	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	DNDI1417722	chembl:CHEMBL1503190	CHEMBL:CHEMBL1503190	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.036718651	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008503267	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.026045472	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
RBL1	hgnc:9893	RBL1	NCI	14-Sep-17	NULL	15.00219178162699	HMBA	ncit:C1125	HEXAMETHYLENE BISACETAMIDE	FALSE	FALSE	FALSE
MCOLN3	hgnc:13358	MCOLN3	DTC	9/2/20	NULL	6.563458904461812	TCMDC-124500	iuphar.ligand:6404	SF-11	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:223	iuphar.ligand:223	[3H]RAUWOLSCINE	FALSE	FALSE	FALSE
OTC	hgnc:8512	OTC	PharmGKB	4/5/24	NULL	0.3070624048871023	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P08185	hgnc:1540	SERPINA6	TEND	1-Aug-11	NULL	0.2853677784548614	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	activator	0.7501095890813501	IUPHAR.LIGAND:2619	iuphar.ligand:2619	BATRACHOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:9278	ncit:C152707	TRADIPITANT	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	AG-126	chembl:CHEMBL77387	CHEMBL:CHEMBL77387	FALSE	FALSE	FALSE
JUNB	hgnc:6205	JUNB	NCI	14-Sep-17	NULL	0.4070362111294147	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.347732922	NITROVIN	chembl:CHEMBL1395447	NITROVIN	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.031189588	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.2224901323546377	IUPHAR.LIGAND:262	iuphar.ligand:262	[3H]5-CT	FALSE	FALSE	FALSE
PSMB4	hgnc:9541	PSMB4	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.7501095890813501	MIVACURIUM CHLORIDE	rxcui:52796	MIVACURIUM CHLORIDE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	DTC	9/2/20	NULL	0.07631929	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	3.182283105193606	CALCDPWW	chembl:CHEMBL1213646	CALCDPWW	FALSE	FALSE	FALSE
SLC22A7	hgnc:10971	SLC22A7	PharmGKB	4/5/24	NULL	0.3241214273808302	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
CD19	hgnc:1633	CD19	ChEMBL	33	binder	1.280674908	DENINTUZUMAB	ncit:C166425	DENINTUZUMAB	FALSE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	DTC	9/2/20	NULL	4.375639269641208	PHANTASMIDINE	chembl:CHEMBL1086654	PHANTASMIDINE	FALSE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TEND	1-Aug-11	NULL	0.4167275494896388	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	NCI	14-Sep-17	NULL	0.045639002	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.045421861	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.017739078	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.157680694	JNK INHIBITOR VIII	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	3.500511415712966	bucillamine	ncit:C83561	BUCILLAMINE	FALSE	FALSE	FALSE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	agonist	0.4375639269641208	INTERFERON BETA-1A	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	NCI	14-Sep-17	NULL	0.4861821410712453	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	ChEMBL	33	modulator	2.763561643983921	CAMOTESKIMAB	ncit:C179215	CAMOTESKIMAB	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.1988926940746003	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:4607	iuphar.ligand:4607	RHODAMINE123	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4299	iuphar.ligand:4299	RO4938581	FALSE	FALSE	FALSE
NCBIGENE:2514	hgnc:11120	SMPD1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10639	iuphar.ligand:10639	WJYK50	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.4234489615781814	IUPHAR.LIGAND:532	iuphar.ligand:532	CGP 12177	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00517674	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR-4	hgnc:3682	FGF4	TTD	2020.06.01	NULL	6.300920548283339	Pentosan Polysulfate	rxcui:155046	PENTOSAN POLYSULFATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:773	iuphar.ligand:773	HIV-TAT	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.046221542	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	2-ACETYLAMINOFLUORENE	chembl:CHEMBL311469	2-ACETYLAMINOFLUORENE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.010389329	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:388	hgnc:668	RHOB	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:5412	iuphar.ligand:5412	PGF1&ALPHA;	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.019318496	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2983390411119005	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:8159	iuphar.ligand:8159	COMPOUND 25 [PMID: 20855207]	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	DNDI1417932	chembl:CHEMBL1334191	CHEMBL:CHEMBL1334191	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.1193356164447602	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.037884323	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:413	hgnc:716	ARSC2	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	PharmGKB	4/5/24	NULL	0.034118045	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P27037	hgnc:173	ACVR2A	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	ACE-011	ncit:C80038	SOTATERCEPT	FALSE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	MILNACIPRAN HYDROCHLORIDE	rxcui:30003	MILNACIPRAN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2738	hgnc:4320	GLI4	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:7915	iuphar.ligand:7915	PFI-3	FALSE	FALSE	FALSE
MMP13	hgnc:7159	MMP13	ChEMBL	33	inhibitor	2.625383561784725	APRATASTAT	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.027347745	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	PIFITHRIN-ALPHA	chembl:CHEMBL198759	CHEMBL:CHEMBL198759	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	5.250767123569449	AMD070	ncit:C126660	MAVORIXAFOR	FALSE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.093931433	PS-341	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1215455352678113	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	L-21649	chembl:CHEMBL333021	L-21649	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3184	iuphar.ligand:3184	NE10575	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TEND	1-Aug-11	NULL	0.3864200913449379	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5787	iuphar.ligand:5787	PARA-COUMARIC ACID	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.08178765	ALLYLESTRENOL	rxcui:525	ALLYLESTRENOL	TRUE	FALSE	FALSE
NCBIGENE:3169	hgnc:5021	FOXA1	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:11395	iuphar.ligand:11395	MK-7110	FALSE	FALSE	FALSE
PRSS1	hgnc:9475	PRSS1	DTC	9/2/20	NULL	2.917092846427472	CYANOPEPTOLIN S	chembl:CHEMBL1076838	CYANOPEPTOLIN S	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	FERROUS SULFATE	rxcui:24947	FERROUS SULFATE	TRUE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	1.029562181092049	HER2 INHIBITOR CP-724,714	ncit:C26648	HER2 INHIBITOR CP-724,714	FALSE	FALSE	TRUE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.300043836	IUPHAR.LIGAND:2950	rxcui:596723	CERIVASTATIN	FALSE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	NCI	14-Sep-17	NULL	0.151464436	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
IL12B	hgnc:5970	IL12B	ChEMBL	33	inhibitor	1.250182648468916	MIRIKIZUMAB	rxcui:2668384	MIRIKIZUMAB	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	4.773424657790408	ASTRAGALIN	chembl:CHEMBL233930	ASTRAGALIN	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1750255707856483	PROPARGITE	chembl:CHEMBL1416084	PROPARGITE	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:9862	ncit:C141273	POSELTINIB	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:729	iuphar.ligand:729	2-ARACHIDONOYLGLYCEROL	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8982	iuphar.ligand:8982	INCB-38579	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.7160136986685613	BUNOLOL	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	3.750547945	AUTOLOGOUS LYMPHOCYTES	ncit:C28681	THERAPEUTIC AUTOLOGOUS LYMPHOCYTES	FALSE	FALSE	FALSE
IFI27	hgnc:5397	IFI27	NCI	14-Sep-17	NULL	1.093909817410302	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
NCBIGENE:1252	hgnc:5187	PRMT1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7028	iuphar.ligand:7028	AMI-1	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	GNF-PF-3012	chembl:CHEMBL582715	CHEMBL:CHEMBL582715	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.00881889	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1591141552596803	ANISOMYCIN	ncit:C95312	ANISOMYCIN	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.750109589	BMS-777607	drugbank:DB12064	BMS-777607	FALSE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.2536602475154323	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.00984765	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.061628722	E-10030	chembl:CHEMBL3301576	PEGPLERANIB SODIUM	FALSE	FALSE	FALSE
GDA	hgnc:4212	GDA	NCI	14-Sep-17	NULL	1.060761035064535	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:6511	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TEND	1-Aug-11	NULL	0.1593072549626653	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	0.789589041	Ramatroban	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	blocker	0.2419708351875322	LANICEMINE	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1047	iuphar.ligand:1047	HUMANIN	FALSE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	binder	2.100306849	MOC31-PE	chembl:CHEMBL2109265	MOC31-PE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.046059361	IUPHAR.LIGAND:360	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	inhibitor	0.023867123	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.068757317	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	0.4296082192011368	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8572	iuphar.ligand:8572	LP99	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:2213	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	1.272913242077442	GSK126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
RB1	hgnc:9884	RB1	DTC	9/2/20	NULL	0.062434805	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.028229931	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	DEFERIPRONE	rxcui:11645	DEFERIPRONE	TRUE	FALSE	FALSE
PARD3B	hgnc:14446	PARD3B	PharmGKB	4/5/24	NULL	1.280674908	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002436325	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:10401	iuphar.ligand:10401	RIPK3 INHIBITOR 42	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.0191914	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	0.4861821410712453	Dezapelisib	ncit:C107686	DEZAPELISIB	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	1.312691780892362	SULFAMIDE	chembl:CHEMBL355001	SULFAMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	GNF-PF-2298	chembl:CHEMBL578905	CHEMBL:CHEMBL578905	FALSE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE 1	hgnc:44465	RAB4B-EGLN2	TTD	2020.06.01	NULL	17.50255707856483	BAY-85-3934	chembl:CHEMBL3646118	MOLIDUSTAT	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	modulator	1.166837138570988	IUPHAR.LIGAND:7945	iuphar.ligand:7945	MK-2206	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:6914	iuphar.ligand:6914	[SAR1,ILE4,ILE8]ANG-II	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.2734774543525755	ERGOCORNINE	chembl:CHEMBL1385840	ERGOCORNINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.0023813	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	NCI	14-Sep-17	NULL	0.012026494	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	DTC	9/2/20	NULL	1.363835616511545	IC261	drugbank:DB03083	IC261	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.1530835896084387	MELAGATRAN	ncit:C66077	MELAGATRAN	FALSE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	ChEMBL	33	inhibitor	2.386712328895204	ENARODUSTAT	ncit:C169944	ENARODUSTAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
TNIK	hgnc:30765	TNIK	DTC	9/2/20	NULL	0.7292732116068681	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.016921583	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:4334	iuphar.ligand:4092	[3H]UBP310	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.040515178	Sitravatinib	ncit:C117734	SITRAVATINIB	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.364636606	BENZPHETAMINE	rxcui:1422	BENZPHETAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.017709164	tropisetron	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
C3	hgnc:1318	C3	DTC	9/2/20	NULL	11.66837138570988	COMPSTATIN	iuphar.ligand:9218	COMPSTATIN	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1325951293830669	(-)-DEMECOLCINE	ncit:C419	DEMECOLCINE	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.021484317	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.002976625	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.009430257	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.085239726	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:5820	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	2.917092846427472	BL22	chembl:CHEMBL2109352	BL22	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000673287	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.008027468	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.012067955	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.2573905452730122	5-BROMODEOXYURIDINE	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
ALOX5AP	hgnc:436	ALOX5AP	PharmGKB	4/5/24	NULL	0.1613138901250215	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	PharmGKB	4/5/24	NULL	0.8204323630577265	nusinersen	rxcui:1863556	NUSINERSEN	TRUE	FALSE	FALSE
UNIPROT:P04818	hgnc:12441	TYMS	TdgClinicalTrial	Jan-14	NULL	0.31919557	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:101	ncit:C73303	TIOSPIRONE	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	DTC	9/2/20	NULL	2.500365296937833	4-ANDROSTENE-3,17-DIONE-DELTA-4-DIONE	chembl:CHEMBL1077603	CHEMBL:CHEMBL1077603	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:552	iuphar.ligand:552	CICLOPROLOL	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:3466	ncit:C152958	ZINTEROL	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	ChEMBL	33	inhibitor	0.1544343271638073	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PSMD3	hgnc:9560	PSMD3	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.4134462302023188	FRAXINE	chembl:CHEMBL293864	FRAXINE	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.059667808	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.138178082	LY-2874455	drugbank:DB13022	LY-2874455	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.016434326	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.7778914257139926	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	1.944728564284981	Talotrexin	ncit:C29341	TALOTREXIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TRIS(2,3-DIBROMOPROPYL)PHOSPHATE	chembl:CHEMBL1904600	TRIS(2,3-DIBROMOPROPYL)PHOSPHATE	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.3365876361262467	ADRENOCORTICOTROPIN	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
ALDH1A2	hgnc:15472	ALDH1A2	PharmGKB	4/5/24	NULL	0.4565884455277782	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	0.8751278539282416	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
UNIPROT:P22455	hgnc:3691	FGFR4	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	TRAFERMIN	ncit:C152708	TRAFERMIN	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4179	iuphar.ligand:4179	DMCM	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:3792	iuphar.ligand:3792	[125I]KISSPEPTIN-13 (HUMAN)	FALSE	FALSE	FALSE
IFNA1	hgnc:5417	IFNA1	NCI	14-Sep-17	NULL	9.546849315580817	CORYNEBACTERIUM GRANULOSUM P40	ncit:C990	CORYNEBACTERIUM GRANULOSUM P40	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.9723642821424906	DEXMETHYLPHENIDATE HYDROCHLORIDE	rxcui:352372	DEXMETHYLPHENIDATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.017009288	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	1-BENZYLMALEIMIDE	chembl:CHEMBL388979	CHEMBL:CHEMBL388979	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CORYNANTHEINE	iuphar.ligand:5345	CORYNANTHINE	FALSE	FALSE	FALSE
NCBIGENE:1838	hgnc:3058	DTNB	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.030133527	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	ChEMBL	33	modulator	0.42006137	ATX08-001	chembl:CHEMBL3545278	ATX08-001	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.029766254	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1131630845596864	IUPHAR.LIGAND:2018	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.046549354	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.085796848	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
BCL2L11	hgnc:994	BCL2L11	DTC	9/2/20	NULL	3.750547945406749	KERACYANIN	rxcui:28165	KERACYANIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	VINPOCETINE	rxcui:24506	VINPOCETINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	VER-3323	iuphar.ligand:168	VER-3323	FALSE	FALSE	FALSE
STAT5A	hgnc:11366	STAT5A	DTC	9/2/20	NULL	17.50255707856483	AZD-1480	drugbank:DB12588	AZD-1480	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009974862	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	GS-39783	iuphar.ligand:5446	GS39783	FALSE	FALSE	FALSE
UNIPROT:P08253	hgnc:7166	MMP2	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	TST10088	drugbank:DB05151	TST10088	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007749066	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.1682938180631233	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1111273465305703	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.070010228	LANIFIBRANOR	ncit:C166556	LANIFIBRANOR	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BUTONATE	ncit:C75966	BUTONATE	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.006071655	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:1913	iuphar.ligand:1913	MB-28767	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:10615	ncit:C169802	BALOVAPTAN	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.729273212	LH-RH ANALOGS	ncit:C1910	GONADOTROPIN-RELEASING HORMONE ANALOG	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.012990517	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
MT-ND4	hgnc:7459	MT-ND4	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.2734774543525755	IUPHAR.LIGAND:262	iuphar.ligand:262	[3H]5-CT	FALSE	FALSE	FALSE
NCBIGENE:3128	hgnc:4954	HLA-DRB6	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11067	iuphar.ligand:11067	EXAMPLE 265 [WO2019097515A1]	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.045421861	IUPHAR.LIGAND:2714	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2430910705356226	GNF-PF-4798	chembl:CHEMBL584635	CHEMBL:CHEMBL584635	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	TCMDC-124166	chembl:CHEMBL528712	CHEMBL:CHEMBL528712	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.009106429	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CYCLIN-DEPENDENT KINASE 6	hgnc:1777	CDK6	TTD	2020.06.01	NULL	0.6141248097742047	LY2835219	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.1265245090016735	IUPHAR.LIGAND:92	rxcui:33739	PIPAMPERONE	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	0.1088116604009326	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	0.1785975212098452	MELAGATRAN	ncit:C66077	MELAGATRAN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.042481935	ERGOCORNINE	chembl:CHEMBL1385840	ERGOCORNINE	FALSE	FALSE	FALSE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547591	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.2300445618212245	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.4773424657790409	PD-360324	chembl:CHEMBL2109513	PD-360324	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6110	iuphar.ligand:6110	GAL-(K)4	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006990459	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P38484	hgnc:5440	IFNGR2	TdgClinicalTrial	Jan-14	NULL	105.0153424713889	INTERFERON GAMMA-1B	rxcui:5882	INTERFERON GAMMA-1B	TRUE	TRUE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TdgClinicalTrial	Jan-14	NULL	0.6035364509849942	VIGABATRIN	rxcui:14851	VIGABATRIN	TRUE	FALSE	FALSE
NCBIGENE:2089	ncbigene:2089	ERVT1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9964	iuphar.ligand:9964	NIK SMI1	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	NS-1619	iuphar.ligand:4272	NS1619	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.2273059360852575	SOBUZOXANE	ncit:C66540	SOBUZOXANE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.01823183	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
NOX3	hgnc:7890	NOX3	PharmGKB	4/5/24	NULL	1.750255707856483	propylthiouracil	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
UNIPROT:P06126	hgnc:1634	CD1A	TEND	1-Aug-11	NULL	4.773424657790409	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
FGF6	hgnc:3684	FGF6	NCI	14-Sep-17	NULL	6.177373086552294	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.4688184931758437	TOMUDEX	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	2.143170254518142	BIAFINE	ncit:C1807	BIAFINE CREAM	FALSE	FALSE	FALSE
LEUKOCYTE ANTIGEN CD37	hgnc:1666	CD37	TTD	2020.06.01	NULL	52.50767123569449	TRU-016	ncit:C74006	OTLERTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:1573	iuphar.ligand:1573	THR10CONTULAKIN-G	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.085239726	VER-49009	chembl:CHEMBL365617	CHEMBL:CHEMBL365617	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	DEXPROPRANOLOL	ncit:C77944	DEXPROPRANOLOL	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.072026984	ANTIHISTAMINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.5556367326528519	THP-ADRIAMYCIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.2430910705356226	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
UNIPROT:Q06187	hgnc:1133	BTK	TdgClinicalTrial	Jan-14	NULL	0.6863747873946993	AVL-292	ncit:C97037	SPEBRUTINIB	FALSE	FALSE	FALSE
PSMB1	hgnc:9537	PSMB1	MyCancerGenome	20-Jun-17	other/unknown	0.5233322714521046	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:P30559	hgnc:8529	OXTR	TEND	1-Aug-11	NULL	4.118248724368195	CARBETOCIN	ncit:C96858	CARBETOCIN	TRUE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	JAX-CKB	10-Apr-24	NULL	1.306751999078369	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.061197752	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
RIBONUCLEOTIDE REDUCTASE	hgnc:581	APBB1	TTD	2020.06.01	NULL	0.5834185692854944	Trimidox	wikidata:Q7842230	TRIMETHOPRIM/SULFADOXINE	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	DTC	9/2/20	NULL	0.1130007271930297	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
FERRITIN	hgnc:3976	FTH1	TTD	2020.06.01	NULL	52.50767123569449	Ferritarg P	drugbank:DB17375	FERRITARG P	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.041739007	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
EMBRYONIC ECTODERM DEVELOPMENT PROTEIN	hgnc:3188	EED	TTD	2020.06.01	NULL	8.751278539282415	MAK683	iuphar.ligand:10515	MAK683	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	Naloxegol	rxcui:1551777	NALOXEGOL	TRUE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.071341945	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	ANAZOLENE	chembl:CHEMBL1555467	ANAZOLENE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GNF-PF-3792	chembl:CHEMBL582983	CHEMBL:CHEMBL582983	FALSE	FALSE	FALSE
DDR2	hgnc:2731	DDR2	ChEMBL	33	inhibitor	0.6364566210387212	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.6250913242344582	PANCURONIUM BROMIDE	rxcui:7884	PANCURONIUM BROMIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
GPD2	hgnc:4456	GPD2	ChEMBL	33	inhibitor	0.4688184931758437	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.5770073762164231	IUPHAR.LIGAND:12956	iuphar.ligand:12956	BRORPHINE	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	0.4565884455277782	TSR-011	ncit:C114287	ALK/TRK INHIBITOR TSR-011	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.003423818	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1795134059339983	CALCIUM CHANNEL BLOCKER	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.061055432	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4252	rxcui:6694	MEFLOQUINE	TRUE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	CART-BCMA cells	ncit:C156272	AUTOLOGOUS ANTI-BCMA-CAR-TCRZ/4-1BB-EXPRESSING T-LYMPHOCYTES CART-BCMA	FALSE	FALSE	FALSE
NCBIGENE:1634	hgnc:2705	DCN	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12669	iuphar.ligand:12669	MMP13 TRACER  [18F]5J	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.9546849315580818	TASPOGLUTIDE	ncit:C152518	TASPOGLUTIDE	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.750109589	SL-0101	chembl:CHEMBL240954	CHEMBL:CHEMBL240954	FALSE	FALSE	FALSE
COL27A1	hgnc:22986	COL27A1	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1750255707856483	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
EPHA10	hgnc:19987	EPHA10	ChEMBL	33	inhibitor	0.9053046764774914	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
FN1	hgnc:3778	FN1	ChEMBL	33	binder	4.039051633514961	RADRETUMAB	ncit:C152144	RADRETUMAB	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.3043922970185189	amprenavir	rxcui:228656	AMPRENAVIR	TRUE	FALSE	FALSE
NCBIGENE:99	hgnc:4487	GPR32	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:3934	iuphar.ligand:3934	RESOLVIN D1	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.074797252	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.043430663	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.1988926940746003	DIFLORASONE	rxcui:23033	DIFLORASONE DIACETATE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1344626664166312	MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.006309501	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.1268301237577161	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.4167275494896388	remifentanil	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
SERPINA5	hgnc:8723	SERPINA5	PharmGKB	4/5/24	NULL	0.2822993077187876	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.046303061	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
PLEKHJ1	hgnc:18211	PLEKHJ1	PharmGKB	4/5/24	NULL	7.001022831425933	candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.056097939	ranolazine	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	ISOFLUROPHATE	rxcui:6027	ISOFLUROPHATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	(E),(E)-2,4-DECACIENAL	chembl:CHEMBL443949	CHEMBL:CHEMBL443949	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.086789539	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	1.779921058837101	MUSCLE RELAXANT	ncit:C29696	MUSCLE RELAXANT	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	2.282942227638891	NEBENTAN	ncit:C81108	NEBENTAN	FALSE	FALSE	FALSE
UNIPROT:Q8N9I0	hgnc:11510	SYT2	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	BOTULINUM TOXIN TYPE B	rxcui:2167673	BOTULINUM TOXIN TYPE B	TRUE	FALSE	FALSE
CASR	hgnc:1514	CASR	ChEMBL	33	modulator	3.281729452230906	TECALCET HYDROCHLORIDE	ncit:C76683	TECALCET HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	1.790034246671403	INDECAINIDE	ncit:C65910	INDECAINIDE	TRUE	FALSE	FALSE
KCNB1	hgnc:6231	KCNB1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
TNFRSF17	hgnc:11913	TNFRSF17	ChEMBL	33	binder	0.16256245	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	AMPEROZIDE HYDROCHLORIDE	ncit:C77259	AMPEROZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.006874531	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	DNDI1417072	chembl:CHEMBL1310701	CHEMBL:CHEMBL1310701	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	PSORALEN	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	8.751278539282417	ledipasvir	rxcui:1591922	LEDIPASVIR	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.2386712328895204	OXAPROZIN	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	UBP-302	iuphar.ligand:4333	UBP302	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	VIOMYCIN SULFATE	ncit:C66655	VIOMYCIN SULFATE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	OGLEMILAST	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 1 ALPHA	hgnc:4910	HIF1A	TTD	2020.06.01	NULL	0.036212187	2-Methoxyestradiol	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.1154014752432846	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.042793538	Ceralasertib	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.092606122	AMG888	ncit:C78853	PATRITUMAB	FALSE	TRUE	TRUE
PTK6	hgnc:9617	PTK6	ChEMBL	33	inhibitor	0.1131630845596864	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.042310775	Fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	AZOCYCLOTIN	chembl:CHEMBL1358709	AZOCYCLOTIN	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:2459	iuphar.ligand:2459	DECAVANADATE	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.021541609	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.021036727	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.062808219	IUPHAR.LIGAND:7792	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	1.050153425	ALLYL ISOTHIOCYANATE	iuphar.ligand:2420	ALLYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.00598378	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:4251	iuphar.ligand:4251	LY503430	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6129	iuphar.ligand:6129	GALANIN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	CALOTHRIXIN A	chembl:CHEMBL435295	CALOTHRIXIN A	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.04593847	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	3.938075342677087	Imiquimod	rxcui:59943	IMIQUIMOD	TRUE	TRUE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Belladonna	rxcui:89781	BELLADONNA EXTRACT, USP	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.032252869	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.1205533268166455	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
ADH5	hgnc:253	ADH5	ChEMBL	33	inhibitor	1.071585127259071	NITREFAZOLE	ncit:C72626	NITREFAZOLE	TRUE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:7912	iuphar.ligand:7912	LCL161	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.050597611	MECLIZINE	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.2019525816757481	PTC299	drugbank:DB05173	PTC299	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:1488	iuphar.ligand:1488	[125I]EYF	FALSE	FALSE	FALSE
NCBIGENE:2751	hgnc:4340	GLUD1P5	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:1024	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.032055965	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.076934317	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	7.001022831425932	RG7625	ncit:C174598	PETESICATIB	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	FLAVOXATE	rxcui:4440	FLAVOXATE	TRUE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:4613	rxcui:3268	DEXFENFLURAMINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.150021918	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.1976759387696734	PIOGLITAZONE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3821	iuphar.ligand:3821	[3H]GASTRIN	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	NULL	0.5000730593875666	IUPHAR.LIGAND:5088	iuphar.ligand:5088	VEGFD	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	0.2734774543525755	IUPHAR.LIGAND:2098	iuphar.ligand:2098	SUBSTANCE P	FALSE	FALSE	FALSE
NCBIGENE:1530	hgnc:10435	RPS6KA6	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.078545507	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.035478156	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	1.166837138570988	5,6,7-TRIBROMOISATIN	chembl:CHEMBL376616	CHEMBL:CHEMBL376616	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006397133	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.091159151	CYCLIC ADENOSINE MONOPHOSPHATE	drugbank:DB02527	CYCLIC ADENOSINE MONOPHOSPHATE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.022730594	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1226814748497534	Gestrinone	rxcui:4792	GESTRINONE	FALSE	FALSE	FALSE
NCBIGENE:718	hgnc:1318	C3	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:2366	iuphar.ligand:2366	BILOBALIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	2.080014029626545	ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:2680	hgnc:9886	KDM5A	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:7026	iuphar.ligand:7026	PBIT	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	blocker	0.1250182648468916	IUPHAR.LIGAND:2624	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:12004	iuphar.ligand:12004	DS69910557	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	1.312691780892362	PETROSIOL A	chembl:CHEMBL2349065	PETROSIOL A	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:5644	iuphar.ligand:5644	BASS ANTAGONIST	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.079758488	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	DTC	9/2/20	NULL	8.751278539282415	ERUCIN	chembl:CHEMBL2151143	ERUCIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	ACEPROMAZINE	rxcui:155	ACEPROMAZINE	TRUE	FALSE	FALSE
KCNK3	hgnc:6278	KCNK3	PharmGKB	4/5/24	NULL	0.6081969641200136	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	inhibitor	0.7721716358190367	ELZASONAN HYDROCHLORIDE	ncit:C73806	ELZASONAN HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	2-BROMOETHANOL	chembl:CHEMBL468583	2-BROMOETHANOL	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1773907812016706	ATROPINE SULFATE	rxcui:153971	ATROPINE SULFATE	TRUE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.3281729452230906	XL-418	chembl:CHEMBL2016893	XL-418	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.052090944	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:6458	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.1435420208739598	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.384671584	NG-MONOMETHYL-L-ARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.5147810905460244	GLYCYRRHETINIC ACID	rxcui:1311506	GLYCYRRHETINIC ACID	TRUE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.6908904109959803	JQ1	drugbank:DB17021	JQ1	FALSE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.040235763	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
LRP1	hgnc:6692	LRP1	NCI	14-Sep-17	NULL	1.060761035064535	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1100789753368857	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006987979	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	METRAZOLINE OXALATE	chembl:CHEMBL1255866	METRAZOLINE OXALATE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	GSK961081	chembl:CHEMBL3039518	BATEFENTEROL	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.028413242	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	binder	3.281729452230906	VRC-01LS	chembl:CHEMBL4298127	VRC-01LS	FALSE	FALSE	FALSE
NCBIGENE:1995	hgnc:3314	ELAVL3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:5940	iuphar.ligand:5940	D4476	FALSE	FALSE	FALSE
NCBIGENE:714	hgnc:1245	C1QC	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009922085	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.1548898856510162	IUPHAR.LIGAND:9193	iuphar.ligand:9193	ZYKLOPHIN	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:9391	iuphar.ligand:9391	COMPOUND 36 [PMID: 21958547]	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.028146701	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012977675	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
ITGA2B	hgnc:6138	ITGA2B	NCI	14-Sep-17	NULL	0.4375639269641209	RECOMBINANT TISSUE PLASMINOGEN ACTIVATOR	rxcui:8410	ALTEPLASE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	A-70108	iuphar.ligand:6077	A68930	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.2546668357992238	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	0.1902451856365742	HYDROCHLOROTHIAZIDE	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
PSMC5	hgnc:9552	PSMC5	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	TOMUZOTUXIMAB	ncit:C152692	TOMUZOTUXIMAB	FALSE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	ALBUVIRTIDE	drugbank:DB15166	ALBUVIRTIDE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.013113804	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.027781837	CPT-11	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NOCICEPTIN RECEPTOR	hgnc:8155	OPRL1	TTD	2020.06.01	NULL	6.563458904461812	LY-2940094	iuphar.ligand:9462	LY2940094	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:1137	iuphar.ligand:1137	[125I]EXENDIN-(9-39)	FALSE	FALSE	FALSE
CD3EAP	hgnc:24219	POLR1G	PharmGKB	4/5/24	NULL	0.3763990769583835	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	STIROFOS	chembl:CHEMBL1452359	STIROFOS	FALSE	FALSE	FALSE
CALMODULIN	hgnc:14986	SNAP91	TTD	2020.06.01	NULL	5.834185692854944	Aprindine	rxcui:1054	APRINDINE	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.1396480617970598	ISOPROPAMIDE IODIDE	rxcui:6051	ISOPROPAMIDE IODIDE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:10615	ncit:C169802	BALOVAPTAN	FALSE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TdgClinicalTrial	Jan-14	NULL	0.3763990769583835	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
NCBIGENE:2340	hgnc:2097	CMA1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9779	iuphar.ligand:9779	TY-51469	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:4082	iuphar.ligand:4082	[3H]CPP	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	ZAPA	chembl:CHEMBL20562	ZAPA	FALSE	FALSE	FALSE
NCBIGENE:252	hgnc:10608	SCTR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1152	iuphar.ligand:1152	VIP	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002529881	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.019447286	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.014464923	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.022632617	DEQUALINIUM	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.055563673	SIB-1757	iuphar.ligand:1431	SIB-1757	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.00402481	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.00804962	rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.1166837138570988	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
CARBONIC ANHYDRASE VI	hgnc:1380	CA6	TTD	2020.06.01	NULL	0.1136529680426288	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
CASPASE-1	hgnc:1499	CASP1	TTD	2020.06.01	NULL	1.346350544504987	Nivocasan	ncit:C98213	NIVOCASAN	FALSE	FALSE	FALSE
SRD5A2	hgnc:11285	SRD5A2	ChEMBL	33	inhibitor	4.375639269641208	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1221108633388244	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:1029	iuphar.ligand:1029	T-BOC-MET-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:6084	iuphar.ligand:6084	GALANIN(1-11)	FALSE	FALSE	FALSE
NCBIGENE:1633	hgnc:2704	DCK	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:10887	iuphar.ligand:10887	(R)-ND-336	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2248	iuphar.ligand:2248	L-368,228	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.034590034	IUPHAR.LIGAND:6057	iuphar.ligand:6057	VEGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.069454592	IUPHAR.LIGAND:8969	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.004920134	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
GATA4	hgnc:4173	GATA4	DTC	9/2/20	NULL	17.50255707856483	NSC-126866	chembl:CHEMBL1684099	CHEMBL:CHEMBL1684099	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.027811267	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.1223955040459079	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	1.693795846312725	Pirmenol	ncit:C81434	PIRMENOL	FALSE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.3684748858645228	N-ACETYLCYSTEINE	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
VON WILLEBRAND FACTOR	hgnc:12726	VWF	TTD	2020.06.01	NULL	8.290684931951763	ALX-0081	rxcui:2110604	CAPLACIZUMAB-YHDP	TRUE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.201178817	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	1.207072901969988	NIACINAMIDE	rxcui:7405	NIACINAMIDE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.5357925636295356	APIXABAN	rxcui:1364430	APIXABAN	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	MIRIPIRIUM	chembl:CHEMBL1393904	MIRIPIRIUM	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.086361301	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.030386384	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	3.500511415712966	NSC-607097	chembl:CHEMBL1374370	CHEMBL:CHEMBL1374370	FALSE	FALSE	FALSE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.106290832	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 70	hgnc:5232	HSPA1A	TTD	2020.06.01	NULL	13.12691780892362	Minnelide	drugbank:DB17309	MINNELIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	PharmGKB	4/5/24	NULL	0.003301746	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:2688	iuphar.ligand:2688	L-783483	FALSE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.2019525816757481	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2493241749083309	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	1.500219178	ZD2079	chembl:CHEMBL1354284	TALIBEGRON HYDROCHLORIDE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.1480479452134243	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
PROTO-ONCOGENE C-ROS	hgnc:10261	ROS1	TTD	2020.06.01	NULL	1.346350544504987	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.076709527	chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	DTC	9/2/20	NULL	4.375639269641208	ISOPROPYL ISOTHIOCYANATE	chembl:CHEMBL2208211	ISOPROPYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	3-CHLOROBENZOPEROXOIC ACID	chembl:CHEMBL458855	CHEMBL:CHEMBL458855	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.051885051	ONC201	iuphar.ligand:9978	ONC201	FALSE	FALSE	FALSE
ABCC9	hgnc:60	ABCC9	PharmGKB	4/5/24	NULL	0.4339476961627644	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
P-SELECTIN GLYCOPROTEIN LIGAND 1	hgnc:10722	SELPLG	TTD	2020.06.01	NULL	13.12691780892362	RO-4905417	iuphar.ligand:12312	INCLACUMAB	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.092443083	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	DECA-1,9-DIENE	chembl:CHEMBL31020	CHEMBL:CHEMBL31020	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.2775246894064191	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NDUFS6	hgnc:7713	NDUFS6	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.3182283105193605	ROFECOXIB	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.8468979231563628	TALAMPANEL	ncit:C38139	TALAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P15056	hgnc:1097	BRAF	TdgClinicalTrial	Jan-14	NULL	0.1832728489902076	XL281	drugbank:DB05190	XL281	FALSE	FALSE	TRUE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:6175	iuphar.ligand:6175	GASTRIN RELEASING PEPTIDE(14-27) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2888	hgnc:4565	GRB14	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9023	iuphar.ligand:9023	PSB-0963	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:9696	iuphar.ligand:9696	OCLACITINIB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CHELIDAMIC ACID	chembl:CHEMBL252909	CHELIDAMIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	AY-9944	chembl:CHEMBL1513392	CHEMBL:CHEMBL1513392	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.027752469	TOPIRAMATE	rxcui:38404	TOPIRAMATE	TRUE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.1166837138570989	IUPHAR.LIGAND:10387	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1402073998282897	PRN1371	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.1450488155682168	TCMDC-125480	chembl:CHEMBL546257	CHEMBL:CHEMBL546257	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS	ncit:C90775	LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS	FALSE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.128537751	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
LHCGR	hgnc:6585	LHCGR	DTC	9/2/20	NULL	6.563458904461812	CYCLOPENTYLCARBAMIC ACID BIPHENYL-3-YL ESTER	chembl:CHEMBL448753	CHEMBL:CHEMBL448753	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000130653	chembl:CHEMBL590212	CHEMBL:CHEMBL590212	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-3	hgnc:4077	GABRA3	TTD	2020.06.01	NULL	0.5834185692854944	NS-2710	chembl:CHEMBL381625	CHEMBL:CHEMBL381625	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	1.810609352954982	TENOVIN-1	chembl:CHEMBL1436543	CHEMBL:CHEMBL1436543	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.2160809515872201	HEPTACHLOR	chembl:CHEMBL194400	HEPTACHLOR	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:4131	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	inhibitor	5.250767123569449	MAVORIXAFOR	ncit:C126660	MAVORIXAFOR	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.075333818	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
SDHB	hgnc:10681	SDHB	NCI	14-Sep-17	NULL	0.6403374540938354	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.045226246	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
UNIPROT:P05362	hgnc:5344	ICAM1	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	BI-505	chembl:CHEMBL2109482	BI-505	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	OPC-28326	drugbank:DB05461	OPC-28326	FALSE	FALSE	FALSE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.056459862	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.065799087	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.2917092846427472	3-HYDROXYBENZYLHYDRAZINE DIHYDROCHLORIDE	iuphar.ligand:5116	3-HYDROXYBENZYLHYDRAZINE	FALSE	FALSE	FALSE
CD37	hgnc:1666	CD37	ChEMBL	33	binder	52.50767123569449	OTLERTUZUMAB	ncit:C74006	OTLERTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2135	hgnc:3516	EXTL2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8939	iuphar.ligand:8939	FRAX597	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:12040	iuphar.ligand:12040	OCEDURENONE	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.3889457128569963	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
CHUK	hgnc:1974	CHUK	DTC	9/2/20	NULL	7.501095891	GLAUCARUBINONE	chembl:CHEMBL458347	GLAUCARUBINONE	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.032412143	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
GABA(A) RECEPTOR DELTA	hgnc:4084	GABRD	TTD	2020.06.01	NULL	0.064944553	ALLOPREGNANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	agonist	0.2243917574174978	IUPHAR.LIGAND:710	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.045382603	IUPHAR.LIGAND:7794	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:9696	iuphar.ligand:9696	OCLACITINIB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	DNDI1417072	chembl:CHEMBL1310701	CHEMBL:CHEMBL1310701	FALSE	FALSE	FALSE
ATP7A	hgnc:869	ATP7A	NCI	14-Sep-17	NULL	0.1977690065374557	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	0.2500365296937833	HYDROXYUREA	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
PSMC2	hgnc:9548	PSMC2	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.1022876712383659	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q03181	hgnc:9235	PPARD	TdgClinicalTrial	Jan-14	NULL	0.7895890411382631	MBX-8025	chembl:CHEMBL3545019	MBX-8025	FALSE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6980	iuphar.ligand:6980	AZIDOPINE	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:11716	iuphar.ligand:11716	LONDAMOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:732	hgnc:1353	C8B	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:2821	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5554	iuphar.ligand:5554	O-ARACHIDONOYL ETHANOLAMINE	FALSE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:8312	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5628	iuphar.ligand:5628	[67GA]NODAGA-[TYR3]OCTREOTIDE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.015655239	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.017114626	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2134458180312784	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
STAT5B	hgnc:11367	STAT5B	DTC	9/2/20	NULL	1.500219178162699	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2225	iuphar.ligand:2225	D[PEN1,TYR(ME)2]AVP	FALSE	FALSE	FALSE
UNIPROT:P31785	hgnc:6010	IL2RG	TEND	1-Aug-11	NULL	1.750255707856483	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	OLVANIL	ncit:C166774	OLVANIL	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.6731752722524935	BELUMOSUDIL MESYLATE	rxcui:2565692	BELUMOSUDIL MESYLATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	0.750109589	Bopindolol	rxcui:19605	BOPINDOLOL	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:1213	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.023420014	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.1223955040459079	IUPHAR.LIGAND:3439	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.029090123	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:588	rxcui:83515	EPROSARTAN	TRUE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:9821	iuphar.ligand:9821	RO5508887	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.4487835148349957	4-HYDROPEROXYCYCLOPHOSPHAMIDE	ncit:C1423	PERFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.6886251965336985	NORGESTIMATE	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
DUX1	hgnc:3079	DUX1	PharmGKB	4/5/24	NULL	3.889457128569963	isoniazid	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.039778539	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.076765601	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.050007306	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.023420014	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2273059360852575	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1751	iuphar.ligand:1751	UP3U	FALSE	FALSE	FALSE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	1.009762908	MRX-4	iuphar.ligand:10796	CONTEZOLID ACEFOSAMIL (PARENT)	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.041508041	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.058733413	VALERIAN	rxcui:253206	VALERIAN ROOT EXTRACT	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.024896952	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
RRM2B	hgnc:17296	RRM2B	ChEMBL	33	inhibitor	0.7501095890813498	GALLIUM NITRATE	rxcui:25544	GALLIUM NITRATE	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TEND	1-Aug-11	NULL	0.056459862	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
5-HT 1B RECEPTOR	hgnc:5287	HTR1B	TTD	2020.06.01	NULL	0.926605963	Frovatriptan	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
EFNB2	hgnc:3227	EFNB2	ChEMBL	33	inhibitor	1.009762908	SEPHB4-HSA	drugbank:DB14797	SEPHB4-HSA	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	CancerCommons	25-Jul-13	inhibitor	0.6783936852156912	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	CancerCommons	25-Jul-13	inhibitor	0.082754407	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-703	chembl:CHEMBL609030	CHEMBL:CHEMBL609030	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CancerCommons	25-Jul-13	inhibitor	0.182318303	REOLYSIN	chembl:CHEMBL3545069	PELAREOREP	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	CGI	2/1/22	NULL	0.9590442234830044	AZD6738	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
DHRS9	hgnc:16888	DHRS9	DTC	9/2/20	NULL	15.00219178	PROTECTED SIPHONODICTYAL C	chembl:CHEMBL456845	PROTECTED SIPHONODICTYAL C	FALSE	FALSE	FALSE
BCL6	hgnc:1001	BCL6	CGI	2/1/22	NULL	4.375639269641208	Onalespib	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.056622219	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.056622219	Anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.026572708	Anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.012154554	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
IDH2	hgnc:5383	IDH2	CGI	2/1/22	NULL	5.469549087051511	AG-221	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
CRBN	hgnc:30185	CRBN	CGI	2/1/22	NULL	0.8975670296699916	Lenalidomide	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	0.192335792	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.546954909	BCL2 inhibitor	ncit:C159200	BCL-2 INHIBITOR	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.025003653	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
UNIPROT:P40238	hgnc:7217	MPL	TdgClinicalTrial	Jan-14	NULL	9.546849315580817	LGD-4665	ncit:C152703	TOTROMBOPAG	FALSE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	CGI	2/1/22	NULL	0.1666910197958555	Mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.013716738	DAUNORUBICIN HYDROCHLORIDE	rxcui:81992	DAUNORUBICIN HYDROCHLORIDE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.4526523382387456	ETOPOSIDE PHOSPHATE	rxcui:24614	ETOPOSIDE PHOSPHATE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2094720926955897	SCOPOLAMINE	rxcui:9601	SCOPOLAMINE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	BIPERIDEN LACTATE	rxcui:19377	BIPERIDEN LACTATE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.7160136986685613	LEVOBUNOLOL HYDROCHLORIDE	rxcui:1813	LEVOBUNOLOL	TRUE	FALSE	FALSE
UNIPROT:P07949	hgnc:9967	RET	TdgClinicalTrial	Jan-14	NULL	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
MPL	hgnc:7217	MPL	ChEMBL	33	agonist	2.983390411119005	ELTROMBOPAG OLAMINE	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	0.4861821410712453	TRICHLORMETHIAZIDE	rxcui:10772	TRICHLORMETHIAZIDE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.2456499239096818	ONDANSETRON	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
CASR	hgnc:1514	CASR	ChEMBL	33	positive modulator	1.640864726115453	CINACALCET HYDROCHLORIDE	rxcui:384379	CINACALCET HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	IMIPRAMINE PAMOATE	rxcui:91118	IMIPRAMINE PAMOATE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.2128689374420047	VILAZODONE HYDROCHLORIDE	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	SAXAGLIPTIN HYDROCHLORIDE	rxcui:1043560	SAXAGLIPTIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1171	hgnc:14679	SLC38A4	GuideToPharmacology	2024.1	NULL	5.250767124	IUPHAR.LIGAND:4542	rxcui:426	ALANINE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1124502911321247	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP PROMPT PURIFIED PORK	chembl:CHEMBL1201643	INSULIN ZINC SUSP PROMPT PURIFIED PORK	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	1.500219178	INSULIN GLARGINE	rxcui:2563969	INSULIN GLARGINE-YFGN	TRUE	FALSE	FALSE
MGAM	hgnc:7043	MGAM	ChEMBL	33	inhibitor	4.773424657790408	MIGLITOL	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:2163	iuphar.ligand:2163	S6716	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.3271505995993426	DEXMETHYLPHENIDATE HYDROCHLORIDE	rxcui:352372	DEXMETHYLPHENIDATE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.138178082	DIBUCAINE HYDROCHLORIDE	rxcui:235402	DIBUCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	ChEMBL	33	inhibitor	0.1141471113819445	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	1.640864726115453	ZICONOTIDE ACETATE	rxcui:486126	ZICONOTIDE ACETATE	TRUE	FALSE	FALSE
MMP8	hgnc:7175	MMP8	ChEMBL	33	inhibitor	0.326134604	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.074975256	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
MMP8	hgnc:7175	MMP8	ChEMBL	33	inhibitor	0.326134604	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.1356787370431382	ISOPROTERENOL SULFATE	rxcui:82031	ISOPROTERENOL SULFATE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	inhibitor	0.057700738	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.1848861663228679	GUANABENZ ACETATE	rxcui:227225	GUANABENZ ACETATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.093763699	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1093909817410302	OXAPROZIN	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.060772768	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
ABCC9	hgnc:60	ABCC9	ChEMBL	33	potentiator	1.193356164447602	PINACIDIL	rxcui:33717	PINACIDIL	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.068115956	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.096167896	METOCLOPRAMIDE HYDROCHLORIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
COL6A1	hgnc:2211	COL6A1	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL2A1	hgnc:2200	COL2A1	ChEMBL	33	cleavage	1.875273972703375	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
PSMB9	hgnc:9546	PSMB9	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB7	hgnc:9544	PSMB7	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.6250913242344582	PANCURONIUM BROMIDE	rxcui:7884	PANCURONIUM BROMIDE	TRUE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.015608701	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
EPHA6	hgnc:19296	EPHA6	ChEMBL	33	inhibitor	0.1810609352954982	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.3750547945406749	VECURONIUM BROMIDE	rxcui:11153	VECURONIUM BROMIDE	TRUE	FALSE	FALSE
NDUFB11	hgnc:20372	NDUFB11	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.028413242	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
ATP1B1	hgnc:804	ATP1B1	ChEMBL	33	inhibitor	0.145450613	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
ATP1B2	hgnc:805	ATP1B2	ChEMBL	33	inhibitor	0.4605936073306535	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
ATP1A2	hgnc:800	ATP1A2	ChEMBL	33	inhibitor	0.8334550989792778	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
FXYD2	hgnc:4026	FXYD2	ChEMBL	33	inhibitor	0.4861821410712454	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.030996264	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.021554873	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.068757317	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.070448575	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	agonist	0.035574303	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	agonist	0.037884323	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.078682824	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.073885091	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.072125922	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.081872668	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.058212496	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.030527716	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.019695301	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.022889133	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.019695301	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.032016873	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
BLK	hgnc:1057	BLK	ChEMBL	33	inhibitor	0.016236138	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	modulator	0.093763699	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	modulator	0.1458546423213736	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	ChEMBL	33	modulator	0.077217164	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	modulator	0.082043236	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	modulator	0.062509132	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	modulator	0.024767769	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNG3	hgnc:1407	CACNG3	ChEMBL	33	modulator	0.1458546423213736	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	modulator	0.031254566	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	modulator	0.030527716	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.054243462	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.07699072	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.062808219	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.020836377	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.016485925	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.070860555	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	ARTICAINE HYDROCHLORIDE	rxcui:2117	ARTICAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.070322774	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.040703621	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.040703621	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	inhibitor	0.150021918	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.066297565	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.1666910197958555	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.082171629	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.045226246	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.055563673	APOMORPHINE HYDROCHLORIDE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.025942525	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.4070362111294147	PARAMETHADIONE	rxcui:32894	PARAMETHADIONE	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	agonist	0.3671865121377238	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	2.080014029626545	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	agonist	0.3512218811752141	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	0.3125456621172291	MIBEFRADIL DIHYDROCHLORIDE	rxcui:83214	MIBEFRADIL DIHYDROCHLORIDE	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	modulator	8.353493151133215	LUMACAFTOR	rxcui:1655922	LUMACAFTOR	TRUE	FALSE	FALSE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	0.3125456621172291	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.4167275494896388	BAY-1082439	chembl:CHEMBL3545245	BAY-1082439	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.076765601	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	ChEMBL	33	inhibitor	0.2287915957982331	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	GSK-610677	chembl:CHEMBL3544968	GSK-610677	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	ChEMBL	33	inhibitor	0.056097939	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.2917092846427472	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.091636424	LY-3009120	chembl:CHEMBL3545195	LY-3009120	FALSE	FALSE	FALSE
NDUFA4	hgnc:7687	NDUFA4	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFA11	hgnc:20371	NDUFA11	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFS7	hgnc:7714	NDUFS7	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFV2	hgnc:7717	NDUFV2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFS1	hgnc:7707	NDUFS1	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFA5	hgnc:7688	NDUFA5	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB11	hgnc:20372	NDUFB11	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFAF2	hgnc:28086	NDUFAF2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB3	hgnc:7698	NDUFB3	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFB8	hgnc:7703	NDUFB8	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFS1	hgnc:7707	NDUFS1	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.2590839041234926	TUCATINIB	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
NDUFB1	hgnc:7695	NDUFB1	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFV1	hgnc:7716	NDUFV1	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	TAK-285	chembl:CHEMBL1614725	TAK-285	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inverse agonist	1.009762908	TEMANOGREL	ncit:C96894	TEMANOGREL	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.3889457128569963	XL-418	chembl:CHEMBL2016893	XL-418	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	1.280674908	PHE377	chembl:CHEMBL3545148	PHE377	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.037884323	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	ChEMBL	33	inhibitor	0.1286952726365061	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PRKD1	hgnc:9407	PRKD1	ChEMBL	33	inhibitor	0.3088686543276147	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	ChEMBL	33	inhibitor	0.07182992	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.025256215	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	ChEMBL	33	inhibitor	0.1342907192728759	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	ChEMBL	33	inhibitor	0.2573905452730122	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
TTK	hgnc:12401	TTK	ChEMBL	33	inhibitor	5.834185692854944	BAY-1217389	iuphar.ligand:12705	BAY1217389	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	0.2287915957982331	AC-201	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.1470803115845784	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
MAP3K1	hgnc:6848	MAP3K1	ChEMBL	33	inhibitor	2.917092846427472	E-6201	drugbank:DB11687	E-6201	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.061737415	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.2991890098899972	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
CXCR2	hgnc:6027	CXCR2	ChEMBL	33	modulator	1.458546423213736	LADARIXIN	ncit:C170087	LADARIXIN	FALSE	FALSE	FALSE
KRT20	hgnc:20412	KRT20	NCI	14-Sep-17	NULL	0.3621218705909965	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
MC3R	hgnc:6931	MC3R	ChEMBL	33	agonist	26.25383561784724	MODIMELANOTIDE	ncit:C175147	MODIMELANOTIDE	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.6731752722524935	RISLENEMDAZ	ncit:C152228	RISLENEMDAZ	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	blocker	0.5556367326528517	LANICEMINE	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	2.282942227638891	ABT-126	chembl:CHEMBL3545231	ABT-126	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.6250913242344582	VIXOTRIGINE	ncit:C152899	VIXOTRIGINE	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	positive modulator	10.74020548002842	TEZACAFTOR	rxcui:1999382	TEZACAFTOR	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.064347636	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	AMA0076	chembl:CHEMBL3545073	AMA0076	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	positive modulator	0.596678082	MIBAMPATOR	ncit:C174617	MIBAMPATOR	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	agonist	0.039068208	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	inverse agonist	0.042073455	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	inverse agonist	0.039068208	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.2083637747448194	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.021751314	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.9907107780319716	CUDRAFLAVONE B	chembl:CHEMBL221907	CUDRAFLAVONE B	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	ChEMBL	33	activator	1.875273972703375	SERELAXIN	ncit:C152342	SERELAXIN	FALSE	FALSE	FALSE
TRAC	hgnc:12029	TRAC	ChEMBL	33	inhibitor	3.281729452230906	MEDI-500	chembl:CHEMBL2109592	MEDI-500	FALSE	FALSE	FALSE
RYANODINE RECEPTOR	hgnc:10483	RYR1	TTD	2020.06.01	NULL	2.083637747448194	Dantrolene	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
IFNLR1	hgnc:18584	IFNLR1	ChEMBL	33	agonist	17.50255707856483	PEGINTERFERON LAMBDA-1A	ncit:C166435	PEGINTERFERON LAMBDA-1A	FALSE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	ChEMBL	33	inhibitor	0.077217164	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
FABP1	hgnc:3555	FABP1	NCI	14-Sep-17	NULL	0.1077448794166097	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
XPNPEP3	hgnc:28052	XPNPEP3	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	CIViC	10-Apr-24	NULL	0.086219493	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
METAP1D	hgnc:32583	METAP1D	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PSMB7	hgnc:9544	PSMB7	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMB11	hgnc:31963	PSMB11	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMB10	hgnc:9538	PSMB10	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	1.750255707856483	NESVACUMAB	ncit:C95712	NESVACUMAB	FALSE	FALSE	FALSE
IL4	hgnc:6014	IL4	ChEMBL	33	inhibitor	21.00306849427779	PASCOLIZUMAB	ncit:C88618	PASCOLIZUMAB	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.2822993077187876	ABBV-257	chembl:CHEMBL4297682	ABBV-257	FALSE	FALSE	FALSE
LTA	hgnc:6709	LTA	ChEMBL	33	inhibitor	13.12691780892362	PATECLIZUMAB	ncit:C174894	PATECLIZUMAB	FALSE	FALSE	FALSE
EGFL7	hgnc:20594	EGFL7	ChEMBL	33	inhibitor	35.00511415712966	PARSATUZUMAB	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.1491695205559502	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	binder	2.059124362184098	LMB-2	chembl:CHEMBL2109367	LMB-2	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	ChEMBL	33	inhibitor	0.6035364509849942	ROVELIZUMAB	ncit:C152264	ROVELIZUMAB	FALSE	FALSE	FALSE
FN1	hgnc:3778	FN1	ChEMBL	33	other/unknown	4.039051633514961	L19SIP 131I	chembl:CHEMBL2109412	L19SIP 131I	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	1.193356164447602	NAVEGLITAZAR	ncit:C75191	NAVEGLITAZAR	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	ChEMBL	33	inhibitor	2.625383561784724	SCH-708980	chembl:CHEMBL2109460	SCH-708980	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.041739007	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.1988926940746003	DILEVALOL HYDROCHLORIDE	ncit:C174786	DILEVALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
CDK19	hgnc:19338	CDK19	ChEMBL	33	inhibitor	0.1250182648468916	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	FENCLOFENAC	ncit:C65643	FENCLOFENAC	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.4773424657790409	LUMIRACOXIB	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	ENCAINIDE HYDROCHLORIDE	rxcui:281189	ENCAINIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADH7	hgnc:256	ADH7	ChEMBL	33	inhibitor	3.750547945406749	NITREFAZOLE	ncit:C72626	NITREFAZOLE	TRUE	FALSE	FALSE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12267	iuphar.ligand:12267	LLL12	FALSE	FALSE	FALSE
ADH4	hgnc:252	ADH4	ChEMBL	33	inhibitor	0.6250913242344582	NITREFAZOLE	ncit:C72626	NITREFAZOLE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	1.514644363	VANUCIZUMAB	ncit:C118578	VANUCIZUMAB	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.9546849315580818	EMACTUZUMAB	ncit:C125548	EMACTUZUMAB	FALSE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	ChEMBL	33	agonist	1.250182648468916	ARGIPRESSIN TANNATE	ncit:C166779	ARGIPRESSIN TANNATE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.061055432	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.080656945	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	blocker	0.1881995384791917	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	0.070574827	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	blocker	0.130291988	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	blocker	0.1881995384791917	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	ChEMBL	33	inhibitor	1.029562181092049	CDP-484	chembl:CHEMBL2109459	CDP-484	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	2.187819634820604	HUPAM4	chembl:CHEMBL2109365	HUPAM4	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.050879526	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.056826484	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	ChEMBL	33	blocker	0.003648646	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	ChEMBL	33	blocker	0.091476779	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	1.591141552596803	ELAGOLIX SODIUM	rxcui:2049847	ELAGOLIX SODIUM	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
RARB	hgnc:9865	RARB	ChEMBL	33	agonist	2.059124362184097	TAMIBAROTENE	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.037213091	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	1,5-ISOQUINOLINEDIOL	chembl:CHEMBL338314	CHEMBL:CHEMBL338314	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	MANIDIPINE 6300	rxcui:29275	MANIDIPINE	FALSE	FALSE	FALSE
NPTN	hgnc:17867	NPTN	NCI	14-Sep-17	NULL	17.50255707856483	GP100	ncit:C2386	GP100 ANTIGEN	FALSE	FALSE	FALSE
C1S	hgnc:1247	C1S	ChEMBL	33	inhibitor	1.312691780892362	HUMAN C1-ESTERASE INHIBITOR	ncit:C87730	HUMAN C1-ESTERASE INHIBITOR	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.9053046764774912	GEPOTIDACIN	ncit:C170025	GEPOTIDACIN	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	0.9723642821424906	ODRONEXTAMAB	ncit:C119615	ODRONEXTAMAB	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.1116392726485354	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.1103102336884338	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	ChEMBL	33	inhibitor	2.763561643983921	MARSTACIMAB	ncit:C166436	MARSTACIMAB	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.3125456621172291	GSK-256066	drugbank:DB12137	GSK-256066	FALSE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	NCI	14-Sep-17	NULL	0.172722603	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	ChEMBL	33	inhibitor	1.531473744374423	NAVTEMADLIN	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	1.166837138570988	OGLEMILAST	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	ChEMBL	33	inhibitor	0.1352294697019358	NAVTEMADLIN	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
RPS27	hgnc:10416	RPS27	ChEMBL	33	modulator	0.093763699	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL15	hgnc:10306	RPL15	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL5	hgnc:10360	RPL5	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL6	hgnc:10362	RPL6	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.018193926	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
GPR84	hgnc:4535	GPR84	ChEMBL	33	negative modulator	26.25383561784724	GLPG-1205	drugbank:DB15346	GLPG-1205	FALSE	FALSE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	inhibitor	2.187819634820604	SGS-742	drugbank:DB05010	SGS-742	FALSE	FALSE	FALSE
EIF2AK4	hgnc:19687	EIF2AK4	PharmGKB	4/5/24	NULL	0.2612321952024601	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	ChEMBL	33	inhibitor	7.501095891	BIMEKIZUMAB	rxcui:2668041	BIMEKIZUMAB	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.5707355569097228	BIIB021	drugbank:DB12359	BIIB021	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.1810609352954982	BIIB021	drugbank:DB12359	BIIB021	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.2536602475154323	BUNAZOSIN	rxcui:19850	BUNAZOSIN	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.6482428547616604	AMITIFADINE	ncit:C169780	AMITIFADINE	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.3977853881492006	AMITIFADINE	ncit:C169780	AMITIFADINE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:405	drugbank:DB08770	4-{2-[(7-AMINO-2-FURAN-2-YL[1,2,4]TRIAZOLO[1,5-A][1,3,5]TRIAZIN-5-YL)AMINO]ETHYL}PHENOL	FALSE	FALSE	FALSE
GPR119	hgnc:19060	GPR119	ChEMBL	33	agonist	8.751278539282415	GSK-1292263	drugbank:DB12627	GSK-1292263	FALSE	FALSE	FALSE
DLL3	hgnc:2909	DLL3	ChEMBL	33	binder	78.76150685354175	ROVALPITUZUMAB TESIRINE	ncit:C107678	ROVALPITUZUMAB TESIRINE	FALSE	FALSE	TRUE
NCBIGENE:66	hgnc:139	ACTBP6	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:3657	iuphar.ligand:3657	[125I]CCL25 (HUMAN)	FALSE	FALSE	FALSE
KIF11	hgnc:6388	KIF11	ChEMBL	33	inhibitor	9.845188356692718	FILANESIB	ncit:C68937	FILANESIB	FALSE	FALSE	TRUE
TNFRSF4	hgnc:11918	TNFRSF4	ChEMBL	33	inhibitor	3.500511415712966	TELAZORLIMAB	ncit:C175859	TELAZORLIMAB	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.2692701089009974	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
IMPDH2	hgnc:6053	IMPDH2	ChEMBL	33	inhibitor	5.250767123569449	AVN-944	drugbank:DB05500	AVN-944	FALSE	FALSE	FALSE
PSMA5	hgnc:9534	PSMA5	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
LAG3	hgnc:6476	LAG3	ChEMBL	33	inhibitor	6.563458904461812	MK-4280	chembl:CHEMBL4297784	MK-4280	FALSE	FALSE	FALSE
KIR3DL2	hgnc:6339	KIR3DL2	ChEMBL	33	inhibitor	26.25383561784724	LACUTAMAB	ncit:C124999	LACUTAMAB	FALSE	FALSE	FALSE
AKR1B1	hgnc:381	AKR1B1	ChEMBL	33	inhibitor	0.8078103267029924	SORBINIL	ncit:C97357	SORBINIL	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	ChEMBL	33	inhibitor	0.1389091831632129	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
TFRC	hgnc:11763	TFRC	ChEMBL	33	binder	8.751278539282415	PABINAFUSP ALFA	ncit:C170281	PABINAFUSP ALFA	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	CLN-081	iuphar.ligand:11889	ZIPALERTINIB	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013887244	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
CYP3A7	hgnc:2640	CYP3A7	ChEMBL	33	inhibitor	0.1389091831632129	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	4.039051633514961	TAFOLECIMAB	ncit:C171839	TAFOLECIMAB	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.2019525816757481	SARPOGRELATE	ncit:C73158	SARPOGRELATE	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	ChEMBL	33	inhibitor	2.282942227638891	COFORMYCIN	chembl:CHEMBL284483	COFORMYCIN	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.052824619	AEE788	iuphar.ligand:7643	AEE788	FALSE	FALSE	TRUE
GIPR	hgnc:4271	GIPR	ChEMBL	33	agonist	4.375639269641208	TIRZEPATIDE	rxcui:2601723	TIRZEPATIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.091159151	BUCINDOLOL HYDROCHLORIDE	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
EGLN2	hgnc:14660	EGLN2	ChEMBL	33	inhibitor	2.100306849	MOLIDUSTAT	rxcui:2637535	MOLIDUSTAT	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	1.111273465305703	MOBOCERTINIB	rxcui:2570736	MOBOCERTINIB	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
ALCAM	hgnc:400	ALCAM	ChEMBL	33	binder	0.084146909	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	ODRONEXTAMAB	ncit:C119615	ODRONEXTAMAB	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
CFLAR	hgnc:1876	CFLAR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.064984742	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PRKAG2	hgnc:9386	PRKAG2	ChEMBL	33	activator	1.875273972703374	ACADESINE	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.1810609352954983	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	ChEMBL	33	activator	0.031479419	OMAVELOXOLONE	rxcui:2631931	OMAVELOXOLONE	TRUE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	ChEMBL	33	inhibitor	0.5147810905460244	BAZLITORAN	ncit:C114975	BAZLITORAN	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.014617949	IUPHAR.LIGAND:2199	ncit:C80380	SATAVAPTAN	FALSE	FALSE	FALSE
SOAT2	hgnc:11178	SOAT2	ChEMBL	33	inhibitor	17.50255707856483	PACTIMIBE	ncit:C66290	PACTIMIBE	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC, EXTENDED	chembl:CHEMBL2108492	INSULIN ZINC, EXTENDED	TRUE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	inhibitor	0.8751278539282416	ENPATORAN	ncit:C177069	ENPATORAN	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.1093909817410302	TALETRECTINIB	ncit:C118948	TALETRECTINIB	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3509871071904712	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1100789753368857	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.088866948	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1374546367426557	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.4948366922735607	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.546954909	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1367387271762877	PD-325901	iuphar.ligand:7935	MIRDAMETINIB	FALSE	FALSE	TRUE
NF1	hgnc:7765	NF1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.5707355569097228	PD-325901	iuphar.ligand:7935	MIRDAMETINIB	FALSE	FALSE	TRUE
NF1	hgnc:7765	NF1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2282942227638891	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.012026494	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.182318303	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
AKT2	hgnc:392	AKT2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.7778914257139926	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
TEK	hgnc:11724	TEK	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1491695205559502	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	DTC	9/2/20	NULL	0.4118248724368196	DIMETHYLCURCUMIN	drugbank:DB06133	DIMETHYLCURCUMIN	FALSE	FALSE	FALSE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.041214813	NVP-BEZ241	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.039420174	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.014369915	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.017456008	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1280674908187671	GAMMA-INTERFERON	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.059532507	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
UNIPROT:P05106	hgnc:6156	ITGB3	TEND	1-Aug-11	NULL	2.800409132570373	TIROFIBAN	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
SLC29A4	hgnc:23097	SLC29A4	DTC	9/2/20	NULL	4.039051633514962	HISTAMINE	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	PYRIMETHAMINE	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	inhibitor	0.025739055	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	DNDI1417025	chembl:CHEMBL1320453	CHEMBL:CHEMBL1320453	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.2853677784548614	VX-745	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	BENZYL ISOTHIOCYANATE	drugbank:DB16860	BENZYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.022789788	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.020117882	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	L-750667	iuphar.ligand:978	L-750,667	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.029170928	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	APIOL	chembl:CHEMBL1560118	APIOL	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.3070624048871023	TCMDC-125536	chembl:CHEMBL528463	CHEMBL:CHEMBL528463	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.008310806	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	CLOPERASTINE HYDROCLORIDE	chembl:CHEMBL1492516	CLOPERASTINE HYDROCLORIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	TCMDC-125756	chembl:CHEMBL536599	CHEMBL:CHEMBL536599	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	CHLOROTRIANISENE	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	SJ000067611	chembl:CHEMBL602126	CHEMBL:CHEMBL602126	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	NIALAMIDE	rxcui:7394	NIALAMIDE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	1,2-DIMETHOXY-ANTHRAQUINONE	chembl:CHEMBL52884	CHEMBL:CHEMBL52884	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	PENTOSALEN	ncit:C63672	PENTOSALEN	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.037884323	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.072026984	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.073643298	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.002590157	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.5707355569097228	2,4-DINITRO-PHENYLAMINE	chembl:CHEMBL354318	CHEMBL:CHEMBL354318	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.0065923	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	5-NITROQUINOLINE	chembl:CHEMBL164449	CHEMBL:CHEMBL164449	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	CHLORPYRIFOS	ncit:C163641	CHLORPYRIFOS	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	3.889457128569962	(S)-FTY720P	chembl:CHEMBL1213480	(S)-FTY720P	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1112450661773188	CIPROFIBRATE	rxcui:21149	CIPROFIBRATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	CHRYSOPHANOL	chembl:CHEMBL41092	CHRYSOPHANOL	FALSE	FALSE	FALSE
HEXA	hgnc:4878	HEXA	DTC	9/2/20	NULL	2.864054794674245	PYRIMETHAMINE	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	NSC-36398	chembl:CHEMBL483206	CHEMBL:CHEMBL483206	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GYKI-52895	chembl:CHEMBL1256984	CHEMBL:CHEMBL1256984	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.014537008	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	DTC	9/2/20	NULL	0.4227670791923872	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	DTC	9/2/20	NULL	0.3571950424196904	MEMANTINE	rxcui:236685	MEMANTINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.082171629	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	TCMDC-124059	chembl:CHEMBL530733	CHEMBL:CHEMBL530733	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	1.019566431761058	AMMONIA SOLUTION, STRONG	chembl:CHEMBL1160819	AMMONIA SOLUTION, STRONG	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	inhibitor	0.024767769	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.022632617	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1415301111474245	GNF-PF-2335	chembl:CHEMBL601146	CHEMBL:CHEMBL601146	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	HYDROXYSTILBAMIDINE ISETHIONATE	ncit:C65871	HYDROXYSTILBAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	1.141471113819445	3-EPI-ISOCUCURBITACIN D	chembl:CHEMBL2022241	CHEMBL:CHEMBL2022241	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.008511537	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.066297565	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	OXYQUINOLINE SULFATE	rxcui:42836	OXYQUINOLINE SULFATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	CAULIBUGULONE C	chembl:CHEMBL445969	CAULIBUGULONE C	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	QUINOLIN-6-YLAMINE	chembl:CHEMBL99408	CHEMBL:CHEMBL99408	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.2811655755592744	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	HISTIDINE	rxcui:5340	HISTIDINE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.078958904	ENCLOMIPHENE	ncit:C28211	ENCLOMIPHENE	FALSE	FALSE	FALSE
STK38L	hgnc:17848	STK38L	DTC	9/2/20	inhibitor	1.312691780892362	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	MONTELUKAST	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.099071078	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.084963869	TANSHINONE IIA SULFONATE	chembl:CHEMBL1473252	TANSHINONE IIA SULFONATE	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	PINORESINOL	chembl:CHEMBL487611	PINORESINOL	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.046221542	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.051177067	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	SERICETIN DIACETATE	chembl:CHEMBL1594132	SERICETIN DIACETATE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006940869	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TDR77582	chembl:CHEMBL1329349	CHEMBL:CHEMBL1329349	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.087952548	MUNDULONE ACETATE	chembl:CHEMBL1372368	MUNDULONE ACETATE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IIIE	chembl:CHEMBL1095027	AESCULIOSIDE IIIE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.029766254	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	BERGAPTOL	chembl:CHEMBL242711	BERGAPTOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	SJ000002502	chembl:CHEMBL591630	CHEMBL:CHEMBL591630	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	GNF-PF-1319	chembl:CHEMBL235891	CHEMBL:CHEMBL235891	FALSE	FALSE	FALSE
BRDT	hgnc:1105	BRDT	DTC	9/2/20	NULL	0.2083637747448194	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	1.875273972703374	MG-132	iuphar.ligand:8616	MG-132	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001067099	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	LAVENDUSTIN C	ncit:C1487	LAVENDUSTIN C	FALSE	FALSE	FALSE
PTPN6	hgnc:9658	PTPN6	DTC	9/2/20	NULL	0.1535312024435511	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.033903258	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	PHENELZINE SULFATE	rxcui:8124	PHENELZINE SULFATE	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.011399842	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.08334551	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.3962843112127887	SORBINIL	ncit:C97357	SORBINIL	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.014369915	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002188184	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.026837552	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	ACTINONIN	drugbank:DB04310	2-[(FORMYL-HYDROXY-AMINO)-METHYL]-HEPTANOIC ACID [1-(2-HYDROXYMETHYL-PYRROLIDINE-1-CARBONYL)-2-METHYL-PROPYL]-AMIDE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.1450488155682168	GNF-PF-4791	chembl:CHEMBL583555	CHEMBL:CHEMBL583555	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.085796848	SCH-23390	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.2323348284765243	TCMDC-125454	chembl:CHEMBL535714	CHEMBL:CHEMBL535714	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	GNF-PF-840	chembl:CHEMBL601605	CHEMBL:CHEMBL601605	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.2678962818147678	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.00333997	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.049770304	PHENYLSTIBONIC ACID	chembl:CHEMBL1369257	PHENYLSTIBONIC ACID	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.010966514	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.029301156	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.038894571	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.091159151	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW434756X	chembl:CHEMBL485745	GW434756X	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	BETANAPHTHOL	ncit:C81517	BETANAPHTHOL	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1041818873724097	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.020257589	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.030688294	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.039068208	WB-4101	iuphar.ligand:499	WB 4101	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	GNF-PF-3501	chembl:CHEMBL581910	CHEMBL:CHEMBL581910	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003703461	PIOGLITAZONE HYDROCHLORIDE	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.045461187	SJ000001592	chembl:CHEMBL591834	CHEMBL:CHEMBL591834	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006054153	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	BENZOTHIAZYL DISULFIDE	chembl:CHEMBL508112	BENZOTHIAZYL DISULFIDE	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	inhibitor	0.027347745	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	NARINGIN	rxcui:31538	NARINGIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.028977744	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	TCMDC-125465	chembl:CHEMBL536151	CHEMBL:CHEMBL536151	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DEXBROMPHENIRAMINE	rxcui:1767	BROMPHENIRAMINE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.006596441	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	KANZONOL W	chembl:CHEMBL591772	KANZONOL W	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.04321619	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	GLUTARAL	rxcui:4888	GLUTARAL	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.4375639269641208	4-HYDROXYEVODIAMINE	chembl:CHEMBL2171794	CHEMBL:CHEMBL2171794	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	MONASTROL	drugbank:DB04331	MONASTROL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00299804	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	GNF-PF-1399	chembl:CHEMBL578504	CHEMBL:CHEMBL578504	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	GNF-PF-4798	chembl:CHEMBL584635	CHEMBL:CHEMBL584635	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	chembl:CHEMBL284028	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.046673486	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.029531874	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004287741	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	BENZOTHIAZOLE-2,6-DIAMINE	chembl:CHEMBL328540	CHEMBL:CHEMBL328540	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004937716	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1810609352954982	CHLOROETHYLCLONIDINE	chembl:CHEMBL326967	CHLOROETHYLCLONIDINE	FALSE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.4339476961627644	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.042379073	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.001538551	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SALSOLINOL HYDROBROMIDE	chembl:CHEMBL553751	SALSOLINOL HYDROBROMIDE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.061773731	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
FPR1	hgnc:3826	FPR1	DTC	9/2/20	NULL	3.500511415712966	AG-14	iuphar.ligand:5835	AG-14	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	FTI-277	chembl:CHEMBL135561	CHEMBL:CHEMBL135561	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006113363	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.025147352	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	BENZO[B]FLUORANTHENE	chembl:CHEMBL1337502	BENZO[B]FLUORANTHENE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV667489	chembl:CHEMBL2028066	CHEMBL:CHEMBL2028066	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	TANSHINONE IIA SULFONATE	chembl:CHEMBL1473252	TANSHINONE IIA SULFONATE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.039214094	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.108040476	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DL-CATECHIN TRIHYDRATE	chembl:CHEMBL1172228	CHEMBL:CHEMBL1172228	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PIPOXOLAN HYDROCHLORIDE	rxcui:235861	PIPOXOLAN HYDROCHLORIDE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	HISTAMINE	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.546954909	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.364636606	2-CINNAMAMIDOBENZAMIDE	chembl:CHEMBL1522743	CHEMBL:CHEMBL1522743	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.1041818873724097	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.42006137	HYDROXYSTILBAMIDINE ISETHIONATE	ncit:C65871	HYDROXYSTILBAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2580229544751573	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2220197515251353	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2447910080918158	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2580229544751573	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	4-(4-CHLOROPHENOXY)ANILINE	chembl:CHEMBL1521156	CHEMBL:CHEMBL1521156	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	3-HYDROXYBENZYLHYDRAZINE DIHYDROCHLORIDE	iuphar.ligand:5116	3-HYDROXYBENZYLHYDRAZINE	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.5834185692854944	8-BROMO-CAMP SODIUM	chembl:CHEMBL1256796	CHEMBL:CHEMBL1256796	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002784371	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	2.500365296937833	CINNAMIC ACID HYDROXAMATE	chembl:CHEMBL237370	CINNAMIC ACID HYDROXAMATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006419031	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1367387271762877	APOCIDEINE	chembl:CHEMBL154709	APOCIDEINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	HOMOVANILLIC ACID	chembl:CHEMBL1562	HOMOVANILLIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	TCMDC-124479	chembl:CHEMBL587259	CHEMBL:CHEMBL587259	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	SJ000082805	chembl:CHEMBL531043	CHEMBL:CHEMBL531043	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	CORYNANTHEINE	iuphar.ligand:5345	CORYNANTHINE	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.7955707762984014	4-(4-CHLOROPHENOXY)ANILINE	chembl:CHEMBL1521156	CHEMBL:CHEMBL1521156	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	5,7-DIMETHOXYISOFLAVONE	chembl:CHEMBL308688	5,7-DIMETHOXYISOFLAVONE	FALSE	FALSE	FALSE
PLAT	hgnc:9051	PLAT	DTC	9/2/20	NULL	0.1110098757625676	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.05664258	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.03233231	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	GNF-PF-4384	chembl:CHEMBL602763	CHEMBL:CHEMBL602763	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	1-BENZYLMALEIMIDE	chembl:CHEMBL388979	CHEMBL:CHEMBL388979	FALSE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.546954909	NORGESTREL	rxcui:7518	NORGESTREL	TRUE	FALSE	FALSE
PSMB7	hgnc:9544	PSMB7	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB9	hgnc:9546	PSMB9	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB4	hgnc:9541	PSMB4	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	0.1878628666751144	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD4	hgnc:9561	PSMD4	DTC	9/2/20	NULL	0.3488881809680698	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD8	hgnc:9566	PSMD8	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.009430257	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.182318303	JNK INHIBITOR VIII	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.1136529680426287	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.4375639269641208	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	2.838252499226729	PARGYLINE	rxcui:7930	PARGYLINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	PIRETANIDE	rxcui:33770	PIRETANIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005448974	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	CHLORPYRIFOS	ncit:C163641	CHLORPYRIFOS	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.059163573	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	TPKI-24	iuphar.ligand:9403	RO3280	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.044535769	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.077444943	SJ000024939	chembl:CHEMBL590691	CHEMBL:CHEMBL590691	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	TCMDC-123600	chembl:CHEMBL531296	CHEMBL:CHEMBL531296	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00095957	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005308631	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002678689	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	NILE RED	chembl:CHEMBL144472	NILE RED	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	PANTOPRAZOLE	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002622106	AMITRIPTYLINE HYDROCHLORIDE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	SB-334867	iuphar.ligand:1703	SB-334867	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.7242437411819931	MANASSANTIN B	chembl:CHEMBL461308	MANASSANTIN B	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	inhibitor	0.041021618	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.6604738520213144	KAEMPFERIDE	chembl:CHEMBL40919	KAEMPFERIDE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.108711535	ETHOPROPAZINE HYDROCHLORIDE	rxcui:6541	ETHOPROPAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.089298761	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	SB-334867	iuphar.ligand:1703	SB-334867	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	OXOPURPUREINE	chembl:CHEMBL456295	OXOPURPUREINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	ESOXYBUTYNIN	ncit:C166661	ESOXYBUTYNIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.027929612	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	4,4'-DITHIODIPYRIDINE	chembl:CHEMBL1232076	CHEMBL:CHEMBL1232076	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.027752469	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.021554873	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	PICOTAMIDE	ncit:C73157	PICOTAMIDE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.021309932	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.021189536	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	KOJIC ACID	rxcui:1426451	KOJIC ACID	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	NSC-747266	chembl:CHEMBL609570	CHEMBL:CHEMBL609570	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	inhibitor	0.019592415	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004458114	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	NSC-45382	chembl:CHEMBL1214274	CHEMBL:CHEMBL1214274	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SJ000201788	chembl:CHEMBL602923	CHEMBL:CHEMBL602923	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.033615667	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	NSC-125034	chembl:CHEMBL239439	CHEMBL:CHEMBL239439	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
F11	hgnc:3529	F11	DTC	9/2/20	NULL	5.527123287967842	SULFATED PENTAGALLOYLGLUCOSIDE	chembl:CHEMBL2314388	SULFATED PENTAGALLOYLGLUCOSIDE	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.010012905	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.210030685	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.1116392726485354	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.108711535	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	chembl:CHEMBL1333512	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.1103102336884338	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1296485709523321	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1773907812016706	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	1.944728564284981	LORGLUMIDE SODIUM	chembl:CHEMBL1255589	LORGLUMIDE SODIUM	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.021805511	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.074797252	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	SJ000044417	chembl:CHEMBL609438	CHEMBL:CHEMBL609438	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.011603905	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	TCMDC-125103	chembl:CHEMBL530281	CHEMBL:CHEMBL530281	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.028708404	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CALMODULIN	hgnc:14986	SNAP91	TTD	2020.06.01	NULL	8.751278539282415	Halofantrine	rxcui:50749	HALOFANTRINE	FALSE	FALSE	FALSE
SF3B2	hgnc:10769	SF3B2	DTC	9/2/20	NULL	35.00511415712966	SPLICEOSTATIN-A	chembl:CHEMBL1221944	CHEMBL:CHEMBL1221944	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.9907107780319716	GNF-PF-4867	chembl:CHEMBL583997	CHEMBL:CHEMBL583997	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	1.193356164447602	DIHYDRODAPHNODORIN B	chembl:CHEMBL1532097	DIHYDRODAPHNODORIN B	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	BUTOCONAZOLE NITRATE	rxcui:19884	BUTOCONAZOLE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.003316134	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	2.019525817	BERKELEYACETAL A	chembl:CHEMBL252920	BERKELEYACETAL A	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	HTS-05057	chembl:CHEMBL372629	CHEMBL:CHEMBL372629	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1483267549030917	R(-)-APOCODEINE HCL	chembl:CHEMBL1256735	CHEMBL:CHEMBL1256735	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.2172731223545979	NOVOBIOCIN	rxcui:7538	NOVOBIOCIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	TCMDC-123762	chembl:CHEMBL547483	CHEMBL:CHEMBL547483	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.060492709	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.031254566	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	MAPROTILINE HYDROCHLORIDE	rxcui:203126	MAPROTILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.063568609	N,N-HEXAMETHYLENEAMILORIDE	iuphar.ligand:1192	5-(N,N-HEXAMETHYLENE)-AMILORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	SJ000114961	chembl:CHEMBL590168	CHEMBL:CHEMBL590168	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000673287	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.182318303	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	IPCONAZOLE	chembl:CHEMBL3185422	IPCONAZOLE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	CALANOLIDE A	drugbank:DB04886	CALANOLIDE A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	OXYPHENISATINE	rxcui:8136	OXYPHENISATIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	SJ000112730	chembl:CHEMBL591178	CHEMBL:CHEMBL591178	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009922085	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.7001022831425933	DEMETON S	chembl:CHEMBL1900921	DEMETON S	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	TDR77585	chembl:CHEMBL1333386	CHEMBL:CHEMBL1333386	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.007244436	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.020819854	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.082559232	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	GUANFACINE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.001999911	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.128537751	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	2.282942227638891	KRM-189	chembl:CHEMBL449063	CHEMBL:CHEMBL449063	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004172574	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	MAGNOLOL	rxcui:2562549	MAGNOLOL	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	chembl:CHEMBL1449651	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.018619742	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.00218782	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.005632662	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	4-((2-PHENETHYLPHENOXY)METHYL)PYRIDINE	chembl:CHEMBL270688	CHEMBL:CHEMBL270688	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	DTC	9/2/20	NULL	0.6819178082557726	KERACYANIN	rxcui:28165	KERACYANIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	PHENYLSTIBONIC ACID	chembl:CHEMBL1369257	PHENYLSTIBONIC ACID	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.003979361	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005483257	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TCMDC-124681	chembl:CHEMBL536008	CHEMBL:CHEMBL536008	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1000146118775133	XANTHOHUMOL	ncit:C121950	XANTHOHUMOL	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.046881849	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	QUININE SULFATE	rxcui:9071	QUININE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.0135995	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
NECTIN4	hgnc:19688	NECTIN4	PharmGKB	4/5/24	NULL	1.029562181092049	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	DIBENZOYLMETHANE	chembl:CHEMBL371523	DIBENZOYLMETHANE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	TRICITRINOL B	chembl:CHEMBL1822982	TRICITRINOL B	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.004542186	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TOCOPHEROL ACETATE	rxcui:1046243	ALPHA-TOCOPHEROL ACETATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TRICHLORMETHINE	ncit:C161524	NITROGEN MUSTARD HN-3	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	NILE RED	chembl:CHEMBL144472	NILE RED	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.002955515	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
SPHK1	hgnc:11240	SPHK1	DTC	9/2/20	NULL	8.751278539282415	DIMETHYLSPINGOSINE	chembl:CHEMBL322333	DIMETHYLSPINGOSINE	FALSE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.5357925636295356	FACTOR VIII	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1023541349623674	CUMENE HYDROPEROXIDE	chembl:CHEMBL1518369	CUMENE HYDROPEROXIDE	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.1909369863116163	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.027177884	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	inhibitor	0.016408647	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	TRIFLUPROMAZINE HYDROCHLORIDE	rxcui:91125	TRIFLUPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.055563673	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	ETHOPROPAZINE HYDROCHLORIDE	rxcui:6541	ETHOPROPAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	DICHLON	chembl:CHEMBL318782	DICHLON	FALSE	FALSE	FALSE
IDO1	hgnc:6059	IDO1	DTC	9/2/20	NULL	3.750547945	PHENYLHYDRAZINE	rxcui:8167	PHENYLHYDRAZINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	OXOTREMORINE	iuphar.ligand:302	OXOTREMORINE	FALSE	FALSE	FALSE
TXN2	hgnc:17772	TXN2	DTC	9/2/20	NULL	17.50255707856483	GAMBOGENIC ACID	chembl:CHEMBL2205166	GAMBOGENIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV396635	chembl:CHEMBL2028045	CHEMBL:CHEMBL2028045	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.016485925	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.042276708	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	TANSHINONE IIA SULFONATE	chembl:CHEMBL1473252	TANSHINONE IIA SULFONATE	FALSE	FALSE	FALSE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
STK10	hgnc:11388	STK10	DTC	9/2/20	inhibitor	0.4375639269641209	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	1.750255707856483	AZD-1480	drugbank:DB12588	AZD-1480	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.013313304	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	MELENGESTROL ACETATE	rxcui:1537798	MELENGESTROL ACETATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	5-METHOXYTRYPTAMINE	rxcui:1426888	5-METHOXYTRYPTAMINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003403842	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	SALICYLALDEHYDE THIOSEMICARBAZONE	chembl:CHEMBL242112	SALICYLALDEHYDE THIOSEMICARBAZONE	FALSE	FALSE	FALSE
SLC9A1	hgnc:11071	SLC9A1	DTC	9/2/20	NULL	52.50767123569449	CARIPORIDE	ncit:C76028	CARIPORIDE	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.212581665	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.094608417	CHIR-99021	ncit:C177060	LADUVIGLUSIB	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	ANDROSTERONE	rxcui:1312359	ANDROSTERONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011806109	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	2'-HYDROXYCHALCONE	chembl:CHEMBL32147	2'-HYDROXYCHALCONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	SJ000032159	chembl:CHEMBL591361	CHEMBL:CHEMBL591361	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.091796628	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	PIRINIXIC ACID	iuphar.ligand:2666	PIRINIXIC ACID	FALSE	FALSE	FALSE
CARM1	hgnc:23393	CARM1	DTC	9/2/20	NULL	35.00511415712966	EOSIN	drugbank:DB13706	EOSIN	FALSE	FALSE	FALSE
DUSP3	hgnc:3069	DUSP3	DTC	9/2/20	NULL	1.071585127259071	TDR77585	chembl:CHEMBL1333386	CHEMBL:CHEMBL1333386	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	BENZO[DE]ISOCHROMEN-1(3H)-ONE	chembl:CHEMBL1479195	CHEMBL:CHEMBL1479195	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	KARANJIN	chembl:CHEMBL208484	KARANJIN	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1165542091802319	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.003270487	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.032173818	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.012454381	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
CTSB	hgnc:2527	CTSB	DTC	9/2/20	NULL	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE	iuphar.ligand:5445	N-DOCOSATETRA-7,10,13,16-ENOYLETHANOLAMINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.037505479	RO-318220	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	FLUNARIZINE DIHYDROCHLORIDE	chembl:CHEMBL539027	FLUNARIZINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.1103102336884338	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	BISINDOLYLMALEIMIDE IX	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.1442518440541057	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.2476776945079929	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011738804	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	DTC	9/2/20	NULL	0.2365210416022274	METHYSERGIDE MALEATE	rxcui:203190	METHYSERGIDE MALEATE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008916229	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	DTC	9/2/20	NULL	2.333674277141977	OCTOPAMINE	rxcui:1311141	OCTOPAMINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	SAPPANONE A TRIMETHYL ETHER	chembl:CHEMBL1606022	SAPPANONE A TRIMETHYL ETHER	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	ARISTOYUNNOLIN A	chembl:CHEMBL2333541	ARISTOYUNNOLIN A	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	GW0742	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.5645986154375752	SOY PROTEIN	ncit:C1803	SOY PROTEIN ISOLATE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.038159645	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007813642	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	SJ000264145	chembl:CHEMBL590675	CHEMBL:CHEMBL590675	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GNF-PF-4325	chembl:CHEMBL598263	CHEMBL:CHEMBL598263	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	L-701324	iuphar.ligand:4240	L701324	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003038638	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
TMPRSS15	hgnc:9490	TMPRSS15	DTC	9/2/20	NULL	0.9546849315580819	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.057073556	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.020542907	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.027929612	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	BENZIDINE	chembl:CHEMBL15901	BENZIDINE	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.3431873936973497	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	SB-218795	iuphar.ligand:5764	SB 218795	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.005602013	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	N-(4-NITROPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1574420	CHEMBL:CHEMBL1574420	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	N-DEACETYLCOLCHICEINE	ncit:C1264	TRIMETHYLCOLCHICINIC ACID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.044124093	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1562728310586145	KETANSERIN TARTRATE	ncit:C2036	KETANSERIN TARTRATE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.026385764	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	ESOXYBUTYNIN	ncit:C166661	ESOXYBUTYNIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.9376369863516875	SJ000036432	chembl:CHEMBL591135	CHEMBL:CHEMBL591135	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.1143957978991165	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.012233847	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	TRIFLUPROMAZINE HYDROCHLORIDE	rxcui:91125	TRIFLUPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PTAEROXYLIN	chembl:CHEMBL1527943	PTAEROXYLIN	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.6667640791834221	PF-04217903	drugbank:DB12848	PF-04217903	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TDR77582	chembl:CHEMBL1329349	CHEMBL:CHEMBL1329349	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.065799087	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	VER-3323	iuphar.ligand:168	VER-3323	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.027476542	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.050781113	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1524170427741495	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	0.4375639269641208	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.052824619	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	TELENZEPINE	ncit:C75285	TELENZEPINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	ALEXIDINE DIHYDROCHLORIDE	chembl:CHEMBL554041	ALEXIDINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.009632668	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	CINOBUFAGIN	ncit:C95021	CINOBUFAGIN	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.017456008	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	TCMDC-124317	chembl:CHEMBL586937	CHEMBL:CHEMBL586937	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	PYRENE	chembl:CHEMBL279564	PYRENE	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1100789753368857	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	PIPENZOLATE	rxcui:33743	PIPENZOLATE	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.017456008	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	1,2-DIMETHOXY-ANTHRAQUINONE	chembl:CHEMBL52884	CHEMBL:CHEMBL52884	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.001135154	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	2,2,3,3,4,4,5,5,6,6,7,7,8,8,8-PENTADECAFLUORO-OCTANOIC ACID	chembl:CHEMBL172988	CHEMBL:CHEMBL172988	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.169927739	QUINALDINE BLUE	chembl:CHEMBL1433292	QUINALDINE BLUE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	HTS-05057	chembl:CHEMBL372629	CHEMBL:CHEMBL372629	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	BENZOPHENONE-THIOSEMICARBAZONE	chembl:CHEMBL1269809	BENZOPHENONE-THIOSEMICARBAZONE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.021951368	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1415301111474245	SJ000001592	chembl:CHEMBL591834	CHEMBL:CHEMBL591834	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.089756703	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001678098	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
EP300	hgnc:3373	EP300	DTC	9/2/20	NULL	5.834185692854944	DIETHYL-2-TETRADECYLIDENEMALONATE	chembl:CHEMBL257748	CHEMBL:CHEMBL257748	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.009270422	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	GNF-PF-2947	chembl:CHEMBL581677	CHEMBL:CHEMBL581677	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.085796848	D-LEUCINE	rxcui:6308	LEUCINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	6-BROMOFLAVONE	chembl:CHEMBL52825	6-BROMOFLAVONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1193356164447602	(-)-DICENTRINE	chembl:CHEMBL478754	CHEMBL:CHEMBL478754	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	MONASTROL	drugbank:DB04331	MONASTROL	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	DIOSMIN	rxcui:3489	DIOSMIN	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	7-METHOXY-BAPTIGENIN	chembl:CHEMBL583578	CHEMBL:CHEMBL583578	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE	chembl:CHEMBL460508	CHEMBL:CHEMBL460508	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	ICI-199,441	iuphar.ligand:11691	ICI-199441	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE	chembl:CHEMBL344469	0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	NSC-748113	chembl:CHEMBL2063687	CHEMBL:CHEMBL2063687	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW819230X	chembl:CHEMBL182283	GW819230X	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.003256492	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	ALLOXAZINE	iuphar.ligand:456	ALLOXAZINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	ENCLOMIPHENE	ncit:C28211	ENCLOMIPHENE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003405608	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
CAMK1	hgnc:1459	CAMK1	DTC	9/2/20	NULL	0.1508841127462485	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1250182648468916	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.4953553890159858	DNDI1417629	chembl:CHEMBL1731432	CHEMBL:CHEMBL1731432	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.013336975	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	AM580	iuphar.ligand:2647	RO 40-6055	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.3596415838061266	NAFTIFINE HYDROCHLORIDE	rxcui:31476	NAFTIFINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	SULFADOXINE	rxcui:10173	SULFADOXINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00299804	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	(S)-FELODIPINE	chembl:CHEMBL428768	(S)-FELODIPINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.056157937	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.010902756	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010375838	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.07458476	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.6250913242344582	NSC-37136	chembl:CHEMBL1370674	CHEMBL:CHEMBL1370674	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.072524408	DIOSMIN	rxcui:3489	DIOSMIN	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1544343271638073	NSC-37642	chembl:CHEMBL1707907	CHEMBL:CHEMBL1707907	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	BENZOPHENONE-THIOSEMICARBAZONE	chembl:CHEMBL1269809	BENZOPHENONE-THIOSEMICARBAZONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.010715851	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.0287871	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	NSC-67746	chembl:CHEMBL333177	CHEMBL:CHEMBL333177	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	DNDI1417607	chembl:CHEMBL1588679	CHEMBL:CHEMBL1588679	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	inhibitor	0.031254566	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	DNDI1417072	chembl:CHEMBL1310701	CHEMBL:CHEMBL1310701	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	CAULIBUGULONE C	chembl:CHEMBL445969	CAULIBUGULONE C	FALSE	FALSE	FALSE
CAMK1D	hgnc:19341	CAMK1D	DTC	9/2/20	NULL	0.056581542	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.023493365	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.086933231	GNF-PF-4078	chembl:CHEMBL584883	CHEMBL:CHEMBL584883	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.012020987	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK1023156A	chembl:CHEMBL518953	GSK-1023156A	FALSE	FALSE	FALSE
CDK16	hgnc:8749	CDK16	DTC	9/2/20	inhibitor	0.2625383561784725	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	DESMETHYLENYLNOCARDAMINE	chembl:CHEMBL517615	DESMETHYLENYLNOCARDAMINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.01186614	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.046881849	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.4375639269641209	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	DIBENZOYLMETHANE	chembl:CHEMBL371523	DIBENZOYLMETHANE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	GNF-PF-2776	chembl:CHEMBL578294	CHEMBL:CHEMBL578294	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	AY-9944	chembl:CHEMBL1513392	CHEMBL:CHEMBL1513392	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	PSB-1115	iuphar.ligand:3286	PSB1115	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	IODOFORM	rxcui:27748	IODOFORM	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	SJ000018298	chembl:CHEMBL591412	CHEMBL:CHEMBL591412	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.004776899	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	PERVILLEINE F	chembl:CHEMBL485486	PERVILLEINE F	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	(E)-2-STYRYLCHROMONE	chembl:CHEMBL388823	CHEMBL:CHEMBL388823	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.052824619	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.009803523	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	MONTELUKAST	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.003708169	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.009954061	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.034118045	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.025147352	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.040051618	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
MAP3K10	hgnc:6849	MAP3K10	DTC	9/2/20	NULL	0.108040476	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	PROSULTIAMINE	ncit:C82256	PROSULTIAMINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002669701	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.027010119	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013299815	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.002318219	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.03378872	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
TNIK	hgnc:30765	TNIK	DTC	9/2/20	inhibitor	0.3281729452230906	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.009487052	Fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.0545251	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.030886865	Lidocaine	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	FDA	10-Apr-24	NULL	0.6775183385250904	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	MyCancerGenome	20-Jun-17	inhibitor	0.6035364509849942	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	MyCancerGenome	20-Jun-17	inhibitor	0.2083637747448194	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.1736364789540161	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.1480479452134243	CANERTINIB	ncit:C77588	CANERTINIB	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.1808115400678185	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.5125748858722557	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.750109589	BMS-777607	drugbank:DB12064	BMS-777607	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.1842374429322613	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.047626006	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.1666910197958555	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.08572681	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.061737415	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.1111273465305703	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.084146909	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1143957978991165	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.182318303	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.08334551	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.094535416	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.074797252	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.046303061	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1666910197958555	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2917092846427472	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2625383561784725	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.009481342	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
AKT3	hgnc:393	AKT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.046881849	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
AKT3	hgnc:393	AKT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.082043236	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.062509132	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1151484018326633	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4526523382387456	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1250182648468916	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.080781033	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.08334551	1058137-23-7	ncit:C95726	LUCITANIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2651902587661338	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.7501095890813498	BAY869766	hemonc:437	REFAMETINIB	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1704794520639431	BAY869766	hemonc:437	REFAMETINIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1346350544504987	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
MAP2K4	hgnc:6844	MAP2K4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.8334550989792776	BAY869766	hemonc:437	REFAMETINIB	FALSE	FALSE	TRUE
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.9376369863516874	BAY869766	hemonc:437	REFAMETINIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1223955040459079	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.004931687	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	1.029066006546944	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.1121958787087489	MARIJUANA	ncit:C26659	MARIJUANA	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.053937002	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.044498026	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
AKR1C1	hgnc:384	AKR1C1	NCI	14-Sep-17	NULL	1.334940794127826	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
ALB	hgnc:399	ALB	NCI	14-Sep-17	NULL	0.1403948428761885	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
APOA1	hgnc:600	APOA1	NCI	14-Sep-17	NULL	0.050174554	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.058212496	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.3621218705909966	GINKGO BILOBA	rxcui:236809	GINKGO BILOBA EXTRACT	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.100589408	IMMUNOSUPPRESSANT	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.1852122442176172	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.075333818	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.071148606	CD271	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.037121012	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.032837818	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1707566544250227	PROTEIN KINASE INHIBITOR	ncit:C1404	PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.8537832721251137	POLYSIALIC ACID	ncit:C1201	POLYSIALIC ACID	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1707566544250227	HYPERBARIC OXYGEN	ncit:C2351	HYPERBARIC OXYGEN	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.056826484	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.03409589	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.029833904	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	NCI	14-Sep-17	NULL	0.066591847	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
CALR	hgnc:1455	CALR	NCI	14-Sep-17	NULL	0.1442518440541057	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
CANX	hgnc:1473	CANX	NCI	14-Sep-17	NULL	52.50767123569449	MPO	ncit:C1846	LERIDISTIM	FALSE	FALSE	FALSE
CAST	hgnc:1515	CAST	NCI	14-Sep-17	NULL	0.326134604	12-O-TETRADECANOYLPHORBOL-13-ACETATE	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	NCI	14-Sep-17	NULL	0.096167896	ANTIDEPRESSANTS	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
CHAT	hgnc:1912	CHAT	NCI	14-Sep-17	NULL	2.333674277141978	DIHYDROTESTOSTERONE	ncit:C29619	DIHYDROTESTOSTERONE	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.9723642821424906	INTERFERON BETA	chembl:CHEMBL2108510	INTERFERON BETA	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.096167896	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.1470803115845784	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.004786261	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.006811217	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.050026364	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
CYR61	hgnc:2654	CCN1	NCI	14-Sep-17	NULL	1.060761035064535	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
DCK	hgnc:2704	DCK	NCI	14-Sep-17	NULL	0.1304538415793652	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.4375639269641208	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
DCK	hgnc:2704	DCK	NCI	14-Sep-17	NULL	2.282942227638891	TETRAHYDROURIDINE	ncit:C868	TETRAHYDROURIDINE	FALSE	FALSE	FALSE
DCN	hgnc:2705	DCN	NCI	14-Sep-17	NULL	0.5770073762164232	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.07182992	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.1367387271762877	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.054243462	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	2.386712328895204	ZEBULARINE	ncit:C37455	ZEBULARINE	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.6604738520213144	UFT	ncit:C9506	TEGAFUR-URACIL	FALSE	FALSE	FALSE
DUSP6	hgnc:3072	DUSP6	NCI	14-Sep-17	NULL	2.187819634820604	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
DUSP6	hgnc:3072	DUSP6	NCI	14-Sep-17	NULL	0.384671584	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.5834185692854945	ANESTHETIC AGENT	ncit:C245	ANESTHETIC AGENT	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1442518440541057	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	1.29648571	CANNABINOL	rxcui:1976	CANNABINOL	FALSE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.2375912725597036	ETANERCEPT	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	0.6482428547616605	FUROSEMIDE	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.021344582	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1029562181092049	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.072474356	CPT-11	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.055010656	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.175610941	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1286952726365061	NICARDIPINE	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.2344092465879218	NG-MONOMETHYL-L-ARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.045758319	6-MP	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	1.810609352954982	MIP-1 ALPHA	ncit:C1391	RECOMBINANT MACROPHAGE INFLAMMATORY PROTEIN-1 ALPHA	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.2414145803939977	RECOMBINANT INTERFERON BETA-1A	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.048083948	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.097236428	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1750255707856483	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
KRT18	hgnc:6430	KRT18	NCI	14-Sep-17	NULL	1.093909817410302	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
LAMP1	hgnc:6499	LAMP1	NCI	14-Sep-17	NULL	6.563458904461812	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.2083637747448194	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
LCAT	hgnc:6522	LCAT	NCI	14-Sep-17	NULL	2.625383561784724	TESTOSTERONE PROPIONATE	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.4861821410712454	CALCIUM CHANNEL BLOCKER	ncit:C333	CALCIUM CHANNEL BLOCKER	FALSE	FALSE	FALSE
LPAR2	hgnc:3168	LPAR2	NCI	14-Sep-17	NULL	1.944728564284981	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.2000292237550266	6-HYDROXYMETHYLACYLFULVENE	ncit:C1717	IROFULVEN	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.5147810905460245	KEYHOLE LIMPET HEMOCYANIN	ncit:C1139	KEYHOLE LIMPET HEMOCYANIN	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.2573905452730122	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	NCI	14-Sep-17	NULL	0.093763699	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
MATK	hgnc:6906	MATK	NCI	14-Sep-17	NULL	0.5770073762164232	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.030950587	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	3.500511415712966	XANTHINE OXIDASE INHIBITOR	ncit:C1637	XANTHINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	1.875273972703375	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.020002922	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	1.093909817410302	GLYCYRRHETINIC ACID	rxcui:1311506	GLYCYRRHETINIC ACID	TRUE	FALSE	FALSE
NODAL	hgnc:7865	NODAL	NCI	14-Sep-17	NULL	105.0153424713889	FGF4	ncit:C1309	RECOMBINANT FIBROBLAST GROWTH FACTOR 4	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.28382525	RHIL-11	rxcui:1311380	INTERLEUKIN-11	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.042073455	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.078136416	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	NCI	14-Sep-17	NULL	0.1047012387551236	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PER1	hgnc:8845	PER1	NCI	14-Sep-17	NULL	1.141471113819445	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1154014752432845	SULFORAPHANE	ncit:C1424	SULFORAPHANE	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	2.019525817	AROMATASE INHIBITOR	ncit:C1740	AROMATASE INHIBITOR	FALSE	FALSE	TRUE
PLAT	hgnc:9051	PLAT	NCI	14-Sep-17	NULL	0.561579372	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.048083948	ANTIDEPRESSANTS	ncit:C265	ANTIDEPRESSANT AGENT	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.089298761	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
PRKAB1	hgnc:9378	PRKAB1	NCI	14-Sep-17	NULL	0.2224901323546377	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
RBP4	hgnc:9922	RBP4	NCI	14-Sep-17	NULL	2.386712328895204	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.034572952	STI571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	NCI	14-Sep-17	NULL	0.015386863	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
RPS6KA3	hgnc:10432	RPS6KA3	NCI	14-Sep-17	NULL	0.3333820395917111	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
RTN4	hgnc:14085	RTN4	NCI	14-Sep-17	NULL	0.6364566210387212	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	1.312691780892362	LISINOPRIL	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
SHH	hgnc:10848	SHH	NCI	14-Sep-17	NULL	0.2885036881082115	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SI	hgnc:10856	SI	NCI	14-Sep-17	NULL	0.4688184931758437	RU-38486	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.027383401	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	NCI	14-Sep-17	NULL	0.1296485709523321	N-ACETYL-L-CYSTEINE	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	NCI	14-Sep-17	NULL	0.2651902587661338	ACLARUBICIN	rxcui:239	ACLARUBICIN	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	NCI	14-Sep-17	NULL	0.036673771	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
SOAT1	hgnc:11177	SOAT1	NCI	14-Sep-17	NULL	0.4773424657790409	6-HYDROXYDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	NCI	14-Sep-17	NULL	0.059667808	SODIUM 4-PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	NCI	14-Sep-17	NULL	0.1136529680426287	AMIKACIN	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	NCI	14-Sep-17	NULL	0.4167275494896388	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
SRI	hgnc:11292	SRI	NCI	14-Sep-17	NULL	0.6563458904461812	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
SYP	hgnc:11506	SYP	NCI	14-Sep-17	NULL	2.187819634820604	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
SULT2A1	hgnc:11458	SULT2A1	NCI	14-Sep-17	NULL	0.9546849315580819	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.1186614039224734	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.093346971	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.2500365296937833	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	NCI	14-Sep-17	NULL	0.090922374	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.1881995384791917	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.2309721608608262	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.055839424	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.11707396	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.077387872	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	NCI	14-Sep-17	NULL	0.1472865953315413	INFLIXIMAB	rxcui:1790539	INFLIXIMAB-DYYB	TRUE	TRUE	FALSE
THBS2	hgnc:11786	THBS2	NCI	14-Sep-17	NULL	6.563458904461812	ADRENOCORTICOTROPIC HORMONE	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	NCI	14-Sep-17	NULL	0.1372749574789398	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.2991890098899971	ANTICARCINOGENIC	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.2991890098899971	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	OncoKB	23-Jul-20	NULL	0.3309307010653015	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	OncoKB	23-Jul-20	NULL	0.088866948	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	OncoKB	23-Jul-20	NULL	1.029066006546944	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	OncoKB	23-Jul-20	NULL	0.1196983386831941	Niraparib	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
ANKFN1	hgnc:26766	ANKFN1	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	OncoKB	23-Jul-20	NULL	0.2660861718025059	AZD8186	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
KCNMB1	hgnc:6285	KCNMB1	PharmGKB	4/5/24	NULL	4.667348554283955	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
ADD1	hgnc:243	ADD1	PharmGKB	4/5/24	NULL	2.187819634820604	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.3889457128569963	terfenadine	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.070197421	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADCY9	hgnc:240	ADCY9	PharmGKB	4/5/24	NULL	1.615620653405984	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
SLC24A4	hgnc:10978	SLC24A4	PharmGKB	4/5/24	NULL	8.078103267029924	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
IGF2R	hgnc:5467	IGF2R	PharmGKB	4/5/24	NULL	4.039051633514962	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
SCGB3A1	hgnc:18384	SCGB3A1	PharmGKB	4/5/24	NULL	1.810609352954982	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.016126435	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.01169957	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADH1A	hgnc:249	ADH1A	PharmGKB	4/5/24	NULL	0.1930429089547592	fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.009862448	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	0.1704794520639432	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.1103102336884338	fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.022949157	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.1491695205559502	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	0.1704794520639432	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.016807833	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.091796628	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	PharmGKB	4/5/24	NULL	0.2375912725597036	fludarabine	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	PharmGKB	4/5/24	NULL	0.09699693	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.069638821	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.071471422	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CYP3A7	hgnc:2640	CYP3A7	PharmGKB	4/5/24	NULL	1.500219178	etonogestrel	rxcui:14584	ETONOGESTREL	TRUE	FALSE	FALSE
CDCA3	hgnc:14624	CDCA3	PharmGKB	4/5/24	NULL	1.141471113819445	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	PharmGKB	4/5/24	NULL	0.1216662358986632	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.027811267	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.1640864726115453	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.157680694	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.053038052	cabazitaxel	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.7292732116068681	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.3070624048871023	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
GRIA1	hgnc:4571	GRIA1	PharmGKB	4/5/24	NULL	0.1881995384791917	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.072919531	chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
WWOX	hgnc:12799	WWOX	PharmGKB	4/5/24	NULL	0.3763990769583835	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NME1	hgnc:7849	NME1	PharmGKB	4/5/24	NULL	1.166837138570989	adefovir dipivoxil	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
MT-ND1	hgnc:7455	MT-ND1	PharmGKB	4/5/24	NULL	5.250767123569449	micronomicin	rxcui:29996	MICRONOMICIN	FALSE	FALSE	FALSE
SERPINA6	hgnc:1540	SERPINA6	PharmGKB	4/5/24	NULL	0.087512785	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.017260904	maprotiline	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.009756163	erythromycin	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.561579372	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.024467694	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003356195	primidone	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.05913026	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	1.009762908	lumefantrine	rxcui:847728	LUMEFANTRINE	TRUE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	PharmGKB	4/5/24	NULL	0.218327115	anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
GSTM3	hgnc:4635	GSTM3	PharmGKB	4/5/24	NULL	0.384671584	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
P2RY12	hgnc:18124	P2RY12	PharmGKB	4/5/24	NULL	3.828684360936057	prasugrel	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	PharmGKB	4/5/24	NULL	0.4795221117415022	prasugrel	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.2169738480813822	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.1229687850953032	neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
CES1P1	hgnc:18546	CES1P1	PharmGKB	4/5/24	NULL	0.9723642821424907	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.040703621	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.005903055	flupenthixol	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.03219848	ciprofloxacin	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.050597611	brexpiprazole	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.050597611	meclizine	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.027244868	hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.2447910080918158	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
PIN1	hgnc:8988	PIN1	PharmGKB	4/5/24	NULL	0.1164249916534246	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
GCKR	hgnc:4196	GCKR	PharmGKB	4/5/24	NULL	0.3659071166250487	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
NAT1	hgnc:7645	NAT1	PharmGKB	4/5/24	NULL	0.088396753	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
EOMES	hgnc:3372	EOMES	PharmGKB	4/5/24	NULL	15.00219178162699	glatiramer acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
MGAT4A	hgnc:7047	MGAT4A	PharmGKB	4/5/24	NULL	0.6403374540938354	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.049793903	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
NR1H3	hgnc:7966	NR1H3	PharmGKB	4/5/24	NULL	0.1111273465305703	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
GRK4	hgnc:4543	GRK4	PharmGKB	4/5/24	NULL	1.166837138570988	verapamil	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
GRK5	hgnc:4544	GRK5	PharmGKB	4/5/24	NULL	0.1630673019742065	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
SPINK5	hgnc:15464	SPINK5	PharmGKB	4/5/24	NULL	3.621218705909965	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.167488584	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HDAC11	hgnc:19086	HDAC11	PharmGKB	4/5/24	NULL	0.167488584	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.021933029	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
MDM4	hgnc:6974	MDM4	PharmGKB	4/5/24	NULL	0.2108741816694558	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
SCNN1G	hgnc:10602	SCNN1G	PharmGKB	4/5/24	NULL	0.2536602475154323	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.016611095	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.09869863	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	0.3454452054979901	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.04339477	etravirine	rxcui:475969	ETRAVIRINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.030996264	iguratimod	ncit:C65886	IGURATIMOD	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.004172574	oxazepam	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
CD38	hgnc:1667	CD38	PharmGKB	4/5/24	NULL	23.33674277141977	isatuximab	rxcui:2282018	ISATUXIMAB	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.4773424657790409	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
ALG10	hgnc:23162	ALG10	PharmGKB	4/5/24	NULL	1.129197231	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
KCNK2	hgnc:6277	KCNK2	PharmGKB	4/5/24	NULL	0.6081969641200136	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
C18ORF21	hgnc:28802	C18orf21	PharmGKB	4/5/24	NULL	1.875273972703374	sotalol	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.1591141552596803	pyrimethamine	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.047304208	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	PharmGKB	4/5/24	NULL	0.036387853	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.006811217	hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.062733179	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SLC22A17	hgnc:23095	SLC22A17	PharmGKB	4/5/24	NULL	0.5770073762164231	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
IL10	hgnc:5962	IL10	PharmGKB	4/5/24	NULL	0.2625383561784725	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
DCP1B	hgnc:24451	DCP1B	PharmGKB	4/5/24	NULL	1.129197231	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.016724851	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NRP2	hgnc:8005	NRP2	PharmGKB	4/5/24	NULL	1.154014752432846	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
COL1A2	hgnc:2198	COL1A2	PharmGKB	4/5/24	NULL	0.1282238613814273	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CBR1	hgnc:1548	CBR1	PharmGKB	4/5/24	NULL	0.384671584	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	0.258658479	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1296485709523321	sibutramine	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	PharmGKB	4/5/24	NULL	0.015557829	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.1392776425349986	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.058341857	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.064824285	lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	PharmGKB	4/5/24	NULL	0.128537751	entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
TET2	hgnc:25941	TET2	PharmGKB	4/5/24	NULL	0.1902451856365742	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.3535870116881784	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.051143836	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
PRDX4	hgnc:17169	PRDX4	PharmGKB	4/5/24	NULL	1.265245090016735	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
GAD2	hgnc:4093	GAD2	PharmGKB	4/5/24	NULL	2.187819634820604	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.546954909	hydralazine / isosorbide dinitrate	wikidata:Q48566743	HYDRALAZINE / ISOSORBIDE DINITRATE	FALSE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TEND	1-Aug-11	NULL	1.312691780892362	ZUCLOPENTHIXOL	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.2734774543525755	procainamide	rxcui:8700	PROCAINAMIDE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.036673771	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	2.100306849	elbasvir / grazoprevir	wikidata:Q22673321	ELBASVIR/GRAZOPREVIR	FALSE	FALSE	FALSE
NFATC1	hgnc:7775	NFATC1	PharmGKB	4/5/24	NULL	0.6105543166941221	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:12075	iuphar.ligand:12075	VULOLISIB	FALSE	FALSE	FALSE
PLCE1	hgnc:17175	PLCE1	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
PML	hgnc:9113	PML	PharmGKB	4/5/24	NULL	1.346350544504987	arsenic trioxide	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	0.03136659	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.6364566210387212	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.020164236	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
AKR1D1	hgnc:388	AKR1D1	PharmGKB	4/5/24	NULL	2.187819634820604	cholic acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	PharmGKB	4/5/24	NULL	0.042793538	venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
GPX5	hgnc:4557	GPX5	PharmGKB	4/5/24	NULL	0.3763990769583835	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ASTN2	hgnc:17021	ASTN2	PharmGKB	4/5/24	NULL	5.834185692854945	isoniazid	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.010620484	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
CNTN4	hgnc:2174	CNTN4	PharmGKB	4/5/24	NULL	3.387591692625451	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	PharmGKB	4/5/24	NULL	0.9546849315580818	liraglutide	rxcui:475968	LIRAGLUTIDE	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.081533651	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.4118248724368196	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	1.848379561100067	captopril	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
PRKCB	hgnc:9395	PRKCB	PharmGKB	4/5/24	NULL	0.5966780822238011	dexmedetomidine	rxcui:228054	DEXMEDETOMIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	0.030598876	regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	1,2-BENZANTHRACENE	chembl:CHEMBL1873684	CHEMBL:CHEMBL1873684	FALSE	FALSE	FALSE
RNF8	hgnc:10071	RNF8	PharmGKB	4/5/24	NULL	0.4217483633389116	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.2580229544751573	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	TALC	12-May-16	inhibitor	0.1356787370431382	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.2128689374420047	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.138178082	DIMETHYLCURCUMIN	drugbank:DB06133	DIMETHYLCURCUMIN	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.1495945049449985	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.3918482928036902	DANUSERTIB	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.082171629	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	BUPRENORPHINE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
UNIPROT:Q01668	hgnc:1391	CACNA1D	TdgClinicalTrial	Jan-14	NULL	0.2442217266776488	AMLODIPINE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.297915865	AMLODIPINE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	ALTROPANE	drugbank:DB04947	ALTROPANE	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
UNIPROT:P10696	hgnc:441	ALPG	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	AMIFOSTINE	rxcui:1545987	AMIFOSTINE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q02880	hgnc:11990	TOP2B	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	AMONAFIDE	rxcui:1440270	AMONAFIDE	FALSE	FALSE	FALSE
UNIPROT:P01583	hgnc:5991	IL1A	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	AMG-108	chembl:CHEMBL2109458	AMG-108	FALSE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.021087418	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
GRIK1	hgnc:4579	GRIK1	ChEMBL	33	inhibitor	1.166837138570989	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
UNIPROT:P13688	hgnc:1814	CEACAM1	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	ARCITUMOMAB	ncit:C1494	ARCITUMOMAB	TRUE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.2590839041234926	ARRY-380	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.016603216	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.024422173	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.024709492	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P19338	hgnc:7667	NCL	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	AS1411	ncit:C91721	ANTI-NUCLEOLIN APTAMER AS1411	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.4167275494896388	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
UNIPROT:Q14957	hgnc:4587	GRIN2C	TdgClinicalTrial	Jan-14	NULL	0.2419708351875322	AZD-6765	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	2.423430980108977	BAPINEUZUMAB	ncit:C79569	BAPINEUZUMAB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.029235897	SEVITERONEL	ncit:C113652	SEVITERONEL	FALSE	FALSE	FALSE
UNIPROT:Q96RJ0	hgnc:17734	TAAR1	TdgClinicalTrial	Jan-14	NULL	0.1905904582057876	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TdgClinicalTrial	Jan-14	NULL	0.729273212	ROSUVASTATIN	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	0.5250767123569451	ETILEVODOPA	rxcui:1421444	ETILEVODOPA	FALSE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TdgClinicalTrial	Jan-14	NULL	18.37768493249307	FOLLITROPIN ALPHA	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.305277158	FOSPROPOFOL	rxcui:828682	FOSPROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.926605963	FROVATRIPTAN	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.1442518440541057	FLIBANSERIN	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	N-2-NAPHTHYLIMIDODICARBONIMIDIC DIAMIDE	chembl:CHEMBL43078	CHEMBL:CHEMBL43078	FALSE	FALSE	FALSE
UNIPROT:P63316	hgnc:11943	TNNC1	TdgClinicalTrial	Jan-14	NULL	4.500657534	LEVOSIMENDAN	rxcui:73107	LEVOSIMENDAN	TRUE	FALSE	FALSE
UNIPROT:P24530	hgnc:3180	EDNRB	TdgClinicalTrial	Jan-14	NULL	2.250328767244049	AMBRISENTAN	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
UNIPROT:P09038	hgnc:3676	FGF2	TdgClinicalTrial	Jan-14	NULL	0.024896952	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.016449772	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
UNIPROT:Q86VZ1	hgnc:15524	P2RY8	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
NCBIGENE:2487	hgnc:3959	FRZB	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9525	iuphar.ligand:9525	A-395	FALSE	FALSE	FALSE
UNIPROT:Q99677	hgnc:4478	LPAR4	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:Q96G91	hgnc:8540	P2RY11	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:Q15077	hgnc:8543	P2RY6	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:P14784	hgnc:6009	IL2RB	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	INTERLEUKIN 2	chembl:CHEMBL1201438	ALDESLEUKIN	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5532	iuphar.ligand:5532	DECANOIC ACID	FALSE	FALSE	FALSE
UNIPROT:P32970	hgnc:11937	CD70	TdgClinicalTrial	Jan-14	NULL	12.11715490054488	MDX-1411	chembl:CHEMBL2109492	MDX-1411	FALSE	FALSE	FALSE
UNIPROT:P51582	hgnc:8542	P2RY4	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.1110098757625676	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.1290114772375786	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.1325951293830669	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.075732218	MIRTAZAPINE	rxcui:15996	MIRTAZAPINE	TRUE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:4291	rxcui:8701	PROCAINE	TRUE	FALSE	FALSE
UNIPROT:Q13200	hgnc:9559	PSMD2	TdgClinicalTrial	Jan-14	NULL	0.5385402178019948	MLN-9708	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
UNIPROT:P04141	hgnc:2434	CSF2	TdgClinicalTrial	Jan-14	NULL	2.100306849	MOR103	ncit:C170271	OTILIMAB	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.2386712328895204	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:Q86VQ6	hgnc:20667	TXNRD3	TdgClinicalTrial	Jan-14	NULL	7.501095890813499	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	1.29648571	MitoQ	chembl:CHEMBL4074884	MITOQUINONE MESYLATE	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.3409589041278864	MOTESANIB	ncit:C71896	MOTESANIB	FALSE	FALSE	TRUE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.6168664383892681	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
UNIPROT:P13612	hgnc:6140	ITGA4	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	NATALIZUMAB	rxcui:354770	NATALIZUMAB	TRUE	TRUE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.5147810905460244	NARATRIPTAN	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	NEBIVOLOL	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P34972	hgnc:2160	CNR2	TdgClinicalTrial	Jan-14	NULL	1.514644363	NABILONE	rxcui:31447	NABILONE	TRUE	FALSE	FALSE
UNIPROT:Q06187	hgnc:1133	BTK	TdgClinicalTrial	Jan-14	NULL	0.4055851016423223	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:8974	iuphar.ligand:8974	OMIPALISIB	FALSE	FALSE	FALSE
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	PEGVISOMANT	rxcui:278739	PEGVISOMANT	TRUE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.09699693	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
UNIPROT:P31751	hgnc:392	AKT2	TdgClinicalTrial	Jan-14	NULL	0.3889457128569963	PERIFOSINE	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
SFN	hgnc:10773	SFN	DTC	9/2/20	NULL	1.400204566285186	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:Q9Y243	hgnc:393	AKT3	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	PERIFOSINE	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.7573221812840553	PIMAVANSERIN	rxcui:1791685	PIMAVANSERIN	TRUE	FALSE	FALSE
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	POZANICLINE	ncit:C81045	POZANICLINE	FALSE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	3.828684360936057	PRASUGREL	rxcui:613391	PRASUGREL	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.400821918	PMI-001	drugbank:DB05730	PMI-001	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.1244257612220248	PAMOIC ACID	iuphar.ligand:2920	PAMOIC ACID	FALSE	FALSE	FALSE
UNIPROT:Q08752	hgnc:9257	PPID	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	SCY-635	drugbank:DB12451	SCY-635	FALSE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TdgClinicalTrial	Jan-14	NULL	0.201178817	DEXLANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:O60832	hgnc:2890	DKC1	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	V934/V935	ncit:C80055	HTERT VACCINE V934/V935	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006100578	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
UNIPROT:O14746	hgnc:11730	TERT	TdgClinicalTrial	Jan-14	NULL	0.5000730593875666	V934/V935	ncit:C80055	HTERT VACCINE V934/V935	FALSE	FALSE	FALSE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	VIGABATRIN	rxcui:14851	VIGABATRIN	TRUE	FALSE	FALSE
UNIPROT:P54284	hgnc:1403	CACNB3	TdgClinicalTrial	Jan-14	NULL	0.1795134059339982	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P07437	hgnc:20778	TUBB	TdgClinicalTrial	Jan-14	NULL	0.082429625	VINORELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	0.072424374	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:Q9H293	hgnc:13765	IL25	TdgClinicalTrial	Jan-14	NULL	5.250767124	VIDOFLUDIMUS	ncit:C152873	VIDOFLUDIMUS	FALSE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	3.750547945	CHLORMERODRIN	ncit:C65315	CHLORMERODRIN	TRUE	FALSE	FALSE
UNIPROT:Q9H3N8	hgnc:17383	HRH4	TdgClinicalTrial	Jan-14	NULL	0.098421127	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	CYCLOPENTOLATE	rxcui:3001	CYCLOPENTOLATE	TRUE	FALSE	FALSE
UNIPROT:P54710	hgnc:4026	FXYD2	TdgClinicalTrial	Jan-14	NULL	0.9723642821424908	CYCLOTHIAZIDE	rxcui:22033	CYCLOTHIAZIDE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.2983390411119005	Dibucaine	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
UNIPROT:P02458	hgnc:2200	COL2A1	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.2243917574174978	CYCLOBENZAPRINE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.011940798	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P23415	hgnc:4326	GLRA1	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	DESFLURANE	rxcui:27340	DESFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	ENCAINIDE	rxcui:42368	ENCAINIDE	FALSE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	1.334940794127826	EPROSARTAN	rxcui:83515	EPROSARTAN	TRUE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.111481255	ERGOCALCIFEROL	rxcui:4018	ERGOCALCIFEROL	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.1166837138570989	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	0.3017682254924971	GLIBENCLAMIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	GONADORELIN	rxcui:6384	GONADORELIN	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.2234368988752957	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
PSMA7	hgnc:9536	PSMA7	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.1280674908187671	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.736088849	GUANADREL SULFATE	rxcui:91239	GUANADREL SULFATE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.1118771404169627	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.1411496538593938	HYDROXYZINE	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1204304386139782	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1562728310586145	METARAMINOL	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
UNIPROT:P48039	hgnc:7463	MTNR1A	TdgClinicalTrial	Jan-14	NULL	1.034633915974276	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.1600843635234588	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q8NET8	hgnc:18084	TRPV3	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	MENTHOL	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TdgClinicalTrial	Jan-14	NULL	1.050153425	METHAZOLAMIDE	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.596678082	METIPRANOLOL	rxcui:10824	METIPRANOLOL	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	1.334940794127826	MOEXIPRIL	rxcui:30131	MOEXIPRIL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.05814803	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TdgClinicalTrial	Jan-14	NULL	0.078136416	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.060984519	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.7242437411819932	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.073885091	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.06757744	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.1693795846312726	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.7778914257139926	ORPHENADRINE	rxcui:7715	ORPHENADRINE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.059532507	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.072125922	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	1.944728564284981	SODIUM OXYBATE	rxcui:9899	SODIUM OXYBATE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1223955040459079	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1835932560688619	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.083257407	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.088396753	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.091796628	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.092988792	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.2625383561784725	TENOXICAM	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
UNIPROT:P37088	hgnc:10599	SCNN1A	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
UNIPROT:P23945	hgnc:3969	FSHR	TdgClinicalTrial	Jan-14	NULL	18.37768493249307	UROFOLLITROPIN	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:Q9GZZ6	hgnc:13800	CHRNA10	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	TRIMETHAPHAN	rxcui:10828	TRIMETHAPHAN	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	3.750547945	CHLORMERODRIN	ncit:C65315	CHLORMERODRIN	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	MODOTUXIMAB	ncit:C152075	MODOTUXIMAB	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.096050618	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P02458	hgnc:2200	COL2A1	TEND	1-Aug-11	NULL	1.875273972703375	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.3739862623624964	COCAINE	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.2243917574174978	CYCLOBENZAPRINE	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TEND	1-Aug-11	NULL	0.099446347	DANAZOL	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	1.666910197958555	DECAMETHONIUM	ncit:C77363	DECAMETHONIUM	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TEND	1-Aug-11	NULL	0.1842374429322614	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TEND	1-Aug-11	NULL	0.095295229	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.056142926	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	1.334940794127826	EPROSARTAN	rxcui:83515	EPROSARTAN	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	0.3671865121377238	ERGOTAMINE	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.4257378748840094	FESOTERODINE	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TEND	1-Aug-11	NULL	0.068115956	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.1909369863116163	FENOPROFEN	rxcui:4331	FENOPROFEN	TRUE	FALSE	FALSE
UNIPROT:O60664	hgnc:16893	PLIN3	TEND	1-Aug-11	NULL	26.25383561784724	IDURSULFASE	rxcui:644101	IDURSULFASE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TEND	1-Aug-11	NULL	1.419126249613364	ISOCARBOXAZID	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
UNIPROT:P47712	hgnc:9035	PLA2G4A	TEND	1-Aug-11	NULL	1.093909817410302	FLUOCINONIDE	rxcui:4462	FLUOCINONIDE	TRUE	FALSE	FALSE
UNIPROT:Q01718	hgnc:6930	MC2R	TEND	1-Aug-11	NULL	2.461297089173179	CORTICOTROPIN	rxcui:376	CORTICOTROPIN	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.926605963	FROVATRIPTAN	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:Q969P6	hgnc:29787	TOP1MT	TdgClinicalTrial	Jan-14	NULL	0.1666910197958555	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P19838	hgnc:7794	NFKB1	TEND	1-Aug-11	NULL	0.029876342	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.6908904109959803	HEXYLCAINE	rxcui:26879	HEXYLCAINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.8950171233357017	HEXYLCAINE	rxcui:26879	HEXYLCAINE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.3889457128569962	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.085147575	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.080781033	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.07160137	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.596678082	METIPRANOLOL	rxcui:10824	METIPRANOLOL	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.081281225	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TEND	1-Aug-11	NULL	3.750547945	DINOPROST TROMETHAMINE	rxcui:23321	DINOPROST TROMETHAMINE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TEND	1-Aug-11	NULL	0.2456499239096818	ONDANSETRON	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
UNIPROT:O60895	hgnc:9844	RAMP2	TEND	1-Aug-11	NULL	7.501095890813499	PRAMLINTIDE	rxcui:139953	PRAMLINTIDE	TRUE	FALSE	TRUE
UNIPROT:P16066	hgnc:7943	NPR1	TEND	1-Aug-11	NULL	0.4039051633514962	NITRIC OXIDE	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.05593857	NORTRIPTYLINE	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.9723642821424906	PROCYCLIDINE	rxcui:8718	PROCYCLIDINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	PROCYCLIDINE	rxcui:8718	PROCYCLIDINE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.087537101	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.059085902	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.074690855	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P03886	hgnc:7455	MT-ND1	TEND	1-Aug-11	NULL	0.2838252499226729	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.108711535	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P18405	hgnc:11284	SRD5A1	TEND	1-Aug-11	NULL	6.563458904461812	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.078136416	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.1635752997996713	SIBUTRAMINE	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.017643707	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.1731022128649269	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.1262203635473425	Zicronapine	ncit:C152950	ZICRONAPINE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Lasofoxifene	ncit:C80679	LASOFOXIFENE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR-LIKE PROTEIN 7	hgnc:20594	EGFL7	TTD	2020.06.01	NULL	35.00511415712966	MEGF0444A	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.2465148884304905	ARQ 751	ncit:C128250	PAN-AKT INHIBITOR ARQ751	FALSE	FALSE	FALSE
ATM SERINE/THREONINE KINASE	hgnc:795	ATM	TTD	2020.06.01	NULL	0.4795221117415022	AZD1390	iuphar.ligand:11277	AZD1390	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	1.111273465305703	AP32788	rxcui:2570736	MOBOCERTINIB	TRUE	FALSE	TRUE
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	2.386712328895204	CA-4948	ncit:C148455	EMAVUSERTIB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	M7583	ncit:C129710	BTK INHIBITOR TL-895	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 8	hgnc:15632	TLR8	TTD	2020.06.01	NULL	3.281729452230906	NKTR-262	ncit:C148289	PEG-CONJUGATED TLR7/8 AGONIST NKTR-262	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	1.897867635025102	PLX9486	ncit:C121647	BEZUCLASTINIB	FALSE	FALSE	FALSE
EXPORTIN-1	hgnc:12825	XPO1	TTD	2020.06.01	NULL	8.751278539282415	SL-801	ncit:C171660	FELEZONEXOR	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1	hgnc:2432	CSF1	TTD	2020.06.01	NULL	7.501095891	PLX73086	ncit:C129688	CSF1R INHIBITOR PLX73086	FALSE	FALSE	FALSE
PROTEIN KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	0.070574827	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
G1/S-SPECIFIC CYCLIN-D1	hgnc:1582	CCND1	TTD	2020.06.01	NULL	0.039068208	ABT-263	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
CALGRANULIN D	hgnc:10489	S100A12	TTD	2020.06.01	NULL	3.500511415712966	BMS-927711	rxcui:2282307	RIMEGEPANT	TRUE	FALSE	FALSE
INTERLEUKIN-37	hgnc:15563	IL37	TTD	2020.06.01	NULL	17.50255707856483	Tildrakizumab	rxcui:2053436	TILDRAKIZUMAB	TRUE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR	hgnc:6008	IL2RA	TTD	2020.06.01	NULL	0.2573905452730122	BNZ-1	ncit:C146636	IL-2/9/15 GAMMA CHAIN RECEPTOR INHIBITOR BNZ-1	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	2.386712328895204	Remogliflozin etabonate	ncit:C91023	REMOGLIFLOZIN ETABONATE	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	1.250182648468916	Setmelanotide	rxcui:2469247	SETMELANOTIDE	TRUE	FALSE	FALSE
ACTIVIN	hgnc:24029	INHBE	TTD	2020.06.01	NULL	26.25383561784724	STM 434	iuphar.ligand:8991	STM 434	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	2.080014029626545	Ceritinib	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	2.917092846427472	SB-656933	ncit:C174724	ELUBRIXIN	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.3680444245492605	ARQ-087	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.8078103267029922	Systebryl	drugbank:DB18298	PTI-110	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	Simotaxel	ncit:C116871	SIMOTAXEL	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 4	hgnc:1605	CCR4	TTD	2020.06.01	NULL	3.088686543276147	GSK-2239633	chembl:CHEMBL2178575	GSK-2239633	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE 2	hgnc:812	ATP2A2	TTD	2020.06.01	NULL	0.760980743	Gallopamil	rxcui:4648	GALLOPAMIL	FALSE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.8204323630577265	Leuvectin	drugbank:DB17303	LEUVECTIN	FALSE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.729273212	Rosuvastatin	rxcui:301542	ROSUVASTATIN	TRUE	FALSE	FALSE
PROLYL 4-HYDROXYLASESUBUNIT ALPHA-1	hgnc:8546	P4HA1	TTD	2020.06.01	NULL	17.50255707856483	SAFIRONIL	ncit:C74278	SAFIRONIL	FALSE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	1.500219178	Epithalon	drugbank:DB17882	EPITALON	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.5357925636295356	Trimidox	wikidata:Q7842230	TRIMETHOPRIM/SULFADOXINE	FALSE	FALSE	FALSE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	3.580068493342807	YF-476	ncit:C87692	NETAZEPIDE	FALSE	FALSE	FALSE
CATIONIC TRYPSINOGEN	hgnc:9475	PRSS1	TTD	2020.06.01	NULL	1.250182648468916	MELAGATRAN	ncit:C66077	MELAGATRAN	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.045898314	METHYLENEDIOXYMETHAMPHETAMINE	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	0.1988926940746004	METHYLENEDIOXYMETHAMPHETAMINE	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.096264064	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	1.029066006546944	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.3281729452230906	TKI258	ncit:C62435	DOVITINIB LACTATE	FALSE	FALSE	FALSE
GABA(A) RECEPTOR BETA-2	hgnc:4082	GABRB2	TTD	2020.06.01	NULL	0.07631929	Ethchlorvynol	rxcui:4118	ETHCHLORVYNOL	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.3689063552859098	Medroxyprogesterone	rxcui:6691	MEDROXYPROGESTERONE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	3.750547945	Methyclothiazide	rxcui:6860	METHYCLOTHIAZIDE	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	4.449802647092754	Cilazapril	rxcui:21102	CILAZAPRIL	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	0.099446347	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV7.3	hgnc:6297	KCNQ3	TTD	2020.06.01	NULL	1.500219178	ICA-105665	drugbank:DB06089	ICA-105665	FALSE	FALSE	FALSE
LIVER CARBOXYLESTERASE	hgnc:1863	CES1	TTD	2020.06.01	NULL	0.760980743	PACTIMIBE	ncit:C66290	PACTIMIBE	FALSE	FALSE	FALSE
SERUM ALBUMIN	hgnc:399	ALB	TTD	2020.06.01	NULL	1.193356164447602	Gadobenate Dimeglumine	rxcui:68173	GADOBENATE DIMEGLUMINE	TRUE	FALSE	FALSE
MAP KINASE P38	hgnc:6874	MAPK12	TTD	2020.06.01	NULL	0.6482428547616604	SM-101	chembl:CHEMBL4298105	VALZIFLOCEPT	FALSE	FALSE	FALSE
INTERFERON-GAMMA	hgnc:5438	IFNG	TTD	2020.06.01	NULL	1.875273972703375	Fumaric acid	rxcui:25389	FUMARIC ACID	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.4773424657790409	Lumiracoxib	ncit:C66041	LUMIRACOXIB	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1132444383228493	Cocaine	rxcui:2653	COCAINE	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.4234489615781814	Oxybuprocaine	rxcui:18889	BENOXINATE	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.317586721	Epinastine	rxcui:39684	EPINASTINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.062645859	Estradiol	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.1842374429322614	Nimodipine	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2044691247495891	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	2.423430980108977	Bapineuzumab	ncit:C79569	BAPINEUZUMAB	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	1.029066006546944	STI571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	0.020002922	STI571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
THROMBOSPONDIN-1	hgnc:11785	THBS1	TTD	2020.06.01	NULL	7.501095891	CVX-045	ncit:C82384	TSP-1 MIMETIC FUSION PROTEIN CVX-045	FALSE	FALSE	TRUE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	2.423430980108977	Ponezumab	ncit:C97941	PONEZUMAB	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR GAMMA	hgnc:9866	RARG	TTD	2020.06.01	NULL	6.177373086552294	Palovarotene	rxcui:2663954	PALOVAROTENE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.014617949	Antiandrogens	ncit:C242	ANTI-ANDROGEN	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.1219690388750162	RG7601	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
C-X-C MOTIF CHEMOKINE 10	hgnc:10637	CXCL10	TTD	2020.06.01	NULL	6.177373086552294	BMS-936557	iuphar.ligand:9047	ELDELUMAB	FALSE	FALSE	FALSE
COMPLEMENT RECEPTOR TYPE 1	hgnc:2334	CR1	TTD	2020.06.01	NULL	13.12691780892362	CDX-1135	drugbank:DB17607	CDX-1135	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	AZD-3514	chembl:CHEMBL2346976	AZD3514	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	1.591141552596803	K-877	chembl:CHEMBL3545412	K-877	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.073437302	ZSTK474	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	0.8751278539282416	LBR-101	rxcui:2056691	FREMANEZUMAB	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE PIM-2	hgnc:8987	PIM2	TTD	2020.06.01	NULL	4.375639269641208	LGH-447	drugbank:DB14943	LGH-447	FALSE	FALSE	FALSE
VITAMIN K-DEPENDENT PROTEIN C	hgnc:9451	PROC	TTD	2020.06.01	NULL	1.312691780892362	Ancrod	rxcui:772	ANCROD	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.7059854956059763	Avelumab	rxcui:1875534	AVELUMAB	TRUE	FALSE	TRUE
CALGRANULIN B	hgnc:10499	S100A9	TTD	2020.06.01	NULL	26.25383561784724	Paquinimod	ncit:C87681	PAQUINIMOD	FALSE	FALSE	FALSE
LOW-AFFINITY NERVE GROWTH FACTOR RECEPTOR	hgnc:7809	NGFR	TTD	2020.06.01	NULL	4.375639269641208	Cenegermin	rxcui:2104331	CENEGERMIN-BKBJ	TRUE	FALSE	FALSE
LYMPHOTOXIN BETA RECEPTOR	hgnc:6718	LTBR	TTD	2020.06.01	NULL	6.563458904461812	Baminercept	ncit:C96762	BAMINERCEPT ALFA	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	P-BCMA-101	drugbank:DB17371	P-BCMA-101	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.9723642821424906	Ioflupane i-123	rxcui:1426874	IOFLUPANE I-123	TRUE	FALSE	FALSE
PROTOPORPHYRINOGEN OXIDASE	hgnc:9280	PPOX	TTD	2020.06.01	NULL	26.25383561784724	Aminolevulinic Acid Hydrochloride	rxcui:261715	AMINOLEVULINIC ACID HYDROCHLORIDE	TRUE	FALSE	FALSE
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	2.019525817	CALAA-01	ncit:C78450	TRANSFERRIN RECEPTOR-TARGETED ANTI-RRM2 SIRNA CALAA-01	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	L-377202	chembl:CHEMBL3093499	L-377202	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.8204323630577265	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
JUN N TERMINAL KINASE	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	0.5147810905460245	AM-111	iuphar.ligand:9101	BRIMAPITIDE	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	4.773424657790408	RO-4998452	chembl:CHEMBL2105711	TOFOGLIFLOZIN	FALSE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	0.1438566335224507	Altiratinib	ncit:C118290	ALTIRATINIB	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	2.386712328895204	BAY-X-7195	chembl:CHEMBL314115	CHEMBL:CHEMBL314115	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	0.6250913242344582	Aldosterone	rxcui:1312358	ALDOSTERONE	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.045898314	Acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.031929262	Amisulpride	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
HISTAMINE H2 RECEPTOR	hgnc:5183	HRH2	TTD	2020.06.01	NULL	2.187819634820604	Famotidine	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.111481255	Ergocalciferol	rxcui:4018	ERGOCALCIFEROL	TRUE	FALSE	FALSE
GUANYLATE CYCLASE	hgnc:4187	GC	TTD	2020.06.01	NULL	1.458546423213736	Erythrityl Tetranitrate	rxcui:4040	ERYTHRITYL TETRANITRATE	TRUE	FALSE	FALSE
N-ACETYLGALACTOSAMINE 6 SULFATASE	hgnc:4122	GALNS	TTD	2020.06.01	NULL	105.0153424713889	Elosulfase alfa	rxcui:1489914	ELOSULFASE ALFA	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.1875273972703375	Hydrocodone	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.3409589041278863	Meclofenamic acid	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
CHLORIDE CHANNEL PROTEIN 2	hgnc:2020	CLCN2	TTD	2020.06.01	NULL	35.00511415712966	Lubiprostone	rxcui:623033	LUBIPROSTONE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1383601350084176	Molindone	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	2.917092846427472	Ocrelizumab	rxcui:1876366	OCRELIZUMAB	TRUE	FALSE	FALSE
SOLUBLE GUANYLATE CYCLASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	0.4039051633514962	Nitroglycerin	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.1411496538593938	Oxatomide	rxcui:54236	OXATOMIDE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Perazine	rxcui:8042	PERAZINE	FALSE	FALSE	FALSE
SQUALENE MONOOXYGENASE	hgnc:11279	SQLE	TTD	2020.06.01	NULL	4.375639269641208	Tolnaftate	rxcui:10637	TOLNAFTATE	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.6819178082557726	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	6.563458904461812	BMS-184476	ncit:C1843	BMS-184476	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	1.312691780892362	LOXORIBINE	ncit:C1470	LOXORIBINE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	MEHD-7945A	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
LEUKOCYTE ANTIGEN CD37	hgnc:1666	CD37	TTD	2020.06.01	NULL	52.50767123569449	Otlertuzumab	ncit:C74006	OTLERTUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	activator	0.1154014752432846	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
MITOCHONDRIAL MATRIX PROTEIN P1	hgnc:5261	HSPD1	TTD	2020.06.01	NULL	17.50255707856483	DiaPep-277	chembl:CHEMBL4297934	DIAPEP-277	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:77	iuphar.ligand:77	SB 714786	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1223955040459079	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.05853698	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.024513385	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.064111931	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:173	ncit:C61919	QUIPAZINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:161	iuphar.ligand:161	BW723C86	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.069089041	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:157	iuphar.ligand:157	(R)-DOI	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.010434752	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
ATR	hgnc:882	ATR	JAX-CKB	10-Apr-24	NULL	1.166837138570988	PJ34	iuphar.ligand:11348	PJ34	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:8425	iuphar.ligand:8425	VELUSETRAG	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.047561296	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.045579576	IUPHAR.LIGAND:63	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.040051618	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:219	iuphar.ligand:219	[3H]LSD	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.076765601	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:154	iuphar.ligand:154	(+)-LSD	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.041872146	IUPHAR.LIGAND:204	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1784	ncbigene:1784	DNCM	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8481	iuphar.ligand:8481	LDN-214117	FALSE	FALSE	FALSE
NCBIGENE:315	hgnc:1611	ACKR4	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:810	iuphar.ligand:810	CCL19	FALSE	FALSE	FALSE
NCBIGENE:1784	ncbigene:1784	DNCM	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:8155	iuphar.ligand:8155	COMPOUND 13A [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:8155	iuphar.ligand:8155	COMPOUND 13A [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8481	iuphar.ligand:8481	LDN-214117	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:8206	iuphar.ligand:8206	COMPOUND 5M [PMID: 20483621]	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.2651902587661338	4'-EPICHAETOVIRIDIN A	chembl:CHEMBL1306556	CHEMBL:CHEMBL1306556	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:480	iuphar.ligand:480	A61603	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.085378327	IUPHAR.LIGAND:502	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:8459	iuphar.ligand:8459	REC 15/2615	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:489	iuphar.ligand:489	5-METHYLURAPIDIL	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:73	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:489	iuphar.ligand:489	5-METHYLURAPIDIL	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.070197421	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.062808219	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.067317527	IUPHAR.LIGAND:502	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.027290889	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:528	iuphar.ligand:526	RX821002	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:7100	rxcui:10382	TESTOSTERONE PROPIONATE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.2586584789935689	IUPHAR.LIGAND:2865	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:5607	iuphar.ligand:5607	LUF5981	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:5606	iuphar.ligand:5606	FK-453	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1682938180631233	IUPHAR.LIGAND:5622	iuphar.ligand:5622	MRS5151	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:5608	rxcui:2199015	ISTRADEFYLLINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:5606	iuphar.ligand:5606	FK-453	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1804387327687096	IUPHAR.LIGAND:412	iuphar.ligand:412	SAKURANETIN	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:582	iuphar.ligand:582	ANGIOTENSIN-(1-7)	FALSE	FALSE	FALSE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.06584034	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:11931	iuphar.ligand:11931	COMPOUND 2 [PMID: 28379944]	FALSE	FALSE	FALSE
NCBIGENE:2794	hgnc:4413	GNL1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:7733	iuphar.ligand:7733	GDC-0152	FALSE	FALSE	FALSE
NCBIGENE:969	hgnc:1694	CD69	GuideToPharmacology	2024.1	inhibitor	0.4861821410712454	IUPHAR.LIGAND:4837	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
NCBIGENE:1886	hgnc:17755	TNFRSF13C	GuideToPharmacology	2024.1	NULL	5.834185692854944	IUPHAR.LIGAND:5069	iuphar.ligand:5069	BAFF	FALSE	FALSE	FALSE
NCBIGENE:2791	hgnc:4403	GNG11	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:12704	iuphar.ligand:12704	TOLINAPANT	FALSE	FALSE	FALSE
NCBIGENE:1466	hgnc:2470	CSRP2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.2465148884304905	Carfentanil	ncit:C80574	CARFENTANIL	FALSE	FALSE	FALSE
NCBIGENE:3232	hgnc:5137	HOXD3	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12672	iuphar.ligand:12672	BCL3 INHIBITOR JS6	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:11261	iuphar.ligand:11261	COMPOUND A [PMID: 28324017]	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.2344092465879218	IUPHAR.LIGAND:9512	ncit:C96754	SOLABEGRON	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:9821	iuphar.ligand:9821	RO5508887	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.041872146	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.2344092465879218	IUPHAR.LIGAND:7129	rxcui:19484	BISOPROLOL	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:12581	iuphar.ligand:12581	ICI-89406	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:7246	rxcui:236883	NEBIVOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.1356787370431382	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.07631929	IUPHAR.LIGAND:6004	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:7518	iuphar.ligand:7518	I-BET151	FALSE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	ChEMBL	33	inhibitor	0.5073204950308647	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9146	iuphar.ligand:9146	BI-7273	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10076	iuphar.ligand:10076	BTK INHIBITOR 16 [PMID: 30122225]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:10625	ncit:C173549	TOLEBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:651	iuphar.ligand:651	AC-LYS-[MEALA6,LEU8,DES-ARG9]BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3826	iuphar.ligand:3826	[3H]LYS-[LEU8][DES-ARG9]BK	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5763	iuphar.ligand:5763	JPE1375	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:5776	iuphar.ligand:5776	YSFKPMPLAR	FALSE	FALSE	FALSE
NCBIGENE:1997	hgnc:3316	ELF1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5940	iuphar.ligand:5940	D4476	FALSE	FALSE	FALSE
NCBIGENE:531	hgnc:1393	CACNA1F	GuideToPharmacology	2024.1	inhibitor	0.1315981735230438	IUPHAR.LIGAND:2523	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:782	iuphar.ligand:782	SB-282241	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.5000730593875666	IUPHAR.LIGAND:773	iuphar.ligand:773	HIV-TAT	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:9430	iuphar.ligand:9430	BMS-681	FALSE	FALSE	FALSE
RPS14	hgnc:10387	RPS14	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:9478	iuphar.ligand:9478	COMPOUND 8IC [PMID: 19081254]	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	antibody	12.35474617310458	IUPHAR.LIGAND:6477	rxcui:2054068	MOGAMULIZUMAB	TRUE	TRUE	TRUE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4136	drugbank:DB07352	APIGENIN	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:9684	iuphar.ligand:9684	COMPOUND 12A [PMID: 29031075]	FALSE	FALSE	FALSE
NCBIGENE:725	hgnc:1328	C4BPB	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:722	hgnc:1325	C4BPA	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:715	hgnc:1246	C1R	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:820	iuphar.ligand:820	CXCL6	FALSE	FALSE	FALSE
NCBIGENE:727	hgnc:1331	C5	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:849	iuphar.ligand:849	[125I]CXCL12&ALPHA; (HUMAN)	FALSE	FALSE	FALSE
RPS29	hgnc:10419	RPS29	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:854	iuphar.ligand:854	T22	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:9883	iuphar.ligand:9883	COMPOUND 46C [PMID: 29350534]	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5974	drugbank:DB03444	6-BROMOINDIRUBIN-3'-OXIME	FALSE	FALSE	FALSE
NCBIGENE:1966	hgnc:1733	CDK13	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:10063	iuphar.ligand:10063	CDK12 INHIBITOR 2	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:5680	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:12511	iuphar.ligand:12511	QR-6401	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4598	iuphar.ligand:4598	GSK931145	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:11885	iuphar.ligand:11885	TANUXICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:9626	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:10426	ncit:C151988	EBVACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:11885	iuphar.ligand:11885	TANUXICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:5680	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8203	iuphar.ligand:8203	RO-0505124	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:9626	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.1256164383629055	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.095295229	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:11189	iuphar.ligand:11189	DALPICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:11356	iuphar.ligand:11356	LY3405105	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.16256245	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:8871	iuphar.ligand:8871	(2S,4S)-KETOCONAZOLE	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:1231	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8872	iuphar.ligand:8872	COMPOUND 1A [PMID: 18573659]	FALSE	FALSE	FALSE
NCBIGENE:1366	hgnc:2049	CLDN7	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11380	iuphar.ligand:11380	R116010	FALSE	FALSE	FALSE
NCBIGENE:1321	ncbigene:1321	CORD4	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8755	iuphar.ligand:8755	COMPOUND 38A [PMID: 15634016]	FALSE	FALSE	FALSE
NCBIGENE:3002	hgnc:4709	GZMB	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9935	iuphar.ligand:9935	GKT136901	FALSE	FALSE	FALSE
NCBIGENE:1443	hgnc:2441	CSH2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:5136	iuphar.ligand:5136	AMINOOXYACETIC ACID	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:4638	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.5097832158805291	IUPHAR.LIGAND:2639	ncit:C81539	SOBETIROME	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:10518	iuphar.ligand:10518	BILORPHIN	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.4646696569530486	IUPHAR.LIGAND:3816	iuphar.ligand:3816	[3H]DELTORPHIN II	FALSE	FALSE	FALSE
NCBIGENE:2821	hgnc:4458	GPI	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7832	iuphar.ligand:7832	COMPOUND 23N [PMID: 24900877]	FALSE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.001552563	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	modulator	0.058997383	IUPHAR.LIGAND:7694	iuphar.ligand:7694	SB269652	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.030850571	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:948	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.040546464	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:2011	hgnc:3332	MARK2	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:8167	iuphar.ligand:8167	LEUCETTINE L41	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:8162	iuphar.ligand:8162	ML315	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:8236	iuphar.ligand:8236	I-CBP112	FALSE	FALSE	FALSE
NCBIGENE:2358	hgnc:3827	FPR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6441	ncit:C66539	SIVELESTAT	FALSE	FALSE	FALSE
NR1I3	hgnc:7969	NR1I3	DTC	9/2/20	NULL	3.750547945	PK-11195	iuphar.ligand:8703	PK 11195	FALSE	FALSE	FALSE
NCBIGENE:2832	hgnc:4530	NPBWR2	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:8456	rxcui:2637535	MOLIDUSTAT	FALSE	FALSE	FALSE
NCBIGENE:1615	hgnc:2678	DARS1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6562	iuphar.ligand:6562	COMPOUND 22 [PMID: 19899765]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:9176	iuphar.ligand:9176	WZ4002	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:9409	iuphar.ligand:9409	TARLOXOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1401	hgnc:2367	CRP	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:4339	iuphar.ligand:4339	URB597	FALSE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:1049	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:12861	iuphar.ligand:12861	CPTB	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:12655	iuphar.ligand:12655	TUG-2304	FALSE	FALSE	FALSE
NCBIGENE:2024	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:8136	iuphar.ligand:8136	COMPOUND 2 [PMID: 15546730]	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.065799087	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.024756092	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.2273059360852575	IUPHAR.LIGAND:9786	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.2778183663264259	IUPHAR.LIGAND:10387	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.056601873	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.013022736	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.091159151	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:10597	iuphar.ligand:10597	BAY-985	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004961042	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.015193192	IUPHAR.LIGAND:5705	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.082043236	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9937	iuphar.ligand:9937	COMPOUND 7D [PMID: 29672049]	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:1023	iuphar.ligand:1023	FMET-MET-TYR-ALA-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6275	iuphar.ligand:6275	SHAAGTIDE	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6198	iuphar.ligand:6198	[125I-TYR]AC2-26	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.3889457128569962	IUPHAR.LIGAND:1023	iuphar.ligand:1023	FMET-MET-TYR-ALA-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1961	rxcui:43611	LATANOPROST	TRUE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.1017590527823536	IUPHAR.LIGAND:4326	iuphar.ligand:4326	TP003	FALSE	FALSE	FALSE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.3947945205691315	IUPHAR.LIGAND:8136	iuphar.ligand:8136	COMPOUND 2 [PMID: 15546730]	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:4179	iuphar.ligand:4179	DMCM	FALSE	FALSE	FALSE
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	1.875273972703375	ryanodine	iuphar.ligand:4303	RYANODINE	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.172722603	IUPHAR.LIGAND:4297	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6136	iuphar.ligand:6136	GALANIN(9-25) (RAT/MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:5357	iuphar.ligand:5357	GALANIN(2-11)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6137	iuphar.ligand:6137	GALANIN(1-20)  (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6075	iuphar.ligand:6075	J18 (GALANIN ANALOGUE)	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6100	iuphar.ligand:6100	M617	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:3592	iuphar.ligand:3592	GALANIN	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6090	iuphar.ligand:6090	GALANIN(2-30) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6129	iuphar.ligand:6129	GALANIN	FALSE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.1164249916534246	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3899	iuphar.ligand:3899	M40	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3186	iuphar.ligand:3186	COMPOUND 51 [PMID: 18800762]	FALSE	FALSE	FALSE
NCBIGENE:2977	hgnc:4684	GUCY1A2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12844	iuphar.ligand:12844	GRASP	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	blocker	0.8751278539282416	IUPHAR.LIGAND:4229	iuphar.ligand:4229	JORO SPIDER TOXIN	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:1148	iuphar.ligand:1148	HGCGR ANTAGONIST	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	CIViC	10-Apr-24	NULL	0.6250913242344582	VENETOCLAX	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4154	iuphar.ligand:4154	CGP37849	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:4086	iuphar.ligand:4086	[3H]L689560	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12110	iuphar.ligand:12110	ICLEPERTIN	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	1.166837138570989	IUPHAR.LIGAND:2817	drugbank:DB04468	AFIMOXIFENE	FALSE	FALSE	FALSE
SLC30A8	hgnc:20303	SLC30A8	PharmGKB	4/5/24	NULL	52.50767123569449	zinc acetate	rxcui:1299637	ANHYDROUS ZINC ACETATE	TRUE	FALSE	FALSE
NCBIGENE:1465	hgnc:2469	CSRP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514962	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:4847	iuphar.ligand:4847	[125I]CNP (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.056097939	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:9664	iuphar.ligand:9664	BML-281	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.080656945	IUPHAR.LIGAND:7007	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.065145994	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.1829535583125243	IUPHAR.LIGAND:12609	iuphar.ligand:12609	COMPOUND 30 [PMID: 37057760]	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:9664	iuphar.ligand:9664	BML-281	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:9426	ncit:C121641	CITARINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:4026	iuphar.ligand:4026	HISTAPRODIFEN	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1197	iuphar.ligand:1197	2-PYRIDYLETHYLAMINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:1193	iuphar.ligand:1193	2-(2-THIAZOLYL)ETHANAMINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:6976	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:1210	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:8982	iuphar.ligand:8982	INCB-38579	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:1208	iuphar.ligand:1208	(+)-CIS-H2-PAT	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1252	iuphar.ligand:1252	IMPENTAMINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1252	iuphar.ligand:1252	IMPENTAMINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:12570	iuphar.ligand:12570	ST-1505	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:7346	iuphar.ligand:7346	MK-0249	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:7346	iuphar.ligand:7346	MK-0249	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:10736	iuphar.ligand:10736	GSK-189254	FALSE	FALSE	FALSE
NCBIGENE:2763	ncbigene:2763	GMFA	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12121	iuphar.ligand:12121	INCB13739	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:729	iuphar.ligand:729	2-ARACHIDONOYLGLYCEROL	FALSE	FALSE	FALSE
NCBIGENE:112	hgnc:237	ADCY6	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:5512	iuphar.ligand:5512	DIOLEOYLPHOSPHATIDIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2885	hgnc:4566	GRB2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8960	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:7954	iuphar.ligand:7954	BMS-911543	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:10459	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:10156	iuphar.ligand:10156	JAK3 INHIBITOR 32	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1604	iuphar.ligand:1604	(-)-CYCLAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1616	iuphar.ligand:1616	DIHYDROMORPHINE	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:9006	iuphar.ligand:9006	UFP-512	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:1633	ncit:C80570	QUADAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.069180068	IUPHAR.LIGAND:9930	iuphar.ligand:9930	HENATINIB	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1284	iuphar.ligand:1284	KISSPEPTIN-13	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.011530011	IUPHAR.LIGAND:5705	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.00854061	IUPHAR.LIGAND:9914	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	inhibitor	0.2344092465879218	IUPHAR.LIGAND:9425	ncit:C174798	NEMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:540	hgnc:870	ATP7B	GuideToPharmacology	2024.1	blocker	0.8751278539282418	IUPHAR.LIGAND:2328	iuphar.ligand:2328	CHARYBDOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:545	hgnc:882	ATR	GuideToPharmacology	2024.1	blocker	0.3500511415712967	IUPHAR.LIGAND:2328	iuphar.ligand:2328	CHARYBDOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	blocker	4.375639269641208	IUPHAR.LIGAND:11477	iuphar.ligand:11477	JNJ303	FALSE	FALSE	FALSE
NCBIGENE:3082	hgnc:4893	HGF	GuideToPharmacology	2024.1	NULL	1.944728564284981	IUPHAR.LIGAND:10364	iuphar.ligand:10364	NSC61610	FALSE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.1615620653405984	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:2882	hgnc:4559	GPX7	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:8923	iuphar.ligand:8923	OPICINUMAB	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:9391	iuphar.ligand:9391	COMPOUND 36 [PMID: 21958547]	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.1154014752432846	IUPHAR.LIGAND:7731	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	agonist	0.5707355569097228	IUPHAR.LIGAND:2936	iuphar.ligand:2936	2-OLEOYL-LPA	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:2751	iuphar.ligand:2751	24(S), 25-EPOXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:6579	iuphar.ligand:6579	H2L5186303	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8590	iuphar.ligand:8590	ONO-9910539	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:2913	iuphar.ligand:2913	ALKYL OMPT	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8588	iuphar.ligand:8588	ONO-3080573	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1295	iuphar.ligand:1295	S36077	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:1328	iuphar.ligand:1328	HS024	FALSE	FALSE	FALSE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:1322	iuphar.ligand:1322	MS05	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:11292	iuphar.ligand:11292	AP1189	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6214	iuphar.ligand:6214	COMPOUND 11Q [PMID: 19433355]	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3216	iuphar.ligand:3216	FARNESYL THIODIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1393	iuphar.ligand:1393	EGLUMEGAD	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1411	ncit:C169894	DEXFOSFOSERINE	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:9911	iuphar.ligand:9911	TAK-733	FALSE	FALSE	TRUE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:7935	iuphar.ligand:7935	MIRDAMETINIB	FALSE	FALSE	TRUE
ALDH1A2	hgnc:15472	ALDH1A2	NCI	14-Sep-17	NULL	1.166837138570989	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.1136529680426287	IUPHAR.LIGAND:12661	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.1262203635473425	IUPHAR.LIGAND:345	ncit:C152880	VINBURNINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.042073455	IUPHAR.LIGAND:360	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.050488145	IUPHAR.LIGAND:328	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.046059361	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:286	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.022889133	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	ChEMBL	33	inhibitor	0.050007306	MK-8353	iuphar.ligand:9974	MK-8353	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:8215	iuphar.ligand:8215	CCT244747	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.024241769	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.5147810905460245	PEITC	ncit:C2233	PHENETHYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	5-CARBOXAMIDOTRYPTAMINE MALEATE	chembl:CHEMBL1256863	CHEMBL:CHEMBL1256863	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:8583	iuphar.ligand:8583	UH-AH 37	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:286	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:316	rxcui:56092	METHSCOPOLAMINE BROMIDE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:345	ncit:C152880	VINBURNINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.054243462	IUPHAR.LIGAND:355	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.049723174	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1988926940746003	IUPHAR.LIGAND:290	iuphar.ligand:290	MCN-A-343	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:8583	iuphar.ligand:8583	UH-AH 37	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:7438	rxcui:155080	METHACHOLINE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1988926940746003	IUPHAR.LIGAND:326	iuphar.ligand:326	LITHOCHOLYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:8591	iuphar.ligand:8591	ML381	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.7955707762984014	IUPHAR.LIGAND:7631	iuphar.ligand:7631	ML375	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.7955707762984014	IUPHAR.LIGAND:3257	iuphar.ligand:3257	VU0238429	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.066297565	IUPHAR.LIGAND:360	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:1360	iuphar.ligand:1360	S20928	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	1.419126249613364	IUPHAR.LIGAND:7778	iuphar.ligand:7778	CBOBNEA	FALSE	FALSE	FALSE
NCBIGENE:970	hgnc:11937	CD70	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:4838	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 23 MEMBER 2	hgnc:10973	SLC23A2	TTD	2020.06.01	NULL	2.019525816757481	Vitamin C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
NCBIGENE:3004	hgnc:4712	GZMM	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9934	iuphar.ligand:9934	COMPOUND 87 [PMID: 20942471]	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	activator	0.9546849315580819	IUPHAR.LIGAND:2619	iuphar.ligand:2619	BATRACHOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:981	hgnc:23089	SLC13A5	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:11242	iuphar.ligand:11242	BI01383298	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11734	iuphar.ligand:11734	ZANDATRIGINE	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:4007	iuphar.ligand:4007	&ALPHA;-CONOTOXIN ARIB	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:2131	iuphar.ligand:2131	SB 222200	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1475	iuphar.ligand:1475	[125I]NEUROMEDIN U-23 (RAT)	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	N-(3-METHOXYPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1328677	CHEMBL:CHEMBL1328677	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	inhibitor	0.175610941	IUPHAR.LIGAND:3439	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
NCBIGENE:1763	hgnc:2939	DNA2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8887	iuphar.ligand:8887	ML130	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	inhibitor	0.008746905	IUPHAR.LIGAND:1024	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.1831662950082366	OXYMETAZOLINE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1027	hgnc:1785	CDKN1B	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:8798	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
NCBIGENE:1025	hgnc:1780	CDK9	GuideToPharmacology	2024.1	inhibitor	0.1767935058440892	IUPHAR.LIGAND:4357	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TEND	1-Aug-11	NULL	1.071585127259071	COAGULATION FACTOR VIIA	rxcui:2386863	COAGULATION FACTOR VIIA (RECOMBINANT)-JNCW	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.1909369863116163	IUPHAR.LIGAND:10615	ncit:C169802	BALOVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.2386712328895204	IUPHAR.LIGAND:2187	iuphar.ligand:2187	D[CHA4]AVP	FALSE	FALSE	FALSE
NCBIGENE:1276	hgnc:8109	ODC1	GuideToPharmacology	2024.1	inhibitor	2.864054794674245	IUPHAR.LIGAND:5176	rxcui:569	EFLORNITHINE	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2249	iuphar.ligand:2249	L-368,899	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:2219	iuphar.ligand:2219	D(CH2)5[TYR(ME)2,THR4,PHE(3I,4N3)-NH29]OVT	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	REV-5901	chembl:CHEMBL8747	REV-5901	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:1723	iuphar.ligand:1723	MRS2496	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:1739	iuphar.ligand:1739	REACTIVE BLUE-2	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:3883	iuphar.ligand:3883	GYPGKF-NH2	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	METHOXYARACHIDONOYL FLUOROPHOSPHONATE	chembl:CHEMBL113262	METHOXYARACHIDONOYL FLUOROPHOSPHONATE	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.061197752	IUPHAR.LIGAND:7186	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:12737	ncit:C166556	LANIFIBRANOR	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:2688	iuphar.ligand:2688	L-783483	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.036770078	IUPHAR.LIGAND:2694	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:2703	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2677	iuphar.ligand:2677	MK-0767	FALSE	FALSE	FALSE
AQP1	hgnc:633	AQP1	NCI	14-Sep-17	NULL	0.16256245	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:6743	iuphar.ligand:6743	MRL24	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:10030	iuphar.ligand:10030	VCE-004.3	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:11204	iuphar.ligand:11204	AZD8154	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.2949869170544634	IUPHAR.LIGAND:10234	iuphar.ligand:10234	COMPOUND 22 [PMID: 24754609]	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	inhibitor	0.018385039	IUPHAR.LIGAND:2714	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1966579447029756	IUPHAR.LIGAND:12720	iuphar.ligand:12720	PF-06843195	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.084281976	IUPHAR.LIGAND:9425	ncit:C174798	NEMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:7963	iuphar.ligand:7963	PILARALISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:10702	iuphar.ligand:10702	COMPOUND 15A [PMID: 32069401]	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.026045472	IUPHAR.LIGAND:6004	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
TNFRSF10A	hgnc:11904	TNFRSF10A	TALC	12-May-16	agonist	42.00613698855559	MAPATUMUMAB	ncit:C61502	MAPATUMUMAB	FALSE	TRUE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.017859752	IUPHAR.LIGAND:7955	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:9636	iuphar.ligand:9636	INAVOLISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:8917	iuphar.ligand:8917	AMG319	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:10234	iuphar.ligand:10234	COMPOUND 22 [PMID: 24754609]	FALSE	FALSE	FALSE
NCBIGENE:1310	hgnc:2196	COL19A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8757	iuphar.ligand:8757	COMPOUND 27 [PMID: 22142545]	FALSE	FALSE	FALSE
NCBIGENE:3207	hgnc:5101	HOXA11	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12222	iuphar.ligand:12222	COMPOUND 1 [PMID: 26055709]	FALSE	FALSE	FALSE
NCBIGENE:1299	hgnc:2219	COL9A3	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:5167	ncit:C76315	CILOSTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:5167	ncit:C76315	CILOSTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1314	hgnc:2230	COPA	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10400	iuphar.ligand:10400	PDE4 INHIBITOR 16	FALSE	FALSE	FALSE
NCBIGENE:1314	hgnc:2230	COPA	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:4743	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.2143170254518143	IUPHAR.LIGAND:10626	ncit:C124226	UZANSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2738	hgnc:4320	GLI4	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:12206	iuphar.ligand:12206	GNE-064	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:12806	iuphar.ligand:12806	COMPOUND 9 [LIN ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.1256164383629055	IUPHAR.LIGAND:7736	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NCBIGENE:3145	hgnc:4982	HMBS	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11166	iuphar.ligand:11166	GNF-6231	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.1422972120208522	IUPHAR.LIGAND:3448	iuphar.ligand:3448	ZK112993	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:5574	iuphar.ligand:5574	[ALA1,12,AIB3,GLN10,HARG11,TRP14,ARG19]PTH-(1-28)-NH2 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1797	iuphar.ligand:1797	[ILE5,TRP23,TYR36]PTHRP-(1-36)-NH2 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:4448	rxcui:32915	TERIPARATIDE	TRUE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1790	iuphar.ligand:1790	PTHRP-(1-36)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1809	iuphar.ligand:1809	[TRP23]PTHRP-(1-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:9815	iuphar.ligand:9815	CCT196969	FALSE	FALSE	FALSE
NCBIGENE:2144	hgnc:8812	PDK4	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9350	iuphar.ligand:9350	VER-246608	FALSE	FALSE	FALSE
NCBIGENE:737	hgnc:20573	PANX3	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:12096	ncit:C175553	TINLORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:9749	iuphar.ligand:9749	6E11	FALSE	FALSE	FALSE
NCBIGENE:1293	hgnc:2213	COL6A3	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:7917	iuphar.ligand:7917	ESI-09	FALSE	FALSE	FALSE
NCBIGENE:3016	hgnc:9878	RASGRP1	GuideToPharmacology	2024.1	activator	5.834185692854944	IUPHAR.LIGAND:10066	iuphar.ligand:10066	RASGRP ACTIVATOR 1	FALSE	FALSE	FALSE
NCBIGENE:1292	hgnc:2212	COL6A2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7917	iuphar.ligand:7917	ESI-09	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8197	iuphar.ligand:8197	COMPOUND 11D [DOI: 10.1039/C0MD00194E]	FALSE	FALSE	FALSE
NCBIGENE:2630	hgnc:4178	GBA1LP	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12113	iuphar.ligand:12113	TAS1553	FALSE	FALSE	FALSE
NCBIGENE:1528	hgnc:2570	CYB5A	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9358	iuphar.ligand:9358	FMK	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:5398	iuphar.ligand:5398	[125I]RELAXIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	inhibitor	0.1835932560688619	IUPHAR.LIGAND:551	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:2925	iuphar.ligand:2925	AUY954	FALSE	FALSE	FALSE
NCBIGENE:2198	ncbigene:2198	FAUNA@	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9581	iuphar.ligand:9581	ARN-3236	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:11311	drugbank:DB11987	GSK-2018682	FALSE	FALSE	FALSE
NCBIGENE:2632	hgnc:4180	GBE1	GuideToPharmacology	2024.1	activator	2.625383561784724	IUPHAR.LIGAND:6811	rxcui:221095	ENOXAPARIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2714	ncbigene:2714	GKP4	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8953	iuphar.ligand:8953	BAY-598	FALSE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:12335	rxcui:2627044	BEXAGLIFLOZIN	TRUE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:9394	ncit:C166685	IPRAGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:8312	rxcui:2638675	SOTAGLIFLOZIN	TRUE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:9395	ncit:C152676	TOFOGLIFLOZIN ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:4594	rxcui:1486966	DAPAGLIFLOZIN PROPANEDIOL	TRUE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:10428	iuphar.ligand:10428	COMPOUND 25 [PMID: 31260299]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2037	iuphar.ligand:2037	BIM 23059	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2005	iuphar.ligand:2005	CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:2070	iuphar.ligand:2070	BN-81,644	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2014	iuphar.ligand:2014	L-362,855	FALSE	FALSE	FALSE
NCBIGENE:2418	hgnc:3929	FRA8A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:11956	iuphar.ligand:11956	N-0385	FALSE	FALSE	FALSE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:12611	ncit:C174060	BASROPARIB	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.2273059360852575	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:2262	hgnc:4453	GPC5	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
NCBIGENE:1722	hgnc:7217	MPL	GuideToPharmacology	2024.1	agonist	2.983390411119005	IUPHAR.LIGAND:6961	rxcui:711942	ELTROMBOPAG	TRUE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.084963869	IUPHAR.LIGAND:2636	iuphar.ligand:2636	RT3	FALSE	FALSE	FALSE
NCBIGENE:2526	hgnc:4015	FUT4	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12154	iuphar.ligand:12154	MITIPERSTAT	FALSE	FALSE	FALSE
NCBIGENE:1757	hgnc:10536	SARDH	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:11307	ncit:C177069	ENPATORAN	FALSE	FALSE	FALSE
NCBIGENE:1795	hgnc:2989	DOCK3	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:8155	iuphar.ligand:8155	COMPOUND 13A [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6472	iuphar.ligand:6472	DIBENZOXAZEPINE	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6296	iuphar.ligand:6296	NITROOLEIC ACID	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:4134	iuphar.ligand:4134	AP18	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:4134	iuphar.ligand:4134	AP18	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	1.544343271638073	IUPHAR.LIGAND:12526	iuphar.ligand:12526	OPTODARG	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:4309	iuphar.ligand:4309	SB366791	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:2460	iuphar.ligand:2460	BCTC	FALSE	FALSE	FALSE
NCBIGENE:508	ncbigene:508	ATP5BL2	GuideToPharmacology	2024.1	blocker	0.3454452054979901	IUPHAR.LIGAND:7216	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:6347	iuphar.ligand:6347	AMG 9810	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.3723948314588262	IUPHAR.LIGAND:9399	iuphar.ligand:9399	MPI-0479605	FALSE	FALSE	FALSE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.060772768	IUPHAR.LIGAND:2770	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2272	iuphar.ligand:2272	PG 99-465	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2190	iuphar.ligand:2190	D[LEU4]AVP	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2194	iuphar.ligand:2194	L023103	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:1513	iuphar.ligand:1513	PANCREATIC POLYPEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1515	iuphar.ligand:1515	PEPTIDE YY	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.6482428547616604	IUPHAR.LIGAND:1546	iuphar.ligand:1546	[PRO34]PYY (HUMAN)	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.009471081	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.020320306	PILARALISIB	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	CIViC	10-Apr-24	NULL	0.005085489	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	CIViC	10-Apr-24	NULL	0.128537751	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.012026494	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.018540844	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.2778183663264259	ANTI-PD1 MONOCLONAL ANTIBODY	ncit:C128037	ANTI-PD1 MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.092606122	ANTI-PD-L1 MONOCLONAL ANTIBODY	ncit:C128057	ANTI-PD-L1 MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
ACVR1	hgnc:171	ACVR1	CIViC	10-Apr-24	NULL	2.500365296937833	MEK-1/MEKK-1 INHIBITOR E6201	ncit:C79848	MEK-1/MEKK-1 INHIBITOR E6201	FALSE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.018540844	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.016086909	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.2792961235941196	PIDNARULEX	ncit:C126798	PIDNARULEX	FALSE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	CIViC	10-Apr-24	NULL	1.458546423213736	ANTI-PD-1 MONOCLONAL ANTIBODY MEDI0680	ncit:C113332	ANTI-PD-1 MONOCLONAL ANTIBODY MEDI0680	FALSE	FALSE	TRUE
KDM6A	hgnc:12637	KDM6A	CIViC	10-Apr-24	NULL	10.50153424713889	EZH2 INHIBITOR	ncit:C156804	EZH2 INHIBITOR	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.029465584	SAPANISERTIB	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	0.1088116604009326	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CRBN	hgnc:30185	CRBN	CIViC	10-Apr-24	NULL	0.8975670296699916	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.047432404	NVP-AST487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1773907812016706	PI3KBETA INHIBITOR AZD8186	ncit:C107684	PI3KBETA INHIBITOR AZD8186	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	CIViC	10-Apr-24	NULL	0.1283806142682017	MUTANT IDH1 INHIBITOR DS-1001	ncit:C148134	SAFUSIDENIB	FALSE	FALSE	TRUE
CSF3R	hgnc:2439	CSF3R	CIViC	10-Apr-24	NULL	1.306751999078369	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.02726255	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
CSF3R	hgnc:2439	CSF3R	DoCM	10-Apr-24	NULL	1.306751999078369	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DoCM	10-Apr-24	NULL	0.2007335520076852	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
BTK	hgnc:1133	BTK	DoCM	10-Apr-24	NULL	0.4055851016423223	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	DoCM	10-Apr-24	NULL	0.6168664383892681	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
PLCG2	hgnc:9066	PLCG2	DoCM	10-Apr-24	NULL	4.773424657790409	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.011273789	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.4565884455277782	HJC0152	iuphar.ligand:12140	HJC0152	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.040230625	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	PF-00477736	chembl:CHEMBL3545137	PF-00477736	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	ERAS-007	ncit:C150248	ERK1/2 INHIBITOR ERAS-007	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	PF-07284890	ncit:C175553	TINLORAFENIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.005912027	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.026181836	Entinostat	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	AZD3514	chembl:CHEMBL2346976	AZD3514	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.024991752	Axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	SY-5609	drugbank:DB17099	SY-5609	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.042293734	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.054355767	Ixazomib	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.084214389	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1547594520630995	Nintedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	Alofanib	ncit:C170744	ALOFANIB	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.02654584	Dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.6326225450083675	THE-630	drugbank:DB16750	THE-630	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.1265245090016735	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.375054795	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.086361301	Dacinostat	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.078136416	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	1.312691780892362	Milademetan	ncit:C141432	MILADEMETAN	FALSE	FALSE	FALSE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.8751278539282416	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.2243917574174979	Baicalein	rxcui:1592893	BAICALEIN	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	ASTX029	iuphar.ligand:11727	ASTX029	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	GDC-0623	drugbank:DB11982	GDC-0623	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.056459862	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.4145342465975881	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.094535416	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	TGX-221	iuphar.ligand:8244	TGX-221	FALSE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	0.4487835148349957	Tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.011858101	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.02896176	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.01689436	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.034612835	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.05068308	Vistusertib	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.047304208	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.9723642821424906	Telaglenastat	ncit:C114381	TELAGLENASTAT	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1440539677248134	Apitolisib	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1944728564284981	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CancerCommons	25-Jul-13	inhibitor	0.094535416	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	CancerCommons	25-Jul-13	inhibitor	0.2311077079035849	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.4688184931758437	LEVETIRACETAM	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	blocker	0.546954909	Z160	iuphar.ligand:7765	NP118809	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.037948209	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.051885051	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
C18ORF21	hgnc:28802	C18orf21	PharmGKB	4/5/24	NULL	3.750547945406749	ibutilide	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
ALDH3A1	hgnc:405	ALDH3A1	PharmGKB	4/5/24	NULL	0.020002922	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:10156	iuphar.ligand:10156	JAK3 INHIBITOR 32	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5805	iuphar.ligand:5805	PFIZER COMPOUND 67 [PMID:18445527]	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:7947	ncit:C79844	VOLASERTIB	FALSE	FALSE	TRUE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.042898424	IUPHAR.LIGAND:2714	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.061628722	MTOR INHIBITOR	ncit:C2201	MTOR INHIBITOR	FALSE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	CHRYSOPHANOL	chembl:CHEMBL41092	CHRYSOPHANOL	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1161674142382621	sulfisoxazole	rxcui:10207	SULFISOXAZOLE	TRUE	FALSE	FALSE
COL2A1	hgnc:2200	COL2A1	PharmGKB	4/5/24	NULL	2.692701089009974	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	GNF-PF-1529	chembl:CHEMBL586078	CHEMBL:CHEMBL586078	FALSE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	0.2651902587661338	Pyrimethamine	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:5907	iuphar.ligand:5907	AR-C118925XX	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.006496866	IUPHAR.LIGAND:2200	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	CGI	2/1/22	NULL	0.1017590527823536	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NDUFB4	hgnc:7699	NDUFB4	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
PSMB11	hgnc:31963	PSMB11	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.052090944	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
UNIPROT:P49768	hgnc:9508	PSEN1	TdgClinicalTrial	Jan-14	NULL	0.577007376	GSI-136	drugbank:DB12819	GSI-136	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.1280674908187671	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.16256245	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.036387853	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
NCBIGENE:2985	hgnc:3621	FCGRT	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:9801	iuphar.ligand:9801	ROZANOLIXIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:6088	iuphar.ligand:6088	GALANIN(1-19) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.018540844	IUPHAR.LIGAND:6000	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1824	iuphar.ligand:1824	[ILE5,TRP23]PTHRP-(5-36) (HUMAN)	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	IMM-1-104	ncit:C192810	MEK INHIBITOR IMM-1-104	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.5357925636295356	RISLENEMDAZ	ncit:C152228	RISLENEMDAZ	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.066297565	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	CICLOPIROX OLAMINE	rxcui:52172	CICLOPIROX OLAMINE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.2734774543525755	SK&F-86466	chembl:CHEMBL123349	CHEMBL:CHEMBL123349	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001701921	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.061992528	IUPHAR.LIGAND:384	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:12766	ncit:C171708	TOLUDESVENLAFAXINE	FALSE	FALSE	FALSE
CCNE1	hgnc:1589	CCNE1	CIViC	10-Apr-24	NULL	0.8751278539282416	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	5.250767123569449	PEGINESATIDE ACETATE	rxcui:1248797	PEGINESATIDE ACETATE	TRUE	FALSE	FALSE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	1.750255707856483	MYCOPHENOLATE MOFETIL HYDROCHLORIDE	rxcui:237112	MYCOPHENOLATE MOFETIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1411496538593938	IUPHAR.LIGAND:5992	drugbank:DB04716	2-TERT-BUTYL-9-FLUORO-1,6-DIHYDROBENZO[H]IMIDAZO[4,5-F]ISOQUINOLIN-7-ONE	FALSE	FALSE	TRUE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1041818873724097	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	(-)-U-50488	chembl:CHEMBL58033	(-)-U-50488	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.00962384	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	2'-EPI-TUBERATOLIDE B	chembl:CHEMBL1668775	2'-EPI-TUBERATOLIDE B	FALSE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.5147810905460244	ELETRIPTAN	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1077080435603989	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.2692701089009974	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.3431873936973496	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TEND	1-Aug-11	NULL	0.6081969641200136	RASAGILINE	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:8170	iuphar.ligand:8170	COMPOUND 8H [PMID: 21561767]	FALSE	FALSE	FALSE
TPH1	hgnc:12008	TPH1	ChEMBL	33	inhibitor	6.563458904461812	TELOTRISTAT ETHYL	rxcui:1872441	TELOTRISTAT ETHYL	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.375054795	NORHARMANE	iuphar.ligand:8222	BETA-CARBOLINE	FALSE	FALSE	FALSE
STAT2	hgnc:11363	STAT2	NCI	14-Sep-17	NULL	6.563458904461812	13-CIS-RETINOIC ACID	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9919	iuphar.ligand:9919	SELATINIB	FALSE	FALSE	FALSE
MIF	hgnc:7097	MIF	NCI	14-Sep-17	NULL	2.500365296937833	PPD	rxcui:1362740	4-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.3777530304726222	IUPHAR.LIGAND:9792	drugbank:DB15396	VAMOTINIB	FALSE	FALSE	FALSE
PIP4K2A	hgnc:8997	PIP4K2A	DTC	9/2/20	NULL	0.8078103267029924	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
EIF4E	hgnc:3287	EIF4E	NCI	14-Sep-17	NULL	0.6035364509849942	MTOR INHIBITOR	ncit:C2201	MTOR INHIBITOR	FALSE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.020257589	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SLC2A3	hgnc:11007	SLC2A3	NCI	14-Sep-17	NULL	0.8078103267029924	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.028626235	THIORIDAZINE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.045579576	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
NPEPPS	hgnc:7900	NPEPPS	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.108711535	PERZINFOTEL	ncit:C72122	PERZINFOTEL	FALSE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	DTC	9/2/20	NULL	1.591141552596803	PHANTASMIDINE	chembl:CHEMBL1086654	PHANTASMIDINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2035181055647073	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	AG1295	iuphar.ligand:5914	AG 1295	FALSE	FALSE	TRUE
KAT5	hgnc:5275	KAT5	DTC	9/2/20	NULL	17.50255707856483	6-DECYLSALICYLIC ACID	chembl:CHEMBL416038	CHEMBL:CHEMBL416038	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.097236428	BUPRENORPHINE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:5706	iuphar.ligand:5706	TAMATINIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.070244376	Saracatinib	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.002861999	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.009862448	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.1060761035064535	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	0.3818739726232327	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NCBIGENE:434	hgnc:745	ASIP	GuideToPharmacology	2024.1	activator	10.50153424713889	IUPHAR.LIGAND:7768	iuphar.ligand:7768	ML297	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	MyCancerGenome	20-Jun-17	inhibitor	0.4375639269641208	GSK461364	ncit:C70948	POLO-LIKE KINASE 1 INHIBITOR GSK461364	FALSE	FALSE	TRUE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	1.584283183835609	AMONAFIDE	rxcui:1440270	AMONAFIDE	FALSE	FALSE	FALSE
UNIPROT:P08254	hgnc:7173	MMP3	TdgClinicalTrial	Jan-14	NULL	0.7501095890813501	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
PLATELET-DERIVED GROWTH FACTOR B	hgnc:8800	PDGFB	TTD	2020.06.01	NULL	2.917092846427472	PDGF-BB	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.2083637747448194	TGR-1202	rxcui:2478439	UMBRALISIB	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:10462	iuphar.ligand:10462	IMNOPITANT	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:11919	iuphar.ligand:11919	INSL5-A13NR	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	2.341819737097098	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.6226206075378794	bromperidol	rxcui:19777	BROMPERIDOL	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.1235474617310458	ETILEVODOPA	rxcui:1421444	ETILEVODOPA	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	4.039051633514961	Pegfilgrastim	rxcui:2048018	PEGFILGRASTIM-JMDB	TRUE	FALSE	FALSE
METHIONINE AMINOPEPTIDASE 2	hgnc:16672	METAP2	TTD	2020.06.01	NULL	13.12691780892362	PPI-2458	drugbank:DB05864	PPI-2458	FALSE	FALSE	FALSE
RXFP2	hgnc:17318	RXFP2	DTC	9/2/20	NULL	1.250182648468916	N6-PHENYLADENOSINE	chembl:CHEMBL262083	N6-PHENYLADENOSINE	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	Levalbuterol	rxcui:237159	LEVALBUTEROL	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	4.375639269641208	Insulin Zinc Susp Recombinant Human	chembl:CHEMBL1201644	INSULIN ZINC SUSP RECOMBINANT HUMAN	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:5933	iuphar.ligand:5933	AZD1480	FALSE	FALSE	TRUE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:12335	rxcui:2627044	BEXAGLIFLOZIN	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	0.5385402178019949	CLORGILINE	ncit:C77522	CLORGILINE	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.5147810905460244	AT-13148	chembl:CHEMBL3544960	AT-13148	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.033338204	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.035216413	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
ITGA5	hgnc:6141	ITGA5	ChEMBL	33	inhibitor	1.640864726115453	ATN-161	drugbank:DB05491	ATN-161	FALSE	FALSE	FALSE
NDUFS4	hgnc:7711	NDUFS4	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.42006137	BALAGLITAZONE	ncit:C78125	BALAGLITAZONE	FALSE	FALSE	FALSE
PSMD2	hgnc:9559	PSMD2	ChEMBL	33	inhibitor	0.5385402178019948	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.019447286	Nintedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.022249013	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.4150804050252529	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	7-METHOXY-BAPTIGENIN	chembl:CHEMBL583578	CHEMBL:CHEMBL583578	FALSE	FALSE	FALSE
SOLUBLE EPOXIDE HYDROLASE	hgnc:3402	EPHX2	TTD	2020.06.01	NULL	2.250328767244049	AR9281	drugbank:DB06345	AR-9281	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	Propoxyphene Hydrochloride	rxcui:71517	PROPOXYPHENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2768	hgnc:4380	GNA12	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7419	ncit:C82174	ZOPOLRESTAT	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.007496384	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	binder	2.282942227638891	YTTRIUM Y 90 LABETUZUMAB	chembl:CHEMBL2108818	YTTRIUM Y 90 LABETUZUMAB	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	agonist	0.038159645	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.1579178082276526	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
RARA	hgnc:9864	RARA	ChEMBL	33	agonist	0.1511209794852536	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.42006137	TCMDC-124022	chembl:CHEMBL548017	CHEMBL:CHEMBL548017	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:3290	ncit:C74246	APADENOSON	FALSE	FALSE	FALSE
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	1.125164383622024	USTEKINUMAB	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.210030685	dimercaprol	rxcui:3445	DIMERCAPROL	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.018974104	levomepromazine	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:P10398	hgnc:646	ARAF	TdgClinicalTrial	Jan-14	NULL	0.6364566210387211	XL281	drugbank:DB05190	XL281	FALSE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:5924	drugbank:DB07364	6-PHENYL[5H]PYRROLO[2,3-B]PYRAZINE	FALSE	FALSE	FALSE
NCBIGENE:2789	hgnc:4409	GNG5P1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12154	iuphar.ligand:12154	MITIPERSTAT	FALSE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.3125456621172291	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	PD-146176	iuphar.ligand:11390	PD-146176	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4154	iuphar.ligand:4154	CGP37849	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.103633562	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.059030547	ANTIPSYCHOTIC AGENT	ncit:C29710	ANTIPSYCHOTIC AGENT	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2081	iuphar.ligand:2081	H-C[DCYS-PHE-LAGL(N&BETA;ME,BENZOYL)-DTRP-LYS-THR-PHE-CYS]-OH	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.016429184	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.020836377	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7498	rxcui:1796	BUFEXAMAC	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	MMV007764	chembl:CHEMBL609628	CHEMBL:CHEMBL609628	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1700	iuphar.ligand:1700	[ALA11, D-LEU15]OREXIN-B	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.2210849315187137	RO4987655	ncit:C82696	MEK INHIBITOR RO4987655	FALSE	FALSE	TRUE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	1.810609352954982	E1001	chembl:CHEMBL1255831	E1001	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.9293393139060973	THEONELLASTEROL D	chembl:CHEMBL1782600	THEONELLASTEROL D	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.5114383561918295	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:1546	iuphar.ligand:1546	[PRO34]PYY (HUMAN)	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.087512785	NEOMYCIN	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	NCI	14-Sep-17	NULL	0.035083077	DIHYDROTESTOSTERONE	ncit:C29619	DIHYDROTESTOSTERONE	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	PharmGKB	4/5/24	NULL	0.046059361	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	GNF-PF-4085	chembl:CHEMBL528181	CHEMBL:CHEMBL528181	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	L-750667	iuphar.ligand:978	L-750,667	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	TUBERATOLIDE B	chembl:CHEMBL1668774	TUBERATOLIDE B	FALSE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12080	iuphar.ligand:12080	EDECESERTIB	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.041150213	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.1547594520630995	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	inhibitor	0.3000438356325399	IUPHAR.LIGAND:1606	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.090634645	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.375054795	IL-5	iuphar.ligand:4997	IL-5	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1944728564284981	NOMIFENSINE MALEATE	rxcui:262302	NOMIFENSINE MALEATE	TRUE	FALSE	FALSE
PTGFR	hgnc:9600	PTGFR	ChEMBL	33	agonist	1.250182648468916	DINOPROST TROMETHAMINE	rxcui:23321	DINOPROST TROMETHAMINE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.093098708	TREQUINSIN	ncit:C152731	TREQUINSIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.045461187	DNDI1417719	chembl:CHEMBL1420370	CHEMBL:CHEMBL1420370	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	ARASERTACONAZOLE	ncit:C79926	ARASERTACONAZOLE	FALSE	FALSE	FALSE
CTSB	hgnc:2527	CTSB	NCI	14-Sep-17	NULL	2.187819634820604	COUMARIN	rxcui:2898	COUMARIN	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:1957	iuphar.ligand:1957	[3H]PGF2&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1731	iuphar.ligand:1731	5BRUTP	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.5672124979164529	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CHLOROXYLENOL	rxcui:20877	CHLOROXYLENOL	TRUE	FALSE	FALSE
DTNBP1	hgnc:17328	DTNBP1	PharmGKB	4/5/24	NULL	0.8751278539282416	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:P38435	hgnc:4247	GGCX	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	ANISINDIONE	rxcui:17941	ANISINDIONE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.082429625	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3896	iuphar.ligand:3896	M15	FALSE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.1785975212098452	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:5841	iuphar.ligand:5841	FMET-ILE-VAL-THR-LEU-PHE	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.021484317	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	0.2692701089009974	Chloroprocaine	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TEND	1-Aug-11	NULL	0.4892019059226195	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:6048	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
PSMC4	hgnc:9551	PSMC4	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CancerCommons	25-Jul-13	inhibitor	0.6721614540713904	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:8591	iuphar.ligand:8591	ML381	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.061055432	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.067317527	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.1233298208706858	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:12078	iuphar.ligand:12078	INIXACICLIB	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:7556	ncit:C66358	PEROSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:768	iuphar.ligand:768	VMIP-II	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,7-BIS[3-(PIPERAZINO)PROPIONAMIDO]ANTHRAQUINONE	chembl:CHEMBL520095	CHEMBL:CHEMBL520095	FALSE	FALSE	FALSE
RHOB	hgnc:668	RHOB	DTC	9/2/20	NULL	23.33674277141977	NSC-126188	chembl:CHEMBL1797159	CHEMBL:CHEMBL1797159	FALSE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.1235474617310458	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CD3EAP	hgnc:24219	POLR1G	PharmGKB	4/5/24	NULL	0.2414145803939976	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NGB	hgnc:14077	NGB	NCI	14-Sep-17	NULL	26.25383561784724	SODIUM SALICYLATE	rxcui:9907	SODIUM SALICYLATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.003936697	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.092851762	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TEND	1-Aug-11	NULL	0.2027323213733378	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	CINOBUFOTALIN	ncit:C151929	CINOBUFOTALIN	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	JCAR017	ncit:C125192	LISOCABTAGENE MARALEUCEL	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	8.078103267029922	MK 1775	hemonc:32625	ADAVOSERTIB	FALSE	FALSE	TRUE
IL6ST	hgnc:6021	IL6ST	DTC	9/2/20	NULL	0.7001022831425933	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.078722146	12-O-TETRADECANOYLPHORBOL-13-ACETATE	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
TAT	hgnc:11573	TAT	NCI	14-Sep-17	NULL	0.2592971419046642	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.068847471	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
NDUFS2	hgnc:7708	NDUFS2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:412	hgnc:11425	STS	GuideToPharmacology	2024.1	blocker	0.1521961485092594	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	0.8401227397711121	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:12582	rxcui:2580	CLENBUTEROL	TRUE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:12354	iuphar.ligand:12354	COMPOUND G1 [PMID: 36689364]	FALSE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	activator	0.1773907812016706	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.4861821410712453	ANTIPSYCHOTIC AGENT	ncit:C29710	ANTIPSYCHOTIC AGENT	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:12661	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.031861451	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1442518440541057	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.009320613	aripiprazole lauroxil	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.057574201	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6358	iuphar.ligand:6358	COMPOUND 22 [PMID: 17276684]	FALSE	FALSE	FALSE
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	1.009762908	oxazepam	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.031659735	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	METOLAZONE	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	ROXINDOLE	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	PharmGKB	4/5/24	NULL	0.014385663	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.1178623372293928	VCR	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
T-CELL ANTIGEN CD7	hgnc:1695	CD7	TTD	2020.06.01	NULL	26.25383561784724	Anti-CD7 CAR-T cells	ncit:C201177	ANTI-CD7 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
NCBIGENE:2939	hgnc:4627	GSTA2	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:11649	iuphar.ligand:11649	FELADILIMAB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.059397818	IUPHAR.LIGAND:7794	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.025942525	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
CD3EAP	hgnc:24219	POLR1G	PharmGKB	4/5/24	NULL	1.666910197958555	melphalan	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	NSC-67746	chembl:CHEMBL333177	CHEMBL:CHEMBL333177	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.013673873	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	1.500219178162699	HMBA	ncit:C1125	HEXAMETHYLENE BISACETAMIDE	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	1.090323227845022	CP-868596	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.089756703	NOREPINEPHRINE BITARTRATE	rxcui:7508	NOREPINEPHRINE BITARTRATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.049192122	Modafinil	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9909	iuphar.ligand:9909	GDC-0623	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	1.875273972703375	NSC-675972	chembl:CHEMBL1379243	CHEMBL:CHEMBL1379243	FALSE	FALSE	FALSE
NOTCH2	hgnc:7882	NOTCH2	CGI	2/1/22	NULL	15.00219178	OMP-59R5	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.2213645498975316	eliglustat	rxcui:1547220	ELIGLUSTAT	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.063110182	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.5114383561918295	REFAMETINIB	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.052639269	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
LYSYL HYDROXYLASE 1	hgnc:9081	PLOD1	TTD	2020.06.01	NULL	2.019525816757481	Ascorbate	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	ChEMBL	33	agonist	6.563458904461812	TELRATOLIMOD	ncit:C124653	TELRATOLIMOD	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.03357268	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.045579576	A-70108	iuphar.ligand:6077	A68930	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.1325951293830669	AVUTOMETINIB	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.032899543	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	FLEROXACIN	rxcui:42322	FLEROXACIN	FALSE	FALSE	FALSE
GSTM3	hgnc:4635	GSTM3	PharmGKB	4/5/24	NULL	0.2333674277141977	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	SKF-75670 HYDROBROMIDE	chembl:CHEMBL1256698	CHEMBL:CHEMBL1256698	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.3860858179095183	Lorcaserin	rxcui:1300701	LORCASERIN	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	0.6819178082557728	Tubocurarine	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TEND	1-Aug-11	NULL	0.7292732116068681	GOSERELIN	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.2224901323546377	CIS(Z)-FLUPENTIXOL DIHYDROCHLORIDE	chembl:CHEMBL1496351	CHEMBL:CHEMBL1496351	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(+)-3-DEOXYTHYSANONE	chembl:CHEMBL593570	CHEMBL:CHEMBL593570	FALSE	FALSE	FALSE
NCBIGENE:630	hgnc:7981	NR4A2	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:12997	iuphar.ligand:12997	COMPOUND 111 [PMID: 37918435]	FALSE	FALSE	FALSE
NCBIGENE:2709	hgnc:4287	GJB5	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8778	iuphar.ligand:8778	COMPOUND 17 [PMID: 23570514]	FALSE	FALSE	FALSE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2651902587661338	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.019339842	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	SJ000160630	chembl:CHEMBL591404	CHEMBL:CHEMBL591404	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.001937267	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5672124979164529	4'-N-BENZOYLSTAUROSPORINE	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.023823807	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5996	iuphar.ligand:5996	JNK INHIBITOR IX	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.2778183663264259	SYM004	ncit:C91381	FUTUXIMAB/MODOTUXIMAB MIXTURE	FALSE	TRUE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002796829	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2724	ncbigene:2724	GLC1D	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8573	iuphar.ligand:8573	NI-57	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:12485	iuphar.ligand:12485	COMPOUND 7 [NGUYEN ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	blocker	0.3977853881492007	IUPHAR.LIGAND:3963	ncit:C75979	HEXAMETHONIUM	FALSE	FALSE	FALSE
UNIPROT:P24394	hgnc:6015	IL4R	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	PRX-321	chembl:CHEMBL4298027	PRX-321	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.039778539	COLFORSIN	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	NCI	14-Sep-17	NULL	0.039793612	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
MYOSIN	hgnc:23212	MYH14	TTD	2020.06.01	NULL	5.834185692854945	Mavacamten	rxcui:2600867	MAVACAMTEN	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.015443433	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
NDUFAF1	hgnc:18828	NDUFAF1	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:376	iuphar.ligand:376	LUF5831	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:6168	iuphar.ligand:6168	[LEU8]-PHYLLOLITORIN	FALSE	FALSE	FALSE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.2243917574174979	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
UNIPROT:Q9NY47	hgnc:1400	CACNA2D2	TEND	1-Aug-11	NULL	0.2812910959055062	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
LEUKOCYTE PROTEINASE-3	hgnc:9495	PRTN3	TTD	2020.06.01	NULL	6.563458904461812	Tiprelestat	ncit:C152650	TIPRELESTAT	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.044763573	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	CROCIN	rxcui:2262278	CROCIN	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:10280	iuphar.ligand:10280	CP-1	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.056097939	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
NCBIGENE:2857	hgnc:4490	GPR34	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	ChEMBL	33	inhibitor	3.281729452230906	METHOTREXATE SODIUM	rxcui:287734	METHOTREXATE SODIUM	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.018918275	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:2814	iuphar.ligand:2814	LG100754	FALSE	FALSE	FALSE
NCBIGENE:1784	ncbigene:1784	DNCM	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:11888	ncit:C175551	ZILURGISERTIB	FALSE	FALSE	FALSE
NCBIGENE:726	hgnc:1482	CAPN5	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.5303805175322677	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.2273059360852575	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	1.544343271638073	Litenimod	ncit:C166612	LITENIMOD	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:847	iuphar.ligand:847	CXCL12-(1-9)	FALSE	FALSE	FALSE
NOTCH-2 RECEPTOR	hgnc:7882	NOTCH2	TTD	2020.06.01	NULL	15.00219178	Tarextumab	ncit:C95719	TAREXTUMAB	FALSE	FALSE	TRUE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3166	iuphar.ligand:3166	NE58062	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	4.118248724368196	MM-121	chembl:CHEMBL2109402	MM-121	FALSE	TRUE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.03357268	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.068191781	IUPHAR.LIGAND:204	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	activator	0.1193356164447602	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.032961501	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	1.312691780892362	Afeletecan	ncit:C79725	AFELETECAN	FALSE	FALSE	FALSE
CYP27A1	hgnc:2605	CYP27A1	PharmGKB	4/5/24	NULL	0.546954909	cholic acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MACROPHAGE MIGRATION INHIBITORY FACTOR	hgnc:7097	MIF	TTD	2020.06.01	NULL	8.751278539282415	ISO-1	iuphar.ligand:9984	ISO-1	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	GNF-PF-2947	chembl:CHEMBL581677	CHEMBL:CHEMBL581677	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.1988926940746003	APRINDINE	rxcui:1054	APRINDINE	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9071	iuphar.ligand:9071	NABILONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.001302144	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2160809515872201	AG1295	iuphar.ligand:5914	AG 1295	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.009779786	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.1831662950082366	OXYMETAZOLINE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	TCMDC-125653	chembl:CHEMBL580918	CHEMBL:CHEMBL580918	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	2,2,3,3,4,4,5,5,6,6,7,7,8,8,8-PENTADECAFLUORO-OCTANOIC ACID	chembl:CHEMBL172988	CHEMBL:CHEMBL172988	FALSE	FALSE	FALSE
RPL17	hgnc:10307	RPL17	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.4861821410712454	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	GNF-PF-4078	chembl:CHEMBL584883	CHEMBL:CHEMBL584883	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	CID 660258	chembl:CHEMBL259805	CHEMBL:CHEMBL259805	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	NOR-BINALTORPHIMINE DIHYDROCHLORIDE	chembl:CHEMBL2374078	CHEMBL:CHEMBL2374078	FALSE	FALSE	FALSE
NCBIGENE:726	hgnc:1482	CAPN5	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.1773907812016706	IUPHAR.LIGAND:7158	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:10489	iuphar.ligand:10489	COMPOUND 12B [PMID: 31465220]	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.596678082	Brasofensine	ncit:C76391	BRASOFENSINE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.050879526	CELIPROLOL	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
KCNC2	hgnc:6234	KCNC2	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.079557078	IUPHAR.LIGAND:286	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.300043836	GNF-PF-1731	chembl:CHEMBL581251	CHEMBL:CHEMBL581251	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DoCM	10-Apr-24	NULL	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
SH2D5	hgnc:28819	SH2D5	PharmGKB	4/5/24	NULL	1.129197231	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.025147352	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	negative modulator	0.1790542923638346	KETAMINE HYDROCHLORIDE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	2-BROMO-HEXADECANOIC ACID	chembl:CHEMBL118417	CHEMBL:CHEMBL118417	FALSE	FALSE	FALSE
UNIPROT:O60840	hgnc:1393	CACNA1F	TEND	1-Aug-11	NULL	0.08334551	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.020986279	CHEMOPREVENTIVE	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	DNDI1416985	chembl:CHEMBL593211	CHEMBL:CHEMBL593211	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.046059361	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	BIOALLETHRIN S-CYCLOPENTENYL ISOMER	chembl:CHEMBL1887350	BIOALLETHRIN S-CYCLOPENTENYL ISOMER	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	PharmGKB	4/5/24	NULL	1.750255707856483	mivacurium	rxcui:30077	MIVACURIUM	TRUE	FALSE	FALSE
NISCH	hgnc:18006	NISCH	ChEMBL	33	agonist	6.563458904461812	RILMENIDINE	rxcui:55679	RILMENIDINE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.058212496	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.031958412	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.2286255641612242	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P54760	hgnc:3395	EPHB4	TdgClinicalTrial	Jan-14	NULL	5.469549087051511	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.07458476	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.070291394	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	KN-62	iuphar.ligand:6001	KN-62	FALSE	FALSE	FALSE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	2.386712328895204	BSO	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
SLC22A17	hgnc:23095	SLC22A17	PharmGKB	4/5/24	NULL	0.3500511415712966	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	CGI	2/1/22	NULL	0.016791708	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	FLOTETUZUMAB	ncit:C117238	FLOTETUZUMAB	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1091635576625665	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	activator	0.1232574442152452	INDOXIMOD	ncit:C71535	INDOXIMOD	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:5965	iuphar.ligand:5965	EGFR/ERBB-2/ERBB-4 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:669	hgnc:1093	BPGM	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:12455	iuphar.ligand:12455	PHENYL-&BETA;-D-GLUCOPYRANOSIDE	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9121	iuphar.ligand:9121	LSN2424100	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	Encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	SUFENTANIL CITRATE	rxcui:58964	SUFENTANIL CITRATE	TRUE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	0.098513454	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.3677319929494733	Lapatinib	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	0.2895643634321387	PYRIDOSTIGMINE	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.088248187	SJ000071854	chembl:CHEMBL602127	CHEMBL:CHEMBL602127	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:9307	iuphar.ligand:9307	MK-3697	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	TRIPARANOL	ncit:C152752	TRIPARANOL	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.087512785	temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SB-262470	iuphar.ligand:716	NPS 2143	FALSE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	2.282942227638891	sofosbuvir	rxcui:1484911	SOFOSBUVIR	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.028498058	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.039068208	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9943	iuphar.ligand:9943	PF-06751979	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	agonist	0.9211872146613068	IUPHAR.LIGAND:3412	iuphar.ligand:3353	LTD4	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-3906	chembl:CHEMBL599102	CHEMBL:CHEMBL599102	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123456	chembl:CHEMBL534084	CHEMBL:CHEMBL534084	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004375639	DECITABINE	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NDUFS8	hgnc:7715	NDUFS8	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFB8	hgnc:7703	NDUFB8	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.027390543	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1376949420516464	FLUVOXAMINE	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:11697	iuphar.ligand:11697	COMPOUND 11D [PMID: 34406006]	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:10649	iuphar.ligand:10649	COMPOUND 7 [PMID: 31955578]	FALSE	FALSE	FALSE
PRKAB1	hgnc:9378	PRKAB1	NCI	14-Sep-17	NULL	0.6250913242344582	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
UGT2B15	hgnc:12546	UGT2B15	PharmGKB	4/5/24	NULL	0.4526523382387457	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	inhibitor	0.077217164	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
PTK6	hgnc:9617	PTK6	DTC	9/2/20	NULL	0.085239726	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	PIRINIXIC ACID	iuphar.ligand:2666	PIRINIXIC ACID	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.1035654265003836	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1296485709523321	DIACEREIN	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	OSM-S-55	chembl:CHEMBL1363033	CHEMBL:CHEMBL1363033	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.3977853881492006	Naproxcinod	ncit:C83989	NAPROXCINOD	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003677523	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.073437302	Ergotamine	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
MAP3K10	hgnc:6849	MAP3K10	DTC	9/2/20	NULL	0.1136529680426288	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
RPL27A	hgnc:10329	RPL27A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.8751278539282416	GIMATECAN	ncit:C65804	GIMATECAN	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	1.381780822	LEPIRUDIN	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:7449	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:2929	iuphar.ligand:2929	COMPOUND 26 [PMID: 16190743]	FALSE	FALSE	FALSE
B3GAT1	hgnc:921	B3GAT1	NCI	14-Sep-17	NULL	11.66837138570989	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003132729	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	5-HYDROXYINDOLE	iuphar.ligand:2295	5-HYDROXYINDOLE	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	2.019525817	Mivebresib	ncit:C121829	MIVEBRESIB	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.073062622	BAY 10-00394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
NF2	hgnc:7773	NF2	CIViC	10-Apr-24	NULL	0.049723174	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.070010228	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.089756703	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:4131	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:1229	iuphar.ligand:1229	BURIMAMIDE	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:2909	iuphar.ligand:2909	VPC12249	FALSE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	PharmGKB	4/5/24	NULL	0.4018444227221517	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
NCBIGENE:543	hgnc:880	ALDH7A1P3	GuideToPharmacology	2024.1	blocker	2.625383561784725	IUPHAR.LIGAND:2328	iuphar.ligand:2328	CHARYBDOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:3448	iuphar.ligand:3448	ZK112993	FALSE	FALSE	FALSE
F11	hgnc:3529	F11	ChEMBL	33	inhibitor	0.6908904109959803	HUMAN C1-ESTERASE INHIBITOR	ncit:C87730	HUMAN C1-ESTERASE INHIBITOR	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.054953083	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:10211	iuphar.ligand:10211	MUTANT ANP	FALSE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1875273972703375	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:2905	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:9258	iuphar.ligand:9258	BIIB021	FALSE	FALSE	FALSE
NCBIGENE:1434	hgnc:2431	CSE1L	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5287	iuphar.ligand:5287	VU0364739	FALSE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.4039051633514961	Renzapride	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.017456008	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	modulator	0.8607814956671229	TELAPRISTONE ACETATE	ncit:C104055	TELAPRISTONE ACETATE	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	1.750255707856483	ATOGEPANT	rxcui:2571813	ATOGEPANT	TRUE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	inhibitor	0.1223955040459079	IUPHAR.LIGAND:150	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.6250913242344582	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.029366707	trimethadione	rxcui:10827	TRIMETHADIONE	TRUE	FALSE	FALSE
PRKAB1	hgnc:9378	PRKAB1	NCI	14-Sep-17	NULL	0.4688184931758437	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.253049018	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.2446009529613098	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.01261294	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1278595890479573	Fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.2625383561784725	FENOPROFEN	rxcui:4331	FENOPROFEN	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	DNDI1417264	chembl:CHEMBL1467200	CHEMBL:CHEMBL1467200	FALSE	FALSE	FALSE
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	0.6604738520213144	MM-141	ncit:C103863	ISTIRATUMAB	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.138178082	AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	Z-PRO-PROLINAL	drugbank:DB03535	Z-PRO-PROLINAL	FALSE	FALSE	FALSE
NCBIGENE:940	hgnc:1653	CD28	GuideToPharmacology	2024.1	inhibitor	0.1842374429322614	IUPHAR.LIGAND:7216	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:9231	ncit:C81420	TARANABANT	FALSE	FALSE	FALSE
NCBIGENE:730	hgnc:1346	C7	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:1640	hgnc:7162	MMP16	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.091796628	IUPHAR.LIGAND:7938	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TEND	1-Aug-11	NULL	1.458546423213736	FONDAPARINUX	rxcui:321208	FONDAPARINUX	TRUE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.9053046764774912	ACETYLCHOLINE CHLORIDE	rxcui:20814	ACETYLCHOLINE CHLORIDE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.013022736	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	CGP-71683A	chembl:CHEMBL17645	CGP-71683A	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.7955707762984014	Bezafibrate	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.075010959	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	2.386712328895204	Benzimidazole	rxcui:1362885	BENZIMIDAZOLE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	CID 5310655	chembl:CHEMBL408563	CHEMBL:CHEMBL408563	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.100976291	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
CEACAM1	hgnc:1814	CEACAM1	NCI	14-Sep-17	NULL	2.187819634820604	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	TALC	12-May-16	inhibitor	0.2692701089009974	NEOVASTAT	drugbank:DB05387	NEOVASTAT	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	7-O-METHYLCRYPTOCHINONE A	chembl:CHEMBL1223742	7-O-METHYLCRYPTOCHINONE A	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.021240967	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.8899605294185507	salvianolic acid b	chembl:CHEMBL541265	SALVIANOLIC ACID B	FALSE	FALSE	FALSE
PSMB1	hgnc:9537	PSMB1	ChEMBL	33	inhibitor	0.3571950424196904	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.305277158	LEVAMLODIPINE MALEATE	rxcui:2377031	LEVAMLODIPINE MALEATE	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.4145342465975881	Margetuximab	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
UNIPROT:Q9UPY5	hgnc:11059	SLC7A11	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	RILUZOLE	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.072725306	IUPHAR.LIGAND:2398	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:10365	iuphar.ligand:10365	COMPOUND 2Q [PMID: 30986068]	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005867434	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	4-FORMYL-BENZOIC ACID	chembl:CHEMBL113897	CHEMBL:CHEMBL113897	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.030176823	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
PERP	hgnc:17637	PERP	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	(-)-U-50488	chembl:CHEMBL58033	(-)-U-50488	FALSE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	PharmGKB	4/5/24	NULL	0.2401265452851883	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	THIOPERAMIDE	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-8	hgnc:7175	MMP8	TTD	2020.06.01	NULL	7.501095891	CIPEMASTAT	ncit:C96297	CIPEMASTAT	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.056826484	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.5147810905460244	SJ000047240	chembl:CHEMBL590706	CHEMBL:CHEMBL590706	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE	chembl:CHEMBL1599728	2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	BENZIODARONE	ncit:C74127	BENZIODARONE	TRUE	FALSE	FALSE
UNIPROT:O60391	hgnc:16768	GRIN3B	TdgClinicalTrial	Jan-14	NULL	0.577007376	AZD-6765	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	1.166837138570989	ALVERINE CITRATE	rxcui:71767	ALVERINE CITRATE	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	2.218633995874415	Asimadoline	ncit:C72137	ASIMADOLINE	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:8214	iuphar.ligand:8214	COMPOUND 14K [PMID: 21982499]	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.053145416	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:4082	iuphar.ligand:4082	[3H]CPP	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.022789788	AZD5438	iuphar.ligand:8473	AZD5438	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	ACETOSIDE	chembl:CHEMBL444478	ACETOSIDE	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5976	drugbank:DB08454	N-(5-METHYL-1H-PYRAZOL-3-YL)-2-PHENYLQUINAZOLIN-4-AMINE	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1415301111474245	GNF-PF-2298	chembl:CHEMBL578905	CHEMBL:CHEMBL578905	FALSE	FALSE	FALSE
SERINC5	hgnc:18825	SERINC5	PharmGKB	4/5/24	NULL	10.50153425	meperidine	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	N,N-HEXAMETHYLENEAMILORIDE	iuphar.ligand:1192	5-(N,N-HEXAMETHYLENE)-AMILORIDE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW852849X	chembl:CHEMBL514162	GW852849X	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002186317	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
BCL2L1	hgnc:992	BCL2L1	DTC	9/2/20	NULL	2.812910959055062	ABT-737	drugbank:DB17023	ABT-737	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	CIViC	10-Apr-24	NULL	0.035622572	COPANLISIB	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.1111273465305703	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
CHRM2	hgnc:1951	CHRM2	DTC	9/2/20	NULL	0.3684748858645228	ENDO-ATROPINE	chembl:CHEMBL2449003	ENDO-ATROPINE	FALSE	FALSE	FALSE
SIGLEC10	hgnc:15620	SIGLEC10	ChEMBL	33	modulator	8.751278539282415	CD24FC	chembl:CHEMBL4297717	CD24FC	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	NSC-47924	chembl:CHEMBL1269845	CHEMBL:CHEMBL1269845	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	0.5608295993131588	ROGARATINIB	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenome	20-Jun-17	inhibitor	0.073922431	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.8899605294185507	MOEXIPRIL HYDROCHLORIDE	rxcui:236066	MOEXIPRIL HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	DTC	9/2/20	NULL	0.1130007271930297	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.2586584789935689	IUPHAR.LIGAND:10357	iuphar.ligand:10357	CDK INHIBITOR 4.35	FALSE	FALSE	FALSE
UNIPROT:Q9BPV8	hgnc:4537	P2RY13	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.088770366	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.096758608	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	DNDI1417719	chembl:CHEMBL1420370	CHEMBL:CHEMBL1420370	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.6241137025199848	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	DTC	9/2/20	NULL	1.029562181092048	6-DECYLSALICYLIC ACID	chembl:CHEMBL416038	CHEMBL:CHEMBL416038	FALSE	FALSE	FALSE
PSMB1	hgnc:9537	PSMB1	ChEMBL	33	inhibitor	0.5233322714521046	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9415	iuphar.ligand:9415	COMPOUND 11 [PMID: 15261275]	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	inverse agonist	0.025439763	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
RPS14	hgnc:10387	RPS14	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.008118069	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
FNTA	hgnc:3782	FNTA	ChEMBL	33	inhibitor	0.9723642821424908	LONAFARNIB	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
TENT4A	hgnc:16705	TENT4A	PharmGKB	4/5/24	NULL	1.129197231	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005867434	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
NDUFAF3	hgnc:29918	NDUFAF3	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.1458546423213736	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
PAGA	hgnc:9352	PRDX1	ChEMBL	33	binder	8.751278539282415	RAXIBACUMAB	rxcui:1366567	RAXIBACUMAB	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.1628144844517658	PHENTOLAMINE	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.089756703	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P51170	hgnc:10602	SCNN1G	TdgClinicalTrial	Jan-14	NULL	1.620607136904151	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.2885036881082115	IUPHAR.LIGAND:7010	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1560	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:11538	iuphar.ligand:11538	OPIORPHIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	SULFANITRAN	ncit:C76978	SULFANITRAN	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.025256215	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.007378818	Paliperidone	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	1.500219178	MK-4618	rxcui:2472254	VIBEGRON	TRUE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.1530835896084387	IUPHAR.LIGAND:1431	iuphar.ligand:1431	SIB-1757	FALSE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 1 ALPHA	hgnc:4910	HIF1A	TTD	2020.06.01	NULL	0.7242437411819931	ENMD-1198	drugbank:DB05959	ENMD-1198	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.300043836	CCT018159	chembl:CHEMBL399530	CHEMBL:CHEMBL399530	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.071780822	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
CBL	hgnc:1541	CBL	NCI	14-Sep-17	NULL	0.1591141552596803	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	modulator	0.2812910959055062	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:7504	iuphar.ligand:7504	NEXTURASTAT A	FALSE	FALSE	FALSE
NCBIGENE:2046	hgnc:3391	EPHA8	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:10428	iuphar.ligand:10428	COMPOUND 25 [PMID: 31260299]	FALSE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TEND	1-Aug-11	NULL	0.1470803115845784	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:7656	iuphar.ligand:7656	ICA-105574	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1493	iuphar.ligand:1493	[125I]TYR10NPS (HUMAN)	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	BENZO[B]FLUORANTHENE	chembl:CHEMBL1337502	BENZO[B]FLUORANTHENE	FALSE	FALSE	FALSE
IDO1	hgnc:6059	IDO1	DTC	9/2/20	NULL	7.501095891	4-PHENYLIMIDAZOLE	chembl:CHEMBL14145	CHEMBL:CHEMBL14145	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:10257	iuphar.ligand:10257	GR-389988	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1966579447029756	IUPHAR.LIGAND:10142	iuphar.ligand:10142	PQR620	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.108711535	DELUCEMINE	ncit:C76776	DELUCEMINE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:1220	iuphar.ligand:1220	[3H]PYRILAMINE	FALSE	FALSE	FALSE
PSMA3	hgnc:9532	PSMA3	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:8075	iuphar.ligand:8075	LY2109761	FALSE	FALSE	FALSE
MELANOCORTIN RECEPTOR 1	hgnc:6929	MC1R	TTD	2020.06.01	NULL	4.500657534488099	afamelanotide	rxcui:2262250	AFAMELANOTIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.003429856	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.081830137	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1215455352678113	BAY-1082439	chembl:CHEMBL3545245	BAY-1082439	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.108040476	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
CD33	hgnc:1659	CD33	ChEMBL	33	other/unknown	4.039051633514961	M195	chembl:CHEMBL2109267	M195	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.8078103267029922	EB-101	ncit:C175196	PRADEMAGENE ZAMIKERACEL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002421494	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005563432	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	PROPANTHELINE	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	PharmGKB	4/5/24	NULL	0.008334551	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	PharmGKB	4/5/24	NULL	2.151953739167807	olaratumab	rxcui:1855735	OLARATUMAB	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.024932417	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	NCI	14-Sep-17	NULL	0.1077080435603989	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
NERVE GROWTH FACTOR	hgnc:7808	NGF	TTD	2020.06.01	NULL	15.00219178	Fasinumab	ncit:C166446	FASINUMAB	FALSE	FALSE	FALSE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	1.019566431761058	Axitirome	ncit:C75992	AXITIROME	FALSE	FALSE	FALSE
CAMK1	hgnc:1459	CAMK1	DTC	9/2/20	NULL	0.2187819634820604	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:1913	iuphar.ligand:1913	MB-28767	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	(+/-)-OCTOCLOTHEPIN MALEATE	chembl:CHEMBL1256660	CHEMBL:CHEMBL1256660	FALSE	FALSE	FALSE
RPS6KB2	hgnc:10437	RPS6KB2	ChEMBL	33	inhibitor	1.312691780892362	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
IL13	hgnc:5973	IL13	ChEMBL	33	inhibitor	4.375639269641208	CENDAKIMAB	ncit:C174792	CENDAKIMAB	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.1228249619548409	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.1154014752432846	Oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	NCI	14-Sep-17	NULL	0.4546118721705151	BSO	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.5834185692854944	MISONIDAZOLE	ncit:C657	MISONIDAZOLE	FALSE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.2302968036653267	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.014354202	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	TALC	12-May-16	vaccine	0.028977744	EP-2101	ncit:C26645	MULTI-NEO-EPITOPE VACCINE OSE 2101	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	RS-17053	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.8751278539282417	Eluxadoline	rxcui:1653781	ELUXADOLINE	TRUE	FALSE	FALSE
TBXA2R	hgnc:11608	TBXA2R	ChEMBL	33	inhibitor	1.875273972703375	SERATRODAST	ncit:C90671	SERATRODAST	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	GNF-PF-4046	chembl:CHEMBL600090	CHEMBL:CHEMBL600090	FALSE	FALSE	FALSE
TLR2	hgnc:11848	TLR2	ChEMBL	33	inhibitor	7.501095891	TOMARALIMAB	ncit:C120554	TOMARALIMAB	FALSE	FALSE	FALSE
S100A12	hgnc:10489	S100A12	NCI	14-Sep-17	NULL	0.1875273972703374	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NCBIGENE:1924	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:12383	iuphar.ligand:12383	RISVODETINIB	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1600843635234588	IUPHAR.LIGAND:73	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:544	iuphar.ligand:544	LK 204-545	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:1022	iuphar.ligand:1022	FMET-LEU-PHE	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:746	ncit:C184881	ONTERNABEZ	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:9175	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:322	iuphar.ligand:322	HEXAHYDRODIFENIDOL	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:10312	iuphar.ligand:10312	CYM-50358	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	1.678633990910949	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	4-PHENOXYPHENOL	chembl:CHEMBL224318	CHEMBL:CHEMBL224318	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	MR1-1	ncit:C88307	ANTI-EGFRVIII IMMUNOTOXIN MR1-1	FALSE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TEND	1-Aug-11	NULL	5.000730593875666	STREPTOKINASE	rxcui:10106	STREPTOKINASE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.013199515	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006265084	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.05853698	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.041021618	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
POLO-LIKE KINASE 2	hgnc:19699	PLK2	TTD	2020.06.01	NULL	3.750547945406749	BI2536	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.1093909817410302	PHA-665752	iuphar.ligand:5700	PHA-665752	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	PharmGKB	4/5/24	NULL	0.2273059360852575	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.2778183663264259	AMIVANTAMAB	rxcui:2549198	AMIVANTAMAB-VMJW	TRUE	FALSE	TRUE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.1041818873724097	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.075496292	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
RAMP1	hgnc:9843	RAMP1	ChEMBL	33	inhibitor	6.563458904461812	ZAVEGEPANT	rxcui:2637955	ZAVEGEPANT	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.071341945	IZENCITINIB	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.051545489	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1458546423213736	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	0.099446347	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.02091106	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
INSULIN-DEGRADING ENZYME	hgnc:5381	IDE	TTD	2020.06.01	NULL	3.500511415712966	Bacitracin	rxcui:1291	BACITRACIN	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.4861821410712453	AZM-475271	chembl:CHEMBL3545150	AZM-475271	FALSE	FALSE	FALSE
CASR	hgnc:1514	CASR	ChEMBL	33	inhibitor	6.563458904461812	RONACALERET	ncit:C81351	RONACALERET	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6563458904461813	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	inhibitor	0.7292732116068681	IUPHAR.LIGAND:1765	rxcui:1116632	TICAGRELOR	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.458240639	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
TERT	hgnc:11730	TERT	CIViC	10-Apr-24	NULL	1.500219178	IODINE I-131	rxcui:1546394	IODINE I-131	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.1293292394967845	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:10453	iuphar.ligand:10453	CR4056	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	1.381780822	Drospirenone	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	CARBARIL	ncit:C76389	CARBARIL	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.037721028	IDARUBICIN HYDROCHLORIDE	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.092443083	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.094608417	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
ATM SERINE/THREONINE KINASE	hgnc:795	ATM	TTD	2020.06.01	NULL	0.2397610558707511	VE-822	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.4861821410712454	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.032173818	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.2375912725597036	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.1422972120208523	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:10063	iuphar.ligand:10063	CDK12 INHIBITOR 2	FALSE	FALSE	FALSE
SOCS1	hgnc:19383	SOCS1	NCI	14-Sep-17	NULL	0.9907107780319716	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	agonist	0.037398626	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.073954467	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1565	iuphar.ligand:1565	L-152,804	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.038131933	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	METHYL YELLOW	chembl:CHEMBL1090440	METHYL YELLOW	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	1.591141552596803	TDR77403	chembl:CHEMBL1534035	CHEMBL:CHEMBL1534035	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	CAULIBUGULONE D	chembl:CHEMBL447876	CAULIBUGULONE D	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.062139256	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	0.6429510763554428	EDOXABAN TOSYLATE	rxcui:1599538	EDOXABAN	TRUE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.295540363	CRA-024781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
NDUFS5	hgnc:7712	NDUFS5	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.088248187	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.1320947704042629	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.4261986301598579	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.1520492410300034	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.9211872146613069	IUPHAR.LIGAND:8433	iuphar.ligand:8433	AS-19	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.004660306	Clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.090843722	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:8137	iuphar.ligand:8137	COMPOUND 8E [PMID: 24432909]	FALSE	FALSE	FALSE
GASTRIN	hgnc:4164	GAST	TTD	2020.06.01	NULL	35.00511415712966	G17DT	ncit:C1692	GASTRIN IMMUNOTOXIN	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	CancerCommons	25-Jul-13	inhibitor	0.4861821410712454	AV951	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
GALNT2	hgnc:4124	GALNT2	PharmGKB	4/5/24	NULL	0.9723642821424908	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	CancerCommons	25-Jul-13	inhibitor	0.1136529680426287	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.038382801	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	CGI	2/1/22	NULL	0.044198376	Letrozole	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.026572708	Tamoxifen	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.1630673019742065	PLX3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
NF2	hgnc:7773	NF2	CGI	2/1/22	NULL	0.2430910705356227	Octreotide	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CGI	2/1/22	NULL	1.090323227845022	Crenolanib	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
CYP11A1	hgnc:2590	CYP11A1	ChEMBL	33	inhibitor	3.500511415712967	LEVOKETOCONAZOLE	rxcui:2588846	LEVOKETOCONAZOLE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	CLEMASTINE FUMARATE	rxcui:142430	CLEMASTINE FUMARATE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.8468979231563628	DEXCHLORPHENIRAMINE MALEATE	rxcui:54828	DEXCHLORPHENIRAMINE MALEATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	modulator	0.2075402025126264	BENZQUINAMIDE HYDROCHLORIDE	rxcui:91272	BENZQUINAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.2734774543525755	PHENYLPROPANOLAMINE HYDROCHLORIDE	rxcui:3266	PHENYLPROPANOLAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.038966732	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.5585922471882393	DIPHEMANIL METHYLSULFATE	rxcui:23364	DIPHEMANIL METHYLSULFATE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	1.166837138570988	GRANISETRON HYDROCHLORIDE	rxcui:142149	GRANISETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1B	hgnc:5287	HTR1B	ChEMBL	33	agonist	0.5147810905460244	ALMOTRIPTAN MALATE	rxcui:283792	ALMOTRIPTAN MALATE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.9944634703730019	FENOFIBRIC ACID	rxcui:24852	FENOFIBRIC ACID	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.2237542808339254	RANOLAZINE	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
KLKB1	hgnc:6371	KLKB1	ChEMBL	33	inhibitor	1.875273972703375	APROTININ	rxcui:1056	APROTININ	TRUE	FALSE	FALSE
PTGIR	hgnc:9602	PTGIR	ChEMBL	33	agonist	0.9376369863516875	ILOPROST	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.3241214273808302	ARMODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.010434752	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.048172175	FENTANYL CITRATE	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.048172175	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.801643836	BETAMETHASONE BENZOATE	rxcui:1517	BETAMETHASONE BENZOATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.03262504	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.6081969641200136	RASAGILINE MESYLATE	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	inhibitor	0.057260274	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1591141552596802	ZALCITABINE	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	inhibitor	0.091159151	METHYLERGONOVINE MALEATE	rxcui:84158	METHYLERGONOVINE MALEATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.035358701	ZIDOVUDINE	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.067839369	TCMDC-124544	chembl:CHEMBL531322	CHEMBL:CHEMBL531322	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	HYDROCODONE POLISTIREX	rxcui:221107	HYDROCODONE POLISTIREX	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	HYDROCODONE BITARTRATE	rxcui:142439	HYDROCODONE BITARTRATE	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1205533268166455	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	negative modulator	0.3195192975802911	KETAMINE HYDROCHLORIDE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.02926849	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.048958202	IBUPROFEN SODIUM	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.003365876	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.157680694	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.076098074	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	AMLODIPINE MALEATE	ncit:C65230	AMLODIPINE MALEATE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.07182992	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.003650422	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.082559232	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.1356787370431382	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	ChEMBL	33	inhibitor	2.187819634820604	PENTOLINIUM TARTRATE	ncit:C66345	PENTOLINIUM TARTRATE	TRUE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TEND	1-Aug-11	NULL	0.9376369863516875	ILOPROST	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
CHRNA3	hgnc:1957	CHRNA3	ChEMBL	33	inhibitor	0.7955707762984014	PENTOLINIUM TARTRATE	ncit:C66345	PENTOLINIUM TARTRATE	TRUE	FALSE	FALSE
CD52	hgnc:1804	CD52	ChEMBL	33	inhibitor	70.01022831425932	ALEMTUZUMAB	rxcui:117055	ALEMTUZUMAB	TRUE	TRUE	TRUE
GC	hgnc:4187	GC	ChEMBL	33	inhibitor	0.546954909	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
FANCC	hgnc:3584	FANCC	CIViC	10-Apr-24	NULL	0.4375639269641208	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
GM	hgnc:9291	PPP1R3A	ChEMBL	33	inhibitor	6.563458904461812	DOCOSANOL	rxcui:594680	DOCOSANOL	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.1415301111474245	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
COL6A3	hgnc:2213	COL6A3	ChEMBL	33	cleavage	0.4688184931758437	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
COL4A5	hgnc:2207	COL4A5	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
ADRM1	hgnc:15759	ADRM1	ChEMBL	33	inhibitor	0.3663325900164732	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB8	hgnc:9545	PSMB8	ChEMBL	33	inhibitor	0.2220197515251353	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMC1	hgnc:9547	PSMC1	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:P08235	hgnc:7979	NR3C2	TdgClinicalTrial	Jan-14	NULL	1.381780822	DROSPIRENONE	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	ChEMBL	33	inhibitor	0.3488881809680698	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD12	hgnc:9557	PSMD12	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD6	hgnc:9564	PSMD6	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	2.100306849	TETRABENAZINE	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.2763561643983921	DEXTROAMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.5250767123569451	MIVACURIUM CHLORIDE	rxcui:52796	MIVACURIUM CHLORIDE	TRUE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.2419708351875322	TOFACITINIB CITRATE	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	1.467605717767858	TOFACITINIB CITRATE	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
MT-ND1	hgnc:7455	MT-ND1	ChEMBL	33	inhibitor	0.093763699	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GLRA1	hgnc:4326	GLRA1	ChEMBL	33	positive modulator	0.1539814405738841	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.2038341274677581	TOFACITINIB CITRATE	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	0.1357664414626878	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
RARG	hgnc:9866	RARG	ChEMBL	33	agonist	0.1930429089547591	ACITRETIN	rxcui:16818	ACITRETIN	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.061197752	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.060423097	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.053038052	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.080781033	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.085147575	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.070010228	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
EED	hgnc:3188	EED	DTC	9/2/20	NULL	3.281729452230906	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.050007306	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.08780547	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.077827576	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.020164236	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.02091106	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.033232703	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.4526523382387456	MOXIFLOXACIN HYDROCHLORIDE	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
FGR	hgnc:3697	FGR	ChEMBL	33	inhibitor	0.032472277	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
FRK	hgnc:3955	FRK	ChEMBL	33	inhibitor	0.024354207	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
SRMS	hgnc:11298	SRMS	ChEMBL	33	inhibitor	0.1704794520639432	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	1.544343271638073	Diethylcarbamazine	rxcui:3384	DIETHYLCARBAMAZINE	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.055155117	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.1389091831632129	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.063110182	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.045898314	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	1.712206670729168	MACITENTAN	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.1091635576625665	VORTIOXETINE HYDROBROMIDE	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.059667808	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.093763699	DROXIDOPA	rxcui:1489913	DROXIDOPA	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	ChEMBL	33	inhibitor	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.07939668	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	0.1521961485092594	ALECTINIB HYDROCHLORIDE	rxcui:1727454	ALECTINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	1.184383561707394	KD3010	drugbank:DB05188	KD3010	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.210030685	DB959	chembl:CHEMBL3545176	DB959	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.3431873936973496	AG-24322	drugbank:DB13035	AG-24322	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.172722603	ALLITINIB	ncit:C179280	ALLITINIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	0.4565884455277782	ASP-3026	drugbank:DB12729	ASP-3026	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.596678082	AS-703988	chembl:CHEMBL3545243	AS-703988	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.201952582	CAL-263	chembl:CHEMBL3545247	CAL-263	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.029766254	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.729273212	BENZENETHIOL	chembl:CHEMBL119405	BENZENETHIOL	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1111273465305703	FALNIDAMOL	ncit:C80868	FALNIDAMOL	FALSE	FALSE	FALSE
NDUFA11	hgnc:20371	NDUFA11	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA10	hgnc:7684	NDUFA10	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFB5	hgnc:7700	NDUFB5	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.027010119	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.2734774543525755	PLX-7486	chembl:CHEMBL3545381	PLX-7486	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.046303061	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.041085815	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.2386712328895204	PLX-7486	chembl:CHEMBL3545381	PLX-7486	FALSE	FALSE	FALSE
PIM2	hgnc:8987	PIM2	ChEMBL	33	inhibitor	2.187819634820604	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	TAK-285	chembl:CHEMBL1614725	TAK-285	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.1241316104862754	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.2885036881082115	DELUCEMINE	ncit:C76776	DELUCEMINE	FALSE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1100789753368857	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	blocker	0.3889457128569963	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.2651902587661338	SODELGLITAZAR	ncit:C75193	SODELGLITAZAR	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	ChEMBL	33	agonist	0.2333674277141977	IRX-4204	chembl:CHEMBL75133	IRX-4204	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	modulator	0.42006137	MK-0533	drugbank:DB15242	MK-0533	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	2.407466349146467	BRIGATINIB	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.5181678082469852	VARLITINIB	ncit:C62530	VARLITINIB	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.047561296	AT-9283	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.095122593	AT-9283	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	ChEMBL	33	inhibitor	0.7212592202705288	ADAVOSERTIB	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1888765152363111	AZM-475271	chembl:CHEMBL3545150	AZM-475271	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.065308049	AT-9283	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.1480479452134243	SAPITINIB	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.4118248724368196	RIVICICLIB	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.079236928	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.5707355569097228	NS-018	chembl:CHEMBL3545217	NS-018	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.1666910197958555	VORUCICLIB	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.049026771	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.079197091	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.088248187	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.029918901	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.6482428547616604	IPATASERTIB	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1056492378987816	FAMITINIB	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.3443125982668492	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1682938180631233	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.2218633995874415	X-82	chembl:CHEMBL3545401	X-82	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.052090944	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1682938180631233	ZSTK-474	drugbank:DB12904	ZSTK-474	FALSE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	1.500219178	VIBEGRON	rxcui:2472254	VIBEGRON	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.4817217544559128	AXELOPRAN	ncit:C171856	AXELOPRAN	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	ChEMBL	33	inhibitor	3.424413341458336	ILACIRNON	ncit:C175798	ILACIRNON	FALSE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	4.145342465975881	OC000459	iuphar.ligand:9277	TIMAPIPRANT	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	AZD3199	chembl:CHEMBL3545103	AZD3199	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	0.729273212	AMP579	chembl:CHEMBL3545163	AMP579	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	agonist	0.040021091	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.458546423213736	ALTINICLINE	ncit:C77841	ALTINICLINE	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	inverse agonist	0.038159645	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.6482428547616604	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.042174836	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
ERAP1	hgnc:18173	ERAP1	ChEMBL	33	inhibitor	0.4375639269641209	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.1428780169678761	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
ERAP2	hgnc:29499	ERAP2	ChEMBL	33	inhibitor	0.4375639269641209	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ChEMBL	33	inhibitor	0.7395446652914718	RIDAFOROLIMUS	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
ENPEP	hgnc:3355	ENPEP	ChEMBL	33	inhibitor	0.6563458904461813	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
LVRN	hgnc:26904	LVRN	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PSMD8	hgnc:9566	PSMD8	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB1	hgnc:9537	PSMB1	ChEMBL	33	inhibitor	0.384671584	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMA7	hgnc:9536	PSMA7	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMB6	hgnc:9543	PSMB6	ChEMBL	33	inhibitor	0.2243917574174978	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMD1	hgnc:9554	PSMD1	ChEMBL	33	inhibitor	0.5385402178019948	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
PSMC4	hgnc:9551	PSMC4	ChEMBL	33	inhibitor	0.2692701089009974	OPROZOMIB	ncit:C91388	OPROZOMIB	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.2616661357260523	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.2678962818147679	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.042174836	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
CHRNA10	hgnc:13800	CHRNA10	ChEMBL	33	inhibitor	1.166837138570989	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	ChEMBL	33	inhibitor	0.2001054544043235	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.7395446652914718	NALFURAFINE HYDROCHLORIDE	ncit:C80586	NALFURAFINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	ChEMBL	33	inhibitor	0.596678082	BEGACESTAT	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	negative modulator	0.096167896	ESKETAMINE HYDROCHLORIDE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	0.3000438356325399	VILDAGLIPTIN	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	ChEMBL	33	inhibitor	0.4688184931758437	BEGACESTAT	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	ChEMBL	33	inhibitor	0.546954909	BEGACESTAT	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
PLA2G7	hgnc:9040	PLA2G7	ChEMBL	33	inhibitor	13.12691780892362	DARAPLADIB	ncit:C72985	DARAPLADIB	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	negative modulator	0.2586584789935689	ESKETAMINE HYDROCHLORIDE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
SLC9A3	hgnc:11073	SLC9A3	ChEMBL	33	inhibitor	13.12691780892362	SQUALAMINE LACTATE	ncit:C1482	SQUALAMINE LACTATE	FALSE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.182318303	FALDAPREVIR	ncit:C171746	FALDAPREVIR	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.084553416	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.074797252	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
MGAM	hgnc:7043	MGAM	ChEMBL	33	inhibitor	4.773424657790408	VOGLIBOSE	ncit:C95221	VOGLIBOSE	TRUE	FALSE	FALSE
FGF1	hgnc:3665	FGF1	ChEMBL	33	inhibitor	0.4861821410712453	SURAMIN HEXASODIUM	chembl:CHEMBL413376	SURAMIN HEXASODIUM	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.4145342465975881	MARGETUXIMAB	rxcui:2473850	MARGETUXIMAB-CMKB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	0.561579372	DURVALUMAB	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	inhibitor	1.009762908	ETARACIZUMAB	ncit:C1800	ETARACIZUMAB	FALSE	FALSE	TRUE
CD4	hgnc:1678	CD4	ChEMBL	33	inhibitor	3.281729452230906	CEDELIZUMAB	chembl:CHEMBL2108266	CEDELIZUMAB	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	ChEMBL	33	other/unknown	0.6908904109959803	EMICIZUMAB	rxcui:1989794	EMICIZUMAB	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	2.151953739167807	OLARATUMAB	rxcui:1855735	OLARATUMAB	TRUE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	other/unknown	6.300920548	ING-1	drugbank:DB05831	ING-1	FALSE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	ChEMBL	33	inhibitor	1.458546423213736	ROVELIZUMAB	ncit:C152264	ROVELIZUMAB	FALSE	FALSE	FALSE
KIR2DL1	hgnc:6329	KIR2DL1	ChEMBL	33	inhibitor	10.50153424713889	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	1.458546423213736	RUCAPARIB CAMSYLATE	rxcui:1862578	RUCAPARIB CAMSYLATE	TRUE	FALSE	FALSE
TNFRSF9	hgnc:11924	TNFRSF9	ChEMBL	33	agonist	52.50767123569449	UTOMILUMAB	ncit:C116619	UTOMILUMAB	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.6226206075378794	BROMPERIDOL	rxcui:19777	BROMPERIDOL	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	agonist	0.7955707762984013	ARGIPRESSIN TANNATE	ncit:C166779	ARGIPRESSIN TANNATE	TRUE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	ChEMBL	33	inhibitor	3.125456621172291	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.093763699	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.097236428	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.031254566	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	blocker	0.1209854175937661	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA2D1	hgnc:1399	CACNA2D1	ChEMBL	33	blocker	0.080656945	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	inhibitor	0.1145205479513511	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.1539814405738841	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
SRD5A1	hgnc:11284	SRD5A1	ChEMBL	33	inhibitor	0.729273212	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	binder	0.2344092465879218	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TRAC	hgnc:12029	TRAC	ChEMBL	33	inhibitor	3.281729452230906	MASLIMOMAB	ncit:C188519	MASLIMOMAB	FALSE	FALSE	FALSE
HBEGF	hgnc:3059	HBEGF	ChEMBL	33	inhibitor	3.387591692625451	KHK-2866	chembl:CHEMBL2109437	KHK-2866	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	modulator	0.364636606	IMC-GP100	chembl:CHEMBL2109434	IMC-GP100	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	3.500511415712966	MEDI-3617	chembl:CHEMBL2109298	MEDI-3617	FALSE	FALSE	FALSE
KCNQ5	hgnc:6299	KCNQ5	ChEMBL	33	blocker	0.071148606	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNG3	hgnc:18306	KCNG3	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNG4	hgnc:19697	KCNG4	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNG1	hgnc:6248	KCNG1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1182605208011137	REVEFENACIN	rxcui:2102775	REVEFENACIN	TRUE	FALSE	FALSE
KCNG2	hgnc:6249	KCNG2	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	ChEMBL	33	inhibitor	0.3977853881492006	BMS-986158	drugbank:DB15435	BMS-986158	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	ChEMBL	33	inhibitor	0.4605936073306534	BMS-986158	drugbank:DB15435	BMS-986158	FALSE	FALSE	FALSE
BRDT	hgnc:1105	BRDT	ChEMBL	33	inhibitor	0.6250913242344582	BMS-986158	drugbank:DB15435	BMS-986158	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.060353645	CD24FC	chembl:CHEMBL4297717	CD24FC	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	ChEMBL	33	positive modulator	0.1988926940746003	ONASEMNOGENE ABEPARVOVEC	rxcui:2170225	ONASEMNOGENE ABEPARVOVEC-XIOI	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.1666910197958555	ADOPRAZINE	ncit:C81482	ADOPRAZINE	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	1.628144844517658	PEMIGATINIB	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	ChEMBL	33	agonist	1.000146118775133	BEPERMINOGENE PERPLASMID	chembl:CHEMBL2108332	BEPERMINOGENE PERPLASMID	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	BENZHYDROCODONE HYDROCHLORIDE	rxcui:2122776	BENZHYDROCODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	LEVAMLODIPINE MALEATE	rxcui:2377031	LEVAMLODIPINE MALEATE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.2476776945079929	LEVAMLODIPINE MALEATE	rxcui:2377031	LEVAMLODIPINE MALEATE	TRUE	FALSE	FALSE
CCDC6	hgnc:18782	CCDC6	ChEMBL	33	inhibitor	6.563458904461812	SELPERCATINIB	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.093098708	SOFPIRONIUM BROMIDE	ncit:C152384	SOFPIRONIUM BROMIDE	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.305277158	BARNIDIPINE	rxcui:39879	MEPIRODIPINE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	2.917092846427472	MAGNESIUM OXYBATE	rxcui:2387308	MAGNESIUM OXYBATE	TRUE	FALSE	FALSE
AXL	hgnc:905	AXL	ChEMBL	33	binder	0.068369364	ENAPOTAMAB VEDOTIN	ncit:C132017	ENAPOTAMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.8537832721251137	SPARTALIZUMAB	ncit:C121625	SPARTALIZUMAB	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	2.625383561784724	BMS-813160	drugbank:DB16240	BMS-813160	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	CABOTEGRAVIR	rxcui:2475077	CABOTEGRAVIR	TRUE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.3201687270469177	CAMRELIZUMAB	ncit:C123816	CAMRELIZUMAB	FALSE	FALSE	FALSE
CD47	hgnc:1682	CD47	ChEMBL	33	inhibitor	4.375639269641208	MAGROLIMAB	ncit:C117730	MAGROLIMAB	FALSE	FALSE	FALSE
IL31RA	hgnc:18969	IL31RA	ChEMBL	33	inhibitor	26.25383561784724	NEMOLIZUMAB	ncit:C170211	NEMOLIZUMAB	FALSE	FALSE	FALSE
LAG3	hgnc:6476	LAG3	ChEMBL	33	inhibitor	13.12691780892362	IERAMILIMAB	ncit:C122683	IERAMILIMAB	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	agonist	0.041540879	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	agonist	0.025439763	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	agonist	0.039068208	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	agonist	0.042073455	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	negative modulator	0.3281729452230906	TAS-117	drugbank:DB15054	TAS-117	FALSE	FALSE	FALSE
PCSK9	hgnc:20001	PCSK9	ChEMBL	33	inhibitor	4.039051633514961	FROVOCIMAB	ncit:C175068	FROVOCIMAB	FALSE	FALSE	FALSE
RPS10	hgnc:10383	RPS10	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS3	hgnc:10420	RPS3	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS17	hgnc:10397	RPS17	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS16	hgnc:10396	RPS16	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS4Y1	hgnc:10425	RPS4Y1	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL7	hgnc:10363	RPL7	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL27	hgnc:10328	RPL27	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL22	hgnc:10315	RPL22	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL10A	hgnc:10299	RPL10A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL28	hgnc:10330	RPL28	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
PPP2CB	hgnc:9300	PPP2CB	ChEMBL	33	inhibitor	10.50153425	LB-100	drugbank:DB15412	LB-100	FALSE	FALSE	FALSE
TIGIT	hgnc:26838	TIGIT	ChEMBL	33	inhibitor	3.281729452230906	TIRAGOLUMAB	ncit:C131291	TIRAGOLUMAB	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.065799087	LANIFIBRANOR	ncit:C166556	LANIFIBRANOR	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	CONTEZOLID	ncit:C171693	CONTEZOLID	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.041672755	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.6403374540938354	CETRELIMAB	ncit:C129448	CETRELIMAB	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	ChEMBL	33	agonist	3.088686543276147	TILSOTOLIMOD SODIUM	ncit:C125080	TILSOTOLIMOD SODIUM	FALSE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	inhibitor	2.917092846427472	SGS-742	drugbank:DB05010	SGS-742	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.6977763619361395	RICOLINOSTAT	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
MME	hgnc:7154	MME	ChEMBL	33	inhibitor	4.773424657790408	ILEPATRIL	ncit:C87731	ILEPATRIL	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	0.4565884455277782	CONTELTINIB	ncit:C169863	CONTELTINIB	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.2275522047050683	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	ChEMBL	33	inhibitor	0.3804903712731485	ALECTINIB HYDROCHLORIDE	rxcui:1727454	ALECTINIB HYDROCHLORIDE	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	ChEMBL	33	inhibitor	0.1767935058440892	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	TECLISTAMAB	rxcui:2619425	TECLISTAMAB-CQYV	TRUE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	TECLISTAMAB	rxcui:2619425	TECLISTAMAB-CQYV	TRUE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	vaccine	0.8078103267029922	VANUTIDE CRIDIFICAR	ncit:C152829	VANUTIDE CRIDIFICAR	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	1.909369863116163	AXATILIMAB	ncit:C155813	AXATILIMAB	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	3.500511415712966	CROVALIMAB	ncit:C169867	CROVALIMAB	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	positive modulator	1.193356164447602	OLACAFTOR	ncit:C170243	OLACAFTOR	FALSE	FALSE	FALSE
EEF1A2	hgnc:3192	EEF1A2	ChEMBL	33	inhibitor	26.25383561784724	PLITIDEPSIN	ncit:C1689	PLITIDEPSIN	FALSE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	ChEMBL	33	potentiator	0.6819178082557726	EZOGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	agonist	2.019525817	PEGENZILEUKIN	drugbank:DB17495	PEGENZILEUKIN	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
PTH1R	hgnc:9608	PTH1R	ChEMBL	33	agonist	2.500365296937833	OSTABOLIN-C	chembl:CHEMBL4802222	OSTABOLIN-C	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	VILANTEROL .ALPHA.-PHENYL CINNAMATE	chembl:CHEMBL1084173	VILANTEROL .ALPHA.-PHENYL CINNAMATE	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.081407242	IUPHAR.LIGAND:4156	iuphar.ligand:4156	CGS8216	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	ChEMBL	33	vaccine	0.596678082	SVN53-67/M57-KLH PEPTIDE VACCINE	ncit:C95705	SVN53-67/M57-KLH PEPTIDE VACCINE	FALSE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.305277158	LACIDIPINE	rxcui:28382	LACIDIPINE	TRUE	FALSE	FALSE
PKLR	hgnc:9020	PKLR	ChEMBL	33	activator	11.66837138570988	MITAPIVAT	rxcui:2594468	MITAPIVAT	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.034318739	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
PKLR	hgnc:9020	PKLR	ChEMBL	33	activator	8.751278539282415	ETAVOPIVAT	ncit:C176893	ETAVOPIVAT	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.03151721	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.037666909	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:1589	iuphar.ligand:1589	(+)-5-(5-BROMOTHIOPHEN-3-YL)-5-METHYL-4-OXO-4,5-DIHYDRO-FURAN-2-CARBOXYLIC ACID	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2983390411119005	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
PARP1	hgnc:270	PARP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3818739726232327	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:4239	iuphar.ligand:4239	L689560	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1008469998124734	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:7739	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.029698909	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1750255707856483	BKM120	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2778183663264258	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.07767407	LENALIDOMIDE	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	COSMIC	4-Sep-20	NULL	2.407466349146467	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.018019105	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	LEVISOPRENALINE	ncit:C74197	LEVISOPRENALINE	FALSE	FALSE	FALSE
NCBIGENE:1722	hgnc:7217	MPL	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5063	iuphar.ligand:5063	THROMBOPOIETIN	FALSE	FALSE	FALSE
LMNA	hgnc:6636	LMNA	DTC	9/2/20	NULL	1.346350544504987	HISTAMINE	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.055563673	TDR77585	chembl:CHEMBL1333386	CHEMBL:CHEMBL1333386	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002737341	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003740928	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	CHALCONE	rxcui:2592960	CHALCONE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.007544206	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.6848826682916673	CELASTROL	iuphar.ligand:10386	CELASTROL	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1448487482363986	CELASTROL	iuphar.ligand:10386	CELASTROL	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1557	iuphar.ligand:1557	NPY-(18-36) (HUMAN, PIG)	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.01635753	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	HEMATOXYLIN	drugbank:DB16871	HEMATOXYLIN	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.025427444	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.7001022831425933	NARINGIN	rxcui:31538	NARINGIN	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	0.1154014752432846	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	DNDI1417719	chembl:CHEMBL1420370	CHEMBL:CHEMBL1420370	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.003819851	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1274458039701322	HARMALOL	chembl:CHEMBL129177	HARMALOL	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.088396753	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	AM580	iuphar.ligand:2647	RO 40-6055	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.7501095890813501	DELAVIRDINE	rxcui:83816	DELAVIRDINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	METHYLMALONIC ACID	drugbank:DB04183	METHYLMALONIC ACID	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	CIViC	10-Apr-24	NULL	0.2273059360852575	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	HARMALINE	drugbank:DB13875	HARMALINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FLUCYTOSINE	rxcui:4451	FLUCYTOSINE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	RESACTIN A	chembl:CHEMBL509617	RESACTIN A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007727398	CLADRIBINE	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.182318303	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ESTRADIOL CYPIONATE	rxcui:1000146	ESTRADIOL CYPIONATE	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.031707531	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.020446912	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	GLIOTOXIN	rxcui:1661743	GLIOTOXIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.033919684	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV007474	chembl:CHEMBL601534	CHEMBL:CHEMBL601534	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.5147810905460245	5-HYDROXYFLAVONE	chembl:CHEMBL16807	5-HYDROXYFLAVONE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1426838892274307	DICYCLOHEXYLCARBODIIMIDE	chembl:CHEMBL162598	DICYCLOHEXYLCARBODIIMIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	3-AMINOBENZAMIDE	chembl:CHEMBL81977	3-AMINOBENZAMIDE	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1744440904840348	ANTINEOPLASTIC	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.013589562	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1620607136904151	13-CIS-RETINAL	iuphar.ligand:6671	13-CIS-RETINAL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003053304	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.8751278539282416	DEXTROAMPHETAMINE ADIPATE	chembl:CHEMBL1200782	DEXTROAMPHETAMINE ADIPATE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.012230997	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.1902451856365742	ARRY-797	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.021422958	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.1400204566285186	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	SJ000071854	chembl:CHEMBL602127	CHEMBL:CHEMBL602127	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.043866058	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01256465	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.019059046	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	METHABENZTHIAZURON	chembl:CHEMBL1890813	METHABENZTHIAZURON	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.1238388472539964	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	NCI	14-Sep-17	NULL	0.2027323213733378	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.029665351	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.4526523382387456	SIMOCYCLINONE D8	chembl:CHEMBL1235969	SIMOCYCLINONE D8	FALSE	FALSE	FALSE
HTR2B	hgnc:5294	HTR2B	DTC	9/2/20	NULL	2.187819634820604	ATC-0175	iuphar.ligand:1305	ATC0175	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	(E)-2-STYRYLCHROMONE	chembl:CHEMBL388823	CHEMBL:CHEMBL388823	FALSE	FALSE	FALSE
SRMS	hgnc:11298	SRMS	DTC	9/2/20	NULL	0.1704794520639432	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.00854617	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.1842374429322614	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.008287196	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007937668	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.032412143	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000928124	IRINOTECAN HYDROCHLORIDE	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.8899605294185507	LOSARTAN	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.072324616	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.2641895408085258	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.039068208	RACEPINEPHRINE	rxcui:66887	RACEPINEPHRINE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.006730027	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	1-BENZYLMALEIMIDE	chembl:CHEMBL388979	CHEMBL:CHEMBL388979	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.079798892	PIFEXOLE	ncit:C76774	PIFEXOLE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	TCMDC-125587	chembl:CHEMBL532160	CHEMBL:CHEMBL532160	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.01214331	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CYPRODINIL	chembl:CHEMBL521027	CYPRODINIL	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.054355767	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	RS-17053	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	0.046881849	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.036770078	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.1172046232939609	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.042073455	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.049192122	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	TCMDC-125653	chembl:CHEMBL580918	CHEMBL:CHEMBL580918	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	NSC-353720	chembl:CHEMBL1408276	CHEMBL:CHEMBL1408276	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	0.1511209794852536	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.364636606	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.2381300282797936	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TEND	1-Aug-11	NULL	8.204323630577266	UDENAFIL	ncit:C74086	UDENAFIL	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.013299815	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	3.889457128569962	DIETHYL-2-UNDECYLIDENEMALONATE	chembl:CHEMBL1797707	CHEMBL:CHEMBL1797707	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	A-315456	chembl:CHEMBL362863	CHEMBL:CHEMBL362863	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.046303061	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
GPR35	hgnc:4492	GPR35	DTC	9/2/20	NULL	0.051127236	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	PRODINE HYDROCHLORIDE	chembl:CHEMBL1529817	ALPHAPRODINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
KDM1A	hgnc:29079	KDM1A	DTC	9/2/20	NULL	21.00306849427779	NAMOLINE	chembl:CHEMBL2426136	NAMOLINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	OBTUSAQUINONE	chembl:CHEMBL1333653	OBTUSAQUINONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	(+)-TETRAHYDROBERBERINE	chembl:CHEMBL476501	CHEMBL:CHEMBL476501	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	ZM-336372	iuphar.ligand:9130	ZM336372	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.095122593	METHYLTESTOSTERONE	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.037239483	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.1438566335224507	FLUNARIZINE DIHYDROCHLORIDE	chembl:CHEMBL539027	FLUNARIZINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.021370644	MAPROTILINE HYDROCHLORIDE	rxcui:203126	MAPROTILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	8-(3-BROMOPHENOXYMETHYL)CAFFEINE	chembl:CHEMBL2088301	CHEMBL:CHEMBL2088301	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1232574442152452	TCMDC-124422	chembl:CHEMBL527620	CHEMBL:CHEMBL527620	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	5-PHENOXYPHTHALIMIDE	chembl:CHEMBL1813518	CHEMBL:CHEMBL1813518	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.014206621	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2430910705356226	SJ000044417	chembl:CHEMBL609438	CHEMBL:CHEMBL609438	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	FLUOXASTROBIN	chembl:CHEMBL1902591	FLUOXASTROBIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	SJ000001592	chembl:CHEMBL591834	CHEMBL:CHEMBL591834	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.037693949	7-NITROINDAZOLE	drugbank:DB02207	7-NITROINDAZOLE	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.014699796	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	BUDESONIDE	rxcui:19831	BUDESONIDE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.027177884	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.021534247	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.1136529680426287	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.008047153	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.004278656	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001624217	MIDAZOLAM HYDROCHLORIDE	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.00346174	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.5676505	SORBINIL	ncit:C97357	SORBINIL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	CARFENTRAZONE-ETHYL	chembl:CHEMBL2145069	CARFENTRAZONE-ETHYL	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	PTAEROXYLIN	chembl:CHEMBL1527943	PTAEROXYLIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.018019105	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.010518364	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	RO-166491	chembl:CHEMBL1256177	CHEMBL:CHEMBL1256177	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	(E)-2-STYRYLCHROMONE	chembl:CHEMBL388823	CHEMBL:CHEMBL388823	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	NSC-98938	chembl:CHEMBL1939691	CHEMBL:CHEMBL1939691	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TENOVIN-1	chembl:CHEMBL1436543	CHEMBL:CHEMBL1436543	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PHENAZINE	chembl:CHEMBL119870	PHENAZINE	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.042006137	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	URAPIDIL	rxcui:39230	URAPIDIL	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	0.2907401508067248	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.014857858	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.030176823	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	RO-0505082	chembl:CHEMBL2164761	CHEMBL:CHEMBL2164761	FALSE	FALSE	FALSE
DAO	hgnc:2671	DAO	DTC	9/2/20	NULL	21.00306849427779	5-CARBOXYFURO[3,2-B]PYRROLE	chembl:CHEMBL492591	CHEMBL:CHEMBL492591	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	INDOMETHACIN MORPHOLINYLAMIDE	chembl:CHEMBL72631	INDOMETHACIN MORPHOLINYLAMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	TCMDC-125293	chembl:CHEMBL548629	CHEMBL:CHEMBL548629	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	BIPHENYL-4-AMINE	chembl:CHEMBL44201	BIPHENYL-4-AMINE	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.062509132	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.055563673	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	LULICONAZOLE	rxcui:1482680	LULICONAZOLE	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.2365210416022274	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.2853677784548614	(E),(E)-2,4-DECACIENAL	chembl:CHEMBL443949	CHEMBL:CHEMBL443949	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.043180651	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	INDOMETHACIN MORPHOLINYLAMIDE	chembl:CHEMBL72631	INDOMETHACIN MORPHOLINYLAMIDE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1962903597596056	CHLOROTRIANISENE	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	DEFERIPRONE	rxcui:11645	DEFERIPRONE	TRUE	FALSE	FALSE
TRPV4	hgnc:18083	TRPV4	DTC	9/2/20	NULL	1.29648571	NSC-677436	chembl:CHEMBL120580	CHEMBL:CHEMBL120580	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-124022	chembl:CHEMBL548017	CHEMBL:CHEMBL548017	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011806109	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	SJ000299520	chembl:CHEMBL592305	CHEMBL:CHEMBL592305	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.011098641	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.5966780822238011	GW501516	iuphar.ligand:2687	GW501516	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	MG-132	iuphar.ligand:8616	MG-132	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.294655843	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	FRAXETIN	chembl:CHEMBL54909	FRAXETIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	BAS-8770931	chembl:CHEMBL515495	CHEMBL:CHEMBL515495	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.070197421	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	0.3590268118679965	Marimastat	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.014206621	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.2917092846427472	GNF-PF-4078	chembl:CHEMBL584883	CHEMBL:CHEMBL584883	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	3.750547945	LOMIFYLLINE	rxcui:164423	LOMIFYLLINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	FENBENDAZOLE	rxcui:4325	FENBENDAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001048811	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	META-SIRTINOL	chembl:CHEMBL200762	CHEMBL:CHEMBL200762	FALSE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	DTC	9/2/20	NULL	1.875273972703374	MG-132	iuphar.ligand:8616	MG-132	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006113363	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	5,7-DIMETHOXYISOFLAVONE	chembl:CHEMBL308688	5,7-DIMETHOXYISOFLAVONE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.010987167	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	3,4-METHYLENEDIOXYB-NITROSTYRENE	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.2573905452730122	BEMESETRON	ncit:C80766	BEMESETRON	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.04321619	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.049302978	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	1.250182648468916	RETINYLRETINOATE	chembl:CHEMBL451039	RETINYLRETINOATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	NSC-98938	chembl:CHEMBL1939691	CHEMBL:CHEMBL1939691	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006397133	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
STAT6	hgnc:11368	STAT6	DTC	9/2/20	NULL	0.5000730593875666	NSC-119889	chembl:CHEMBL516616	CHEMBL:CHEMBL516616	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.305277158	PENICILLIOL B	chembl:CHEMBL513800	PENICILLIOL B	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-1782	chembl:CHEMBL579315	CHEMBL:CHEMBL579315	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007813642	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	SERTACONAZOLE NITRATE	rxcui:236601	SERTACONAZOLE NITRATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	AROMATICIN	chembl:CHEMBL494255	AROMATICIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	NSC-119889	chembl:CHEMBL516616	CHEMBL:CHEMBL516616	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	OXYPHENCYCLIMINE HYDROCHLORIDE	rxcui:91164	OXYPHENCYCLIMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	TCMDC-125140	chembl:CHEMBL525106	CHEMBL:CHEMBL525106	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.015477574	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	DIOXYBENZONE	rxcui:23350	DIOXYBENZONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BENSULIDE	chembl:CHEMBL1895252	BENSULIDE	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:3357	iuphar.ligand:3357	L902688	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	ALEXIDINE DIHYDROCHLORIDE	chembl:CHEMBL554041	ALEXIDINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.004565091	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011143394	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	DTC	9/2/20	NULL	0.080042182	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:4247	iuphar.ligand:4247	LY382884	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	DTC	9/2/20	NULL	0.072927321	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	DTC	9/2/20	NULL	0.084146909	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	DTC	9/2/20	NULL	0.084146909	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1686	iuphar.ligand:1686	[(PF)PHE4]N/OFQ-(1-13)-NH2	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	DTC	9/2/20	NULL	0.085239726	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	FENBENDAZOLE	rxcui:4325	FENBENDAZOLE	TRUE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.069454592	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.014369915	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TRIPHENYL PHOSPHATE	chembl:CHEMBL454511	TRIPHENYL PHOSPHATE	FALSE	FALSE	FALSE
STEROID 17-ALPHA-MONOOXYGENASE	hgnc:2593	CYP17A1	TTD	2020.06.01	NULL	3.125456621172291	Abiraterone acetate	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	E927A	chembl:CHEMBL28517	E927A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ETHYLESTRENOL	rxcui:4162	ETHYLESTRENOL	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.035890411	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.06714536	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	1.009762908	NSC-37642	chembl:CHEMBL1707907	CHEMBL:CHEMBL1707907	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.013975957	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	DIHYDROERGOCRISTINE MESYLATE	ncit:C75939	DIHYDROERGOCRISTINE MESYLATE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1000146118775133	5,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484662	CHEMBL:CHEMBL484662	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10642	iuphar.ligand:10642	MRL-871	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.063722902	CHLOROPHENYLPIPERAZINE	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	NILE RED	chembl:CHEMBL144472	NILE RED	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007749066	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.082171629	GNF-PF-4384	chembl:CHEMBL602763	CHEMBL:CHEMBL602763	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.002186317	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001276441	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001807182	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.072826174	BENZO[B]FLUORANTHENE	chembl:CHEMBL1337502	BENZO[B]FLUORANTHENE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	ENCLOMIPHENE	ncit:C28211	ENCLOMIPHENE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	OncoKB	23-Jul-20	NULL	1.944728564284981	BLU-667	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
BRSK2	hgnc:11405	BRSK2	DTC	9/2/20	inhibitor	1.312691780892362	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	ANISOMYCIN	ncit:C95312	ANISOMYCIN	FALSE	FALSE	FALSE
ZNF697	hgnc:32034	ZNF697	PharmGKB	4/5/24	NULL	3.500511415712966	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.008529511	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.006215397	E-DOXEPIN	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.017059022	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
TDP2	hgnc:17768	TDP2	DTC	9/2/20	NULL	3.500511415712967	(-)-DICENTRINE	chembl:CHEMBL478754	CHEMBL:CHEMBL478754	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.3454452054979901	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1562728310586145	EZETIMIBE	rxcui:341248	EZETIMIBE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002359895	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	GNF-PF-2947	chembl:CHEMBL581677	CHEMBL:CHEMBL581677	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.070574827	BERGAPTOL	chembl:CHEMBL242711	BERGAPTOL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007749066	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	TCMDC-124479	chembl:CHEMBL587259	CHEMBL:CHEMBL587259	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.729273212	GNF-PF-4322	chembl:CHEMBL604100	CHEMBL:CHEMBL604100	FALSE	FALSE	FALSE
NR2F2	hgnc:7976	NR2F2	DTC	9/2/20	NULL	1.250182648468916	TCMDC-125620	chembl:CHEMBL530291	CHEMBL:CHEMBL530291	FALSE	FALSE	FALSE
TEK	hgnc:11724	TEK	DTC	9/2/20	NULL	0.546954909	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
IDE	hgnc:5381	IDE	DTC	9/2/20	NULL	1.750255707856483	N-(4-NITROPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1574420	CHEMBL:CHEMBL1574420	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.005697447	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.013313304	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP3A43	hgnc:17450	CYP3A43	PharmGKB	4/5/24	NULL	0.2083637747448194	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	OXOGLAUCINE	iuphar.ligand:12559	OXOGLAUCINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.020575106	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.020721259	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.045461187	GNF-PF-4085	chembl:CHEMBL528181	CHEMBL:CHEMBL528181	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.02302968	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.002210756	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	DNDI1417413	chembl:CHEMBL1343568	CHEMBL:CHEMBL1343568	FALSE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	DTC	9/2/20	NULL	4.039051633514961	SB-744185	chembl:CHEMBL490417	CHEMBL:CHEMBL490417	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.003070624	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.011993529	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004101201	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	1.400204566285186	SPLICEOSTATIN-A	chembl:CHEMBL1221944	CHEMBL:CHEMBL1221944	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	1-[2-(TRIFLUOROMETHYL)PHENYL]IMIDAZOLE	iuphar.ligand:4331	TRIM	FALSE	FALSE	FALSE
PNLIP	hgnc:9155	PNLIP	DTC	9/2/20	NULL	13.12691780892362	HOOKEROSIDE B	chembl:CHEMBL444815	HOOKEROSIDE B	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.021449212	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	RIFAMYCIN SODIUM	rxcui:236475	RIFAMYCIN SODIUM	TRUE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	0.4339476961627644	PYRIMETHAMINE	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.018942161	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.1553481397505754	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.1528607605114832	BISDEMETHOXYCURCUMIN	chembl:CHEMBL105350	BISDEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	SJ000018298	chembl:CHEMBL591412	CHEMBL:CHEMBL591412	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.014622019	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.003001124	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.014369915	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	1.280674908	ISOPROPYL ISOTHIOCYANATE	chembl:CHEMBL2208211	ISOPROPYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-525334	chembl:CHEMBL401570	CHEMBL:CHEMBL401570	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.041672755	MESO-2,3-DIMERCAPTOSUCCINIC ACID	rxcui:3446	SUCCIMER	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	2.282942227638891	30-NORHEDERAGENIN	chembl:CHEMBL1081326	CHEMBL:CHEMBL1081326	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.01484106	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NOX1	hgnc:7889	NOX1	DTC	9/2/20	NULL	1.093909817410302	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	4-HYDROXYBENZALDEHYDE PHENYLHYDRAZONE	chembl:CHEMBL224032	CHEMBL:CHEMBL224032	FALSE	FALSE	FALSE
PIP4K2A	hgnc:8997	PIP4K2A	DTC	9/2/20	NULL	1.750255707856483	GNF-PF-1678	chembl:CHEMBL580340	CHEMBL:CHEMBL580340	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.026519026	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.009260612	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003767907	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB]	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	SANTIN	chembl:CHEMBL161957	SANTIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.031555091	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	DESACETYL SALANNIN	chembl:CHEMBL2270444	DESACETYL SALANNIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	chembl:CHEMBL1333512	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.2414145803939976	RADICICOL	ncit:C1462	RADICICOL	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	3.500511415712966	BPR-890	chembl:CHEMBL498746	CHEMBL:CHEMBL498746	FALSE	FALSE	FALSE
PTGES	hgnc:9599	PTGES	DTC	9/2/20	NULL	0.2612321952024602	CELECOXIB	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1000146118775133	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
TGFBR1	hgnc:11772	TGFBR1	DTC	9/2/20	inhibitor	0.1875273972703375	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1378154100674396	GALLAMINE	rxcui:4638	GALLAMINE	FALSE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	DTC	9/2/20	NULL	0.5357925636295356	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.002362018	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	HEPTACHLOR	chembl:CHEMBL194400	HEPTACHLOR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00299804	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	OBTUSAQUINONE	chembl:CHEMBL1333653	OBTUSAQUINONE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.026519026	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
CCBL1	hgnc:1564	KYAT1	DTC	9/2/20	NULL	35.00511415712966	TRANS-3-INDOLEACRYLIC ACID	chembl:CHEMBL445966	CHEMBL:CHEMBL445966	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	CLORGILINE	ncit:C77522	CLORGILINE	FALSE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.1411496538593938	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.4688184931758437	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	GNF-PF-1319	chembl:CHEMBL235891	CHEMBL:CHEMBL235891	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	(S)-PROMETHAZINE	chembl:CHEMBL251904	(S)-PROMETHAZINE	FALSE	FALSE	FALSE
EPHA3	hgnc:3387	EPHA3	DTC	9/2/20	inhibitor	0.1458546423213736	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.024241769	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-3906	chembl:CHEMBL599102	CHEMBL:CHEMBL599102	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	TCMDC-125465	chembl:CHEMBL536151	CHEMBL:CHEMBL536151	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.035890411	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001631484	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015201989	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	APOCIDEINE	chembl:CHEMBL154709	APOCIDEINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.019107595	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2083637747448194	GNF-PF-1399	chembl:CHEMBL578504	CHEMBL:CHEMBL578504	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	A-70108	iuphar.ligand:6077	A68930	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.017243899	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	chembl:CHEMBL1348974	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.050781113	D-ASPARTATE	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.029170928	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.038131933	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.013120358	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	TCMDC-125140	chembl:CHEMBL525106	CHEMBL:CHEMBL525106	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1250182648468916	CARBARIL	ncit:C76389	CARBARIL	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	CICLOPIROX OLAMINE	rxcui:52172	CICLOPIROX OLAMINE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.061412481	QUINOXALINE-2-CARBOXYLIC ACID	chembl:CHEMBL151797	CHEMBL:CHEMBL151797	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	DIOSMIN	rxcui:3489	DIOSMIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	GW0742	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	DTC	9/2/20	NULL	0.051782713	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004931224	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	TYRPHOSTIN 25	chembl:CHEMBL310798	TYRPHOSTIN 25	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.013814173	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.021554873	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	PHENOXYBENZAMINE HYDROCHLORIDE	rxcui:71512	PHENOXYBENZAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.007952093	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.076765601	4,4'-DIMETHOXYDALBERGIONE	chembl:CHEMBL1436980	4,4'-DIMETHOXYDALBERGIONE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000642547	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	DIAMIDE	chembl:CHEMBL1255835	DIAMIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00517674	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	KARANJIN	chembl:CHEMBL208484	KARANJIN	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.3302369260106572	XANTHOHUMOL	ncit:C121950	XANTHOHUMOL	FALSE	FALSE	FALSE
FPR1	hgnc:3826	FPR1	DTC	9/2/20	NULL	0.2500365296937833	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.032173818	DEQUALINIUM	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	DNDI1417413	chembl:CHEMBL1343568	CHEMBL:CHEMBL1343568	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.024861587	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
CA12	hgnc:1371	CA12	DTC	9/2/20	NULL	0.7501095890813501	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.017059022	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.020510809	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	12-METHYL TETRADECANOIC ACID	chembl:CHEMBL495852	CHEMBL:CHEMBL495852	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	FANCHININ	drugbank:DB14066	TETRANDRINE	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.7955707762984013	BISDEMETHOXYCURCUMIN	chembl:CHEMBL105350	BISDEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	METHABENZTHIAZURON	chembl:CHEMBL1890813	METHABENZTHIAZURON	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	DTC	9/2/20	NULL	0.068169648	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.042276708	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	SR-59230A	iuphar.ligand:547	SR59230A	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	BENPERIDOL	rxcui:1373	BENPERIDOL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	DEXPROPRANOLOL	ncit:C77944	DEXPROPRANOLOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007003824	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.0135995	DISOPYRAMIDE PHOSPHATE	rxcui:203178	DISOPYRAMIDE PHOSPHATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	DNDI1417207	chembl:CHEMBL256062	CHEMBL:CHEMBL256062	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1182605208011137	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003499578	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	DEGUELIN	ncit:C63666	DEGUELIN	FALSE	FALSE	FALSE
PTK6	hgnc:9617	PTK6	DTC	9/2/20	NULL	0.364636606	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	8-(3-CHLOROSTYRYL)CAFFEINE	iuphar.ligand:5609	CSC	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	THIOPERAMIDE	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	CIMIRACEMATE A	chembl:CHEMBL1076184	CIMIRACEMATE A	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.1535312024435511	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.04464938	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	6-DESOXYMORPHINE	chembl:CHEMBL410907	CHEMBL:CHEMBL410907	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	5-NITROACENAPHTHENE	chembl:CHEMBL423081	CHEMBL:CHEMBL423081	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010629083	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00626658	ENALAPRIL MALEATE	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.2465148884304905	ICOSAPENT	rxcui:90	EICOSAPENTAENOIC ACID	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.0055883	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.093098708	SQ-22536	chembl:CHEMBL64239	CHEMBL:CHEMBL64239	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	ALAZANINE	chembl:CHEMBL578063	ALAZANINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	BENZYL ISOTHIOCYANATE	drugbank:DB16860	BENZYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.4688184931758437	PHENYLETHENYLSEMICARBAZONE	chembl:CHEMBL74635	PHENYLETHENYLSEMICARBAZONE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NAPROPAMIDE	chembl:CHEMBL1877460	NAPROPAMIDE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.003120442	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.012710644	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.3621218705909965	NVP-AUY922	iuphar.ligand:9261	LUMINESPIB	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	7,3',4'-TRIMETHOXYISOFLAVONE	chembl:CHEMBL273891	CHEMBL:CHEMBL273891	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.3205596534535683	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003767907	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.011741429	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.048618214	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.022632617	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008176218	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.2263261691193728	GNF-PF-4337	chembl:CHEMBL277148	CHEMBL:CHEMBL277148	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	inhibitor	0.046881849	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	HARMALOL	chembl:CHEMBL129177	HARMALOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.029845209	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	2-PICOLINIC ACID	chembl:CHEMBL72628	2-PICOLINIC ACID	FALSE	FALSE	FALSE
SLC28A2	hgnc:11002	SLC28A2	DTC	9/2/20	NULL	0.7001022831425934	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	2.019525817	BERKELEYACETAL B	chembl:CHEMBL252921	BERKELEYACETAL B	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.6035364509849942	(+)-CIS-DIOXOLANE IODIDE	chembl:CHEMBL387632	CHEMBL:CHEMBL387632	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FANETIZOLE	ncit:C72775	FANETIZOLE	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.031032903	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.020836377	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	1,5-NAPHTHALENEDIAMINE	chembl:CHEMBL538965	CHEMBL:CHEMBL538965	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	GNF-PF-1509	chembl:CHEMBL576412	CHEMBL:CHEMBL576412	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.013411921	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	1.312691780892362	PEVONEDISTAT	ncit:C77906	PEVONEDISTAT	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.091159151	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	STROPHANTHIDIN	chembl:CHEMBL111743	STROPHANTHIDIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.004191225	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.012486961	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
SLC28A3	hgnc:16484	SLC28A3	DTC	9/2/20	NULL	1.000146118775133	ADENOSINE	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.081030357	TCMDC-125465	chembl:CHEMBL536151	CHEMBL:CHEMBL536151	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.057260274	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.033919684	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.8204323630577265	XR-9544	chembl:CHEMBL444075	CHEMBL:CHEMBL444075	FALSE	FALSE	FALSE
TXNRD2	hgnc:18155	TXNRD2	DTC	9/2/20	NULL	1.009762908	ARSENIC TRIOXIDE	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	DTC	9/2/20	NULL	0.023440925	CLOPIDOGREL	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	SPARFLOXACIN	rxcui:18469	SPARFLOXACIN	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007086055	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.750109589	DNDI1417773	chembl:CHEMBL1379900	CHEMBL:CHEMBL1379900	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.1071585127259071	NSC-8186	chembl:CHEMBL122355	CHEMBL:CHEMBL122355	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	SJ000112730	chembl:CHEMBL591178	CHEMBL:CHEMBL591178	FALSE	FALSE	FALSE
CDK19	hgnc:19338	CDK19	DTC	9/2/20	NULL	0.08334551	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
MMP12	hgnc:7158	MMP12	DTC	9/2/20	NULL	0.8975670296699916	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	0.3182283105193606	PYRIMETHAMINE	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.036013492	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	FLAVOKAWAIN B	chembl:CHEMBL104255	FLAVOKAWAIN B	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	0.5385402178019949	NAPHTHOQUINONE	chembl:CHEMBL55934	NAPHTHOQUINONE	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.2500365296937833	MIGALASTAT	rxcui:2054252	MIGALASTAT	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.046549354	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	DIAMIDE	chembl:CHEMBL1255835	DIAMIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.005046873	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.042619863	NSC-92207	chembl:CHEMBL139935	CHEMBL:CHEMBL139935	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.029416062	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
PRKCI	hgnc:9404	PRKCI	DTC	9/2/20	NULL	0.045265234	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	PHENYLHYDRAZINE	rxcui:8167	PHENYLHYDRAZINE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.041085815	3,4-METHYLENEDIOXYB-NITROSTYRENE	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	inhibitor	0.030527716	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007792334	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.032472277	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.040235763	PHENYLSTIBONIC ACID	chembl:CHEMBL1369257	PHENYLSTIBONIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	PAPAVERINE HYDROCHLORIDE	rxcui:203132	PAPAVERINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	2-MERCAPTOBENZOTHIAZOLE	rxcui:1358845	2-MERCAPTOBENZOTHIAZOLE	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.011757204	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.1491695205559502	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.3225286930939465	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PHENOXYCARB	chembl:CHEMBL15780	PHENOXYCARB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	PERGOLIDE	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
MARK4	hgnc:13538	MARK4	DTC	9/2/20	NULL	0.108040476	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
MUSK	hgnc:7525	MUSK	DTC	9/2/20	inhibitor	0.6563458904461813	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	SALSOLINOL HYDROBROMIDE	chembl:CHEMBL553751	SALSOLINOL HYDROBROMIDE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.027563082	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
PSMB8	hgnc:9545	PSMB8	DTC	9/2/20	NULL	4.773424657790408	LACTACYSTIN	chembl:CHEMBL374308	LACTACYSTIN	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.078136416	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.032173818	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002610374	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.015123177	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	inhibitor	0.028536778	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
GDA	hgnc:4212	GDA	DTC	9/2/20	NULL	35.00511415712966	NSC-7861	chembl:CHEMBL321248	7-METHYLXANTHINE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.016558711	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.019680536	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	OXOTREMORINE	iuphar.ligand:302	OXOTREMORINE	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	DTC	9/2/20	NULL	0.049864835	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	DTC	9/2/20	NULL	0.7955707762984013	AZD-4017	drugbank:DB14875	AZD-4017	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	HARMOL HYDROCHLORIDE	chembl:CHEMBL1449575	HARMOL HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000991047	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002165622	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	DTC	9/2/20	NULL	1.121958787087489	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.016377939	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW827099X	chembl:CHEMBL365297	GW827099X	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	GALANGIN	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.037505479	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.08334551	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.098884503	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CLINAFLOXACIN	ncit:C74372	CLINAFLOXACIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.009242681	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	CID 660258	chembl:CHEMBL259805	CHEMBL:CHEMBL259805	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	OXYMETHOLONE	rxcui:7813	OXYMETHOLONE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	DIHYDROERGOCRISTINE MESYLATE	ncit:C75939	DIHYDROERGOCRISTINE MESYLATE	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	2.838252499226729	RO-4746092	chembl:CHEMBL2203706	CHEMBL:CHEMBL2203706	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.1902451856365742	AG-1296	iuphar.ligand:5915	AG 1296	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2083637747448194	BI-2536	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	chembl:CHEMBL1348974	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.02646556	DIHYDROXIDINE	chembl:CHEMBL1224528	DIHYDROXIDINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	SALMETEROL XINAFOATE	rxcui:72616	SALMETEROL XINAFOATE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.070765056	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	INDIGO	rxcui:1426889	INDIGO	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001365893	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1141471113819445	CHLOROTRIANISENE	rxcui:2397	CHLOROTRIANISENE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	GUANFACINE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.009115915	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.1902451856365742	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2430910705356226	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2243917574174978	SCRIPTAID	drugbank:DB17053	SCRIPTAID	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	inhibitor	0.057073556	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.3977853881492007	GW305074X	chembl:CHEMBL1880739	GW305074X	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	1.312691780892362	N-DEACETYLCOLCHICEINE	ncit:C1264	TRIMETHYLCOLCHICINIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	ENCLOMIPHENE	ncit:C28211	ENCLOMIPHENE	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.088333021	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.031032903	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.040515178	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.081030357	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.065389379	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.1973972602845657	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
GLA	hgnc:4296	GLA	DTC	9/2/20	NULL	0.2885036881082115	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
TRPC5	hgnc:12337	TRPC5	DTC	9/2/20	NULL	7.001022831425932	NSC-677436	chembl:CHEMBL120580	CHEMBL:CHEMBL120580	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	SB-200646	chembl:CHEMBL85194	CHEMBL:CHEMBL85194	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.010440977	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.026830696	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.015075415	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.8751278539282416	2,4-DIAMINOTOLUENE	chembl:CHEMBL541230	CHEMBL:CHEMBL541230	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.050978322	NSC-130813	chembl:CHEMBL463783	CHEMBL:CHEMBL463783	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	DTC	9/2/20	NULL	0.1750255707856483	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.1458546423213736	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	SAPPANONE A DIMETHYL ETHER	chembl:CHEMBL1489223	SAPPANONE A DIMETHYL ETHER	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	DTC	9/2/20	inhibitor	0.027929612	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	GNF-PF-1678	chembl:CHEMBL580340	CHEMBL:CHEMBL580340	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	KARANJIN	chembl:CHEMBL208484	KARANJIN	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.03070624	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.049302978	(-)-DICENTRINE	chembl:CHEMBL478754	CHEMBL:CHEMBL478754	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	(-)-U-50488	chembl:CHEMBL58033	(-)-U-50488	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	BENZO[DEF]CHRYSENE	chembl:CHEMBL31184	BENZO[DEF]CHRYSENE	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.0095957	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	7-HYDROXY ISOFLAVONE	chembl:CHEMBL491981	7-HYDROXY ISOFLAVONE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	7-HYDROXY ISOFLAVONE	chembl:CHEMBL491981	7-HYDROXY ISOFLAVONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000217742	chembl:CHEMBL591887	CHEMBL:CHEMBL591887	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.008651783	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	R(-)-APOCODEINE HCL	chembl:CHEMBL1256735	CHEMBL:CHEMBL1256735	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	2-METHOXYPHENAZINE	chembl:CHEMBL1420181	CHEMBL:CHEMBL1420181	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.019687916	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	DTC	9/2/20	NULL	1.750255707856483	SB-269970	drugbank:DB13988	SB-269970	FALSE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.036013492	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.0023813	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	DTC	9/2/20	NULL	0.1203384367510187	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	DTC	9/2/20	NULL	0.1172918940484613	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	DTC	9/2/20	NULL	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	BERBERINE	rxcui:1437	BERBERINE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.018540844	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	(S)-PINACIDIL	chembl:CHEMBL251647	(S)-PINACIDIL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.009357988	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	GS-39783	iuphar.ligand:5446	GS39783	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	5-PHENOXYPHTHALIMIDE	chembl:CHEMBL1813518	CHEMBL:CHEMBL1813518	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	7-HYDROXY ISOFLAVONE	chembl:CHEMBL491981	7-HYDROXY ISOFLAVONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	MONTELUKAST	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1861974157294131	INDOMETHACIN MORPHOLINYLAMIDE	chembl:CHEMBL72631	INDOMETHACIN MORPHOLINYLAMIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00506733	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.046798281	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	GNF-PF-5183	chembl:CHEMBL577660	CHEMBL:CHEMBL577660	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00551957	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.045461187	GNF-PF-3201	chembl:CHEMBL581872	CHEMBL:CHEMBL581872	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.025840389	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.01186614	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	1.458546423213736	DIMETHYLSPINGOSINE	chembl:CHEMBL322333	DIMETHYLSPINGOSINE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	FDA	10-Apr-24	NULL	0.2778183663264258	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.008804103	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	FDA	10-Apr-24	NULL	2.407466349146467	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.075550606	Blinatumomab	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.2631963470460877	Busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
STXBP2	hgnc:11445	STXBP2	FDA	10-Apr-24	NULL	13.12691780892362	Emapalumab-lzsg	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
RAB27A	hgnc:9766	RAB27A	FDA	10-Apr-24	NULL	13.12691780892362	Emapalumab-lzsg	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	FDA	10-Apr-24	NULL	0.2083637747448194	Emapalumab-lzsg	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	FDA	10-Apr-24	NULL	1.282909942931453	Encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.003405608	Duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SH2D1A	hgnc:10820	SH2D1A	FDA	10-Apr-24	NULL	13.12691780892362	Emapalumab-lzsg	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.029170928	Hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.525076712	Sulfadiazine	rxcui:10171	SULFADIAZINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.1151484018326633	Tipiracil	rxcui:10803	TRIFLURIDINE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	FDA	10-Apr-24	NULL	0.1511209794852536	Tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	0.1582152052299645	ALISERTIB	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.1618941559168381	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.1480479452134243	AZD8931	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
MAPKAP1	hgnc:18752	MAPKAP1	MyCancerGenome	20-Jun-17	inhibitor	0.7955707762984016	MLN0128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	MyCancerGenome	20-Jun-17	inhibitor	0.2083637747448194	BI2536	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
SRC	hgnc:11283	SRC	MyCancerGenome	20-Jun-17	inhibitor	0.4167275494896389	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.065799087	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
CD74	hgnc:1697	CD74	MyCancerGenome	20-Jun-17	antibody	52.50767123569449	MILATUZUMAB	ncit:C66983	MILATUZUMAB	FALSE	TRUE	TRUE
TNFRSF10A	hgnc:11904	TNFRSF10A	MyCancerGenome	20-Jun-17	antibody	42.00613698855559	MAPATUMUMAB	ncit:C61502	MAPATUMUMAB	FALSE	TRUE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	MyCancerGenome	20-Jun-17	other/unknown	0.9512259281828714	TANESPIMYCIN	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.059364241	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ABCB4	hgnc:45	ABCB4	NCI	14-Sep-17	NULL	0.8751278539282416	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.058602312	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.652269208	NG-MONOMETHYL-L-ARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.760980743	2,3-DIDEOXYADENOSINE	ncit:C429	DIDEOXYADENOSINE	FALSE	FALSE	FALSE
ADK	hgnc:257	ADK	NCI	14-Sep-17	NULL	1.750255707856483	2,3-DIDEOXYADENOSINE	ncit:C429	DIDEOXYADENOSINE	FALSE	FALSE	FALSE
ADH1C	hgnc:251	ADH1C	NCI	14-Sep-17	NULL	0.025644772	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	NCI	14-Sep-17	NULL	0.012175692	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.091476779	5-FLUORODEOXYURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.960506181	ISIS 3521	rxcui:2634355	APRINOCARSEN	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.2561349816375342	SAPONIN	ncit:C823	SAPONIN	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.029106248	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
CCK	hgnc:1569	CCK	NCI	14-Sep-17	NULL	35.00511415712966	VIRGINIAMYCIN M1	drugbank:DB01669	VIRGINIAMYCIN M1	FALSE	FALSE	FALSE
CCL5	hgnc:10632	CCL5	NCI	14-Sep-17	NULL	26.25383561784724	OX40 LIGAND	ncit:C1548	RECOMBINANT OX40 LIGAND	FALSE	FALSE	FALSE
CCL8	hgnc:10635	CCL8	NCI	14-Sep-17	NULL	1.346350544504987	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	13.12691780892362	MIP-1BETA	ncit:C1467	RECOMBINANT HUMAN MACROPHAGE INFLAMMATORY PROTEIN-1 BETA	FALSE	FALSE	FALSE
CD1A	hgnc:1634	CD1A	NCI	14-Sep-17	NULL	2.282942227638891	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	0.3750547945406749	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
CD86	hgnc:1705	CD86	NCI	14-Sep-17	NULL	1.296485709523321	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
CD86	hgnc:1705	CD86	NCI	14-Sep-17	NULL	0.2917092846427472	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
CDC25C	hgnc:1727	CDC25C	NCI	14-Sep-17	NULL	0.1810609352954982	CDDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.026227608	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.053771297	CPT-11	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.038937836	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.065923002	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.3535870116881784	BSO	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.4667348554283955	ACLARUBICIN	rxcui:239	ACLARUBICIN	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	1.400204566285186	BCG VACCINE	ncit:C298	BCG VACCINE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1000146118775133	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
CSH1	hgnc:2440	CSH1	NCI	14-Sep-17	NULL	26.25383561784724	MARIJUANA	ncit:C26659	MARIJUANA	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1272913242077442	MECHLORETHAMINE	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.2800409132570373	PROCARBAZINE	rxcui:8702	PROCARBAZINE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.2187819634820604	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.5834185692854944	BISPECIFIC ANTIBODIES	ncit:C1454	BISPECIFIC ANTIBODY	FALSE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.1250182648468916	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	1.093909817410302	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	1.875273972703375	VALERIAN	rxcui:253206	VALERIAN ROOT EXTRACT	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.3454452054979901	AUTOLOGOUS DENDRITIC CELLS	ncit:C2594	THERAPEUTIC AUTOLOGOUS DENDRITIC CELLS	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.022080602	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.4953553890159858	LACTULOSE	rxcui:6218	LACTULOSE	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.2273059360852575	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.042741287	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.1234022825750752	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	1.050153425	MAGNESIUM SULFATE	rxcui:1311625	MAGNESIUM SULFATE ANHYDROUS	TRUE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.091317689	12-O-TETRADECANOYLPHORBOL-13-ACETATE	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
GCLC	hgnc:4311	GCLC	NCI	14-Sep-17	NULL	2.386712328895204	BUTHIONINE SULFOXIMINE	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	2.019525817	PD 098059	ncit:C1625	MEK INHIBITOR PD-98059	FALSE	FALSE	FALSE
GGH	hgnc:4248	GGH	NCI	14-Sep-17	NULL	0.7955707762984016	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
GFRA1	hgnc:4243	GFRA1	NCI	14-Sep-17	NULL	1.591141552596803	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
HGF	hgnc:4893	HGF	NCI	14-Sep-17	NULL	0.051859428	STI571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	0.6848826682916673	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	NCI	14-Sep-17	NULL	0.074690855	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
HMOX2	hgnc:5014	HMOX2	NCI	14-Sep-17	NULL	2.100306849	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
HOXB1	hgnc:5111	HOXB1	NCI	14-Sep-17	NULL	0.3462044257298538	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
HPRT1	hgnc:5157	HPRT1	NCI	14-Sep-17	NULL	1.093909817410302	3TC	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.6908904109959803	L-744,832	ncit:C1682	L-744,832	FALSE	FALSE	FALSE
HPRT1	hgnc:5157	HPRT1	NCI	14-Sep-17	NULL	13.12691780892362	NITROSOUREAS	ncit:C699	NITROSOUREA COMPOUND	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.2713574740862765	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.066005872	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.2035181055647073	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	NCI	14-Sep-17	NULL	0.1795134059339982	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	NCI	14-Sep-17	NULL	0.094608417	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
IBSP	hgnc:5341	IBSP	NCI	14-Sep-17	NULL	1.105424657593568	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	NCI	14-Sep-17	NULL	0.5834185692854945	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
IL11	hgnc:5966	IL11	NCI	14-Sep-17	NULL	0.3281729452230906	AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
IL6R	hgnc:6019	IL6R	NCI	14-Sep-17	NULL	0.218327115	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
IL8RB	hgnc:6027	CXCR2	NCI	14-Sep-17	NULL	0.3889457128569963	N-ACETYL-L-CYSTEINE	rxcui:197	ACETYLCYSTEINE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.6482428547616604	TOCOPHEROL ACETATE	rxcui:1046243	ALPHA-TOCOPHEROL ACETATE	TRUE	FALSE	FALSE
LOH19CR1	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.3940538179038987	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.060737619	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.5357925636295356	LYMPHOKINES	ncit:C621	RECOMBINANT LYMPHOKINE	FALSE	FALSE	FALSE
MAP2	hgnc:6839	MAP2	NCI	14-Sep-17	NULL	1.009762908	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.1286952726365061	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.024814589	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.2059124362184098	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.05051243	CPT-11	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.1223955040459079	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.2187819634820604	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.525076712	IMMUNOMODULATING AGENT	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.750109589	ELSAMICIN A	ncit:C1080	ELSAMITRUCIN	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	COBALT 60	ncit:C28239	COBALT CO-60	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.060008767	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.4688184931758437	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.3860858179095184	BUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.061628722	ICI 182,780	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.067231333	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
NR2C1	hgnc:7971	NR2C1	NCI	14-Sep-17	NULL	1.154014752432846	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	5.527123287967842	TINIDAZOLE	rxcui:10612	TINIDAZOLE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.017543492	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.1553481397505754	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	NCI	14-Sep-17	NULL	0.2375912725597036	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.040515178	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.092606122	SELECTIVE ESTROGEN RECEPTOR MODULATOR	ncit:C1821	SELECTIVE ESTROGEN RECEPTOR MODULATOR	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.062509132	AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1470803115845784	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	NCI	14-Sep-17	NULL	0.6250913242344582	LEPIRUDIN	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.056097939	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.010058941	CDDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.729273212	HYPERICUM PERFORATUM	rxcui:1310069	HYPOXIS HEMEROCALLIDEA ROOT EXTRACT	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	CALCIUM GLUCONATE	rxcui:1908	CALCIUM GLUCONATE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.029170928	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	TESTOLACTONE	rxcui:10378	TESTOLACTONE	TRUE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.4487835148349957	CONJUGATED ESTROGENS	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.3365876361262467	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.2243917574174978	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
PTHLH	hgnc:9607	PTHLH	NCI	14-Sep-17	NULL	4.375639269641208	MAGNESIUM SULFATE	rxcui:1311625	MAGNESIUM SULFATE ANHYDROUS	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.4487835148349957	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.5385402178019949	PROTEIN KINASE INHIBITOR	ncit:C1404	PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
RPS19	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.2991890098899971	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
SCD	hgnc:10571	SCD	NCI	14-Sep-17	NULL	0.5556367326528519	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.085796848	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
SAA1	hgnc:10513	SAA1	NCI	14-Sep-17	NULL	3.088686543276147	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.6035364509849942	ETHER	ncit:C29819	ETHER	FALSE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.1400204566285186	RECOMBINANT HUMAN INTERLEUKIN-2	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.8401227397711121	CANCER VACCINES	ncit:C1663	ANTINEOPLASTIC VACCINE	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.070574827	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.3763990769583834	TIMOLOL MALEATE	rxcui:42933	TIMOLOL MALEATE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.2822993077187876	MAGNESIUM SULFATE	rxcui:1311625	MAGNESIUM SULFATE ANHYDROUS	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.029845209	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
TNFRSF8	hgnc:11923	TNFRSF8	NCI	14-Sep-17	NULL	0.2430910705356226	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.04636439	SAPONIN	ncit:C823	SAPONIN	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:8793	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.325124899	DELTA 9-TETRAHYDROCANNABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	2.234368988752957	CARBOGEN	ncit:C1038	CARBOGEN	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	0.502465753	MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	NCI	14-Sep-17	NULL	0.1591141552596803	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.1875273972703374	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.08937476	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UMOD	hgnc:12559	UMOD	NCI	14-Sep-17	NULL	1.29648571	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.002562787	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.006314054	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.1493817104856173	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.3454452054979901	trastuzumab deruxtecan	rxcui:2267574	FAM-TRASTUZUMAB DERUXTECAN-NXKI	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.2734774543525755	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.28382525	carbidopa	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
ADO	hgnc:23506	ADO	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.8751278539282416	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.037505479	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.020203029	erythromycin	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.016304198	sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.012228149	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.023813003	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
USP5	hgnc:12628	USP5	PharmGKB	4/5/24	NULL	0.760980743	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
PHC1	hgnc:3182	PHC1	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NUCB2	hgnc:8044	NUCB2	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.7001022831425933	TNP-470	drugbank:DB08633	TNP-470	FALSE	FALSE	FALSE
OGDH	hgnc:8124	OGDH	PharmGKB	4/5/24	NULL	0.9211872146613069	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
MUC16	hgnc:15582	MUC16	NCI	14-Sep-17	NULL	22.50328767	B43.13	ncit:C1784	OREGOVOMAB	FALSE	FALSE	FALSE
NRXN1	hgnc:8008	NRXN1	PharmGKB	4/5/24	NULL	2.019525816757481	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.038467158	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TCF7L2	hgnc:11641	TCF7L2	PharmGKB	4/5/24	NULL	0.4565884455277782	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
MIEF2	hgnc:17920	MIEF2	PharmGKB	4/5/24	NULL	4.039051633514962	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MYBBP1A	hgnc:7546	MYBBP1A	PharmGKB	4/5/24	NULL	5.834185692854945	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
PYGL	hgnc:9725	PYGL	PharmGKB	4/5/24	NULL	1.458546423213736	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.1241316104862754	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	PharmGKB	4/5/24	NULL	0.013140058	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
HBEGF	hgnc:3059	HBEGF	PharmGKB	4/5/24	NULL	0.047049885	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
WWOX	hgnc:12799	WWOX	PharmGKB	4/5/24	NULL	0.3070624048871023	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.015925894	etidronic acid	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
AK4	hgnc:363	AK4	PharmGKB	4/5/24	NULL	2.917092846427472	adefovir dipivoxil	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
AKR7A2	hgnc:389	AKR7A2	PharmGKB	4/5/24	NULL	0.5770073762164231	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.057955487	pirtobrutinib	rxcui:2629338	PIRTOBRUTINIB	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.2169738480813822	normeperidine	chembl:CHEMBL1052	NORMEPERIDINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	PharmGKB	4/5/24	NULL	0.022078281	venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	0.729273212	lisinopril	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
RPL13	hgnc:10303	RPL13	PharmGKB	4/5/24	NULL	0.1807492985738192	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	0.6482428547616605	chlorthalidone	rxcui:2409	CHLORTHALIDONE	TRUE	FALSE	FALSE
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	0.1268301237577161	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
GALNT17	hgnc:16347	GALNT17	PharmGKB	4/5/24	NULL	4.773424657790409	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
SCNN1G	hgnc:10602	SCNN1G	PharmGKB	4/5/24	NULL	0.9723642821424906	torasemide	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
UHRF1	hgnc:12556	UHRF1	PharmGKB	4/5/24	NULL	0.5933070196123672	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
UNIPROT:Q9UQD0	hgnc:10596	SCN8A	TdgClinicalTrial	Jan-14	NULL	0.088996053	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
GPR83	hgnc:4523	GPR83	PharmGKB	4/5/24	NULL	3.500511415712966	candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
EPM2A	hgnc:3413	EPM2A	PharmGKB	4/5/24	NULL	0.4054646427466756	chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.1121958787087489	vindesine	rxcui:11204	VINDESINE	FALSE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1166837138570989	fluconazole	rxcui:4450	FLUCONAZOLE	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.1083749664307419	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.009788902	ivabradine	rxcui:1649480	IVABRADINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003454907	alprazolam	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.1187956362798518	alprazolam	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
GSTA2	hgnc:4627	GSTA2	PharmGKB	4/5/24	NULL	0.384671584	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
TBL1X	hgnc:11585	TBL1X	PharmGKB	4/5/24	NULL	3.281729452230906	levothyroxine	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
GSTM3	hgnc:4635	GSTM3	PharmGKB	4/5/24	NULL	0.4605936073306535	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
ACSS2	hgnc:15814	ACSS2	PharmGKB	4/5/24	NULL	0.2258394461750301	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
PSPH	hgnc:9577	PSPH	PharmGKB	4/5/24	NULL	21.00306849	methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
CBS	hgnc:1550	CBS	PharmGKB	4/5/24	NULL	4.200613698855561	methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.007341677	astemizole	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004894451	tolterodine	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006525935	artemisinin	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011012515	miconazole	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	0.4734548598913698	cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
LMNB2	hgnc:6638	LMNB2	PharmGKB	4/5/24	NULL	10.50153425	metreleptin	rxcui:1491625	METRELEPTIN	TRUE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.7955707762984016	telmisartan	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.1151484018326633	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:1520	hgnc:2545	CTSS	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:5677	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
DLG2	hgnc:2901	DLG2	PharmGKB	4/5/24	NULL	8.078103267029924	anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
UGT1A	hgnc:12529	UGT1A	PharmGKB	4/5/24	NULL	2.386712328895204	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.071731791	fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.08780547	troglitazone	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.8751278539282416	dolutegravir	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
MAP2K6	hgnc:6846	MAP2K6	PharmGKB	4/5/24	NULL	0.092118721	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	PharmGKB	4/5/24	NULL	0.017218453	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.01439355	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CDH13	hgnc:1753	CDH13	PharmGKB	4/5/24	NULL	0.070860555	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.013350539	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	1.105424657593568	methazolamide	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
SLC15A2	hgnc:10921	SLC15A2	PharmGKB	4/5/24	NULL	0.070860555	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.1001290450718812	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	PharmGKB	4/5/24	NULL	0.073922431	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MLLT3	hgnc:7136	MLLT3	PharmGKB	4/5/24	NULL	2.386712328895204	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
ANK3	hgnc:494	ANK3	PharmGKB	4/5/24	NULL	0.04321619	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
MGAT4A	hgnc:7047	MGAT4A	PharmGKB	4/5/24	NULL	0.4861821410712453	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
MIR2054	hgnc:37070	MIR2054	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
EXO1	hgnc:3511	EXO1	PharmGKB	4/5/24	NULL	0.6482428547616604	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.043902735	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.037121012	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
CSMD1	hgnc:14026	CSMD1	PharmGKB	4/5/24	NULL	0.2763561643983921	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.108711535	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.5114383561918295	glatiramer acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
EIF2AK4	hgnc:19687	EIF2AK4	PharmGKB	4/5/24	NULL	0.2302968036653267	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.7343730242754476	ciprofloxacin	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
SLC7A5	hgnc:11063	SLC7A5	PharmGKB	4/5/24	NULL	2.500365296937833	melphalan	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.095468493	ciprofloxacin	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	PharmGKB	4/5/24	NULL	0.060585775	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	PharmGKB	4/5/24	NULL	0.458240639	vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.9883796938483671	pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
SLC13A3	hgnc:14430	SLC13A3	PharmGKB	4/5/24	NULL	0.5770073762164231	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1166837138570989	meperidine	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CDH4	hgnc:1763	CDH4	PharmGKB	4/5/24	NULL	3.387591692625451	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	PharmGKB	4/5/24	NULL	0.5147810905460245	pirtobrutinib	rxcui:2629338	PIRTOBRUTINIB	TRUE	FALSE	FALSE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	0.3750547945406749	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
DIAPH3	hgnc:15480	DIAPH3	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	0.4000584475100533	ponatinib	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
SPP1	hgnc:11255	SPP1	ChEMBL	33	inhibitor	3.500511415712966	ASK-8007	chembl:CHEMBL2109530	ASK-8007	FALSE	FALSE	FALSE
AGPAT2	hgnc:325	AGPAT2	PharmGKB	4/5/24	NULL	10.50153425	metreleptin	rxcui:1491625	METRELEPTIN	TRUE	FALSE	FALSE
GALNT14	hgnc:22946	GALNT14	PharmGKB	4/5/24	NULL	0.1750255707856483	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCC6	hgnc:57	ABCC6	PharmGKB	4/5/24	NULL	0.021087418	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1750255707856483	nitrofurazone	rxcui:7455	NITROFURAZONE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	PharmGKB	4/5/24	NULL	0.008374429	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.1154014752432846	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
EPM2A	hgnc:3413	EPM2A	PharmGKB	4/5/24	NULL	0.1973972602845657	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UGT2B10	hgnc:12544	UGT2B10	PharmGKB	4/5/24	NULL	0.4605936073306535	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
AKR1C4	hgnc:387	AKR1C4	PharmGKB	4/5/24	NULL	0.5770073762164231	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
BTRC	hgnc:1144	BTRC	PharmGKB	4/5/24	NULL	1.129197231	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.2917092846427472	tadalafil	rxcui:358263	TADALAFIL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.003053304	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.078722146	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.044161204	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	PharmGKB	4/5/24	NULL	0.6563458904461812	galantamine	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.049107011	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	4.773424657790408	db-289	rxcui:718967	PAFURAMIDINE	FALSE	FALSE	FALSE
AKR1C3	hgnc:386	AKR1C3	PharmGKB	4/5/24	NULL	0.070010228	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SLC28A2	hgnc:11002	SLC28A2	PharmGKB	4/5/24	NULL	1.500219178162699	boceprevir	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1166837138570989	pitavastatin	rxcui:861634	PITAVASTATIN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1166837138570989	artemether	rxcui:18343	ARTEMETHER	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1166837138570989	pantoprazole	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
BSCL2	hgnc:15832	BSCL2	PharmGKB	4/5/24	NULL	10.50153425	metreleptin	rxcui:1491625	METRELEPTIN	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	3.818739726232327	artemether	rxcui:18343	ARTEMETHER	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.4412409347537353	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PSPH	hgnc:9577	PSPH	PharmGKB	4/5/24	NULL	21.00306849	l-methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.05073205	tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	1.500219178	entacapone	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.00591236	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	PharmGKB	4/5/24	NULL	0.048663273	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.3454452054979901	AV-412	drugbank:DB06021	AV-412	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.1695984213039228	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.069454592	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.4717670371580817	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	TALC	12-May-16	inhibitor	0.1620607136904151	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.3864200913449379	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
FOLR1	hgnc:3791	FOLR1	TALC	12-May-16	NULL	2.917092846427472	EPOFOLATE	drugbank:DB12266	EPOFOLATE	FALSE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.3062196950280639	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.2282942227638891	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.3205596534535683	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.1944728564284981	GIVINOSTAT	ncit:C71716	GIVINOSTAT	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.073954467	NEOVASTAT	drugbank:DB05387	NEOVASTAT	FALSE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	TALC	12-May-16	vaccine	0.6731752722524935	S-3304	drugbank:DB12149	S-3304	FALSE	FALSE	TRUE
BCL2	hgnc:990	BCL2	TALC	12-May-16	inhibitor	0.2001054544043235	NAVITOCLAX	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.1440539677248134	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	TALC	12-May-16	inhibitor	1.367387271762877	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	TALC	12-May-16	inhibitor	0.4375639269641208	GSK461364	ncit:C70948	POLO-LIKE KINASE 1 INHIBITOR GSK461364	FALSE	FALSE	TRUE
SRC	hgnc:11283	SRC	TALC	12-May-16	inhibitor	0.1136529680426287	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	TALC	12-May-16	inhibitor	0.2019525816757481	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.3968833804663227	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.1852122442176172	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.007496384	TESTOSTERONE	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	0.8078103267029922	ACC-001	chembl:CHEMBL2108058	VANUTIDE CRIDIFICAR	FALSE	FALSE	FALSE
UNIPROT:P01584	hgnc:5992	IL1B	TdgClinicalTrial	Jan-14	NULL	0.2287915957982331	AC-201	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
UNIPROT:P18510	hgnc:6000	IL1RN	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	AC-201	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2442217266776488	SALMETEROL	rxcui:36117	SALMETEROL	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.058622403945453	AZELASTINE	rxcui:18603	AZELASTINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1204304386139782	BUPRENORPHINE	rxcui:1819	BUPRENORPHINE	TRUE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	DRONABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
UNIPROT:P00915	hgnc:1368	CA1	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	CG100649	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
UNIPROT:P19438	hgnc:11916	TNFRSF1A	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	CYT-6091	ncit:C62538	COLLOIDAL GOLD-BOUND TUMOR NECROSIS FACTOR	FALSE	FALSE	FALSE
UNIPROT:Q13093	hgnc:9040	PLA2G7	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	DARAPLADIB	ncit:C72985	DARAPLADIB	FALSE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	CX717	chembl:CHEMBL4791762	CX-717	FALSE	FALSE	FALSE
UNIPROT:P42263	hgnc:4573	GRIA3	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	CX717	chembl:CHEMBL4791762	CX-717	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.075496292	DULOXETINE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.3977853881492007	CX717	chembl:CHEMBL4791762	CX-717	FALSE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	DEGARELIX	rxcui:475230	DEGARELIX	TRUE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.069454592	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.6429510763554428	EDOXABAN	rxcui:1599538	EDOXABAN	TRUE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.1434635826111871	E-10030	chembl:CHEMBL3301576	PEGPLERANIB SODIUM	FALSE	FALSE	FALSE
UNIPROT:Q16665	hgnc:4910	HIF1A	TdgClinicalTrial	Jan-14	NULL	0.7242437411819931	ENMD-1198	drugbank:DB05959	ENMD-1198	FALSE	FALSE	FALSE
UNIPROT:P07947	hgnc:12841	YES1	TdgClinicalTrial	Jan-14	NULL	0.008143249	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P05771	hgnc:9395	PRKCB	TdgClinicalTrial	Jan-14	NULL	1.367387271762877	ENZASTAURIN	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
UNIPROT:P07949	hgnc:9967	RET	TdgClinicalTrial	Jan-14	NULL	0.02091106	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	EPLIVANSERINE	ncit:C65517	EPLIVANSERIN	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	GANTACURIUM	drugbank:DB05710	GANTACURIUM	FALSE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	0.7955707762984014	NBI-42902	iuphar.ligand:1178	NBI-42902	FALSE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	NBI-42902	iuphar.ligand:1178	NBI-42902	FALSE	FALSE	FALSE
UNIPROT:P49354	hgnc:3782	FNTA	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	GGTI-2418	chembl:CHEMBL3218390	GGTI-2418	FALSE	FALSE	FALSE
UNIPROT:P15056	hgnc:1097	BRAF	TdgClinicalTrial	Jan-14	NULL	2.341819737097098	GSK2118436	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	1.544343271638073	ISS-1018	drugbank:DB05463	ISS-1018	FALSE	FALSE	FALSE
UNIPROT:P16070	hgnc:1681	CD44	TdgClinicalTrial	Jan-14	NULL	0.9211872146613068	HYALURONAN	rxcui:5463	HYALURONIC ACID	TRUE	FALSE	FALSE
UNIPROT:P29459	hgnc:5969	IL12A	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	HUMANIZED SMART ANTI-IL-12 ANTIBODY	drugbank:DB05848	HUMANIZED SMART ANTI-IL-12 ANTIBODY	FALSE	FALSE	FALSE
UNIPROT:Q08493	hgnc:8782	PDE4C	TdgClinicalTrial	Jan-14	NULL	0.2263261691193728	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
UNIPROT:Q16853	hgnc:550	AOC3	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
UNIPROT:Q9NR82	hgnc:6299	KCNQ5	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	ICA-105665	drugbank:DB06089	ICA-105665	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	2.151953739167807	IMC-3G3	rxcui:1855735	OLARATUMAB	TRUE	FALSE	FALSE
UNIPROT:P28845	hgnc:5208	HSD11B1	TdgClinicalTrial	Jan-14	NULL	3.088686543276147	INCB13739	drugbank:DB05064	INCB13739	FALSE	FALSE	FALSE
UNIPROT:P55157	hgnc:7467	MTTP	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	IMPLITAPIDE	ncit:C65901	IMPLITAPIDE	FALSE	FALSE	FALSE
UNIPROT:P15260	hgnc:5439	IFNGR1	TdgClinicalTrial	Jan-14	NULL	39.38075342677087	INTERFERON GAMMA-1B	rxcui:5882	INTERFERON GAMMA-1B	TRUE	TRUE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.729273212	INTERFERON BETA	chembl:CHEMBL2108510	INTERFERON BETA	TRUE	FALSE	FALSE
UNIPROT:Q13509	hgnc:20772	TUBB3	TdgClinicalTrial	Jan-14	NULL	0.058212496	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.090821275	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
UNIPROT:P04035	hgnc:5006	HMGCR	TdgClinicalTrial	Jan-14	NULL	1.121958787087489	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
UNIPROT:P17752	hgnc:12008	TPH1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	LX1032	rxcui:1872441	TELOTRISTAT ETHYL	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.091796628	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.029106248	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	TIZANIDINE	rxcui:236460	TIZANIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.030598876	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.028413242	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.032252869	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.1831662950082366	OXYMETAZOLINE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FGF1	hgnc:3665	FGF1	ChEMBL	33	activator	1.944728564284981	ALDAFERMIN	ncit:C169769	ALDAFERMIN	FALSE	FALSE	FALSE
UNIPROT:Q9Y277	hgnc:12674	VDAC3	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	OLESOXIME	ncit:C174604	OLESOXIME	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.082043236	OXYMETAZOLINE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.3697723326457359	OPC-28326	drugbank:DB05461	OPC-28326	FALSE	FALSE	FALSE
UNIPROT:P15502	hgnc:3327	ELN	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	PRT-201	chembl:CHEMBL3545070	VONAPANITASE	FALSE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.100976291	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
UNIPROT:P06737	hgnc:9725	PYGL	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	PSN357	drugbank:DB05044	PSN357	FALSE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	0.6081969641200136	RASAGILINE	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.1320947704042629	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.08334551	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.097236428	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P41180	hgnc:1514	CASR	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	RONACALERET	ncit:C81351	RONACALERET	FALSE	FALSE	FALSE
UNIPROT:P06276	hgnc:983	BCHE	TdgClinicalTrial	Jan-14	NULL	0.5625821918110125	RIVASTIGMINE	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:4079	iuphar.ligand:4079	[3H]CGP61594	FALSE	FALSE	FALSE
UNIPROT:Q02108	hgnc:4685	GUCY1A1	TdgClinicalTrial	Jan-14	NULL	1.400204566285186	RIOCIGUAT	rxcui:1439816	RIOCIGUAT	TRUE	FALSE	FALSE
UNIPROT:P56199	hgnc:6134	ITGA1	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	SAN-300	chembl:CHEMBL4297822	SAN-300	FALSE	FALSE	FALSE
NCBIGENE:401	hgnc:691	PHOX2A	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:2358	ncit:C66687	ZATEBRADINE	FALSE	FALSE	FALSE
UNIPROT:Q12882	hgnc:3012	DPYD	TdgClinicalTrial	Jan-14	NULL	1.981421556063943	GIMESTAT	ncit:C2416	GIMERACIL	FALSE	FALSE	FALSE
UNIPROT:P29474	hgnc:7876	NOS3	TdgClinicalTrial	Jan-14	NULL	0.7501095890813501	TETRAHYDROBIOPTERIN	rxcui:753340	SAPROPTERIN	TRUE	FALSE	FALSE
UNIPROT:Q9P1W9	hgnc:8987	PIM2	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	SGI-1776	drugbank:DB12494	SGI-1776	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00675253	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	SIFALIMUMAB	ncit:C95061	SIFALIMUMAB	FALSE	FALSE	FALSE
UNIPROT:P16471	hgnc:9446	PRLR	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	SOMATROPIN	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	TAS-108	drugbank:DB05966	TAS-108	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.074690855	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RICTOR	hgnc:28611	RICTOR	TALC	12-May-16	inhibitor	3.750547945	OSI 027	chembl:CHEMBL3120215	OSI-027	FALSE	FALSE	TRUE
UNIPROT:P06731	hgnc:1817	CEACAM5	TdgClinicalTrial	Jan-14	NULL	2.282942227638891	TF2	ncit:C82355	ANTI-CEA/ANTI-HSG BISPECIFIC MONOCLONAL ANTIBODY TF2	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.096967075	PILOCARPINE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P31350	hgnc:10452	RRM2	TdgClinicalTrial	Jan-14	NULL	3.029288725136221	TRIAPINE	ncit:C2242	TRIAPINE	FALSE	FALSE	TRUE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	0.7955707762984014	TRIPTORELIN PAMOATE	rxcui:338529	TRIPTORELIN PAMOATE	TRUE	FALSE	FALSE
UNIPROT:Q92847	hgnc:4267	GHSR	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	TZP-102	drugbank:DB16129	TZP-102	FALSE	FALSE	FALSE
UNIPROT:Q02750	hgnc:6840	MAP2K1	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
UNIPROT:P06028	hgnc:4703	GYPB	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	WX-G250	ncit:C1960	GIRENTUXIMAB	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.011124507	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
UNIPROT:O14733	hgnc:6847	MAP2K7	TdgClinicalTrial	Jan-14	NULL	0.7501095890813498	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.1151484018326633	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.2991890098899971	AMINOGLYCOSIDES	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1008469998124734	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
UNIPROT:P15941	hgnc:7508	MUC1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	YTTRIUM (90Y) CLIVATUZUMAB TETRAXETAN	iuphar.ligand:8087	YTTRIUM (90Y) CLIVATUZUMAB TETRAXETAN	FALSE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.1852122442176172	XP13512	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
UNIPROT:Q9NY47	hgnc:1400	CACNA2D2	TdgClinicalTrial	Jan-14	NULL	0.2778183663264259	XP13512	rxcui:1101333	GABAPENTIN ENACARBIL	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	YKP-10A	chembl:CHEMBL4297620	SOLRIAMFETOL	FALSE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.048618214	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.9376369863516875	5-CHLORO-[1,10]PHENANTHROLINE	chembl:CHEMBL317115	CHEMBL:CHEMBL317115	FALSE	FALSE	FALSE
UNIPROT:Q8NER1	hgnc:12716	TRPV1	TdgClinicalTrial	Jan-14	NULL	0.3659071166250487	ZUCAPSAICIN	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
UNIPROT:Q16678	hgnc:2597	CYP1B1	TdgClinicalTrial	Jan-14	NULL	1.591141552596803	ZYC300	drugbank:DB04986	ZYC300	FALSE	FALSE	FALSE
UNIPROT:P08185	hgnc:1540	SERPINA6	TEND	1-Aug-11	NULL	3.281729452230906	CICLESONIDE	rxcui:274964	CICLESONIDE	TRUE	FALSE	FALSE
UNIPROT:P03952	hgnc:6371	KLKB1	TdgClinicalTrial	Jan-14	NULL	3.750547945	BCX4161	ncit:C169799	AVORALSTAT	FALSE	FALSE	FALSE
UNIPROT:P20701	hgnc:6148	ITGAL	TdgClinicalTrial	Jan-14	NULL	0.6584034010745392	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.064944553	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.061737415	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.059532507	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.060984519	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.057700738	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.063300387	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.1117184494376478	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:O95069	hgnc:6277	KCNK2	TdgClinicalTrial	Jan-14	NULL	1.154014752432846	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TdgClinicalTrial	Jan-14	NULL	0.9053046764774914	DIVALPROEX SODIUM	rxcui:266856	DIVALPROEX SODIUM	TRUE	FALSE	FALSE
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	0.3424413341458336	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.4605936073306534	FLAVOXATE	rxcui:4440	FLAVOXATE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.099446347	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1553481397505754	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.032899543	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TdgClinicalTrial	Jan-14	NULL	7.001022831425932	PHENINDIONE	rxcui:8130	PHENINDIONE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1704794520639432	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.078136416	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.079798892	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.1470803115845784	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.2408608772279564	PROPOXYPHENE	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.1315981735230438	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.108711535	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	CancerCommons	25-Jul-13	inhibitor	0.046860929	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.2895643634321387	PYRIDOSTIGMINE	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	0.5515511684421691	TACRINE	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.087318744	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	5.000730593875666	STREPTOKINASE	rxcui:10106	STREPTOKINASE	TRUE	FALSE	FALSE
UNIPROT:P42684	hgnc:77	ABL2	TEND	1-Aug-11	NULL	0.039341412	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P62158	hgnc:1442	CALM1	TEND	1-Aug-11	NULL	2.917092846427472	APRINDINE	rxcui:1054	APRINDINE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	CancerCommons	25-Jul-13	inhibitor	0.1512704997187101	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
UNIPROT:O00305	hgnc:1404	CACNB4	TEND	1-Aug-11	NULL	0.1795134059339982	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TEND	1-Aug-11	NULL	0.1093909817410302	AMLODIPINE	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TEND	1-Aug-11	NULL	0.6177373086552295	MARINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	1.336059069138614	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.2234368988752957	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P50416	hgnc:2328	CPT1A	TEND	1-Aug-11	NULL	1.154014752432846	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
UNIPROT:P23786	hgnc:2330	CPT2	TEND	1-Aug-11	NULL	0.326134604	PERHEXILINE	rxcui:8050	PERHEXILINE	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.4734548598913698	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
UNIPROT:P21964	hgnc:2228	COMT	TEND	1-Aug-11	NULL	1.500219178	ENTACAPONE	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.058622403945453	AZELASTINE	rxcui:18603	AZELASTINE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.4861821410712453	BENZTROPINE	rxcui:1424	BENZTROPINE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	CGI	2/1/22	NULL	0.014881721	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P04626	hgnc:3430	ERBB2	TEND	1-Aug-11	NULL	0.3677319929494733	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.063300387	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.082429625	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.060984519	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.059532507	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
ERCC1	hgnc:3433	ERCC1	CGI	2/1/22	NULL	0.3319450480417468	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.061737415	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.5585922471882393	BUCLIZINE	rxcui:59636	BUCLIZINE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.064944553	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.1250182648468916	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.063110182	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1785975212098452	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.089298761	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.08334551	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.05814803	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.087222045	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.2817943000126717	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1875273972703375	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1346350544504987	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
AR	hgnc:644	AR	CGI	2/1/22	NULL	0.014617949	Abiraterone	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.097236428	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.030598876	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P14784	hgnc:6009	IL2RB	TEND	1-Aug-11	NULL	1.346350544504987	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.061725319	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
ERCC2	hgnc:3434	ERCC2	CGI	2/1/22	NULL	0.1646008502686348	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P29460	hgnc:5970	IL12B	TEND	1-Aug-11	NULL	1.125164383622024	USTEKINUMAB	rxcui:847083	USTEKINUMAB	TRUE	FALSE	FALSE
UNIPROT:P23415	hgnc:4326	GLRA1	TEND	1-Aug-11	NULL	0.1539814405738841	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	0.8899605294185507	LOSARTAN	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.069240885	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.070010228	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.077789143	LORAZEPAM	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TEND	1-Aug-11	NULL	0.036951211	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
MYD88	hgnc:7562	MYD88	CGI	2/1/22	NULL	1.591141552596803	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
UNIPROT:P07225	hgnc:9456	PROS1	TEND	1-Aug-11	NULL	0.258658479	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P00740	hgnc:3551	F9	TEND	1-Aug-11	NULL	0.047647615	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.062833272	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
UNIPROT:Q9P0X4	hgnc:1396	CACNA1I	TEND	1-Aug-11	NULL	2.500365296937833	PARAMETHADIONE	rxcui:32894	PARAMETHADIONE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.1363835616511545	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.736088849	PHENMETRAZINE	rxcui:8133	PHENMETRAZINE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.1615620653405984	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	CGI	2/1/22	NULL	0.090821275	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
UNIPROT:P12931	hgnc:11283	SRC	TEND	1-Aug-11	NULL	0.1136529680426287	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P07333	hgnc:2433	CSF1R	TEND	1-Aug-11	NULL	0.038966732	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TEND	1-Aug-11	NULL	0.1205533268166455	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.074006584	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TEND	1-Aug-11	NULL	4.861821410712453	TOSITUMOMAB	rxcui:263010	TOSITUMOMAB	TRUE	FALSE	TRUE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.036463661	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.013836014	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	CGI	2/1/22	NULL	0.019138936	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TEND	1-Aug-11	NULL	1.325951293830669	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
UNIPROT:O43451	hgnc:7043	MGAM	TEND	1-Aug-11	NULL	4.773424657790408	VOGLIBOSE	ncit:C95221	VOGLIBOSE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.01992701	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	0.8078103267029924	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P30939	hgnc:5292	HTR1F	TEND	1-Aug-11	NULL	0.9546849315580819	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.057700738	PF-03084014	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	1.628144844517658	INCB54828	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
CD40L RECEPTOR	hgnc:11919	CD40	TTD	2020.06.01	NULL	2.187819634820604	ABBV-323	chembl:CHEMBL4298212	RAVAGALIMAB	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.064824285	CP-868596	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.007478127	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.061628722	Enzastaurin	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
LIVER AND ACTIVATION-REGULATED CHEMOKINE	hgnc:10619	CCL20	TTD	2020.06.01	NULL	52.50767123569449	GSK3050002	iuphar.ligand:9623	GSK3050002	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.2365210416022274	BETHANECHOL CHLORIDE	rxcui:47088	BETHANECHOL CHLORIDE	TRUE	FALSE	FALSE
B-CELL-SPECIFIC GLYCOPROTEIN B29	hgnc:1699	CD79B	TTD	2020.06.01	NULL	6.563458904461812	MGD010	chembl:CHEMBL4298039	MGD-010	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	Bb2121	ncit:C117729	IDECABTAGENE VICLEUCEL	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	1.029562181092049	Seribantumab	ncit:C78859	SERIBANTUMAB	FALSE	FALSE	TRUE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.175415383	DT-200	chembl:CHEMBL3545417	GLPG0492	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.1312691780892362	DCC-2618	rxcui:2369389	RIPRETINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.009659248	Mitomycin C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.4773424657790409	Revamilast	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	2.917092846427472	ADX-48621	ncit:C171677	DIPRAGLURANT	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	2.386712328895204	KLH-2109	rxcui:2621019	LINZAGOLIX	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.6105543166941221	BAY1179470	ncit:C107683	APRUTUMAB	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.074690855	PILOCARPINE HYDROCHLORIDE	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TISSUE FACTOR	hgnc:3541	F3	TTD	2020.06.01	NULL	3.500511415712966	MORAb-066	drugbank:DB17347	MORAB-066	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.052824619	LY3023414	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	2.625383561784724	BCI-838	chembl:CHEMBL4594408	MGS-0210	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	2.019525817	Tedalinab	ncit:C152534	TEDALINAB	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	2.128689374420047	LY-686017	ncit:C152707	TRADIPITANT	FALSE	FALSE	FALSE
PTH1R	hgnc:9608	PTH1R	ChEMBL	33	agonist	2.812910959055062	TERIPARATIDE	rxcui:32915	TERIPARATIDE	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 70	hgnc:5232	HSPA1A	TTD	2020.06.01	NULL	26.25383561784724	AG-858	drugbank:DB05502	AG-858	FALSE	FALSE	FALSE
ILEAL SODIUM/BILE ACID COTRANSPORTER	hgnc:10906	SLC10A2	TTD	2020.06.01	NULL	2.692701089009974	LUM001	iuphar.ligand:11708	MARALIXIBAT	FALSE	FALSE	FALSE
ISOCITRATE DEHYDROGENASE	hgnc:5382	IDH1	TTD	2020.06.01	NULL	0.064190307	AG-221	rxcui:1940332	ENASIDENIB	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1773907812016706	TROSPIUM CHLORIDE	rxcui:236778	TROSPIUM	TRUE	FALSE	FALSE
CHOLINEPHOSPHATE CYTIDYLYLTRANSFERASE	hgnc:8755	PCYT1B	TTD	2020.06.01	NULL	26.25383561784724	CT-2584	drugbank:DB13098	CT-2584	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.1	hgnc:1394	CACNA1G	TTD	2020.06.01	NULL	0.729273212	Penfluridol	rxcui:7974	PENFLURIDOL	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	0.042073455	NBQX	iuphar.ligand:4264	NBQX	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.2187819634820604	XR-5000	ncit:C2203	ACRIDINE CARBOXAMIDE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	XR-5000	ncit:C2203	ACRIDINE CARBOXAMIDE	FALSE	FALSE	FALSE
IMPA1	hgnc:6050	IMPA1	ChEMBL	33	inhibitor	5.250767124	LITHIUM CARBONATE	rxcui:42351	LITHIUM CARBONATE	TRUE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.082043236	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	0.1075976869583903	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	3.750547945	Desmoteplase	ncit:C87246	DESMOTEPLASE	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.027855529	Amlexanox	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.4782119420372905	Megestrol	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	Levobetaxolol	rxcui:353497	LEVOBETAXOLOL	FALSE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.1367387271762877	Phenyltoloxamine	rxcui:33408	PHENYLTOLOXAMINE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.3125456621172291	Piclamilast	ncit:C96718	PICLAMILAST	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	Carebastine	ncit:C77432	CAREBASTINE	FALSE	FALSE	FALSE
CHOLECYSTOKININ RECEPTOR TYPE A	hgnc:1570	CCKAR	TTD	2020.06.01	NULL	1.312691780892362	A-71378	iuphar.ligand:894	A-71378	FALSE	FALSE	FALSE
NEUTRAL ENDOPEPTIDASE	hgnc:7154	MME	TTD	2020.06.01	NULL	1.591141552596802	Gallopamil	rxcui:4648	GALLOPAMIL	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.06697407	DOLASTATIN-10	chembl:CHEMBL39541	DOLASTATIN-10	FALSE	FALSE	FALSE
PTGER1	hgnc:9593	PTGER1	ChEMBL	33	agonist	0.4892019059226195	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.021370644	Nitroglycerin	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	1.193356164447602	Naveglitazar	ncit:C75191	NAVEGLITAZAR	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1109316997937207	XL999	drugbank:DB05014	XL999	FALSE	FALSE	TRUE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	0.036821649	Ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.4449802647092754	LISINOPRIL	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	5.834185692854944	Org-24461	chembl:CHEMBL59821	CHEMBL:CHEMBL59821	FALSE	FALSE	FALSE
HISTAMINE H2 RECEPTOR	hgnc:5183	HRH2	TTD	2020.06.01	NULL	6.563458904461812	Nizatidine	rxcui:42319	NIZATIDINE	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.4449802647092754	Lisinopril	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.081030357	Romiplostim	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	3.088686543276147	XOMA 052	ncit:C97945	GEVOKIZUMAB	FALSE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	3.281729452230906	MK-5442	chembl:CHEMBL2105731	ENCALERET SULFATE	FALSE	FALSE	FALSE
MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN	hgnc:7467	MTTP	TTD	2020.06.01	NULL	8.751278539282415	Granotapide	ncit:C174852	GRANOTAPIDE	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.1491695205559502	Ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	CYCLIZINE LACTATE	rxcui:91071	CYCLIZINE LACTATE	TRUE	FALSE	FALSE
CHOLINEPHOSPHATE CYTIDYLYLTRANSFERASE	hgnc:8755	PCYT1B	TTD	2020.06.01	NULL	8.751278539282415	Sphingosine	drugbank:DB03203	SPHINGOSINE	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.7395446652914718	YN-968D1	ncit:C74012	RIVOCERANIB MESYLATE	FALSE	FALSE	FALSE
ALKALINE PHOSPHATASE TISSUE-NONSPECIFIC	hgnc:438	ALPL	TTD	2020.06.01	NULL	0.9907107780319716	Asfotase alfa	rxcui:1720259	ASFOTASE ALFA	TRUE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	2.561349816375341	PAC-14028	drugbank:DB12428	PAC-14028	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V6	hgnc:14006	TRPV6	TTD	2020.06.01	NULL	10.50153424713889	SOR-C13	drugbank:DB15366	SOR-C13	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	0.7955707762984014	TRIPTORELIN PAMOATE	rxcui:338529	TRIPTORELIN PAMOATE	TRUE	FALSE	FALSE
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	0.6908904109959803	RG6013	rxcui:1989794	EMICIZUMAB	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	1.009762908	MP-0112	chembl:CHEMBL4297684	ABICIPAR PEGOL	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	0.4039051633514961	KD025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
IMMUNE CHECKPOINT	hgnc:2203	COL4A2	TTD	2020.06.01	NULL	17.50255707856483	NLG919	ncit:C113793	NAVOXIMOD	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	0.1097721349875146	MK-3475	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	GRC-6211	chembl:CHEMBL3545107	GRC-6211	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.9546849315580819	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	0.1595977849109255	ASM-024	chembl:CHEMBL3707249	ASM-024	FALSE	FALSE	FALSE
E2 UBIQUITIN-CONJUGATING ENZYME T	hgnc:25009	UBE2T	TTD	2020.06.01	NULL	8.751278539282415	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	BI-754091	chembl:CHEMBL4802172	EZABENLIMAB	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	8.751278539282417	QUINETHAZONE	rxcui:59743	QUINETHAZONE	TRUE	FALSE	FALSE
P53-BINDING PROTEIN MDM4	hgnc:6974	MDM4	TTD	2020.06.01	NULL	2.917092846427472	ALRN-6924	ncit:C118669	SULANEMADLIN	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.069180068	Thiothixene	rxcui:10510	THIOTHIXENE	TRUE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	4.773424657790408	SC-49483	chembl:CHEMBL4297283	GLYCOVIR	FALSE	FALSE	FALSE
SLC12A3	hgnc:10912	SLC12A3	ChEMBL	33	inhibitor	0.9723642821424906	METHYCLOTHIAZIDE	rxcui:6860	METHYCLOTHIAZIDE	TRUE	FALSE	FALSE
G-PROTEIN COUPLED BILE ACID RECEPTOR 1	hgnc:19680	GPBAR1	TTD	2020.06.01	NULL	8.751278539282415	Sodium taurocholate	chembl:CHEMBL443728	SODIUM TAUROCHOLATE	FALSE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	1.567393171214761	TAK-901	drugbank:DB12756	TAK-901	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1226814748497534	Clomiphene Citrate	rxcui:142431	CLOMIPHENE CITRATE	TRUE	FALSE	FALSE
SSTR1	hgnc:11330	SSTR1	ChEMBL	33	agonist	1.093909817410302	PASIREOTIDE DIASPARTATE	rxcui:1364104	PASIREOTIDE DIASPARTATE	TRUE	FALSE	FALSE
DUFFY ANTIGEN CHEMOKINE RECEPTOR	hgnc:4035	ACKR1	TTD	2020.06.01	NULL	1.640864726115453	Chloroquine	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.4930297768609811	Nalbuphine	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.095468493	Paroxetine	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.3241214273808302	Modafinil	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
E3 UBIQUITIN-PROTEIN LIGASE COP1	hgnc:17440	COP1	TTD	2020.06.01	NULL	0.8078103267029924	Quinine	rxcui:9071	QUININE	TRUE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	6.563458904461812	NIZATIDINE	rxcui:42319	NIZATIDINE	TRUE	FALSE	FALSE
TRYPTOPHAN HYDROXYLASE	hgnc:12008	TPH1	TTD	2020.06.01	NULL	6.563458904461812	Telotristat ethyl	rxcui:1872441	TELOTRISTAT ETHYL	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.4145342465975881	Ropivacaine	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	0.7001022831425933	KB-003	iuphar.ligand:8935	LENZILUMAB	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.1400204566285186	Topotecan	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.027870314	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-10	hgnc:13800	CHRNA10	TTD	2020.06.01	NULL	10.50153424713889	ACV-1	drugbank:DB05724	ALPHA-CONOTOXIN VC 1.1	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA 2	hgnc:4572	GRIA2	TTD	2020.06.01	NULL	1.591141552596803	Paliroden	ncit:C82298	PALIRODEN	FALSE	FALSE	FALSE
GLUCOSE-DEPENDENT INSULINOTROPIC RECEPTOR	hgnc:19060	GPR119	TTD	2020.06.01	NULL	8.751278539282415	GSK1292263	chembl:CHEMBL3187503	GSK-1292263	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	1.009762908	LY2886721	iuphar.ligand:6475	LY2886721	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.07767407	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1008469998124734	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.028498058	Celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.077827576	Cabergoline	rxcui:47579	CABERGOLINE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	1.432027397337122	Etoricoxib	rxcui:307296	ETORICOXIB	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Levocabastine	rxcui:28627	LEVOCABASTINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.1356787370431382	Indacaterol	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.5357925636295356	Nadroparin calcium	ncit:C61320	NADROPARIN CALCIUM	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3040984820600068	OPC-34712	rxcui:1658314	BREXPIPRAZOLE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.094099769	Oxcarbazepine	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.075496292	DULOXETINE HYDROCHLORIDE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Promestriene	rxcui:34625	PROMESTRIENE	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Tripelennamine	rxcui:10847	TRIPELENNAMINE	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.3062196950280639	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	0.2019525816757481	JWH-015	iuphar.ligand:5558	JWH015	FALSE	FALSE	FALSE
NEUROTROPHIC TYROSINE KINASE ROR1	hgnc:10256	ROR1	TTD	2020.06.01	NULL	52.50767123569449	Cirmtuzumab	chembl:CHEMBL4297728	CIRMTUZUMAB	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1635752997996713	PROTRIPTYLINE HYDROCHLORIDE	rxcui:203199	PROTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.2001054544043235	ABT-263	ncit:C64776	NAVITOCLAX	FALSE	FALSE	TRUE
PURINE NUCLEOSIDE PHOSPHORYLASE	hgnc:7892	PNP	TTD	2020.06.01	NULL	8.751278539282415	Forodesine	ncit:C65755	FORODESINE	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3 EPSILON	hgnc:1674	CD3E	TTD	2020.06.01	NULL	0.9723642821424906	Ertumaxomab	ncit:C2658	ERTUMAXOMAB	FALSE	FALSE	FALSE
PROTEINASE ACTIVATED RECEPTOR 1	hgnc:3537	F2R	TTD	2020.06.01	NULL	2.019525817	E5555	ncit:C169794	ATOPAXAR	FALSE	FALSE	FALSE
ENDOTHELIN B RECEPTOR	hgnc:3180	EDNRB	TTD	2020.06.01	NULL	2.500365296937833	SPI-1620	ncit:C74027	SOVATELTIDE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.1090501998664475	MESTRANOL	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
INTEGRIN BETA-7	hgnc:6162	ITGB7	TTD	2020.06.01	NULL	17.50255707856483	Rhumab Beta7	ncit:C97944	ETROLIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1388	hgnc:2349	ATF6B	GuideToPharmacology	2024.1	modulator	13.12691780892362	IUPHAR.LIGAND:9141	iuphar.ligand:9141	PKUMDL_MH_1001	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.041150213	IUPHAR.LIGAND:31	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:19	iuphar.ligand:19	LY293284	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:30	iuphar.ligand:30	U92016A	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:24	iuphar.ligand:24	S-14506	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.8078103267029922	BUPIVACAINE HYDROCHLORIDE	rxcui:267396	BUPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.013313304	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:78	iuphar.ligand:78	SDZ-216525	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.062509132	IUPHAR.LIGAND:60	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.032899543	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:117	ncit:C77255	ALNIDITAN	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.056826484	IUPHAR.LIGAND:31	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.093098708	IUPHAR.LIGAND:125	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.048573239	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.4907258993990139	PSEUDOEPHEDRINE SULFATE	rxcui:91169	PSEUDOEPHEDRINE SULFATE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1241316104862754	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.034727296	IUPHAR.LIGAND:130	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.013890918	IUPHAR.LIGAND:214	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
F5	hgnc:3542	F5	ChEMBL	33	inhibitor	0.2949869170544634	DROTRECOGIN ALFA (ACTIVATED)	ncit:C80267	DROTRECOGIN ALFA (ACTIVATED)	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.019844169	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:219	iuphar.ligand:219	[3H]LSD	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.007272531	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.077217164	IUPHAR.LIGAND:145	iuphar.ligand:145	5-MEO-DMT	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.096521454	IUPHAR.LIGAND:154	iuphar.ligand:154	(+)-LSD	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.080905503	IUPHAR.LIGAND:39	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:71	iuphar.ligand:71	MPDT	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.059330702	IUPHAR.LIGAND:201	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.043866058	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.1842374429322614	IUPHAR.LIGAND:71	iuphar.ligand:71	MPDT	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.9211872146613069	IUPHAR.LIGAND:3929	iuphar.ligand:3929	E55888	FALSE	FALSE	FALSE
NCBIGENE:1385	hgnc:2345	CREB1	GuideToPharmacology	2024.1	inhibitor	0.5303805175322677	IUPHAR.LIGAND:5297	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
F8	hgnc:3546	F8	ChEMBL	33	inhibitor	1.544343271638073	DROTRECOGIN ALFA (ACTIVATED)	ncit:C80267	DROTRECOGIN ALFA (ACTIVATED)	TRUE	FALSE	FALSE
NCBIGENE:768	hgnc:1383	CA9	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12787	ncit:C111994	ENCEQUIDAR	FALSE	FALSE	FALSE
NCBIGENE:1784	ncbigene:1784	DNCM	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8121	iuphar.ligand:8121	ML347	FALSE	FALSE	FALSE
NCBIGENE:1231	hgnc:1603	CCR2	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:5130	iuphar.ligand:5130	A134974	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.09814518	IMIPRAMINE HYDROCHLORIDE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1677	hgnc:2773	DFFB	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8553	iuphar.ligand:8553	COMPOUND 15C [PMID: 21536437]	FALSE	FALSE	FALSE
NCBIGENE:1279	hgnc:2199	COL1AR	GuideToPharmacology	2024.1	activator	26.25383561784724	IUPHAR.LIGAND:10214	iuphar.ligand:10214	FD1	FALSE	FALSE	FALSE
NCBIGENE:3068	hgnc:4856	HDGF	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12309	iuphar.ligand:12309	TDI-11861	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	ChEMBL	33	inhibitor	0.108711535	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2466	hgnc:3863	FRA17B	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8841	iuphar.ligand:8841	4-ACRYLOYLPHENOL	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:12216	iuphar.ligand:12216	MS15	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.1238388472539964	IUPHAR.LIGAND:73	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.052142673	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.1526385791735305	IUPHAR.LIGAND:6360	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:6501	ncit:C72915	FASIDOTRIL	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:6575	rxcui:36908	SPIRAPRIL	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:6571	rxcui:30131	MOEXIPRIL	TRUE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:6314	iuphar.ligand:6314	ML233	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.08178765	NORTRIPTYLINE HYDROCHLORIDE	rxcui:203130	NORTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:8524	iuphar.ligand:8524	ELABELA/TODDLER-32	FALSE	FALSE	FALSE
NCBIGENE:696	hgnc:1135	BTN1A1	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:4285	drugbank:DB07810	PHLORETIN	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:6186	iuphar.ligand:6186	MM54	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	2.341819737097098	DABRAFENIB MESYLATE	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
NCBIGENE:2951	hgnc:4640	GSTP1P1	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:9642	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
NCBIGENE:1245	ncbigene:1245	CMR1A	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9017	iuphar.ligand:9017	COMPOUND 9 [PMID: 23472952]	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	0.021905578	IUPHAR.LIGAND:4139	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.201178817	IUPHAR.LIGAND:5622	iuphar.ligand:5622	MRS5151	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:5619	iuphar.ligand:5619	PSB-10	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.201178817	IUPHAR.LIGAND:4252	rxcui:6694	MEFLOQUINE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:429	iuphar.ligand:429	MRS1088	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:395	iuphar.ligand:395	MRS1065	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:459	iuphar.ligand:459	MRE 3008F20	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:402	iuphar.ligand:402	MRS928	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.018430211	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:3281	ncit:C96199	DERENOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:382	iuphar.ligand:382	AS70	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.1810609352954983	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.061992528	IUPHAR.LIGAND:5617	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:5607	iuphar.ligand:5607	LUF5981	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5614	ncit:C76394	PRELADENANT	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.049210563	IUPHAR.LIGAND:384	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.090219366	IUPHAR.LIGAND:409	rxcui:1536070	FLAVONE	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.5000730593875666	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:463	ncit:C1465	DEXNIGULDIPINE	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.5413161983061289	IUPHAR.LIGAND:460	iuphar.ligand:460	MPC-MECA	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11647	ncit:C129693	GARTISERTIB	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8041	iuphar.ligand:8041	KU-60019	FALSE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	0.035719504	IUPHAR.LIGAND:7950	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:8466	iuphar.ligand:8466	COMPOUND 10 [PMID: 19402633]	FALSE	FALSE	FALSE
NCBIGENE:2901	hgnc:4583	GRIK5	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9142	iuphar.ligand:9142	PF-8380	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1715936968486748	IUPHAR.LIGAND:10387	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
NCBIGENE:2901	hgnc:4583	GRIK5	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9791	iuphar.ligand:9791	BI-2545	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.021155387	IUPHAR.LIGAND:5718	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.7759754369807069	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:1938	hgnc:3214	EEF2	GuideToPharmacology	2024.1	inhibitor	0.2651902587661338	IUPHAR.LIGAND:12661	iuphar.ligand:12661	BI-847325	FALSE	FALSE	TRUE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:618	iuphar.ligand:618	RANATENSIN	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:3788	iuphar.ligand:3788	[125I]GRP (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:3840	iuphar.ligand:3840	[D-PHE6, LEU13, CPA14,&PSI;13-14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6184	iuphar.ligand:6184	[D-ARG1,D-TRP7,9,LEU11]SUBSTANCE P	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10394	iuphar.ligand:10394	COMPOUND 3L [PMID: 30637955]	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:6540	iuphar.ligand:6540	EXAMPLE 98 [WO2011020806]	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:7804	iuphar.ligand:7804	AZ3971	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.039068208	IUPHAR.LIGAND:63	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:12580	iuphar.ligand:12580	NDD-825	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.042073455	IUPHAR.LIGAND:564	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.5645986154375752	IUPHAR.LIGAND:567	iuphar.ligand:567	BRL 37344	FALSE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:3325	iuphar.ligand:3325	U75302	FALSE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6157	iuphar.ligand:6157	ONO-4057	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:12239	iuphar.ligand:12239	JNJ-64264681	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:9815	iuphar.ligand:9815	CCT196969	FALSE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:9269	iuphar.ligand:9269	BMX-IN-1	FALSE	FALSE	FALSE
NCBIGENE:1786	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:8121	iuphar.ligand:8121	ML347	FALSE	FALSE	FALSE
NCBIGENE:2731	hgnc:4313	GLDC	GuideToPharmacology	2024.1	NULL	8.751278539282415	IUPHAR.LIGAND:9523	iuphar.ligand:9523	OF-1	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.1250182648468916	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:2730	hgnc:4312	GCLM	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:7809	iuphar.ligand:7809	COMPOUND 1 [PMID: 25408830]	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:12096	ncit:C175553	TINLORAFENIB	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:10387	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
NCBIGENE:2721	ncbigene:2721	GLC#	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8233	iuphar.ligand:8233	GSK2801	FALSE	FALSE	FALSE
NCBIGENE:2599	hgnc:1375	CA4	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:10433	iuphar.ligand:10433	COMPOUND 5A [PMID: 31287314]	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:9476	iuphar.ligand:9476	SB-423562	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.2465148884304905	NALMEFENE HYDROCHLORIDE	rxcui:236069	NALMEFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1620	hgnc:2687	BRINP1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9034	iuphar.ligand:9034	VRT-043198	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:9475	iuphar.ligand:9475	ATF936	FALSE	FALSE	FALSE
NCBIGENE:2351	ncbigene:2351	FOLR2L	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:11701	iuphar.ligand:11701	UAWJ9-36-3	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:7862	ncit:C66512	RELACATIB	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9705	iuphar.ligand:9705	AM2201	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:11149	iuphar.ligand:11149	GW405833	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:9231	ncit:C81420	TARANABANT	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.07614901	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:757	iuphar.ligand:757	CCL4	FALSE	FALSE	FALSE
NCBIGENE:67	hgnc:140	ACTBP7	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:3649	iuphar.ligand:3649	CCL28	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:762	iuphar.ligand:762	[125I]CCL2 (HUMAN)	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
NCBIGENE:3126	hgnc:4952	HLA-DRB4	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:11326	iuphar.ligand:11326	ATIBUCLIMAB	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:803	iuphar.ligand:803	[3H]MARAVIROC	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:801	ncit:C166464	CENICRIVIROC	FALSE	FALSE	FALSE
NCBIGENE:65	ncbigene:65	ACTBP5	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:772	iuphar.ligand:772	CCL8	FALSE	FALSE	FALSE
NCBIGENE:2764	hgnc:4373	GMFB	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:7992	iuphar.ligand:7992	INEBILIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:9833	iuphar.ligand:9833	BSAB (CD89-CD20)	FALSE	FALSE	FALSE
NCBIGENE:65	ncbigene:65	ACTBP5	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:768	iuphar.ligand:768	VMIP-II	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:10106	iuphar.ligand:10106	CCR5 ANTAGONIST 34	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.1030370314672184	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:64	hgnc:137	ACTBP4	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:810	iuphar.ligand:810	CCL19	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:6781	rxcui:263010	TOSITUMOMAB	TRUE	FALSE	TRUE
NCBIGENE:2601	hgnc:4153	GAPDHP60	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:9434	iuphar.ligand:9434	VADASTUXIMAB TALIRINE	FALSE	FALSE	FALSE
NCBIGENE:1993	hgnc:3313	ELAVL2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8162	iuphar.ligand:8162	ML315	FALSE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11746	iuphar.ligand:11746	MONZOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:9365	iuphar.ligand:9365	CHIR-124	FALSE	FALSE	FALSE
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	blocker	6.563458904461812	IUPHAR.LIGAND:4199	iuphar.ligand:4199	GATX2	FALSE	FALSE	FALSE
NCBIGENE:3248	hgnc:5154	HPGD	GuideToPharmacology	2024.1	inhibitor	0.1058622403945453	IUPHAR.LIGAND:8400	ncit:C75251	ANACETRAPIB	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	ChEMBL	33	inhibitor	0.2282942227638891	LITHIUM CARBONATE	rxcui:42351	LITHIUM CARBONATE	TRUE	FALSE	FALSE
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	activator	0.6563458904461813	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:395	hgnc:676	ARHGAP6	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:2313	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NCBIGENE:1255	ncbigene:1255	CNA1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:7030	iuphar.ligand:7030	BMS PYRAZOLE INHIBITOR 7F	FALSE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7408	ncit:C77994	ERIBAXABAN	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:8942	ncit:C101519	EDICOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.009809018	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	0.4000584475100533	PONATINIB HYDROCHLORIDE	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:917	iuphar.ligand:917	[125I]UROCORTIN 1 (MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:714	hgnc:1245	C1QC	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:714	hgnc:1245	C1QC	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:683	iuphar.ligand:683	ADRENOMEDULLIN	FALSE	FALSE	FALSE
NCBIGENE:721	hgnc:1324	C4B	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:722	hgnc:1325	C4BPA	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.0296486	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:719	hgnc:1319	C3AR1	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:730	hgnc:1346	C7	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:729	hgnc:1339	C6	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:732	hgnc:1353	C8B	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:733	hgnc:1354	C8G	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:730	hgnc:1346	C7	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:821	iuphar.ligand:821	CXCL8	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	inhibitor	0.008043455	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:836	iuphar.ligand:836	CXCL11	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.300043836	IUPHAR.LIGAND:768	iuphar.ligand:768	VMIP-II	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1060761035064535	IUPHAR.LIGAND:7938	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1328	hgnc:2621	CYP2C19	GuideToPharmacology	2024.1	inhibitor	0.027121731	IUPHAR.LIGAND:8777	iuphar.ligand:8777	COMPOUND 51 [CROSIGNANI ET AL., 2011]	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	agonist	0.9211872146613068	IUPHAR.LIGAND:3353	iuphar.ligand:3353	LTD4	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:10346	iuphar.ligand:10346	MK-571	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3381	iuphar.ligand:3381	BAYU9773	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.1428780169678761	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10481	iuphar.ligand:10481	COMPOUND 1 [PMID: 31477924]	FALSE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9906	ncit:C87623	TENELIGLIPTIN	FALSE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12238	iuphar.ligand:12238	ICED-2	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9906	ncit:C87623	TENELIGLIPTIN	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.1121958787087489	IUPHAR.LIGAND:5820	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1363835616511545	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.050488145	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:1899	iuphar.ligand:1899	[3H]BWA868C	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:9277	iuphar.ligand:9277	TIMAPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:10180	ncit:C152348	SETIPIPRANT	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	IBUPROFEN LYSINE	rxcui:36761	IBUPROFEN LYSINE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:945	iuphar.ligand:945	[125I]SCH23982	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.046673486	IUPHAR.LIGAND:948	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:8441	iuphar.ligand:8441	A-381393	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	0.3804903712731485	IUPHAR.LIGAND:80	iuphar.ligand:3251	[3H]WAY100635	FALSE	FALSE	FALSE
NCBIGENE:1232	hgnc:1604	CCR3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12355	iuphar.ligand:12355	COMPOUND 49 [PMID: 36529947]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:10477	iuphar.ligand:10477	FIRMONERTINIB	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.1458546423213736	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:11941	iuphar.ligand:11941	COMPOUND 17B [PMID: 35286086]	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12951	ncit:C175747	BEFOTERTINIB	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:6068	iuphar.ligand:6068	MF266-1	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1925	iuphar.ligand:1925	11-DEOXY-PGE1	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:5857	iuphar.ligand:5857	CJ-042794	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	ChEMBL	33	inhibitor	0.3337351985319565	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:1931	iuphar.ligand:1931	ONO-AE-248	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	inhibitor	0.3201687270469177	IUPHAR.LIGAND:9283	iuphar.ligand:9283	TG6-129	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.3182283105193606	IUPHAR.LIGAND:2817	drugbank:DB04468	AFIMOXIFENE	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.3182283105193606	IUPHAR.LIGAND:2817	drugbank:DB04468	AFIMOXIFENE	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.1446492320542548	IUPHAR.LIGAND:2818	rxcui:4103	ESTRONE	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2821	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.018942161	IUPHAR.LIGAND:2801	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:2827	iuphar.ligand:2827	HPTE	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	IBUPROFEN LYSINE	rxcui:36761	IBUPROFEN LYSINE	TRUE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:2743	iuphar.ligand:2743	GW4064	FALSE	FALSE	FALSE
NCBIGENE:1718	hgnc:2859	DHCR24	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:7447	rxcui:1248798	PEGINESATIDE	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	blocker	0.4605936073306534	IUPHAR.LIGAND:4369	iuphar.ligand:4369	[35S]TBPS	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.3201687270469177	IUPHAR.LIGAND:4326	iuphar.ligand:4326	TP003	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	INDOMETHACIN SODIUM	rxcui:1294612	INDOMETHACIN SODIUM	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.1600843635234588	IUPHAR.LIGAND:4297	iuphar.ligand:4297	RO19-4603	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:4346	iuphar.ligand:4346	ZK93423	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.086219493	IUPHAR.LIGAND:4108	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	0.08334551	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.06466462	IUPHAR.LIGAND:10773	rxcui:2265690	CENOBAMATE	TRUE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:5357	iuphar.ligand:5357	GALANIN(2-11)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6105	iuphar.ligand:6105	GAL-B2	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6075	iuphar.ligand:6075	J18 (GALANIN ANALOGUE)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6106	iuphar.ligand:6106	GAL-B2-DPEG24	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.4953553890159858	IUPHAR.LIGAND:6107	iuphar.ligand:6107	GAL-B5	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6112	iuphar.ligand:6112	GAL-B2-C10	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:6111	iuphar.ligand:6111	GAL-B2-C8	FALSE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:6512	iuphar.ligand:6512	(R)-EF-1520	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:4138	iuphar.ligand:4138	ARGIOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:250	hgnc:439	ALPP	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:10685	ncit:C171811	APRAGLUTIDE	FALSE	FALSE	FALSE
NCBIGENE:250	hgnc:439	ALPP	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:1140	iuphar.ligand:1140	GLUCAGON-LIKE PEPTIDE 2	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	blocker	0.4688184931758437	IUPHAR.LIGAND:4138	iuphar.ligand:4138	ARGIOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	blocker	0.4167275494896388	IUPHAR.LIGAND:4229	iuphar.ligand:4229	JORO SPIDER TOXIN	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:4249	iuphar.ligand:4249	LY404187	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:4162	iuphar.ligand:4162	CONCANAVALIN A	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.6563458904461813	IUPHAR.LIGAND:4068	iuphar.ligand:4068	(RS)-(TETRAZOL-5-YL)GLYCINE	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4082	iuphar.ligand:4082	[3H]CPP	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	blocker	0.1790542923638346	IUPHAR.LIGAND:4233	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:4086	iuphar.ligand:4086	[3H]L689560	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.2117244807890907	IUPHAR.LIGAND:4282	ncit:C738	PHENCYCLIDINE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:4082	iuphar.ligand:4082	[3H]CPP	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4155	ncit:C152322	SELFOTEL	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4155	ncit:C152322	SELFOTEL	FALSE	FALSE	FALSE
NCBIGENE:1272	hgnc:2171	CNTN1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:5267	iuphar.ligand:5267	S-ALLYLGLYCINE	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:4086	iuphar.ligand:4086	[3H]L689560	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	inhibitor	0.577007376	IUPHAR.LIGAND:731	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:2360	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:4289	iuphar.ligand:4289	PMBA	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.098884503	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.046840028	IUPHAR.LIGAND:5989	drugbank:DB02052	INDIRUBIN-3'-MONOXIME	FALSE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:11412	ncit:C156792	ELRAGLUSIB	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	NULL	3.281729452230906	IUPHAR.LIGAND:4584	iuphar.ligand:4584	[35S]ACPPB	FALSE	FALSE	FALSE
NCBIGENE:311	hgnc:535	ANXA11	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:11197	iuphar.ligand:11197	COMPOUND 2 [PMID: 31932225]	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:8981	iuphar.ligand:8981	CONESSINE	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:1226	iuphar.ligand:1226	IMPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5750	iuphar.ligand:5750	COMPOUND 20F [PMID: 21536438]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:3621	iuphar.ligand:3621	SEA	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5738	iuphar.ligand:5738	COMPOUND 3J [PMID: 21444206]	FALSE	FALSE	FALSE
NCBIGENE:99	hgnc:4487	GPR32	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:1034	iuphar.ligand:1034	LXA4	FALSE	FALSE	FALSE
NCBIGENE:105	hgnc:227	ADARB2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:7800	iuphar.ligand:7800	COMPOUND 1 [PMID: 24900608]	FALSE	FALSE	FALSE
NCBIGENE:101	hgnc:215	ADAM8	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12947	iuphar.ligand:12947	YL-365	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:5846	iuphar.ligand:5846	6-N-OCTYLAMINOURACIL	FALSE	FALSE	FALSE
NCBIGENE:114	hgnc:239	ADCY8	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:10570	iuphar.ligand:10570	OSTN (115-133)	FALSE	FALSE	FALSE
NCBIGENE:150	hgnc:281	ADRA2A	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:7040	iuphar.ligand:7040	CGEN-857	FALSE	FALSE	FALSE
NCBIGENE:2625	hgnc:4172	GATA3	GuideToPharmacology	2024.1	inhibitor	0.072725306	IUPHAR.LIGAND:6842	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	0.4487835148349958	IUPHAR.LIGAND:7113	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
NCBIGENE:2443	hgnc:3841	FRA11F	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10511	ncit:C169828	CAROTEGRAST	FALSE	FALSE	FALSE
NCBIGENE:2451	hgnc:3848	FRA12D	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9720	iuphar.ligand:9720	BIRT 377	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12445	iuphar.ligand:12445	LUPULONE	FALSE	FALSE	FALSE
NCBIGENE:674	ncbigene:674	BRAFPS1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:12470	iuphar.ligand:12470	CYCLAMATE	FALSE	FALSE	FALSE
NCBIGENE:674	ncbigene:674	BRAFPS1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:5432	rxcui:9509	SACCHARIN	TRUE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:12499	iuphar.ligand:12499	LACTUCOPICRIN	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:7954	iuphar.ligand:7954	BMS-911543	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:10459	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.09869863	IUPHAR.LIGAND:11304	ncit:C177760	NEZULCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:11613	ncit:C180657	ROPSACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.036362653	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:12318	iuphar.ligand:12318	GDC-0214	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:9193	iuphar.ligand:9193	ZYKLOPHIN	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:8942	ncit:C101519	EDICOTINIB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:9105	iuphar.ligand:9105	PLX5622	FALSE	FALSE	FALSE
NCBIGENE:521	hgnc:846	ATP5ME	GuideToPharmacology	2024.1	activator	0.7501095890813501	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	0.4167275494896389	IUPHAR.LIGAND:710	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:943	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	0.062808219	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:549	hgnc:890	AUH	GuideToPharmacology	2024.1	blocker	52.50767123569449	IUPHAR.LIGAND:2549	iuphar.ligand:2549	SHK TOXIN	FALSE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11404	iuphar.ligand:11404	COMPOUND 23A [PMID: 33417443]	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:1338	iuphar.ligand:1338	THIQ	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:1328	iuphar.ligand:1328	HS024	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.024920584	IUPHAR.LIGAND:7950	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:10649	iuphar.ligand:10649	COMPOUND 7 [PMID: 31955578]	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:9571	iuphar.ligand:9571	ECF309	FALSE	FALSE	FALSE
NCBIGENE:2381	hgnc:3893	FRA2I	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8828	iuphar.ligand:8828	COMPOUND 7B [PMID: 17583500]	FALSE	FALSE	FALSE
NCBIGENE:2988	hgnc:4694	GUK2	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:9805	iuphar.ligand:9805	IMAPRELIMAB	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12093	iuphar.ligand:12093	ZANZALINTINIB	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6409	iuphar.ligand:6409	CTEP	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6429	iuphar.ligand:6429	COMPOUND 16M [PMID: 19931453]	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1406	iuphar.ligand:1406	(R,S)-4-PPG	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1411	ncit:C169894	DEXFOSFOSERINE	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1393	iuphar.ligand:1393	EGLUMEGAD	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	0.145450613	IUPHAR.LIGAND:2523	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:9974	iuphar.ligand:9974	MK-8353	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:11095	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
NCBIGENE:2066	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:9380	iuphar.ligand:9380	BIX02189	FALSE	FALSE	FALSE
NCBIGENE:2072	hgnc:3436	ERCC4	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11506	iuphar.ligand:11506	GDC-0134	FALSE	FALSE	FALSE
NCBIGENE:2074	hgnc:3438	ERCC6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8174	iuphar.ligand:8174	COMPOUND 31 [PMID: 23374866]	FALSE	FALSE	FALSE
NCBIGENE:2074	hgnc:3438	ERCC6	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
NCBIGENE:2086	hgnc:3454	ERV3-1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
NCBIGENE:1638	hgnc:2709	DCT	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10887	iuphar.ligand:10887	(R)-ND-336	FALSE	FALSE	FALSE
NCBIGENE:990	hgnc:1744	CDC6	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8818	iuphar.ligand:8818	7ACC2	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:1457	iuphar.ligand:1457	MOTILIN	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1445	iuphar.ligand:1445	EM-523	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.050488145	IUPHAR.LIGAND:286	ncit:C81044	ACECLIDINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.055271233	IUPHAR.LIGAND:328	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.040235763	IUPHAR.LIGAND:1357	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:7781	iuphar.ligand:7781	ISOAMYL-AGOMELATINE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1604	iuphar.ligand:1604	(-)-CYCLAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:1633	ncit:C80570	QUADAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:1553	hgnc:2608	CYP2A13	GuideToPharmacology	2024.1	activator	2.625383561784725	IUPHAR.LIGAND:2351	iuphar.ligand:2351	CALMODULIN	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.28382525	IUPHAR.LIGAND:4797	rxcui:6664	MAZINDOL	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.2365210416022274	IUPHAR.LIGAND:7477	rxcui:787390	TAPENTADOL	TRUE	FALSE	FALSE
NCBIGENE:1251	hgnc:7872	NOS1	GuideToPharmacology	2024.1	inhibitor	0.7395446652914718	IUPHAR.LIGAND:5127	iuphar.ligand:5127	7NI	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:12392	iuphar.ligand:12392	ZIDESAMTINIB	FALSE	FALSE	FALSE
NCBIGENE:1819	hgnc:3030	DRG2	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:10257	iuphar.ligand:10257	GR-389988	FALSE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:6492	ncit:C171870	CANDOXATRIL	TRUE	FALSE	FALSE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:6501	ncit:C72915	FASIDOTRIL	FALSE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3984	iuphar.ligand:3984	WAGLERIN-1	FALSE	FALSE	FALSE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:4001	rxcui:7883	PANCURONIUM	TRUE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:3973	iuphar.ligand:3973	&ALPHA;-CONOTOXIN AUIB	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3974	iuphar.ligand:3974	[3H]A-585539	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2091	iuphar.ligand:2091	NEUROPEPTIDE K	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:11492	iuphar.ligand:11492	CPN-223	FALSE	FALSE	FALSE
NCBIGENE:299	hgnc:16454	NMUR2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:1475	iuphar.ligand:1475	[125I]NEUROMEDIN U-23 (RAT)	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1482	iuphar.ligand:1482	Y-RFRP-3	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:4020	iuphar.ligand:4020	AC263093	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:12606	iuphar.ligand:12606	(R)-YNT-3708	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1699	iuphar.ligand:1699	OREXIN-B	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:12606	iuphar.ligand:12606	(R)-YNT-3708	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:11447	iuphar.ligand:11447	COMPOUND 1 [PMID: 33547286]	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:9302	rxcui:2272403	LEMBOREXANT	TRUE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2890	rxcui:1547099	SUVOREXANT	TRUE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:9467	iuphar.ligand:9467	[3H]EMPA	FALSE	FALSE	FALSE
NCBIGENE:2136	hgnc:16059	PAK4	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:8939	iuphar.ligand:8939	FRAX597	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:4298	iuphar.ligand:4298	RO3	FALSE	FALSE	FALSE
NCBIGENE:484	hgnc:807	ATP1B3P1	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:9062	iuphar.ligand:9062	PF-04905428	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:5905	iuphar.ligand:5905	COMPOUND 4 [PMID: 22984835]	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:6200	iuphar.ligand:6200	N4-PHENYLETHOXYCYTIDINE-5'-TRIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1854	iuphar.ligand:1854	SCH 40338	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.04464938	IUPHAR.LIGAND:8918	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:10633	iuphar.ligand:10633	GSK2292767	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:10098	ncit:C113434	PARSACLISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.039068208	IUPHAR.LIGAND:6004	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:6024	iuphar.ligand:6024	PI 3-KG INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.070197421	IUPHAR.LIGAND:7965	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
NCBIGENE:1300	hgnc:2185	COL10A1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11865	iuphar.ligand:11865	ENSIFENTRINE	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7320	rxcui:306674	VARDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:5275	iuphar.ligand:5275	T0156	FALSE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6066	iuphar.ligand:6066	PKR-A	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1868	iuphar.ligand:1868	PROKINETICIN-2&BETA;	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:6433	iuphar.ligand:6433	TRIAZINE COMPOUND PC10	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.058341857	IUPHAR.LIGAND:5705	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
NCBIGENE:2864	hgnc:4498	FFAR1	GuideToPharmacology	2024.1	inhibitor	0.085239726	IUPHAR.LIGAND:7519	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11349	rxcui:21090	CICLOPIROX	TRUE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10671	iuphar.ligand:10671	MC2050	FALSE	FALSE	FALSE
NCBIGENE:1486	hgnc:2496	CTBS	GuideToPharmacology	2024.1	activator	2.500365296937833	IUPHAR.LIGAND:10066	iuphar.ligand:10066	RASGRP ACTIVATOR 1	FALSE	FALSE	FALSE
NCBIGENE:1491	hgnc:2501	CTH	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:8012	iuphar.ligand:8012	PIK-75	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9766	ncit:C120036	PEPOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:9733	ncit:C123882	TRODUSQUEMINE	FALSE	FALSE	FALSE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9732	iuphar.ligand:9732	HPN	FALSE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:2814	iuphar.ligand:2814	LG100754	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:2654	iuphar.ligand:2654	CD2665	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9356	iuphar.ligand:9356	GSK429286A	FALSE	FALSE	FALSE
NCBIGENE:1528	hgnc:2570	CYB5A	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8039	iuphar.ligand:8039	BIX 02565	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:11907	iuphar.ligand:11907	WNN0109-C011	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:11907	iuphar.ligand:11907	WNN0109-C011	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6522	iuphar.ligand:6522	EUROPIUM-LABELLED MOUSE INSL5	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1998	iuphar.ligand:1998	R3/I5	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.300043836	IUPHAR.LIGAND:9331	rxcui:2668045	ETRASIMOD	TRUE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	activator	0.1640864726115453	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:12570	iuphar.ligand:12570	ST-1505	FALSE	FALSE	FALSE
NCBIGENE:2708	hgnc:10886	SIRT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8778	iuphar.ligand:8778	COMPOUND 17 [PMID: 23570514]	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:6677	iuphar.ligand:6677	(+)-SKF 10.047	FALSE	FALSE	FALSE
NCBIGENE:2707	hgnc:4285	GJB3	GuideToPharmacology	2024.1	activator	8.751278539282415	IUPHAR.LIGAND:7703	iuphar.ligand:7703	SRT1720	FALSE	FALSE	FALSE
NCBIGENE:2712	hgnc:4291	GK2	GuideToPharmacology	2024.1	modulator	26.25383561784724	IUPHAR.LIGAND:10123	iuphar.ligand:10123	MDL-800	FALSE	FALSE	FALSE
NCBIGENE:2199	hgnc:3601	FBLN2	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:12157	ncit:C175865	TILPISERTIB	FALSE	FALSE	FALSE
NCBIGENE:959	hgnc:11935	CD40LG	GuideToPharmacology	2024.1	inhibitor	0.020811602	IUPHAR.LIGAND:1024	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
NCBIGENE:960	hgnc:1681	CD44	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:6529	iuphar.ligand:6529	264W94	FALSE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:4594	rxcui:1486966	DAPAGLIFLOZIN PROPANEDIOL	TRUE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11146	iuphar.ligand:11146	COMPOUND 59 [PMID: 30889352]	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:2009	iuphar.ligand:2009	DES-AA1,2,5,12,13-[D-TRP8]SRIF	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:2012	iuphar.ligand:2012	DES-AA5-[D-TRP8]SRIF	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2057	iuphar.ligand:2057	[111IN,90Y]DOTA-NOC	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:2068	iuphar.ligand:2068	BIM 23058	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:2077	iuphar.ligand:2077	SST3-ODN-8	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2005	iuphar.ligand:2005	CGP 23996	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:2016	iuphar.ligand:2016	L-817,818	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2012	iuphar.ligand:2012	DES-AA5-[D-TRP8]SRIF	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2058	iuphar.ligand:2058	[111IN,90Y]DOTA-OC	FALSE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:10127	iuphar.ligand:10127	STING AGONIST 2	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.019142425	IUPHAR.LIGAND:7113	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:9761	iuphar.ligand:9761	COMPOUND 9 [PMID: 26006010]	FALSE	FALSE	FALSE
NCBIGENE:2642	hgnc:4192	GCGR	GuideToPharmacology	2024.1	inhibitor	0.3750547945406749	IUPHAR.LIGAND:7403	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	1.019566431761058	IUPHAR.LIGAND:12026	ncit:C170368	RESMETIROM	TRUE	FALSE	FALSE
NCBIGENE:1752	hgnc:11848	TLR2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:8888	iuphar.ligand:8888	COMPOUND 13 [PMID: 23098072]	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	OXAPROZIN POTASSIUM	rxcui:660767	OXAPROZIN POTASSIUM	TRUE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1971	iuphar.ligand:1971	EP 171	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.069089041	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1976	ncit:C76408	VAPIPROST	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1983	iuphar.ligand:1983	[125I]SQ-29548	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.6482428547616604	IUPHAR.LIGAND:9380	iuphar.ligand:9380	BIX02189	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.596678082	IUPHAR.LIGAND:6308	iuphar.ligand:6308	OLEOCANTHAL	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	blocker	0.760980743	IUPHAR.LIGAND:9968	iuphar.ligand:9968	SH045	FALSE	FALSE	FALSE
NCBIGENE:488	hgnc:812	ATP2A2	GuideToPharmacology	2024.1	activator	1.141471113819445	IUPHAR.LIGAND:2436	iuphar.ligand:2436	OAG	FALSE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.1831662950082366	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.2386712328895204	IUPHAR.LIGAND:4339	iuphar.ligand:4339	URB597	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	0.2763561643983921	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	1.875273972703375	IUPHAR.LIGAND:12536	iuphar.ligand:12536	LBA	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	activator	0.375054795	IUPHAR.LIGAND:2459	iuphar.ligand:2459	DECAVANADATE	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:12535	iuphar.ligand:12535	PENTAFLUORO-TRITYL CLOTRIMAZOLE ANALOGUE 29A	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.05853698	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:2480	rxcui:29209	MALIC ACID	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	0.1767935058440892	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.094099769	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:7954	iuphar.ligand:7954	BMS-911543	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2779	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.082043236	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2645	hgnc:4195	GCK	GuideToPharmacology	2024.1	inhibitor	0.1060761035064535	IUPHAR.LIGAND:6853	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2259	iuphar.ligand:2259	RO 25-1553	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:2281	iuphar.ligand:2281	[125I]BAY 55-9837	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.032055965	IUPHAR.LIGAND:2174	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:2179	iuphar.ligand:2179	[THR4,GLY7]OT	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2196	iuphar.ligand:2196	OPC-21268	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.014617949	IUPHAR.LIGAND:2190	iuphar.ligand:2190	D[LEU4]AVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2217	iuphar.ligand:2217	D(CH2)5[TYR(ET)2,VAL4,DES-GLY9]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.1093909817410302	IUPHAR.LIGAND:2213	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.1262203635473425	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2235	iuphar.ligand:2235	D(CH2)5[D-ILE2,ILE4,TYR-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2208	iuphar.ligand:2208	[PHAA1,D-TYR(ET)2,LYS6,DES-GLY9]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2215	iuphar.ligand:2215	D(CH2)5[D-ILE2,ILE4,ALA-NH2]AVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2232	iuphar.ligand:2232	[125I]D(CH2)5[D-TYR(ET)2,ILE4,TYR-NH29]AVP	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.072125922	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
NCBIGENE:75	hgnc:148	ACTG1P3	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:4370	iuphar.ligand:4370	XCL2	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2208	iuphar.ligand:2208	[PHAA1,D-TYR(ET)2,LYS6,DES-GLY9]AVP	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:7733	iuphar.ligand:7733	GDC-0152	FALSE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
SCNN1G	hgnc:10602	SCNN1G	ChEMBL	33	blocker	1.620607136904151	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:1505	iuphar.ligand:1505	NPY	FALSE	FALSE	FALSE
NCBIGENE:587	hgnc:977	BCAT2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:4164	iuphar.ligand:4164	CU2+	FALSE	FALSE	FALSE
NCBIGENE:587	hgnc:977	BCAT2	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.1215455352678113	ENCORAFENIB	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
IKZF1	hgnc:13176	IKZF1	CIViC	10-Apr-24	NULL	0.1296485709523321	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
RUNX1	hgnc:10471	RUNX1	CIViC	10-Apr-24	NULL	0.018521224	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
SCNN1B	hgnc:10600	SCNN1B	ChEMBL	33	blocker	1.823183029	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.1396480617970598	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.022225469	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
IGF2	hgnc:5466	IGF2	CIViC	10-Apr-24	NULL	0.4167275494896388	LINSITINIB	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.5000730593875666	C-MET INHIBITOR	ncit:C143099	C-MET INHIBITOR	FALSE	FALSE	TRUE
HAVCR2	hgnc:18437	HAVCR2	CIViC	10-Apr-24	NULL	4.375639269641208	PD1 INHIBITOR	ncit:C124946	PD1 INHIBITOR	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.006945459	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
CTAG1B	hgnc:2491	CTAG1B	CIViC	10-Apr-24	NULL	1.640864726115453	LETETRESGENE AUTOLEUCEL	ncit:C121379	LETETRESGENE AUTOLEUCEL	FALSE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	CIViC	10-Apr-24	NULL	0.01354163	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	CIViC	10-Apr-24	NULL	0.6482428547616604	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.2035181055647073	RITODRINE HYDROCHLORIDE	rxcui:105470	RITODRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	CIViC	10-Apr-24	NULL	0.2019525816757481	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.108040476	IDELALISIB	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1060761035064535	ATAZANAVIR SULFATE	rxcui:343047	ATAZANAVIR	TRUE	FALSE	FALSE
FOXF1	hgnc:3809	FOXF1	CIViC	10-Apr-24	NULL	1.312691780892362	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
IGF1R	hgnc:5465	IGF1R	CIViC	10-Apr-24	NULL	0.9907107780319716	LINSITINIB	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.108711535	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1767935058440892	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
ADH1C	hgnc:251	ADH1C	ChEMBL	33	inhibitor	0.8751278539282417	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.068503159	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
ATR	hgnc:882	ATR	JAX-CKB	10-Apr-24	NULL	0.1944728564284981	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
ATR	hgnc:882	ATR	JAX-CKB	10-Apr-24	NULL	1.750255707856483	VE-821	iuphar.ligand:8042	VE-821	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.019980088	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.052630476	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
PDE6C	hgnc:8787	PDE6C	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	1.282909942931453	Encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Tiragolumab	ncit:C131291	TIRAGOLUMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.02287916	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.4118248724368195	Sintilimab	ncit:C132992	SINTILIMAB	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.043430663	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.4039051633514962	Ulixertinib	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.5303805175322676	BAY1161909	ncit:C116074	EMPESERTIB	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.1001290450718812	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.175610941	Saracatinib	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.4070362111294147	3D185	ncit:C175460	FGFR/CSF-1R INHIBITOR 3D185	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.047647615	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.005787883	Methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	Glasdegib	rxcui:2105845	GLASDEGIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.2160809515872201	Saridegib	ncit:C80063	PATIDEGIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.172722603	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
PDE1A	hgnc:8774	PDE1A	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.006583621	Metformin	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.019750864	Saracatinib	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	4.375639269641208	SH1573	ncit:C180425	IDH2 MUTANT INHIBITOR SH1573	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.2282942227638891	INCB053914	ncit:C124226	UZANSERTIB	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.6351734423672721	Lifirafenib	ncit:C124995	LIFIRAFENIB	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1209854175937661	I-BET151	iuphar.ligand:7518	I-BET151	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.3947945205691315	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
PDE6B	hgnc:8786	PDE6B	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.045016865	Apitolisib	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.108040476	Idelalisib	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.037398626	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.182318303	LY2780301	ncit:C95737	AKT INHIBITOR LY2780301	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.034727296	Floxuridine	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	CC-115	drugbank:DB12740	CC-115	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	APS03118	ncit:C198976	RET INHIBITOR APS03118	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.088322407	BAY 61-3606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	1.009762908	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.5173169579871378	Vistusertib	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
PDE6D	hgnc:8788	PDE6D	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.077273983	Obinutuzumab	rxcui:974779	OBINUTUZUMAB	TRUE	FALSE	FALSE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.022078281	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.006439499	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	GSK2830371	iuphar.ligand:11103	GSK2830371	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.007478127	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.069546584	Milademetan	ncit:C141432	MILADEMETAN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.028977744	Tanespimycin	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.00551957	Ixazomib	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.019318496	Epirubicin	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.013636585	Ruxolitinib	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
PDE6G	hgnc:8789	PDE6G	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.057197899	3,4-METHYLENEDIOXYB-NITROSTYRENE	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.015911416	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.5173169579871378	LYMPHOKINES	ncit:C621	RECOMBINANT LYMPHOKINE	FALSE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.3633748874442526	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.068191781	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	SAN-300	chembl:CHEMBL4297822	SAN-300	FALSE	FALSE	FALSE
UNIPROT:P00790	hgnc:8885	PGA3	TEND	1-Aug-11	NULL	17.50255707856483	SUCRALFATE	rxcui:10156	SUCRALFATE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.038837035	IUPHAR.LIGAND:551	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NCBIGENE:623	hgnc:1029	BDKRB1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:2828	iuphar.ligand:2828	DAIDZEIN	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.027010119	Cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.054020238	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	PLAZOMICIN SULFATE	rxcui:2052872	PLAZOMICIN SULFATE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.015002192	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.069824031	LERCANIDIPINE	rxcui:135056	LERCANIDIPINE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	7-METHOXYISOFLAVONE	chembl:CHEMBL563919	CHEMBL:CHEMBL563919	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	BENZO[DE]ISOCHROMEN-1(3H)-ONE	chembl:CHEMBL1479195	CHEMBL:CHEMBL1479195	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.00770359	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.056826484	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:10257	iuphar.ligand:10257	GR-389988	FALSE	FALSE	FALSE
NCBIGENE:2082	ncbigene:2082	ERPL1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8196	iuphar.ligand:8196	COMPOUND 17D [PMID: 23099093]	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:6073	ncit:C90753	TERUTROBAN	FALSE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.4861821410712454	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
CLNK	hgnc:17438	CLNK	PharmGKB	4/5/24	NULL	13.12691780892362	Antihypertensives	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	5.250767123569449	Piperaquine	ncit:C87634	PIPERAQUINE	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.030527716	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
MLST8	hgnc:24825	MLST8	ChEMBL	33	activator	4.375639269641208	INDOXIMOD	ncit:C71535	INDOXIMOD	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	1.678633990910949	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	7-NITROINDAZOLE	drugbank:DB02207	7-NITROINDAZOLE	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.03409589	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	0.6035364509849942	ENOXACIN	rxcui:3925	ENOXACIN	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DIBUCAINE HYDROCHLORIDE	rxcui:235402	DIBUCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.016449772	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.0023813	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.062733179	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
GIPR	hgnc:4271	GIPR	PharmGKB	4/5/24	NULL	0.6908904109959803	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:732	hgnc:1353	C8B	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.018819954	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
PROTEIN KINASE C BETA	hgnc:9395	PRKCB	TTD	2020.06.01	NULL	1.367387271762877	Enzastaurin	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.038608582	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	LADIRATUZUMAB VEDOTIN	ncit:C112001	LADIRATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.005723531	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	1.250182648468916	ETHER	ncit:C29819	ETHER	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.030527716	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
C5ORF56	hgnc:33838	CARINH	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.039390601	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	TALC	12-May-16	inhibitor	3.443125982668491	MEDI-575	ncit:C82684	TOVETUMAB	FALSE	TRUE	TRUE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	0.5469549087051511	BG-9928	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:4013	iuphar.ligand:4013	[125I]KISSPEPTIN-14 (HUMAN)	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.033658764	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9102	iuphar.ligand:9102	SC-22716	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.016434326	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	HEMATOXYLIN	drugbank:DB16871	HEMATOXYLIN	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.2822993077187876	PF-04236921	chembl:CHEMBL2109613	PF-04236921	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.082429625	CHLORDIAZEPOXIDE	rxcui:2356	CHLORDIAZEPOXIDE	TRUE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.561579372	Durvalumab	rxcui:1919503	DURVALUMAB	TRUE	FALSE	TRUE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.020656047	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	0.3500511415712967	IUPHAR.LIGAND:6228	iuphar.ligand:6228	VU0001171	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DICHLOROXYLENOL	ncit:C77048	DICHLOROXYLENOL	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.1130007271930297	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	CGI	2/1/22	NULL	0.2540693769469088	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.069454592	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PARP1	hgnc:270	PARP1	MyCancerGenome	20-Jun-17	other/unknown	0.3818739726232327	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.2051080907644316	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.1203384367510187	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3004	iuphar.ligand:3004	COMPOUND 2C [PMID: 2153213]	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	negative modulator	0.1143957978991165	KETAMINE HYDROCHLORIDE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.3500511415712966	CLINAFLOXACIN	ncit:C74372	CLINAFLOXACIN	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.3365876361262467	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	FLURBIPROFEN SODIUM	rxcui:91351	FLURBIPROFEN SODIUM	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.015434354	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.084553416	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
NCBIGENE:2352	hgnc:3795	FOLR3	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9855	ncit:C174598	PETESICATIB	FALSE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	modulator	0.087512785	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.9907107780319716	INSM-18	chembl:CHEMBL3545025	INSM-18	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.00881889	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.1172918940484613	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.019447286	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	LAVENDUSTIN C	ncit:C1487	LAVENDUSTIN C	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007003824	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.014172111	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.010948222	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.041021618	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
RPS2	hgnc:10404	RPS2	ChEMBL	33	modulator	0.1093909817410302	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	chembl:CHEMBL1348974	(4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE	FALSE	FALSE	FALSE
NCBIGENE:2835	hgnc:4466	GPR12	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:12615	ncit:C167347	TULMIMETOSTAT	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:7361	iuphar.ligand:7361	COMPOUND 24 [PMID: 16451050]	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	HYDROXYTYROSOL	rxcui:1314227	HYDROXYTYROSOL	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.1565523888959287	ZOLPIDEM TARTRATE	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.138178082	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2651902587661338	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	TCMDC-123951	chembl:CHEMBL587849	CHEMBL:CHEMBL587849	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.035005114	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
ATAT1	hgnc:21186	ATAT1	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:1298	iuphar.ligand:1298	MELANIN-CONCENTRATING HORMONE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	ALLITRIDIN	chembl:CHEMBL123040	ALLITRIDIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	GNF-PF-5183	chembl:CHEMBL577660	CHEMBL:CHEMBL577660	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.8401227397711121	SAPONIN	ncit:C823	SAPONIN	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
ASNS	hgnc:753	ASNS	PharmGKB	4/5/24	NULL	14.58546423213736	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
UNIPROT:P50391	hgnc:9329	NPY4R	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	OBINEPITIDE	ncit:C175168	OBINEPITIDE	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C9	hgnc:60	ABCC9	TTD	2020.06.01	NULL	0.596678082	Glimepiride	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
POLA1	hgnc:9173	POLA1	ChEMBL	33	inhibitor	0.070574827	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	1.712206670729168	Macitentan	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:3777	iuphar.ligand:3777	[125I]CT (SALMON)	FALSE	FALSE	FALSE
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.5357925636295356	Tasidotin hydrochloride	ncit:C142999	TASIDOTIN HYDROCHLORIDE	FALSE	FALSE	FALSE
CACNB2	hgnc:1402	CACNB2	ChEMBL	33	modulator	0.1262203635473425	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
ADH1A	hgnc:249	ADH1A	ChEMBL	33	inhibitor	0.4688184931758437	NITREFAZOLE	ncit:C72626	NITREFAZOLE	TRUE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:6126	iuphar.ligand:6126	SNAP 37889	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.027010119	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.076934317	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MT-RNR1	hgnc:7470	MT-RNR1	PharmGKB	4/5/24	NULL	7.501095891	micronomicin	rxcui:29996	MICRONOMICIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
DUSP1	hgnc:3064	DUSP1	NCI	14-Sep-17	NULL	0.212152207	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.1921012362281506	SODIUM PHENYLBUTYRATE	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.1442518440541057	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	TOLMETIN	rxcui:10636	TOLMETIN	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	modulator	0.063110182	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.07458476	Bethanidine	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	1.250182648468916	IUPHAR.LIGAND:6941	rxcui:974779	OBINUTUZUMAB	TRUE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:4209	iuphar.ligand:4209	GYKI53655	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2259	iuphar.ligand:2259	RO 25-1553	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.063160791	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1008469998124734	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.5527123287967841	IUPHAR.LIGAND:215	iuphar.ligand:215	NORFENFLURAMINE	FALSE	FALSE	FALSE
CACNB4	hgnc:1404	CACNB4	ChEMBL	33	modulator	0.1553481397505754	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	3.889457128569962	LFB-R603	chembl:CHEMBL2109348	LFB-R603	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.525076712	nalidixic acid	rxcui:7240	NALIDIXIC ACID	TRUE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:873	iuphar.ligand:873	CI-988	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.045016865	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
TNFRSF17	hgnc:11913	TNFRSF17	ChEMBL	33	binder	0.6908904109959803	TECLISTAMAB	rxcui:2619425	TECLISTAMAB-CQYV	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	OLVANIL	ncit:C166774	OLVANIL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000942602	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.3271505995993426	AMITIFADINE	ncit:C169780	AMITIFADINE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.3697723326457359	GNF-PF-3770	chembl:CHEMBL597874	CHEMBL:CHEMBL597874	FALSE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	1.875273972703375	GNF-PF-3971	chembl:CHEMBL599890	CHEMBL:CHEMBL599890	FALSE	FALSE	FALSE
KCNK10	hgnc:6273	KCNK10	ChEMBL	33	potentiator	0.2838252499226729	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.012710644	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.039763477	Busulfan	rxcui:1828	BUSULFAN	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.1187188949127459	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	inhibitor	5.527123287967842	IUPHAR.LIGAND:9774	ncit:C169937	ELISMETREP	FALSE	FALSE	FALSE
PSMD7	hgnc:9565	PSMD7	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.062808219	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.045658845	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
NDUFS4	hgnc:7711	NDUFS4	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
KCNH8	hgnc:18864	KCNH8	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.2051080907644316	2-(2-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL112060	CHEMBL:CHEMBL112060	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.1682938180631234	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NDUFA3	hgnc:7686	NDUFA3	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.069089041	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.015892152	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	0.7501095890813501	GNF-PF-5183	chembl:CHEMBL577660	CHEMBL:CHEMBL577660	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.2857560339357523	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.067317527	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P09960	hgnc:6710	LTA4H	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	DG051	drugbank:DB05177	DG051	FALSE	FALSE	FALSE
UNIPROT:P45880	hgnc:12672	VDAC2	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	OLESOXIME	ncit:C174604	OLESOXIME	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.049723174	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:5976	drugbank:DB08454	N-(5-METHYL-1H-PYRAZOL-3-YL)-2-PHENYLQUINAZOLIN-4-AMINE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.016077058	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	DTC	9/2/20	NULL	0.1790542923638346	KETAMINE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	SKF-38393	iuphar.ligand:935	SKF-38393	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	S(+)-ISOPROTERENOL-BITARTRATE	chembl:CHEMBL1257092	CHEMBL:CHEMBL1257092	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.1105424657593568	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.039778539	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	1.121958787087489	Lovastatin	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CHRND	hgnc:1965	CHRND	ChEMBL	33	inhibitor	0.5357925636295356	VECURONIUM BROMIDE	rxcui:11153	VECURONIUM BROMIDE	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	3.750547945	DESMOTEPLASE	ncit:C87246	DESMOTEPLASE	TRUE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.3750547945406749	GNF-PF-4085	chembl:CHEMBL528181	CHEMBL:CHEMBL528181	FALSE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.1054370908347279	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	0.4565884455277782	AZD3463	iuphar.ligand:7706	AZD3463	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.201178817	PENICILLIOL A	chembl:CHEMBL457041	PENICILLIOL A	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005669763	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	GW0742	iuphar.ligand:2686	GW0742X	FALSE	FALSE	FALSE
UNIPROT:P30291	hgnc:12761	WEE1	TdgClinicalTrial	Jan-14	NULL	0.7212592202705288	MK-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
NCBIGENE:1264	hgnc:2155	CNN1	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10669	iuphar.ligand:10669	A-908292	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.018106094	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.049676132	GNF-PF-1319	chembl:CHEMBL235891	CHEMBL:CHEMBL235891	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	4,4'-DITHIODIPYRIDINE	chembl:CHEMBL1232076	CHEMBL:CHEMBL1232076	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.092606122	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.1174668260306364	24-OXOCYCLOARTANOL	chembl:CHEMBL225869	CHEMBL:CHEMBL225869	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	SCH-23390	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	NITAZOXANIDE	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:10142	iuphar.ligand:10142	PQR620	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	GNF-PF-2776	chembl:CHEMBL578294	CHEMBL:CHEMBL578294	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.093763699	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
HSPG2	hgnc:5273	HSPG2	NCI	14-Sep-17	NULL	0.4023576339899961	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
HPD	hgnc:5147	HPD	NCI	14-Sep-17	NULL	1.750255707856483	6-HYDROXYDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.2763561643983921	DEXTROAMPHETAMINE SULFATE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.088945801	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
HAVCR2	hgnc:18437	HAVCR2	ChEMBL	33	inhibitor	4.375639269641208	RO-7121661	chembl:CHEMBL4594602	RO-7121661	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002553627	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-156744	chembl:CHEMBL1481453	CHEMBL:CHEMBL1481453	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.4734548598913698	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	modulator	0.054695491	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.1666910197958555	ARRY-300	chembl:CHEMBL3545359	ARRY-300	FALSE	FALSE	FALSE
PSMA7	hgnc:9536	PSMA7	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	REMIMAZOLAM BESYLATE	rxcui:2383942	REMIMAZOLAM BESYLATE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012977675	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	agonist	0.040021091	ABP-700	drugbank:DB15411	ABP-700	FALSE	FALSE	FALSE
NCBIGENE:2652	hgnc:4206	OPN1MW	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8238	iuphar.ligand:8238	A-366	FALSE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.4688184931758437	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	inverse agonist	0.038159645	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
CUL4A	hgnc:2554	CUL4A	ChEMBL	33	inhibitor	3.281729452230906	POMALIDOMIDE	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
NCBIGENE:2792	hgnc:4411	GNGT1	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:7729	drugbank:DB16305	XEVINAPANT	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.090821275	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.4907258993990139	1-HYDROXY-6-(4-HYDROXY-PHENYL)-1-PHENYL-HEXAN-3-ONE (ENANTIOMERIC MIX)	chembl:CHEMBL1095870	1-HYDROXY-6-(4-HYDROXY-PHENYL)-1-PHENYL-HEXAN-3-ONE (ENANTIOMERIC MIX)	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	agonist	0.097236428	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.067839369	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1607377690888607	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5744	iuphar.ligand:5744	COMPOUND 2 [PMID: 21939274]	FALSE	FALSE	FALSE
NCBIGENE:385	hgnc:18865	KCNT1	GuideToPharmacology	2024.1	activator	0.3889457128569963	IUPHAR.LIGAND:8494	rxcui:7402	NICLOSAMIDE	TRUE	FALSE	FALSE
NCBIGENE:2871	hgnc:4547	GRK6P1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8515	iuphar.ligand:8515	MJN228	FALSE	FALSE	FALSE
NCBIGENE:1213	hgnc:2092	CLTC	GuideToPharmacology	2024.1	NULL	0.2027323213733378	IUPHAR.LIGAND:6690	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
CACNA1F	hgnc:1393	CACNA1F	PharmGKB	4/5/24	NULL	0.043866058	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.019739726	pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.044498026	PD-404182	chembl:CHEMBL595227	CHEMBL:CHEMBL595227	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006356861	SKF-82526	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	2.625383561784724	IUPHAR.LIGAND:9313	iuphar.ligand:9313	GW542573X	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:12720	iuphar.ligand:12720	PF-06843195	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	HARMALINE	drugbank:DB13875	HARMALINE	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	3.088686543276147	5,6,7-TRIBROMOISATIN	chembl:CHEMBL376616	CHEMBL:CHEMBL376616	FALSE	FALSE	FALSE
MAGEA3	hgnc:6801	MAGEA3	NCI	14-Sep-17	NULL	5.834185692854944	INCOMPLETE FREUND&APOS;S ADJUVANT	ncit:C1573	INCOMPLETE FREUND'S ADJUVANT	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.8975670296699914	MISONIDAZOLE	ncit:C657	MISONIDAZOLE	FALSE	FALSE	FALSE
BLMH	hgnc:1059	BLMH	PharmGKB	4/5/24	NULL	1.230648544586589	bleomycin	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.9053046764774912	VALRUBICIN	rxcui:31435	VALRUBICIN	TRUE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:9913	iuphar.ligand:9913	FLUMBATINIB	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:6992	iuphar.ligand:6992	VPC03090-P	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	modulator	0.8468979231563628	IUPHAR.LIGAND:10432	rxcui:2612087	DEUCRAVACITINIB	TRUE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.305277158	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NSC-270156	chembl:CHEMBL471226	CHEMBL:CHEMBL471226	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.041672755	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	GNF-PF-1000	chembl:CHEMBL600554	CHEMBL:CHEMBL600554	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PYRAFLUFEN-ETHYL	chembl:CHEMBL1905010	PYRAFLUFEN-ETHYL	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.5147810905460245	MAFOSFAMIDE	ncit:C1150	MAFOSFAMIDE	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.091476779	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.1154014752432846	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
NF1	hgnc:7765	NF1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2853677784548614	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
GADD45A	hgnc:4095	GADD45A	NCI	14-Sep-17	NULL	0.5357925636295356	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.8334550989792777	MATUZUMAB	ncit:C2012	MATUZUMAB	FALSE	FALSE	TRUE
UNIPROT:Q9UQL6	hgnc:14068	HDAC5	TdgClinicalTrial	Jan-14	NULL	0.094608417	RESMINOSTAT	ncit:C84856	RESMINOSTAT	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	TCMDC-125204	chembl:CHEMBL588028	CHEMBL:CHEMBL588028	FALSE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.035098711	METHYLENEDIOXYMETHAMPHETAMINE	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	ISOGINKGETIN	chembl:CHEMBL1208903	ISOGINKGETIN	FALSE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	0.1097721349875146	PEMBROLIZUMAB	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.1615620653405984	EGANELISIB	ncit:C125471	EGANELISIB	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	ChEMBL	33	inhibitor	0.218327115	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	GNF-PF-1935	chembl:CHEMBL588250	CHEMBL:CHEMBL588250	FALSE	FALSE	FALSE
ADH6	hgnc:255	ADH6	ChEMBL	33	inhibitor	0.7501095890813498	NITREFAZOLE	ncit:C72626	NITREFAZOLE	TRUE	FALSE	FALSE
RPS9	hgnc:10442	RPS9	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	DTC	9/2/20	NULL	0.1583941817064691	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
NR2F2	hgnc:7976	NR2F2	DTC	9/2/20	NULL	1.458546423213736	GNF-PF-1678	chembl:CHEMBL580340	CHEMBL:CHEMBL580340	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:766	iuphar.ligand:766	[125I]CCL8 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:3293	iuphar.ligand:3293	[ARG16]CHICKEN SECRETIN	FALSE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	1.419126249613364	MN-305	drugbank:DB05339	MN-305	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.008937476	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	3.750547945	AM-1638	chembl:CHEMBL2152070	CHEMBL:CHEMBL2152070	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	NSC-3323	chembl:CHEMBL1270169	CHEMBL:CHEMBL1270169	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	ZAPA	chembl:CHEMBL20562	ZAPA	FALSE	FALSE	FALSE
PSMC6	hgnc:9553	PSMC6	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD11	hgnc:9556	PSMD11	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.036770078	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.036770078	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.058471794	IUPHAR.LIGAND:2227	iuphar.ligand:2227	[3H]D[CHA4]AVP	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.075333818	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	GS-39783	iuphar.ligand:5446	GS39783	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	1.141471113819445	OM-174	ncit:C169880	DEFOSLIMOD	FALSE	FALSE	FALSE
UNIPROT:P45985	hgnc:6844	MAP2K4	TdgClinicalTrial	Jan-14	NULL	0.8334550989792776	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
5-HT 1D RECEPTOR	hgnc:5289	HTR1D	TTD	2020.06.01	NULL	0.8078103267029924	Zolmitriptan	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.2224901323546377	IUPHAR.LIGAND:219	iuphar.ligand:219	[3H]LSD	FALSE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.01816246	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
RPS24	hgnc:10411	RPS24	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	FENEBRUTINIB	ncit:C116844	FENEBRUTINIB	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.056826484	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	1.235474617310458	GEN1046	ncit:C172194	ACASUNLIMAB	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CYCLIC ADENOSINE MONOPHOSPHATE	drugbank:DB02527	CYCLIC ADENOSINE MONOPHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TEND	1-Aug-11	NULL	2.072671233	XIMELAGATRAN	ncit:C77996	XIMELAGATRAN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.2804896967718723	PSC-833	ncit:C1405	VALSPODAR	FALSE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	0.7001022831425933	fexofenadine	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
WHSC1	hgnc:12766	NSD2	DTC	9/2/20	NULL	0.546954909	NSC-36398	chembl:CHEMBL483206	CHEMBL:CHEMBL483206	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	(S,R)-MEFLOQUINE	chembl:CHEMBL172	(S,R)-MEFLOQUINE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	GNF-PF-2776	chembl:CHEMBL578294	CHEMBL:CHEMBL578294	FALSE	FALSE	FALSE
TNF-RELATED WEAK INDUCER OF APOPTOSIS	hgnc:11927	TNFSF12	TTD	2020.06.01	NULL	78.76150685354175	RO-5458640	chembl:CHEMBL2109600	RO-5458640	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.1565523888959287	Zolpidem	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.2273059360852575	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.081830137	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE	chembl:CHEMBL344469	0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002196239	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	1.071585127259071	ELSILIMOMAB	ncit:C188564	ELSILIMOMAB	FALSE	FALSE	FALSE
DDB1	hgnc:2717	DDB1	ChEMBL	33	modulator	3.281729452230906	IBERDOMIDE	ncit:C129048	IBERDOMIDE	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:12078	iuphar.ligand:12078	INIXACICLIB	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.049535539	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.082429625	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	8.751278539282415	BMS-833923	drugbank:DB16844	BMS-833923	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:12734	iuphar.ligand:12734	COMPOUND 4G [PMID: 30893553]	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.068847471	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
ANGPTL3	hgnc:491	ANGPTL3	ChEMBL	33	inhibitor	26.25383561784724	EVINACUMAB	rxcui:2478335	EVINACUMAB	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	RALOXIFEN	chembl:CHEMBL1079109	RALOXIFEN	TRUE	FALSE	FALSE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TdgClinicalTrial	Jan-14	NULL	0.1873044158229292	GLIBENCLAMIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:1783	iuphar.ligand:1783	UDP-GLUCOSE	FALSE	FALSE	FALSE
NCBIGENE:669	hgnc:1093	BPGM	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:12452	iuphar.ligand:12452	BETA-GENTIOBIOSE	FALSE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.1646008502686348	IUPHAR.LIGAND:7938	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
NCBIGENE:984	hgnc:1729	CDK11B	GuideToPharmacology	2024.1	NULL	1.029562181092048	IUPHAR.LIGAND:4659	iuphar.ligand:4659	[3H]GLYSAR	FALSE	FALSE	FALSE
NCBIGENE:716	hgnc:1247	C1S	GuideToPharmacology	2024.1	inhibitor	0.1312691780892362	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1495945049449985	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.7778914257139926	RIVICICLIB	ncit:C64762	RIVICICLIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PYRVINIUM PAMOATE	rxcui:55347	PYRVINIUM PAMOATE	TRUE	FALSE	FALSE
HPSE	hgnc:5164	HPSE	DTC	9/2/20	NULL	0.3241214273808303	METERGOLINE	rxcui:6834	METERGOLINE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	inhibitor	0.022249013	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.024513385	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1193356164447602	HYDROXYSTILBAMIDINE ISETHIONATE	ncit:C65871	HYDROXYSTILBAMIDINE ISETHIONATE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.4930297768609811	POLYESTRADIOL PHOSPHATE	rxcui:34120	POLYESTRADIOL PHOSPHATE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.5385402178019948	THEAFLAVINS	ncit:C29855	THEAFLAVIN	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.033002936	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.025757994	Pirarubicin	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	DTC	9/2/20	NULL	0.1172046232939609	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1166837138570988	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:7922	iuphar.ligand:7922	(HYDROXYMETHYLPHENYL)AGOMELATINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	PharmGKB	4/5/24	NULL	0.011054247	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.07699072	IUPHAR.LIGAND:7792	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:9324	iuphar.ligand:9324	HINSL5: A8-21 (T9R)	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.1396480617970598	IUPHAR.LIGAND:2018	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.089756703	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6482428547616604	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.2035181055647073	NAFTOPIDIL	ncit:C72927	NAFTOPIDIL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005424346	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.060772768	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
INSRR	hgnc:6093	INSRR	DTC	9/2/20	inhibitor	0.6563458904461813	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.056018141	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.086551106	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.080781033	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	COSMIC	4-Sep-20	NULL	0.2639729920045843	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.089756703	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
HTR2B	hgnc:5294	HTR2B	ChEMBL	33	agonist	0.1286952726365061	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	TELISOTUZUMAB VEDOTIN	ncit:C118571	TELISOTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	ARMODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.062262061	ROTIGOTINE	rxcui:616739	ROTIGOTINE	TRUE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1979	ncit:C65463	DOMITROBAN	FALSE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	NCI	14-Sep-17	NULL	0.2206204673768676	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.1250182648468916	ROPINIROLE HYDROCHLORIDE	rxcui:236553	ROPINIROLE HYDROCHLORIDE	TRUE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	1.325951293830669	Zafirlukast	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	0.105015342	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:4005	iuphar.ligand:4005	METHYLLYCACONITINE	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1693	iuphar.ligand:1693	SB 612111	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.085796848	2-MESATP	iuphar.ligand:1711	2MESATP	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.028626235	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	CARBARIL	ncit:C76389	CARBARIL	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.018206543	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.09741683	RG-547	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.017243899	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.2083637747448194	AG-13958	chembl:CHEMBL3545335	AG-13958	FALSE	FALSE	FALSE
ELANE	hgnc:3309	ELANE	ChEMBL	33	inhibitor	1.141471113819445	ALVELESTAT	ncit:C125714	ALVELESTAT	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.072927321	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
UNIPROT:P06756	hgnc:6150	ITGAV	TdgClinicalTrial	Jan-14	NULL	0.3671865121377238	ANTITHYMOCYTE GLOBULIN	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.2333674277141977	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
NCBIGENE:1042	hgnc:10973	SLC23A2	GuideToPharmacology	2024.1	NULL	2.019525816757481	IUPHAR.LIGAND:4532	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.010177878	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PTH1R	hgnc:9608	PTH1R	ChEMBL	33	agonist	2.500365296937833	PARATHYROID HORMONE	rxcui:1427222	PARATHYROID HORMONE	TRUE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	1.346350544504987	SUVN-D4010	iuphar.ligand:12749	USMARAPRIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.036977233	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	inhibitor	0.037505479	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	N-METHYLHISTAMINE	iuphar.ligand:1241	N-[3H]METHYLHISTAMINE	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1415301111474245	DNDI1417413	chembl:CHEMBL1343568	CHEMBL:CHEMBL1343568	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.078136416	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	ROPIVACAINE HYDROCHLORIDE	rxcui:236539	ROPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9799	iuphar.ligand:9799	SCH.336	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5785	iuphar.ligand:5785	MK 1903	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.018106094	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.01214331	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.6908904109959803	CP-724714	drugbank:DB12302	CP-724714	FALSE	FALSE	FALSE
SETD4	hgnc:1258	SETD4	PharmGKB	4/5/24	NULL	0.5770073762164231	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.1389091831632129	INCB40093	ncit:C107686	DEZAPELISIB	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.03070624	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.1356787370431382	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.061340737	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	0.046303061	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
NCBIGENE:608	hgnc:11913	TNFRSF17	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:6695	iuphar.ligand:6695	BI6015	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	0.081533651	IUPHAR.LIGAND:1456	rxcui:4053	ERYTHROMYCIN	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.046221542	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	DTC	9/2/20	NULL	1.875273972703375	CORTISONE	rxcui:2878	CORTISONE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	2.333674277141977	TELEOCIDIN B	chembl:CHEMBL488007	TELEOCIDIN B	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	PBCAR0191	ncit:C158558	AZERCABTAGENE ZAPRELEUCEL	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.011738804	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007551801	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
S1PR4	hgnc:3170	S1PR4	DTC	9/2/20	NULL	0.5303805175322677	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.007624172	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
DDR2	hgnc:2731	DDR2	CGI	2/1/22	NULL	1.067952635302261	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	VAPITADINE DIHYDROCHLORIDE	ncit:C96722	VAPITADINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2778183663264258	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:4209	iuphar.ligand:4209	GYKI53655	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:6676	iuphar.ligand:6676	(RS)-PPCC	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.1226814748497534	SURUFATINIB	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.008013991	mifepristone	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.026779381	Ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
PAX2	hgnc:8616	PAX2	NCI	14-Sep-17	NULL	2.187819634820604	AG 490	iuphar.ligand:5916	AG 490	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	1.591141552596802	DIETHYL-2-DODECYLIDENEMALONATE	chembl:CHEMBL1797708	CHEMBL:CHEMBL1797708	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1961681366215236	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2225	iuphar.ligand:2225	D[PEN1,TYR(ME)2]AVP	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	S(+)-ISOPROTERENOL-BITARTRATE	chembl:CHEMBL1257092	CHEMBL:CHEMBL1257092	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ChEMBL	33	inhibitor	0.1374546367426557	LGX-806	chembl:CHEMBL3545263	LGX-806	FALSE	FALSE	FALSE
DDR2	hgnc:2731	DDR2	CIViC	10-Apr-24	NULL	1.067952635302261	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.02617531	SEMAXANIB	ncit:C1831	SEMAXANIB	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1250182648468916	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
HSD3B7	hgnc:18324	HSD3B7	PharmGKB	4/5/24	NULL	4.375639269641208	cholic acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	2.700394520692859	boceprevir	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.253049018	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.073922431	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.1526385791735305	LY-2874455	drugbank:DB13022	LY-2874455	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.089756703	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:6188	iuphar.ligand:6188	BAG-1	FALSE	FALSE	FALSE
PTHR1	hgnc:9608	PTH1R	NCI	14-Sep-17	NULL	0.3409589041278864	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
GATA3	hgnc:4172	GATA3	PharmGKB	4/5/24	NULL	0.036847489	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
TRANSFORMING GROWTH FACTOR BETA 1	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	0.1483267549030917	LY2157299	ncit:C116891	GALUNISERTIB	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	TENOFOVIR ALAFENAMIDE FUMARATE	rxcui:1721604	TENOFOVIR ALAFENAMIDE FUMARATE	TRUE	FALSE	FALSE
CDK20	hgnc:21420	CDK20	ChEMBL	33	inhibitor	0.6250913242344582	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
KCNH6	hgnc:18862	KCNH6	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
UNIPROT:P11169	hgnc:11007	SLC2A3	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	ChEMBL	33	inhibitor	0.5707355569097228	R-348	drugbank:DB06321	R-348	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.072125922	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.090634645	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.077217164	IUPHAR.LIGAND:17	ncit:C76104	LYSERGIDE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW642125X	chembl:CHEMBL196022	GW642125X	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.015118823	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TEND	1-Aug-11	NULL	0.4150804050252529	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.024309107	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00449706	PENTACHLOROPHENOL	chembl:CHEMBL75967	PENTACHLOROPHENOL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.1852122442176172	PEXIDARTINIB	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.2625383561784725	TAK-593	drugbank:DB13093	TAK-593	FALSE	FALSE	FALSE
KCNE1	hgnc:6240	KCNE1	PharmGKB	4/5/24	NULL	1.607377690888607	sotalol	rxcui:9947	SOTALOL	TRUE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	inhibitor	0.6563458904461813	IUPHAR.LIGAND:4086	iuphar.ligand:4086	[3H]L689560	FALSE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	0.3671865121377238	IUPHAR.LIGAND:2604	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1312691780892362	Glimepiride	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.1785975212098452	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
BCHE	hgnc:983	BCHE	FDA	10-Apr-24	NULL	2.148041096005684	Succinylcholine	rxcui:10154	SUCCINYLCHOLINE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.061055432	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.2778183663264258	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.364636606	GNF-PF-4337	chembl:CHEMBL277148	CHEMBL:CHEMBL277148	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	BPI-9016	chembl:CHEMBL3545236	BPI-9016	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.4565884455277783	OLEANOLIC_ACID	iuphar.ligand:3306	OLEANOLIC ACID	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.5707355569097228	XL-019	chembl:CHEMBL3545328	XL-019	FALSE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	CGI	2/1/22	NULL	0.026519026	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.6019397937072561	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.069332312	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
NCBIGENE:394	hgnc:675	ARHGAP5	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2313	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.2143170254518142	IUPHAR.LIGAND:62	iuphar.ligand:62	(+)-BUTACLAMOL	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	agonist	1.458546423213736	GS-9667	chembl:CHEMBL3545011	GS-9667	FALSE	FALSE	FALSE
FAT1	hgnc:3595	FAT1	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	DTC	9/2/20	NULL	0.050879526	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.026779381	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.014617949	IUPHAR.LIGAND:2219	iuphar.ligand:2219	D(CH2)5[TYR(ME)2,THR4,PHE(3I,4N3)-NH29]OVT	FALSE	FALSE	FALSE
GSTA1	hgnc:4626	GSTA1	PharmGKB	4/5/24	NULL	0.3663325900164732	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	ChEMBL	33	inhibitor	2.386712328895204	CI-988	iuphar.ligand:873	CI-988	FALSE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ChEMBL	33	inhibitor	0.3365876361262468	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.2000292237550266	ETILEVODOPA	rxcui:1421444	ETILEVODOPA	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.5339763176511304	RESCINNAMINE	rxcui:9259	RESCINNAMINE	TRUE	FALSE	FALSE
NCBIGENE:2099	hgnc:3467	ESR1	GuideToPharmacology	2024.1	inhibitor	0.061340737	IUPHAR.LIGAND:8196	iuphar.ligand:8196	COMPOUND 17D [PMID: 23099093]	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:1749	drugbank:DB03435	URIDINE-5'-DIPHOSPHATE	FALSE	FALSE	FALSE
FES	hgnc:3657	FES	DTC	9/2/20	inhibitor	0.3281729452230906	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	DTC	9/2/20	NULL	0.1029562181092049	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:257	iuphar.ligand:257	SB 207710	FALSE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.8334550989792776	TRILACICLIB	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
COL5A3	hgnc:14864	COL5A3	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
MT-ND2	hgnc:7456	MT-ND2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	8.290684931951763	AM-211	chembl:CHEMBL2181753	AM-211	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.2160809515872201	NERAMEXANE MESYLATE	ncit:C75163	NERAMEXANE MESYLATE	FALSE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	0.8751278539282416	ETARACIZUMAB	ncit:C1800	ETARACIZUMAB	FALSE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.037666909	BELANTAMAB MAFODOTIN	rxcui:2387833	BELANTAMAB MAFODOTIN-BLMF	TRUE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:11955	iuphar.ligand:11955	BMS-189532	FALSE	FALSE	FALSE
NCBIGENE:1530	hgnc:10435	RPS6KA6	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10597	iuphar.ligand:10597	BAY-985	FALSE	FALSE	FALSE
NCBIGENE:2235	hgnc:3647	FECH	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.6250913242344582	XEN403	chembl:CHEMBL3545091	XEN403	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001656812	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	2.282942227638891	Clazosentan	ncit:C79486	CLAZOSENTAN	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.013645445	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.1315981735230438	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	1.064344687210023	DIPHEMANIL METHYLSULFATE	rxcui:23364	DIPHEMANIL METHYLSULFATE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.046965717	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.201952582	ANTIANDROGENS	ncit:C242	ANTI-ANDROGEN	FALSE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	SANGIVAMYCIN	chembl:CHEMBL101892	SANGIVAMYCIN	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.1613138901250215	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.9460841664089098	KAEMPFERIDE	chembl:CHEMBL40919	KAEMPFERIDE	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.2442217266776488	SALMETEROL	rxcui:36117	SALMETEROL	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.6035364509849942	GLYCYRRHETINIC ACID	rxcui:1311506	GLYCYRRHETINIC ACID	TRUE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	agonist	0.078958904	IUPHAR.LIGAND:43	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:9664	iuphar.ligand:9664	BML-281	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.4375639269641209	IUPHAR.LIGAND:12438	iuphar.ligand:12438	ARISTOLOCHIC ACID	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:6579	iuphar.ligand:6579	H2L5186303	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	3.621218705909965	IUPHAR.LIGAND:3516	ncit:C66298	PALOSURAN	FALSE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.3125456621172291	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00359617	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.082429625	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	3-HYDROXYBENZYLHYDRAZINE DIHYDROCHLORIDE	iuphar.ligand:5116	3-HYDROXYBENZYLHYDRAZINE	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	DTC	9/2/20	NULL	0.081030357	AZIETOMIDATE	iuphar.ligand:5404	[3H]AZIETOMIDATE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.081407242	tiotropium	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	0.5707355569097228	PHA-543613	iuphar.ligand:3998	PHA-543613	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.014683353	ranolazine	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.008418738	regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	agonist	0.096167896	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	ChEMBL	33	inhibitor	0.1223955040459079	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
RPS28	hgnc:10418	RPS28	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.2465148884304905	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
NCBIGENE:2719	hgnc:4451	GPC3	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8640	iuphar.ligand:8640	COMPOUND 57 [PMID: 26155854]	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:597	iuphar.ligand:597	PD123319	FALSE	FALSE	FALSE
NCBIGENE:239	hgnc:429	ALOX12	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:8198	ncit:C80063	PATIDEGIB	FALSE	FALSE	TRUE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:10283	iuphar.ligand:10283	SAR7334	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE	chembl:CHEMBL344469	0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1041818873724097	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	4.375639269641208	Pankomab-GEX	ncit:C94220	GATIPOTUZUMAB	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	2.341819737097098	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.010711479	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	agonist	0.3182283105193606	IUPHAR.LIGAND:772	iuphar.ligand:772	CCL8	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1852122442176172	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
NCBIGENE:2363	hgnc:3871	FRA1D	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11585	drugbank:DB13000	PCI-27483	FALSE	FALSE	FALSE
NCBIGENE:1800	hgnc:3002	DPEP1	GuideToPharmacology	2024.1	inhibitor	0.043323161	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	0.5966780822238011	IUPHAR.LIGAND:4743	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.011585982	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.8140724222588294	MN-221	chembl:CHEMBL2218893	BEDORADRINE SULFATE	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.075768645	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	4'-METHOXY-AURONE	chembl:CHEMBL611941	4'-METHOXY-AURONE	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1019566431761058	ANAZOLENE	chembl:CHEMBL1555467	ANAZOLENE	FALSE	FALSE	FALSE
SLC29A1	hgnc:11003	SLC29A1	PharmGKB	4/5/24	NULL	0.5933070196123671	trifluridine	rxcui:10803	TRIFLURIDINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.1141471113819445	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TdgClinicalTrial	Jan-14	NULL	2.461297089173179	ZICONOTIDE	rxcui:68503	ZICONOTIDE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:3284	iuphar.ligand:3284	PSB603	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.006912542	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1630673019742065	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.4167275494896388	LYMPHOKINES	ncit:C621	RECOMBINANT LYMPHOKINE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	INDIBULIN	ncit:C2049	INDIBULIN	FALSE	FALSE	FALSE
TDGF1	hgnc:11701	CRIPTO	ChEMBL	33	binder	52.50767123569449	BIIB-015	chembl:CHEMBL2109575	BIIB-015	FALSE	FALSE	FALSE
KCNV1	hgnc:18861	KCNV1	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.037213091	SOBLIDOTIN	ncit:C26672	SOBLIDOTIN	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.2108741816694558	IUPHAR.LIGAND:77	iuphar.ligand:77	SB 714786	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.4605936073306534	FLAVOXATE	rxcui:4440	FLAVOXATE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.1902451856365742	LOSMAPIMOD	ncit:C96532	LOSMAPIMOD	FALSE	FALSE	FALSE
TSLP	hgnc:30743	TSLP	ChEMBL	33	inhibitor	52.50767123569449	TEZEPELUMAB	rxcui:2587789	TEZEPELUMAB	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TEND	1-Aug-11	NULL	0.072927321	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.2282942227638891	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	modulator	1.029562181092048	IUPHAR.LIGAND:7945	iuphar.ligand:7945	MK-2206	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:11568	iuphar.ligand:11568	LUT014	FALSE	FALSE	FALSE
NCBIGENE:2063	hgnc:7977	NR2F6	GuideToPharmacology	2024.1	modulator	3.281729452230906	IUPHAR.LIGAND:7942	iuphar.ligand:7942	REFAMETINIB	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:2000	iuphar.ligand:2000	INSL5	FALSE	FALSE	FALSE
NCBIGENE:2234	ncbigene:2234	FEB2	GuideToPharmacology	2024.1	inhibitor	5.834185692854945	IUPHAR.LIGAND:12186	iuphar.ligand:12186	AMG28	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:6389	iuphar.ligand:6389	SF-22	FALSE	FALSE	FALSE
PROSTAGLANDIN E2 RECEPTOR EP3	hgnc:9595	PTGER3	TTD	2020.06.01	NULL	3.889457128569962	ONO-9054	ncit:C152337	SEPETAPROST	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.8204323630577265	IUPHAR.LIGAND:10286	iuphar.ligand:10286	HC-070	FALSE	FALSE	FALSE
NUDT15	hgnc:23063	NUDT15	FDA	10-Apr-24	NULL	0.7955707762984016	Thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	0.062808219	IUPHAR.LIGAND:2523	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:8591	iuphar.ligand:8591	ML381	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	ChEMBL	33	inhibitor	0.3431873936973496	TANZISERTIB	ncit:C152510	TANZISERTIB	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.4861821410712453	LISDEXAMFETAMINE DIMESYLATE	rxcui:673579	LISDEXAMFETAMINE DIMESYLATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.6563458904461812	ANTIPYRINE	rxcui:1001	ANTIPYRINE	TRUE	FALSE	FALSE
RPS13	hgnc:10386	RPS13	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
BACE1	hgnc:933	BACE1	ChEMBL	33	inhibitor	4.039051633514961	LANABECESTAT	ncit:C170091	LANABECESTAT	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	SEW-03621	chembl:CHEMBL1271059	CHEMBL:CHEMBL1271059	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002359895	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	MMV007764	chembl:CHEMBL609628	CHEMBL:CHEMBL609628	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.066213961	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1888765152363111	REBASTINIB	ncit:C152162	REBASTINIB	FALSE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	MyCancerGenome	20-Jun-17	antibody	1.372749574789398	MEHD7945A	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.010195664	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	inhibitor	0.017982079	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.016748858	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	N,N-HEXAMETHYLENEAMILORIDE	iuphar.ligand:1192	5-(N,N-HEXAMETHYLENE)-AMILORIDE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.1346350544504987	CAPESEROD	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:12609	iuphar.ligand:12609	COMPOUND 30 [PMID: 37057760]	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:12720	iuphar.ligand:12720	PF-06843195	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1852122442176172	Pexidartinib	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	2.386712328895204	LINZAGOLIX	rxcui:2621019	LINZAGOLIX	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NB-ACETYLTRYPTAMINE	chembl:CHEMBL33171	NB-ACETYLTRYPTAMINE	FALSE	FALSE	FALSE
SYNDECAN-1	hgnc:10658	SDC1	TTD	2020.06.01	NULL	52.50767123569449	BT-062	ncit:C78840	INDATUXIMAB RAVTANSINE	FALSE	FALSE	FALSE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:2936	iuphar.ligand:2936	2-OLEOYL-LPA	FALSE	FALSE	FALSE
NCBIGENE:150	hgnc:281	ADRA2A	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:11279	iuphar.ligand:11279	AR234958	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:10400	iuphar.ligand:10400	PDE4 INHIBITOR 16	FALSE	FALSE	FALSE
B2M	hgnc:914	B2M	JAX-CKB	10-Apr-24	NULL	1.312691780892362	Interferon gamma	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002159654	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ESTRADIOL DIPROPIONATE	ncit:C29770	ESTRADIOL DIPROPIONATE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	AG-126	chembl:CHEMBL77387	CHEMBL:CHEMBL77387	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW876790X	chembl:CHEMBL506153	GW876790X	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003013526	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ALEXIDINE DIHYDROCHLORIDE	chembl:CHEMBL554041	ALEXIDINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
UGT1A9	hgnc:12541	UGT1A9	NCI	14-Sep-17	NULL	4.565884455277782	ALOE VERA GEL	ncit:C1565	ALOE VERA GEL	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.063110182	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NDUFS6	hgnc:7713	NDUFS6	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	positive modulator	0.3125456621172291	MIBAMPATOR	ncit:C174617	MIBAMPATOR	FALSE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.729273212	CINACIGUAT	ncit:C87280	CINACIGUAT	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:962	iuphar.ligand:962	[3H]NEMONAPRIDE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.029845209	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.1511209794852536	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.002977976	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	2.187819634820604	DEOXYCYTIDINE	rxcui:2642208	DEOXYCYTIDINE	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.017751072	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.4782119420372905	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.2557191780959147	Nirogacestat	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
IL18	hgnc:5986	IL18	NCI	14-Sep-17	NULL	0.1973972602845657	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
CDK2	hgnc:1771	CDK2	CancerCommons	25-Jul-13	inhibitor	0.073062622	BAY1000394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CancerCommons	25-Jul-13	inhibitor	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
CYP17A1	hgnc:2593	CYP17A1	CancerCommons	25-Jul-13	inhibitor	3.125456621172291	ABIRATERONE ACETATE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	CancerCommons	25-Jul-13	inhibitor	0.9907107780319716	LINSITINIB	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	CancerCommons	25-Jul-13	inhibitor	0.3697723326457359	CC-223	ncit:C92575	ONATASERTIB	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CGI	2/1/22	NULL	0.736088849	GDC-0810	ncit:C106235	BRILANESTRANT	FALSE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CGI	2/1/22	NULL	0.1372749574789398	Pertuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ERBB3	hgnc:3431	ERBB3	CGI	2/1/22	NULL	0.1372749574789398	Trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.9845188356692719	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	0.5672124979164529	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CGI	2/1/22	NULL	0.1875273972703375	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	1.064344687210023	DIPHEMANIL METHYLSULFATE	rxcui:23364	DIPHEMANIL METHYLSULFATE	TRUE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	2.917092846427472	TABIMORELIN	ncit:C76887	TABIMORELIN	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	DARIFENACIN HYDROBROMIDE	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	1.381780822	DESIRUDIN	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1935172158563679	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
LIPF	hgnc:6622	LIPF	ChEMBL	33	inhibitor	2.692701089009974	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	2.763561643983921	BIVALIRUDIN	rxcui:60819	BIVALIRUDIN	TRUE	FALSE	FALSE
F2R	hgnc:3537	F2R	ChEMBL	33	inhibitor	2.019525817	ATOPAXAR	ncit:C169794	ATOPAXAR	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	0.2019525816757481	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
HTR1F	hgnc:5292	HTR1F	ChEMBL	33	agonist	1.591141552596802	ALMOTRIPTAN MALATE	rxcui:283792	ALMOTRIPTAN MALATE	TRUE	FALSE	FALSE
AXL	hgnc:905	AXL	ChEMBL	33	inhibitor	0.172722603	GILTERITINIB	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.8899605294185507	FOSINOPRIL SODIUM	rxcui:227278	FOSINOPRIL SODIUM	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	ChEMBL	33	inhibitor	1.381780822	LEPIRUDIN	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	ANTAZOLINE PHOSPHATE	rxcui:866	ANTAZOLINE PHOSPHATE	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	0.3860858179095183	BALSALAZIDE DISODIUM	rxcui:153718	BALSALAZIDE DISODIUM	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.4189441853911795	ANISOTROPINE METHYLBROMIDE	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.022894123	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.596678082	METOPROLOL FUMARATE	rxcui:102313	METOPROLOL FUMARATE	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.2853677784548614	ACUMAPIMOD	ncit:C166567	ACUMAPIMOD	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	METOPROLOL SUCCINATE	rxcui:221124	METOPROLOL SUCCINATE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.08334551	METOCLOPRAMIDE HYDROCHLORIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.2333674277141978	ALOSETRON HYDROCHLORIDE	rxcui:85247	ALOSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	0.251232877	DONITRIPTAN	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	ChEMBL	33	inhibitor	1.346350544504987	ALLOPURINOL SODIUM	rxcui:80566	ALLOPURINOL SODIUM	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	1.458546423213736	DANAPAROID SODIUM	rxcui:103843	DANAPAROID SODIUM	TRUE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	0.3500511415712966	LINAGLIPTIN	rxcui:1100699	LINAGLIPTIN	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.2365210416022274	BUSPIRONE HYDROCHLORIDE	rxcui:203116	BUSPIRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	agonist	0.1530835896084387	RAPASTINEL	ncit:C152156	RAPASTINEL	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.4906052389860809	SUNITINIB MALATE	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.6058577450272442	DIHYDROERGOTAMINE MESYLATE	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ASPART PROTAMINE RECOMBINANT	chembl:CHEMBL1201664	INSULIN ASPART PROTAMINE RECOMBINANT	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.351221881	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	positive modulator	0.108711535	NEBOGLAMINE	ncit:C66222	NEBOGLAMINE	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN LISPRO	rxcui:2376838	INSULIN LISPRO-AABC	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1154649175056503	BUPROPION HYDROCHLORIDE	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.4907258993990139	BRETYLIUM TOSYLATE	rxcui:1737	BRETYLIUM TOSYLATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.0701037	MAPROTILINE HYDROCHLORIDE	rxcui:203126	MAPROTILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	ChEMBL	33	inhibitor	0.1446492320542548	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	inhibitor	0.092226589	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
TEK	hgnc:11724	TEK	ChEMBL	33	inhibitor	0.3977853881492008	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FDPS	hgnc:3631	FDPS	ChEMBL	33	inhibitor	1.458546423213736	ALENDRONATE SODIUM	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
PGF	hgnc:8893	PGF	ChEMBL	33	inhibitor	7.001022831425934	AFLIBERCEPT	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
FDPS	hgnc:3631	FDPS	ChEMBL	33	inhibitor	1.633571993999384	ZOLEDRONIC ACID	rxcui:1546014	ZOLEDRONIC ACID ANHYDROUS	TRUE	FALSE	TRUE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.1325951293830669	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	agonist	0.2586584789935689	RAPASTINEL	ncit:C152156	RAPASTINEL	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.3117023117067671	NALOXONE HYDROCHLORIDE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.029106248	IXABEPILONE	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.1988926940746003	ISOPROTERENOL SULFATE	rxcui:82031	ISOPROTERENOL SULFATE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.1526385791735305	GUANABENZ ACETATE	rxcui:227225	GUANABENZ ACETATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	OXAPROZIN	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.1041818873724097	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	agonist	0.108711535	APIMOSTINEL	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.089756703	PHENTOLAMINE MESYLATE	rxcui:227240	PHENTOLAMINE MESYLATE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1512704997187101	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.067231333	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1100789753368857	NICARDIPINE HYDROCHLORIDE	rxcui:235230	NICARDIPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.058277105	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.073540156	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
COL4A6	hgnc:2208	COL4A6	ChEMBL	33	cleavage	0.9376369863516874	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	agonist	0.1209854175937661	APIMOSTINEL	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
PSMC4	hgnc:9551	PSMC4	ChEMBL	33	inhibitor	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA7	hgnc:9536	PSMA7	ChEMBL	33	inhibitor	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.4773424657790409	TIPRANAVIR	rxcui:190548	TIPRANAVIR	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.2302968036653267	ATROPINE SULFATE	rxcui:153971	ATROPINE SULFATE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.3454452054979901	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
EPHA7	hgnc:3390	EPHA7	ChEMBL	33	inhibitor	0.050294704	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
EPHB3	hgnc:3394	EPHB3	ChEMBL	33	inhibitor	0.015608701	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CHRNA1	hgnc:1955	CHRNA1	ChEMBL	33	inhibitor	0.3571950424196904	VECURONIUM BROMIDE	rxcui:11153	VECURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.5357925636295356	VECURONIUM BROMIDE	rxcui:11153	VECURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	3.424413341458336	TC-6987	drugbank:DB14854	TC-6987	FALSE	FALSE	FALSE
EPHB6	hgnc:3396	EPHB6	ChEMBL	33	inhibitor	0.9053046764774914	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	0.017751072	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	0.1902451856365742	RG3487	chembl:CHEMBL2151439	RG3487	FALSE	FALSE	FALSE
EPHB2	hgnc:3393	EPHB2	ChEMBL	33	inhibitor	0.011911904	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	positive modulator	0.2885036881082115	NEBOGLAMINE	ncit:C66222	NEBOGLAMINE	FALSE	FALSE	FALSE
EPHA4	hgnc:3388	EPHA4	ChEMBL	33	inhibitor	0.9053046764774914	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NDUFA13	hgnc:17194	NDUFA13	ChEMBL	33	inhibitor	0.2344092465879218	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFV1	hgnc:7716	NDUFV1	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFS1	hgnc:7707	NDUFS1	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFAF4	hgnc:21034	NDUFAF4	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFS7	hgnc:7714	NDUFS7	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFAF2	hgnc:28086	NDUFAF2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFA4L2	hgnc:29836	NDUFA4L2	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NDUFB1	hgnc:7695	NDUFB1	ChEMBL	33	inhibitor	0.3125456621172291	METFORMIN HYDROCHLORIDE	rxcui:235743	METFORMIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ATP1A4	hgnc:14073	ATP1A4	ChEMBL	33	inhibitor	0.2917092846427472	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.030598876	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
ATP1A4	hgnc:14073	ATP1A4	ChEMBL	33	inhibitor	0.138178082	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.029465584	METHOXYFLURANE	rxcui:6857	METHOXYFLURANE	TRUE	FALSE	FALSE
ATP1B2	hgnc:805	ATP1B2	ChEMBL	33	inhibitor	0.9723642821424908	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
ATP1B3	hgnc:806	ATP1B3	ChEMBL	33	inhibitor	0.4605936073306535	DIGITOXIN	rxcui:3403	DIGITOXIN	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.069638821	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.061725319	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.06466462	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.060353645	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.067059606	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	agonist	0.036925226	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	agonist	0.1041818873724097	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	0.4565884455277783	BRADANICLINE	ncit:C169814	BRADANICLINE	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	agonist	0.039420174	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.072125922	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	agonist	0.034727296	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	agonist	0.1067229090156392	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.046965717	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	agonist	0.090452491	MEPROBAMATE	rxcui:6760	MEPROBAMATE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.054243462	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.061055432	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.021997349	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.020656047	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.061055432	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
GRIK3	hgnc:4581	GRIK3	ChEMBL	33	inhibitor	1.666910197958555	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	ChEMBL	33	inhibitor	0.064944553	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.1136529680426287	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	GENTAMICIN SULFATE	rxcui:1870193	GENTAMICIN SULFATE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.050007306	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	modulator	0.027929612	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	ChEMBL	33	modulator	0.1230648544586589	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	modulator	0.082043236	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
KCNK10	hgnc:6273	KCNK10	ChEMBL	33	potentiator	0.3387591692625452	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.1767935058440892	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	QUINIDINE POLYGALACTURONATE	rxcui:41875	QUINIDINE POLYGALACTURONATE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.087512785	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	MEXILETINE HYDROCHLORIDE	rxcui:142138	MEXILETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	0.2651902587661338	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.021933029	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.019233579	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.020164236	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.018799739	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.012756966	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.017859752	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.017283631	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.458546423213736	AZD1446	chembl:CHEMBL2179529	AZD1446	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.080781033	LABETALOL HYDROCHLORIDE	rxcui:202693	LABETALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.060772768	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.045791574	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.060585775	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.082171629	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.084553416	MEPHENTERMINE SULFATE	rxcui:82042	MEPHENTERMINE SULFATE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.08334551	DROPERIDOL	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inverse agonist	0.051885051	HALOPERIDOL LACTATE	rxcui:217483	HALOPERIDOL LACTATE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inverse agonist	0.1250182648468916	HALOPERIDOL LACTATE	rxcui:217483	HALOPERIDOL LACTATE	TRUE	FALSE	FALSE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	2.500365296937833	PARAMETHADIONE	rxcui:32894	PARAMETHADIONE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.1519026168824334	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.1744440904840348	MIBEFRADIL DIHYDROCHLORIDE	rxcui:83214	MIBEFRADIL DIHYDROCHLORIDE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	1.000146118775133	JNJ-38877605	drugbank:DB13113	JNJ-38877605	FALSE	FALSE	FALSE
RAF1	hgnc:9829	RAF1	ChEMBL	33	inhibitor	0.6731752722524935	LY-3009120	chembl:CHEMBL3545195	LY-3009120	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.1000146118775133	MERESTINIB	ncit:C95729	MERESTINIB	FALSE	FALSE	FALSE
NDUFS8	hgnc:7715	NDUFS8	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	LY-3007113	chembl:CHEMBL3544998	LY-3007113	FALSE	FALSE	FALSE
MT-ND6	hgnc:7462	MT-ND6	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB7	hgnc:7702	NDUFB7	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.041021618	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.5834185692854944	MK-1496	drugbank:DB12763	MK-1496	FALSE	FALSE	FALSE
NDUFA2	hgnc:7685	NDUFA2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFAF3	hgnc:29918	NDUFAF3	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFS3	hgnc:7710	NDUFS3	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFB2	hgnc:7697	NDUFB2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFC2	hgnc:7706	NDUFC2	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFAF4	hgnc:21034	NDUFAF4	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFA7	hgnc:7691	NDUFA7	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFAB1	hgnc:7694	NDUFAB1	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NDUFB8	hgnc:7703	NDUFB8	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFA9	hgnc:7693	NDUFA9	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFA3	hgnc:7686	NDUFA3	ChEMBL	33	inhibitor	0.3431873936973497	ME-344	drugbank:DB13062	ME-344	FALSE	FALSE	FALSE
NDUFAF3	hgnc:29918	NDUFAF3	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFB11	hgnc:20372	NDUFB11	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA3	hgnc:7686	NDUFA3	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFS3	hgnc:7710	NDUFS3	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA4L2	hgnc:29836	NDUFA4L2	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFB4	hgnc:7699	NDUFB4	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
NDUFA5	hgnc:7688	NDUFA5	ChEMBL	33	inhibitor	0.3500511415712966	NV-128	chembl:CHEMBL3545135	NV-128	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.1470803115845784	RG-547	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.063415062	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	2.625383561784724	VICRIVIROC MALEATE	ncit:C73146	VICRIVIROC MALEATE	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	0.8468979231563628	TRICETAMIDE	ncit:C74378	TRICETAMIDE	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1666910197958555	PWT-33587	chembl:CHEMBL3545006	PWT-33587	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	S-222611	chembl:CHEMBL3545200	S-222611	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.1136529680426287	ZOTIRACICLIB	ncit:C171725	ZOTIRACICLIB	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.095122593	ZOTIRACICLIB	ncit:C171725	ZOTIRACICLIB	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	4.565884455277782	ZIBOTENTAN	ncit:C48430	ZIBOTENTAN	FALSE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.3500511415712966	ZOTIRACICLIB	ncit:C171725	ZOTIRACICLIB	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.3241214273808302	ZOTIRACICLIB	ncit:C171725	ZOTIRACICLIB	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	HEMAY-022	chembl:CHEMBL3545111	HEMAY-022	FALSE	FALSE	FALSE
CCR9	hgnc:1610	CCR9	ChEMBL	33	inhibitor	26.25383561784724	MLN3126	chembl:CHEMBL3545268	MLN3126	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	IRDABISANT	ncit:C170078	IRDABISANT	FALSE	FALSE	FALSE
BDKRB1	hgnc:1029	BDKRB1	ChEMBL	33	inhibitor	5.834185692854944	BI113823	chembl:CHEMBL3545386	BI113823	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.7095631248066824	PBF-999	iuphar.ligand:13188	PBF-999	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.064347636	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1223955040459079	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	ChEMBL	33	inhibitor	2.500365296937833	IMD-2560	chembl:CHEMBL3545147	IMD-2560	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	1.141471113819445	TEZOSENTAN	ncit:C97358	TEZOSENTAN	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.075768645	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.033615667	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
PRKCB	hgnc:9395	PRKCB	ChEMBL	33	inhibitor	0.1930429089547592	CEP-2563	chembl:CHEMBL3545332	CEP-2563	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1363835616511545	PUQUITINIB	ncit:C162555	PUQUITINIB	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.062509132	NKTR-171	chembl:CHEMBL3545209	NKTR-171	FALSE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.092606122	ELPETRIGINE	ncit:C166519	ELPETRIGINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	ChEMBL	33	inhibitor	0.2083637747448194	BI-2536	iuphar.ligand:5666	BI-2536	FALSE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.6000876712650799	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.023780648	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1875273972703374	FAMITINIB	ncit:C97512	FAMITINIB	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.064111931	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.5469549087051511	TONAPOFYLLINE	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1111273465305703	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.2035181055647073	FADOLMIDINE HYDROCHLORIDE	ncit:C77297	FADOLMIDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	inhibitor	2.100306849	BALIXAFORTIDE	ncit:C91094	BALIXAFORTIDE	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	blocker	0.577007376	LANICEMINE	ncit:C77601	LANICEMINE	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.6908904109959803	PF-04531083	drugbank:DB12468	PF-04531083	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	positive modulator	0.4234489615781814	FARAMPATOR	ncit:C65620	FARAMPATOR	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.3182283105193605	SEMAGLUTIDE	rxcui:1991302	SEMAGLUTIDE	TRUE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.3125456621172291	BECAMPANEL	ncit:C79860	BECAMPANEL	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	inverse agonist	0.040021091	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	agonist	0.03729238	ADIPIPLON	ncit:C76933	ADIPIPLON	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	inverse agonist	0.036062961	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	LOREDIPLON	ncit:C170129	LOREDIPLON	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	inverse agonist	0.044347695	RESEQUINIL	chembl:CHEMBL2107801	RESEQUINIL	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.4861821410712454	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	ChEMBL	33	inhibitor	0.1037701012563132	BARICITINIB	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	ChEMBL	33	inhibitor	0.2983390411119005	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	2.282942227638891	CLAZOSENTAN	ncit:C79486	CLAZOSENTAN	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.082171629	CEBRANOPADOL	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.053524639	CEBRANOPADOL	ncit:C112002	CEBRANOPADOL	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inverse agonist	0.463302981	PITOLISANT	rxcui:2197878	PITOLISANT	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	1.591141552596803	ZOPTARELIN DOXORUBICIN	ncit:C74025	ZOPTARELIN DOXORUBICIN	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	ChEMBL	33	agonist	1.071585127259071	BREMELANOTIDE	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	ChEMBL	33	other/unknown	22.50328767	OREGOVOMAB	ncit:C1784	OREGOVOMAB	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.5645986154375752	NERELIMOMAB	ncit:C166480	NERELIMOMAB	FALSE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	other/unknown	9.845188356692718	ZANOLIMUMAB	ncit:C91701	ZANOLIMUMAB	FALSE	FALSE	FALSE
CA9	hgnc:1383	CA9	ChEMBL	33	binder	3.750547945	CG250 177LU	chembl:CHEMBL3707297	CG250 177LU	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.042689164	PACLITAXEL POLIGLUMEX	rxcui:2473230	PACLITAXEL POLIGLUMEX	FALSE	FALSE	FALSE
TLR3	hgnc:11849	TLR3	ChEMBL	33	agonist	10.50153424713889	RINTATOLIMOD	ncit:C1001	RINTATOLIMOD	FALSE	FALSE	FALSE
IL10RB	hgnc:5965	IL10RB	ChEMBL	33	agonist	5.834185692854944	PEGINTERFERON LAMBDA-1A	ncit:C166435	PEGINTERFERON LAMBDA-1A	FALSE	FALSE	FALSE
METAP1	hgnc:15789	METAP1	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
ALOX5AP	hgnc:436	ALOX5AP	ChEMBL	33	inhibitor	7.501095891	FIBOFLAPON	ncit:C169978	FIBOFLAPON	FALSE	FALSE	FALSE
NPEPL1	hgnc:16244	NPEPL1	ChEMBL	33	inhibitor	2.625383561784725	TOSEDOSTAT	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	8.204323630577266	UDENAFIL	ncit:C74086	UDENAFIL	TRUE	FALSE	FALSE
PSMB9	hgnc:9546	PSMB9	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMA8	hgnc:22985	PSMA8	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMA2	hgnc:9531	PSMA2	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
PSMB3	hgnc:9540	PSMB3	ChEMBL	33	inhibitor	0.4167275494896388	MARIZOMIB	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.1810609352954982	RETASPIMYCIN HYDROCHLORIDE	ncit:C48401	RETASPIMYCIN HYDROCHLORIDE	FALSE	FALSE	TRUE
CD40	hgnc:11919	CD40	ChEMBL	33	inhibitor	4.375639269641208	DACETUZUMAB	ncit:C62179	DACETUZUMAB	FALSE	FALSE	FALSE
CD74	hgnc:1697	CD74	ChEMBL	33	inhibitor	52.50767123569449	MILATUZUMAB	ncit:C66983	MILATUZUMAB	FALSE	TRUE	TRUE
KIR2DL3	hgnc:6331	KIR2DL3	ChEMBL	33	inhibitor	7.876150685354174	IPH-2101	hemonc:260	IPH-2101	FALSE	FALSE	FALSE
IGHE	hgnc:5522	IGHE	ChEMBL	33	inhibitor	8.751278539282415	AL-901	chembl:CHEMBL2109455	AL-901	FALSE	FALSE	FALSE
TPH2	hgnc:20692	TPH2	ChEMBL	33	inhibitor	1.458546423213736	TELOTRISTAT ETHYL	rxcui:1872441	TELOTRISTAT ETHYL	TRUE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	agonist	0.1816874437221263	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	agonist	0.2059124362184098	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR5A	hgnc:5300	HTR5A	ChEMBL	33	agonist	0.7721716358190368	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	ChEMBL	33	agonist	0.1029562181092049	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	inhibitor	0.5000730593875666	DILEVALOL HYDROCHLORIDE	ncit:C174786	DILEVALOL HYDROCHLORIDE	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.6731752722524935	MEBANAZINE	ncit:C80969	MEBANAZINE	TRUE	FALSE	FALSE
MALT1	hgnc:6819	MALT1	ChEMBL	33	inhibitor	17.50255707856483	MEPAZINE ACETATE	chembl:CHEMBL1712842	MEPAZINE ACETATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.2187819634820604	IBUFENAC	ncit:C96750	IBUFENAC	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.022889133	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	ChEMBL	33	binder	3.750547945	IGOVOMAB	ncit:C188577	IGOVOMAB	TRUE	FALSE	FALSE
ITGA4	hgnc:6140	ITGA4	ChEMBL	33	inhibitor	3.889457128569962	ABRILUMAB	ncit:C139025	ABRILUMAB	FALSE	FALSE	FALSE
ITGB7	hgnc:6162	ITGB7	ChEMBL	33	inhibitor	5.834185692854944	ABRILUMAB	ncit:C139025	ABRILUMAB	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	ACEMETACIN	rxcui:16695	ACEMETACIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.02505934	CYPROTERONE ACETATE	rxcui:22054	CYPROTERONE ACETATE	TRUE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	CORTIVAZOL	rxcui:21660	CORTIVAZOL	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.090064616	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.1136529680426287	CINNARIZINE	rxcui:2549	CINNARIZINE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.0701037	DEBRISOQUIN	rxcui:3118	DEBRISOQUIN	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.086551106	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	blocker	0.1209854175937661	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.07631929	CELIPROLOL	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	blocker	0.1693795846312726	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.014617949	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
PTH1R	hgnc:9608	PTH1R	ChEMBL	33	agonist	3.750547945	ABALOPARATIDE	rxcui:1921069	ABALOPARATIDE	TRUE	FALSE	FALSE
PAGA	hgnc:9352	PRDX1	ChEMBL	33	inhibitor	8.751278539282415	MDX-1303	drugbank:DB05945	MDX-1303	FALSE	FALSE	FALSE
TRBV7-9	hgnc:12243	TRBV7-9	ChEMBL	33	inhibitor	4.375639269641208	MASLIMOMAB	ncit:C188519	MASLIMOMAB	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	modulator	0.525076712	IMC-GP100	chembl:CHEMBL2109434	IMC-GP100	FALSE	FALSE	FALSE
CD6	hgnc:1691	CD6	ChEMBL	33	inhibitor	52.50767123569449	ITOLIZUMAB	ncit:C95787	ITOLIZUMAB	FALSE	FALSE	FALSE
TNFSF12	hgnc:11927	TNFSF12	ChEMBL	33	inhibitor	78.76150685354175	RO-5458640	chembl:CHEMBL2109600	RO-5458640	FALSE	FALSE	FALSE
PDCD1LG2	hgnc:18731	PDCD1LG2	ChEMBL	33	modulator	26.25383561784724	RHIGM12B7	chembl:CHEMBL2109309	RHIGM12B7	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.03043923	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	OZENOXACIN	rxcui:1994739	OZENOXACIN	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.03043923	DOXYCYCLINE HYCLATE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.053361455	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
BHMT	hgnc:1047	BHMT	ChEMBL	33	other/unknown	5.250767124	BETAINE	rxcui:1512	BETAINE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.055387839	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
KCND3	hgnc:6239	KCND3	ChEMBL	33	blocker	0.1600843635234588	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNA3	hgnc:6221	KCNA3	ChEMBL	33	blocker	0.1829535583125243	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
KCNA7	hgnc:6226	KCNA7	ChEMBL	33	blocker	0.2134458180312784	AMIFAMPRIDINE PHOSPHATE	rxcui:2106337	AMIFAMPRIDINE PHOSPHATE	TRUE	FALSE	FALSE
IFNAR2	hgnc:5433	IFNAR2	ChEMBL	33	positive modulator	0.8204323630577265	ROPEGINTERFERON ALFA-2B	rxcui:2587059	ROPEGINTERFERON ALFA-2B	TRUE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.7001022831425934	PRALICIGUAT	ncit:C174906	PRALICIGUAT	FALSE	FALSE	FALSE
GUCY1A1	hgnc:4685	GUCY1A1	ChEMBL	33	activator	0.8751278539282416	CINACIGUAT	ncit:C87280	CINACIGUAT	FALSE	FALSE	FALSE
ATP2A3	hgnc:813	ATP2A3	ChEMBL	33	inhibitor	1.093909817410302	MIPSAGARGIN	ncit:C90554	MIPSAGARGIN	FALSE	FALSE	FALSE
PPIA	hgnc:9253	PPIA	ChEMBL	33	inhibitor	7.501095891	SCY 635	chembl:CHEMBL1269597	SCY 635	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	agonist	5.834185692854944	TZP-102	drugbank:DB16129	TZP-102	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
CD40	hgnc:11919	CD40	ChEMBL	33	inhibitor	2.187819634820604	ISCALIMAB	ncit:C175096	ISCALIMAB	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	NAVAFENTEROL	ncit:C174920	NAVAFENTEROL	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	GSK-256066	drugbank:DB12137	GSK-256066	FALSE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	BISEGLIPTIN	ncit:C171768	BISEGLIPTIN	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.5834185692854944	MK-0873	drugbank:DB13029	MK-0873	FALSE	FALSE	FALSE
RPS19	hgnc:10402	RPS19	ChEMBL	33	modulator	0.050488145	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPS20	hgnc:10405	RPS20	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL9P9	hgnc:30334	RPL9P8	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL9P8	hgnc:30334	RPL9P8	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL19	hgnc:10312	RPL19	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL7A	hgnc:10364	RPL7A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL13	hgnc:10303	RPL13	ChEMBL	33	modulator	0.093763699	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL32	hgnc:10336	RPL32	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL13A	hgnc:10304	RPL13A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.033487035	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.036463661	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.182318303	BUNAZOSIN	rxcui:19850	BUNAZOSIN	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	modulator	1.312691780892362	AFELETECAN	ncit:C79725	AFELETECAN	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.640864726115453	IPRAGLIFLOZIN	ncit:C166685	IPRAGLIFLOZIN	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	ChEMBL	33	inhibitor	2.763561643983921	CONCIZUMAB	ncit:C166914	CONCIZUMAB	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	ABIVERTINIB MALEATE	ncit:C169756	ABIVERTINIB MALEATE	FALSE	FALSE	FALSE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	0.9376369863516875	APROCITENTAN	ncit:C174728	APROCITENTAN	TRUE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	ChEMBL	33	negative modulator	1.750255707856483	NIMACIMAB	ncit:C175163	NIMACIMAB	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	3.500511415712966	POZELIMAB	rxcui:2663938	POZELIMAB	TRUE	FALSE	FALSE
EPHX2	hgnc:3402	EPHX2	ChEMBL	33	inhibitor	2.250328767244049	AR9281	drugbank:DB06345	AR-9281	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.295540363	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.1223955040459079	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.2983390411119005	XAMOTEROL	rxcui:39801	XAMOTEROL	TRUE	FALSE	FALSE
GPR119	hgnc:19060	GPR119	ChEMBL	33	agonist	17.50255707856483	MBX-2982	drugbank:DB12345	MBX-2982	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.3365876361262467	ABEXINOSTAT	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
ATP2A2	hgnc:812	ATP2A2	ChEMBL	33	activator	0.5073204950308647	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
FXYD2	hgnc:4026	FXYD2	ChEMBL	33	inhibitor	0.4861821410712454	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
CXCR2	hgnc:6027	CXCR2	ChEMBL	33	inhibitor	1.458546423213736	SX-682	chembl:CHEMBL4297480	SX-682	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.069454592	KBP5209	chembl:CHEMBL4650289	KBP5209	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	ChEMBL	33	inhibitor	1.981421556063943	GIMERACIL	ncit:C2416	GIMERACIL	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	FLOTETUZUMAB	ncit:C117238	FLOTETUZUMAB	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.6250913242344582	FIPAMEZOLE	ncit:C65684	FIPAMEZOLE	FALSE	FALSE	FALSE
TBXA2R	hgnc:11608	TBXA2R	ChEMBL	33	inhibitor	0.9376369863516875	PICOTAMIDE	ncit:C73157	PICOTAMIDE	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	agonist	0.7684049449126024	RESINIFERATOXIN	ncit:C1214	RESINIFERATOXIN	FALSE	FALSE	FALSE
FGB	hgnc:3662	FGB	ChEMBL	33	positive modulator	1.166837138570988	FIBRINOGEN, HUMAN	rxcui:2264108	FIBRINOGEN, HUMAN	TRUE	FALSE	FALSE
F8	hgnc:3546	F8	ChEMBL	33	positive modulator	3.088686543276147	GIROCTOCOGENE FITELPARVOVEC	ncit:C174651	GIROCTOCOGENE FITELPARVOVEC	FALSE	FALSE	FALSE
FGG	hgnc:3694	FGG	ChEMBL	33	positive modulator	2.187819634820604	FIBRINOGEN, HUMAN	rxcui:2264108	FIBRINOGEN, HUMAN	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
ROR1	hgnc:10256	ROR1	ChEMBL	33	inhibitor	52.50767123569449	CIRMTUZUMAB	chembl:CHEMBL4297728	CIRMTUZUMAB	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	PRALUZATAMAB RAVTANSINE	ncit:C134697	PRALUZATAMAB RAVTANSINE	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	CENSAVUDINE	ncit:C166942	CENSAVUDINE	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	1.458546423213736	DIANICLINE	ncit:C76073	DIANICLINE	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.2333674277141978	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.2500365296937833	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	ChEMBL	33	activator	0.2344092465879218	ACADESINE	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
PRKAB1	hgnc:9378	PRKAB1	ChEMBL	33	activator	0.9376369863516874	ACADESINE	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2386712328895204	ROLIPRAM	ncit:C72842	ROLIPRAM	FALSE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	ChEMBL	33	activator	1.363835616511545	ACADESINE	ncit:C71537	ACADESINE	FALSE	FALSE	FALSE
MPL	hgnc:7217	MPL	ChEMBL	33	agonist	4.773424657790408	HETROMBOPAG OLAMINE	ncit:C173439	HETROMBOPAG OLAMINE	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	ZURANOLONE	rxcui:2669905	ZURANOLONE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.037734582	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	ChEMBL	33	inhibitor	0.2804896967718723	VALSPODAR	ncit:C1405	VALSPODAR	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	inhibitor	4.375639269641208	GATIPOTUZUMAB	ncit:C94220	GATIPOTUZUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	1.336059069138614	TRAMETINIB	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3923362732430473	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	ClearityFoundationBiomarkers	26-Jul-13	NULL	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.4782119420372905	MEGESTROL ACETATE	rxcui:29451	MEGESTROL ACETATE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.072927321	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.4167275494896389	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.6482428547616604	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.049275217	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
AKT1	hgnc:391	AKT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.443726799	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3697723326457359	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.0403388	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
FOLH1	hgnc:3788	FOLH1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.046860929	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1008469998124734	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NTSR1	hgnc:8039	NTSR1	ChEMBL	33	inhibitor	5.834185692854944	REMINERTANT	ncit:C156766	MECLINERTANT	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.093098708	CYSTAMINE	rxcui:1426401	CYSTAMINE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013192882	OXIDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.087629625	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.009430257	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	DEGUELIN	ncit:C63666	DEGUELIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005315618	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	TRIMETAZIDINE	rxcui:10826	TRIMETAZIDINE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.085796848	DIAMIDE	chembl:CHEMBL1255835	DIAMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	1-[2-(TRIFLUOROMETHYL)PHENYL]IMIDAZOLE	iuphar.ligand:4331	TRIM	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-4809	chembl:CHEMBL585439	CHEMBL:CHEMBL585439	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	ICI-199,441	iuphar.ligand:11691	ICI-199441	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003001553	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	FERROUS SULFATE	rxcui:24947	FERROUS SULFATE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	LAVENDUSTIN C	ncit:C1487	LAVENDUSTIN C	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	URAPIDIL	rxcui:39230	URAPIDIL	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.005497034	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00487265	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.024932417	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1988926940746003	TRACAZOLATE	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	TCMDC-124059	chembl:CHEMBL530733	CHEMBL:CHEMBL530733	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-742864	chembl:CHEMBL103080	CHEMBL:CHEMBL103080	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.4717670371580817	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	LINOPIRDINE	ncit:C82306	LINOPIRDINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003541833	RALOXIFENE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.032412143	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	DNDI1417080	chembl:CHEMBL1498652	CHEMBL:CHEMBL1498652	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	IPCONAZOLE	chembl:CHEMBL3185422	IPCONAZOLE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00684585	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.073954467	THUNBERGINOL B	chembl:CHEMBL70501	THUNBERGINOL B	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	ARACHIDONYL TRIFLUOROMETHYLKETONE	iuphar.ligand:5142	ARACHIDONYL TRIFLUOROMETHYL KETONE	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.1207072901969988	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.000747185	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	DESONIDE	rxcui:3254	DESONIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	GNF-PF-5183	chembl:CHEMBL577660	CHEMBL:CHEMBL577660	FALSE	FALSE	FALSE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	0.106290832	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.008188969	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.1159109740302306	PROFLAVINE	rxcui:8723	PROFLAVINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.4070362111294147	DICHLOROISOPROTERENOL	drugbank:DB12803	DICHLOROISOPROTERENOL	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.030246354	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	1-BENZYLMALEIMIDE	chembl:CHEMBL388979	CHEMBL:CHEMBL388979	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006439499	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ROCAGLAMIDE	drugbank:DB15495	ROCAGLAMIDE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.03262504	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	TCMDC-124447	chembl:CHEMBL587229	CHEMBL:CHEMBL587229	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	TCMDC-124479	chembl:CHEMBL587259	CHEMBL:CHEMBL587259	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	PAPAVERINE HYDROCHLORIDE	rxcui:203132	PAPAVERINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	2,4-DIMETHYLPHENOL	chembl:CHEMBL29878	CHEMBL:CHEMBL29878	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV274073	chembl:CHEMBL1740701	CHEMBL:CHEMBL1740701	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	BENZETHONIUM	rxcui:1390	BENZETHONIUM	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.016327012	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
S1PR4	hgnc:3170	S1PR4	DTC	9/2/20	NULL	0.2243917574174979	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.08914715	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.043109746	7-NITROINDAZOLE	drugbank:DB02207	7-NITROINDAZOLE	FALSE	FALSE	FALSE
HSP90	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.7242437411819931	EFUNGUMAB	ncit:C87763	EFUNGUMAB	FALSE	FALSE	FALSE
PRSS2	hgnc:9483	PRSS2	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.059297201	LUMATEPERONE	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	1.842374429322613	SETIPIPRANT	ncit:C152348	SETIPIPRANT	FALSE	FALSE	FALSE
NGF	hgnc:7808	NGF	ChEMBL	33	inhibitor	22.50328767	TANEZUMAB	ncit:C71522	TANEZUMAB	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.050246575	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	TYRPHOSTIN AG-1478	iuphar.ligand:4862	AG1478	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
CASP7	hgnc:1508	CASP7	DTC	9/2/20	NULL	0.5147810905460244	3-HYDROXYANTHRANILIC ACID	drugbank:DB03644	3-HYDROXYANTHRANILIC ACID	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.035719504	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	DOLASTATIN 12	chembl:CHEMBL448114	DOLASTATIN 12	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	(S)-3,5-DIHYDROXYPHENYLGLYCINE	drugbank:DB04228	DIHYDROXYPHENYLGLYCINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	chembl:CHEMBL284028	2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.002214392	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	TCMDC-124422	chembl:CHEMBL527620	CHEMBL:CHEMBL527620	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.2845944240417046	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.078958904	SB-222200	iuphar.ligand:2131	SB 222200	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GNF-PF-2094	chembl:CHEMBL578928	CHEMBL:CHEMBL578928	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	NAFTOPIDIL	ncit:C72927	NAFTOPIDIL	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.1117184494376478	7-HYDROXY ISOFLAVONE	chembl:CHEMBL491981	7-HYDROXY ISOFLAVONE	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	ChEMBL	33	inhibitor	0.2476776945079929	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
HRH4	hgnc:17383	HRH4	DTC	9/2/20	NULL	1.790034246671403	THIOPERAMIDE	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
PARP1	hgnc:270	PARP1	ChEMBL	33	inhibitor	0.3818739726232327	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
TXK	hgnc:12434	TXK	DTC	9/2/20	inhibitor	0.6563458904461813	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	SB-222200	iuphar.ligand:2131	SB 222200	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.05664258	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	OBTUSAQUINONE	chembl:CHEMBL1333653	OBTUSAQUINONE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
RHD	hgnc:10009	RHD	ChEMBL	33	other/unknown	13.12691780892362	ATOROLIMUMAB	ncit:C188669	ATOROLIMUMAB	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011049594	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.9907107780319716	AVE-1642	chembl:CHEMBL2109357	AVE-1642	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	1.009762908	TARANABANT	ncit:C81420	TARANABANT	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.2568509424527334	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.1262203635473425	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.032412143	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
KIR2DL1	hgnc:6329	KIR2DL1	ChEMBL	33	inhibitor	4.375639269641208	LIRILUMAB	ncit:C103820	LIRILUMAB	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.036212187	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	TCMDC-123762	chembl:CHEMBL547483	CHEMBL:CHEMBL547483	FALSE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	3.088686543276147	NSC-640556	chembl:CHEMBL1983317	CHEMBL:CHEMBL1983317	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	GALANGIN	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.009053047	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.075768645	JNK INHIBITOR VIII	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	DEFERIPRONE	rxcui:11645	DEFERIPRONE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01715937	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
TSPO	hgnc:1158	TSPO	ChEMBL	33	agonist	2.763561643983921	ALPIDEM	ncit:C80669	ALPIDEM	TRUE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.045265234	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	QUESTIOMYCIN B	chembl:CHEMBL28319	QUESTIOMYCIN B	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	1.981421556063943	BROMOPYROGALLOL RED	chembl:CHEMBL210287	BROMOPYROGALLOL RED	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.014330696	SENNOSIDE B	rxcui:56161	SENNOSIDE B	FALSE	FALSE	FALSE
EP300	hgnc:3373	EP300	DTC	9/2/20	NULL	5.834185692854944	DIETHYL-2-UNDECYLIDENEMALONATE	chembl:CHEMBL1797707	CHEMBL:CHEMBL1797707	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.032412143	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	EMETINE DIHYDROCHLORIDE	chembl:CHEMBL493439	EMETINE HYDROCHLORIDE	FALSE	FALSE	FALSE
TRPV4	hgnc:18083	TRPV4	ChEMBL	33	inhibitor	0.3241214273808302	BUTAMBEN	rxcui:19861	BUTAMBEN	TRUE	FALSE	FALSE
GPER1	hgnc:4485	GPER1	DTC	9/2/20	NULL	1.117184494376478	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE	iuphar.ligand:5445	N-DOCOSATETRA-7,10,13,16-ENOYLETHANOLAMINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
CYBB	hgnc:2578	CYBB	DTC	9/2/20	NULL	1.875273972703374	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1861974157294131	D-64131	chembl:CHEMBL140220	CHEMBL:CHEMBL140220	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.059667808	DIPYRONE	rxcui:1537943	METAMIZOLE SODIUM	TRUE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.02234369	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009579944	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.019607047	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.097236428	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.00279415	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.006487234	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.028413242	CHRYSIN	rxcui:1362888	CHRYSIN	TRUE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	6.177373086552294	PF-06465469	chembl:CHEMBL2179805	CHEMBL:CHEMBL2179805	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	LAVENDUSTIN C	ncit:C1487	LAVENDUSTIN C	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.039778539	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.2075402025126264	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	L-THREO-BENZYLOXY ASPARTATE	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.01715937	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	DNDI1417155	chembl:CHEMBL1548739	CHEMBL:CHEMBL1548739	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.2386712328895204	ISOXICAM	ncit:C80558	ISOXICAM	TRUE	FALSE	FALSE
PPP1CA	hgnc:9281	PPP1CA	DTC	9/2/20	NULL	5.250767123569449	DEMETHYL-CANTHARIDIN	chembl:CHEMBL8327	DEMETHYL-CANTHARIDIN	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	GNF-PF-3501	chembl:CHEMBL581910	CHEMBL:CHEMBL581910	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.072324616	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.036062961	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.364636606	GNF-PF-5159	chembl:CHEMBL1493528	CHEMBL:CHEMBL1493528	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	2.386712328895204	HEXAHYDROCURCUMIN	chembl:CHEMBL479650	HEXAHYDROCURCUMIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PERBROMOBENZENE	chembl:CHEMBL375600	PERBROMOBENZENE	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.063415062	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	2'-HYDROXYCHALCONE	chembl:CHEMBL32147	2'-HYDROXYCHALCONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003063458	CLOMETHIAZOLE	rxcui:2372	CHLORMETHIAZOLE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.08178765	CUMENE HYDROPEROXIDE	chembl:CHEMBL1518369	CUMENE HYDROPEROXIDE	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.008496387	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
RGS12	hgnc:9994	RGS12	DTC	9/2/20	NULL	2.187819634820604	LAVENDUSTIN C	ncit:C1487	LAVENDUSTIN C	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	(R)-SARGACHROMENOL	chembl:CHEMBL1668777	(R)-SARGACHROMENOL	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.024547766	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	(S)-FELODIPINE	chembl:CHEMBL428768	(S)-FELODIPINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.6035364509849942	DINOPROST TROMETHAMINE	rxcui:23321	DINOPROST TROMETHAMINE	TRUE	FALSE	FALSE
MARK4	hgnc:13538	MARK4	DTC	9/2/20	inhibitor	0.2187819634820604	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.0296486	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	DTC	9/2/20	NULL	0.1312691780892362	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.050781113	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1193356164447602	NOMIFENSINE MALEATE	rxcui:262302	NOMIFENSINE MALEATE	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.1426838892274307	CLOFIBRATE	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
EPHA6	hgnc:19296	EPHA6	DTC	9/2/20	inhibitor	0.2625383561784725	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	PAPAVERINE HYDROCHLORIDE	rxcui:203132	PAPAVERINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004384042	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	1.500219178	NSC-73753	chembl:CHEMBL1506226	CHEMBL:CHEMBL1506226	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	CID 695758	chembl:CHEMBL260028	CHEMBL:CHEMBL260028	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005308631	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.2983390411119005	PRONETALOL	ncit:C82257	PRONETALOL	TRUE	FALSE	FALSE
TYR	hgnc:12442	TYR	DTC	9/2/20	NULL	7.160136986685614	KOJIC ACID	rxcui:1426451	KOJIC ACID	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.033148782	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	BENZOTHIAZYL DISULFIDE	chembl:CHEMBL508112	BENZOTHIAZYL DISULFIDE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.1187188949127459	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.016764901	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	ZINC 03369470	chembl:CHEMBL599013	CHEMBL:CHEMBL599013	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	FUTUXIMAB	ncit:C152971	FUTUXIMAB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006434764	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
CLK1	hgnc:2068	CLK1	DTC	9/2/20	NULL	3.500511415712966	NU-2058	chembl:CHEMBL269881	CHEMBL:CHEMBL269881	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	CARMINOMYCIN	ncit:C352	CARUBICIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124653	chembl:CHEMBL533921	CHEMBL:CHEMBL533921	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	KETANSERIN TARTRATE	ncit:C2036	KETANSERIN TARTRATE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	GNF-PF-254	iuphar.ligand:5919	AKT INHIBITOR IV	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.030814361	LOPERAMIDE	rxcui:6468	LOPERAMIDE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.014002046	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.1193356164447602	CEPHALOTHIN	rxcui:2236	CEPHALOTHIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.068907705	REVERSETRIIODOTHYRONINE	iuphar.ligand:2636	RT3	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004674828	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.006265084	DOPAMINE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	PHENSERINE	drugbank:DB04892	PHENSERINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	MACLURAXANTHONE	chembl:CHEMBL478960	MACLURAXANTHONE	FALSE	FALSE	FALSE
GPA33	hgnc:4445	GPA33	ChEMBL	33	binder	13.12691780892362	A33 131I	chembl:CHEMBL2109642	A33 131I	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2328499833068492	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2651902587661338	4-(4-AMINOPHENYL)BUTANOIC ACID	chembl:CHEMBL1650245	CHEMBL:CHEMBL1650245	FALSE	FALSE	FALSE
ACVRL1	hgnc:175	ACVRL1	DTC	9/2/20	inhibitor	0.1458546423213736	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	P-1075	chembl:CHEMBL11458	CHEMBL:CHEMBL11458	FALSE	FALSE	FALSE
PLD2	hgnc:9068	PLD2	DTC	9/2/20	NULL	0.5385402178019949	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	L-THREO-BENZYLOXY ASPARTATE	iuphar.ligand:4631	DL-TBOA	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.023823807	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	DTC	9/2/20	NULL	3.621218705909965	CASEARINOL B	chembl:CHEMBL459192	CASEARINOL B	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	BENZAMIL HYDROCHLORIDE	chembl:CHEMBL1256878	BENZAMIL HYDROCHLORIDE	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.3621218705909966	5-FLUOROURIDINE	drugbank:DB01629	5-FLUOROURIDINE	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	0.8751278539282418	NILE RED	chembl:CHEMBL144472	NILE RED	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	ETHYLESTRENOL	rxcui:4162	ETHYLESTRENOL	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	PHENAMIL	iuphar.ligand:4281	PHENAMIL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	TELOMESTATIN	chembl:CHEMBL443683	TELOMESTATIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	5,7-DIMETHOXYISOFLAVONE	chembl:CHEMBL308688	5,7-DIMETHOXYISOFLAVONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003217973	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.039899446	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	ChEMBL	33	inhibitor	0.7501095890813501	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	GNF-PF-3876	chembl:CHEMBL596631	CHEMBL:CHEMBL596631	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.099071078	2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE	chembl:CHEMBL201325	CHEMBL:CHEMBL201325	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	ChEMBL	33	inhibitor	0.729273212	BUTAMBEN	rxcui:19861	BUTAMBEN	TRUE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	ChEMBL	33	inhibitor	0.3590268118679965	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
ICAM1	hgnc:5344	ICAM1	ChEMBL	33	inhibitor	8.751278539282415	ENLIMOMAB	ncit:C188612	ENLIMOMAB	FALSE	FALSE	FALSE
IL3RA	hgnc:6012	IL3RA	ChEMBL	33	inhibitor	5.250767123569449	CSL-360	chembl:CHEMBL2109327	CSL-360	FALSE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	DTC	9/2/20	NULL	0.3488881809680698	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB1	hgnc:9537	PSMB1	DTC	9/2/20	NULL	0.5233322714521046	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB8	hgnc:9545	PSMB8	DTC	9/2/20	NULL	0.2220197515251353	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
ADRM1	hgnc:15759	ADRM1	DTC	9/2/20	NULL	0.3663325900164732	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
AKT2	hgnc:392	AKT2	ChEMBL	33	inhibitor	0.4167275494896389	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
PSMC1	hgnc:9547	PSMC1	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA7	hgnc:9536	PSMA7	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.8607814956671229	SEGESTERONE ACETATE	rxcui:2055977	SEGESTERONE ACETATE	TRUE	FALSE	FALSE
PSMC6	hgnc:9553	PSMC6	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.067317527	FISETIN	rxcui:2667741	FISETIN	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.1785975212098452	CILNIDIPINE	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
PSMD6	hgnc:9564	PSMD6	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD12	hgnc:9557	PSMD12	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	blocker	0.1415301111474245	CILNIDIPINE	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
PSMD7	hgnc:9565	PSMD7	DTC	9/2/20	NULL	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA6	hgnc:9535	PSMA6	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMC4	hgnc:9551	PSMC4	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD11	hgnc:9556	PSMD11	DTC	9/2/20	NULL	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	2.218633995874415	ASIMADOLINE	ncit:C72137	ASIMADOLINE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.095122593	GNF-PF-2950	chembl:CHEMBL602807	CHEMBL:CHEMBL602807	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.5357925636295356	TCMDC-124317	chembl:CHEMBL586937	CHEMBL:CHEMBL586937	FALSE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	ChEMBL	33	agonist	2.625383561784724	CPG-52852	drugbank:DB12476	CPG-52852	FALSE	FALSE	FALSE
PTPN11	hgnc:9644	PTPN11	DTC	9/2/20	NULL	3.750547945	OLTIPRAZ	ncit:C1177	OLTIPRAZ	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.026599631	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	1.050153425	OLTIPRAZ	ncit:C1177	OLTIPRAZ	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.2442217266776488	FLUNARIZINE DIHYDROCHLORIDE	chembl:CHEMBL539027	FLUNARIZINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.023151531	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	THIOPERAMIDE	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.2500365296937833	DIFAMILAST	ncit:C169909	DIFAMILAST	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	(S)-MIDODRINE	chembl:CHEMBL255027	(S)-MIDODRINE	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	2-ETHYLANTHRAQUINONE	chembl:CHEMBL42355	CHEMBL:CHEMBL42355	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	ZARDAVERINE	ncit:C66686	ZARDAVERINE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015088411	OXIDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.018430211	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	TCMDC-125630	chembl:CHEMBL548619	CHEMBL:CHEMBL548619	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.003191956	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	DNDI1417072	chembl:CHEMBL1310701	CHEMBL:CHEMBL1310701	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.082689246	BENZIODARONE	ncit:C74127	BENZIODARONE	TRUE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.024008995	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.007300844	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RPS5	hgnc:10426	RPS5	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.026045472	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	7,3'-DIHYDROXYFLAVONE	chembl:CHEMBL253786	CHEMBL:CHEMBL253786	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	PIRETANIDE	rxcui:33770	PIRETANIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	TCMDC-123762	chembl:CHEMBL547483	CHEMBL:CHEMBL547483	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	RS-17053	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	(E)-2-STYRYLCHROMONE	chembl:CHEMBL388823	CHEMBL:CHEMBL388823	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	H-89 CHLORIDE	chembl:CHEMBL1315166	CHEMBL:CHEMBL1315166	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.3443125982668492	DELAVIRDINE	rxcui:83816	DELAVIRDINE	TRUE	FALSE	FALSE
GALK1	hgnc:4118	GALK1	DTC	9/2/20	NULL	0.055387839	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	ELIPRODIL	ncit:C80994	ELIPRODIL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV020403	chembl:CHEMBL548338	CHEMBL:CHEMBL548338	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	PHENELZINE SULFATE	rxcui:8124	PHENELZINE SULFATE	TRUE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.041182487	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.2344092465879218	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.2169738480813822	PROTOPORPHYRIN DISODIUM	ncit:C76666	PROTOPORPHYRIN DISODIUM	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010588359	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.004370177	TRICHOSTATIN	drugbank:DB04297	TRICHOSTATIN A	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DARBUFELONE MESYLATE	ncit:C81062	DARBUFELONE MESYLATE	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	DTC	9/2/20	NULL	0.6105543166941221	SANDARACOPIMARIC ACID	chembl:CHEMBL513197	SANDARACOPIMARIC ACID	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.011555385	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	DTC	9/2/20	NULL	0.4070362111294147	SANDARACOPIMARIC ACID	chembl:CHEMBL513197	SANDARACOPIMARIC ACID	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.041442519	S(+)-ISOPROTERENOL-BITARTRATE	chembl:CHEMBL1257092	CHEMBL:CHEMBL1257092	FALSE	FALSE	FALSE
GRM6	hgnc:4598	GRM6	DTC	9/2/20	NULL	1.166837138570988	N-(3-CHLOROPHENYL)PICOLINAMIDE	iuphar.ligand:6234	VU0364770	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	GABAZINE	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	SAPPANONE A DIMETHYL ETHER	chembl:CHEMBL1489223	SAPPANONE A DIMETHYL ETHER	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1100789753368857	6,4'-DIMETHOXYFLAVONE	chembl:CHEMBL1410006	6,4'-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
CTSL	hgnc:2537	CTSL	DTC	9/2/20	NULL	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.4667348554283956	NAPHTHOQUINONE	chembl:CHEMBL55934	NAPHTHOQUINONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002356506	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	OLEAMIDE	iuphar.ligand:284	OLEAMIDE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.009158847	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.009430257	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	SJ000018298	chembl:CHEMBL591412	CHEMBL:CHEMBL591412	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.1881995384791917	R-1487	drugbank:DB06518	R-1487	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.047176704	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	MELITRACEN	rxcui:446248	MELITRACEN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.020117882	DICHLOROPHEN	rxcui:3351	DICHLOROPHEN	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	1.810609352954982	S-(2-CHLOROBENZYL)ISOTHIOUREA HCL	chembl:CHEMBL1224310	CHEMBL:CHEMBL1224310	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.024651489	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.026519026	OLEIC ACID	rxcui:7631	OLEIC ACID	TRUE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.1041818873724097	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.010082118	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.2966535098061835	EUPATORIN	chembl:CHEMBL487402	EUPATORIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004172574	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	DIOXYBENZONE	rxcui:23350	DIOXYBENZONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.002856317	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
SUMO1	hgnc:12502	SUMO1	DTC	9/2/20	NULL	0.1973972602845657	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	DTC	9/2/20	NULL	2.100306849	DIMETHYL FUMARATE	rxcui:1373478	DIMETHYL FUMARATE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.1130007271930297	ABT-751	drugbank:DB12254	ABT-751	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	2.500365296937833	6-METHOXYCOMAPARVIN	chembl:CHEMBL401565	CHEMBL:CHEMBL401565	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1238388472539964	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004176557	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	5,7-DIMETHOXYISOFLAVONE	chembl:CHEMBL308688	5,7-DIMETHOXYISOFLAVONE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.073922431	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001303599	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	DNDI1417447	chembl:CHEMBL1307453	CHEMBL:CHEMBL1307453	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	BISINDOLYLMALEIMIDE IX	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.033658764	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	PYROXAMINE MALEATE	ncit:C76677	PYROXAMINE MALEATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	DNDI1417234	chembl:CHEMBL2094549	CHEMBL:CHEMBL2094549	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002331809	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.2638576444004749	SENNOSIDE A	chembl:CHEMBL2368547	SENNOSIDE A	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	GNF-PF-3964	chembl:CHEMBL599088	CHEMBL:CHEMBL599088	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	TRACAZOLATE	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-124576	chembl:CHEMBL579420	CHEMBL:CHEMBL579420	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1508841127462485	SJ000047240	chembl:CHEMBL590706	CHEMBL:CHEMBL590706	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	PROFLAVINE	rxcui:8723	PROFLAVINE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.072826174	QUERCETIN DIHYDRATE	ncit:C75768	QUERCETIN DIHYDRATE	FALSE	FALSE	FALSE
SMAD2	hgnc:6768	SMAD2	DTC	9/2/20	NULL	4.375639269641208	BISDEMETHOXYCURCUMIN	chembl:CHEMBL105350	BISDEMETHOXYCURCUMIN	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.011176601	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005903055	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	PIPLARTINE	chembl:CHEMBL465843	PIPLARTINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.018962684	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	0.5357925636295356	CYCLOVALONE	ncit:C81040	CYCLOVALONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	(-)-U-50488	chembl:CHEMBL58033	(-)-U-50488	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	PIPERIDOLATE HYDROCHLORIDE	rxcui:102170	PIPERIDOLATE HYDROCHLORIDE	FALSE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	DTC	9/2/20	NULL	2.250328767	MG-132	iuphar.ligand:8616	MG-132	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.064944553	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.006210251	METHYSERGIDE	rxcui:6911	METHYSERGIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.1900426678745596	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	GNF-PF-5134	chembl:CHEMBL602969	CHEMBL:CHEMBL602969	FALSE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	0.1256164383629055	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	DTC	9/2/20	NULL	0.046940525	FLUOROURACIL	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.027347745	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	AG-1296	iuphar.ligand:5915	AG 1296	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	AG-1296	iuphar.ligand:5915	AG 1296	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.061055432	GALUTEOLIN	chembl:CHEMBL233929	GALUTEOLIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	INDOLE-3-CARBINOL	rxcui:2598119	INDOLE-3-CARBINOL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.054243462	NSC-42384	chembl:CHEMBL1270168	CHEMBL:CHEMBL1270168	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001450208	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.2817943000126717	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	4,2',4',6'-TETRAHYDROXYCHALCONE	chembl:CHEMBL338066	4,2',4',6'-TETRAHYDROXYCHALCONE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.056826484	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	GW282974X	chembl:CHEMBL30432	GW282974X	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	GNF-PF-2335	chembl:CHEMBL601146	CHEMBL:CHEMBL601146	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	AMPEROZIDE HYDROCHLORIDE	ncit:C77259	AMPEROZIDE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.1630673019742065	KERACYANIN	rxcui:28165	KERACYANIN	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	inhibitor	0.009244308	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	CID 739615	chembl:CHEMBL260560	CHEMBL:CHEMBL260560	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.030176823	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	NSC-19803	chembl:CHEMBL522983	CHEMBL:CHEMBL522983	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.005602013	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
HTR7	hgnc:5302	HTR7	DTC	9/2/20	NULL	0.2692701089009974	5-CARBOXAMIDOTRYPTAMINE	iuphar.ligand:4	5-CT	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.084553416	3R14S-OCHRATOXIN A	iuphar.ligand:4672	OCHRATOXIN A	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	GNF-PF-2776	chembl:CHEMBL578294	CHEMBL:CHEMBL578294	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003405608	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	3,4-METHYLENEDIOXYB-NITROSTYRENE	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	1,2-DINITRO-BENZENE	chembl:CHEMBL168075	CHEMBL:CHEMBL168075	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	DIBENZOYLMETHANE	chembl:CHEMBL371523	DIBENZOYLMETHANE	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.016166155	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007232462	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	SALIRASIB	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
TRPC5	hgnc:12337	TRPC5	DTC	9/2/20	NULL	4.200613698855561	4,4'-DITHIODIPYRIDINE	chembl:CHEMBL1232076	CHEMBL:CHEMBL1232076	FALSE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	inhibitor	0.093763699	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.028290771	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.525076712	GNF-PF-1935	chembl:CHEMBL588250	CHEMBL:CHEMBL588250	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.1367387271762877	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.008428198	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	1.666910197958555	NSC-37136	chembl:CHEMBL1370674	CHEMBL:CHEMBL1370674	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	KINETIN RIBOSIDE	chembl:CHEMBL411066	KINETIN RIBOSIDE	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.3860858179095183	DIHYDRODAPHNODORIN B	chembl:CHEMBL1532097	DIHYDRODAPHNODORIN B	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	(S)-3,5-DIHYDROXYPHENYLGLYCINE	drugbank:DB04228	DIHYDROXYPHENYLGLYCINE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.01327292	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	SJ000262801	chembl:CHEMBL605077	CHEMBL:CHEMBL605077	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	DTC	9/2/20	NULL	0.029074015	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	NSC-172614	chembl:CHEMBL1317506	CHEMBL:CHEMBL1317506	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	1-BENZYLMALEIMIDE	chembl:CHEMBL388979	CHEMBL:CHEMBL388979	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	DTC	9/2/20	NULL	0.015385511	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	GNF-PF-3201	chembl:CHEMBL581872	CHEMBL:CHEMBL581872	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	APIOL	chembl:CHEMBL1560118	APIOL	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.02232469	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	NAFAMOSTAT	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	NSC-45382	chembl:CHEMBL1214274	CHEMBL:CHEMBL1214274	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	MECLIZINE DIHCL	chembl:CHEMBL1085765	MECLIZINE DIHCL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	DNDI1417215	chembl:CHEMBL1390650	CHEMBL:CHEMBL1390650	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	TCMDC-123650	chembl:CHEMBL580727	CHEMBL:CHEMBL580727	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.082559232	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	HARMOL HYDROCHLORIDE	chembl:CHEMBL1449575	HARMOL HYDROCHLORIDE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	DTC	9/2/20	NULL	0.7955707762984013	CHOLIC ACID	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	STROPHANTHIDIN	chembl:CHEMBL111743	STROPHANTHIDIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	QUESTIOMYCIN B	chembl:CHEMBL28319	QUESTIOMYCIN B	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	4-HYDROXYBENZALDEHYDE PHENYLHYDRAZONE	chembl:CHEMBL224032	CHEMBL:CHEMBL224032	FALSE	FALSE	FALSE
RIPK2	hgnc:10020	RIPK2	DTC	9/2/20	NULL	0.2917092846427472	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	5,7-DIHYDROXY-4-METHYLCOUMARIN	chembl:CHEMBL12252	5,7-DIHYDROXY-4-METHYLCOUMARIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	DTC	9/2/20	NULL	2.187819634820604	ALLYL ISOTHIOCYANATE	iuphar.ligand:2420	ALLYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.2344092465879218	INDIRUBIN SULFATE	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
ESRRA	hgnc:3471	ESRRA	DTC	9/2/20	NULL	0.3723948314588262	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.015627283	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	CID 660258	chembl:CHEMBL259805	CHEMBL:CHEMBL259805	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.003116552	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.005686341	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.1835932560688619	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	LERCANIDIPINE	rxcui:135056	LERCANIDIPINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007727398	E-FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.012137696	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	PHENTHOATE	ncit:C163686	PHENTHOATE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.050007306	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	ALPHA,BETA-DEHYDROCURVULARIN	chembl:CHEMBL482050	CHEMBL:CHEMBL482050	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.3889457128569962	BENZALDEHYDE O-4-METHOXYPHENYLCARBAMOYL OXIME	chembl:CHEMBL599469	CHEMBL:CHEMBL599469	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	2.059124362184098	ARUNCIN B	chembl:CHEMBL2203686	ARUNCIN B	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006439499	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	PSORALEN	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009170044	SJ000113257	chembl:CHEMBL528694	CHEMBL:CHEMBL528694	FALSE	FALSE	FALSE
USP2	hgnc:12618	USP2	DTC	9/2/20	NULL	0.065145994	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	QUERCETIN DIHYDRATE	ncit:C75768	QUERCETIN DIHYDRATE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	NSC-327705	chembl:CHEMBL1317986	CHEMBL:CHEMBL1317986	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	DEGUELIN	ncit:C63666	DEGUELIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	5-HYDROXYINDOLACETIC ACID	iuphar.ligand:11900	5-HYDROXYINDOLEACETIC ACID	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.5303805175322676	TCMDC-123653	chembl:CHEMBL548540	CHEMBL:CHEMBL548540	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-124409	chembl:CHEMBL587801	CHEMBL:CHEMBL587801	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.2983390411119005	TRACAZOLATE	ncit:C152706	TRACAZOLATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.001493605	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PRSS2	hgnc:9483	PRSS2	DTC	9/2/20	NULL	5.834185692854944	CYANOPEPTOLIN S	chembl:CHEMBL1076838	CYANOPEPTOLIN S	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.6863747873946993	FENAMIC ACID	iuphar.ligand:4182	DIPHENYLAMINE-2-CARBOXYLIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.00299189	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	PALMITOYL-CARNITINE	chembl:CHEMBL301722	PALMITOYL-CARNITINE	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.027519744	SB-202190	iuphar.ligand:4307	SB202190	FALSE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	0.577007376	OXOPURPUREINE	chembl:CHEMBL456295	OXOPURPUREINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	GNF-PF-5051	chembl:CHEMBL600773	CHEMBL:CHEMBL600773	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	inhibitor	0.006311018	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	(S)APOMORPHINE	iuphar.ligand:8285	S(+)-APOMORPHINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	DNDI1416985	chembl:CHEMBL593211	CHEMBL:CHEMBL593211	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2917092846427472	ALDICARB	ncit:C163578	ALDICARB	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.020575106	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
TDP2	hgnc:17768	TDP2	DTC	9/2/20	NULL	1.944728564284981	GNF-PF-4418	chembl:CHEMBL604321	CHEMBL:CHEMBL604321	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.041182487	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	CHLOROPHENYLPIPERAZINE	iuphar.ligand:142	M-CHLOROPHENYLPIPERAZINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TCMDC-123920	chembl:CHEMBL1606	CHEMBL:CHEMBL1606	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	P-HYDROXYCINNAMALDEHYDE	chembl:CHEMBL431836	P-HYDROXYCINNAMALDEHYDE	FALSE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	0.1434635826111871	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
APH1B	hgnc:24080	APH1B	DTC	9/2/20	NULL	2.019525817	LY-411575	chembl:CHEMBL392068	CHEMBL:CHEMBL392068	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.031707531	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	FENBENDAZOLE	rxcui:4325	FENBENDAZOLE	TRUE	FALSE	FALSE
CAPN1	hgnc:1476	CAPN1	DTC	9/2/20	NULL	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	ANETHOLTRITHION	rxcui:820	ANETHOLE TRITHIONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	QUINACRINE	rxcui:9061	QUINACRINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00202529	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.023274677	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.001831769	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.023482858	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007866318	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
RPS12	hgnc:10385	RPS12	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
GYPA	hgnc:4702	GYPA	DTC	9/2/20	NULL	15.00219178	YESSOTOXIN	chembl:CHEMBL1077126	YESSOTOXIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	METHOCTRAMINE	iuphar.ligand:327	METHOCTRAMINE	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	inhibitor	0.036463661	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.169927739	CAULIBUGULONE C	chembl:CHEMBL445969	CAULIBUGULONE C	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.2638576444004749	EUFLAVINE	drugbank:DB13326	EUFLAVINE	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	MAKALUVAMINE F	chembl:CHEMBL509890	MAKALUVAMINE F	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	3,4-DIMETHOXYDALBERGIONE	chembl:CHEMBL1591258	3,4-DIMETHOXYDALBERGIONE	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.029715717	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.026319635	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.6141248097742046	7,8-DIHYDROXYISOFLAVONE	chembl:CHEMBL241813	CHEMBL:CHEMBL241813	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.004310975	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
RPS17	hgnc:10397	RPS17	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	DEOXYVASICINONE	chembl:CHEMBL456881	DEOXYVASICINONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.022410444	DNDI1417523	chembl:CHEMBL598663	CHEMBL:CHEMBL598663	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.034970144	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.008103036	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.029590122	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	BUTOCONAZOLE NITRATE	rxcui:19884	BUTOCONAZOLE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.017243899	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	DTC	9/2/20	NULL	0.057073556	THIRAM	rxcui:10517	THIRAM	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.014114965	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	GUANFACINE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPS11	hgnc:10384	RPS11	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.081533651	NSC-107022	chembl:CHEMBL1601846	CHEMBL:CHEMBL1601846	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	MELPHALAN	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000217121	chembl:CHEMBL607308	CHEMBL:CHEMBL607308	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.2734774543525755	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.006836936	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-1938	chembl:CHEMBL587728	CHEMBL:CHEMBL587728	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.7778914257139925	25-HYDROXYCHOLESTEROL	drugbank:DB04705	25-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	A-77636	iuphar.ligand:9637	A77636	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.052090944	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	1.640864726115453	RETUSIN	chembl:CHEMBL77966	RETUSIN	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	inhibitor	0.052507671	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.034118045	POMIFERIN	rxcui:2593691	POMIFERIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.014369915	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.1470803115845784	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.007651949	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
RPS3A	hgnc:10421	RPS3A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	TCMDC-123912	iuphar.ligand:3930	JP1302	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.750109589	SULFANITRAN	ncit:C76978	SULFANITRAN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1810609352954982	NSC-1010	chembl:CHEMBL1688556	CHEMBL:CHEMBL1688556	FALSE	FALSE	FALSE
NR2F2	hgnc:7976	NR2F2	DTC	9/2/20	NULL	2.187819634820604	RESACTIN A	chembl:CHEMBL509617	RESACTIN A	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004579424	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.014537008	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	CICLOPIROX OLAMINE	rxcui:52172	CICLOPIROX OLAMINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-633	chembl:CHEMBL602408	CHEMBL:CHEMBL602408	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	BENZO[D]ISOTHIAZOL-3-ONE	chembl:CHEMBL297304	CHEMBL:CHEMBL297304	FALSE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.8751278539282416	(-)-DEMECOLCINE	ncit:C419	DEMECOLCINE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	GBR-12935	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.026227608	BETA-LAPACHONE	ncit:C28694	LAPACHONE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	GNF-PF-1339	chembl:CHEMBL600353	CHEMBL:CHEMBL600353	FALSE	FALSE	FALSE
RPS15A	hgnc:10389	RPS15A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.009673484	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	ANISOMYCIN	ncit:C95312	ANISOMYCIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	HERNIARIN	chembl:CHEMBL49732	HERNIARIN	FALSE	FALSE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	3.889457128569962	6-DECYLSALICYLIC ACID	chembl:CHEMBL416038	CHEMBL:CHEMBL416038	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	HALOFANTRINE HYDROCHLORIDE	rxcui:58130	HALOFANTRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TDP2	hgnc:17768	TDP2	DTC	9/2/20	NULL	0.6731752722524936	9,10-PHENANTHRENEQUINONE	chembl:CHEMBL51931	9,10-PHENANTHRENEQUINONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00239313	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.054695491	VINPOCETINE	rxcui:24506	VINPOCETINE	FALSE	FALSE	FALSE
RPS4Y1	hgnc:10425	RPS4Y1	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RAC1	hgnc:9801	RAC1	DTC	9/2/20	NULL	11.66837138570988	NSC-23766	iuphar.ligand:11057	NSC 23766	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007479725	IMIPRAMINE HYDROCHLORIDE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007946076	DEQUALINIUM	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	CID 695758	chembl:CHEMBL260028	CHEMBL:CHEMBL260028	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	(20S,21S)-7-CYCLOHEXYLFLUOROCAMPTOTHECIN	chembl:CHEMBL2435339	(20S,21S)-7-CYCLOHEXYLFLUOROCAMPTOTHECIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	QUINOXALINE-2-CARBOXYLIC ACID	chembl:CHEMBL151797	CHEMBL:CHEMBL151797	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	SPERMIDINE	rxcui:1483262	SPERMIDINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013299815	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.2381300282797936	2,5-BIS(4-ISOPROPYLSTYRYL)PYRAZINE	chembl:CHEMBL2181040	CHEMBL:CHEMBL2181040	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
RPS8	hgnc:10441	RPS8	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
EPHA7	hgnc:3390	EPHA7	DTC	9/2/20	inhibitor	0.072927321	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
DYRK3	hgnc:3094	DYRK3	DTC	9/2/20	NULL	0.1136529680426287	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.066803653	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	TCMDC-124059	chembl:CHEMBL530733	CHEMBL:CHEMBL530733	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	1.944728564284981	1,2,4,5-BENZENETETRAAMINE TETRAHYDROCHLORIDE	chembl:CHEMBL456559	CHEMBL:CHEMBL456559	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	CLORGILINE	ncit:C77522	CLORGILINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	ESOXYBUTYNIN	ncit:C166661	ESOXYBUTYNIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007374673	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1446492320542548	DNDI1417400	chembl:CHEMBL1362503	CHEMBL:CHEMBL1362503	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	SUPROFEN METHYL ESTER	chembl:CHEMBL1474177	SUPROFEN METHYL ESTER	FALSE	FALSE	FALSE
RPL29	hgnc:10331	RPL29	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GNF-PF-4325	chembl:CHEMBL598263	CHEMBL:CHEMBL598263	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.014287802	PURPURIN	chembl:CHEMBL294264	PURPURIN	FALSE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.075768645	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	STAUROSPORINE AGLYCON	chembl:CHEMBL268368	STAUROSPORINE AGLYCON	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	STROPHANTHIDIN	chembl:CHEMBL111743	STROPHANTHIDIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	NSC-172614	chembl:CHEMBL1317506	CHEMBL:CHEMBL1317506	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.009309871	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.023823807	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	SJ000032159	chembl:CHEMBL591361	CHEMBL:CHEMBL591361	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007962947	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
IGF1	hgnc:5464	IGF1	ChEMBL	33	inhibitor	13.12691780892362	XENTUZUMAB	ncit:C106118	XENTUZUMAB	FALSE	FALSE	FALSE
KLK7	hgnc:6368	KLK7	DTC	9/2/20	NULL	52.50767123569449	CASTANIN	chembl:CHEMBL464404	CASTANIN	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	INDIGO	rxcui:1426889	INDIGO	TRUE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	2.100306849	MORONIC ACID	chembl:CHEMBL472646	MORONIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	AG-126	chembl:CHEMBL77387	CHEMBL:CHEMBL77387	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.729273212	DNDI1417470	chembl:CHEMBL1422873	CHEMBL:CHEMBL1422873	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	SR-59230A	iuphar.ligand:547	SR59230A	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	SEROTONIN	rxcui:1311214	SEROTONIN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.027319288	AURINTRICARBOXYLIC ACID	chembl:CHEMBL275938	AURINTRICARBOXYLIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.003324322	AMITRIPTYLINE HYDROCHLORIDE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	(S)-SARGACHROMENOL	chembl:CHEMBL1668778	(S)-SARGACHROMENOL	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.004920134	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005107253	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
RPL37A	hgnc:10348	RPL37A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
FGF22	hgnc:3679	FGF22	DTC	9/2/20	NULL	1.250182648468916	N-(4-NITROPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1574420	CHEMBL:CHEMBL1574420	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	IODOACETAMIDE	iuphar.ligand:6271	2-IODOACETAMIDE	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.033487035	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.2900976311364336	PICEID	chembl:CHEMBL142652	PICEID	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.033487035	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	INDOCATE	ncit:C65912	INDOCATE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW678313X	chembl:CHEMBL372474	GW678313X	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
PTP4A3	hgnc:9636	PTP4A3	DTC	9/2/20	NULL	2.019525816757481	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	DNDI1417213	chembl:CHEMBL2094532	CHEMBL:CHEMBL2094532	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	FLUPIRTINE MALEATE	rxcui:236774	FLUPIRTINE MALEATE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
EIF4A1	hgnc:3282	EIF4A1	DTC	9/2/20	NULL	2.019525817	HIPPURISTANOL	chembl:CHEMBL1098427	HIPPURISTANOL	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	QUINOXALINE-2-CARBOXYLIC ACID	chembl:CHEMBL151797	CHEMBL:CHEMBL151797	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	SJ000117451	chembl:CHEMBL592123	CHEMBL:CHEMBL592123	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	4-PHENYLPHENOL	chembl:CHEMBL73380	CHEMBL:CHEMBL73380	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	EFONIDIPINE	ncit:C73026	EFONIDIPINE	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.100589408	CEFOTETAN	rxcui:2187	CEFOTETAN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	ATRACURIUM BESYLATE	rxcui:1219	ATRACURIUM BESYLATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.1190650141398968	BENZOXAZOLINONE	chembl:CHEMBL280323	BENZOXAZOLINONE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	DENDROAMIDE A	chembl:CHEMBL516542	DENDROAMIDE A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	CHOLECALCIFEROL	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00449706	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.072424374	DNDI1417607	chembl:CHEMBL1588679	CHEMBL:CHEMBL1588679	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1640864726115453	ERGOCRYPTINE	iuphar.ligand:271	&ALPHA;-ERGOCRYPTINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	CLOBENPROPIT	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	0.1110098757625676	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.042741287	PLUMBAGIN	drugbank:DB17048	PLUMBAGIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	NSC-93392	chembl:CHEMBL53738	CHEMBL:CHEMBL53738	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	CALCIMYCIN	ncit:C83573	CALCIMYCIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.039538909	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.03140411	Ixabepilone	rxcui:337523	IXABEPILONE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	1.250182648468916	Inotuzumab Ozogamicin	rxcui:1942950	INOTUZUMAB OZOGAMICIN	TRUE	FALSE	FALSE
F5	hgnc:3542	F5	FDA	10-Apr-24	NULL	0.1966579447029756	Lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
BCHE	hgnc:983	BCHE	FDA	10-Apr-24	NULL	1.750255707856483	Mivacurium	rxcui:30077	MIVACURIUM	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	0.5498185469706229	RO5212054	ncit:C92591	BRAF(V600E) KINASE INHIBITOR RO5212054	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.6019397937072561	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.07661359	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.4375639269641208	BELOTECAN	ncit:C73305	BELOTECAN	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	MyCancerGenome	20-Jun-17	inhibitor	1.678633990910949	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.2678962818147679	PD0325901	drugbank:DB07101	MIRDAMETINIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.027390543	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.2275522047050683	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.090821275	SIROLIMUS	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	inhibitor	1.090323227845022	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.088248187	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.2778183663264258	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
CD38	hgnc:1667	CD38	ChEMBL	33	inhibitor	5.834185692854944	FELZARTAMAB	ncit:C97954	FELZARTAMAB	FALSE	FALSE	FALSE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.2051080907644316	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.2051080907644316	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.045016865	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.1215455352678113	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.052090944	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.1215455352678113	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.029918901	GDC-0980	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.2243917574174978	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.3241214273808303	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.1620607136904151	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
POLE3	hgnc:13546	POLE3	ChEMBL	33	inhibitor	0.7955707762984016	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.2243917574174978	PX-866	ncit:C78848	SONOLISIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.040328473	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
MLST8	hgnc:24825	MLST8	MyCancerGenome	20-Jun-17	inhibitor	0.5966780822238011	MLN0128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
RPTOR	hgnc:30287	RPTOR	MyCancerGenome	20-Jun-17	inhibitor	0.1491695205559502	MLN0128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
MAP2K5	hgnc:6845	MAP2K5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3281729452230906	MEK162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.042259695	EVEROLIMUS	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
RET	hgnc:9967	RET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5303805175322677	CABOZANTINIB	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.073437302	BAY80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.8334550989792776	BAY869766	hemonc:437	REFAMETINIB	FALSE	FALSE	TRUE
MAP2K7	hgnc:6847	MAP2K7	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.7501095890813498	BAY869766	hemonc:437	REFAMETINIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1519026168824334	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.150021918	GSK2126458	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
AANAT	hgnc:19	AANAT	NCI	14-Sep-17	NULL	0.03729238	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.062331044	ANTIHISTAMINE	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4398548375764984	1096708-71-2	ncit:C106254	TOVORAFENIB	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.2804896967718723	PSC 833	ncit:C1405	VALSPODAR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02926849	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
ALDH1A2	hgnc:15472	ALDH1A2	NCI	14-Sep-17	NULL	1.166837138570989	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
BACE1	hgnc:933	BACE1	ChEMBL	33	inhibitor	4.039051633514961	ATABECESTAT	ncit:C166553	ATABECESTAT	FALSE	FALSE	FALSE
AGTR2	hgnc:338	AGTR2	NCI	14-Sep-17	NULL	0.4339476961627644	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
ARSB	hgnc:714	ARSB	NCI	14-Sep-17	NULL	1.009762908	ASCORBIC ACID	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
AQP1	hgnc:633	AQP1	NCI	14-Sep-17	NULL	2.763561643983921	CARBONIC ANHYDRASE INHIBITOR	ncit:C29577	CARBONIC ANHYDRASE INHIBITOR	FALSE	FALSE	FALSE
AQP1	hgnc:633	AQP1	NCI	14-Sep-17	NULL	0.172722603	DIMETHYL SULFOXIDE	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.046303061	ABIVERTINIB	ncit:C147125	ABIVERTINIB	FALSE	FALSE	FALSE
ATF2	hgnc:784	ATF2	NCI	14-Sep-17	NULL	1.750255707856483	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.035574303	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.042689164	6-HYDROXYDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.023075224	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.5676505	DIHYDROTESTOSTERONE	ncit:C29619	DIHYDROTESTOSTERONE	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.4730420832044549	GLYCYRRHETINIC ACID	rxcui:1311506	GLYCYRRHETINIC ACID	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.1988926940746003	CALCITONIN	rxcui:1311287	CALCITONIN	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.008230043	DDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.03849536	GW572016	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
GABRD	hgnc:4084	GABRD	ChEMBL	33	agonist	0.042619863	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	agonist	0.042073455	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	NCI	14-Sep-17	NULL	0.025390557	MITOXANTRONE	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
CARTPT	hgnc:24323	CARTPT	NCI	14-Sep-17	NULL	0.5122699632750682	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.1555782851427985	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.078136416	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.038467158	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.8334550989792776	ANABOLIC-ANDROGENIC STEROIDS	ncit:C2360	ANABOLIC STEROID	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.007378818	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	3.281729452230906	GISADENAFIL	ncit:C83728	GISADENAFIL	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.2187819634820604	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.1988926940746003	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.1174668260306364	MICAFUNGIN	rxcui:325887	MICAFUNGIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.029366707	METRONIDAZOLE	rxcui:6922	METRONIDAZOLE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.041672755	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.1346350544504987	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1221108633388244	6-HYDROXYDOPAMINE	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
CYP3A7	hgnc:2640	CYP3A7	NCI	14-Sep-17	NULL	0.5770073762164232	QUININE	rxcui:9071	QUININE	TRUE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	1.400204566285186	SAPONIN	ncit:C823	SAPONIN	FALSE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.2917092846427472	MITOMYCIN-C	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
DCT	hgnc:2709	DCT	NCI	14-Sep-17	NULL	1.346350544504987	FUNGIZONE	rxcui:236594	AMPHOTERICIN B LIPOSOMAL	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.029424304	TAXOTERE	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	1.093909817410302	ANTIFOLATES	ncit:C511	FOLATE ANTAGONIST	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.1367387271762877	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.3697723326457359	OLINVACIMAB	ncit:C102877	OLINVACIMAB	FALSE	FALSE	FALSE
DPYSL3	hgnc:3015	DPYSL3	NCI	14-Sep-17	NULL	0.2381300282797936	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
EPO	hgnc:3415	EPO	NCI	14-Sep-17	NULL	15.00219178	INTERLEUKIN-1-ALPHA	ncit:C1754	RECOMBINANT INTERLEUKIN-1-ALPHA	FALSE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	NCI	14-Sep-17	NULL	0.2983390411119005	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.2641895408085258	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.151537291	METHIMAZOLE	rxcui:6835	METHIMAZOLE	TRUE	FALSE	FALSE
GCLM	hgnc:4312	GCLM	NCI	14-Sep-17	NULL	1.154014752432846	SULFORAPHANE	ncit:C1424	SULFORAPHANE	FALSE	FALSE	FALSE
ACACA	hgnc:84	ACACA	ChEMBL	33	inhibitor	1.141471113819445	OLUMACOSTAT GLASARETIL	ncit:C166791	OLUMACOSTAT GLASARETIL	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.151537291	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.6482428547616604	CHEMOPREVENTIVE	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	3.088686543276147	PLANT STEROLS	ncit:C28178	PHYTOSTEROL	FALSE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.1691068316769549	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
GPT	hgnc:4552	GPT	NCI	14-Sep-17	NULL	0.9376369863516874	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	1.591141552596802	MISONIDAZOLE	ncit:C657	MISONIDAZOLE	FALSE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.1835932560688619	CARVEDILOL	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
GSTA1	hgnc:4626	GSTA1	NCI	14-Sep-17	NULL	3.500511415712966	PHYTOCHEMICALS	ncit:C28269	PHYTOCHEMICAL	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.050007306	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.652269208	SULFORAPHANE	ncit:C1424	SULFORAPHANE	FALSE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1211249624814175	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	0.1970269089519493	CORTICOSTEROIDS	ncit:C211	THERAPEUTIC CORTICOSTEROID	FALSE	FALSE	FALSE
KLKB1	hgnc:6371	KLKB1	ChEMBL	33	inhibitor	3.750547945	AVORALSTAT	ncit:C169799	AVORALSTAT	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.071341945	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.546954909	MONOCLONAL ANTIBODY 17-1A	rxcui:80726	EDRECOLOMAB	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	RCD4	ncit:C2342	RECOMBINANT SOLUBLE HUMAN CD4 PROTEIN	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1172046232939609	METOCLOPRAMIDE	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1093909817410302	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.4102161815288632	MARIJUANA	ncit:C26659	MARIJUANA	FALSE	FALSE	FALSE
INPPL1	hgnc:6080	INPPL1	NCI	14-Sep-17	NULL	3.182283105193606	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1040580087905162	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.7242437411819932	CLOBETASOL PROPIONATE	rxcui:21245	CLOBETASOL PROPIONATE	TRUE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.1902451856365742	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	NCI	14-Sep-17	NULL	1.131630845596864	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
KCNA5	hgnc:6224	KCNA5	NCI	14-Sep-17	NULL	1.400204566285186	DIHYDROTESTOSTERONE	ncit:C29619	DIHYDROTESTOSTERONE	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.019233579	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.031631127	DOCETAXEL	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
LDHA	hgnc:6535	LDHA	NCI	14-Sep-17	NULL	4.375639269641208	ANTHRACYCLINES	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	1.129197231	CHOLESTYRAMINE	rxcui:2447	CHOLESTYRAMINE RESIN	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.095468493	PAROXETINE HYDROCHLORIDE HEMIHYDRATE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	1.693795846312725	FAT EMULSION	ncit:C2575	FAT EMULSION	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.1268301237577161	8-METHOXYPSORALEN	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.1071585127259071	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.2083637747448194	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.1495945049449985	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1029562181092049	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
MUC2	hgnc:7512	MUC2	NCI	14-Sep-17	NULL	1.666910197958555	CHEMOPREVENTIVE AGENT	ncit:C1892	CHEMOPREVENTIVE AGENT	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	agonist	0.3659071166250487	ZUCAPSAICIN	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	NCI	14-Sep-17	NULL	0.026680727	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.01573971	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.00674559	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.087005255	NSAID	ncit:C257	NONSTEROIDAL ANTIINFLAMMATORY DRUG	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	2.187819634820604	PD 153035	ncit:C1547	COMPOUND 32	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.068369364	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.1620607136904151	THEAFLAVINS	ncit:C29855	THEAFLAVIN	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1346350544504987	MTOR INHIBITOR	ncit:C2201	MTOR INHIBITOR	FALSE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.036718651	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	0.3804903712731485	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.2692701089009974	THEAFLAVINS	ncit:C29855	THEAFLAVIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	2.917092846427472	ETIDRONATE DISODIUM	rxcui:9872	ETIDRONATE DISODIUM	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.085796848	BUPROPION	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
REG1A	hgnc:9951	REG1A	NCI	14-Sep-17	NULL	26.25383561784724	LINOMIDE	ncit:C1519	ROQUINIMEX	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	NCI	14-Sep-17	NULL	0.090064616	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
RUNX2	hgnc:10472	RUNX2	NCI	14-Sep-17	NULL	3.182283105193606	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.4907258993990139	VILOXAZINE HYDROCHLORIDE	rxcui:142143	VILOXAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.072125922	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.546954909	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.031069628	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1346350544504987	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
SMARCA4	hgnc:11100	SMARCA4	NCI	14-Sep-17	NULL	0.1442518440541057	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SMAD2	hgnc:6768	SMAD2	NCI	14-Sep-17	NULL	0.8204323630577265	BLEOMYCIN	rxcui:1622	BLEOMYCIN	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.1635752997996713	FGFR INHIBITOR DEBIO 1347	chembl:CHEMBL3907479	FGFR INHIBITOR DEBIO 1347	FALSE	FALSE	FALSE
SMAD4	hgnc:6770	SMAD4	NCI	14-Sep-17	NULL	0.9546849315580819	TGF	ncit:C899	RECOMBINANT TRANSFORMING GROWTH FACTOR	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.2500365296937833	WORTMANNIN	ncit:C1277	WORTMANNIN	FALSE	FALSE	FALSE
SPP1	hgnc:11255	SPP1	NCI	14-Sep-17	NULL	0.3889457128569963	IMMUNOSUPPRESSANT	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
STAT4	hgnc:11365	STAT4	NCI	14-Sep-17	NULL	17.50255707856483	DNA METHYLTRANSFERASE INHIBITOR	ncit:C2083	DNA METHYLTRANSFERASE INHIBITOR	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	NCI	14-Sep-17	NULL	0.5000730593875666	RECOMBINANT INTERLEUKIN	ncit:C593	RECOMBINANT INTERLEUKIN	FALSE	FALSE	FALSE
STS	hgnc:11425	STS	NCI	14-Sep-17	NULL	0.1186614039224734	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
TERC	hgnc:11727	TERC	NCI	14-Sep-17	NULL	0.1810609352954982	CDDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TBXA2R	hgnc:11608	TBXA2R	NCI	14-Sep-17	NULL	0.1630673019742065	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.1814781263906492	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.6731752722524935	ACIVICIN	ncit:C986	ACIVICIN	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.2778183663264259	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.2143170254518142	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	0.133155548	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
WRN	hgnc:12791	WRN	NCI	14-Sep-17	NULL	0.035299275	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.019382677	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	OncoKB	23-Jul-20	NULL	0.6019397937072561	Dacomitinib	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	OncoKB	23-Jul-20	NULL	0.3923362732430473	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	2.341819737097098	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	OncoKB	23-Jul-20	NULL	0.2639729920045843	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PDGFB	hgnc:8800	PDGFB	OncoKB	23-Jul-20	NULL	0.3500511415712966	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
ERCC2	hgnc:3434	ERCC2	OncoKB	23-Jul-20	NULL	0.1646008502686348	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.029235897	GT-0918	iuphar.ligand:11992	PRUXELUTAMIDE	FALSE	FALSE	FALSE
NELFCD	hgnc:15934	NELFCD	PharmGKB	4/5/24	NULL	1.141471113819445	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
MUSK	hgnc:7525	MUSK	PharmGKB	4/5/24	NULL	2.625383561784725	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
CHRNA1	hgnc:1955	CHRNA1	PharmGKB	4/5/24	NULL	0.2500365296937833	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	PharmGKB	4/5/24	NULL	0.1117184494376478	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.2263261691193728	galantamine	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
STMN1	hgnc:6510	STMN1	PharmGKB	4/5/24	NULL	1.346350544504987	vinorelbine	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
ERCC1	hgnc:3433	ERCC1	PharmGKB	4/5/24	NULL	0.087512785	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SCNN1G	hgnc:10602	SCNN1G	PharmGKB	4/5/24	NULL	0.6482428547616605	furosemide	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
ATP2B1	hgnc:814	ATP2B1	PharmGKB	4/5/24	NULL	0.4102161815288632	Antihypertensives	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
LAG3	hgnc:6476	LAG3	ChEMBL	33	inhibitor	3.281729452230906	TEBOTELIMAB	ncit:C143957	TEBOTELIMAB	FALSE	FALSE	FALSE
KCNK3	hgnc:6278	KCNK3	PharmGKB	4/5/24	NULL	1.000146118775133	candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	BUDIGALIMAB	ncit:C137682	BUDIGALIMAB	FALSE	FALSE	FALSE
CSF3R	hgnc:2439	CSF3R	ChEMBL	33	inhibitor	2.019525817	CSL-324	chembl:CHEMBL4650461	CSL-324	FALSE	FALSE	FALSE
IL6R	hgnc:6019	IL6R	ChEMBL	33	inhibitor	4.039051633514961	LEVILIMAB	ncit:C173804	LEVILIMAB	FALSE	FALSE	FALSE
SV2B	hgnc:16874	SV2B	ChEMBL	33	modulator	2.763561643983921	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.077444943	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
NCOA3	hgnc:7670	NCOA3	PharmGKB	4/5/24	NULL	0.8078103267029924	salbutamol	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.005099813	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.085239726	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.07458476	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.003399875	doxepin	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	agonist	2.625383561784724	DASIGLUCAGON	rxcui:2535233	DASIGLUCAGON	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.1215455352678113	encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.2822993077187876	encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	1.282909942931453	encorafenib	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.082300425	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1131630845596864	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
CXCL8	hgnc:6025	CXCL8	PharmGKB	4/5/24	NULL	0.033529803	pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
SLC28A3	hgnc:16484	SLC28A3	PharmGKB	4/5/24	NULL	0.4546118721705152	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.048618214	pitavastatin	rxcui:861634	PITAVASTATIN	TRUE	FALSE	FALSE
CHD4	hgnc:1919	CHD4	PharmGKB	4/5/24	NULL	0.4773424657790409	vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.045579576	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	1.909369863116163	cerivastatin	rxcui:596723	CERIVASTATIN	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.059667808	DOTHIEPIN	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
ZNF385D	hgnc:26191	ZNF385D	PharmGKB	4/5/24	NULL	6.058577450272442	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.2853677784548614	sumatriptan	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.2651902587661338	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
MIR3117	hgnc:38385	MIR3117	PharmGKB	4/5/24	NULL	0.7292732116068681	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
LEUS	hgnc:6512	LARS1	ChEMBL	33	inhibitor	52.50767123569449	EPETRABOROLE	ncit:C166950	EPETRABOROLE	FALSE	FALSE	FALSE
CPA2	hgnc:2297	CPA2	PharmGKB	4/5/24	NULL	1.944728564284981	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.00804962	rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
NME2	hgnc:7850	NME2	PharmGKB	4/5/24	NULL	1.166837138570989	adefovir dipivoxil	rxcui:141400	ADEFOVIR DIPIVOXIL	TRUE	FALSE	FALSE
LYN	hgnc:6735	LYN	PharmGKB	4/5/24	NULL	0.084689792	ziprasidone	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	PharmGKB	4/5/24	NULL	0.053145416	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	inhibitor	0.8899605294185507	NBI-921352	iuphar.ligand:11734	ZANDATRIGINE	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	PharmGKB	4/5/24	NULL	0.210030685	hydralazine	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
LRRC15	hgnc:20818	LRRC15	PharmGKB	4/5/24	NULL	0.760980743	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
SH2B3	hgnc:29605	SH2B3	PharmGKB	4/5/24	NULL	3.500511415712966	candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.056097939	bromperidol	rxcui:19777	BROMPERIDOL	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.074797252	trabectedin	rxcui:1716278	TRABECTEDIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.008013991	romidepsin	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.2804896967718723	Valspodar	ncit:C1405	VALSPODAR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.037398626	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.064111931	iguratimod	ncit:C65886	IGURATIMOD	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.032055965	azithromycin	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.062331044	terfenadine	rxcui:42330	TERFENADINE	TRUE	FALSE	FALSE
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	0.1000146118775133	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.2243917574174978	lenvatinib	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
ABCB11	hgnc:42	ABCB11	PharmGKB	4/5/24	NULL	0.3292017005372696	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	PharmGKB	4/5/24	NULL	0.081407242	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NAMPT	hgnc:30092	NAMPT	PharmGKB	4/5/24	NULL	2.100306849	nitric oxide	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.305277158	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.2220197515251353	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
IL1RL2	hgnc:5999	IL1RL2	ChEMBL	33	inhibitor	8.751278539282415	IMSIDOLIMAB	ncit:C177088	IMSIDOLIMAB	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	PharmGKB	4/5/24	NULL	4.861821410712453	tositumomab	rxcui:263010	TOSITUMOMAB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.015875335	pembrolizumab	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.3968833804663227	neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.030868707	tremelimumab	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
PRKAB2	hgnc:9379	PRKAB2	PharmGKB	4/5/24	NULL	0.2763561643983921	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	2.461297089173179	aflatoxin b1	rxcui:2282017	AFLATOXIN B1	FALSE	FALSE	FALSE
ATP1A1	hgnc:799	ATP1A1	PharmGKB	4/5/24	NULL	3.500511415712966	eplerenone	rxcui:298869	EPLERENONE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.020741723	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	10.50153424713889	sofosbuvir	rxcui:1484911	SOFOSBUVIR	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.033204682	galantamine	rxcui:4637	GALANTAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.08854582	umeclidinium / vilanterol	wikidata:Q17125410	UMECLIDINIUM BROMIDE/VILANTEROL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.035418328	mirabegron	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.011068227	ranolazine	rxcui:35829	RANOLAZINE	TRUE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	PharmGKB	4/5/24	NULL	0.095122593	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
FIP1L1	hgnc:19124	FIP1L1	PharmGKB	4/5/24	NULL	3.500511415712967	meperidine	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.045791574	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.088770366	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.041989341	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.1164249916534246	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.053854022	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BDKRB2	hgnc:1030	BDKRB2	PharmGKB	4/5/24	NULL	0.075442056	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
HCP5	hgnc:21659	HCP5	PharmGKB	4/5/24	NULL	0.3763990769583835	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	PharmGKB	4/5/24	NULL	0.020692678	glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
MIR1912	hgnc:35396	MIR1912	PharmGKB	4/5/24	NULL	0.3454452054979901	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.1228249619548409	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
SLC26A9	hgnc:14469	SLC26A9	PharmGKB	4/5/24	NULL	0.6908904109959803	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
PRKAA2	hgnc:9377	PRKAA2	PharmGKB	4/5/24	NULL	0.167488584	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
F5	hgnc:3542	F5	PharmGKB	4/5/24	NULL	0.1966579447029756	lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	PharmGKB	4/5/24	NULL	0.042845917	valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.056097939	astemizole	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
SZRD1	hgnc:30232	SZRD1	PharmGKB	4/5/24	NULL	1.154014752432846	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.5073204950308646	glucose	rxcui:349730	ANHYDROUS DEXTROSE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.3117023117067671	naloxone	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
AMACR	hgnc:451	AMACR	PharmGKB	4/5/24	NULL	2.187819634820604	cholic acid	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.010848692	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.015498132	cimetidine	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
PVT1	hgnc:9709	PVT1	PharmGKB	4/5/24	NULL	7.501095890813499	glatiramer acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
IFNAR1	hgnc:5432	IFNAR1	PharmGKB	4/5/24	NULL	0.8334550989792776	glatiramer acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.089756703	hydromorphone	rxcui:203177	HYDROMORPHONE HYDROCHLORIDE	TRUE	FALSE	FALSE
IKBKG	hgnc:5961	IKBKG	PharmGKB	4/5/24	NULL	2.386712328895204	pyrimethamine	rxcui:9010	PYRIMETHAMINE	TRUE	FALSE	FALSE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.3182283105193606	thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	0.3500511415712966	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
ABCC10	hgnc:52	ABCC10	PharmGKB	4/5/24	NULL	0.192335792	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
SLCO4C1	hgnc:23612	SLCO4C1	PharmGKB	4/5/24	NULL	0.384671584	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
SLCO6A1	hgnc:23613	SLCO6A1	PharmGKB	4/5/24	NULL	0.5770073762164231	daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.058341857	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1458546423213736	labetalol	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
CETP	hgnc:1869	CETP	PharmGKB	4/5/24	NULL	0.6731752722524935	fluvastatin	rxcui:41127	FLUVASTATIN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.027135747	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	PharmGKB	4/5/24	NULL	0.088333021	entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
FMO3	hgnc:3771	FMO3	PharmGKB	4/5/24	NULL	1.750255707856483	teneligliptin	ncit:C87623	TENELIGLIPTIN	FALSE	FALSE	FALSE
SLC6A9	hgnc:11056	SLC6A9	PharmGKB	4/5/24	NULL	0.4861821410712453	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
SLIT1	hgnc:11085	SLIT1	PharmGKB	4/5/24	NULL	1.141471113819445	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.026359273	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.0545251	goserelin	rxcui:203146	GOSERELIN ACETATE	TRUE	FALSE	TRUE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	0.094099769	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	3.500511415712966	elbasvir / grazoprevir	wikidata:Q22673321	ELBASVIR/GRAZOPREVIR	FALSE	FALSE	FALSE
DOCK8	hgnc:19191	DOCK8	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.038837035	vortioxetine	rxcui:1439834	VORTIOXETINE HYDROBROMIDE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	PharmGKB	4/5/24	NULL	0.048083948	arsenic trioxide	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
XRCC4	hgnc:12831	XRCC4	PharmGKB	4/5/24	NULL	1.265245090016735	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ABCC10	hgnc:52	ABCC10	PharmGKB	4/5/24	NULL	0.2108741816694558	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
AKR1C3	hgnc:386	AKR1C3	PharmGKB	4/5/24	NULL	0.084349673	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
NCF4	hgnc:7662	NCF4	PharmGKB	4/5/24	NULL	0.4884434533552976	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
CYP11B2	hgnc:2592	CYP11B2	ChEMBL	33	inhibitor	1.750255707856483	LEVOKETOCONAZOLE	rxcui:2588846	LEVOKETOCONAZOLE	TRUE	FALSE	FALSE
NELL1	hgnc:7750	NELL1	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
CBS	hgnc:1550	CBS	PharmGKB	4/5/24	NULL	4.200613698855561	l-methionine	rxcui:6837	METHIONINE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.03505185	neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.561579372	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.6364566210387212	acetaminophen glucuronide	chembl:CHEMBL1647	ACETAMINOPHEN GLUCURONIDE	FALSE	FALSE	FALSE
TTC6	hgnc:19739	TTC6	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
UGGT2	hgnc:15664	UGGT2	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
HSD3B1	hgnc:5217	HSD3B1	PharmGKB	4/5/24	NULL	1.141471113819445	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
ILKAP	hgnc:15566	ILKAP	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
XYLT2	hgnc:15517	XYLT2	PharmGKB	4/5/24	NULL	0.5645986154375753	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	PharmGKB	4/5/24	NULL	0.6250913242344582	venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CYP3A7	hgnc:2640	CYP3A7	PharmGKB	4/5/24	NULL	3.750547945	cortisone acetate	rxcui:21655	CORTISONE ACETATE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.031112584	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	0.750109589	interferon alfa-2b, recombinant	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
F7	hgnc:3544	F7	ChEMBL	33	positive modulator	1.250182648468916	EPTACOG ALFA	rxcui:2386863	COAGULATION FACTOR VIIA (RECOMBINANT)-JNCW	TRUE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.097326545	docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	TALC	12-May-16	inhibitor	0.421837528	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.3725599732909588	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	0.060956201	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	1.981421556063943	ROBATUMUMAB	ncit:C71527	ROBATUMUMAB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.2465148884304905	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
UNIPROT:Q9Y5Y4	hgnc:4502	PTGDR2	TdgClinicalTrial	Jan-14	NULL	8.290684931951763	AM-211	chembl:CHEMBL2181753	AM-211	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.1442518440541058	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	ARQ-501	drugbank:DB11948	LAPACHONE	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.2275522047050683	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.2817943000126717	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	0.1400204566285186	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.010939098	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.021878196	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P47898	hgnc:5300	HTR5A	TdgClinicalTrial	Jan-14	NULL	0.525076712	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.037505479	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.020002922	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.070010228	ASENAPINE	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.4861821410712454	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	4.922594178346359	AVANAFIL	rxcui:1291301	AVANAFIL	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.4070362111294147	OLODATEROL	rxcui:1546059	OLODATEROL	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	0.2763561643983921	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P34972	hgnc:2160	CNR2	TdgClinicalTrial	Jan-14	NULL	0.1187956362798518	DRONABINOL	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.6563458904461813	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	CG100649	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	0.7955707762984014	BEZAFIBRATE	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	PEG-SN38	ncit:C70651	FIRTECAN PEGOL	FALSE	FALSE	FALSE
UNIPROT:P22455	hgnc:3691	FGFR4	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	1.826353782111113	AMBRISENTAN	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	LEVETIRACETAM	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	0.6058577450272442	DIHYDROERGOTAMINE	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P68371	hgnc:20771	TUBB4B	TdgClinicalTrial	Jan-14	NULL	0.1265245090016735	MEBENDAZOLE	rxcui:6672	MEBENDAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q15391	hgnc:16442	P2RY14	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:O00398	hgnc:19906	P2RY10	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	0.2734774543525755	MC-1	drugbank:DB05315	MC-1	FALSE	FALSE	FALSE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.212152207	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.3864200913449379	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.421837528	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.3725599732909588	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.3062196950280639	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.1136529680426287	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
UNIPROT:P49721	hgnc:9539	PSMB2	TdgClinicalTrial	Jan-14	NULL	0.3365876361262467	MLN-9708	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
UNIPROT:P41597	hgnc:1603	CCR2	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	MLN-1202	iuphar.ligand:8921	PLOZALIZUMAB	FALSE	FALSE	FALSE
UNIPROT:P20618	hgnc:9537	PSMB1	TdgClinicalTrial	Jan-14	NULL	0.384671584	MLN-9708	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
UNIPROT:P23921	hgnc:10451	RRM1	TdgClinicalTrial	Jan-14	NULL	0.8824818695074704	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
UNIPROT:Q7LG56	hgnc:17296	RRM2B	TdgClinicalTrial	Jan-14	NULL	1.500219178162699	MOTEXAFIN GADOLINIUM	ncit:C1881	MOTEXAFIN GADOLINIUM	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.3968833804663227	NERATINIB	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.6035364509849942	NERAMEXANE	ncit:C76781	NERAMEXANE	FALSE	FALSE	FALSE
UNIPROT:Q9NZ42	hgnc:30100	PSENEN	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	NIC5-15	chembl:CHEMBL493737	METHYLINOSITOL	FALSE	FALSE	FALSE
UNIPROT:Q96BI3	hgnc:29509	APH1A	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	NIC5-15	chembl:CHEMBL493737	METHYLINOSITOL	FALSE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.3182283105193605	NN9924	chembl:CHEMBL4084119	LIRAGLUTIDE	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.2408608772279564	NKTR-181	ncit:C170277	OXYCODEGOL	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.030996264	OCINAPLON	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.089756703	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.1565523888959287	ZOLPIDEM	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
UNIPROT:P15056	hgnc:1097	BRAF	TdgClinicalTrial	Jan-14	NULL	1.657092009619794	VEMURAFENIB	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
UNIPROT:P11532	hgnc:2928	DMD	TdgClinicalTrial	Jan-14	NULL	7.501095891	PRO044	drugbank:DB17003	BMN-044	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	POZANICLINE	ncit:C81045	POZANICLINE	FALSE	FALSE	FALSE
UNIPROT:P11216	hgnc:9723	PYGB	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	PSN357	drugbank:DB05044	PSN357	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	3.424413341458336	TC-6987	drugbank:DB14854	TC-6987	FALSE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	TRAFERMIN	ncit:C152708	TRAFERMIN	FALSE	FALSE	FALSE
UNIPROT:P35225	hgnc:5973	IL13	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	TNX-650	chembl:CHEMBL2109466	TNX-650	FALSE	FALSE	FALSE
UNIPROT:P20618	hgnc:9537	PSMB1	TdgClinicalTrial	Jan-14	NULL	0.5233322714521046	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	VARDENAFIL	rxcui:306674	VARDENAFIL	TRUE	FALSE	FALSE
UNIPROT:O60840	hgnc:1393	CACNA1F	TdgClinicalTrial	Jan-14	NULL	0.08334551	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:Q16552	hgnc:5981	IL17A	TdgClinicalTrial	Jan-14	NULL	0.4039051633514962	VIDOFLUDIMUS	ncit:C152873	VIDOFLUDIMUS	FALSE	FALSE	FALSE
UNIPROT:O00305	hgnc:1404	CACNB4	TdgClinicalTrial	Jan-14	NULL	0.1795134059339982	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.093763699	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	0.2365210416022275	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.008730906	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.012736852	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.3043922970185189	DAPIPRAZOLE	rxcui:22298	DAPIPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	CYCLIZINE	rxcui:2977	CYCLIZINE	TRUE	FALSE	FALSE
UNIPROT:P21817	hgnc:10483	RYR1	TdgClinicalTrial	Jan-14	NULL	2.083637747448194	DANTROLENE	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
MMP13	hgnc:7159	MMP13	ChEMBL	33	inhibitor	1.093909817410302	REBIMASTAT	ncit:C1875	REBIMASTAT	FALSE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	1.400204566285186	DESLANOSIDE	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.1250182648468916	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	GONADORELIN	rxcui:6384	GONADORELIN	TRUE	FALSE	FALSE
UNIPROT:Q13002	hgnc:4580	GRIK2	TdgClinicalTrial	Jan-14	NULL	0.4565884455277783	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.3182283105193606	HEXOBARBITAL	rxcui:5302	HEXOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.09814518	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	3.750547945	HYDROFLUMETHIAZIDE	rxcui:5495	HYDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.089501712	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	INTERFERON ALFACON-1	rxcui:59744	INTERFERON ALFACON-1	TRUE	TRUE	TRUE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	0.8899605294185507	LOSARTAN	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.1219218372345847	LEVOBUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
UNIPROT:P08253	hgnc:7166	MMP2	TdgClinicalTrial	Jan-14	NULL	0.3590268118679965	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	NEPAFENAC	rxcui:298665	NEPAFENAC	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	NIZATIDINE	rxcui:42319	NIZATIDINE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.067317527	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.059532507	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.063300387	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.071341945	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.05814803	NITRAZEPAM	rxcui:7440	NITRAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.051277023	NOREPINEPHRINE	rxcui:7512	NOREPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.8950171233357017	PENBUTOLOL	rxcui:7973	PENBUTOLOL	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.091796628	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P21964	hgnc:2228	COMT	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	TOLCAPONE	rxcui:72937	TOLCAPONE	TRUE	FALSE	FALSE
UNIPROT:P51168	hgnc:10600	SCNN1B	TdgClinicalTrial	Jan-14	NULL	1.823183029	TRIAMTERENE	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
UNIPROT:P18031	hgnc:9642	PTPN1	TdgClinicalTrial	Jan-14	NULL	1.400204566285186	TILUDRONATE	rxcui:11476	TILUDRONIC ACID	TRUE	FALSE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TEND	1-Aug-11	NULL	0.9053046764774914	DIVALPROEX SODIUM	rxcui:266856	DIVALPROEX SODIUM	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.6819178082557728	TUBOCURARINE	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
UNIPROT:P51164	hgnc:820	ATP4B	TEND	1-Aug-11	NULL	0.1442518440541058	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.063160791	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.06466462	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.060353645	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.069638821	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.067059606	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TEND	1-Aug-11	NULL	0.2344092465879218	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.2453629496995069	ESTRIOL	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.280789686	ERGOTAMINE	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.3684748858645228	FESOTERODINE	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.3256289689035318	FORMOTEROL	rxcui:236216	FORMOTEROL FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TEND	1-Aug-11	NULL	0.037721028	IDARUBICIN	rxcui:5650	IDARUBICIN	TRUE	FALSE	TRUE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.4321619031744403	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TEND	1-Aug-11	NULL	0.064111931	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TEND	1-Aug-11	NULL	0.1092771513750145	ISOFLURANE	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	2.500365296937833	MIVACURIUM	rxcui:30077	MIVACURIUM	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.05073205	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.6141248097742046	MIVACURIUM	rxcui:30077	MIVACURIUM	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.693795846312725	OLOPATADINE	rxcui:135391	OLOPATADINE	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TEND	1-Aug-11	NULL	6.563458904461812	NIZATIDINE	rxcui:42319	NIZATIDINE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.116943588	OXANDROLONE	rxcui:7779	OXANDROLONE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.008317388	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.4605936073306534	PROCYCLIDINE	rxcui:8718	PROCYCLIDINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.072927321	PRAZOSIN	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.062733179	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.058799184	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P35499	hgnc:10591	SCN4A	TEND	1-Aug-11	NULL	0.052116795	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.043180651	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TEND	1-Aug-11	NULL	0.091556532	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.0296486	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TEND	1-Aug-11	NULL	0.4906052389860809	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	0.5515511684421691	TACRINE	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.013659644	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.1790034246671403	ZOPICLONE	rxcui:40001	ZOPICLONE	TRUE	FALSE	FALSE
HLA CLASS II ANTIGEN DR10	hgnc:4948	HLA-DRB1	TTD	2020.06.01	NULL	2.386712328895204	Oncolym	chembl:CHEMBL2109447	LYM-1	FALSE	FALSE	FALSE
DOPAMINE D1 RECEPTOR	hgnc:3020	DRD1	TTD	2020.06.01	NULL	0.068369364	Zicronapine	ncit:C152950	ZICRONAPINE	FALSE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.4102161815288632	Carboxyamidotriazole orotate	ncit:C91090	CARBOXYAMIDOTRIAZOLE OROTATE	FALSE	FALSE	FALSE
THYROID HORMONE RECEPTOR BETA	hgnc:11799	THRB	TTD	2020.06.01	NULL	0.5097832158805291	VK-2809	drugbank:DB15137	VK-2809	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.2822993077187876	ATI-2042	ncit:C83563	BUDIODARONE	FALSE	FALSE	FALSE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	1.944728564284981	AB928	ncit:C159564	ETRUMADENANT	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	0.7001022831425933	GMI-1359	drugbank:DB18092	GMI-1359	FALSE	FALSE	FALSE
CYTOTOXIC T-LYMPHOCYTE PROTEIN 4	hgnc:2505	CTLA4	TTD	2020.06.01	NULL	3.500511415712966	MK-1308	ncit:C150679	QUAVONLIMAB	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.6177373086552294	LY3300054	ncit:C128138	LODAPOLIMAB	FALSE	FALSE	FALSE
PROTEIN-SERINE O-PALMITOLEOYLTRANSFERASE PORCUPINE	hgnc:17652	PORCN	TTD	2020.06.01	NULL	26.25383561784724	LGK974	drugbank:DB12561	WNT-974	FALSE	FALSE	FALSE
ANGIOPOIETIN-2	hgnc:485	ANGPT2	TTD	2020.06.01	NULL	3.500511415712966	LY3127804	ncit:C177075	ZANSECIMAB	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE PIM	hgnc:8986	PIM1	TTD	2020.06.01	NULL	0.375054795	PIM447	iuphar.ligand:9790	PIM447	FALSE	FALSE	FALSE
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	1.381780822	PLX2853	ncit:C146825	BRD4 INHIBITOR PLX2853	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.4773424657790409	REVAMILAST	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.2051080907644316	BNZ-1	ncit:C146636	IL-2/9/15 GAMMA CHAIN RECEPTOR INHIBITOR BNZ-1	FALSE	FALSE	FALSE
INTERLEUKIN 15 RECEPTOR ALPHA	hgnc:5978	IL15RA	TTD	2020.06.01	NULL	3.281729452230906	BNZ-1	ncit:C146636	IL-2/9/15 GAMMA CHAIN RECEPTOR INHIBITOR BNZ-1	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	0.2905562835176771	TPX-0005	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
F8	hgnc:3546	F8	ChEMBL	33	positive modulator	3.088686543276147	OCTOCOG ALFA	chembl:CHEMBL2108455	OCTOCOG ALFA	FALSE	FALSE	FALSE
PROTEIN KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	0.182318303	TG02	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
CALGRANULIN D	hgnc:10489	S100A12	TTD	2020.06.01	NULL	3.500511415712966	Eptinezumab	rxcui:2282660	EPTINEZUMAB	TRUE	FALSE	FALSE
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	4.375639269641208	Omaveloxolone	rxcui:2631931	OMAVELOXOLONE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	1.193356164447602	LEO-32731	chembl:CHEMBL3654384	ORISMILAST	FALSE	FALSE	FALSE
INTERLEUKIN-12 ALPHA	hgnc:5969	IL12A	TTD	2020.06.01	NULL	1.750255707856483	Mirikizumab	rxcui:2668384	MIRIKIZUMAB	TRUE	FALSE	FALSE
ATR	hgnc:882	ATR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1944728564284981	BMN673	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	5.250767123569449	AZD7687	iuphar.ligand:7827	AZD7687	FALSE	FALSE	FALSE
INTERLEUKIN-33	hgnc:16028	IL33	TTD	2020.06.01	NULL	4.375639269641208	AMG 282	ncit:C171824	ASTEGOLIMAB	FALSE	FALSE	FALSE
C5A ANAPHYLATOXIN CHEMOTACTIC RECEPTOR	hgnc:1338	C5AR1	TTD	2020.06.01	NULL	6.563458904461812	CCX-168	iuphar.ligand:9450	AVACOPAN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.2465148884304905	Brimonidine	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
PROTON-COUPLED FOLATE TRANSPORTER	hgnc:30521	SLC46A1	TTD	2020.06.01	NULL	0.6250913242344582	Methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.1232574442152452	PQR309	ncit:C111898	BIMIRALISIB	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.4930297768609811	ARQ092	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	0.7134194461371536	ASP-015K	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	1.591141552596802	Alpha-glucosidase	rxcui:2475360	LYSOSOMAL ALPHA-GLUCOSIDASE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4907258993990139	Bicifadine	ncit:C79930	BICIFADINE	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.375054795	Alfentanil	rxcui:203203	ALFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
SERINE PROTEASE UNSPECIFIC	hgnc:11756	TFF2	TTD	2020.06.01	NULL	2.187819634820604	Aprotinin	rxcui:1056	APROTININ	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.5339763176511304	Rescinnamine	rxcui:9259	RESCINNAMINE	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.3704244884352345	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.020688602	Aspirin	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	2.282942227638891	Darusentan	ncit:C75991	DARUSENTAN	FALSE	FALSE	FALSE
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1	hgnc:2357	CRHR1	TTD	2020.06.01	NULL	1.458546423213736	CRA1000	iuphar.ligand:3498	CRA1000	FALSE	FALSE	FALSE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	1.400204566285186	Deslanoside	rxcui:3248	DESLANOSIDE	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.2	hgnc:1389	CACNA1B	TTD	2020.06.01	NULL	0.4102161815288632	LOMERIZINE	ncit:C66029	LOMERIZINE	FALSE	FALSE	FALSE
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	1.750255707856483	Spermidine	rxcui:1483262	SPERMIDINE	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	Dopexamine	rxcui:23638	DOPEXAMINE	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.069454592	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.3977853881492006	Oxaprozin	rxcui:32613	OXAPROZIN	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.2	hgnc:1389	CACNA1B	TTD	2020.06.01	NULL	0.1640864726115453	Ralfinamide	chembl:CHEMBL2107771	RALFINAMIDE	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION GENE 3 PROTEIN	hgnc:6476	LAG3	TTD	2020.06.01	NULL	13.12691780892362	IMP-701	ncit:C122683	IERAMILIMAB	FALSE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	2.917092846427472	SSR-103800	iuphar.ligand:4778	SSR-103800	FALSE	FALSE	FALSE
VITAMIN K EPOXIDE REDUCTASE COMPLEX 1	hgnc:23663	VKORC1	TTD	2020.06.01	NULL	3.500511415712966	Phenprocoumon	rxcui:8150	PHENPROCOUMON	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.750109589	Diphenoxylate	rxcui:3500	DIPHENOXYLATE	TRUE	FALSE	FALSE
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	0.6563458904461812	MEPTAZINOL	rxcui:6761	MEPTAZINOL	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.01835077	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
PUROMYCIN-SENSITIVE AMINOPEPTIDASE	hgnc:7900	NPEPPS	TTD	2020.06.01	NULL	2.625383561784725	CHR-2797	ncit:C70650	TOSEDOSTAT	FALSE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Fluoroquinolone	wikidata:Q28801726	FLUOROQUINOLONE	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.028356978	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PROTEIN KINASE C THETA	hgnc:9410	PRKCQ	TTD	2020.06.01	NULL	0.5250767123569451	Sotrastaurin acetate	ncit:C80631	SOTRASTAURIN ACETATE	FALSE	FALSE	TRUE
PROTEIN KINASE C ALPHA	hgnc:9393	PRKCA	TTD	2020.06.01	NULL	0.4375639269641209	Sotrastaurin acetate	ncit:C80631	SOTRASTAURIN ACETATE	FALSE	FALSE	TRUE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.2	hgnc:1389	CACNA1B	TTD	2020.06.01	NULL	2.461297089173179	Ziconotide	rxcui:68503	ZICONOTIDE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.090821275	Rapamycin	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	0.055563673	tamatinib	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1B	hgnc:278	ADRA1B	TTD	2020.06.01	NULL	0.5073204950308646	Methoxamine	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2275522047050683	TEMSIROLIMUS	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	0.7001022831425933	Nicotinamide	rxcui:7405	NIACINAMIDE	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.400821918	Mapracorat	ncit:C166458	MAPRACORAT	FALSE	FALSE	FALSE
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	4.861821410712453	Tositumomab	rxcui:263010	TOSITUMOMAB	TRUE	FALSE	TRUE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	0.020399251	Curcumin	rxcui:2955	CURCUMIN	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	8.204323630577266	Udenafil	ncit:C74086	UDENAFIL	TRUE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	4.773424657790408	Voglibose	ncit:C95221	VOGLIBOSE	TRUE	FALSE	FALSE
ACTIVATION B7-1 ANTIGEN	hgnc:1700	CD80	TTD	2020.06.01	NULL	5.250767123569449	Abatacept	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.1666910197958555	P1446A-05	ncit:C141430	VORUCICLIB	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Emedastine	rxcui:28144	EMEDASTINE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1400204566285186	TOPOTECAN	rxcui:266573	TOPOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.7955707762984014	Oxeglitazar	ncit:C66259	OXEGLITAZAR	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE BETA-1	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	0.3547815624033412	PF-4708671	iuphar.ligand:8036	PF-4708671	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.2224901323546377	AMG 900	ncit:C82349	AURORA KINASE INHIBITOR AMG 900	FALSE	FALSE	FALSE
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	6.563458904461812	KGP94	iuphar.ligand:6533	KGP94	FALSE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 1	hgnc:1602	CCR1	TTD	2020.06.01	NULL	5.834185692854944	GSK2941266	chembl:CHEMBL4444976	CCX354	FALSE	FALSE	FALSE
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	1.750255707856483	OPB-31121	ncit:C90588	STAT3 INHIBITOR OPB-31121	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	0.6863747873946993	MM-141	ncit:C103863	ISTIRATUMAB	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
GALACTOSIDE 3(4)-L-FUCOSYLTRANSFERASE	hgnc:4014	FUT3	TTD	2020.06.01	NULL	52.50767123569449	Rebmab-100	drugbank:DB17213	HU3S193	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	0.089298761	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	2.407466349146467	Brigatinib	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
MITOCHONDRIAL RRNA METHYLTRANSFERASE 2	hgnc:16352	MRM2	TTD	2020.06.01	NULL	26.25383561784724	Plazomicin	rxcui:2049549	PLAZOMICIN	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Rosoxacin	rxcui:35797	ROSOXACIN	FALSE	FALSE	FALSE
GABA TRANSPORTER GAT-1	hgnc:11042	SLC6A1	TTD	2020.06.01	NULL	3.500511415712966	CI-966	iuphar.ligand:4612	CI-966	FALSE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	2.059124362184097	AZD-4017	drugbank:DB14875	AZD-4017	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	3,3'-DIMETHOXYBENZIDINE	chembl:CHEMBL398363	CHEMBL:CHEMBL398363	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	TBI-1501	ncit:C150377	AUTOLOGOUS ANTI-CD19 CAR-T CELLS TBI-1501	FALSE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	KITE-585	drugbank:DB17409	KITE-585	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.384671584	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	1.467605717767858	Tofacitinib	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.801643836	Betamethasone Benzoate	rxcui:1517	BETAMETHASONE BENZOATE	TRUE	FALSE	FALSE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.577007376	GSI-136	drugbank:DB12819	GSI-136	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.172722603	Cipatinib	drugbank:DB16752	CIPATINIB	FALSE	FALSE	FALSE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	2.019525817	CHF-5074	iuphar.ligand:7339	CHF-5074	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.1591141552596803	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.2333674277141978	Renzapride	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.067317527	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	Ethylestrenol	rxcui:4162	ETHYLESTRENOL	TRUE	FALSE	FALSE
STEROID 17-ALPHA-MONOOXYGENASE	hgnc:2593	CYP17A1	TTD	2020.06.01	NULL	3.125456621172291	ABIRATERONE	rxcui:1100071	ABIRATERONE ACETATE	TRUE	FALSE	TRUE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.8899605294185507	Alacepril	ncit:C75021	ALACEPRIL	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.9944634703730019	FENOFIBRIC ACID	rxcui:24852	FENOFIBRIC ACID	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.058622403945453	Azelastine	rxcui:18603	AZELASTINE	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.03262504	Dexamethasone	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR	hgnc:1571	CCKBR	TTD	2020.06.01	NULL	3.580068493342807	Pentagastrin	rxcui:7993	PENTAGASTRIN	TRUE	FALSE	FALSE
SQLE	hgnc:11279	SQLE	DTC	9/2/20	NULL	1.009762908	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.1801292323694494	Panobinostat	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
ATP-BINDING CASSETTE TRANSPORTER C9	hgnc:60	ABCC9	TTD	2020.06.01	NULL	0.3409589041278863	Repaglinide	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	1.250182648468916	Testolactone	rxcui:10378	TESTOLACTONE	TRUE	FALSE	TRUE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.458240639	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.546954909	SR13668	chembl:CHEMBL245030	SR-13668	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.2625383561784725	TAK-593	drugbank:DB13093	TAK-593	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	1.944728564284981	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	3.281729452230906	BMS-188797	ncit:C1859	BMS-188797	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.8899605294185507	CL-329167	chembl:CHEMBL275875	CL-329167	FALSE	FALSE	FALSE
GLUCOSYLCERAMIDASE	hgnc:4177	GBA1	TTD	2020.06.01	NULL	1.500219178	Isofagomine tartrate	chembl:CHEMBL2105671	AFEGOSTAT TARTRATE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	TRIMEPRAZINE TARTRATE	rxcui:164308	TRIMEPRAZINE TARTRATE	TRUE	FALSE	FALSE
LEUKOTRIENE B4 RECEPTOR 1	hgnc:6713	LTB4R	TTD	2020.06.01	NULL	0.8204323630577265	LTB4	iuphar.ligand:2487	LTB4	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	0.088396753	METHYLENEDIOXYMETHAMPHETAMINE	ncit:C61081	3,4-METHYLENEDIOXYMETHAMPHETAMINE	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	2.143170254518142	LY-517717	drugbank:DB05713	LY-517717	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	1.372749574789398	MEHD-7945A	ncit:C116628	DULIGOTUZUMAB	FALSE	TRUE	TRUE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	0.7684049449126024	Resiniferatoxin	ncit:C1214	RESINIFERATOXIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	0.1190650141398968	PBT-2	drugbank:DB05565	PBT-1033	FALSE	FALSE	FALSE
THYROTROPIN-RELEASING HORMONE RECEPTOR	hgnc:12299	TRHR	TTD	2020.06.01	NULL	8.751278539282415	AZETIRELIN	ncit:C74408	AZETIRELIN	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.7955707762984014	N-(4-CARBOXYPHENYL)RHODANINE	chembl:CHEMBL450802	CHEMBL:CHEMBL450802	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.05751114	IUPHAR.LIGAND:31	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.079077818	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.5527123287967842	GNF-PF-3542	chembl:CHEMBL598477	CHEMBL:CHEMBL598477	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.2692701089009974	IUPHAR.LIGAND:145	iuphar.ligand:145	5-MEO-DMT	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.053199262	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.08334551	IUPHAR.LIGAND:17	ncit:C76104	LYSERGIDE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:157	iuphar.ligand:157	(R)-DOI	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:144	drugbank:DB01445	BUFOTENINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.052090944	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.005483257	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.061412481	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.061412481	IUPHAR.LIGAND:91	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.03251249	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:167	iuphar.ligand:167	S 16924	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1105424657593568	IUPHAR.LIGAND:17	ncit:C76104	LYSERGIDE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.1779921058837101	IUPHAR.LIGAND:17	ncit:C76104	LYSERGIDE	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	inhibitor	0.064347636	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.098884503	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	agonist	0.1112450661773188	IUPHAR.LIGAND:115	iuphar.ligand:115	TFMPP	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.038693936	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.3777530304726222	IUPHAR.LIGAND:8963	iuphar.ligand:8963	BO1	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.010113188	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:1924	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:8147	iuphar.ligand:8147	COMPOUND 24 [PMID: 23441572]	FALSE	FALSE	FALSE
NCBIGENE:1785	hgnc:2974	DNM2	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:12485	iuphar.ligand:12485	COMPOUND 7 [NGUYEN ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:11588	iuphar.ligand:11588	COMPOUND 17 [PMID: 34176264]	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.1693795846312726	IUPHAR.LIGAND:10474	ncit:C169804	BELIZATINIB	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.01644462	IUPHAR.LIGAND:5714	iuphar.ligand:5714	NVP-TAE684	FALSE	FALSE	FALSE
NCBIGENE:2611	hgnc:4147	GAPDHP69	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:4842	rxcui:30009	MIGLITOL	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1422972120208523	IUPHAR.LIGAND:488	rxcui:236495	TAMSULOSIN HYDROCHLORIDE	TRUE	FALSE	TRUE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:490	iuphar.ligand:490	A-119637	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:502	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	FIPEXIDE	ncit:C65685	FIPEXIDE	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.094438258	IUPHAR.LIGAND:223	iuphar.ligand:223	[3H]RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:502	rxcui:8153	PHENTOLAMINE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3456	ncit:C72100	MIBOLERONE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	PERVILLEINE C	chembl:CHEMBL451845	PERVILLEINE C	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7893	iuphar.ligand:7893	LISINOPRIL-TRYPTOPHAN	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:10557	iuphar.ligand:10557	COMPOUND 15A	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:459	iuphar.ligand:459	MRE 3008F20	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.05486695	IUPHAR.LIGAND:5617	iuphar.ligand:5617	LAS38096	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:3281	ncit:C96199	DERENOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:409	rxcui:1536070	FLAVONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:418	iuphar.ligand:418	CGS 24012	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:469	iuphar.ligand:469	MRS1186	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:467	iuphar.ligand:467	MRS1097	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:5614	ncit:C76394	PRELADENANT	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	OSAJIN	chembl:CHEMBL238188	OSAJIN	FALSE	FALSE	FALSE
NCBIGENE:1934	hgnc:3209	EEF1B2P2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12776	iuphar.ligand:12776	A011	FALSE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8374	iuphar.ligand:8374	OLODANRIGAN	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:6175	iuphar.ligand:6175	GASTRIN RELEASING PEPTIDE(14-27) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:3127	hgnc:4953	HLA-DRB5	GuideToPharmacology	2024.1	antibody	10.50153424713889	IUPHAR.LIGAND:11026	iuphar.ligand:11026	MEPLAZUMAB	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:618	iuphar.ligand:618	RANATENSIN	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7853	iuphar.ligand:7853	EXAMPLE 20 [WO2010128058]	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9761	iuphar.ligand:9761	COMPOUND 9 [PMID: 26006010]	FALSE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.065145994	IUPHAR.LIGAND:551	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.5645986154375752	NSC-127133	chembl:CHEMBL1172911	CHEMBL:CHEMBL1172911	FALSE	FALSE	FALSE
NCBIGENE:2333	hgnc:1067	BMP1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8562	iuphar.ligand:8562	COMPOUND 2 [PMID: 11934595]	FALSE	FALSE	FALSE
NCBIGENE:1786	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:8481	iuphar.ligand:8481	LDN-214117	FALSE	FALSE	FALSE
NCBIGENE:1941	hgnc:18041	BMP2K	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8206	iuphar.ligand:8206	COMPOUND 5M [PMID: 20483621]	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
NCBIGENE:2730	hgnc:4312	GCLM	GuideToPharmacology	2024.1	NULL	2.019525817	IUPHAR.LIGAND:9523	iuphar.ligand:9523	OF-1	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:7034	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
NCBIGENE:2725	hgnc:1104	BRD3	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:6004	drugbank:DB02656	LY-294002	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.1744440904840348	IUPHAR.LIGAND:7034	ncit:C171748	APABETALONE	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7808	iuphar.ligand:7808	ET BROMODOMAIN INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:10534	iuphar.ligand:10534	DBET6	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.077444943	8-FLUOROTRYPTANTHRIN	chembl:CHEMBL1098875	CHEMBL:CHEMBL1098875	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.4070362111294147	IUPHAR.LIGAND:11690	iuphar.ligand:11690	GSK852	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:10044	ncit:C147125	ABIVERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:11628	rxcui:2629338	PIRTOBRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:9761	iuphar.ligand:9761	COMPOUND 9 [PMID: 26006010]	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:670	iuphar.ligand:670	JMV1116	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:650	iuphar.ligand:650	KALLIDIN	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:650	iuphar.ligand:650	KALLIDIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.01823183	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:9449	iuphar.ligand:9449	COMPOUND 17 [PMID: 24257095]	FALSE	FALSE	FALSE
NCBIGENE:2948	hgnc:4636	GSTM4	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:9616	iuphar.ligand:9616	POM2-C-HMBP	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.1597596487901455	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:656	iuphar.ligand:656	JMV1431	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:3846	iuphar.ligand:3846	[PHE8,&PSI;(CH2-NH)ARG9]BK	FALSE	FALSE	FALSE
NCBIGENE:2336	hgnc:1476	CAPN1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11643	iuphar.ligand:11643	CALPEPTIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	SODIUM DIMETHYLCARBAMODITHIOATE	chembl:CHEMBL569460	SODIUM DIMETHYLCARBAMODITHIOATE	FALSE	FALSE	FALSE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:11344	iuphar.ligand:11344	C5APEP	FALSE	FALSE	FALSE
NCBIGENE:2336	hgnc:1476	CAPN1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11701	iuphar.ligand:11701	UAWJ9-36-3	FALSE	FALSE	FALSE
NCBIGENE:1622	hgnc:2690	DBI	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8566	iuphar.ligand:8566	AC-VEID-CHO	FALSE	FALSE	FALSE
NCBIGENE:528	hgnc:856	ATP6V1C1	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:2523	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	activator	0.6105543166941221	IUPHAR.LIGAND:2511	iuphar.ligand:2511	BAYK 8644	FALSE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	0.1544343271638073	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:388	hgnc:668	RHOB	GuideToPharmacology	2024.1	blocker	5.834185692854944	IUPHAR.LIGAND:4212	iuphar.ligand:4212	HC-056456	FALSE	FALSE	FALSE
NCBIGENE:389	hgnc:669	RHOC	GuideToPharmacology	2024.1	activator	0.4375639269641209	IUPHAR.LIGAND:1883	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9607	iuphar.ligand:9607	BMS-202	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.1973972602845657	IUPHAR.LIGAND:731	iuphar.ligand:731	HU-210	FALSE	FALSE	FALSE
NCBIGENE:67	hgnc:140	ACTBP7	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:3646	iuphar.ligand:3646	CCL27	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:9497	iuphar.ligand:9497	BMS-817399	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:3649	iuphar.ligand:3649	CCL28	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:794	iuphar.ligand:794	[125I]CCL11 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	0.070197421	IUPHAR.LIGAND:4190	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:9850	iuphar.ligand:9850	GW406381	FALSE	FALSE	FALSE
NCBIGENE:718	hgnc:1318	C3	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:720	hgnc:1323	C4A	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:725	hgnc:1328	C4BPB	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:724	hgnc:1327	C4BPAP2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:716	hgnc:1247	C1S	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:733	hgnc:1354	C8G	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2899	iuphar.ligand:2899	ISOTHIOUREA-1T	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:12511	iuphar.ligand:12511	QR-6401	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:9903	iuphar.ligand:9903	SAMURACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:10426	ncit:C151988	EBVACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:11189	iuphar.ligand:11189	DALPICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:9626	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:5947	iuphar.ligand:5947	CDK1/5 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:10426	ncit:C151988	EBVACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.3621218705909966	IUPHAR.LIGAND:11885	iuphar.ligand:11885	TANUXICICLIB	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:5662	iuphar.ligand:5662	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:9887	iuphar.ligand:9887	JH-XI-10-02	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.1646008502686348	IUPHAR.LIGAND:7938	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.2586584789935689	IUPHAR.LIGAND:9626	rxcui:2479690	TRILACICLIB	TRUE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:9903	iuphar.ligand:9903	SAMURACICLIB	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:3353	iuphar.ligand:3353	LTD4	FALSE	FALSE	FALSE
NCBIGENE:2743	hgnc:4329	GLRB	GuideToPharmacology	2024.1	antibody	0.5834185692854945	IUPHAR.LIGAND:8462	rxcui:2619313	TREMELIMUMAB	TRUE	TRUE	TRUE
NCBIGENE:1444	hgnc:2442	CSHL1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5136	iuphar.ligand:5136	AMINOOXYACETIC ACID	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:3412	iuphar.ligand:3353	LTD4	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:12766	ncit:C171708	TOLUDESVENLAFAXINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.4646696569530486	IUPHAR.LIGAND:9065	iuphar.ligand:9065	[3H][D-ALA2]DELTORPHIN I	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:1643	iuphar.ligand:1643	&BETA;-ENDORPHIN	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1620	iuphar.ligand:1620	DYNORPHIN A	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:1608	iuphar.ligand:1608	DPDPE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1618	iuphar.ligand:1618	DYNORPHIN-(1-11)	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	inhibitor	0.092933931	IUPHAR.LIGAND:7471	rxcui:1516803	ALVIMOPAN ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:9906	ncit:C87623	TENELIGLIPTIN	FALSE	FALSE	FALSE
NCBIGENE:2357	hgnc:3826	FPR1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:6310	rxcui:596554	VILDAGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.031822831	IUPHAR.LIGAND:204	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.020591244	IUPHAR.LIGAND:90	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.063645662	IUPHAR.LIGAND:177	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.036847489	IUPHAR.LIGAND:7281	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.011799477	IUPHAR.LIGAND:7227	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.016856395	IUPHAR.LIGAND:62	iuphar.ligand:62	(+)-BUTACLAMOL	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.1630673019742065	IUPHAR.LIGAND:62	iuphar.ligand:62	(+)-BUTACLAMOL	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:3304	ncit:C87494	ECOPIPAM HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1896	hgnc:3157	EDA	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:6143	iuphar.ligand:6143	ECTODYSPLASIN A2	FALSE	FALSE	FALSE
NCBIGENE:2487	hgnc:3959	FRZB	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:11784	iuphar.ligand:11784	AZ14117230	FALSE	FALSE	FALSE
NCBIGENE:1566	ncbigene:1566	CYP2D7BP	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9682	iuphar.ligand:9682	COMPOUND 2G [PMID: 27390066]	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7013	iuphar.ligand:7013	EI1	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:7717	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.038467158	IUPHAR.LIGAND:7816	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
NCBIGENE:1400	hgnc:2365	CRMP1	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:5244	iuphar.ligand:5244	PF750	FALSE	FALSE	FALSE
NCBIGENE:1401	hgnc:2367	CRP	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5206	iuphar.ligand:5206	JNJ1661010	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:1051	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:8639	iuphar.ligand:8639	COMPOUND 7R [PMID: 26080733]	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:12485	iuphar.ligand:12485	COMPOUND 7 [NGUYEN ET AL., 2023]	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.2273059360852575	IUPHAR.LIGAND:9786	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:12249	iuphar.ligand:12249	COMPOUND 6LI [CHAN ET AL., 2022]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.008123093	IUPHAR.LIGAND:5962	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:9601	iuphar.ligand:9601	CATEQUENTINIB	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.043180651	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.068369364	IUPHAR.LIGAND:5672	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.071439008	IUPHAR.LIGAND:9428	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.027781837	IUPHAR.LIGAND:5705	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6251	iuphar.ligand:6251	SCK&BETA;8-1	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6249	iuphar.ligand:6249	UPAR FRAGMENT	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:5834	iuphar.ligand:5834	COMPOUND R-(-)-5F [PMID: 22607879]	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1046	iuphar.ligand:1046	HP(2-20)	FALSE	FALSE	FALSE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:1045	iuphar.ligand:1045	F2L-[125I]TYR	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:11283	iuphar.ligand:11283	BAY-6672	FALSE	FALSE	FALSE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:10428	iuphar.ligand:10428	COMPOUND 25 [PMID: 31260299]	FALSE	FALSE	FALSE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:9186	iuphar.ligand:9186	ECF506	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.9907107780319716	IUPHAR.LIGAND:3486	iuphar.ligand:3486	2,3-DIHYDRO-1,4-DITHIIN-1,1,4,4-TETROXIDE	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:3896	iuphar.ligand:3896	M15	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6134	iuphar.ligand:6134	GALANIN(5-29) (RAT/MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:3896	iuphar.ligand:3896	M15	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6075	iuphar.ligand:6075	J18 (GALANIN ANALOGUE)	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3188	drugbank:DB07409	(1-HYDROXY-1-PHOSPHONO-2-[1,1';4',1'']TERPHENYL-3-YL-ETHYL)-PHOSPHONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:4818	rxcui:236875	TIAGABINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.2442217266776488	IUPHAR.LIGAND:7077	rxcui:4461	FLUOCINOLONE ACETONIDE	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	blocker	0.1682938180631233	IUPHAR.LIGAND:4282	ncit:C738	PHENCYCLIDINE	FALSE	FALSE	FALSE
NCBIGENE:936	hgnc:1647	CD24P2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:4667	iuphar.ligand:4667	ORG 25543	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:3878	iuphar.ligand:3878	GNRH III	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12283	rxcui:2621019	LINZAGOLIX	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:5583	iuphar.ligand:5583	[AC-D-2NAL1,D4CPA2,D-3PAL3,6,LEU8, D-ALA10]GNRH-II	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:12394	iuphar.ligand:12394	MERIGOLIX	FALSE	FALSE	FALSE
NCBIGENE:1471	hgnc:2475	CST3	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:2369	hgnc:3877	FRA1J	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8650	iuphar.ligand:8650	COMPOUND 20 [PMID:12127536]	FALSE	FALSE	FALSE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:9066	ncit:C171663	CENDERITIDE	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5789	iuphar.ligand:5789	COMPOUND 21 [PMID: 21185185]	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.2430910705356226	IUPHAR.LIGAND:9426	ncit:C121641	CITARINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:9426	ncit:C121641	CITARINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:9426	ncit:C121641	CITARINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.2134458180312784	IUPHAR.LIGAND:9426	ncit:C121641	CITARINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:12179	iuphar.ligand:12179	COMPOUND 35M [PMID: 36073117]	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:12269	iuphar.ligand:12269	KA2507	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:7007	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.3000438356325399	IUPHAR.LIGAND:7010	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:1221	ncit:C72108	ARPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:7346	iuphar.ligand:7346	MK-0249	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.007941269	IUPHAR.LIGAND:86	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:1226	iuphar.ligand:1226	IMPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.027433475	IUPHAR.LIGAND:204	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:1218	iuphar.ligand:1218	ABT-239	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.2573905452730122	IUPHAR.LIGAND:1242	iuphar.ligand:1241	N-[3H]METHYLHISTAMINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1249	iuphar.ligand:1249	IMBUTAMINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:1248	iuphar.ligand:1248	DIMAPRIT	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1258	iuphar.ligand:1258	A-304121	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:1218	iuphar.ligand:1218	ABT-239	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9873	iuphar.ligand:9873	VUF14738	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:1266	iuphar.ligand:1266	IODOPHENPROPIT	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.096521454	IUPHAR.LIGAND:1267	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2961	iuphar.ligand:2961	COMPOUND 18 [PMID: 8426367]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	0.038467158	IUPHAR.LIGAND:2739	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5564	iuphar.ligand:5564	CID1172084	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:5570	iuphar.ligand:5570	CP55,667	FALSE	FALSE	FALSE
NCBIGENE:3019	hgnc:27269	IDO2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12668	iuphar.ligand:12668	EXAMPLE 184 [WO2014186035]	FALSE	FALSE	FALSE
NCBIGENE:2624	hgnc:4171	GATA2	GuideToPharmacology	2024.1	inhibitor	0.1988926940746004	IUPHAR.LIGAND:6845	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9579	iuphar.ligand:9579	COMPOUND II [PMID: 21329883]	FALSE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8196	iuphar.ligand:8196	COMPOUND 17D [PMID: 23099093]	FALSE	FALSE	FALSE
NCBIGENE:2039	hgnc:3382	DMTN	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:5986	iuphar.ligand:5986	IKK-2 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:11565	iuphar.ligand:11565	COMPOUND 13AC [PMID: 33256400]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.09869863	IUPHAR.LIGAND:1606	rxcui:8001	PENTAZOCINE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:1643	iuphar.ligand:1643	&BETA;-ENDORPHIN	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:9913	iuphar.ligand:9913	FLUMBATINIB	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:12383	iuphar.ligand:12383	RISVODETINIB	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:11963	iuphar.ligand:11963	DIVARASIB	FALSE	FALSE	FALSE
NCBIGENE:521	hgnc:846	ATP5ME	GuideToPharmacology	2024.1	activator	0.9376369863516875	IUPHAR.LIGAND:1051	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
NCBIGENE:526	hgnc:854	ATP6V1B2	GuideToPharmacology	2024.1	activator	1.750255707856483	IUPHAR.LIGAND:2509	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	activator	1.591141552596802	IUPHAR.LIGAND:2308	iuphar.ligand:2308	NS1643	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	0.1262203635473425	IUPHAR.LIGAND:2611	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	activator	0.2430910705356227	IUPHAR.LIGAND:2597	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
NCBIGENE:2830	hgnc:4515	GPR6	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:8232	iuphar.ligand:8232	UNC1215	FALSE	FALSE	FALSE
NCBIGENE:1515	hgnc:2538	CTSV	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:5672	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	activator	0.1620607136904151	IUPHAR.LIGAND:2597	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6712	iuphar.ligand:6712	COMPOUND 4 [PMID: 22533316]	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.2143170254518142	IUPHAR.LIGAND:8136	iuphar.ligand:8136	COMPOUND 2 [PMID: 15546730]	FALSE	FALSE	FALSE
NCBIGENE:1271	hgnc:2170	CNTFR	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:5150	rxcui:1374	BENSERAZIDE	TRUE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:2913	iuphar.ligand:2913	ALKYL OMPT	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:2309	iuphar.ligand:2309	PAXILLINE	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:2688	iuphar.ligand:2688	L-783483	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:10034	iuphar.ligand:10034	IMB-808	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:2912	iuphar.ligand:2912	OMPT	FALSE	FALSE	FALSE
NCBIGENE:274	hgnc:1052	BIN1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:2915	iuphar.ligand:2915	&ALPHA;-FLUOROMETHYLENEPHOSPHONATE	FALSE	FALSE	FALSE
NCBIGENE:2105	hgnc:7111	MKNK2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:12385	iuphar.ligand:12385	TINODASERTIB	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1304	iuphar.ligand:1304	ATC0065	FALSE	FALSE	FALSE
NCBIGENE:281	hgnc:479	AMYP1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1298	iuphar.ligand:1298	MELANIN-CONCENTRATING HORMONE	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:6546	iuphar.ligand:6546	PG-106	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:3052	drugbank:DB07841	GERANYLGERANYL DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:1393	iuphar.ligand:1393	EGLUMEGAD	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:1392	iuphar.ligand:1392	(2R,3R)-APDC	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6213	iuphar.ligand:6213	[18F]FITM	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6334	iuphar.ligand:6334	[18F]MK-1312	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	0.251232877	IUPHAR.LIGAND:7744	iuphar.ligand:7744	RGB-286638	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:7942	iuphar.ligand:7942	REFAMETINIB	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:5441	iuphar.ligand:5441	LY593093	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:8604	iuphar.ligand:8604	BODIPY-PIRENZEPINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:8598	iuphar.ligand:8598	CY3B-TELENZEPINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:329	rxcui:8761	PROPANTHELINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:8583	iuphar.ligand:8583	UH-AH 37	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:326	iuphar.ligand:326	LITHOCHOLYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1491695205559502	IUPHAR.LIGAND:345	ncit:C152880	VINBURNINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.049723174	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:328	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1491695205559502	IUPHAR.LIGAND:322	iuphar.ligand:322	HEXAHYDRODIFENIDOL	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:10104	iuphar.ligand:10104	(S)-DIMETINDENE	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:12324	iuphar.ligand:12324	UCM1341	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:10518	iuphar.ligand:10518	BILORPHIN	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1610	iuphar.ligand:1610	ETHYLKETOCYCLAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:750	hgnc:1197	GAS8-AS1	GuideToPharmacology	2024.1	blocker	13.12691780892362	IUPHAR.LIGAND:4160	iuphar.ligand:4160	CO2+	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	NULL	0.1442518440541057	IUPHAR.LIGAND:10482	iuphar.ligand:10482	COMPOUND 16 [PMID: 31498617]	FALSE	FALSE	FALSE
PSMA6	hgnc:9535	PSMA6	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	blocker	0.1930429089547592	IUPHAR.LIGAND:2623	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3995	iuphar.ligand:3995	A-582941	FALSE	FALSE	FALSE
NCBIGENE:467	hgnc:785	ATF3	GuideToPharmacology	2024.1	blocker	1.875273972703375	IUPHAR.LIGAND:3963	ncit:C75979	HEXAMETHONIUM	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:2110	ncit:C170264	OSANETANT	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:2117	ncit:C166502	IBODUTANT	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:2090	iuphar.ligand:2090	NEUROKININ B	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:2098	iuphar.ligand:2098	SUBSTANCE P	FALSE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	DTC	9/2/20	NULL	0.546954909	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5767	iuphar.ligand:5767	PD 161182	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1468	iuphar.ligand:1468	NEUROMEDIN S-33	FALSE	FALSE	FALSE
NCBIGENE:302	hgnc:537	ANXA2	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:7929	iuphar.ligand:7929	RTI-118	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1482	iuphar.ligand:1482	Y-RFRP-3	FALSE	FALSE	FALSE
NCBIGENE:2129	hgnc:14311	NUAK1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
NCBIGENE:2129	hgnc:14311	NUAK1	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:9176	iuphar.ligand:9176	WZ4002	FALSE	FALSE	TRUE
PSMB10	hgnc:9538	PSMB10	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:3085	ncbigene:3085	HMG1P	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:10384	iuphar.ligand:10384	NUDT7-COV-1	FALSE	FALSE	FALSE
NCBIGENE:1222	hgnc:13819	SLCO1C1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:1608	iuphar.ligand:1608	DPDPE	FALSE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	inhibitor	0.024141458	IUPHAR.LIGAND:1024	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
PSMB9	hgnc:9546	PSMB9	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	inhibitor	0.1615620653405984	IUPHAR.LIGAND:3439	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.2386712328895204	IUPHAR.LIGAND:2190	iuphar.ligand:2190	D[LEU4]AVP	FALSE	FALSE	FALSE
NCBIGENE:1021	hgnc:1777	CDK6	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8826	iuphar.ligand:8826	DISPROCYNIUM24	FALSE	FALSE	FALSE
PSMA8	hgnc:22985	PSMA8	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.3182283105193605	IUPHAR.LIGAND:2196	iuphar.ligand:2196	OPC-21268	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:3338	iuphar.ligand:3338	MRS2365	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:1715	iuphar.ligand:1715	DATP&ALPHA;S	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2670	ncit:C98152	REGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2699	iuphar.ligand:2699	NTZDPA	FALSE	FALSE	FALSE
PSMB4	hgnc:9541	PSMB4	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2659	iuphar.ligand:2659	LY-465608	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:2688	iuphar.ligand:2688	L-783483	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.016856395	IUPHAR.LIGAND:7955	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:10142	iuphar.ligand:10142	PQR620	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:7963	iuphar.ligand:7963	PILARALISIB	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:8012	iuphar.ligand:8012	PIK-75	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.022691301	IUPHAR.LIGAND:8952	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
PSMB6	hgnc:9543	PSMB6	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.2949869170544634	IUPHAR.LIGAND:9826	iuphar.ligand:9826	GSK1059615	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:10702	iuphar.ligand:10702	COMPOUND 15A [PMID: 32069401]	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.053633985	IUPHAR.LIGAND:7965	iuphar.ligand:7965	ZSTK474	FALSE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:11204	iuphar.ligand:11204	AZD8154	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.064111931	IUPHAR.LIGAND:7794	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
NCBIGENE:1297	hgnc:2217	COL9A1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:11626	drugbank:DB14885	PF-05180999	FALSE	FALSE	FALSE
NCBIGENE:3207	hgnc:5101	HOXA11	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12221	iuphar.ligand:12221	COMPOUND 3 [PMID: 26055709]	FALSE	FALSE	FALSE
PSMC1	hgnc:9547	PSMC1	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	8.204323630577266	IUPHAR.LIGAND:11577	ncit:C74086	UDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:9552	iuphar.ligand:9552	NITROSOPRODENAFIL	FALSE	FALSE	FALSE
NCBIGENE:1306	hgnc:2192	COL15A1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5270	iuphar.ligand:5270	SCH51866	FALSE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.2143170254518143	IUPHAR.LIGAND:8214	iuphar.ligand:8214	COMPOUND 14K [PMID: 21982499]	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:10671	iuphar.ligand:10671	MC2050	FALSE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8731	iuphar.ligand:8731	COMPOUND 10B [PMID: 26222319]	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:8662	iuphar.ligand:8662	APR19	FALSE	FALSE	FALSE
PSMD8	hgnc:9566	PSMD8	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:2759	iuphar.ligand:2759	5&BETA;-PREGNANE-3,20-DIONE	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:2766	iuphar.ligand:2766	3-KETO-LITHOCHOLIC ACID	FALSE	FALSE	FALSE
NCBIGENE:3145	hgnc:4982	HMBS	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11167	drugbank:DB12561	WNT-974	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1794	iuphar.ligand:1794	[HIS5]PTH-(1-34) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1790	iuphar.ligand:1790	PTHRP-(1-36)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1798	iuphar.ligand:1798	[ILE5,TRP23]PTHRP-(1-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:8299	rxcui:1921069	ABALOPARATIDE	TRUE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1794	iuphar.ligand:1794	[HIS5]PTH-(1-34) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:735	hgnc:1358	C9	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.00445925	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
NCBIGENE:736	hgnc:8600	PANX2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
SHFM1	hgnc:10845	SEM1	DTC	9/2/20	NULL	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NCBIGENE:2915	hgnc:4597	GRM5	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:9350	iuphar.ligand:9350	VER-246608	FALSE	FALSE	FALSE
NCBIGENE:598	hgnc:992	BCL2L1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:2738	iuphar.ligand:2738	CHOLESTEROL SULPHATE	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10045	iuphar.ligand:10045	CINTIRORGON	FALSE	FALSE	FALSE
NCBIGENE:1529	ncbigene:1529	CYB5P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8139	iuphar.ligand:8139	COMPOUND 25B [PMID: 22564207]	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:11464	iuphar.ligand:11464	NANOLUCIFERASE-LABELLED RELAXIN	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.015193192	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:1525	hgnc:2559	CXADR	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:12617	iuphar.ligand:12617	GLXC-26326	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8331	iuphar.ligand:8331	A(C10/15S)INSL3	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:3885	iuphar.ligand:3885	INSL3 B-CHAIN ANALOGUE	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:12098	iuphar.ligand:12098	ICANBELIMOD	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:6992	iuphar.ligand:6992	VPC03090-P	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:2909	iuphar.ligand:2909	VPC12249	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	DESMETHOXYYANGONIN	chembl:CHEMBL254218	DESMETHOXYYANGONIN	FALSE	FALSE	FALSE
NCBIGENE:3213	hgnc:5114	HOXB3	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:12281	iuphar.ligand:12281	YTK-2205	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:2925	iuphar.ligand:2925	AUY954	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	TODRALAZINE	ncit:C77080	TODRALAZINE	FALSE	FALSE	FALSE
NCBIGENE:3020	hgnc:4764	H3-3A	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10130	iuphar.ligand:10130	SPRI3	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:2929	iuphar.ligand:2929	COMPOUND 26 [PMID: 16190743]	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	DOCONEXENT	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
NCBIGENE:2883	hgnc:10732	SEMA4D	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:8932	iuphar.ligand:8932	PEPINEMAB	FALSE	FALSE	FALSE
NCBIGENE:3103	hgnc:10721	SELP	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:10550	rxcui:2262279	CRIZANLIZUMAB	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.5707355569097228	GEDUNIN	chembl:CHEMBL465226	GEDUNIN	FALSE	FALSE	FALSE
NCBIGENE:2714	ncbigene:2714	GKP4	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:7021	iuphar.ligand:7021	AZ505	FALSE	FALSE	FALSE
NCBIGENE:1041	hgnc:1802	CDSN	GuideToPharmacology	2024.1	NULL	0.5048814541893702	IUPHAR.LIGAND:4532	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:10654	ncit:C150375	LICOGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:9394	ncit:C166685	IPRAGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:833	hgnc:1493	CARS1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6794	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:4588	iuphar.ligand:4588	REMOGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:9395	ncit:C152676	TOFOGLIFLOZIN ANHYDROUS	FALSE	FALSE	FALSE
NCBIGENE:2514	hgnc:11120	SMPD1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10640	iuphar.ligand:10640	COMPOUND 21B [PMID: 31944697]	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3137	iuphar.ligand:3137	YM-75440	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:8136	iuphar.ligand:8136	COMPOUND 2 [PMID: 15546730]	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	GNF-PF-3756	chembl:CHEMBL597035	CHEMBL:CHEMBL597035	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.09869863	IUPHAR.LIGAND:8487	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:2014	iuphar.ligand:2014	L-362,855	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2034	iuphar.ligand:2034	BIM 23030	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.1215455352678113	(-)-USNIC ACID	chembl:CHEMBL461903	(-)-USNIC ACID	FALSE	FALSE	FALSE
NCBIGENE:632	hgnc:1043	BGLAP	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:10484	iuphar.ligand:10484	RJW100	FALSE	FALSE	FALSE
NCBIGENE:2740	hgnc:4324	GLP1R	GuideToPharmacology	2024.1	inhibitor	0.1591141552596802	IUPHAR.LIGAND:7915	iuphar.ligand:7915	PFI-3	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6291	iuphar.ligand:6291	1,6-HEXAMETHYLENE DIISOCYANATE	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.1491695205559502	IUPHAR.LIGAND:4270	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.2386712328895204	IUPHAR.LIGAND:4164	iuphar.ligand:4164	CU2+	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	1.640864726115453	IUPHAR.LIGAND:12527	iuphar.ligand:12527	GFB-8438	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.1750255707856483	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:4232	iuphar.ligand:4232	KB-R7943	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.1491695205559502	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.251232877	IUPHAR.LIGAND:2434	iuphar.ligand:2434	LA3+	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	blocker	1.458546423213736	IUPHAR.LIGAND:11862	iuphar.ligand:11862	PRU-12	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	TCMDC-124585	chembl:CHEMBL587856	CHEMBL:CHEMBL587856	FALSE	FALSE	FALSE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	blocker	0.7292732116068681	IUPHAR.LIGAND:710	rxcui:1483263	SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.068191781	IUPHAR.LIGAND:2461	iuphar.ligand:2461	CAPSAZEPINE	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	1.944728564284981	IUPHAR.LIGAND:4295	iuphar.ligand:4295	RN1747	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.9131768910555564	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1870	hgnc:3114	E2F2	GuideToPharmacology	2024.1	NULL	10.50153424713889	IUPHAR.LIGAND:5074	iuphar.ligand:5074	TUMOUR NECROSIS FACTOR SHED FORM	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.5585922471882393	IUPHAR.LIGAND:9271	iuphar.ligand:9271	MPS1-IN-1	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:10156	iuphar.ligand:10156	JAK3 INHIBITOR 32	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	1.467605717767858	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
NCBIGENE:2429	hgnc:3939	FRA9E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8880	iuphar.ligand:8880	IU1	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.089298761	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
NCBIGENE:2271	hgnc:3700	FH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11340	iuphar.ligand:11340	SBP-7455	FALSE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:2775	ncit:C80885	LEXACALCITOL	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:11454	ncit:C152319	SELEPRESSIN	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2215	iuphar.ligand:2215	D(CH2)5[D-ILE2,ILE4,ALA-NH2]AVP	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:1515	iuphar.ligand:1515	PEPTIDE YY	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.1620607136904151	PI3K-ALPHA INHIBITOR MEN1611	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	CIViC	10-Apr-24	NULL	0.3697723326457359	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	CIViC	10-Apr-24	NULL	0.088333021	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.6019397937072561	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.546954909	ANTI-HER3 MONOCLONAL ANTIBODY GSK2849330	ncit:C111997	ANTI-HER3 MONOCLONAL ANTIBODY GSK2849330	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	0.073054151	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	CIViC	10-Apr-24	NULL	0.028356978	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.006215397	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.546954909	KRAS G12C INHIBITOR GDC-6036	ncit:C173995	DIVARASIB	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.021036727	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
CRLF2	hgnc:14281	CRLF2	CIViC	10-Apr-24	NULL	1.029562181092049	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	CIViC	10-Apr-24	NULL	1.678633990910949	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	CIViC	10-Apr-24	NULL	0.026412309	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
H3-3A	hgnc:4764	H3-3A	CIViC	10-Apr-24	NULL	8.751278539282415	AKT/ERK INHIBITOR ONC201	ncit:C113792	DORDAVIPRONE	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	CIViC	10-Apr-24	NULL	0.4167275494896389	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.1440539677248134	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
KMT2C	hgnc:13726	KMT2C	CIViC	10-Apr-24	NULL	26.25383561784724	AROMATASE INHIBITOR	ncit:C1740	AROMATASE INHIBITOR	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	CIViC	10-Apr-24	NULL	1.944728564284981	ANTI-VEGF MONOCLONAL ANTIBODY	ncit:C2496	ANTI-VEGF MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
TSC2	hgnc:12363	TSC2	CIViC	10-Apr-24	NULL	4.375639269641208	MTOR INHIBITOR	ncit:C2201	MTOR INHIBITOR	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	CIViC	10-Apr-24	NULL	0.038104261	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.05913026	MTOR INHIBITOR	ncit:C2201	MTOR INHIBITOR	FALSE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	CIViC	10-Apr-24	NULL	0.033658764	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
RRM1	hgnc:10451	RRM1	CIViC	10-Apr-24	NULL	0.035098711	CARBOPLATIN	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
MMP9	hgnc:7176	MMP9	CIViC	10-Apr-24	NULL	0.052507671	BEVACIZUMAB	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.032616354	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	1.282909942931453	ENCORAFENIB	rxcui:2049106	ENCORAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	DoCM	10-Apr-24	NULL	2.341819737097098	DABRAFENIB	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	DoCM	10-Apr-24	NULL	1.678633990910949	RUXOLITINIB	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	DoCM	10-Apr-24	NULL	0.9845188356692719	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
ABL1	hgnc:76	ABL1	JAX-CKB	10-Apr-24	NULL	0.6241137025199848	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.043484614	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.031488858	Pazopanib	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.3043922970185188	THZ1	iuphar.ligand:8052	THZ1	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.3409589041278863	Vantictumab	ncit:C96799	VANTICTUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.014995051	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	PAC-1	drugbank:DB13048	PAC-1	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.02036365	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.06109095	Idelalisib	rxcui:1544460	IDELALISIB	TRUE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.7955707762984014	Mps1-IN-1	iuphar.ligand:9271	MPS1-IN-1	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.5527123287967842	Ulixertinib	ncit:C104744	ULIXERTINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	RLY-4008	ncit:C174208	LIRAFUGRATINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.029783137	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.8290684931951763	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.2075402025126264	Baricitinib	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.050609804	Nintedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.8204323630577265	SGC0946	iuphar.ligand:7020	SGC0946	FALSE	FALSE	FALSE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	0.2778183663264258	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.8204323630577265	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	3.000438356	Dostarlimab-gxly	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
MSH2	hgnc:7325	MSH2	JAX-CKB	10-Apr-24	NULL	2.500365296937833	Dostarlimab-gxly	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.2401265452851883	Oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.064824285	Capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.064824285	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4022765134992723	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.051850893	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1411496538593938	Sintilimab	ncit:C132992	SINTILIMAB	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	DEL-22379	wikidata:Q21044462	DEL-22379	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.097236428	TAS-117	drugbank:DB15054	TAS-117	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	WX390	ncit:C159499	PI3K/MTOR KINASE INHIBITOR WXFL10030390	FALSE	FALSE	FALSE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	1.009762908	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.022099188	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
POLD1	hgnc:9175	POLD1	JAX-CKB	10-Apr-24	NULL	0.6250913242344582	Dostarlimab-gxly	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
POLE	hgnc:9177	POLE	JAX-CKB	10-Apr-24	NULL	0.7501095890813498	Dostarlimab-gxly	rxcui:2539967	DOSTARLIMAB	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.022995101	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.3547815624033412	AT13148	ncit:C101786	MULTI-AGC KINASE INHIBITOR AT13148	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.026280116	Apitolisib	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1182605208011137	AZD8835	iuphar.ligand:8915	AZD8835	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.01835077	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	TGX-221	iuphar.ligand:8244	TGX-221	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.070956312	TAS-117	drugbank:DB15054	TAS-117	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.035478156	Ipilimumab	rxcui:1094833	IPILIMUMAB	TRUE	TRUE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.5173169579871378	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.5173169579871378	R547	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.09876051	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.2991890098899972	Saracatinib	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1178623372293928	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	CancerCommons	25-Jul-13	inhibitor	0.3906820776465364	MSC1936369B	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CancerCommons	25-Jul-13	inhibitor	1.657092009619794	ZELBORAF	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CancerCommons	25-Jul-13	inhibitor	0.1350505947420126	XL765	drugbank:DB05241	XL765	FALSE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.052455216	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.055504938	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.079758488	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.065125794	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.076840494	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.07160137	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.083522277	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.07963752	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.086694009	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.01924768	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.033658764	METHARBITAL	rxcui:6825	METHARBITAL	TRUE	FALSE	FALSE
ACE1	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.1483267549030917	MALATHION	rxcui:6606	MALATHION	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.016449772	PHENYTOIN SODIUM	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.053145416	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.096167896	ERLOSAMIDE	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.2500365296937833	TACEDINALINE	ncit:C2202	TACEDINALINE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.042689164	VINFLUNINE	ncit:C61564	VINFLUNINE	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.038894571	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.042689164	PLINABULIN	ncit:C62444	PLINABULIN	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	3.281729452230906	TOFOGLIFLOZIN	ncit:C152675	TOFOGLIFLOZIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	1.944728564284981	ARBACLOFEN PLACARBIL	ncit:C76088	ARBACLOFEN PLACARBIL	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	negative modulator	0.071439008	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	negative modulator	0.2885036881082115	ESKETAMINE HYDROCHLORIDE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	negative modulator	0.042689164	VERUBULIN	ncit:C96747	VERUBULIN	FALSE	FALSE	FALSE
APH1B	hgnc:24080	APH1B	ChEMBL	33	inhibitor	0.5048814541893701	BEGACESTAT	ncit:C76054	BEGACESTAT	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	negative modulator	0.1209854175937661	ESKETAMINE HYDROCHLORIDE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	negative modulator	0.108711535	ESKETAMINE HYDROCHLORIDE	rxcui:2119365	ESKETAMINE	TRUE	FALSE	FALSE
ELN	hgnc:3327	ELN	ChEMBL	33	cleavage	13.12691780892362	VONAPANITASE	ncit:C152909	VONAPANITASE	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	2.187819634820604	TALAZOPARIB TOSYLATE	rxcui:2099703	TALAZOPARIB TOSYLATE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	0.100976291	MUPARFOSTAT	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	ChEMBL	33	inhibitor	0.1419126249613365	MUPARFOSTAT	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
FGF1	hgnc:3665	FGF1	ChEMBL	33	inhibitor	0.5834185692854945	MUPARFOSTAT	ncit:C38690	MUPARFOSTAT	FALSE	FALSE	FALSE
DDB1	hgnc:2717	DDB1	ChEMBL	33	inhibitor	3.281729452230906	POMALIDOMIDE	rxcui:1369713	POMALIDOMIDE	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.4773424657790409	PARECOXIB SODIUM	rxcui:279951	PARECOXIB SODIUM	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	DEXIBUPROFEN	ncit:C166907	DEXIBUPROFEN	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	2.128689374420047	XALIPRODEN	ncit:C152924	XALIPRODEN	FALSE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	binder	6.300920548	CITATUZUMAB BOGATOX	ncit:C71694	CITATUZUMAB BOGATOX	FALSE	FALSE	FALSE
PGF	hgnc:8893	PGF	ChEMBL	33	inhibitor	3.500511415712967	CONBERCEPT	ncit:C162879	CONBERCEPT	FALSE	FALSE	FALSE
CD2	hgnc:1639	CD2	ChEMBL	33	inhibitor	17.50255707856483	SIPLIZUMAB	ncit:C38685	SIPLIZUMAB	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	ChEMBL	33	inhibitor	0.4861821410712453	ROVELIZUMAB	ncit:C152264	ROVELIZUMAB	FALSE	FALSE	FALSE
CD5	hgnc:1685	CD5	ChEMBL	33	binder	5.250767123569449	ZOLIMOMAB ARITOX	ncit:C29549	ZOLIMOMAB ARITOX	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	ChEMBL	33	inhibitor	1.071585127259071	PF-04236921	chembl:CHEMBL2109613	PF-04236921	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	agonist	0.02271093	DEXFENFLURAMINE HYDROCHLORIDE	rxcui:155142	DEXFENFLURAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.3922986931402463	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	CHLORPHENOXAMINE	rxcui:20881	CHLORPHENOXAMINE	TRUE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	inhibitor	0.7721716358190367	ATOSIBAN	rxcui:59639	ATOSIBAN	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.089501712	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.100976291	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.040328473	TERODILINE HYDROCHLORIDE	rxcui:235839	TERODILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.1211249624814175	ACALABRUTINIB	rxcui:1986808	ACALABRUTINIB	TRUE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	binder	0.182318303	PINATUZUMAB VEDOTIN	ncit:C104167	PINATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	binder	2.282942227638891	LABETUZUMAB GOVITECAN	ncit:C95710	LABETUZUMAB GOVITECAN	FALSE	FALSE	FALSE
RPS15A	hgnc:10389	RPS15A	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL11	hgnc:10301	RPL11	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
FAU	hgnc:3597	FAU	ChEMBL	33	modulator	0.065634589	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL12	hgnc:10302	RPL12	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL18	hgnc:10310	RPL18	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPLP0	hgnc:10371	RPLP0	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPL35	hgnc:10344	RPL35	ChEMBL	33	modulator	0.1312691780892362	ELX-02	ncit:C174918	EXALUREN	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	CADAZOLID	ncit:C118642	CADAZOLID	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.040021091	BMS-275183	ncit:C62639	BMS-275183	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.042689164	LAROTAXEL	ncit:C48427	LAROTAXEL	FALSE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	ChEMBL	33	inhibitor	2.500365296937833	M-1095	chembl:CHEMBL4298023	M-1095	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.036463661	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
CEACAM5	hgnc:1817	CEACAM5	ChEMBL	33	binder	0.2853677784548614	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.7721716358190367	TRIAPINE	ncit:C2242	TRIAPINE	FALSE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	TUSAMITAMAB RAVTANSINE	ncit:C117229	TUSAMITAMAB RAVTANSINE	FALSE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	ChEMBL	33	inhibitor	1.658136986390352	VIDOFLUDIMUS	ncit:C152873	VIDOFLUDIMUS	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.1640864726115453	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
RPS6KA2	hgnc:10431	RPS6KA2	ChEMBL	33	inhibitor	2.625383561784725	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	ChEMBL	33	inhibitor	0.073954467	TAS0612	chembl:CHEMBL4650277	TAS0612	FALSE	FALSE	FALSE
DBH	hgnc:2689	DBH	ChEMBL	33	inhibitor	3.500511415712966	ZAMICASTAT	ncit:C152947	ZAMICASTAT	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.037213091	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.037666909	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	ChEMBL	33	inhibitor	0.4861821410712453	CONTELTINIB	ncit:C169863	CONTELTINIB	FALSE	FALSE	FALSE
LIPF	hgnc:6622	LIPF	ChEMBL	33	inhibitor	11.66837138570988	CETILISTAT	ncit:C77404	CETILISTAT	FALSE	FALSE	FALSE
TREM1	hgnc:17760	TREM1	ChEMBL	33	inhibitor	52.50767123569449	NANGIBOTIDE	ncit:C166834	NANGIBOTIDE	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	0.2573905452730122	KBP5209	chembl:CHEMBL4650289	KBP5209	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
NPM1	hgnc:7910	NPM1	ChEMBL	33	inhibitor	0.4167275494896389	CERITINIB	rxcui:1535457	CERITINIB	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	RG-7636	chembl:CHEMBL2109282	RG-7636	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	ChEMBL	33	inhibitor	0.1842374429322613	EDASALONEXENT	ncit:C171665	EDASALONEXENT	FALSE	FALSE	FALSE
PDE10A	hgnc:21160	LINC00473	ChEMBL	33	inhibitor	8.751278539282415	BALIPODECT	ncit:C166905	BALIPODECT	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.8334550989792777	SELETALISIB	ncit:C152320	SELETALISIB	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	binder	0.525076712	TECLISTAMAB	rxcui:2619425	TECLISTAMAB-CQYV	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	BELUMOSUDIL MESYLATE	rxcui:2565692	BELUMOSUDIL MESYLATE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.6105543166941221	FIPAMEZOLE	ncit:C65684	FIPAMEZOLE	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	DEXELVUCITABINE	ncit:C76928	DEXELVUCITABINE	FALSE	FALSE	FALSE
MLNR	hgnc:4495	MLNR	ChEMBL	33	agonist	21.00306849427779	MITEMCINAL FUMARATE	ncit:C170187	MITEMCINAL FUMARATE	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	ChEMBL	33	inhibitor	0.2117244807890907	IZENCITINIB	ncit:C175805	IZENCITINIB	FALSE	FALSE	FALSE
ADM	hgnc:259	ADM	ChEMBL	33	modulator	6.563458904461812	ENIBARCIMAB	ncit:C175779	ENIBARCIMAB	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2035181055647073	BUCINDOLOL HYDROCHLORIDE	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
OPRL1	hgnc:8155	OPRL1	ChEMBL	33	agonist	6.563458904461812	SCH-486757	drugbank:DB12782	SCH-486757	FALSE	FALSE	FALSE
TLR2	hgnc:11848	TLR2	ChEMBL	33	inhibitor	0.9376369863516875	VB-201	drugbank:DB15259	VB-201	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.079557078	TIRZEPATIDE	rxcui:2601723	TIRZEPATIDE	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.8968701608581359	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.258658479	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	SAPPANONE A TRIMETHYL ETHER	chembl:CHEMBL1606022	SAPPANONE A TRIMETHYL ETHER	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.068907705	SCOPOLETIN	chembl:CHEMBL71851	SCOPOLETIN	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	BENZIODARONE	ncit:C74127	BENZIODARONE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.010966514	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.01214331	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	AZETIDINE-2,4-DICARBOXYLIC ACID	chembl:CHEMBL41680	CHEMBL:CHEMBL41680	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.006373064	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.1250182648468916	6,7-ADTN HYDROBROMIDE	chembl:CHEMBL1255656	CHEMBL:CHEMBL1255656	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	AG-808	chembl:CHEMBL68534	CHEMBL:CHEMBL68534	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	AESCULIOSIDE IVC	chembl:CHEMBL1094679	AESCULIOSIDE IVC	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.1691068316769549	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	NS-1619	iuphar.ligand:4272	NS1619	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	SJ000032151	chembl:CHEMBL592600	CHEMBL:CHEMBL592600	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	1.111273465305703	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.375054795	GNF-PF-2094	chembl:CHEMBL578928	CHEMBL:CHEMBL578928	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.025390557	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	2,4,5,10-TETRAHYDROPYRAZOLO[3,4-A]CARBAZOLE	chembl:CHEMBL512649	CHEMBL:CHEMBL512649	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.015075415	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009158847	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.2778183663264259	DIMETHYLADENINE	chembl:CHEMBL407391	DIMETHYLADENINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	5-HYDROXYINDOLE	iuphar.ligand:2295	5-HYDROXYINDOLE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GAMMA-AMINOBUTYRIC ACID	rxcui:4617	GAMMA-AMINOBUTYRIC ACID	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.5556367326528519	3'-NORSPONGIOLACTONE	chembl:CHEMBL1078000	CHEMBL:CHEMBL1078000	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	SULBENTINE	ncit:C72964	SULBENTINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	SJ000032152	chembl:CHEMBL590665	CHEMBL:CHEMBL590665	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	HYDROXYZINE PAMOATE	rxcui:203182	HYDROXYZINE PAMOATE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.276356164	CHELIDAMIC ACID	chembl:CHEMBL252909	CHELIDAMIC ACID	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.00675253	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.019776901	3,4-METHYLENEDIOXYB-NITROSTYRENE	iuphar.ligand:6048	SYK INHIBITOR III	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	GBR-12935	iuphar.ligand:4638	[3H]GBR12935	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005618798	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.4102161815288632	NITROBLUE TETRAZOLIUM	chembl:CHEMBL1185260	NITROBLUE TETRAZOLIUM	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.026319635	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	NCI-10777	chembl:CHEMBL189724	CHEMBL:CHEMBL189724	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	CLOXYQUIN	ncit:C61689	CLOXYQUIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.1653584607713247	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011762471	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.011157601	EMODIN	ncit:C466	EMODIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	ALLITRIDIN	chembl:CHEMBL123040	ALLITRIDIN	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1944728564284981	SCOPOLETIN	chembl:CHEMBL71851	SCOPOLETIN	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.01858569	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-124681	chembl:CHEMBL536008	CHEMBL:CHEMBL536008	FALSE	FALSE	FALSE
CSK	hgnc:2444	CSK	DTC	9/2/20	inhibitor	0.4375639269641209	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	METHYLERGONOVINE	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	TCMDC-125140	chembl:CHEMBL525106	CHEMBL:CHEMBL525106	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.014537008	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.4167275494896388	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012112496	3-O-METHYLQUERCETIN	chembl:CHEMBL163316	3-O-METHYLQUERCETIN	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.006649908	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.026519026	CID 94381	chembl:CHEMBL374632	CHEMBL:CHEMBL374632	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	RS-17053	iuphar.ligand:495	RS-17053	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.3500511415712966	DNDI1417331	chembl:CHEMBL1092508	CHEMBL:CHEMBL1092508	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	OXYTETRACYCLINE HYDROCHLORIDE	rxcui:4780	OXYTETRACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.020351811	LOBARIC ACID	chembl:CHEMBL551842	LOBARIC ACID	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	SJ000299520	chembl:CHEMBL592305	CHEMBL:CHEMBL592305	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	GABAZINE	iuphar.ligand:4083	[3H]GABAZINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TCMDC-124857	chembl:CHEMBL546580	CHEMBL:CHEMBL546580	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	CEFSULODIN SODIUM	rxcui:267417	CEFSULODIN SODIUM	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.023524942	CHRYSENE-1,4-DIONE	chembl:CHEMBL421215	CHEMBL:CHEMBL421215	FALSE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	DTC	9/2/20	NULL	5.250767123569449	LACTACYSTIN	chembl:CHEMBL374308	LACTACYSTIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.013022736	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	MONTELUKAST	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	DTC	9/2/20	NULL	0.2660861718025059	UMECLIDINIUM BROMIDE	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.003531589	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005483257	ELLAGIC ACID	rxcui:1043181	ELLAGIC ACID	FALSE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	DTC	9/2/20	NULL	3.663325900164732	BENZOHYDROXAMATE	chembl:CHEMBL16300	BENZOHYDROXAMATE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	ZAPA	chembl:CHEMBL20562	ZAPA	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.011637338	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	TYRPHOSTIN AG-1478	iuphar.ligand:4862	AG1478	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.6482428547616604	XANTHOHUMOL	ncit:C121950	XANTHOHUMOL	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.1100789753368857	COMBRETASTATIN A4	drugbank:DB14680	COMBRETASTATIN A4	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	3-AMINOBENZAMIDE	chembl:CHEMBL81977	3-AMINOBENZAMIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	PHENELZINE SULFATE	rxcui:8124	PHENELZINE SULFATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	BENZO[B]FLUORANTHENE	chembl:CHEMBL1337502	BENZO[B]FLUORANTHENE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	DNDI1417234	chembl:CHEMBL2094549	CHEMBL:CHEMBL2094549	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.036847489	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.042481935	FUMARPROTOCETRARIC ACID	chembl:CHEMBL366861	FUMARPROTOCETRARIC ACID	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.007254445	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	DTC	9/2/20	NULL	0.2075402025126264	ESTAZOLAM	rxcui:4077	ESTAZOLAM	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	RO-318220	iuphar.ligand:5259	RO31-8220	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2430910705356226	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2365210416022274	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.054243462	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	DNDI1417025	chembl:CHEMBL1320453	CHEMBL:CHEMBL1320453	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	CID 887167	chembl:CHEMBL260342	CHEMBL:CHEMBL260342	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.1112450661773188	6,7-ADTN HYDROBROMIDE	chembl:CHEMBL1255656	CHEMBL:CHEMBL1255656	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002170994	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2243917574174978	7-ETHYL-10-HYDROXY-CAMPTOTHECIN	iuphar.ligand:6925	SN-38	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	GANODERMANONTRIOL	chembl:CHEMBL1915763	GANODERMANONTRIOL	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.1232574442152452	EUPATORIN	chembl:CHEMBL487402	EUPATORIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003616231	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.032412143	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	DIHYDROGAMBOGIC ACID	chembl:CHEMBL1526240	DIHYDROGAMBOGIC ACID	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.011077568	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	2-METHYLAMINOBENZOIC ACID METHYL ESTER	chembl:CHEMBL1409791	2-METHYLAMINOBENZOIC ACID METHYL ESTER	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-5102	chembl:CHEMBL603031	CHEMBL:CHEMBL603031	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	(R)-BICALUTAMIDE	drugbank:DB02932	(R)-BICALUTAMIDE	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.7095631248066824	TG100-115	drugbank:DB05552	TG100-115	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	BENZOTHIAZYL DISULFIDE	chembl:CHEMBL508112	BENZOTHIAZYL DISULFIDE	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	4.200613699	GSK812397	chembl:CHEMBL1242210	CHEMBL:CHEMBL1242210	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	ICI-199,441	iuphar.ligand:11691	ICI-199441	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.046303061	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.091159151	SJ000293754	chembl:CHEMBL486706	CHEMBL:CHEMBL486706	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	1,2-DIMETHOXY-ANTHRAQUINONE	chembl:CHEMBL52884	CHEMBL:CHEMBL52884	FALSE	FALSE	FALSE
ME3	hgnc:6985	ME3	DTC	9/2/20	NULL	8.751278539282415	MALONIC ACID	drugbank:DB02175	MALONIC ACID	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	10,11-DIHYDROEPOTHILONE D	chembl:CHEMBL453818	CHEMBL:CHEMBL453818	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.079557078	NSC-105827	chembl:CHEMBL171699	CHEMBL:CHEMBL171699	FALSE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	0.1842374429322614	ETHOXZOLAMIDE	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	TRIPARANOL	ncit:C152752	TRIPARANOL	TRUE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1136529680426287	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	S(+)-ISOPROTERENOL-BITARTRATE	chembl:CHEMBL1257092	CHEMBL:CHEMBL1257092	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.007693432	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	HOMIDIUM	ncit:C83806	HOMIDIUM	FALSE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	DTC	9/2/20	NULL	0.2885036881082116	(-)-EPICATECHIN	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.018006746	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.019534104	PICEATANNOL	ncit:C1195	PICEATANNOL	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.014172111	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.2734774543525755	ZIMELDINE	ncit:C152954	ZIMELDINE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.015434354	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	0.076934317	TAMOXIFEN	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	DYCLONINE HYDROCHLORIDE	rxcui:91188	DYCLONINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.058931169	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.00211273	DOPAMINE HYDROCHLORIDE	rxcui:3628	DOPAMINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007831122	AMSACRINE	rxcui:739	AMSACRINE	TRUE	FALSE	TRUE
ADRA2A	hgnc:281	ADRA2A	DTC	9/2/20	NULL	0.2616661357260523	MOXONIDINE	rxcui:30257	MOXONIDINE	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.015959778	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	SJ000001592	chembl:CHEMBL591834	CHEMBL:CHEMBL591834	FALSE	FALSE	FALSE
POLG	hgnc:9179	POLG	DTC	9/2/20	NULL	35.00511415712966	KASANOSIN A	chembl:CHEMBL458178	KASANOSIN A	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	PHYSODIC ACID	chembl:CHEMBL171637	PHYSODIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	SJ000018298	chembl:CHEMBL591412	CHEMBL:CHEMBL591412	FALSE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	inhibitor	0.1193356164447602	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	DNDI1417078	chembl:CHEMBL1320798	CHEMBL:CHEMBL1320798	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	DNDI1417601	chembl:CHEMBL1503729	CHEMBL:CHEMBL1503729	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.000679905	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	HALOPROGIN	rxcui:26422	HALOPROGIN	TRUE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.078136416	AZD-1775	ncit:C91725	ADAVOSERTIB	FALSE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.034118045	GNF-PF-5114	chembl:CHEMBL601952	CHEMBL:CHEMBL601952	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.1591141552596803	PYROGALLOL	rxcui:9022	PYROGALLOL	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.030386384	SB-204741	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	SIB-1757	iuphar.ligand:1431	SIB-1757	FALSE	FALSE	FALSE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.012448476	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CYSTAMINE	rxcui:1426401	CYSTAMINE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.003313623	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	DIPHENYLENEIODONIUM	drugbank:DB17025	DIPHENYLENEIODONIUM	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1544343271638073	BI-87E7	chembl:CHEMBL523200	CHEMBL:CHEMBL523200	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.002201026	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.090530468	GNF-PF-4967	chembl:CHEMBL585827	CHEMBL:CHEMBL585827	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.048618214	2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE	chembl:CHEMBL502774	CHEMBL:CHEMBL502774	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002075566	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	1,2-DIPHENYLDISULFANE	chembl:CHEMBL462861	CHEMBL:CHEMBL462861	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.009855043	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.2067231151011594	IOPHENOXIC ACID	chembl:CHEMBL1551165	IOPHENOXIC ACID	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	SJ000089001	chembl:CHEMBL591618	CHEMBL:CHEMBL591618	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	GNF-PF-4967	chembl:CHEMBL585827	CHEMBL:CHEMBL585827	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.002725689	METHOTREXATE	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.1143957978991165	JNK INHIBITOR VIII	iuphar.ligand:5998	JNK INHIBITOR VIII	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.003195452	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	CHLORPYRIFOS	ncit:C163641	CHLORPYRIFOS	FALSE	FALSE	FALSE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.4565884455277783	CCT018159	chembl:CHEMBL399530	CHEMBL:CHEMBL399530	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	DTC	9/2/20	NULL	0.3571950424196904	DIZOCILPINE	ncit:C65450	DIZOCILPINE	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	CIMIRACEMATE A	chembl:CHEMBL1076184	CIMIRACEMATE A	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.052771529	CHRYSOPHANOL	chembl:CHEMBL41092	CHRYSOPHANOL	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.025147352	ILORASERTIB	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	7-BENZYLOXYCOUMARIN	chembl:CHEMBL145781	7-BENZYLOXYCOUMARIN	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	0.8401227397711121	OLEANOLIC_ACID	iuphar.ligand:3306	OLEANOLIC ACID	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.100589408	GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE	chembl:CHEMBL1255944	CHEMBL:CHEMBL1255944	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00195778	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1620607136904151	DINITRO CRESOL	chembl:CHEMBL419564	DINITRO CRESOL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	OXOGLAUCINE	iuphar.ligand:12559	OXOGLAUCINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.013631275	PYRITHIONE ZINC	ncit:C47698	PYRITHIONE ZINC	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	HISTAMINE	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.006823609	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	CEFOPERAZONE	rxcui:2184	CEFOPERAZONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	LINOPIRDINE	ncit:C82306	LINOPIRDINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.009579944	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.00310329	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	(S)-FLUOXETINE	drugbank:DB08544	(S)-FLUOXETINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	(S)-PROMETHAZINE	chembl:CHEMBL251904	(S)-PROMETHAZINE	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.021608095	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	FERROUS SULFATE	rxcui:24947	FERROUS SULFATE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	TCMDC-125567	chembl:CHEMBL530049	CHEMBL:CHEMBL530049	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	E319	chembl:CHEMBL242080	E319	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.018874073	PENTABROMOPHENOL	drugbank:DB03167	PENTABROMOPHENOL	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.052824619	ROTENONE	rxcui:1366666	ROTENONE	FALSE	FALSE	FALSE
NOD1	hgnc:16390	NOD1	DTC	9/2/20	NULL	13.12691780892362	GNF-PF-3971	chembl:CHEMBL599890	CHEMBL:CHEMBL599890	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	AFIMOXIFENE	ncit:C975	AFIMOXIFENE	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	THIOPERAMIDE	iuphar.ligand:1267	THIOPERAMIDE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.092443083	PHENETHYLISOTHIOCYANATE	chembl:CHEMBL151649	PHENETHYLISOTHIOCYANATE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.003285014	PD-98059	drugbank:DB17042	PD-98059	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001844705	DALFAMPRIDINE	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	SJ000059275	chembl:CHEMBL603952	CHEMBL:CHEMBL603952	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	MORUSINOL	chembl:CHEMBL1719948	MORUSINOL	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	1.000146118775133	TYROSOL SINAPATE	chembl:CHEMBL2348314	TYROSOL SINAPATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	GESTRINONE	rxcui:4792	GESTRINONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	TCMDC-124321	chembl:CHEMBL526952	CHEMBL:CHEMBL526952	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	TELENZEPINE	ncit:C75285	TELENZEPINE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.025513932	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	3-ACETYLCOUMARIN	chembl:CHEMBL149463	3-ACETYLCOUMARIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	CARBOXYMETHOXYLAMINE	iuphar.ligand:5136	AMINOOXYACETIC ACID	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	SKF-89976A	iuphar.ligand:4705	SKF89976A	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.019949723	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.015627283	SNS-314	drugbank:DB06134	SNS-314	FALSE	FALSE	TRUE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.7955707762984014	GARDENIN	chembl:CHEMBL77705	GARDENIN	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.3281729452230906	2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE	chembl:CHEMBL412603	CHEMBL:CHEMBL412603	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.015019357	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.007699637	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.038382801	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.021773863	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.029074015	4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL	chembl:CHEMBL1465049	CHEMBL:CHEMBL1465049	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.012079059	DORAMAPIMOD	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	chembl:CHEMBL1333512	N,N'-DIPHENYL-P-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.024286619	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.033615667	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	BIFONAZOLE	rxcui:19295	BIFONAZOLE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	O-METHYLCALOTHRIXIN A	chembl:CHEMBL549880	O-METHYLCALOTHRIXIN A	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	inhibitor	0.054695491	HESPERADIN	rxcui:1552358	HESPERADIN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.006896201	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.072424374	FLUNARIZINE DIHYDROCHLORIDE	chembl:CHEMBL539027	FLUNARIZINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	DTC	9/2/20	NULL	0.1491695205559502	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.2841324201065719	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	P-1075	chembl:CHEMBL11458	CHEMBL:CHEMBL11458	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005669763	5,6,7,8,4'-PENTAHYDROXYFLAVONE	chembl:CHEMBL234338	CHEMBL:CHEMBL234338	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	SJ000024939	chembl:CHEMBL590691	CHEMBL:CHEMBL590691	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	ZAPA	chembl:CHEMBL20562	ZAPA	FALSE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	DTC	9/2/20	NULL	4.375639269641208	AZD-8055	drugbank:DB12774	AZD-8055	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.003708169	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	4-AMINOPHENOL	rxcui:1435279	4-AMINOPHENOL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.021554873	3,8'-BIAPIGENIN	chembl:CHEMBL515252	CHEMBL:CHEMBL515252	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.071439008	PHENANTHROLINE	drugbank:DB02365	1,10-PHENANTHROLINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	2-PICOLINIC ACID	chembl:CHEMBL72628	2-PICOLINIC ACID	FALSE	FALSE	FALSE
TRPA1	hgnc:497	TRPA1	DTC	9/2/20	NULL	8.751278539282415	4-HYDROXYNON-2-ENAL	iuphar.ligand:6274	4-HYDROXYNONENAL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002861765	KETOCONAZOLE	rxcui:6135	KETOCONAZOLE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.040112812	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	NSC-45382	chembl:CHEMBL1214274	CHEMBL:CHEMBL1214274	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.061992528	(R,S)-INDATRALINE	chembl:CHEMBL341898	(R,S)-INDATRALINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	GNF-PF-1000	chembl:CHEMBL600554	CHEMBL:CHEMBL600554	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	5-METHOXYFLAVANONE	chembl:CHEMBL317869	CHEMBL:CHEMBL317869	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.035216413	LINOLENIC ACID	rxcui:52071	LINOLENIC ACID	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	ALRESTATIN	ncit:C72917	ALRESTATIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	3-METHOXYCATECHOL	chembl:CHEMBL1518159	3-METHOXYCATECHOL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	EPOXYCYTOCHALASIN H	chembl:CHEMBL517645	EPOXYCYTOCHALASIN H	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	CITROPTEN	chembl:CHEMBL481049	CITROPTEN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	(+)-CIS-DIOXOLANE IODIDE	chembl:CHEMBL387632	CHEMBL:CHEMBL387632	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	ARACHIDONIC ACID	rxcui:1368624	ARACHIDONIC ACID	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	DTC	9/2/20	NULL	0.030868707	TAMATINIB	drugbank:DB07159	TAMATINIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	DNDI1417072	chembl:CHEMBL1310701	CHEMBL:CHEMBL1310701	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.006896201	RG-1530	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	PYRAFLUFEN-ETHYL	chembl:CHEMBL1905010	PYRAFLUFEN-ETHYL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001223613	KENPAULLONE	iuphar.ligand:6000	KENPAULLONE	FALSE	FALSE	FALSE
RAC1	hgnc:9801	RAC1	DTC	9/2/20	NULL	5.834185692854944	ZU-4194738	chembl:CHEMBL554475	CHEMBL:CHEMBL554475	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	LAPACHOL	chembl:CHEMBL15193	LAPACHOL	FALSE	FALSE	FALSE
ESR	hgnc:3467	ESR1	FDA	10-Apr-24	NULL	0.019629036	Eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
MS4A1	hgnc:7315	MS4A1	FDA	10-Apr-24	NULL	3.889457128569962	Obinutuzumab	rxcui:974779	OBINUTUZUMAB	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.004172574	Rabeprazole	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	FDA	10-Apr-24	NULL	0.02804897	Piroxicam	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
CASR	hgnc:1514	CASR	FDA	10-Apr-24	NULL	1.093909817410302	Parathyroid Hormone	rxcui:1427222	PARATHYROID HORMONE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.047734247	Probenecid	rxcui:8698	PROBENECID	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	FDA	10-Apr-24	NULL	0.2273059360852576	Thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	MyCancerGenome	20-Jun-17	inhibitor	0.8008364246019593	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
HBB	hgnc:4827	HBB	FDA	10-Apr-24	NULL	0.9053046764774912	Voxelotor	rxcui:2265678	VOXELOTOR	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.009040577	Voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	MyCancerGenome	20-Jun-17	inhibitor	0.1193356164447602	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenome	20-Jun-17	inhibitor	0.2778183663264259	AMUVATINIB	ncit:C71750	AMUVATINIB	FALSE	FALSE	TRUE
ARAF	hgnc:646	ARAF	MyCancerGenome	20-Jun-17	inhibitor	0.075369863	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
DEPTOR	hgnc:22953	DEPTOR	MyCancerGenome	20-Jun-17	inhibitor	0.7955707762984016	MLN0128	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.065799087	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.014790893	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.032899543	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.035719504	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4828291607879953	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.760980743	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2041114528112516	PD-0332991	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.023080295	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.08572681	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.042073455	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.011872848	CDDP	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.005540537	VCR	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.044347695	CHLORPROMAZINE	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.6455861217503421	PSC-833	ncit:C1405	VALSPODAR	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.1262203635473425	NITROFURANTOIN	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	0.1544343271638073	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.652269208	RECOMBINANT INTERLEUKIN	ncit:C593	RECOMBINANT INTERLEUKIN	FALSE	FALSE	FALSE
APC	hgnc:583	APC	NCI	14-Sep-17	NULL	0.2651902587661338	HISTONE DEACETYLASE INHIBITOR	ncit:C1946	HISTONE DEACETYLASE INHIBITOR	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1400204566285186	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.017075665	CYCLOPHOSPHAMIDE	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1200632726425941	13-CIS-RETINOIC ACID	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.050007306	PREDNISOLONE	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.053854022	OXYTOCIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1422972120208523	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.2500365296937833	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
CCL11	hgnc:10610	CCL11	NCI	14-Sep-17	NULL	1.944728564284981	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	NCI	14-Sep-17	NULL	0.099258358	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
CD40LG	hgnc:11935	CD40LG	NCI	14-Sep-17	NULL	0.1646008502686348	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
CD80	hgnc:1700	CD80	NCI	14-Sep-17	NULL	0.9723642821424908	ROXITHROMYCIN	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.4234489615781814	DEXTRAN SULFATE SODIUM	ncit:C1284	DEXTRAN SULFATE SODIUM	FALSE	FALSE	FALSE
CEACAM1	hgnc:1814	CEACAM1	NCI	14-Sep-17	NULL	0.2885036881082115	RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
CHST11	hgnc:17422	CHST11	NCI	14-Sep-17	NULL	11.66837138570989	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
CRH	hgnc:2355	CRH	NCI	14-Sep-17	NULL	0.5966780822238011	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.2059124362184098	ANTIBIOTIC	ncit:C258	ANTIBIOTIC	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	4.039051633514961	ACRIDINE	ncit:C203	ACRIDINE	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.252440727	SPIRONOLACTONE	rxcui:9997	SPIRONOLACTONE	TRUE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	0.729273212	BCG	ncit:C77178	BACILLUS CALMETTE-GUERIN ANTIGEN	FALSE	FALSE	FALSE
CTSB	hgnc:2527	CTSB	NCI	14-Sep-17	NULL	2.917092846427472	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
CTSK	hgnc:2536	CTSK	NCI	14-Sep-17	NULL	0.3535870116881784	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	4.375639269641208	BETA-GLUCAN	ncit:C2678	BETA-GLUCAN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.004698673	E7389	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.4861821410712453	PROTEIN SYNTHESIS INHIBITOR	ncit:C784	PROTEIN SYNTHESIS INHIBITOR	FALSE	FALSE	FALSE
EMR2	hgnc:3337	ADGRE2	NCI	14-Sep-17	NULL	11.66837138570989	CHONDROITIN SULFATE	rxcui:2473	CHONDROITIN SULFATES	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.3454452054979901	GREEN TEA POLYPHENOLS	ncit:C2694	GREEN TEA EXTRACT	FALSE	FALSE	FALSE
ERCC6	hgnc:3438	ERCC6	NCI	14-Sep-17	NULL	0.1207072901969988	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	0.1091635576625665	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	1.009762908	LEPIRUDIN	rxcui:114934	DESIRUDIN	TRUE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.1293292394967844	FUDR	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.2011788169949981	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.019896806	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	1.810609352954982	AD-CD154	ncit:C2493	ADENOVIRUS 5-CD40 LIGAND	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.4953553890159858	POLY I:C	ncit:C758	POLY IC	FALSE	FALSE	FALSE
PZP	hgnc:9750	PZP	NCI	14-Sep-17	NULL	0.2966535098061836	PROGESTERONE	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.072125922	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
SAG	hgnc:10521	SAG	NCI	14-Sep-17	NULL	0.201178817	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.4412409347537352	DALTEPARIN	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
SCD	hgnc:10571	SCD	NCI	14-Sep-17	NULL	0.2885036881082116	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
SLC28A1	hgnc:11001	SLC28A1	NCI	14-Sep-17	NULL	5.250767123569449	URIDINE	rxcui:11017	URIDINE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.2386712328895204	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.2282942227638891	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	1.400204566285186	INCOMPLETE FREUND&APOS;S ADJUVANT	ncit:C1573	INCOMPLETE FREUND'S ADJUVANT	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.1448487482363986	PROTOPORPHYRIN	drugbank:DB02285	PROTOPORPHYRIN	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.317586721	13-CIS-RETINOIC ACID	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
TGFBR3	hgnc:11774	TGFBR3	NCI	14-Sep-17	NULL	0.5048814541893702	CYTOKINES	ncit:C1283	RECOMBINANT CYTOKINE	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.192335792	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	1.000146118775133	SAPONIN	ncit:C823	SAPONIN	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.217423069	DOXYCYCLINE	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.09972967	VITAMIN A	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	NCI	14-Sep-17	NULL	0.151537291	UREA	rxcui:11002	UREA	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.1411496538593938	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.112919723	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.049095532	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	NCI	14-Sep-17	NULL	0.3017682254924971	TENIPOSIDE	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.4546118721705151	ANTIOXIDANT	ncit:C275	ANTIOXIDANT	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	NCI	14-Sep-17	NULL	0.077616661	ANTISENSE OLIGONUCLEOTIDES	ncit:C1291	ANTISENSE OLIGONUCLEOTIDES	FALSE	FALSE	FALSE
UMOD	hgnc:12559	UMOD	NCI	14-Sep-17	NULL	5.000730593875666	LYMPHOKINES	ncit:C621	RECOMBINANT LYMPHOKINE	FALSE	FALSE	FALSE
VCAN	hgnc:2464	VCAN	NCI	14-Sep-17	NULL	0.6035364509849942	CSA	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.08780547	GENTAMICIN	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	1.640864726115453	LISINOPRIL	rxcui:1546022	LISINOPRIL ANHYDROUS	TRUE	FALSE	FALSE
VIM	hgnc:12692	VIM	NCI	14-Sep-17	NULL	1.500219178162699	GELDANAMYCIN	ncit:C1112	GELDANAMYCIN	FALSE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	PharmGKB	4/5/24	NULL	0.094244538	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.027635616	eribulin	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.043180651	fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	PharmGKB	4/5/24	NULL	0.057073556	temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	2.187819634820604	calcein	chembl:CHEMBL1973733	OFTASCEINE	FALSE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	PharmGKB	4/5/24	NULL	0.2763561643983921	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	PharmGKB	4/5/24	NULL	0.1141471113819445	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
POR	hgnc:9208	POR	PharmGKB	4/5/24	NULL	0.4773424657790409	clobazam	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
CHRNA5	hgnc:1959	CHRNA5	PharmGKB	4/5/24	NULL	0.8751278539282418	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
CHRNA6	hgnc:15963	CHRNA6	PharmGKB	4/5/24	NULL	0.8751278539282418	rozanolixizumab	rxcui:2642274	ROZANOLIXIZUMAB	TRUE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.1693795846312726	efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1548898856510162	dolutegravir	rxcui:1433867	DOLUTEGRAVIR SODIUM	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1032599237673441	isoniazid	rxcui:6038	ISONIAZID	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.012558639	chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.042242696	diethylstilbestrol	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
TREML4	hgnc:30807	TREML4	PharmGKB	4/5/24	NULL	4.039051633514962	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.008152099	sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.1495945049449985	ivermectin	rxcui:6069	IVERMECTIN	TRUE	FALSE	FALSE
SETD4	hgnc:1258	SETD4	PharmGKB	4/5/24	NULL	0.3500511415712966	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
MT1A	hgnc:7393	MT1A	PharmGKB	4/5/24	NULL	1.280674908	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
HMGCR	hgnc:5006	HMGCR	PharmGKB	4/5/24	NULL	1.750255707856483	cerivastatin	rxcui:596723	CERIVASTATIN	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	0.1346350544504987	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATP10A	hgnc:13542	ATP10A	PharmGKB	4/5/24	NULL	2.019525816757481	duloxetine	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.039598545	clarithromycin	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.017599354	clarithromycin	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	0.729273212	asparaginase	rxcui:1156	ASPARAGINASE	TRUE	FALSE	TRUE
KCNJ11	hgnc:6257	KCNJ11	PharmGKB	4/5/24	NULL	0.1293292394967844	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.1999620096341412	cetuximab	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
BRCA1	hgnc:1100	BRCA1	PharmGKB	4/5/24	NULL	0.1269527834518725	rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	0.1470803115845784	etidronic acid	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
DAOA	hgnc:21191	DAOA	PharmGKB	4/5/24	NULL	2.187819634820604	methamphetamine	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
AKR7A2	hgnc:389	AKR7A2	PharmGKB	4/5/24	NULL	0.3500511415712966	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.1121958787087489	hydroxocobalamin	rxcui:5514	HYDROXOCOBALAMIN	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.2917092846427472	maraviroc	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
IL18	hgnc:5986	IL18	PharmGKB	4/5/24	NULL	0.3947945205691315	interferon alfa-2b, recombinant	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
MMP9	hgnc:7176	MMP9	PharmGKB	4/5/24	NULL	0.525076712	Antihypertensives	ncit:C270	ANTIHYPERTENSIVE AGENT	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	PharmGKB	4/5/24	NULL	0.06375385	vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
CYSLTR1	hgnc:17451	CYSLTR1	PharmGKB	4/5/24	NULL	1.084869240406911	montelukast	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.729273212	torasemide	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.0076065	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	PharmGKB	4/5/24	NULL	0.017450206	erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.007179391	chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.056097939	voriconazole	rxcui:121243	VORICONAZOLE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.018193926	chlorpromazine	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
CYP11B2	hgnc:2592	CYP11B2	PharmGKB	4/5/24	NULL	1.166837138570988	candesartan	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
FCHSD1	hgnc:25463	FCHSD1	PharmGKB	4/5/24	NULL	0.258658479	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	PharmGKB	4/5/24	NULL	0.2983390411119005	nppb	iuphar.ligand:4270	NPPB	FALSE	FALSE	FALSE
VPS13D	hgnc:23595	VPS13D	PharmGKB	4/5/24	NULL	1.944728564284981	capecitabine	rxcui:194000	CAPECITABINE	TRUE	FALSE	TRUE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.03043923	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
BDKRB1	hgnc:1029	BDKRB1	PharmGKB	4/5/24	NULL	2.917092846427472	perindopril	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
TSPAN5	hgnc:17753	TSPAN5	PharmGKB	4/5/24	NULL	15.00219178162699	serotonin	rxcui:1311214	SEROTONIN	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.034318739	alprazolam	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
KLC3	hgnc:20717	KLC3	PharmGKB	4/5/24	NULL	2.012489141437768	oxaliplatin	rxcui:32592	OXALIPLATIN	TRUE	FALSE	TRUE
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	0.087512785	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.036977233	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.03219848	ciprofloxacin	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
BEST3	hgnc:17105	BEST3	PharmGKB	4/5/24	NULL	2.282942227638891	hydrochlorothiazide	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.012141906	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
MTHFD1	hgnc:7432	MTHFD1	PharmGKB	4/5/24	NULL	0.1411496538593938	gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.057073556	epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.078722146	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	0.4861821410712453	lusutrombopag	rxcui:2054984	LUSUTROMBOPAG	TRUE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.1704794520639431	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
CAPN10	hgnc:1477	CAPN10	PharmGKB	4/5/24	NULL	1.875273972703374	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
CYP3A7	hgnc:2640	CYP3A7	PharmGKB	4/5/24	NULL	0.6697407045369196	tacrolimus	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	2.100306849	deleobuvir	ncit:C166826	DELEOBUVIR	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	2.625383561784724	phenazopyridine	rxcui:8120	PHENAZOPYRIDINE	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	2.019525817	pegaptanib	rxcui:498509	PEGAPTANIB	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.3125456621172291	iguratimod	ncit:C65886	IGURATIMOD	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.087512785	perindopril	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.080781033	chloroprocaine	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	PharmGKB	4/5/24	NULL	0.046784382	sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.01123399	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.09869863	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.02302968	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
FMO1	hgnc:3769	FMO1	PharmGKB	4/5/24	NULL	0.4605936073306535	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
PLAGL1	hgnc:9046	PLAGL1	PharmGKB	4/5/24	NULL	1.381780822	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
PTPRN2	hgnc:9677	PTPRN2	PharmGKB	4/5/24	NULL	1.381780822	olanzapine	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UGT1A6	hgnc:12538	UGT1A6	PharmGKB	4/5/24	NULL	0.1973972602845657	phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	0.258658479	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.100589408	MAO inhibitors	ncit:C667	MONOAMINE OXIDASE INHIBITOR	FALSE	FALSE	FALSE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.2442217266776488	prednisone	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.01014641	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ABCC10	hgnc:52	ABCC10	PharmGKB	4/5/24	NULL	0.1166837138570988	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
ERCC2	hgnc:3434	ERCC2	PharmGKB	4/5/24	NULL	0.095468493	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SLC15A1	hgnc:10920	SLC15A1	PharmGKB	4/5/24	NULL	0.1400204566285186	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
SLC22A7	hgnc:10971	SLC22A7	PharmGKB	4/5/24	NULL	0.1166837138570988	doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1544343271638073	ketamine	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	PharmGKB	4/5/24	NULL	0.1151484018326633	entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.04464938	neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
UNIPROT:P12268	hgnc:6053	IMPDH2	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
UNIPROT:P16422	hgnc:11529	EPCAM	TdgClinicalTrial	Jan-14	NULL	1.260184109656668	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.3938075342677087	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	0.091796628	DULOXETINE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P20333	hgnc:11917	TNFRSF1B	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	CYT-6091	ncit:C62538	COLLOIDAL GOLD-BOUND TUMOR NECROSIS FACTOR	FALSE	FALSE	FALSE
UNIPROT:P48058	hgnc:4574	GRIA4	TdgClinicalTrial	Jan-14	NULL	0.596678082	CX717	chembl:CHEMBL4791762	CX-717	FALSE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.591141552596803	DEGARELIX	rxcui:475230	DEGARELIX	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.3006164383722967	DIFLUPREDNATE	rxcui:23043	DIFLUPREDNATE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	DERSALAZINE	ncit:C77949	DERSALAZINE	FALSE	FALSE	FALSE
UNIPROT:O15399	hgnc:4588	GRIN2D	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	DEXANABINOL	ncit:C99381	DEXANABINOL	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.036062961	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1041818873724097	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.047821194	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
UNIPROT:P42263	hgnc:4573	GRIA3	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
UNIPROT:Q08499	hgnc:8783	PDE4D	TdgClinicalTrial	Jan-14	NULL	0.078136416	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.222962511	ED-71	ncit:C87291	ELDECALCITOL	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.042073455	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.042073455	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.7026004179620139	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	0.018410824	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P06241	hgnc:4037	FYN	TdgClinicalTrial	Jan-14	NULL	0.047049885	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.060492709	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P04629	hgnc:8031	NTRK1	TdgClinicalTrial	Jan-14	NULL	0.023202683	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:Q05397	hgnc:9611	PTK2	TdgClinicalTrial	Jan-14	NULL	0.062733179	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.047712559	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
UNIPROT:Q02750	hgnc:6840	MAP2K1	TdgClinicalTrial	Jan-14	NULL	0.5903640284436551	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
UNIPROT:P13866	hgnc:11036	SLC5A1	TdgClinicalTrial	Jan-14	NULL	1.312691780892362	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:Q8IW41	hgnc:6889	MAPKAPK5	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	GLPG0259	chembl:CHEMBL5095028	GLPG-0259	FALSE	FALSE	FALSE
UNIPROT:P31639	hgnc:11037	SLC5A2	TdgClinicalTrial	Jan-14	NULL	0.4102161815288632	GLUFOSFAMIDE	ncit:C1612	GLUFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TdgClinicalTrial	Jan-14	NULL	0.1367387271762877	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
UNIPROT:P37088	hgnc:10599	SCNN1A	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	GS-9411	chembl:CHEMBL4297254	552-02	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.1665148136438514	GUANFACINE	rxcui:203142	GUANFACINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P51172	hgnc:10601	SCNN1D	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	GS-9411	chembl:CHEMBL4297254	552-02	FALSE	FALSE	FALSE
UNIPROT:Q8WW43	hgnc:24080	APH1B	TdgClinicalTrial	Jan-14	NULL	0.577007376	GSI-136	drugbank:DB12819	GSI-136	FALSE	FALSE	FALSE
UNIPROT:P51168	hgnc:10600	SCNN1B	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	GS-9411	chembl:CHEMBL4297254	552-02	FALSE	FALSE	FALSE
UNIPROT:O14746	hgnc:11730	TERT	TdgClinicalTrial	Jan-14	NULL	3.000438356	GV1001	ncit:C62756	TERTOMOTIDE	FALSE	FALSE	FALSE
UNIPROT:P08571	hgnc:1628	CD14	TdgClinicalTrial	Jan-14	NULL	14.32027397337122	IC14	chembl:CHEMBL2109330	IC14	FALSE	FALSE	FALSE
UNIPROT:O75330	hgnc:5012	HMMR	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	HYALURONAN	rxcui:5463	HYALURONIC ACID	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	0.1458546423213736	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
UNIPROT:P56696	hgnc:6298	KCNQ4	TdgClinicalTrial	Jan-14	NULL	1.050153425	ICA-105665	drugbank:DB06089	ICA-105665	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1383601350084176	ITOPRIDE	ncit:C65991	ITOPRIDE	FALSE	FALSE	FALSE
UNIPROT:Q14872	hgnc:7428	MTF1	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	LOR-253	chembl:CHEMBL4297261	APTO-253	FALSE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TdgClinicalTrial	Jan-14	NULL	1.084869240406911	MONTELUKAST	rxcui:115713	MONTELUKAST SODIUM	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.08914715	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	LIXIVAPTAN	ncit:C74429	LIXIVAPTAN	FALSE	FALSE	FALSE
UNIPROT:Q14832	hgnc:4595	GRM3	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	LY2140023	drugbank:DB05096	LY2140023	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.059297201	BUSPIRONE	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.087512785	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2004109589148645	CICLESONIDE	rxcui:274964	CICLESONIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	DOXYLAMINE	rxcui:3642	DOXYLAMINE	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.080550887	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.096167896	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	FLUDROCORTISONE	rxcui:4452	FLUDROCORTISONE	TRUE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.076690854	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.058799184	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.033701971	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.030368809	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1223955040459079	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.087318744	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.081365193	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q9Y271	hgnc:17451	CYSLTR1	TdgClinicalTrial	Jan-14	NULL	7.955707762984016	PRANLUKAST	ncit:C96712	PRANLUKAST	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.085239726	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.055155117	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P07202	hgnc:12015	TPO	TdgClinicalTrial	Jan-14	NULL	2.625383561784725	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.088248187	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.2778183663264258	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	PROPOXYPHENE	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.1154014752432845	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.1013661606866689	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.055504938	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	0.1884246575443582	TEMAZEPAM	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.068191781	SULINDAC	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	2.316514907	AMBENONIUM	rxcui:623	AMBENONIUM	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.064318974	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
UNIPROT:P15056	hgnc:1097	BRAF	TEND	1-Aug-11	NULL	0.091636424	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:Q08289	hgnc:1402	CACNB2	TEND	1-Aug-11	NULL	0.1458546423213736	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P19793	hgnc:10477	RXRA	TEND	1-Aug-11	NULL	0.2333674277141977	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
UNIPROT:Q01668	hgnc:1391	CACNA1D	TEND	1-Aug-11	NULL	0.081407242	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P10826	hgnc:9865	RARB	TEND	1-Aug-11	NULL	0.4412409347537352	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
UNIPROT:P28702	hgnc:10478	RXRB	TEND	1-Aug-11	NULL	0.8334550989792776	ALITRETINOIN	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
UNIPROT:P06729	hgnc:1639	CD2	TEND	1-Aug-11	NULL	11.66837138570988	ALEFACEPT	rxcui:299635	ALEFACEPT	TRUE	TRUE	FALSE
UNIPROT:P51800	hgnc:2026	CLCNKA	TEND	1-Aug-11	NULL	4.039051633514962	NIFLUMIC ACID	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.2282942227638891	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P01589	hgnc:6008	IL2RA	TEND	1-Aug-11	NULL	1.715936968486748	BASILIXIMAB	rxcui:196102	BASILIXIMAB	TRUE	TRUE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.4189441853911795	BENZTROPINE	rxcui:1424	BENZTROPINE	TRUE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TEND	1-Aug-11	NULL	0.093098708	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1595977849109255	BETHANECHOL	rxcui:19257	BETHANECHOL	TRUE	FALSE	FALSE
UNIPROT:P29317	hgnc:3386	EPHA2	TEND	1-Aug-11	NULL	0.4167275494896388	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.2004109589148645	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.7458476027797514	BISOPROLOL	rxcui:19484	BISOPROLOL	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.99446347	BETAXOLOL	rxcui:1520	BETAXOLOL	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.1193356164447602	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.038765353	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P22607	hgnc:3690	FGFR3	TEND	1-Aug-11	NULL	0.138178082	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.06757744	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1785975212098452	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.055563673	BROMAZEPAM	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1221108633388244	BUTABARBITAL	rxcui:477631	BUTABARBITAL	TRUE	FALSE	FALSE
UNIPROT:P07202	hgnc:12015	TPO	TEND	1-Aug-11	NULL	2.625383561784725	PROPYLTHIOURACIL	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
UNIPROT:P20648	hgnc:819	ATP4A	TEND	1-Aug-11	NULL	0.2243917574174979	RABEPRAZOLE	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TEND	1-Aug-11	NULL	0.9845188356692718	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TEND	1-Aug-11	NULL	0.661861402	RIZATRIPTAN	rxcui:237082	RIZATRIPTAN BENZOATE	TRUE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TEND	1-Aug-11	NULL	0.5676504998453459	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P07949	hgnc:9967	RET	TEND	1-Aug-11	NULL	0.3968833804663227	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
UNIPROT:P10721	hgnc:6342	KIT	TEND	1-Aug-11	NULL	0.1331836936859721	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P51692	hgnc:11367	STAT5B	TEND	1-Aug-11	NULL	0.2727671233023091	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:Q02643	hgnc:4266	GHRHR	TEND	1-Aug-11	NULL	19.69037671338543	TESAMORELIN	rxcui:1044584	TESAMORELIN	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.2031244535229961	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.2187819634820604	TOLAZOLINE	rxcui:10634	TOLAZOLINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.2075402025126264	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.051885051	TRIAMCINOLONE	rxcui:10759	TRIAMCINOLONE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	1.721562991334245	ULIPRISTAL	rxcui:1005920	ULIPRISTAL ACETATE	TRUE	FALSE	FALSE
UNIPROT:Q02641	hgnc:1401	CACNB1	TEND	1-Aug-11	NULL	0.1666910197958555	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.01924768	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
PROTEIN TYROSINE PHOSPHATASE	hgnc:10989	SLC25A3	TTD	2020.06.01	NULL	26.25383561784724	KP-100	chembl:CHEMBL5095468	OREMEPERMIN ALFA	FALSE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	0.065145994	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.016131389	ZIPRASIDONE	rxcui:115698	ZIPRASIDONE	TRUE	FALSE	FALSE
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	52.50767123569449	TAK-935	ncit:C166470	SOTICLESTAT	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.1232574442152452	MM-141	ncit:C103863	ISTIRATUMAB	FALSE	FALSE	FALSE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	4.109296009750004	Ensartinib	ncit:C102754	ENSARTINIB	FALSE	FALSE	FALSE
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	0.5469549087051511	Mirvetuximab soravtansine	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.033658764	Enzastaurin	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
INTERCELLULAR ADHESION MOLECULE ICAM-1	hgnc:5344	ICAM1	TTD	2020.06.01	NULL	17.50255707856483	Alicaforsen	ncit:C169771	ALICAFORSEN	FALSE	FALSE	FALSE
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	0.2853677784548614	TAK-828	iuphar.ligand:9867	TAK-828F	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.9546849315580818	Cabiralizumab	ncit:C123831	CABIRALIZUMAB	FALSE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	0.3500511415712966	Cabiralizumab	ncit:C123831	CABIRALIZUMAB	FALSE	FALSE	FALSE
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	5.250767123569449	ERY974	ncit:C129936	ANTI-GLYPICAN 3/CD3 BISPECIFIC ANTIBODY ERY974	FALSE	FALSE	FALSE
OX40L RECEPTOR	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	3.500511415712966	INCAGN1949	ncit:C129967	AGONISTIC ANTI-OX40 MONOCLONAL ANTIBODY INCAGN01949	FALSE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	10.50153424713889	Talacotuzumab	ncit:C102784	TALACOTUZUMAB	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.2453629496995069	BL-1021	chembl:CHEMBL1187120	BL-1021	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	0.2869271652223742	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.2108741816694558	XL-820	chembl:CHEMBL3545402	XL-820	FALSE	FALSE	FALSE
MELANOCYTES LINEAGE-SPECIFIC ANTIGEN GP100	hgnc:10880	PMEL	TTD	2020.06.01	NULL	8.751278539282415	Gp100:209-217(210M) peptide vaccine	ncit:C49022	GP100:209-217(210M) PEPTIDE VACCINE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.097236428	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
FYN TYROSINE PROTEIN KINASE	hgnc:4037	FYN	TTD	2020.06.01	NULL	0.3241214273808303	JNJ-26483327	chembl:CHEMBL3545133	JNJ-26483327	FALSE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.2025758921130189	MLN1117	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	0.1790034246671403	Azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
ANGIOTENSIN-CONVERTING ENZYME 2	hgnc:13557	ACE2	TTD	2020.06.01	NULL	5.250767123569449	ORE-1001	drugbank:DB12271	ORE-1001	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.8899605294185507	Olmesartan medoxomil	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.009437037	Acetaminophen	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.1805819381121768	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
CYSTEINE PROTEASE	hgnc:14650	PPIG	TTD	2020.06.01	NULL	52.50767123569449	MELARSOPROL	ncit:C170159	MELARSOPROL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	PERUVOSIDE	drugbank:DB13756	PERUVOSIDE	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	7.955707762984016	Pranlukast	ncit:C96712	PRANLUKAST	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.2035181055647073	L-796568	chembl:CHEMBL111201	CHEMBL:CHEMBL111201	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.2983390411119005	L-796568	chembl:CHEMBL111201	CHEMBL:CHEMBL111201	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.1190650141398968	BAY 10-00394	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.1491695205559502	Cabazitaxel	rxcui:996051	CABAZITAXEL	TRUE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.693795846312725	Alcaftadine	rxcui:1000082	ALCAFTADINE	TRUE	FALSE	FALSE
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	2.282942227638891	AVX701	ncit:C70644	CARCINOEMBRYONIC ANTIGEN PEPTIDE 1-6D VIRUS-LIKE REPLICON PARTICLES VACCINE	FALSE	FALSE	FALSE
STEROID 17-ALPHA-MONOOXYGENASE	hgnc:2593	CYP17A1	TTD	2020.06.01	NULL	30.00438356	TAK-700	ncit:C90582	ORTERONEL	FALSE	FALSE	TRUE
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	0.4167275494896388	GDC-0152	drugbank:DB12380	GDC-0152	FALSE	FALSE	FALSE
APOPTOSIS MEDIATING SURFACE ANTIGEN FAS	hgnc:11920	FAS	TTD	2020.06.01	NULL	0.4526523382387456	APG-101	ncit:C90562	ASUNERCEPT	FALSE	FALSE	FALSE
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	5.834185692854944	CVT-6883	drugbank:DB05936	CVT-6883	FALSE	FALSE	FALSE
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	3.281729452230906	ARQ 621	ncit:C82694	EG5 KINESIN-RELATED MOTOR PROTEIN INHIBITOR ARQ 621	FALSE	FALSE	FALSE
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.5048814541893701	BMS-708163	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
SH2 DOMAIN INOSITOL 5'-PHOSPHATASE 1	hgnc:6079	INPP5D	TTD	2020.06.01	NULL	26.25383561784724	AQX-1125	ncit:C152258	ROSIPTOR	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.2386712328895204	Darbufelone	ncit:C81061	DARBUFELONE	FALSE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.1159109740302306	SGT-53	ncit:C29474	TRANSFERRIN RECEPTOR-TARGETED LIPOSOMAL P53 CDNA	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	2.625383561784724	MK-1029	chembl:CHEMBL3545031	MK-1029	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.400821918	Dexamethasone sodium phosphate	rxcui:48933	DEXAMETHASONE SODIUM PHOSPHATE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.5556367326528519	EGF816	ncit:C115109	NAZARTINIB	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.2453629496995069	Metaiodobenzylguanidine I-131	rxcui:14448	3-IODOBENZYLGUANIDINE	TRUE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	0.7095631248066824	Netupitant	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
INTEGRIN ALPHA-V	hgnc:6150	ITGAV	TTD	2020.06.01	NULL	1.346350544504987	Abituzumab	ncit:C82422	ABITUZUMAB	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1226814748497534	Rhopressa	rxcui:1992864	NETARSUDIL	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.4234489615781814	LY-2624803	drugbank:DB15092	LY-2624803	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1183271464466354	Intedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
LEPTIN RECEPTOR	hgnc:6554	LEPR	TTD	2020.06.01	NULL	3.500511415712967	Metreleptin	rxcui:1491625	METRELEPTIN	TRUE	FALSE	FALSE
5-HT 7 RECEPTOR	hgnc:5302	HTR7	TTD	2020.06.01	NULL	1.750255707856483	JNJ-18038683	iuphar.ligand:8432	JNJ-18038683	FALSE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	2.500365296937833	ONO-9054	ncit:C152337	SEPETAPROST	FALSE	FALSE	FALSE
INTERLEUKIN-1 ALPHA	hgnc:5991	IL1A	TTD	2020.06.01	NULL	5.250767123569449	ABT-981	ncit:C166465	LUTIKIZUMAB	FALSE	FALSE	FALSE
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	2.625383561784724	LY-2409021	chembl:CHEMBL3707351	ADOMEGLIVANT	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	1.381780822	LY-2623091	drugbank:DB15367	LY-2623091	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	1.050153425	BLZ-100	chembl:CHEMBL3990023	TOZULERISTIDE	FALSE	FALSE	FALSE
ORNITHINE DECARBOXYLASE	hgnc:8109	ODC1	TTD	2020.06.01	NULL	2.100306849	Difluoromethylornithine	ncit:C226	EFLORNITHINE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 19 MEMBER 1	hgnc:10937	SLC19A1	TTD	2020.06.01	NULL	0.026045472	Methotrexate	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NECTIN CELL ADHESION MOLECULE 4	hgnc:19688	NECTIN4	TTD	2020.06.01	NULL	35.00511415712966	ASG-22ME	chembl:CHEMBL3301589	ENFORTUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.019680536	IUPHAR.LIGAND:54	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.045265234	IUPHAR.LIGAND:7227	rxcui:6779	MESORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.06466462	IUPHAR.LIGAND:36	rxcui:1827	BUSPIRONE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.2263261691193728	IUPHAR.LIGAND:58	ncit:C152944	ZALOSPIRONE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.6326225450083675	IUPHAR.LIGAND:3926	iuphar.ligand:3926	[11C]AZ10419369	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.037213091	IUPHAR.LIGAND:102	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.052718545	IUPHAR.LIGAND:130	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:92	rxcui:33739	PIPAMPERONE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:77	iuphar.ligand:77	SB 714786	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.101562227	IUPHAR.LIGAND:149	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:92	rxcui:33739	PIPAMPERONE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.050246575	IUPHAR.LIGAND:177	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.046059361	IUPHAR.LIGAND:221	iuphar.ligand:221	SB 204741	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.096521454	IUPHAR.LIGAND:173	ncit:C61919	QUIPAZINE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.077217164	IUPHAR.LIGAND:161	iuphar.ligand:161	BW723C86	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.096521454	IUPHAR.LIGAND:219	iuphar.ligand:219	[3H]LSD	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.096521454	IUPHAR.LIGAND:84	rxcui:21877	CYAMEMAZINE	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.1620607136904151	IUPHAR.LIGAND:107	iuphar.ligand:107	5-MEOT	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.018385039	IUPHAR.LIGAND:89	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.1458546423213736	IUPHAR.LIGAND:244	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.024052987	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:783	hgnc:1402	CACNB2	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:4743	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:1264	hgnc:2155	CNN1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12242	ncit:C177068	CLESACOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1382	hgnc:2339	CRABP2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:10344	iuphar.ligand:10344	COMPOUND 1 [LOLLI ET AL., 2019]	FALSE	FALSE	FALSE
NCBIGENE:1382	hgnc:2339	CRABP2	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:8769	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1278	hgnc:2198	COL1A2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:10092	iuphar.ligand:10092	ST034307	FALSE	FALSE	FALSE
NCBIGENE:874	hgnc:1549	CBR3	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:4500	iuphar.ligand:4500	BENZYLSERINE	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12216	iuphar.ligand:12216	MS15	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:11355	rxcui:1494066	MILTEFOSINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.026071336	IUPHAR.LIGAND:2398	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.055039488	IUPHAR.LIGAND:7207	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.038104261	IUPHAR.LIGAND:551	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7894	iuphar.ligand:7894	RXP-407	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.2035181055647073	IUPHAR.LIGAND:6339	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:6313	iuphar.ligand:6313	CYCLO APELIN-12 (1-12)	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	activator	0.7721716358190367	IUPHAR.LIGAND:4203	iuphar.ligand:4203	GMQ	FALSE	FALSE	FALSE
NCBIGENE:2951	hgnc:4640	GSTP1P1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11110	ncit:C166897	EZUTROMID	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.016311796	IUPHAR.LIGAND:407	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	1.544343271638073	IUPHAR.LIGAND:11474	iuphar.ligand:11474	NS383	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:881	iuphar.ligand:881	L-740093	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:766	iuphar.ligand:766	[125I]CCL8 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:797	iuphar.ligand:797	CCL17	FALSE	FALSE	FALSE
NCBIGENE:61	hgnc:1605	CCR4	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:798	iuphar.ligand:798	CCL22	FALSE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:8458	iuphar.ligand:8458	OTELIXIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12980	iuphar.ligand:12980	LC52-0332	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.3431873936973497	IUPHAR.LIGAND:8006	iuphar.ligand:8006	BX-795	FALSE	FALSE	FALSE
NCBIGENE:699	hgnc:1148	BUB1	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:4242	rxcui:623033	LUBIPROSTONE	TRUE	FALSE	FALSE
NCBIGENE:3248	hgnc:5154	HPGD	GuideToPharmacology	2024.1	inhibitor	0.1058622403945453	IUPHAR.LIGAND:8401	ncit:C166804	EVACETRAPIB	FALSE	FALSE	FALSE
NCBIGENE:3248	hgnc:5154	HPGD	GuideToPharmacology	2024.1	inhibitor	0.1058622403945453	IUPHAR.LIGAND:10721	iuphar.ligand:10721	DRL-17822	FALSE	FALSE	FALSE
NCBIGENE:701	hgnc:1149	BUB1B	GuideToPharmacology	2024.1	blocker	3.500511415712967	IUPHAR.LIGAND:4177	iuphar.ligand:4177	DIDS	FALSE	FALSE	FALSE
NCBIGENE:2359	hgnc:3828	FPR3	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9602	rxcui:1927851	BETRIXABAN	TRUE	FALSE	FALSE
NCBIGENE:2360	hgnc:3868	FRA1A	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11754	ncit:C175138	MILVEXIAN	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:8975	iuphar.ligand:8975	IL-34	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9684	iuphar.ligand:9684	COMPOUND 12A [PMID: 29031075]	FALSE	FALSE	FALSE
NCBIGENE:1989	hgnc:1974	CHUK	GuideToPharmacology	2024.1	modulator	0.3409589041278864	IUPHAR.LIGAND:5669	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:2896	rxcui:307296	ETORICOXIB	TRUE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:687	ncit:C169781	AMLINTIDE	FALSE	FALSE	FALSE
NCBIGENE:715	hgnc:1246	C1R	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:716	hgnc:1247	C1S	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:724	hgnc:1327	C4BPAP2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2447	rxcui:4453	FLUFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8948	iuphar.ligand:8948	AZD5069	FALSE	FALSE	FALSE
NCBIGENE:734	hgnc:1355	OSGIN2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:8495	iuphar.ligand:8495	HIV-1 MATRIX PROTEIN P17	FALSE	FALSE	FALSE
NCBIGENE:727	hgnc:1331	C5	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:4278	iuphar.ligand:4278	OCTANOL	FALSE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:821	iuphar.ligand:821	CXCL8	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:840	iuphar.ligand:840	DIOSCIN	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:5662	iuphar.ligand:5662	AT-7519	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.022439176	IUPHAR.LIGAND:5925	drugbank:DB04014	ALSTERPAULLONE	FALSE	FALSE	FALSE
NCBIGENE:1965	hgnc:3265	EIF2S1	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:10063	iuphar.ligand:10063	CDK12 INHIBITOR 2	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10581	iuphar.ligand:10581	COMPOUND 13E [PMID: 31811124]	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:11951	iuphar.ligand:11951	ASAPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:1901	iuphar.ligand:1901	13,14-DIHYDRO-15-KETO-PGF2&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1885	iuphar.ligand:1885	PGJ2	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:1905	iuphar.ligand:1905	TM30089	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.036387853	IUPHAR.LIGAND:83	rxcui:2403	CHLORPROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:62	iuphar.ligand:62	(+)-BUTACLAMOL	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:8777	iuphar.ligand:8777	COMPOUND 51 [CROSIGNANI ET AL., 2011]	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	inhibitor	0.2243917574174978	IUPHAR.LIGAND:943	iuphar.ligand:943	SCH-23390	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1000146118775133	IUPHAR.LIGAND:62	iuphar.ligand:62	(+)-BUTACLAMOL	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.041182487	IUPHAR.LIGAND:48	rxcui:8047	PERGOLIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:957	iuphar.ligand:957	(+)-UH232	FALSE	FALSE	FALSE
NCBIGENE:156	hgnc:289	GRK2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:10482	iuphar.ligand:10482	COMPOUND 16 [PMID: 31498617]	FALSE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:5102	iuphar.ligand:5102	1400W	FALSE	FALSE	FALSE
NCBIGENE:2624	hgnc:4171	GATA2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:6842	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
NCBIGENE:1398	hgnc:2362	CRK	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:2338	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
NCBIGENE:2443	hgnc:3841	FRA11F	GuideToPharmacology	2024.1	antibody	1.875273972703375	IUPHAR.LIGAND:6591	rxcui:354770	NATALIZUMAB	TRUE	TRUE	FALSE
NCBIGENE:2451	hgnc:3848	FRA12D	GuideToPharmacology	2024.1	antibody	3.500511415712966	IUPHAR.LIGAND:6593	rxcui:356988	EFALIZUMAB	TRUE	TRUE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:8067	iuphar.ligand:8067	NVP-AEW541	FALSE	FALSE	TRUE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:5048	iuphar.ligand:5048	PQ401	FALSE	FALSE	FALSE
NCBIGENE:1695	hgnc:6008	IL2RA	GuideToPharmacology	2024.1	antibody	1.715936968486748	IUPHAR.LIGAND:6879	rxcui:196102	BASILIXIMAB	TRUE	TRUE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8080	iuphar.ligand:8080	IRAK4 INHIBITOR 4B [PMID: 18474425]	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:4042	iuphar.ligand:4042	RO3244794	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:5855	iuphar.ligand:5855	FK-788	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:9283	iuphar.ligand:9283	TG6-129	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.4375639269641209	IUPHAR.LIGAND:4285	drugbank:DB07810	PHLORETIN	FALSE	FALSE	FALSE
NCBIGENE:666	hgnc:1087	BOK	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:347	drugbank:DB15954	STRYCHNINE	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.1187956362798518	IUPHAR.LIGAND:12497	rxcui:2641822	EPICATECHIN	FALSE	FALSE	FALSE
NCBIGENE:671	hgnc:1095	BPI	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:7608	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
NCBIGENE:669	hgnc:1093	BPGM	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:12454	iuphar.ligand:12454	SALICIN	FALSE	FALSE	FALSE
NCBIGENE:669	hgnc:1093	BPGM	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:12453	iuphar.ligand:12453	4-NITROPHENYL-&BETA;-D-MANNOPYRANOSIDE	FALSE	FALSE	FALSE
NCBIGENE:663	hgnc:1083	BNIP2	GuideToPharmacology	2024.1	agonist	17.50255707856483	IUPHAR.LIGAND:12427	iuphar.ligand:12427	MALVIDIN-3-GLUCOSIDE	FALSE	FALSE	FALSE
NCBIGENE:661	hgnc:1080	POLR3D	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:12423	iuphar.ligand:12423	STEVIOSIDE	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:12467	iuphar.ligand:12467	CYCLOLINOPEPTIDE 1-MSO,3-MET-CL6	FALSE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	0.7501095890813501	IUPHAR.LIGAND:12438	iuphar.ligand:12438	ARISTOLOCHIC ACID	FALSE	FALSE	FALSE
NCBIGENE:663	hgnc:1083	BNIP2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:7608	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
NCBIGENE:665	hgnc:1085	BNIP3L	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:328	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:7792	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:10459	ncit:C161798	BREPOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:12047	iuphar.ligand:12047	COMPOUND 11 [PMID: 35653642]	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.076765601	IUPHAR.LIGAND:12932	iuphar.ligand:12932	COMPOUND 25AP [PMID: 37796543]	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:10518	iuphar.ligand:10518	BILORPHIN	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.040640612	IUPHAR.LIGAND:1639	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0296486	IUPHAR.LIGAND:8155	iuphar.ligand:8155	COMPOUND 13A [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.069180068	IUPHAR.LIGAND:11619	ncit:C80870	TOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.008301608	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.2075402025126264	IUPHAR.LIGAND:6054	iuphar.ligand:6054	VEGF RECEPTOR 2 KINASE INHIBITOR II	FALSE	FALSE	FALSE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1287	iuphar.ligand:1287	KISSPEPTIN-28	FALSE	FALSE	FALSE
NCBIGENE:525	hgnc:853	ATP6V1B1	GuideToPharmacology	2024.1	activator	1.050153425	IUPHAR.LIGAND:2509	rxcui:7442	NITRIC OXIDE	TRUE	FALSE	FALSE
NCBIGENE:527	hgnc:855	ATP6V0C	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	activator	0.9546849315580819	IUPHAR.LIGAND:4272	iuphar.ligand:4272	NS1619	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	blocker	0.1562728310586145	IUPHAR.LIGAND:2313	rxcui:3226	DEQUALINIUM	TRUE	FALSE	FALSE
NCBIGENE:387	hgnc:667	RHOA	GuideToPharmacology	2024.1	activator	1.500219178	IUPHAR.LIGAND:4272	iuphar.ligand:4272	NS1619	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	blocker	3.750547945	IUPHAR.LIGAND:2388	drugbank:DB01917	PUTRESCINE	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	0.062509132	IUPHAR.LIGAND:707	iuphar.ligand:707	CA2+	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	0.5000730593875667	IUPHAR.LIGAND:2328	iuphar.ligand:2328	CHARYBDOTOXIN	FALSE	FALSE	FALSE
NCBIGENE:443	hgnc:756	ASPA	GuideToPharmacology	2024.1	blocker	0.364636606	IUPHAR.LIGAND:2416	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
NCBIGENE:542	hgnc:879	ALDH7A1P2	GuideToPharmacology	2024.1	blocker	0.091159151	IUPHAR.LIGAND:2416	rxcui:897018	DALFAMPRIDINE	TRUE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	modulator	4.375639269641208	IUPHAR.LIGAND:9433	iuphar.ligand:9433	TOLIMIDONE	FALSE	FALSE	FALSE
NCBIGENE:1380	hgnc:2336	CR2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10261	iuphar.ligand:10261	AT-56	FALSE	FALSE	FALSE
NCBIGENE:2682	hgnc:11114	KDM5C	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7026	iuphar.ligand:7026	PBIT	FALSE	FALSE	FALSE
NCBIGENE:2681	hgnc:4253	GGTA1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7026	iuphar.ligand:7026	PBIT	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:7735	iuphar.ligand:7735	AZ13483342	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:3804	iuphar.ligand:3804	[125I]SHU9119	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:1328	iuphar.ligand:1328	HS024	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.093931433	IUPHAR.LIGAND:5892	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.2059124362184097	IUPHAR.LIGAND:12093	iuphar.ligand:12093	ZANZALINTINIB	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6355	iuphar.ligand:6355	A-850002	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6451	iuphar.ligand:6451	COMPOUND 53 [PMID: 23434029]	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:1425	iuphar.ligand:1425	[3H]M-MPEP	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1406	iuphar.ligand:1406	(R,S)-4-PPG	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:1440	iuphar.ligand:1440	MSOPPE	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1412	iuphar.ligand:1410	L-AP4	FALSE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1410	iuphar.ligand:1410	L-AP4	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:2873	rxcui:4452	FLUDROCORTISONE	TRUE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	3.454452054979901	IUPHAR.LIGAND:2876	rxcui:298869	EPLERENONE	TRUE	FALSE	FALSE
NCBIGENE:1502	hgnc:6875	MAPK13	GuideToPharmacology	2024.1	inhibitor	0.1691068316769549	IUPHAR.LIGAND:5668	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1501	hgnc:2516	CTNND2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:5668	ncit:C76770	DORAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:6059	iuphar.ligand:6059	VX-702	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:7838	iuphar.ligand:7838	BMS-582949	FALSE	FALSE	FALSE
NCBIGENE:1494	hgnc:6877	MAPK3	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:9974	iuphar.ligand:9974	MK-8353	FALSE	FALSE	FALSE
NCBIGENE:2088	ncbigene:2088	ERVK3	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8135	iuphar.ligand:8135	COMPOUND 21 [PMID: 23312943]	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:7869	iuphar.ligand:7869	COMPOUND 5  [PMID: 24900526]	FALSE	FALSE	FALSE
NCBIGENE:1636	hgnc:2707	ACE	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:7844	iuphar.ligand:7844	AZD1236	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12669	iuphar.ligand:12669	MMP13 TRACER  [18F]5J	FALSE	FALSE	FALSE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:5281	rxcui:10734	TRANYLCYPROMINE	TRUE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1453	iuphar.ligand:1453	[LEU13]MOTILIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1454	iuphar.ligand:1454	[PHE3,LEU13]MOTILIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1450	iuphar.ligand:1450	[D-BPA5,ILE13]MOTILIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:12305	iuphar.ligand:12305	VU0486846	FALSE	FALSE	FALSE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12888	iuphar.ligand:12888	FRILUGLANSTAT	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:327	iuphar.ligand:327	METHOCTRAMINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.050246575	IUPHAR.LIGAND:355	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.5527123287967841	IUPHAR.LIGAND:3255	iuphar.ligand:3255	THRX160209	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2663	iuphar.ligand:2663	AD-5061	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:8917	iuphar.ligand:8917	AMG319	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.012756966	IUPHAR.LIGAND:7950	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:7963	iuphar.ligand:7963	PILARALISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:9425	ncit:C174798	NEMIRALISIB	FALSE	FALSE	FALSE
NCBIGENE:1294	hgnc:2214	COL7A1	GuideToPharmacology	2024.1	activator	2.625383561784725	IUPHAR.LIGAND:2351	iuphar.ligand:2351	CALMODULIN	FALSE	FALSE	FALSE
NCBIGENE:1303	hgnc:2188	COL12A1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:9992	iuphar.ligand:9992	COMPOUND 29 [MOSLIN ET AL., 2017]	FALSE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:9610	iuphar.ligand:9610	CBS-3595	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:8214	iuphar.ligand:8214	COMPOUND 14K [PMID: 21982499]	FALSE	FALSE	FALSE
NCBIGENE:1432	hgnc:6876	MAPK14	GuideToPharmacology	2024.1	inhibitor	0.1426838892274307	IUPHAR.LIGAND:7376	ncit:C76401	RILAPLADIB	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:5918	iuphar.ligand:5918	AGL 2043	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:5690	iuphar.ligand:5690	KI-20227	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:7886	iuphar.ligand:7886	FAMITINIB	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.042006137	IUPHAR.LIGAND:5936	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
NCBIGENE:1434	hgnc:2431	CSE1L	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:8782	iuphar.ligand:8782	COMPOUND 69 [PMID: 19136975]	FALSE	FALSE	FALSE
NCBIGENE:2388	hgnc:3900	FRA4A	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:7730	iuphar.ligand:7730	BOCOCIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1543	hgnc:2595	CYP1A1	GuideToPharmacology	2024.1	activator	0.8751278539282416	IUPHAR.LIGAND:8821	iuphar.ligand:8821	MT47-100	FALSE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	0.9376369863516874	IUPHAR.LIGAND:8616	iuphar.ligand:8616	MG-132	FALSE	FALSE	FALSE
NCBIGENE:1257	ncbigene:1257	CNC2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:11423	iuphar.ligand:11423	SGC6870	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	0.2524407270946851	IUPHAR.LIGAND:2611	iuphar.ligand:2611	ROTTLERIN	FALSE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	activator	1.591141552596802	IUPHAR.LIGAND:10066	iuphar.ligand:10066	RASGRP ACTIVATOR 1	FALSE	FALSE	FALSE
NCBIGENE:1487	hgnc:2494	CTBP1	GuideToPharmacology	2024.1	inhibitor	2.019525816757481	IUPHAR.LIGAND:8142	drugbank:DB04098	BALANOL	FALSE	FALSE	FALSE
NCBIGENE:1491	hgnc:2501	CTH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8185	iuphar.ligand:8185	COMPOUND 3 [PMID: 19097791]	FALSE	FALSE	FALSE
NCBIGENE:1491	hgnc:2501	CTH	GuideToPharmacology	2024.1	activator	1.312691780892362	IUPHAR.LIGAND:2391	drugbank:DB04557	ARACHIDONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:9643	iuphar.ligand:9643	RIPA-56	FALSE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:10401	iuphar.ligand:10401	RIPK3 INHIBITOR 42	FALSE	FALSE	FALSE
NCBIGENE:611	hgnc:1012	OPN1SW	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:2814	iuphar.ligand:2814	LG100754	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.054355767	IUPHAR.LIGAND:8189	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:2647	iuphar.ligand:2647	RO 40-6055	FALSE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:5706	iuphar.ligand:5706	TAMATINIB	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.086219493	IUPHAR.LIGAND:5181	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	0.2917092846427472	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.006642337	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.02287916	Paclitaxel	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.4118248724368195	LMB-100	drugbank:DB18591	LMB-100	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	PF-07257876	ncit:C180866	ANTI-CD47/ANTI-PD-L1 BISPECIFIC ANTIBODY PF-07257876	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	PF-06801591	ncit:C124058	SASANLIMAB	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.057073556	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	5.136620012187506	Ensartinib	ncit:C102754	ENSARTINIB	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	1.165474011072658	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.059481927	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1744440904840348	PRN1371	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.019844169	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	LAM-003	ncit:C152979	HSP90 INHIBITOR LAM-003	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.3241214273808302	AGS62P1	chembl:CHEMBL4297893	AGS62P1	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.069089041	Uprosertib	ncit:C84870	UPROSERTIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.004426918	Vandetanib	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.106290832	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.023774188	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.006419031	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.6159257622955366	Baricitinib	rxcui:2047232	BARICITINIB	TRUE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.1620607136904151	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	0.1902451856365742	TGX-221	iuphar.ligand:8244	TGX-221	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	Torkinib	iuphar.ligand:5704	PP-242	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.01823183	Bevacizumab	rxcui:2046138	BEVACIZUMAB-AWWB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.024309107	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	0.384671584	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.2586584789935689	Entinostat	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	0.072927321	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.015454797	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.008429889	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.033117421	R547	iuphar.ligand:5707	R547	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.026748686	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.05073205	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	AG-528	chembl:CHEMBL56542	CHEMBL:CHEMBL56542	FALSE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.068191781	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.011049594	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.070432825	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.1553481397505754	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	SJ000032154	chembl:CHEMBL591876	CHEMBL:CHEMBL591876	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CHLOROBENZILATE	chembl:CHEMBL539904	CHLOROBENZILATE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	NSC-74859	chembl:CHEMBL477936	CHEMBL:CHEMBL477936	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.027347745	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
TOP2B	hgnc:11990	TOP2B	DTC	9/2/20	NULL	0.3337351985319565	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	ChEMBL	33	inhibitor	0.6482428547616604	BOS-589	chembl:CHEMBL4650296	BOS-589	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	TRIMETHOBENZAMIDE HYDROCHLORIDE	rxcui:38685	TRIMETHOBENZAMIDE	TRUE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	DNDI1417165	chembl:CHEMBL1406948	CHEMBL:CHEMBL1406948	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.1544343271638073	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	GNF-PF-2491	chembl:CHEMBL577851	CHEMBL:CHEMBL577851	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.2344092465879218	N-(4-FLUOROBENZYLCARBAMOTHIOYL)BENZAMIDE	chembl:CHEMBL1545737	CHEMBL:CHEMBL1545737	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1363835616511545	NSC-11437	chembl:CHEMBL1814509	CHEMBL:CHEMBL1814509	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.050879526	4'-EPICHAETOVIRIDIN A	chembl:CHEMBL1306556	CHEMBL:CHEMBL1306556	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.023151531	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	DNDI1417024	chembl:CHEMBL1462710	CHEMBL:CHEMBL1462710	FALSE	FALSE	FALSE
IL1R1	hgnc:5993	IL1R1	NCI	14-Sep-17	NULL	0.5385402178019949	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
CA10	hgnc:1369	CA10	PharmGKB	4/5/24	NULL	2.763561643983921	fluticasone propionate	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1605739181519709	ALKS 37	chembl:CHEMBL2364619	METHYLSAMIDORPHAN	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.060169218	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.591141552596803	NBI-56418	rxcui:2049846	ELAGOLIX	TRUE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.022015795	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
NCBIGENE:2839	hgnc:584	APCS	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8256	ncit:C153209	MIRIDESAP	FALSE	FALSE	FALSE
NCBIGENE:1344	hgnc:2645	CYP4F2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:11372	iuphar.ligand:11372	SESAMIN	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12984	iuphar.ligand:12984	BI-4020	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.054020238	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.023151531	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CHRNB4	hgnc:1964	CHRNB4	DTC	9/2/20	NULL	4.375639269641208	3-BENZHYDRYLQUINUCLIDINE	chembl:CHEMBL2332279	CHEMBL:CHEMBL2332279	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.013505059	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.018704642	Dexlansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1584738568481725	FRUQUINTINIB	rxcui:2670179	FRUQUINTINIB	TRUE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:11081	iuphar.ligand:11081	PSB-KD107	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.07699072	Promethazine	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.5707355569097228	VINORELBIN DITARTRATE	chembl:CHEMBL538943	VINORELBINE TARTRATE	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.029581787	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.084146909	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
IFNL4	hgnc:44480	IFNL4	PharmGKB	4/5/24	NULL	3.500511415712966	daclatasvir	rxcui:1606218	DACLATASVIR	FALSE	FALSE	FALSE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	1.276228120312019	Brentuximab vedotin	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.050294704	IUPHAR.LIGAND:40	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.3777530304726222	IUPHAR.LIGAND:7906	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	positive modulator	2.386712328895204	BAMOCAFTOR	ncit:C171861	BAMOCAFTOR	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.030996264	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
HCAR2	hgnc:24827	HCAR2	ChEMBL	33	agonist	17.50255707856483	SCH-900271	drugbank:DB12433	SCH-900271	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CRUFOMATE	ncit:C75214	CRUFOMATE	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.006868237	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	ZUCAPSAICIN	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.035890411	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:P08473	hgnc:7154	MME	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	PL37	iuphar.ligand:7896	PL37	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.1479089330582944	Xylometazoline	rxcui:39841	XYLOMETAZOLINE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.071245144	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.039361073	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.5585922471882393	CLIDINIUM	rxcui:21232	CLIDINIUM	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	TALC	12-May-16	NULL	0.8751278539282416	CANFOSFAMIDE HCL	chembl:CHEMBL2107319	CANFOSFAMIDE HYDROCHLORIDE	FALSE	FALSE	TRUE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.2453629496995069	Suronacrine maleate	ncit:C96776	SURONACRINE MALEATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.018354192	dextromethorphan	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
UNIPROT:P05121	hgnc:8583	SERPINE1	TdgClinicalTrial	Jan-14	NULL	0.1930429089547591	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006978691	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.2500365296937833	E-7050	ncit:C82363	GOLVATINIB	FALSE	FALSE	FALSE
SCN3A	hgnc:10590	SCN3A	ChEMBL	33	blocker	0.072927321	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TLR8	hgnc:15632	TLR8	DTC	9/2/20	NULL	4.922594178346359	RESIQUIMOD	ncit:C63958	RESIQUIMOD	FALSE	FALSE	FALSE
CYTOCHROME P450 26	hgnc:2603	CYP26A1	TTD	2020.06.01	NULL	13.12691780892362	LIAROZOLE	ncit:C1433	LIAROZOLE	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	Icotinib hydrochloride	ncit:C99160	ICOTINIB HYDROCHLORIDE	FALSE	FALSE	FALSE
GDNF RECEPTOR ALPHA-3	hgnc:4245	GFRA3	TTD	2020.06.01	NULL	52.50767123569449	Neublastin	drugbank:DB15438	ARTEMIN	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	agonist	0.038467158	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.030185497	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	HISPIDULIN	drugbank:DB14008	HISPIDULIN	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.078840347	OSI-027	drugbank:DB12387	OSI-027	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.2318219480604613	PHA-680632	chembl:CHEMBL363160	PHA-680632	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.004910471	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL201761	SALINAZID	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:6043	drugbank:DB08009	SU-11652	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	CIViC	10-Apr-24	NULL	0.013957382	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.020164236	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	GNF-PF-130	chembl:CHEMBL578890	CHEMBL:CHEMBL578890	FALSE	FALSE	FALSE
ACACB	hgnc:85	ACACB	ChEMBL	33	inhibitor	1.693795846312725	PF-05175157	drugbank:DB12096	PF-05175157	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	DROMETRIZOLE	rxcui:1426903	DROMETRIZOLE	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	0.3671865121377238	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	DI-TERT-BUTYLHYDROQUINONE	chembl:CHEMBL480626	CHEMBL:CHEMBL480626	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	EPITESTOSTERONE	drugbank:DB07768	EPITESTOSTERONE	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.017578732	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.1121958787087489	valinomycin	ncit:C924	VALINOMYCIN	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.088695391	Birinapant	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1383601350084176	Tiapride	rxcui:10588	TIAPRIDE	FALSE	FALSE	FALSE
CASP8	hgnc:1509	CASP8	ChEMBL	33	inhibitor	0.8078103267029924	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
DDB1	hgnc:2717	DDB1	ChEMBL	33	inhibitor	0.3547815624033412	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	0.5147810905460245	ORELABRUTINIB	ncit:C156173	ORELABRUTINIB	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.006071655	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NCBIGENE:3134	hgnc:4963	HLA-F	GuideToPharmacology	2024.1	modulator	13.12691780892362	IUPHAR.LIGAND:11103	iuphar.ligand:11103	GSK2830371	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.039531467	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	GNF-PF-2383	chembl:CHEMBL578915	CHEMBL:CHEMBL578915	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.012466209	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	LY-83583	chembl:CHEMBL312487	CHEMBL:CHEMBL312487	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000069305	chembl:CHEMBL603739	CHEMBL:CHEMBL603739	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002338872	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	1.400204566285186	JX-594	ncit:C71533	PEXASTIMOGENE DEVACIREPVEC	FALSE	FALSE	FALSE
ALPHA-GLUCOSIDASE	hgnc:4296	GLA	TTD	2020.06.01	NULL	1.009762908	Deoxynojirimycin	ncit:C87373	DUVOGLUSTAT	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.040515178	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TEND	1-Aug-11	NULL	5.834185692854944	IBRITUMOMAB	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1629	iuphar.ligand:1629	NALORPHINE	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.056157937	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-220455	chembl:CHEMBL95207	CHEMBL:CHEMBL95207	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	0.6563458904461812	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
NCBIGENE:3101	hgnc:4925	HK3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:10508	iuphar.ligand:10508	MK-8719	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.201952582	RP-6530	chembl:CHEMBL3545141	RP-6530	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	PERUVOSIDE	drugbank:DB13756	PERUVOSIDE	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	TALC	12-May-16	inhibitor	0.2333674277141978	SB939	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.4303907478335614	DIENOGEST	rxcui:22968	DIENOGEST	TRUE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:5839	iuphar.ligand:5839	GG-2P20	FALSE	FALSE	FALSE
PSMB11	hgnc:31963	PSMB11	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
AIP	hgnc:358	AIP	NCI	14-Sep-17	NULL	4.200613699	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	ZM-241385	drugbank:DB08770	4-{2-[(7-AMINO-2-FURAN-2-YL[1,2,4]TRIAZOLO[1,5-A][1,3,5]TRIAZIN-5-YL)AMINO]ETHYL}PHENOL	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FURFURAL	drugbank:DB16856	FURFURAL	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.025489161	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.032016873	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	blocker	0.2983390411119005	IUPHAR.LIGAND:2294	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	CIViC	10-Apr-24	NULL	0.6471533709721451	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	agonist	0.040021091	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.5000730593875666	ABT-925	rxcui:1661017	ABT-925	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	ChEMBL	33	positive modulator	2.763561643983921	NONACOG BETA PEGOL	rxcui:1990855	COAGULATION FACTOR IX (RECOMBINANT), GLYCOPEGYLATED	TRUE	FALSE	FALSE
UNIPROT:P15248	hgnc:6029	IL9	TdgClinicalTrial	Jan-14	NULL	35.00511415712966	MEDI-528	iuphar.ligand:8934	ENOKIZUMAB	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.044573575	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.1056492378987816	AZD2014	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.2651902587661338	P-T-OCTYLPHENOL	chembl:CHEMBL259327	CHEMBL:CHEMBL259327	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.1605739181519709	Ergot alkaloids	rxcui:4023	ERGOT ALKALOIDS	FALSE	FALSE	FALSE
NCBIGENE:1575	hgnc:7900	NPEPPS	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8671	iuphar.ligand:8671	ANTAQ	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1458546423213736	GNF-PF-372	chembl:CHEMBL580155	CHEMBL:CHEMBL580155	FALSE	FALSE	FALSE
OXER1	hgnc:24884	OXER1	DTC	9/2/20	NULL	35.00511415712966	5-OXO-ETE	iuphar.ligand:3391	5-OXO-ETE	FALSE	FALSE	FALSE
SYNE3	hgnc:19861	SYNE3	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	1.381780822	AUTO2	ncit:C150509	AUTOLOGOUS BCMA/TACI-TARGETED CAR T CELLS AUTO2	FALSE	FALSE	FALSE
NCBIGENE:286	hgnc:492	ANK1	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1326	iuphar.ligand:1326	[125I]NDP-MSH	FALSE	FALSE	FALSE
SLC4A1	hgnc:11027	SLC4A1	PharmGKB	4/5/24	NULL	4.039051633514962	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
LYSOSOMAL ALPHA-GLUCOSIDASE	hgnc:4065	GAA	TTD	2020.06.01	NULL	0.5469549087051511	Deoxynojirimycin	ncit:C87373	DUVOGLUSTAT	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.047219129	IUPHAR.LIGAND:136	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:8526	iuphar.ligand:8526	ELABELA/TODDLER-11	FALSE	FALSE	FALSE
NCBIGENE:982	ncbigene:982	CDB2	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8881	iuphar.ligand:8881	COMPOUND 1A [PMID: 23597791]	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.038159645	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
UNIPROT:P47872	hgnc:10608	SCTR	TdgClinicalTrial	Jan-14	NULL	31.50460274141669	RG1068	rxcui:606396	SECRETIN HUMAN, SYNTHETIC	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.3947945205691315	FTORMETAZINE	ncit:C65774	FTORMETAZINE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.014537008	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.040112812	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.6403374540938354	CHEMOSENSITIZER	ncit:C1744	MULTIDRUG RESISTANCE MODULATOR	FALSE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.074797252	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.003001124	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	BISACODYL	rxcui:1596	BISACODYL	TRUE	FALSE	FALSE
CA2	hgnc:1373	CA2	NCI	14-Sep-17	NULL	1.211715490054488	DORZOLAMIDE	rxcui:60207	DORZOLAMIDE	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	8-[METHYL(4-PHENYLBUTYL)AMINO]CAFFEINE	chembl:CHEMBL1927684	CHEMBL:CHEMBL1927684	FALSE	FALSE	FALSE
NCBIGENE:2730	hgnc:4312	GCLM	GuideToPharmacology	2024.1	NULL	4.039051633514961	IUPHAR.LIGAND:8575	iuphar.ligand:8575	PFI-4	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	1.141471113819445	Decernotinib	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.015263858	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.025776962	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.3697723326457359	ANILERIDINE PHOSPHATE	ncit:C87352	ANILERIDINE PHOSPHATE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.080103236	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
UNIPROT:Q14654	hgnc:6257	KCNJ11	TEND	1-Aug-11	NULL	0.5173169579871378	REPAGLINIDE	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	ChEMBL	33	inhibitor	0.6482428547616604	GALCANEZUMAB	rxcui:2058846	GALCANEZUMAB	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	TRAPIDIL	rxcui:10735	TRAPIDIL	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.052090944	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NPM1	hgnc:7910	NPM1	FDA	10-Apr-24	NULL	0.7143900848393808	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.031254566	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.03070624	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.2536602475154323	PHENYLEPHRINE BITARTRATE	rxcui:91167	PHENYLEPHRINE BITARTRATE	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.1944728564284981	RG3487	chembl:CHEMBL2151439	RG3487	FALSE	FALSE	FALSE
CASP4	hgnc:1505	CASP4	ChEMBL	33	inhibitor	4.039051633514962	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.8140724222588294	CLENBUTEROL	rxcui:2580	CLENBUTEROL	TRUE	FALSE	FALSE
RPS13	hgnc:10386	RPS13	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1605739181519709	KP201	chembl:CHEMBL3137310	BENZHYDROCODONE HYDROCHLORIDE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.028360625	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.5385402178019948	Bunazosin	rxcui:19850	BUNAZOSIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	(+/-)-PENTAACETYLCATECHIN	chembl:CHEMBL1336025	(+/-)-PENTAACETYLCATECHIN	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.3962843112127887	DEMETHYLWEDELOLACTONE	chembl:CHEMBL2089002	DEMETHYLWEDELOLACTONE	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.4773424657790409	NAPROXEN ETEMESIL	ncit:C166529	NAPROXEN ETEMESIL	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:3976	iuphar.ligand:3976	[125I]EPIBATIDINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	PERMETHRIN	rxcui:33199	PERMETHRIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004698673	zonisamide	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.063110182	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	2.282942227638891	ATRASENTAN HYDROCHLORIDE	ncit:C1779	ATRASENTAN HYDROCHLORIDE	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.069180068	CLEBOPRIDE	rxcui:21224	CLEBOPRIDE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.044198376	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
NCBIGENE:1230	hgnc:1602	CCR1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:4805	rxcui:8011	PENTOSTATIN	TRUE	FALSE	TRUE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:4008	iuphar.ligand:4008	&ALPHA;-CONOTOXIN RGIA	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:6162	iuphar.ligand:6162	ZK-158252	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.5527123287967842	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.00473106	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.1666910197958555	TIAPRIDE	rxcui:10588	TIAPRIDE	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	ChEMBL	33	inhibitor	0.1556551518844698	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.084553416	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.005893778	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.016460085	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
EZH2	hgnc:3527	EZH2	CIViC	10-Apr-24	NULL	2.333674277141978	GSK126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.048764961	Etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.013415348	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.070129236	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
NCBIGENE:3011	hgnc:12565	UNC119	GuideToPharmacology	2024.1	NULL	52.50767123569449	IUPHAR.LIGAND:9966	iuphar.ligand:9966	SQUARUNKIN A	FALSE	FALSE	FALSE
PTPN6	hgnc:9658	PTPN6	DTC	9/2/20	NULL	1.250182648468916	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.073540156	LUZINDOLE	iuphar.ligand:1363	LUZINDOLE	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	3.281729452230906	KO-143	iuphar.ligand:10007	KO 143	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	agonist	0.2243917574174978	IUPHAR.LIGAND:9637	iuphar.ligand:9637	A77636	FALSE	FALSE	FALSE
NCBIGENE:3097	hgnc:4921	HIVEP2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10486	iuphar.ligand:10486	COMPOUND 21B [PMID: 31430136]	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	DESVENLAFAXINE SUCCINATE	rxcui:683693	DESVENLAFAXINE SUCCINATE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.025827679	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	agonist	0.2885036881082115	APIMOSTINEL	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	0.8468979231563628	IUPHAR.LIGAND:573	iuphar.ligand:573	C5A	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.099446347	VERNAKALANT HYDROCHLORIDE	ncit:C152865	VERNAKALANT HYDROCHLORIDE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.3697723326457359	CEP-5214	chembl:CHEMBL150894	CEP-5214	FALSE	FALSE	FALSE
UNIPROT:P30411	hgnc:1030	BDKRB2	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	ANATIBANT	ncit:C79554	ANATIBANT	FALSE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.09869863	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
NCBIGENE:2844	hgnc:4476	GPR21	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:8318	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:6577	iuphar.ligand:6577	CID16020046	FALSE	FALSE	FALSE
NCBIGENE:540	hgnc:870	ATP7B	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:7972	iuphar.ligand:7972	WP1066	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1773907812016706	LY294002	ncit:C148229	PI3K/BET INHIBITOR LY294002	FALSE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.02832129	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
IFI27	hgnc:5397	IFI27	NCI	14-Sep-17	NULL	0.8468979231563629	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	NCI	14-Sep-17	NULL	0.09869863	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	TALC	12-May-16	inhibitor	0.2991890098899972	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	0.4245903334422736	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
NCBIGENE:748	hgnc:10484	RYR2	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:10161	iuphar.ligand:10161	VK-II-86	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1164249916534246	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.019107595	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.07699072	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1293	iuphar.ligand:1293	MCH6-17	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.053038052	TCMDC-125813	chembl:CHEMBL580076	CHEMBL:CHEMBL580076	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.043629141	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	1.875273972703375	salvianolic acid b	chembl:CHEMBL541265	SALVIANOLIC ACID B	FALSE	FALSE	FALSE
NCBIGENE:1326	hgnc:6860	MAP3K8	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8747	iuphar.ligand:8747	COMPOUND 3 [PMID: 18255300]	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:1220	iuphar.ligand:1220	[3H]PYRILAMINE	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	agonist	0.1071585127259071	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
ETS2	hgnc:3489	ETS2	PharmGKB	4/5/24	NULL	0.3580068493342807	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
DICKKOPF-RELATED PROTEIN 1	hgnc:2891	DKK1	TTD	2020.06.01	NULL	11.66837138570988	BHQ-880	hemonc:57	BHQ-880	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.1256164383629055	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.1229687850953032	SU-014813	chembl:CHEMBL1721885	SU-014813	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.005297384	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.2302968036653267	TOLTERODINE	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:2199	ncit:C80380	SATAVAPTAN	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.074797252	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.1526385791735305	GW632580X	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003703461	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.1215455352678113	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.2500365296937833	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.060492709	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:8793	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:9962	rxcui:2205637	TRIFAROTENE	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:9117	ncit:C121829	MIVEBRESIB	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	NSC-695801	chembl:CHEMBL461193	CHEMBL:CHEMBL461193	FALSE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	DTC	9/2/20	NULL	1.071585127259071	IC261	drugbank:DB03083	IC261	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.099446347	TCMDC-125813	chembl:CHEMBL580076	CHEMBL:CHEMBL580076	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	binder	0.364636606	TALQUETAMAB	rxcui:2644447	TALQUETAMAB	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC, PROMPT	chembl:CHEMBL2108493	INSULIN ZINC, PROMPT	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016621612	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.2083637747448194	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
PIPSL	hgnc:23733	PIPSL	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:6996	iuphar.ligand:6996	(S)-FTY720-PHOSPHATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	SB-215505	iuphar.ligand:190	SB 215505	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	1.458546423213736	Itacitinib	ncit:C116855	ITACITINIB	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.024674658	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1842374429322614	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.013879903	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.007123548	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CGI	2/1/22	NULL	0.009272878	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.047886613	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
AQP4	hgnc:637	AQP4	DTC	9/2/20	NULL	0.065799087	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.012878997	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
UNIPROT:P30872	hgnc:11330	SSTR1	TEND	1-Aug-11	NULL	1.215455352678113	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.026519026	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.076765601	(+)-EPITAXIFOLIN	chembl:CHEMBL9249	(+)-EPITAXIFOLIN	FALSE	FALSE	FALSE
UNIPROT:P11836	hgnc:7315	MS4A1	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	IBRITUMOMAB	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.010128795	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:2745	hgnc:4330	GLRX	GuideToPharmacology	2024.1	NULL	5.250767124	IUPHAR.LIGAND:6891	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
MATK	hgnc:6906	MATK	DTC	9/2/20	NULL	0.069454592	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.093763699	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1988926940746003	IUPHAR.LIGAND:301	ncit:C132273	MILAMELINE	FALSE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	AVICINE	ncit:C30000	CTP-37-DT VACCINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	8.078103267029922	BOMBESIN ANTAGONIST	ncit:C2132	BOMBESIN ANTAGONIST	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	CIViC	10-Apr-24	NULL	0.073540156	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.7895890411382631	GSK3787	chembl:CHEMBL598608	CHEMBL:CHEMBL598608	FALSE	FALSE	FALSE
CAMK2A	hgnc:1460	CAMK2A	DTC	9/2/20	NULL	0.063568609	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2273059360852575	CLODRONATE	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.2206204673768676	BESTATIN	ncit:C1015	UBENIMEX	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.3621218705909966	TCMDC-125142	chembl:CHEMBL528791	CHEMBL:CHEMBL528791	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.031929262	Perphenazine	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	4-METHYLDAPHNETIN	chembl:CHEMBL276618	4-METHYLDAPHNETIN	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.546954909	NICERGOLINE	rxcui:7398	NICERGOLINE	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.3804903712731485	atrasentan	ncit:C61606	ATRASENTAN	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 2	hgnc:3169	S1PR2	TTD	2020.06.01	NULL	2.500365296937833	Jte 013	iuphar.ligand:2917	JTE-013	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	NCI	14-Sep-17	NULL	0.2375912725597036	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.067317527	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	modulator	5.834185692854944	RG7342	chembl:CHEMBL3545203	RG7342	FALSE	FALSE	FALSE
FGA	hgnc:3661	FGA	ChEMBL	33	cleavage	3.182283105193605	ALFIMEPRASE	ncit:C79877	ALFIMEPRASE	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	ChEMBL	33	inhibitor	0.072324616	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	TIRATRICOL	rxcui:13982	TIRATRICOL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	7,4'-DIHYDROXYFLAVONE	chembl:CHEMBL294878	CHEMBL:CHEMBL294878	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	DOXACURIUM	rxcui:23651	DOXACURIUM	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
CASP10	hgnc:1500	CASP10	ChEMBL	33	inhibitor	4.039051633514962	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	DEXTROMORAMIDE	rxcui:3290	DEXTROMORAMIDE	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.06714536	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	DIPHENHYDRAMINE	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
FGB	hgnc:3662	FGB	DTC	9/2/20	NULL	0.1458546423213736	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
MAP3K10	hgnc:6849	MAP3K10	DTC	9/2/20	NULL	0.081030357	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
T-CELL-SPECIFIC SURFACE GLYCOPROTEIN CD28	hgnc:1653	CD28	TTD	2020.06.01	NULL	0.7001022831425934	Belatacept	rxcui:1112973	BELATACEPT	TRUE	FALSE	FALSE
CLU	hgnc:2095	CLU	NCI	14-Sep-17	NULL	3.182283105193606	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003439517	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.019980088	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.084553416	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
TMCO6	hgnc:28814	TMCO6	PharmGKB	4/5/24	NULL	5.527123287967842	fluticasone propionate	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	SALVINORIN A	drugbank:DB12327	SALVINORIN A	FALSE	FALSE	FALSE
SIRT2	hgnc:10886	SIRT2	DTC	9/2/20	NULL	0.3977853881492008	GW5074	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.073540156	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
SELE	hgnc:10718	SELE	DTC	9/2/20	NULL	4.773424657790408	SIALYL LEWIS X	chembl:CHEMBL375586	SIALYL LEWIS X	FALSE	FALSE	FALSE
CCL18	hgnc:10616	CCL18	NCI	14-Sep-17	NULL	1.810609352954982	LD78	ncit:C1391	RECOMBINANT MACROPHAGE INFLAMMATORY PROTEIN-1 ALPHA	FALSE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	NCI	14-Sep-17	NULL	0.258658479	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1221108633388244	HYDRALAZINE	rxcui:5470	HYDRALAZINE	TRUE	FALSE	FALSE
GABPA	hgnc:4071	GABPA	NCI	14-Sep-17	NULL	0.1207072901969988	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P24530	hgnc:3180	EDNRB	TdgClinicalTrial	Jan-14	NULL	2.812910959055062	MACITENTAN	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW861893X	chembl:CHEMBL519881	GW861893X	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE	chembl:CHEMBL1255936	CHEMBL:CHEMBL1255936	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	FLAVONE	rxcui:1536070	FLAVONE	FALSE	FALSE	FALSE
NOTCH3	hgnc:7883	NOTCH3	MyCancerGenome	20-Jun-17	other/unknown	0.7501095890813498	PF-03084014	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:3874	iuphar.ligand:3874	EUROPIUM-LABELLED RELAXIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.035560536	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-74859	chembl:CHEMBL477936	CHEMBL:CHEMBL477936	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.1988926940746003	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007063179	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
ARID4A	hgnc:9885	ARID4A	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.2991890098899972	AZD0530	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:2920	iuphar.ligand:2920	PAMOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:478	hgnc:801	ATP1A3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4267	iuphar.ligand:4267	NF449	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.062833272	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.072524408	GLAUCINE METHIODIDE	chembl:CHEMBL225852	GLAUCINE METHIODIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.092606122	TESEVATINIB	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	DNDI1417221	chembl:CHEMBL1459280	CHEMBL:CHEMBL1459280	FALSE	FALSE	FALSE
NCBIGENE:714	hgnc:1245	C1QC	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.069454592	IUPHAR.LIGAND:40	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:2030	hgnc:11003	SLC29A1	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:8017	iuphar.ligand:8017	IM-12	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.007649719	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.008240375	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.4251633298436802	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005085489	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	PD-168,077	iuphar.ligand:975	PD168,077	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.4375639269641208	DIFLOMOTECAN	ncit:C90824	DIFLOMOTECAN	FALSE	FALSE	FALSE
NOX1	hgnc:7889	NOX1	DTC	9/2/20	NULL	17.50255707856483	TCMDC-125505	chembl:CHEMBL587104	CHEMBL:CHEMBL587104	FALSE	FALSE	FALSE
KLB	hgnc:15527	KLB	ChEMBL	33	activator	4.375639269641208	ALDAFERMIN	ncit:C169769	ALDAFERMIN	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	inhibitor	0.2344092465879218	IUPHAR.LIGAND:4210	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:5437	iuphar.ligand:5437	ML169	FALSE	FALSE	FALSE
CLK3	hgnc:2071	CLK3	DTC	9/2/20	NULL	2.333674277141977	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
RUNX3	hgnc:10473	RUNX3	NCI	14-Sep-17	NULL	1.419126249613364	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
AOX1	hgnc:553	AOX1	PharmGKB	4/5/24	NULL	1.615620653405984	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
PLAUR	hgnc:9053	PLAUR	NCI	14-Sep-17	NULL	13.12691780892362	MCP-2	ncit:C1671	RECOMBINANT HUMAN MONOCYTE CHEMOATTRACTANT PROTEIN-2	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.016807833	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:415	iuphar.ligand:415	(S)-PIA	FALSE	FALSE	FALSE
NCBIGENE:70	hgnc:143	ACTC1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:841	iuphar.ligand:841	DURAMYCIN	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:10507	iuphar.ligand:10507	OMO-1	FALSE	FALSE	FALSE
NCBIGENE:2976	hgnc:4665	GTF3C2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10373	iuphar.ligand:10373	NC1	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.026412309	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Retifanlimab	rxcui:2632981	RETIFANLIMAB	TRUE	FALSE	FALSE
CORTICOSTEROID 11-BETA-DEHYDROGENASE 1	hgnc:5208	HSD11B1	TTD	2020.06.01	NULL	0.7721716358190367	GLYCYRRHIZIN	rxcui:26143	GLYCYRRHIZIC ACID	TRUE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.2500365296937833	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.056581542	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.5357925636295358	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.1000146118775133	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:9928	iuphar.ligand:9928	PUQUITINIB	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.182318303	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	GUANIDINONALTRINDOLE	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
PSMA4	hgnc:9533	PSMA4	DTC	9/2/20	NULL	0.5000730593875666	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	PHOSMET	drugbank:DB11448	PHOSMET	FALSE	FALSE	FALSE
NCBIGENE:2160	hgnc:3529	F11	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:12708	iuphar.ligand:12708	GDC-0339	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	DNDI1417221	chembl:CHEMBL1459280	CHEMBL:CHEMBL1459280	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.041150213	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.039778539	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	4.375639269641208	GO-203-2c	drugbank:DB15008	GO-203-2C	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.029416062	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
APH1A	hgnc:29509	APH1A	DTC	9/2/20	NULL	1.406455479527531	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	DNDI1417692	chembl:CHEMBL1481509	CHEMBL:CHEMBL1481509	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.1751715470748774	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.041396776	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	EMETINE	rxcui:3820	EMETINE	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.1904575128526865	AMETHOPTERIN	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
GSC1	hgnc:4612	GSC	ChEMBL	33	inhibitor	10.50153424713889	MICAFUNGIN SODIUM	rxcui:487070	MICAFUNGIN SODIUM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	EUGENYL BENZOAT	chembl:CHEMBL264141	EUGENYL BENZOAT	FALSE	FALSE	FALSE
NGF	hgnc:7808	NGF	ChEMBL	33	inhibitor	15.00219178	MEDI-578	chembl:CHEMBL2109527	MEDI-578	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:5924	drugbank:DB07364	6-PHENYL[5H]PYRROLO[2,3-B]PYRAZINE	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.011277421	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.01708122	IUPHAR.LIGAND:5698	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1294	iuphar.ligand:1294	S36057	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	activator	0.3088686543276147	IUPHAR.LIGAND:11997	ncit:C175863	TEREVALEFIM	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.031707531	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
NCBIGENE:2405	hgnc:3916	FRA6E	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:10409	iuphar.ligand:10409	ZETOMIPZOMIB	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	TCMDC-124544	chembl:CHEMBL531322	CHEMBL:CHEMBL531322	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.039068208	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	ChEMBL	33	inhibitor	3.281729452230906	PIRITREXIM	ncit:C1031	PIRITREXIM	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	0.5250767123569451	TAE684	ncit:C171615	ALK INHIBITOR TAE684	FALSE	FALSE	TRUE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.364636606	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	1.346350544504987	CORDYCEPIN	rxcui:1989289	CORDYCEPIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	DIMPYLATE	ncit:C169912	DIMPYLATE	FALSE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	7.876150685354174	PEGINESATIDE	rxcui:1248798	PEGINESATIDE	FALSE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	EP-100	chembl:CHEMBL4297748	EP-100	FALSE	FALSE	FALSE
NCBIGENE:2884	hgnc:4561	GPX1P2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10319	rxcui:2623641	OLUTASIDENIB	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.024674658	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.1758069349409414	ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	CIViC	10-Apr-24	NULL	0.058277105	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	NITRILOTRIACETIC ACID	drugbank:DB03040	NITRILOTRIACETIC ACID	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	BUFLOMEDIL	rxcui:19836	BUFLOMEDIL	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
CD9	hgnc:1709	CD9	NCI	14-Sep-17	NULL	0.305277158	HERBIMYCIN A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.023016221	ABT-348	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1230	hgnc:1602	CCR1	GuideToPharmacology	2024.1	inhibitor	1.166837138570989	IUPHAR.LIGAND:5179	iuphar.ligand:5179	EHNA	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.693795846312725	Bepotastine	rxcui:658552	BEPOTASTINE BESILATE	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.018699313	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	PharmGKB	4/5/24	NULL	0.09869863	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
RRM2	hgnc:10452	RRM2	PharmGKB	4/5/24	NULL	0.5385402178019949	cladribine	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
UNIPROT:P35346	hgnc:11334	SSTR5	TEND	1-Aug-11	NULL	0.729273212	OCTREOTIDE	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
INTERFERON ALPHA/BETA RECEPTOR 2	hgnc:5433	IFNAR2	TTD	2020.06.01	NULL	0.9376369863516874	Interferon Alfa-2b, Recombinant	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.2692701089009974	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
GPR12	hgnc:4466	GPR12	DTC	9/2/20	NULL	15.00219178	NEOCYCLOCITRINOL B	chembl:CHEMBL497296	NEOCYCLOCITRINOL B	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.076208521	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.1717808219270267	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
FUS	hgnc:4010	FUS	NCI	14-Sep-17	NULL	0.384671584	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	0.1988926940746003	muraglitazar	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
GLRA2	hgnc:4327	GLRA2	DTC	9/2/20	NULL	0.3125456621172291	WIN-552122	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	APLAVIROC HYDROCHLORIDE	ncit:C76492	APLAVIROC HYDROCHLORIDE	FALSE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	NULL	0.546954909	IUPHAR.LIGAND:5050	iuphar.ligand:5050	PROTEIN S	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.015193192	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:1378	hgnc:2334	CR1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8812	iuphar.ligand:8812	COMPOUND 30 [PMID: 15953724]	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00449706	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
PSMD13	hgnc:9558	PSMD13	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	0.6250913242344582	Adapalene	rxcui:60223	ADAPALENE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.035560536	IRESSA	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	SJ000133784	chembl:CHEMBL589670	CHEMBL:CHEMBL589670	FALSE	FALSE	FALSE
RNF8	hgnc:10071	RNF8	PharmGKB	4/5/24	NULL	0.3977853881492008	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.084146909	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
UNIPROT:Q9H244	hgnc:18124	P2RY12	TdgClinicalTrial	Jan-14	NULL	1.262203635473425	TICLOPIDINE	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
NCBIGENE:1373	hgnc:2323	CPS1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11517	ncit:C166470	SOTICLESTAT	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.00937637	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:7354	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
HRH4	hgnc:17383	HRH4	DTC	9/2/20	NULL	9.546849315580817	VUF-10499	chembl:CHEMBL454890	CHEMBL:CHEMBL454890	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.05010274	URSODIOL	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.03223307	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.4667348554283955	GP100	ncit:C2386	GP100 ANTIGEN	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.3947945205691315	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:7743	iuphar.ligand:7743	IZORLISIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.017274533	lidocaine	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:10253	iuphar.ligand:10253	[125I]26RFA (HUMAN)	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.087512785	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:4033	iuphar.ligand:4033	GW803430	FALSE	FALSE	FALSE
NCBIGENE:1484	ncbigene:1484	CTAA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524936	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.088396753	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	NIGULDIPINE	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	0.054020238	levodopa	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.036162308	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009170044	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.7395446652914718	V-101	chembl:CHEMBL1365576	TETRASUL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CV-3988	iuphar.ligand:6079	CV-3988	FALSE	FALSE	FALSE
ITGB5	hgnc:6160	ITGB5	ChEMBL	33	inhibitor	2.187819634820604	ABITUZUMAB	ncit:C82422	ABITUZUMAB	FALSE	FALSE	FALSE
CACNA1F	hgnc:1393	CACNA1F	ChEMBL	33	blocker	0.3125456621172291	AMLODIPINE BENZOATE	rxcui:2184116	AMLODIPINE BENZOATE	TRUE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.090064616	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
MCHR2	hgnc:20867	MCHR2	DTC	9/2/20	NULL	35.00511415712966	SB-568849	iuphar.ligand:1312	SB-568849	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.042689164	IUPHAR.LIGAND:2880	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	FN-1501	drugbank:DB17383	FN-1501	FALSE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	CIViC	10-Apr-24	NULL	0.1835932560688619	VINORELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
PSMA8	hgnc:22985	PSMA8	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	ZIMELIDINE DIHYDROCHLORIDE	chembl:CHEMBL1257002	ZIMELIDINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
PADI2	hgnc:18341	PADI2	DTC	9/2/20	NULL	1.750255707856483	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	2.573905452730122	Canakinumab	rxcui:853491	CANAKINUMAB	TRUE	TRUE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	GNF-PF-1859	chembl:CHEMBL1520837	CHEMBL:CHEMBL1520837	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TEND	1-Aug-11	NULL	0.6482428547616605	CETUXIMAB	rxcui:318341	CETUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.1595977849109255	DIPHENIDOL	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.006858369	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
BIRC7	hgnc:13702	BIRC7	CIViC	10-Apr-24	NULL	0.1810609352954982	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
IRF6	hgnc:6121	IRF6	PharmGKB	4/5/24	NULL	5.250767124	interferon beta-1b	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
NOS1	hgnc:7872	NOS1	ChEMBL	33	inhibitor	0.2112984757975633	TILARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:8799	ncit:C79817	AZALANSTAT	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6083	iuphar.ligand:6083	GALANIN(7-29) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:2625	hgnc:4172	GATA3	GuideToPharmacology	2024.1	inhibitor	0.1256164383629055	IUPHAR.LIGAND:6832	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
FGFR2	hgnc:3689	FGFR2	DoCM	10-Apr-24	NULL	0.3174882446809434	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1751715470748774	OXYMORPHONE	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.015344147	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.033658764	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.034118045	RELCOVAPTAN	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	1.166837138570988	BISPECIFIC ANTIBODY	ncit:C1454	BISPECIFIC ANTIBODY	FALSE	FALSE	FALSE
TNF ALPHA CONVERTING ENZYME	hgnc:195	ADAM17	TTD	2020.06.01	NULL	3.500511415712967	Apratastat	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.1666910197958555	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.010614043	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
NCBIGENE:2661	hgnc:4224	GDF9	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.021189536	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	CNQX DISODIUM	chembl:CHEMBL1255647	CHEMBL:CHEMBL1255647	FALSE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.218327115	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1204304386139782	ELUXADOLINE	rxcui:1653781	ELUXADOLINE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	1.250182648468916	DUTEPLASE	ncit:C169926	DUTEPLASE	FALSE	FALSE	FALSE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:10139	iuphar.ligand:10139	STAT3 INHIBITOR 8Q	FALSE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	5.527123287967842	ARRY-502	drugbank:DB16053	ARRY-502	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	8-[3-(TRIFLUOROMETHYL)PHENOXYMETHYL]CAFFEINE	chembl:CHEMBL2088303	CHEMBL:CHEMBL2088303	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007727398	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 27	hgnc:5246	HSPB1	TTD	2020.06.01	NULL	4.375639269641208	OGX-427	ncit:C71740	APATORSEN	FALSE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	TALC	12-May-16	antibody	0.8899605294185507	GC-1008	chembl:CHEMBL1743022	FRESOLIMUMAB	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	ORPHENADRINE (CHLORIDE)	chembl:CHEMBL1201023	ORPHENADRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1250182648468916	CLOBETASOL PROPIONATE	rxcui:21245	CLOBETASOL PROPIONATE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
UNIPROT:O14965	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.3236220106976548	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:748	iuphar.ligand:748	L-759,633	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:1312	iuphar.ligand:1312	SB-568849	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	ODM-203	drugbank:DB16843	ODM-203	FALSE	FALSE	FALSE
NCBIGENE:310	hgnc:545	ANXA7	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:1582	ncit:C156766	MECLINERTANT	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.018699313	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.015475294	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	(+)-EPITAXIFOLIN	chembl:CHEMBL9249	(+)-EPITAXIFOLIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PENT-1-ENE	chembl:CHEMBL295337	CHEMBL:CHEMBL295337	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1875273972703374	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.03591496	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
CYSLTR1	hgnc:17451	CYSLTR1	ChEMBL	33	inhibitor	9.546849315580817	CR-3465	chembl:CHEMBL3545273	CR-3465	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.3182283105193606	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:153	iuphar.ligand:153	(+)-DOI	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.087222045	IUPHAR.LIGAND:7247	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
PROTEASOME	hgnc:9338	PRB2	TTD	2020.06.01	NULL	0.3571950424196904	Marizomib	ncit:C64634	MARIZOMIB	FALSE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	2-PYRIDYLKETONE BENZOYL HYDRAZONE	chembl:CHEMBL252151	CHEMBL:CHEMBL252151	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	P-T-OCTYLPHENOL	chembl:CHEMBL259327	CHEMBL:CHEMBL259327	FALSE	FALSE	FALSE
NPAS3	hgnc:19311	NPAS3	PharmGKB	4/5/24	NULL	1.567393171214761	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	0.9546849315580819	LIK-066	ncit:C150375	LICOGLIFLOZIN	FALSE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.062139256	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	agonist	0.040021091	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.041672755	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:136	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:677	hgnc:1107	ZFP36L1	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:9675	drugbank:DB05767	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	blocker	0.5303805175322676	IUPHAR.LIGAND:4000	iuphar.ligand:4000	NS1738	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2252	iuphar.ligand:2252	L-371,257	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.010871153	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1458546423213736	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:12525	iuphar.ligand:12525	OPTOBI-1	FALSE	FALSE	FALSE
KINESIN-LIKE PROTEIN KIF11	hgnc:6388	KIF11	TTD	2020.06.01	NULL	6.563458904461812	AZD-4877	drugbank:DB11671	AZD-4877	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TEND	1-Aug-11	NULL	0.6775183385250904	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.04907259	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.024490518	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
IL11	hgnc:5966	IL11	PharmGKB	4/5/24	NULL	0.5625821918110125	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	N-PROPYL BROMIDE	chembl:CHEMBL1230095	N-PROPYL BROMIDE	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.015921065	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	METHENOLONE ENANTHATE	rxcui:29654	METHENOLONE ENANTHATE	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.026058398	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1968053644516285	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.001870464	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.039214094	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.085332077	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.004235514	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	0.6563458904461812	IUPHAR.LIGAND:2317	iuphar.ligand:2317	NS309	FALSE	FALSE	FALSE
UNIPROT:P47989	hgnc:12805	XDH	TEND	1-Aug-11	NULL	0.31414846	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	DTC	9/2/20	NULL	0.5357925636295356	N6-PHENYLADENOSINE	chembl:CHEMBL262083	N6-PHENYLADENOSINE	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.023274677	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	7-HYDROXYCHLORPROMAZINE	chembl:CHEMBL909	7-HYDROXYCHLORPROMAZINE	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.1835932560688619	FOSPHENYTOIN	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.2075402025126264	Dihydroergotoxine	rxcui:3419	DIHYDROERGOTOXINE	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.1143957978991165	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	inhibitor	7.876150685354174	MK-0893	drugbank:DB12044	MK-0893	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.4278402841426959	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.079557078	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
PML	hgnc:9113	PML	CIViC	10-Apr-24	NULL	0.384671584	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02639903	THC	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
CBR1	hgnc:1548	CBR1	PharmGKB	4/5/24	NULL	0.2134458180312784	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	NCI	14-Sep-17	NULL	0.045265234	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CHI3L1	hgnc:1932	CHI3L1	NCI	14-Sep-17	NULL	4.375639269641208	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	1.944728564284981	CELL SURFACE ANTIGEN	ncit:C269	CELL SURFACE ANTIGEN	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	CancerCommons	25-Jul-13	inhibitor	2.100306849	SNS-032	drugbank:DB05969	SNS-032	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	CancerCommons	25-Jul-13	inhibitor	0.297662535	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	CancerCommons	25-Jul-13	inhibitor	0.3621218705909965	AT13387	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	CancerCommons	25-Jul-13	inhibitor	0.7395446652914718	DS-3078A	chembl:CHEMBL3544963	DS-3078A	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CancerCommons	25-Jul-13	inhibitor	1.184383561707394	BIBW2992	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CGI	2/1/22	NULL	NULL	4OHtestosterone	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.070690956	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.085796848	Gefitinib	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
FANCA	hgnc:3582	FANCA	CGI	2/1/22	NULL	0.3977853881492008	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
GNA11	hgnc:4379	GNA11	CGI	2/1/22	NULL	0.095468493	Vorinostat	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	0.064824285	Azacytidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.043756393	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	CGI	2/1/22	NULL	0.041672755	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	CGI	2/1/22	NULL	0.4102161815288633	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.3547815624033412	MEPENZOLATE BROMIDE	rxcui:52560	MEPENZOLATE BROMIDE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.2365210416022274	OXYPHENONIUM BROMIDE	rxcui:42833	OXYPHENONIUM BROMIDE	TRUE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	3.125456621172291	LANREOTIDE ACETATE	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
IMPA1	hgnc:6050	IMPA1	ChEMBL	33	inhibitor	8.751278539282415	LITHIUM CITRATE	rxcui:52105	LITHIUM CITRATE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.7095631248066824	CYCLOPENTOLATE HYDROCHLORIDE	rxcui:106029	CYCLOPENTOLATE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1182605208011137	IPRATROPIUM BROMIDE	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.8899605294185507	ENALAPRILAT	rxcui:1545989	ENALAPRILAT ANHYDROUS	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	0.5933070196123671	RAMIPRIL	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	0.2019525816757481	METHAZOLAMIDE	rxcui:6826	METHAZOLAMIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2822993077187876	FEXOFENADINE HYDROCHLORIDE	rxcui:236474	FEXOFENADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	0.6177373086552295	EPOETIN ALFA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2792961235941196	MEPENZOLATE BROMIDE	rxcui:52560	MEPENZOLATE BROMIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2031244535229961	DICYCLOMINE HYDROCHLORIDE	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.596678082	BISOPROLOL FUMARATE	rxcui:142146	BISOPROLOL FUMARATE	TRUE	FALSE	FALSE
SLC12A1	hgnc:10910	SLC12A1	ChEMBL	33	inhibitor	0.8334550989792778	FUROSEMIDE	rxcui:4603	FUROSEMIDE	TRUE	FALSE	FALSE
MPL	hgnc:7217	MPL	ChEMBL	33	agonist	2.983390411119005	ROMIPLOSTIM	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
FKBP1A	hgnc:3711	FKBP1A	ChEMBL	33	inhibitor	0.4688184931758437	TACROLIMUS	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2983390411119005	CITALOPRAM HYDROBROMIDE	rxcui:221078	CITALOPRAM HYDROBROMIDE	TRUE	FALSE	FALSE
AVPR1B	hgnc:896	AVPR1B	ChEMBL	33	agonist	1.250182648468916	VASOPRESSIN TANNATE	chembl:CHEMBL1201528	VASOPRESSIN TANNATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	ChEMBL	33	agonist	0.1672218829162245	DOXERCALCIFEROL	rxcui:11516	DOXERCALCIFEROL	TRUE	FALSE	FALSE
GHR	hgnc:4263	GHR	ChEMBL	33	agonist	1.400204566285186	SOMATROPIN	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN SUSP PROTAMINE ZINC PURIFIED BEEF	chembl:CHEMBL1201541	INSULIN SUSP PROTAMINE ZINC PURIFIED BEEF	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.2453629496995069	AMPHETAMINE ASPARTATE	rxcui:221057	AMPHETAMINE ASPARTATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.2453629496995069	MILNACIPRAN HYDROCHLORIDE	rxcui:30003	MILNACIPRAN HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.4907258993990139	GUANETHIDINE MONOSULFATE	rxcui:82023	GUANETHIDINE MONOSULFATE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.272767123	CABOZANTINIB S-MALATE	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	ChEMBL	33	inhibitor	0.057073556	BOSUTINIB	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	agonist	0.305277158	PALIFERMIN	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.9001315068976199	MIRABEGRON	rxcui:1300786	MIRABEGRON	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.8607814956671229	ETHYNODIOL DIACETATE	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	0.3170753093942904	NICOTINE	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	1.790034246671403	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.096167896	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.1848861663228679	CODEINE POLISTIREX	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	CODEINE SULFATE	rxcui:91104	CODEINE SULFATE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.07614901	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.086818239	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.025304902	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	ChEMBL	33	inhibitor	0.3804903712731485	LITHIUM CITRATE	rxcui:52105	LITHIUM CITRATE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.046881849	ISOPROTERENOL HYDROCHLORIDE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.4375639269641209	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.033338204	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.014708031	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.6105543166941221	METHYLDOPATE HYDROCHLORIDE	rxcui:91241	METHYLDOPATE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.2465148884304905	METHYLDOPATE HYDROCHLORIDE	rxcui:91241	METHYLDOPATE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.364636606	CAFFEINE, CITRATED	rxcui:20033	CAFFEINE CITRATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.046881849	PHENYLBUTAZONE	rxcui:8160	PHENYLBUTAZONE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.038049037	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.036977233	OXYMETAZOLINE HYDROCHLORIDE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.1408971500063358	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.084553416	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.2324817828272369	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
RRM2	hgnc:10452	RRM2	ChEMBL	33	inhibitor	0.130291988	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	agonist	0.029235897	METHYLTESTOSTERONE	rxcui:6904	METHYLTESTOSTERONE	TRUE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAXIMIN	rxcui:35619	RIFAXIMIN	TRUE	FALSE	FALSE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAXIMIN	rxcui:35619	RIFAXIMIN	TRUE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAXIMIN	rxcui:35619	RIFAXIMIN	TRUE	FALSE	FALSE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAXIMIN	rxcui:35619	RIFAXIMIN	TRUE	FALSE	FALSE
CHRND	hgnc:1965	CHRND	ChEMBL	33	agonist	0.7501095890813501	DECAMETHONIUM BROMIDE	ncit:C65365	DECAMETHONIUM BROMIDE	TRUE	FALSE	FALSE
GLUCLX	NULL	NULL	ChEMBL	33	modulator	NULL	IVERMECTIN	rxcui:6069	IVERMECTIN	TRUE	FALSE	FALSE
PDE7A	hgnc:8791	PDE7A	ChEMBL	33	inhibitor	0.300043836	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE6H	hgnc:8790	PDE6H	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.1022876712383659	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.1000146118775133	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.091796628	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.055839424	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.016126435	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.091583148	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.034318739	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.1252170220247087	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.039097298	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.1018248310970158	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.1600843635234588	ZALEPLON	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHRADINE	rxcui:2239	CEPHRADINE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.801643836	REL-BENDIGOLE E	chembl:CHEMBL1915270	CHEMBL:CHEMBL1915270	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMENOXIME HYDROCHLORIDE	ncit:C65296	CEFMENOXIME HYDROCHLORIDE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMENOXIME HYDROCHLORIDE	ncit:C65296	CEFMENOXIME HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMENOXIME HYDROCHLORIDE	ncit:C65296	CEFMENOXIME HYDROCHLORIDE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMENOXIME HYDROCHLORIDE	ncit:C65296	CEFMENOXIME HYDROCHLORIDE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMENOXIME HYDROCHLORIDE	ncit:C65296	CEFMENOXIME HYDROCHLORIDE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMENOXIME HYDROCHLORIDE	ncit:C65296	CEFMENOXIME HYDROCHLORIDE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFMENOXIME HYDROCHLORIDE	ncit:C65296	CEFMENOXIME HYDROCHLORIDE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTETAN DISODIUM	rxcui:203141	CEFOTETAN DISODIUM	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFIXIME	rxcui:1546021	CEFIXIME ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	PENICILLIN G POTASSIUM	rxcui:203133	PENICILLIN G POTASSIUM	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.00899104	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	4-METHYL-[1,10]PHENANTHROLINE	chembl:CHEMBL316589	CHEMBL:CHEMBL316589	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	ML-10302	iuphar.ligand:235	ML 10302	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.017608206	WIN-552122	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	S-NITROSOGLUTATHIONE	drugbank:DB17877	S-NITROSOGLUTATHIONE	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
TSSK2	hgnc:11401	TSSK2	DTC	9/2/20	NULL	0.088996053	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002796829	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	6-METHOXY-HARMALAN	chembl:CHEMBL338115	CHEMBL:CHEMBL338115	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.00753879	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	NSC-645827	chembl:CHEMBL95704	CHEMBL:CHEMBL95704	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.106290832	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
AKT1S1	hgnc:28426	AKT1S1	DTC	9/2/20	NULL	0.9376369863516874	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	4-METHYL-[1,10]PHENANTHROLINE	chembl:CHEMBL316589	CHEMBL:CHEMBL316589	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.4102161815288632	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	MMV396678	chembl:CHEMBL1459149	CHEMBL:CHEMBL1459149	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.089298761	BROMOCRIPTINE MESYLATE	rxcui:142426	BROMOCRIPTINE MESYLATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.003894361	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	PROPACHLOR	chembl:CHEMBL1394829	PROPACHLOR	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.093763699	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.1136529680426287	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.021189536	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.596678082	DNDI1395216	chembl:CHEMBL522887	CHEMBL:CHEMBL522887	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.018540844	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	TCMDC-125310	chembl:CHEMBL582030	CHEMBL:CHEMBL582030	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.008353113	PROPACHLOR	chembl:CHEMBL1394829	PROPACHLOR	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
POLD1	hgnc:9175	POLD1	ChEMBL	33	inhibitor	0.047049885	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
POLD4	hgnc:14106	POLD4	ChEMBL	33	inhibitor	0.094099769	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
POLD2	hgnc:9176	POLD2	ChEMBL	33	inhibitor	0.094099769	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CACNA1S	hgnc:1397	CACNA1S	ChEMBL	33	modulator	0.038104261	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNB1	hgnc:1401	CACNB1	ChEMBL	33	modulator	0.1442518440541058	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNG4	hgnc:1408	CACNG4	ChEMBL	33	modulator	0.2243917574174979	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNA2D4	hgnc:20202	CACNA2D4	ChEMBL	33	modulator	0.2019525816757481	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.083744292	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.075768645	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.08334551	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.084689792	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.088996053	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.067839369	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.082171629	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.066297565	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.036337489	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.038467158	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	agonist	0.061055432	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPME2	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPMJ2	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
RPLI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	blocker	0.729273212	PHENSUXIMIDE	rxcui:33309	PHENSUXIMIDE	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.7326651800329465	ETHOSUXIMIDE	rxcui:4135	ETHOSUXIMIDE	TRUE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	modulator	0.3281729452230906	BLINATUMOMAB	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.07631929	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.027524552	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.024238039	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.064944553	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
CDK11B	hgnc:1729	CDK11B	ChEMBL	33	inhibitor	0.1470803115845784	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	1.000146118775133	SAR-125844	drugbank:DB15382	SAR-125844	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1250182648468916	TAK-593	drugbank:DB13093	TAK-593	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	ChEMBL	33	inhibitor	0.546954909	BPI-9016	chembl:CHEMBL3545236	BPI-9016	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.6731752722524935	Y-39983	chembl:CHEMBL571948	Y-39983	FALSE	FALSE	FALSE
ADORA2B	hgnc:264	ADORA2B	ChEMBL	33	inhibitor	1.458546423213736	QAF805	chembl:CHEMBL3545204	QAF805	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.2917092846427472	FK453	iuphar.ligand:5606	FK-453	FALSE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	inhibitor	1.381780822	QAF805	chembl:CHEMBL3545204	QAF805	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	inhibitor	0.5585922471882393	TC-2216	chembl:CHEMBL504652	TC-2216	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	PYROTINIB	ncit:C111895	PYROTINIB	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1223955040459079	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.172722603	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1363835616511545	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1363835616511545	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.3017682254924971	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.061592576	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.1325951293830669	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.1810609352954983	C-1311	chembl:CHEMBL338604	C-1311	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.8140724222588294	CARMOTEROL	ncit:C171749	CARMOTEROL	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	BEDORADRINE SULFATE	ncit:C77933	BEDORADRINE SULFATE	FALSE	FALSE	FALSE
GLP2R	hgnc:4325	GLP2R	ChEMBL	33	agonist	26.25383561784724	ELSIGLUTIDE	ncit:C101131	ELSIGLUTIDE	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	1.280674908	GRC-6211	chembl:CHEMBL3545107	GRC-6211	FALSE	FALSE	FALSE
TACR3	hgnc:11528	TACR3	ChEMBL	33	inhibitor	5.834185692854944	TALNETANT	ncit:C76464	TALNETANT	FALSE	FALSE	FALSE
MAS1	hgnc:6899	MAS1	ChEMBL	33	agonist	17.50255707856483	TXA127	chembl:CHEMBL3545347	TXA127	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	agonist	3.088686543276147	FE 202767	chembl:CHEMBL3545167	FE 202767	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.019676849	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	ChEMBL	33	inhibitor	3.580068493342807	ITRIGLUMIDE	ncit:C65992	ITRIGLUMIDE	FALSE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	agonist	0.3671865121377238	DONITRIPTAN	ncit:C65466	DONITRIPTAN	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.4947116523181093	GILTERITINIB	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	agonist	0.1530835896084387	APIMOSTINEL	ncit:C169785	APIMOSTINEL	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	agonist	0.1209854175937661	RAPASTINEL	ncit:C152156	RAPASTINEL	FALSE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.1530835896084387	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	positive modulator	0.2586584789935689	NEBOGLAMINE	ncit:C66222	NEBOGLAMINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.012695278	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.5147810905460244	RG3487	chembl:CHEMBL2151439	RG3487	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.2792961235941196	SIMPINICLINE	ncit:C179121	SIMPINICLINE	FALSE	FALSE	FALSE
GRIK1	hgnc:4579	GRIK1	ChEMBL	33	inhibitor	3.500511415712966	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
KCNMA1	hgnc:6284	KCNMA1	ChEMBL	33	activator	5.834185692854944	BMS-223131	chembl:CHEMBL222460	BMS-223131	FALSE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	ChEMBL	33	inhibitor	0.2536602475154323	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	inhibitor	0.5303805175322677	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
GRIK5	hgnc:4583	GRIK5	ChEMBL	33	inhibitor	0.5834185692854945	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007003824	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	blocker	0.217423069	CNS-5161	drugbank:DB05824	CNS-5161	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.3763990769583835	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	agonist	0.038159645	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	agonist	0.025439763	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	agonist	0.042073455	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.1595977849109255	BRIVANIB ALANINATE	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1158257453728555	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.024885152	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.039068208	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.151464436	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
HTR6	hgnc:5301	HTR6	ChEMBL	33	inhibitor	3.500511415712966	IDALOPIRDINE	ncit:C166835	IDALOPIRDINE	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.018305561	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	1.250182648468916	VAPREOTIDE	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.03409589	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.8334550989792776	VAPREOTIDE	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
EDNRB	hgnc:3180	EDNRB	ChEMBL	33	inhibitor	1.875273972703375	TEZOSENTAN	ncit:C97358	TEZOSENTAN	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	1.712206670729168	ENCENICLINE	ncit:C166844	ENCENICLINE	FALSE	FALSE	FALSE
ADORA1	hgnc:262	ADORA1	ChEMBL	33	inhibitor	0.8751278539282416	ROLOFYLLINE	ncit:C96195	ROLOFYLLINE	FALSE	FALSE	FALSE
MUC16	hgnc:15582	MUC16	ChEMBL	33	other/unknown	11.25164383622025	ABAGOVOMAB	ncit:C26449	ABAGOVOMAB	FALSE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	ChEMBL	33	inhibitor	19.69037671338543	TABALUMAB	ncit:C91727	TABALUMAB	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	3.000438356	ONARTUZUMAB	ncit:C82348	ONARTUZUMAB	FALSE	TRUE	TRUE
TERT	hgnc:11730	TERT	ChEMBL	33	inhibitor	1.500219178	IMETELSTAT SODIUM	ncit:C84511	IMETELSTAT SODIUM	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	SJ000121029	chembl:CHEMBL591631	CHEMBL:CHEMBL591631	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.4907258993990139	EDIVOXETINE	ncit:C166706	EDIVOXETINE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	inhibitor	1.615620653405984	CRENEZUMAB	ncit:C174789	CRENEZUMAB	FALSE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	ChEMBL	33	agonist	11.66837138570988	DROZITUMAB	ncit:C95784	DROZITUMAB	FALSE	FALSE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.036977233	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
CD248	hgnc:18219	CD248	ChEMBL	33	inhibitor	157.5230137070835	ONTUXIZUMAB	ncit:C82406	ONTUXIZUMAB	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	1.419126249613364	SAFINAMIDE MESYLATE	rxcui:1922449	SAFINAMIDE MESYLATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	CLEMIZOLE	ncit:C81139	CLEMIZOLE	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3281729452230906	ISOXICAM	ncit:C80558	ISOXICAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.039068208	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.040021091	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFADIMETHOXINE SODIUM	rxcui:1306121	SULFADIMETHOXINE SODIUM	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
AOC1	hgnc:80	AOC1	ChEMBL	33	activator	0.596678082	PROXIBARBAL	rxcui:83885	PROXIBARBAL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	PH-011685	chembl:CHEMBL126804	CHEMBL:CHEMBL126804	FALSE	FALSE	FALSE
CD22	hgnc:1643	CD22	ChEMBL	33	inhibitor	2.917092846427472	YTTRIUM Y 90 EPRATUZUMAB TETRAXETAN	chembl:CHEMBL2108666	YTTRIUM Y 90 EPRATUZUMAB TETRAXETAN	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	SUPTAVUMAB	ncit:C152476	SUPTAVUMAB	FALSE	FALSE	FALSE
CSNK1E	hgnc:2453	CSNK1E	DTC	9/2/20	inhibitor	5.250767124	HTS-466284	drugbank:DB03921	4-(3-PYRIDIN-2-YL-1H-PYRAZOL-4-YL)QUINOLINE	FALSE	FALSE	FALSE
TSLP	hgnc:30743	TSLP	ChEMBL	33	inhibitor	26.25383561784724	AMG-157	chembl:CHEMBL2109595	AMG-157	FALSE	FALSE	FALSE
CD27	hgnc:11922	CD27	ChEMBL	33	agonist	15.00219178	VARLILUMAB	ncit:C99127	VARLILUMAB	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIBRENTASVIR	rxcui:1940636	PIBRENTASVIR	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	VOXILAPREVIR	rxcui:1939323	VOXILAPREVIR	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	modulator	0.9723642821424906	FBT-A05	chembl:CHEMBL2109351	FBT-A05	FALSE	FALSE	FALSE
G	NULL	NULL	ChEMBL	33	inhibitor	NULL	RAFIVIRUMAB	ncit:C95793	RAFIVIRUMAB	FALSE	FALSE	FALSE
G	NULL	NULL	ChEMBL	33	inhibitor	NULL	FORAVIRUMAB	ncit:C95786	FORAVIRUMAB	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.080103236	NIMODIPINE	rxcui:7426	NIMODIPINE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.6482428547616604	OPHIOBOLIN O	chembl:CHEMBL1934283	OPHIOBOLIN O	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
CALCA	hgnc:1437	CALCA	ChEMBL	33	inhibitor	0.4861821410712453	FREMANEZUMAB	rxcui:2056691	FREMANEZUMAB	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	ChEMBL	33	inhibitor	0.4688184931758437	EMAPALUMAB	rxcui:2104603	EMAPALUMAB-LZSG	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
POU2F2	hgnc:9213	POU2F2	DTC	9/2/20	NULL	35.00511415712966	LINAGLIPTIN	rxcui:1100699	LINAGLIPTIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.546954909	DANOPREVIR	ncit:C171872	DANOPREVIR	FALSE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.1367387271762877	VANIPREVIR	ncit:C152828	VANIPREVIR	FALSE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CO-TRIMOXAZOLE	chembl:CHEMBL195591	CO-TRIMOXAZOLE	FALSE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CO-TRIMOXAZOLE	chembl:CHEMBL195591	CO-TRIMOXAZOLE	FALSE	FALSE	FALSE
SEM1	hgnc:10845	SEM1	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
SPHK2	hgnc:18859	SPHK2	ChEMBL	33	inhibitor	6.563458904461812	ABC-294640	iuphar.ligand:6624	OPAGANIB	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	FAROPENEM	ncit:C65621	FAROPENEM MEDOXOMIL	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.2381300282797936	TENALISIB	ncit:C113433	TENALISIB	FALSE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	ChEMBL	33	binder	0.024008995	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
AGER	hgnc:320	AGER	ChEMBL	33	inhibitor	5.250767123569449	AZELIRAGON	ncit:C174675	AZELIRAGON	FALSE	FALSE	FALSE
RPS7	hgnc:10440	RPS7	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL30	hgnc:10333	RPL30	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPS28	hgnc:10418	RPS28	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPS23	hgnc:10410	RPS23	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL41	hgnc:10354	RPL41	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
CX3CL1	hgnc:10647	CX3CL1	ChEMBL	33	inhibitor	17.50255707856483	QUETMOLIMAB	ncit:C170361	QUETMOLIMAB	FALSE	FALSE	FALSE
RPLP0	hgnc:10371	RPLP0	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL37	hgnc:10347	RPL37	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLESROVIMAB	ncit:C186415	CLESROVIMAB	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.596678082	HT-0712	drugbank:DB11650	HT-0712	FALSE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	1.458546423213736	DARIDOREXANT	rxcui:2591497	DARIDOREXANT	TRUE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	4.773424657790408	SELTOREXANT	ncit:C152326	SELTOREXANT	FALSE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPODOXIME	rxcui:20489	CEFPODOXIME	TRUE	FALSE	FALSE
NS5A	NULL	NULL	ChEMBL	33	inhibitor	NULL	RUZASVIR	ncit:C152277	RUZASVIR	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.033487035	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.038894571	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.042174836	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
POLE2	hgnc:9178	POLE2	ChEMBL	33	inhibitor	0.7955707762984016	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	GS-9256	drugbank:DB12876	GS-9256	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELEOBUVIR	ncit:C166826	DELEOBUVIR	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.1383601350084176	TIAPRIDE	rxcui:10588	TIAPRIDE	FALSE	FALSE	FALSE
PDE9A	hgnc:8795	PDE9A	ChEMBL	33	inhibitor	6.563458904461812	TOVINONTRINE	ncit:C174928	TOVINONTRINE	FALSE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	ChEMBL	33	inhibitor	3.281729452230906	SELATOGREL	ncit:C166930	SELATOGREL	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.4375639269641208	CAMPTOTHECIN-20-O-PROPIONATE	chembl:CHEMBL124162	CAMPTOTHECIN-20-O-PROPIONATE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	ChEMBL	33	modulator	0.4636438961209227	EPRENETAPOPT	ncit:C85465	EPRENETAPOPT	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	agonist	0.042073455	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	agonist	0.036062961	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	SISUNATOVIR	ncit:C170818	SISUNATOVIR	FALSE	FALSE	FALSE
TNFRSF18	hgnc:11914	TNFRSF18	ChEMBL	33	agonist	13.12691780892362	RAGIFILIMAB	ncit:C126643	RAGIFILIMAB	FALSE	FALSE	FALSE
C1S	hgnc:1247	C1S	ChEMBL	33	inhibitor	10.50153424713889	SUTIMLIMAB	rxcui:2591404	SUTIMLIMAB	TRUE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	ChEMBL	33	inhibitor	0.2333674277141977	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
C3	hgnc:1318	C3	ChEMBL	33	inhibitor	2.917092846427472	PEGCETACOPLAN	rxcui:2557372	PEGCETACOPLAN	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	ChEMBL	33	inhibitor	0.3621218705909965	ONALESPIB	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
HSP90AB1	hgnc:5258	HSP90AB1	ChEMBL	33	inhibitor	0.5707355569097228	ONALESPIB	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
REVERSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	APRICITABINE	ncit:C79871	APRICITABINE	FALSE	FALSE	FALSE
TRANSCRIPTASE	NULL	NULL	ChEMBL	33	inhibitor	NULL	APRICITABINE	ncit:C79871	APRICITABINE	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVAROFLOXACIN	ncit:C171788	ACORAFLOXACIN	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVAROFLOXACIN	ncit:C171788	ACORAFLOXACIN	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	AVAROFLOXACIN	ncit:C171788	ACORAFLOXACIN	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1988926940746003	CENTANAFADINE	ncit:C171666	CENTANAFADINE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	0.4565884455277782	PLB1003	chembl:CHEMBL4650298	PLB1003	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	ChEMBL	33	inhibitor	0.2187819634820604	NINGETINIB	drugbank:DB16256	NINGETINIB	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	CABOTEGRAVIR SODIUM	rxcui:2475076	CABOTEGRAVIR SODIUM	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
TGFBR1	hgnc:11772	TGFBR1	ChEMBL	33	inhibitor	5.000730593875666	VACTOSERTIB	ncit:C116357	VACTOSERTIB	FALSE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	ChEMBL	33	inhibitor	5.834185692854944	DAPANSUTRILE	ncit:C166608	DAPANSUTRILE	FALSE	FALSE	FALSE
GMPS	hgnc:4378	GMPS	ChEMBL	33	inhibitor	13.12691780892362	MIZORIBINE	ncit:C66172	MIZORIBINE	FALSE	FALSE	FALSE
POLR2A	hgnc:9187	POLR2A	ChEMBL	33	inhibitor	5.834185692854944	TAS-106	drugbank:DB06656	TAS-106	FALSE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	4.773424657790408	PRADEFOVIR MESYLATE	ncit:C66454	PRADEFOVIR MESYLATE	FALSE	FALSE	FALSE
SV2C	hgnc:30670	SV2C	ChEMBL	33	modulator	2.763561643983921	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	ETESEVIMAB	rxcui:2477854	ETESEVIMAB	TRUE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	ChEMBL	33	inhibitor	7.501095891	SEVITERONEL	ncit:C113652	SEVITERONEL	FALSE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	ChEMBL	33	inhibitor	5.527123287967842	EMVODODSTAT	ncit:C91100	EMVODODSTAT	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMUBARVIMAB	ncit:C175227	AMUBARVIMAB	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	ENSOVIBEP	ncit:C179065	ENSOVIBEP	FALSE	FALSE	FALSE
CYP11B1	hgnc:2591	CYP11B1	ChEMBL	33	inhibitor	1.750255707856483	LEVOKETOCONAZOLE	rxcui:2588846	LEVOKETOCONAZOLE	TRUE	FALSE	FALSE
PDCD1	hgnc:8760	PDCD1	ChEMBL	33	inhibitor	1.280674908	FINOTONLIMAB	ncit:C170758	FINOTONLIMAB	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	activator	0.3723948314588262	ALDAFERMIN	ncit:C169769	ALDAFERMIN	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	NESBUVIR	ncit:C76498	NESBUVIR	FALSE	FALSE	FALSE
EDNRA	hgnc:3179	EDNRA	ChEMBL	33	inhibitor	4.565884455277782	BQ-123	drugbank:DB12054	BQ-123	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	ChEMBL	33	inhibitor	0.066297565	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
TNNT3	hgnc:11950	TNNT3	ChEMBL	33	activator	8.751278539282415	RELDESEMTIV	ncit:C166781	RELDESEMTIV	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	modulator	0.2004109589148645	VELSECORAT	ncit:C171915	VELSECORAT	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.2639729920045843	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	0.6177373086552294	COSIBELIMAB	ncit:C151947	COSIBELIMAB	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.3454452054979901	ZANIDATAMAB	ncit:C130010	ZANIDATAMAB	FALSE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	2.917092846427472	PALTUSOTINE	ncit:C175836	PALTUSOTINE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	ChEMBL	33	vaccine	1.400204566285186	PEXASTIMOGENE DEVACIREPVEC	ncit:C71533	PEXASTIMOGENE DEVACIREPVEC	FALSE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	ChEMBL	33	inhibitor	1.500219178	LEVOKETOCONAZOLE	rxcui:2588846	LEVOKETOCONAZOLE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.04593847	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.078761507	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	PYRAZINOIC ACID	chembl:CHEMBL613	PYRAZINOIC ACID	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.8899605294185507	TRV-120027	drugbank:DB12199	TRV-120027	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	ChEMBL	33	inhibitor	0.6731752722524935	REBIMASTAT	ncit:C1875	REBIMASTAT	FALSE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	2.386712328895204	DARIDOREXANT HYDROCHLORIDE	rxcui:2591496	DARIDOREXANT HYDROCHLORIDE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	ChEMBL	33	inhibitor	1.029562181092049	ACALABRUTINIB MALEATE	ncit:C174678	ACALABRUTINIB MALEATE	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	1.458546423213736	ENSIFENTRINE	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
TUB2	NULL	NULL	ChEMBL	33	binder	NULL	FENBENDAZOLE	rxcui:4325	FENBENDAZOLE	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.082754407	BMN673	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1101693521639275	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
RRM1	hgnc:10451	RRM1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2324817828272369	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.030945115	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
FLK1	hgnc:6307	KDR	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.018305561	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
RRM1	hgnc:10451	RRM1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2324817828272369	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
RRM2	hgnc:10452	RRM2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.130291988	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	COSMIC	4-Sep-20	NULL	2.212697851403848	Crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.006945459	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.014832675	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.050007306	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DANTHRON	rxcui:22293	DANTHRON	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.014832675	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.210030685	SJ000173328	chembl:CHEMBL591613	CHEMBL:CHEMBL591613	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.050246575	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.03110644	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(+)-7,9-DEOXYTHYSANONE	chembl:CHEMBL607534	CHEMBL:CHEMBL607534	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	CALPHOSTIN C	iuphar.ligand:5156	CALPHOSTIN C	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007330402	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	0.1620607136904151	MOMETASONE FUROATE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.037586021	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.024605282	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PTPN7	hgnc:9659	PTPN7	DTC	9/2/20	NULL	0.9546849315580819	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.267214612	ALISOL A-23 ACETATE	chembl:CHEMBL2059711	CHEMBL:CHEMBL2059711	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.046881849	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.015335184	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	DIHYDROERGOTAMINE MESYLATE	rxcui:203176	DIHYDROERGOTAMINE MESYLATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	MRS-2220	iuphar.ligand:6496	MRS 2219	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.022353202	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.3889457128569962	TRIMEPRAZINE TARTRATE	rxcui:164308	TRIMEPRAZINE TARTRATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SULFAPYRIDINE	rxcui:10188	SULFAPYRIDINE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.059297201	DIHYDREXIDINE	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	0.2692701089009974	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMA1	hgnc:9530	PSMA1	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD13	hgnc:9558	PSMD13	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD11	hgnc:9556	PSMD11	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD7	hgnc:9565	PSMD7	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD3	hgnc:9560	PSMD3	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	NOVIFLUMURON	chembl:CHEMBL1873307	NOVIFLUMURON	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	1R,9S-HYDRASTINE	chembl:CHEMBL475536	1R,9S-HYDRASTINE	FALSE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1446492320542548	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	0.1215455352678113	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.2470949234620917	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	0.2160809515872201	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.1054370908347279	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.1591141552596802	DNDI1416934	chembl:CHEMBL1989750	CHEMBL:CHEMBL1989750	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.4167275494896388	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003483789	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.013673873	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.047734247	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.024605282	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.082043236	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	MEPAZINE ACETATE	chembl:CHEMBL1712842	MEPAZINE ACETATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.1283806142682017	CENTAUREIDIN	chembl:CHEMBL77552	CENTAUREIDIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ALPHA-TERTHIENYL	chembl:CHEMBL90017	ALPHA-TERTHIENYL	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.046303061	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	2-HYDROXYESTRADIOL	ncit:C120474	2-HYDROXYESTRADIOL	FALSE	FALSE	FALSE
PHKG2	hgnc:8931	PHKG2	DTC	9/2/20	NULL	0.049210563	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.150021918	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.089756703	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	1.666910197958555	NSC-127133	chembl:CHEMBL1172911	CHEMBL:CHEMBL1172911	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.039688338	ARUNDINE	chembl:CHEMBL446452	ARUNDINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	NSC-74859	chembl:CHEMBL477936	CHEMBL:CHEMBL477936	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-124570	chembl:CHEMBL546475	CHEMBL:CHEMBL546475	FALSE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	DTC	9/2/20	NULL	0.2430910705356226	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	CL-976	chembl:CHEMBL22373	CL-976	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	GF-109203	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.095122593	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008916229	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	VALNEMULIN	rxcui:2604036	VALNEMULIN	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.024238039	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.06697407	GNF-PF-5061	chembl:CHEMBL601385	CHEMBL:CHEMBL601385	FALSE	FALSE	FALSE
MMP3	hgnc:7173	MMP3	DTC	9/2/20	NULL	3.750547945	BERKELEYACETAL A	chembl:CHEMBL252920	BERKELEYACETAL A	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.304834086	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.040515178	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	DEOXIEPINEPHRINE	chembl:CHEMBL31088	DEOXIEPINEPHRINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	IMAZODAN	ncit:C83787	IMAZODAN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	SORBIC ACID	rxcui:1311139	SORBIC ACID	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	GNF-PF-372	chembl:CHEMBL580155	CHEMBL:CHEMBL580155	FALSE	FALSE	FALSE
SLC6A1	hgnc:11042	SLC6A1	DTC	9/2/20	NULL	7.001022831425932	HINOKININ	chembl:CHEMBL242011	HINOKININ	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	CHRYSENE	chembl:CHEMBL85685	CHRYSENE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	CONICASTEROL D	chembl:CHEMBL1782605	CONICASTEROL D	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.059667808	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.00453826	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ALPHA-PHELLANDRENE	chembl:CHEMBL455041	ALPHA-PHELLANDRENE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.1202465753489187	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	(+)-EPITAXIFOLIN	chembl:CHEMBL9249	(+)-EPITAXIFOLIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.057073556	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.056399217	PROPACHLOR	chembl:CHEMBL1394829	PROPACHLOR	FALSE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.031784305	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.019447286	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.035098711	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.030004384	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.6364566210387212	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	MEBEVERINE HYDROCHLORIDE	rxcui:235827	MEBEVERINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	3,3'-DIMETHOXYBENZIDINE	chembl:CHEMBL398363	CHEMBL:CHEMBL398363	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-4853	chembl:CHEMBL599957	CHEMBL:CHEMBL599957	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.3889457128569963	GW559768X	chembl:CHEMBL237347	GW559768X	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.093763699	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.016352436	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00410569	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.061412481	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1411496538593938	CID 2056784	chembl:CHEMBL261123	CHEMBL:CHEMBL261123	FALSE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.4039051633514962	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	URACIL MUSTARD	rxcui:10996	URACIL MUSTARD	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	HYDROXYFLUTAMIDE	ncit:C63948	HYDROXYFLUTAMIDE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.03151721	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
SENP1	hgnc:17927	SENP1	DTC	9/2/20	NULL	17.50255707856483	ORG-41841	chembl:CHEMBL211405	CHEMBL:CHEMBL211405	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.077789143	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.036237178	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	HYDROCORTISONE 21-OCTANOATE	chembl:CHEMBL253989	CHEMBL:CHEMBL253989	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TRIAMCINOLONE DIACETATE	rxcui:10762	TRIAMCINOLONE DIACETATE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	ACETYLSEROTONIN	iuphar.ligand:5451	N-ACETYLSEROTONIN	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.066047385	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	NSC-209931	chembl:CHEMBL472656	CHEMBL:CHEMBL472656	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	IBUDILAST	ncit:C65876	IBUDILAST	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	TCMDC-125110	chembl:CHEMBL580816	CHEMBL:CHEMBL580816	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.001711742	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.091159151	DNDI1417597	chembl:CHEMBL1330352	CHEMBL:CHEMBL1330352	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.08854582	8-PHENYL THEOPHYLLINE	chembl:CHEMBL62350	8-PHENYL THEOPHYLLINE	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	DESIPRAMINE HYDROCHLORIDE	rxcui:203174	DESIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.021240967	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.018719312	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
MPI	hgnc:7216	MPI	DTC	9/2/20	NULL	0.4339476961627644	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.015892152	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.025123288	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.006397133	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	2.838252499226729	APREPITANT	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008916229	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	DTC	9/2/20	NULL	0.473042083	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.022099188	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003147942	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SULINDAC SULFOXIDE	chembl:CHEMBL1376	SULINDAC SULFOXIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TRIFORINE	chembl:CHEMBL453418	TRIFORINE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.078958904	DIHYDREXIDINE	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
BRD4	hgnc:13575	BRD4	DTC	9/2/20	NULL	0.167488584	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	DEXTROMEPROMAZINE	chembl:CHEMBL1323355	DEXTROMEPROMAZINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.064347636	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	DNDI1416924	chembl:CHEMBL156959	CHEMBL:CHEMBL156959	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	PROTOCATECHUALDEHYDE	rxcui:1362689	PROTOCATECHUALDEHYDE	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.042242696	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TRITON X	chembl:CHEMBL39763	TRITON X	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.3977853881492007	FURAFYLLINE	ncit:C65779	FURAFYLLINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	ISOEUGENITOL	chembl:CHEMBL1371435	ISOEUGENITOL	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	PROTOCATECHUALDEHYDE	rxcui:1362689	PROTOCATECHUALDEHYDE	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.027781837	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	3,6-DIPHENYL-[1,2,4,5]TETRAZINE	chembl:CHEMBL17784	CHEMBL:CHEMBL17784	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	L-765314	iuphar.ligand:506	L-765314	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	GNF-PF-3537	chembl:CHEMBL601110	CHEMBL:CHEMBL601110	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.082043236	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	6-METHOXY-HARMALAN	chembl:CHEMBL338115	CHEMBL:CHEMBL338115	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124183	chembl:CHEMBL534319	CHEMBL:CHEMBL534319	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.020591244	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.3580068493342807	DEXIBUPROFEN	ncit:C166907	DEXIBUPROFEN	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.003458092	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.070860555	DNDI1417692	chembl:CHEMBL1481509	CHEMBL:CHEMBL1481509	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.041344623	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.016116535	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.060008767	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.2083637747448194	DNDI1417195	chembl:CHEMBL1303948	CHEMBL:CHEMBL1303948	FALSE	FALSE	FALSE
CTDSP1	hgnc:21614	CTDSP1	DTC	9/2/20	NULL	0.1535312024435511	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002088278	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.046673486	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.085796848	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.003712364	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.046881849	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005867434	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	NONIVAMIDE	rxcui:31945	NONIVAMIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	BUFLOMEDIL	rxcui:19836	BUFLOMEDIL	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.050978322	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006356861	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	0.046881849	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.017775109	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.045579576	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
ABCB11	hgnc:42	ABCB11	DTC	9/2/20	NULL	0.9546849315580819	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.014299475	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.1164249916534246	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.075010959	MUNDULONE	chembl:CHEMBL465339	MUNDULONE	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.2187819634820604	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.01555322	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.01795748	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	DTC	9/2/20	NULL	0.5385402178019949	DEMETHYLWEDELOLACTONE	chembl:CHEMBL2089002	DEMETHYLWEDELOLACTONE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
GPBAR1	hgnc:19680	GPBAR1	DTC	9/2/20	NULL	2.625383561784724	CHENODIOL	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1025540453822158	DNDI1417597	chembl:CHEMBL1330352	CHEMBL:CHEMBL1330352	FALSE	FALSE	FALSE
PTPN22	hgnc:9652	PTPN22	DTC	9/2/20	NULL	1.050153425	GNF-PF-3542	chembl:CHEMBL598477	CHEMBL:CHEMBL598477	FALSE	FALSE	FALSE
DHRS9	hgnc:16888	DHRS9	DTC	9/2/20	NULL	15.00219178	(+/-)-WIEDENDIOL B	chembl:CHEMBL456619	(+/-)-WIEDENDIOL B	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.049442252	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.039068208	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.046881849	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.043466615	KETOROLAC TROMETHAMINE	rxcui:28200	KETOROLAC TROMETHAMINE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.018106094	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.060492709	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	VU001171	iuphar.ligand:6228	VU0001171	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.007012242	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.018540844	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.049349315	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.025489161	FENOLDOPAM MESYLATE	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.099446347	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.09003373	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.031822831	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.038187397	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003829323	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
CAMKK2	hgnc:1470	CAMKK2	DTC	9/2/20	NULL	0.1909369863116163	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00051291	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005166044	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.072927321	CID 5310655	chembl:CHEMBL408563	CHEMBL:CHEMBL408563	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	SJ000032153	chembl:CHEMBL600862	CHEMBL:CHEMBL600862	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.3281729452230906	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.017799211	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
SLCO1B3	hgnc:10961	SLCO1B3	DTC	9/2/20	NULL	1.400204566285186	MK-8245	drugbank:DB13024	MK-8245	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PENTACHLORONITROBENZENE	chembl:CHEMBL468759	PENTACHLORONITROBENZENE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.041085815	FAGARONINE	chembl:CHEMBL282622	FAGARONINE	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.1100789753368857	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	FLUOROSALAN	ncit:C82318	FLUOROSALAN	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.024309107	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.020226376	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.1250182648468916	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	2.282942227638891	DAUCOSTEROL	chembl:CHEMBL506678	SITOGLUSIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	ORTHO-METHOXYCINNAMALDEHYDE	chembl:CHEMBL83159	CHEMBL:CHEMBL83159	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	GNF-PF-3515	iuphar.ligand:4203	GMQ	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.013320059	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.036718651	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	DTC	9/2/20	NULL	0.212152207	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TROLOX	chembl:CHEMBL153	TROLOX	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2447910080918158	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
CD1D	hgnc:1637	CD1D	DTC	9/2/20	NULL	157.5230137070835	KRN-7000	drugbank:DB12232	KRN-7000	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	BUTANAL	chembl:CHEMBL1478334	BUTANAL	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	(-)-PLAKILACTONE C	chembl:CHEMBL2178586	CHEMBL:CHEMBL2178586	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.138178082	FURAFYLLINE	ncit:C65779	FURAFYLLINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	GNF-PF-2686	chembl:CHEMBL578276	CHEMBL:CHEMBL578276	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1426838892274307	PHENFORMIN HYDROCHLORIDE	rxcui:235288	PHENFORMIN HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	RIMCAZOLE	ncit:C152218	RIMCAZOLE	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.105015342	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006691433	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	NSC-117199	chembl:CHEMBL502257	CHEMBL:CHEMBL502257	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.024513385	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.045579576	MOLINDONE	rxcui:7019	MOLINDONE	TRUE	FALSE	FALSE
NCSTN	hgnc:17091	NCSTN	DTC	9/2/20	NULL	1.790034246671403	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.02832129	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	PIFITHRIN-ALPHA	chembl:CHEMBL198759	CHEMBL:CHEMBL198759	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1651184630053286	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00626658	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.020257589	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	GNF-PF-4590	chembl:CHEMBL529361	CHEMBL:CHEMBL529361	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	GEDUNIN	chembl:CHEMBL465226	GEDUNIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-123747	chembl:CHEMBL530698	CHEMBL:CHEMBL530698	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	CARMOFUR	ncit:C955	CARMOFUR	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.069824031	CANTHARIDIC_ACID	chembl:CHEMBL275516	CANTHARIDIC_ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	1.193356164447602	RO-5068760	chembl:CHEMBL1956073	CHEMBL:CHEMBL1956073	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.2206204673768676	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	POTASSIUM DICHROMATE	rxcui:8595	POTASSIUM DICHROMATE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00236553	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1693795846312726	METHANANDAMIDE	iuphar.ligand:2506	R-(+)-METHANANDAMIDE	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	DTC	9/2/20	NULL	0.4234489615781814	CEFOXITIN	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	GNF-PF-130	chembl:CHEMBL578890	CHEMBL:CHEMBL578890	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006077277	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	BUFEXAMAC	rxcui:1796	BUFEXAMAC	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.091159151	4-HYDROXYESTRADIOL	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.1250182648468916	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.038187397	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	DEXIBUPROFEN	ncit:C166907	DEXIBUPROFEN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	RESOKAEMPFEROL	chembl:CHEMBL242383	RESOKAEMPFEROL	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.027276712	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.1356787370431382	CLENBUTEROL HYDROCHLORIDE	rxcui:235955	CLENBUTEROL HYDROCHLORIDE	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	DTC	9/2/20	NULL	0.1296485709523321	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	4'-EPICHAETOVIRIDIN A	chembl:CHEMBL1306556	CHEMBL:CHEMBL1306556	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	GNF-PF-2298	chembl:CHEMBL578905	CHEMBL:CHEMBL578905	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.093098708	RAFOXANIDE	ncit:C152146	RAFOXANIDE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	ABAMECTIN	ncit:C95196	ABAMECTIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ALCLOMETASONE DIPROPIONATE	rxcui:108088	ALCLOMETASONE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2187819634820604	DESMETHOXYYANGONIN	chembl:CHEMBL254218	DESMETHOXYYANGONIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	ARTEMISIN	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.1060761035064535	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	7-HYDROXYFLAVONE	chembl:CHEMBL276915	7-HYDROXYFLAVONE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.075442056	AVOBENZONE	rxcui:45045	AVOBENZONE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	chembl:CHEMBL1322879	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.009270422	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.4023576339899961	PINOPHILIN A	chembl:CHEMBL2011646	PINOPHILIN A	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.011279843	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	RAFOXANIDE	ncit:C152146	RAFOXANIDE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.067059606	ROBINETIN	chembl:CHEMBL170405	ROBINETIN	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.061412481	PROCARBAZINE	rxcui:8702	PROCARBAZINE	TRUE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1290114772375786	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.00937637	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GNF-PF-3515	iuphar.ligand:4203	GMQ	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.011710007	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.062509132	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	RIMCAZOLE	ncit:C152218	RIMCAZOLE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.091159151	BENZAMIL	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.085239726	BENZAMIL	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.056826484	SB-224289	iuphar.ligand:130	SB 224289	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.012087401	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	PROPARGITE	chembl:CHEMBL1416084	PROPARGITE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.012020987	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012763168	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.015892152	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.03292017	CGS-15943	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	ENDOSULFAN	chembl:CHEMBL194399	ENDOSULFAN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.047518255	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	DEXTROMEPROMAZINE	chembl:CHEMBL1323355	DEXTROMEPROMAZINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007831122	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	1.458546423213736	GNF-PF-4759	chembl:CHEMBL585265	CHEMBL:CHEMBL585265	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.014630168	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.023274677	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.004237907	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	1.750255707856483	HISPIDULIN	drugbank:DB14008	HISPIDULIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.003740928	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.009756163	MORPHINE	rxcui:32926	PAREGORIC	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.2983390411119005	SJ000279525	chembl:CHEMBL600841	CHEMBL:CHEMBL600841	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	GNF-PF-628	chembl:CHEMBL1448140	CHEMBL:CHEMBL1448140	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW829055X	chembl:CHEMBL189148	GW829055X	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	THIOSEMICARBAZIDE	chembl:CHEMBL256250	THIOSEMICARBAZIDE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.347732922	GNF-PF-2324	chembl:CHEMBL577419	CHEMBL:CHEMBL577419	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.3697723326457359	GNF-PF-388	chembl:CHEMBL582278	CHEMBL:CHEMBL582278	FALSE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.6604738520213144	CHRYSOERIOL	drugbank:DB17283	CHRYSOERIOL	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	DITHIAZANINE	ncit:C72743	DITHIAZANINE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.075442056	REV-5901	chembl:CHEMBL8747	REV-5901	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1017590527823536	NSC-127133	chembl:CHEMBL1172911	CHEMBL:CHEMBL1172911	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	0.1041818873724097	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.090452491	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.023420014	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.030368809	NSC-402083	chembl:CHEMBL1546228	CHEMBL:CHEMBL1546228	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.023440925	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	SB-204070	iuphar.ligand:256	SB 204070	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	SJ000059269	chembl:CHEMBL590686	CHEMBL:CHEMBL590686	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	HYDROXYTOLUIC ACID	ncit:C65873	HYDROXYTOLUIC ACID	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.045579576	DEOXIEPINEPHRINE	chembl:CHEMBL31088	DEOXIEPINEPHRINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BETAMETHASONE BUTYRATE PROPIONATE	ncit:C78755	BETAMETHASONE BUTYRATE PROPIONATE	FALSE	FALSE	FALSE
SIRT5	hgnc:14933	SIRT5	DTC	9/2/20	NULL	0.9376369863516874	NSC-74859	chembl:CHEMBL477936	CHEMBL:CHEMBL477936	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	BROXYQUINOLINE	ncit:C73253	BROXYQUINOLINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	3,3'-DIMETHOXYBENZIDINE	chembl:CHEMBL398363	CHEMBL:CHEMBL398363	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.1724389859957126	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.05913026	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	GNF-PF-628	chembl:CHEMBL1448140	CHEMBL:CHEMBL1448140	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.037721028	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.039939912	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	FEBANTEL	rxcui:24805	FEBANTEL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.1032937794800547	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	6-METHOXY-HARMALAN	chembl:CHEMBL338115	CHEMBL:CHEMBL338115	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.029918901	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	5,8-DIPRENYLOXYPSORALEN	chembl:CHEMBL1710181	CHEMBL:CHEMBL1710181	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	SJ000114740	chembl:CHEMBL592068	CHEMBL:CHEMBL592068	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.002602482	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CHUK	hgnc:1974	CHUK	DTC	9/2/20	NULL	7.501095891	6R-SENECIONYLCHAPARRIN	chembl:CHEMBL564009	CHEMBL:CHEMBL564009	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	DNDI1416924	chembl:CHEMBL156959	CHEMBL:CHEMBL156959	FALSE	FALSE	FALSE
RPS6KA4	hgnc:10433	RPS6KA4	DTC	9/2/20	NULL	0.3281729452230906	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.065634589	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	GANCAONIN L	chembl:CHEMBL590636	GANCAONIN L	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1810609352954982	HYDROCORTISONE 21-OCTANOATE	chembl:CHEMBL253989	CHEMBL:CHEMBL253989	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	DTC	9/2/20	NULL	2.019525817	DESMOSTEROL	iuphar.ligand:2748	DESMOSTEROL	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2194678003581797	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.1766448149224373	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	DTC	9/2/20	NULL	0.1724389859957126	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.023284998	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.020257589	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	TCMDC-124544	chembl:CHEMBL531322	CHEMBL:CHEMBL531322	FALSE	FALSE	FALSE
SLC46A1	hgnc:30521	SLC46A1	DTC	9/2/20	NULL	2.100306849	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	2-ARACHIDONOYLGLYCEROL	iuphar.ligand:729	2-ARACHIDONOYLGLYCEROL	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.5073204950308646	MK-8245	drugbank:DB13024	MK-8245	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	HONOKIOL	rxcui:2562546	HONOKIOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	GF-109203	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.005155392	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	2-PHENYLQUINOLINE	chembl:CHEMBL89786	2-PHENYLQUINOLINE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.02339914	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	1.250182648468916	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.035098711	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	LINURON	chembl:CHEMBL448213	LINURON	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.018340088	PROPACHLOR	chembl:CHEMBL1394829	PROPACHLOR	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	DTC	9/2/20	NULL	0.8468979231563628	4-(2-BENZYLPHENOXY)PIPERIDINE	chembl:CHEMBL1923521	CHEMBL:CHEMBL1923521	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	GNF-PF-5037	chembl:CHEMBL585828	CHEMBL:CHEMBL585828	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	SB-218795	iuphar.ligand:5764	SB 218795	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	(-)-ROLIPRAM	chembl:CHEMBL430893	(-)-ROLIPRAM	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.3804903712731485	DERRUBONE	chembl:CHEMBL412010	DERRUBONE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.1207072901969988	DERRUBONE	chembl:CHEMBL412010	DERRUBONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004339477	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.010586224	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	CID 2056784	chembl:CHEMBL261123	CHEMBL:CHEMBL261123	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.022477599	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
GABRB2	hgnc:4082	GABRB2	DTC	9/2/20	NULL	0.6105543166941221	ISOPIMARIC ACID	chembl:CHEMBL512164	ISOPIMARIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	TEMEFOS	drugbank:DB12231	TEMEFOS	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TENATOPRAZOLE	ncit:C90934	TENATOPRAZOLE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.089756703	ETRAVIRINE	rxcui:475969	ETRAVIRINE	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	7-O-METHYLCRYPTOCHINONE B	chembl:CHEMBL1223743	7-O-METHYLCRYPTOCHINONE B	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.0095957	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	NSC-175743	chembl:CHEMBL1609016	CHEMBL:CHEMBL1609016	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.036162308	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	14-[(N-TETRADECYLAMIDO)SUCCINYL]DOXORUBICIN	chembl:CHEMBL2023733	CHEMBL:CHEMBL2023733	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DNDI1417097	chembl:CHEMBL1531222	CHEMBL:CHEMBL1531222	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PELUBIPROFEN	ncit:C66333	PELUBIPROFEN	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.038187397	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.2465148884304905	GNF-PF-3145	chembl:CHEMBL579761	CHEMBL:CHEMBL579761	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.032694689	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.048618214	4'-EPICHAETOVIRIDIN A	chembl:CHEMBL1306556	CHEMBL:CHEMBL1306556	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.027010119	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NR2E3	hgnc:7974	NR2E3	DTC	9/2/20	NULL	0.2344092465879218	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	GNF-PF-5061	chembl:CHEMBL601385	CHEMBL:CHEMBL601385	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.039778539	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.04464938	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003050289	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.08178765	P-T-OCTYLPHENOL	chembl:CHEMBL259327	CHEMBL:CHEMBL259327	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TETRAZOLIUM RED	chembl:CHEMBL401540	TETRAZOLIUM RED	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.023420014	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	ZK-164015	chembl:CHEMBL184074	CHEMBL:CHEMBL184074	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.018443158	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
CA1	hgnc:1368	CA1	DTC	9/2/20	NULL	2.625383561784724	RESORCINOL	rxcui:35382	RESORCINOL	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.01924768	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.2000292237550266	EPICATECHIN GALLATE	iuphar.ligand:12462	EPICATECHIN GALLATE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	INDOCYANINE GREEN	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.099071078	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	GNF-PF-3537	chembl:CHEMBL601110	CHEMBL:CHEMBL601110	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.009270422	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.014268389	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	TOLAZAMIDE	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.020002922	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.061197752	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	TEMEFOS	drugbank:DB12231	TEMEFOS	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.2067231151011594	SDX-101	chembl:CHEMBL1716091	SDX-101	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	VIOLASTYRENE	chembl:CHEMBL1354529	VIOLASTYRENE	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.018860514	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	S-METOLACHLOR	chembl:CHEMBL2251445	S-METOLACHLOR	FALSE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	DTC	9/2/20	NULL	2.838252499226729	RO-4896062	chembl:CHEMBL2203709	CHEMBL:CHEMBL2203709	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	3.500511415712966	COSMOMYCIN C	chembl:CHEMBL2152009	COSMOMYCIN C	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.028598949	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.006077277	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	4-NITROANILINE	chembl:CHEMBL14282	4-NITROANILINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	NSC-123414	chembl:CHEMBL16751	CHEMBL:CHEMBL16751	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.00709659	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.018962684	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.009270422	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.9907107780319716	SPINASAPONIN A METHYL ESTER	chembl:CHEMBL1288830	SPINASAPONIN A METHYL ESTER	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004120188	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.036337489	BROXYQUINOLINE	ncit:C73253	BROXYQUINOLINE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.2734774543525755	PRECLAMOL	ncit:C82251	PRECLAMOL	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	CID 650707	chembl:CHEMBL408653	CHEMBL:CHEMBL408653	FALSE	FALSE	FALSE
CHRNA3	hgnc:1957	CHRNA3	DTC	9/2/20	NULL	1.591141552596803	3-BENZHYDRYLQUINUCLIDINE	chembl:CHEMBL2332279	CHEMBL:CHEMBL2332279	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.007872215	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	TRIACETYLRESVERATROL	chembl:CHEMBL597744	TRIACETYLRESVERATROL	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.061992528	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.054355767	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.014916952	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.005493584	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.024932417	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	chembl:CHEMBL1449651	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.011047269	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PRKDC	hgnc:9413	PRKDC	DTC	9/2/20	NULL	3.750547945406749	KU-0060648	iuphar.ligand:8011	KU-0060648	FALSE	FALSE	TRUE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.026519026	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.044124093	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.1704794520639431	L-765314	iuphar.ligand:506	L-765314	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.012337329	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TGFBR2	hgnc:11773	TGFBR2	DTC	9/2/20	NULL	5.834185692854945	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	NSC-42258	chembl:CHEMBL1410004	CHEMBL:CHEMBL1410004	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.005778964	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006439499	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.00770359	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1363835616511545	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1491695205559502	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	DNDI1417221	chembl:CHEMBL1459280	CHEMBL:CHEMBL1459280	FALSE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.3750547945406749	SB-242235	chembl:CHEMBL95692	SB-242235	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003703461	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.016727516	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.2059124362184098	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.026458892	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.105015342	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	4,4'-OXYDIANILINE	chembl:CHEMBL354663	CHEMBL:CHEMBL354663	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	MEDROXYPROGESTERONE ACETATE	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.1250182648468916	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.108711535	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.006054153	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1296485709523321	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.009935226	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	EMETINE	rxcui:3820	EMETINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	ELATOSIDE D	chembl:CHEMBL1834952	ELATOSIDE D	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	SDZ-205557	iuphar.ligand:258	SDZ 205557	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.050879526	AG-528	chembl:CHEMBL56542	CHEMBL:CHEMBL56542	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	PIFITHRIN-ALPHA	chembl:CHEMBL198759	CHEMBL:CHEMBL198759	FALSE	FALSE	FALSE
MGLL	hgnc:17038	MGLL	DTC	9/2/20	NULL	17.50255707856483	1,4-BIS(MALIMIDO)XYLENE	chembl:CHEMBL565711	CHEMBL:CHEMBL565711	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.035358701	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.1767935058440892	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	2-AMINOETHOXYDIPHENYL BORATE	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FERBAM	chembl:CHEMBL460100	FERBAM	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	0.1944728564284981	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.048618214	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.014565235	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.038382801	FLAVANONE	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	0.4861821410712454	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.081030357	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.007244436	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	BAS 02077837	chembl:CHEMBL1485809	CHEMBL:CHEMBL1485809	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	1.458546423213736	1,4-BIS(4-METHOXYPHENYLSULFONYL)PIPERAZINE	chembl:CHEMBL1091502	CHEMBL:CHEMBL1091502	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.080042182	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-4431	chembl:CHEMBL494669	CHEMBL:CHEMBL494669	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	CETIRIZINE HYDROCHLORIDE	rxcui:203150	CETIRIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.1526385791735305	CEFMETAZOLE SODIUM	rxcui:203140	CEFMETAZOLE SODIUM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008345148	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	ESTRAMUSTINE PHOSPHATE	rxcui:105556	ESTRAMUSTINE PHOSPHATE	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.095468493	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.007177101	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.2651902587661338	2,4,6-TRIBROMOPHENOL	drugbank:DB02417	2,4,6-TRIBROMOPHENOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00449783	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00402481	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	GNF-PF-1859	chembl:CHEMBL1520837	CHEMBL:CHEMBL1520837	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.021155387	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	DNDI1416934	chembl:CHEMBL1989750	CHEMBL:CHEMBL1989750	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006193403	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004919212	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.032016873	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	TCMDC-125821	chembl:CHEMBL547977	CHEMBL:CHEMBL547977	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	N-(4-CARBOXYPHENYL)RHODANINE	chembl:CHEMBL450802	CHEMBL:CHEMBL450802	FALSE	FALSE	FALSE
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.02706581	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PTK6	hgnc:9617	PTK6	DTC	9/2/20	NULL	0.1193356164447602	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.024513385	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DESOXYCORTICOSTERONE ACETATE	rxcui:258333	DESOXYCORTICOSTERONE ACETATE	TRUE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	DTC	9/2/20	NULL	0.099446347	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.020510809	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	HYDROCORTISONE SODIUM SUCCINATE	rxcui:235483	HYDROCORTISONE SODIUM SUCCINATE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.003341458	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.060984519	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.596678082	OLMESARTAN MEDOXOMIL	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	FENOFIBRIC ACID	rxcui:24852	FENOFIBRIC ACID	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	4-(N,NDIMETHYLAMINO)BENZALDOXIME	chembl:CHEMBL498513	CHEMBL:CHEMBL498513	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.3621218705909965	FUROSPONGOLIDE	chembl:CHEMBL1077108	FUROSPONGOLIDE	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	2.715914029432474	SRT-1720	drugbank:DB17057	SRT-1720	FALSE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.048618214	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.07458476	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MONENSIN SODIUM	ncit:C82249	MONENSIN SODIUM	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	BENZODODECINIUM CHLORIDE	rxcui:1311592	BENZODODECINIUM CHLORIDE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	DITHIAZANINE	ncit:C72743	DITHIAZANINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	4-HYDROXYESTRADIOL	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.011575765	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW284372X	chembl:CHEMBL215993	GW284372X	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	CLOBETASOL PROPIONATE	rxcui:21245	CLOBETASOL PROPIONATE	TRUE	FALSE	FALSE
APBA1	hgnc:578	APBA1	DTC	9/2/20	NULL	0.3201687270469177	PHENAZINE-2,3-DIAMINE	chembl:CHEMBL274921	CHEMBL:CHEMBL274921	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	DNDI1417147	chembl:CHEMBL2094484	CHEMBL:CHEMBL2094484	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.018699313	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.068369364	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.052142673	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.034544521	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	GNF-PF-2491	chembl:CHEMBL577851	CHEMBL:CHEMBL577851	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.011767743	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	LUZINDOLE	iuphar.ligand:1363	LUZINDOLE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.013140058	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ISOPROPYL PALMITATE	rxcui:1311179	ISOPROPYL PALMITATE	TRUE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.04573839	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	DTC	9/2/20	NULL	0.010275474	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010093747	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665961	chembl:CHEMBL602312	CHEMBL:CHEMBL602312	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01535312	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.059532507	LY-83583	chembl:CHEMBL312487	CHEMBL:CHEMBL312487	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	6ALPHA-HYDROXYESTRADIOL	chembl:CHEMBL1432305	CHEMBL:CHEMBL1432305	FALSE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.038665443	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.6019397937072561	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	DNDI1417529	chembl:CHEMBL1990783	CHEMBL:CHEMBL1990783	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.013087655	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	SJ000150791	chembl:CHEMBL600572	CHEMBL:CHEMBL600572	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	GNF-PF-3418	chembl:CHEMBL582099	CHEMBL:CHEMBL582099	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.011365297	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.060008767	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	ENOXIMONE	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	DTC	9/2/20	NULL	0.4605936073306534	ZAMIFENACIN	ncit:C66682	ZAMIFENACIN	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1458546423213736	2-AMINO-ANTHRAQUINONE	chembl:CHEMBL84685	CHEMBL:CHEMBL84685	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.026253836	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.023080295	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003001553	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	N-(4-FLUOROBENZYLCARBAMOTHIOYL)BENZAMIDE	chembl:CHEMBL1545737	CHEMBL:CHEMBL1545737	FALSE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.2500365296937833	JNJ-1661010	iuphar.ligand:5206	JNJ1661010	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.013415348	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	DUP-697	chembl:CHEMBL42485	DUP-697	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007292732	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.012087401	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.007841647	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.00747866	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
NPY1R	hgnc:7956	NPY1R	DTC	9/2/20	NULL	0.7501095890813498	N6-PHENYLADENOSINE	chembl:CHEMBL262083	N6-PHENYLADENOSINE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	GEDUNIN	chembl:CHEMBL465226	GEDUNIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW627512B	chembl:CHEMBL443563	GW627512B	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2892984641085096	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.099446347	FAGARONINE	chembl:CHEMBL282622	FAGARONINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.007884035	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	3.000438356	BAS-8770938	chembl:CHEMBL478510	CHEMBL:CHEMBL478510	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.038981196	ALISOL A-23 ACETATE	chembl:CHEMBL2059711	CHEMBL:CHEMBL2059711	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	0.097870776	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.036770078	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TCMDC-123528	chembl:CHEMBL529138	CHEMBL:CHEMBL529138	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.061992528	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1458546423213736	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.1012684112549556	Exemestane	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.1086365611772989	Glyburide	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	FDA	10-Apr-24	NULL	0.1108075556053025	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CYB5R	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Isosorbide Dinitrate	rxcui:6058	ISOSORBIDE DINITRATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.018704642	Lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
NUDT15	hgnc:23063	NUDT15	FDA	10-Apr-24	NULL	0.5834185692854944	Mercaptopurine	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	FDA	10-Apr-24	NULL	0.2108741816694558	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	MyCancerGenome	20-Jun-17	inhibitor	0.2290910612377596	RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenome	20-Jun-17	inhibitor	NULL	ENMD-0276	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	0.1465330360065893	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	MyCancerGenome	20-Jun-17	inhibitor	1.831662950082366	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.1374032518317239	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.3453256329104173	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.1312691780892362	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
PIK3R6	hgnc:27101	PIK3R6	MyCancerGenome	20-Jun-17	inhibitor	0.108040476	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.017042412	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
VEGFR2	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.070129236	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
AKT2	hgnc:392	AKT2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.364636606	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1101693521639275	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.2917092846427472	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.016621612	AZT	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02639903	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02804897	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.02804897	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.044878351	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.023620185	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.1682938180631233	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
AGER	hgnc:320	AGER	NCI	14-Sep-17	NULL	3.000438356325399	MAPK INHIBITORS	ncit:C2149	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
AGTR2	hgnc:338	AGTR2	NCI	14-Sep-17	NULL	0.8678953923255289	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
AKR1C1	hgnc:384	AKR1C1	NCI	14-Sep-17	NULL	0.921187215	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.2573905452730122	ZINC SULFATE	rxcui:1299928	ZINC SULFATE ANHYDROUS	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.045421861	RECOMBINANT ERYTHROPOIETIN	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	NULL	LIGNAN	NULL	NULL	NULL	NULL	NULL
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
APOD	hgnc:612	APOD	NCI	14-Sep-17	NULL	0.4234489615781814	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	3.029288725136221	REVERSE TRANSCRIPTASE INHIBITOR	ncit:C1589	REVERSE TRANSCRIPTASE INHIBITOR	FALSE	FALSE	FALSE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.087732116	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
BCL2L2	hgnc:995	BCL2L2	NCI	14-Sep-17	NULL	0.8751278539282417	2-CDA	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.060984519	DDI	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.8537832721251137	NORMAL SALINE	hemonc:30954	NORMAL SALINE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.017075665	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.050222545	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	1.419126249613364	CSF	ncit:C387	RECOMBINANT COLONY STIMULATING FACTOR	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.224072566	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.05792352	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.097870776	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.025942525	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.026227608	ALL-TRANS-RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.059667808	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
CASR	hgnc:1514	CASR	NCI	14-Sep-17	NULL	0.7292732116068681	AMINOGLYCOSIDE ANTIBIOTICS	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.6482428547616605	AMINOGLYCOSIDES	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
CHI3L1	hgnc:1932	CHI3L1	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
CP	hgnc:2295	CP	NCI	14-Sep-17	NULL	0.1178623372293928	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
CRHR2	hgnc:2358	CRHR2	NCI	14-Sep-17	NULL	0.1415301111474245	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.7001022831425933	CHEMOSENSITIZER	ncit:C1744	MULTIDRUG RESISTANCE MODULATOR	FALSE	FALSE	FALSE
CTSG	hgnc:2532	CTSG	NCI	14-Sep-17	NULL	1.193356164447602	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
CTSK	hgnc:2536	CTSK	NCI	14-Sep-17	NULL	0.9723642821424906	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.064111931	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.1060761035064535	L-TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.4167275494896388	AZTREONAM	rxcui:1272	AZTREONAM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
CYP2B	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	0.4102161815288632	POLY IC	ncit:C758	POLY IC	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.035418328	BETA-BLOCKER	ncit:C29576	BETA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.035358701	L-TRIIODOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.017274533	LIGNOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.003454907	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.010541895	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1221108633388244	PLATINUM	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.025264317	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
DEFB4	hgnc:2767	DEFB4A	NCI	14-Sep-17	NULL	0.4565884455277782	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	0.2075402025126264	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
DFFB	hgnc:2773	DFFB	NCI	14-Sep-17	NULL	0.2414145803939976	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.1367387271762877	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.1904575128526865	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	0.6364566210387212	CLADRIBINE	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.2105922643142827	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
DSP	hgnc:3052	DSP	NCI	14-Sep-17	NULL	1.842374429322614	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	1.810609352954982	HOECHST 33258	chembl:CHEMBL301735	HOECHST 33258	FALSE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.104285345	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.138178082	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.061919424	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.066047385	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.3977853881492007	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.4039051633514962	PANTOPRAZOLE	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
GAPDH	hgnc:4141	GAPDH	NCI	14-Sep-17	NULL	0.1583941817064691	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
GCLM	hgnc:4312	GCLM	NCI	14-Sep-17	NULL	NULL	CAROTENOID	NULL	NULL	NULL	NULL	NULL
GCLM	hgnc:4312	GCLM	NCI	14-Sep-17	NULL	0.055711057	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.561579372	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
GJA1	hgnc:4274	GJA1	NCI	14-Sep-17	NULL	0.5303805175322677	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
GHRL	hgnc:18129	GHRL	NCI	14-Sep-17	NULL	0.2573905452730122	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.2302968036653267	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.2763561643983921	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
GRB2	hgnc:4566	GRB2	NCI	14-Sep-17	NULL	0.600087671	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	NCI	14-Sep-17	NULL	0.7395446652914718	6-DIAZO-5-OXO-L-NORLEUCINE	drugbank:DB17537	6-DIAZO-5-OXO-L-NORLEUCINE	FALSE	FALSE	FALSE
GRB2	hgnc:4566	GRB2	NCI	14-Sep-17	NULL	1.071585127259071	ANTINEOPLASTIC	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	NCI	14-Sep-17	NULL	0.2273059360852575	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	NCI	14-Sep-17	NULL	0.036821649	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.251232877	ONDANSETRON	rxcui:203148	ONDANSETRON HYDROCHLORIDE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	NULL	CAROTENOID	NULL	NULL	NULL	NULL	NULL
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.108374966	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	2.059124362184098	POLYVALENT VACCINE	ncit:C2848	POLYVALENT VACCINE	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.2734774543525755	4-HYDROPEROXYCYCLOPHOSPHAMIDE	ncit:C1423	PERFOSFAMIDE	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	NULL	AUTOLOGOUS TUMOR CELLS	NULL	NULL	NULL	NULL	NULL
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.086361301	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.182318303	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1372749574789398	2-CDA	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.4102161815288632	SIGNAL TRANSDUCTION INHIBITORS	ncit:C2189	SIGNAL TRANSDUCTION INHIBITOR	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.1286952726365061	13-CIS RETINOIC ACID	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	NULL	EF-2	NULL	NULL	NULL	NULL	NULL
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.1293292394967844	FK 506	rxcui:235991	ANHYDROUS TACROLIMUS	TRUE	TRUE	FALSE
ITGA5	hgnc:6141	ITGA5	NCI	14-Sep-17	NULL	0.8204323630577265	DMSO	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.3017682254924971	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.9723642821424908	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
ITGAX	hgnc:6152	ITGAX	NCI	14-Sep-17	NULL	0.760980743	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.2083637747448194	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	2.386712328895204	LAK CELLS	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	2.386712328895204	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	1.458546423213736	MEGAKARYOCYTE GROWTH AND DEVELOPMENT FACTOR	ncit:C878	RECOMBINANT HUMAN THROMBOPOIETIN	FALSE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.8751278539282416	ABARELIX	rxcui:301739	ABARELIX	TRUE	FALSE	TRUE
KRT18	hgnc:6430	KRT18	NCI	14-Sep-17	NULL	1.381780822	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
KRT19	hgnc:6436	KRT19	NCI	14-Sep-17	NULL	0.6105543166941221	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.182318303	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.1121958787087489	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.065308049	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	NCI	14-Sep-17	NULL	0.1346350544504987	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
MARCKSL1	hgnc:7142	MARCKSL1	NCI	14-Sep-17	NULL	0.729273212	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	NCI	14-Sep-17	NULL	0.6563458904461813	IMIPRAMINE	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.6731752722524935	BMS-275291	ncit:C1875	REBIMASTAT	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1029562181092049	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.053854022	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	0.063072278	6-MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
MT1H	hgnc:7400	MT1H	NCI	14-Sep-17	NULL	0.8824818695074707	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.5000730593875666	HYPOXANTHINE	ncit:C29105	HYPOXANTHINE	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.062509132	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	NCI	14-Sep-17	NULL	0.2430910705356227	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.1259176768242074	GENE THERAPY VECTORS	ncit:C2172	GENE TRANSDUCTION AGENT	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	0.1256164383629055	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	NCI	14-Sep-17	NULL	0.252440727	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
NT5E	hgnc:8021	NT5E	NCI	14-Sep-17	NULL	0.4251633298436802	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	1.093909817410302	2&APOS;-AMINO-3&APOS;-METHOXYFLAVONE	ncit:C1625	MEK INHIBITOR PD-98059	FALSE	FALSE	FALSE
PEBP1	hgnc:8630	PEBP1	NCI	14-Sep-17	NULL	2.763561643983921	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.011124507	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PCSK1	hgnc:8743	PCSK1	NCI	14-Sep-17	NULL	0.7430330835239787	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.060772768	HERBIMYCIN A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.023759127	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	NULL	DIPHOSPHONATE	NULL	NULL	NULL	NULL	NULL
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	0.130291988	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.071277382	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	PD-81723	chembl:CHEMBL59532	CHEMBL:CHEMBL59532	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.086551106	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.016156207	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	0.1902451856365742	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.054020238	AZT	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1041818873724097	ANTINEOPLASTIC	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.086219493	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.015075415	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.047176704	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
RBP3	hgnc:9921	RBP3	NCI	14-Sep-17	NULL	1.693795846312725	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
RPS19	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.1408971500063358	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
S100A10	hgnc:10487	S100A10	NCI	14-Sep-17	NULL	0.6105543166941221	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
SDC2	hgnc:10659	SDC2	NCI	14-Sep-17	NULL	8.751278539282415	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	0.2524407270946851	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	IMIDAZOLE ACETIC ACID	chembl:CHEMBL784	IMIDAZOLE ACETIC ACID	FALSE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	0.1981421556063943	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
SFTPA1	hgnc:10798	SFTPA1	NCI	14-Sep-17	NULL	2.187819634820604	RETINYL PALMITATE	rxcui:35406	VITAMIN A PALMITATE	TRUE	FALSE	FALSE
SLC2A3	hgnc:11007	SLC2A3	NCI	14-Sep-17	NULL	0.3962843112127886	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.050488145	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.070244376	STREPTOZOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
SLPI	hgnc:11092	SLPI	NCI	14-Sep-17	NULL	1.230648544586589	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	NCI	14-Sep-17	NULL	0.013957382	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
SOS1	hgnc:11187	SOS1	NCI	14-Sep-17	NULL	5.527123287967842	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.8078103267029924	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.00258837	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
SOCS6	hgnc:16833	SOCS6	NCI	14-Sep-17	NULL	1.981421556063943	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
SV2A	hgnc:20566	SV2A	NCI	14-Sep-17	NULL	0.3962843112127886	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003439517	ATROPINE	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
STIM2	hgnc:19205	STIM2	NCI	14-Sep-17	NULL	11.66837138570989	AMINOGLYCOSIDE ANTIBIOTIC	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.084553416	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
STRAP	hgnc:30796	STRAP	NCI	14-Sep-17	NULL	7.001022831425933	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.2130128650535274	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
TEAD1	hgnc:11714	TEAD1	NCI	14-Sep-17	NULL	1.221108633388244	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.08334551	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
TBXAS1	hgnc:11609	TBXAS1	NCI	14-Sep-17	NULL	0.2853677784548614	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1141471113819445	OXYQUINOLINE	rxcui:110	OXYQUINOLINE	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	NCI	14-Sep-17	NULL	0.5000730593875666	BDNF	iuphar.ligand:4872	BDNF	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.084689792	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.1417211099478933	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.061376588	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
TGFBR3	hgnc:11774	TGFBR3	NCI	14-Sep-17	NULL	2.187819634820604	RANTES	ncit:C1211	RECOMBINANT RANTES	FALSE	FALSE	FALSE
THBD	hgnc:11784	THBD	NCI	14-Sep-17	NULL	0.3500511415712966	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
WT1	hgnc:12796	WT1	NCI	14-Sep-17	NULL	0.5048814541893701	DMSO	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.1417211099478934	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.1389091831632129	17-AAG	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
SMARCB1	hgnc:11103	SMARCB1	OncoKB	23-Jul-20	NULL	7.501095890813499	Tazemetostat	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	OncoKB	23-Jul-20	NULL	0.637458239	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.049026771	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
APH1B	hgnc:24080	APH1B	DTC	9/2/20	NULL	1.514644363	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	OncoKB	23-Jul-20	NULL	0.1766118064547324	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	OncoKB	23-Jul-20	NULL	0.9814517987980279	Debio1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
ARAF	hgnc:646	ARAF	OncoKB	23-Jul-20	NULL	0.1060761035064535	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	OncoKB	23-Jul-20	NULL	0.4947116523181093	Gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	OncoKB	23-Jul-20	NULL	0.1176247115494948	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
EZH2	hgnc:3527	EZH2	OncoKB	23-Jul-20	NULL	2.917092846427472	Tazemetostat	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	OncoKB	23-Jul-20	NULL	0.179119736	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CSRP3	hgnc:2472	CSRP3	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
APOE	hgnc:613	APOE	PharmGKB	4/5/24	NULL	0.4526523382387456	lecanemab	rxcui:2626143	LECANEMAB	TRUE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	0.065799087	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.029399592	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.037345428	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	VU001171	iuphar.ligand:6228	VU0001171	FALSE	FALSE	FALSE
NTS	hgnc:8038	NTS	PharmGKB	4/5/24	NULL	0.1535312024435511	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
HTR3E	hgnc:24005	HTR3E	PharmGKB	4/5/24	NULL	0.092118721	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.002330153	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	1.280674908	POLYGODIAL	iuphar.ligand:10293	POLYGODIAL	FALSE	FALSE	FALSE
ZIC4	hgnc:20393	ZIC4	PharmGKB	4/5/24	NULL	1.381780822	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.106290832	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
TOR1A	hgnc:3098	TOR1A	PharmGKB	4/5/24	NULL	1.381780822	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
DPP6	hgnc:3010	DPP6	PharmGKB	4/5/24	NULL	0.027635616	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
RGS2	hgnc:9998	RGS2	PharmGKB	4/5/24	NULL	1.381780822	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
LEPR	hgnc:6554	LEPR	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
ATAT1	hgnc:21186	ATAT1	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CACNG2	hgnc:1406	CACNG2	PharmGKB	4/5/24	NULL	0.079197091	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	hydroxyphenytoin	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	7-hydroxy r-warfarin	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	7-hydroxy s-warfarin	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.072927321	tenoxicam	rxcui:37790	TENOXICAM	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.003116552	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.003198567	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	NULL	hormonal contraceptives for systemic use	NULL	NULL	NULL	NULL	NULL
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.058602312	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.045265234	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005867434	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.5966780822238011	selegiline	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
ATP5F1E	hgnc:838	ATP5F1E	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.019461702	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	PharmGKB	4/5/24	NULL	0.101562227	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.031612084	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	PharmGKB	4/5/24	NULL	0.008621949	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CCL2	hgnc:10618	CCL2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
BDNF-AS	hgnc:20608	BDNF-AS	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.016690296	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
IBA57	hgnc:27302	IBA57	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
NEFM	hgnc:7734	NEFM	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
PI4KA	hgnc:8983	PI4KA	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
ADCY2	hgnc:233	ADCY2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CACNA1B	hgnc:1389	CACNA1B	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CACNA1E	hgnc:1392	CACNA1E	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CACNA2D3	hgnc:15460	CACNA2D3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CACNB4	hgnc:1404	CACNB4	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CACNG3	hgnc:1407	CACNG3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CHRM4	hgnc:1953	CHRM4	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	3.500511415712966	CUCURBITACIN E	chembl:CHEMBL455056	CUCURBITACIN E	FALSE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
DGKB	hgnc:2850	DGKB	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	1.166837138570988	Ergot alkaloids	rxcui:4023	ERGOT ALKALOIDS	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	PharmGKB	4/5/24	NULL	NULL	Beta blocking agents, selective	NULL	NULL	NULL	NULL	NULL
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	NULL	Antithyroid Preparations	NULL	NULL	NULL	NULL	NULL
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	0.7001022831425934	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.024596061	mianserin	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.3365876361262467	Zosuquidar	ncit:C76198	ZOSUQUIDAR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.6731752722524935	R101933	ncit:C28698	LANIQUIDAR	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.037398626	silibinin	ncit:C152359	SILIBININ	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.018699313	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.010199625	fluphenazine	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.008630452	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
PGLYRP4	hgnc:30015	PGLYRP4	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
NFKB1	hgnc:7794	NFKB1	PharmGKB	4/5/24	NULL	0.042516333	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.05913026	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.056097939	midazolam	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.1481697953740938	osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	PharmGKB	4/5/24	NULL	NULL	Pyrimidine analogues	NULL	NULL	NULL	NULL	NULL
RGS4	hgnc:10000	RGS4	PharmGKB	4/5/24	NULL	0.0230499	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
MS4A1	hgnc:7315	MS4A1	PharmGKB	4/5/24	NULL	5.834185692854944	ibritumomab	rxcui:262323	IBRITUMOMAB TIUXETAN	TRUE	TRUE	TRUE
GSR	hgnc:4623	GSR	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
SCN10A	hgnc:10582	SCN10A	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
NR1I3	hgnc:7969	NR1I3	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
ATP7B	hgnc:870	ATP7B	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	NULL	Beta Blocking Agents	NULL	NULL	NULL	NULL	NULL
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	NULL	Beta Blocking Agents	NULL	NULL	NULL	NULL	NULL
KL	hgnc:6344	KL	PharmGKB	4/5/24	NULL	NULL	Beta Blocking Agents	NULL	NULL	NULL	NULL	NULL
CYP19A1	hgnc:2594	CYP19A1	PharmGKB	4/5/24	NULL	NULL	triglycerides	NULL	NULL	NULL	NULL	NULL
NAGS	hgnc:17996	NAGS	PharmGKB	4/5/24	NULL	NULL	sodium benzoate / sodium phenylacetate	NULL	NULL	NULL	NULL	NULL
ZNF816	hgnc:26995	ZNF816	PharmGKB	4/5/24	NULL	1.009762908	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
HLA-E	hgnc:4962	HLA-E	PharmGKB	4/5/24	NULL	0.6731752722524936	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
PSORS1C1	hgnc:17202	PSORS1C1	PharmGKB	4/5/24	NULL	0.8078103267029924	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.106290832	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
PLA2G4A	hgnc:9035	PLA2G4A	PharmGKB	4/5/24	NULL	NULL	Pyrazolones	NULL	NULL	NULL	NULL	NULL
PLA2G4A	hgnc:9035	PLA2G4A	PharmGKB	4/5/24	NULL	NULL	propionic acid derivatives	NULL	NULL	NULL	NULL	NULL
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.5385402178019949	amlodipine	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
ATF5	hgnc:790	ATF5	PharmGKB	4/5/24	NULL	0.1620607136904151	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.052090944	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
CTNNA2	hgnc:2510	CTNNA2	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
EYA4	hgnc:3522	EYA4	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
IFNG	hgnc:5438	IFNG	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.07631929	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
IFNGR1	hgnc:5439	IFNGR1	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	SJ000089102	chembl:CHEMBL606460	CHEMBL:CHEMBL606460	FALSE	FALSE	FALSE
IFNGR2	hgnc:5440	IFNGR2	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
IL12B	hgnc:5970	IL12B	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
IL17A	hgnc:5981	IL17A	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
IL1RN	hgnc:6000	IL1RN	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.068369364	CID 650707	chembl:CHEMBL408653	CHEMBL:CHEMBL408653	FALSE	FALSE	FALSE
IL5	hgnc:6016	IL5	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
IL9	hgnc:6029	IL9	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
KLRC4	hgnc:6377	KLRC4	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.1392776425349986	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
MAFB	hgnc:6408	MAFB	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
MICA	hgnc:7090	MICA	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
PON1	hgnc:9204	PON1	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
TBX21	hgnc:11599	TBX21	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
TLR2	hgnc:11848	TLR2	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
TLR4	hgnc:11850	TLR4	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
TLR5	hgnc:11851	TLR5	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
TNFAIP3	hgnc:11896	TNFAIP3	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
TNFRSF1A	hgnc:11916	TNFRSF1A	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
SLC12A8	hgnc:15595	SLC12A8	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1296485709523321	itraconazole	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	NULL	Alkylating Agents	NULL	NULL	NULL	NULL	NULL
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.029833904	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	PharmGKB	4/5/24	NULL	0.073850452	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	PharmGKB	4/5/24	NULL	0.022949157	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	PharmGKB	4/5/24	NULL	0.1902451856365742	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.038256955	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.04427291	palonosetron	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	desethyl hydroxychloroquine	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.013622434	clonidine	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.002241666	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	0.3043922970185188	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
SLC22A6	hgnc:10970	SLC22A6	PharmGKB	4/5/24	NULL	0.3547815624033412	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
PROC	hgnc:9451	PROC	PharmGKB	4/5/24	NULL	1.312691780892362	synthetic conjugated estrogens, A	rxcui:253166	SYNTHETIC CONJUGATED ESTROGENS, A	FALSE	FALSE	FALSE
AGBL4	hgnc:25892	AGBL4	PharmGKB	4/5/24	NULL	1.875273972703374	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
ITPA	hgnc:6176	ITPA	PharmGKB	4/5/24	NULL	1.093909817410302	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
ARG1	hgnc:663	ARG1	PharmGKB	4/5/24	NULL	NULL	sodium benzoate / sodium phenylacetate	NULL	NULL	NULL	NULL	NULL
CSNK2A1	hgnc:2457	CSNK2A1	DTC	9/2/20	NULL	0.024309107	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ARG1	hgnc:663	ARG1	PharmGKB	4/5/24	NULL	0.4546118721705151	sildenafil	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.2143170254518142	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
PLCG1	hgnc:9065	PLCG1	PharmGKB	4/5/24	NULL	NULL	Pyrazolones	NULL	NULL	NULL	NULL	NULL
PLCG1	hgnc:9065	PLCG1	PharmGKB	4/5/24	NULL	NULL	propionic acid derivatives	NULL	NULL	NULL	NULL	NULL
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	NULL	desmethylclozapine glucuronide	NULL	NULL	NULL	NULL	NULL
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	NULL	nivolumab / relatlimab	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.007366396	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.033243223	hydroxyzine	rxcui:5553	HYDROXYZINE	TRUE	FALSE	FALSE
EPHA6	hgnc:19296	EPHA6	PharmGKB	4/5/24	NULL	0.2561349816375341	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
SPIDR	hgnc:28971	SPIDR	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.03357268	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
TNRC6A	hgnc:11969	TNRC6A	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NAT2	hgnc:7646	NAT2	PharmGKB	4/5/24	NULL	0.043756393	clonazepam	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.04339477	ambrisentan	rxcui:358274	AMBRISENTAN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	16alpha-hydroxyprogesterone	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.054243462	desoxycortone	rxcui:3256	DESOXYCORTICOSTERONE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.016690296	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.031536139	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	XANTHYLETIN	chembl:CHEMBL303846	XANTHYLETIN	FALSE	FALSE	FALSE
HLA-E	hgnc:4962	HLA-E	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.1137761023525341	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
DUX1	hgnc:3079	DUX1	PharmGKB	4/5/24	NULL	1.250182648468916	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
EPM2A	hgnc:3413	EPM2A	PharmGKB	4/5/24	NULL	0.5000730593875666	trifluoperazine	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	SJ000173328	chembl:CHEMBL591613	CHEMBL:CHEMBL591613	FALSE	FALSE	FALSE
ERICH3	hgnc:25346	ERICH3	PharmGKB	4/5/24	NULL	1.000146118775133	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
TNFRSF8	hgnc:11923	TNFRSF8	PharmGKB	4/5/24	NULL	1.276228120312019	brentuximab vedotin	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2191733444543002	ALBUTEROL	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	NULL	Rubella vaccines	NULL	NULL	NULL	NULL	NULL
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.2651902587661338	codeine	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
APOA5	hgnc:17288	APOA5	PharmGKB	4/5/24	NULL	1.400204566285186	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.1521961485092594	gemtuzumab ozogamicin	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
ADH1A	hgnc:249	ADH1A	PharmGKB	4/5/24	NULL	0.6563458904461813	gemtuzumab ozogamicin	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005903055	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.064824285	hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.072424374	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	PharmGKB	4/5/24	NULL	0.081533651	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PPP1R13L	hgnc:18838	PPP1R13L	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.2430910705356226	8-AZAGUANINE	ncit:C28788	8-AZAGUANINE	FALSE	FALSE	FALSE
MIR582	hgnc:32838	MIR582	PharmGKB	4/5/24	NULL	2.917092846427472	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
ADCY9	hgnc:240	ADCY9	PharmGKB	4/5/24	NULL	10.50153424713889	dalcetrapib	ncit:C81529	DALCETRAPIB	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1193356164447602	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.5073204950308646	valsartan	rxcui:69749	VALSARTAN	TRUE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.025588534	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GALNT18	hgnc:30488	GALNT18	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PROCR	hgnc:9452	PROCR	PharmGKB	4/5/24	NULL	NULL	hormonal contraceptives for systemic use	NULL	NULL	NULL	NULL	NULL
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-1686	chembl:CHEMBL580140	CHEMBL:CHEMBL580140	FALSE	FALSE	FALSE
CDH2	hgnc:1759	CDH2	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
CAMK1D	hgnc:19341	CAMK1D	PharmGKB	4/5/24	NULL	1.193356164447602	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.013890918	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	1.615620653405984	cannabinoids	chembl:CHEMBL3833333	NABIXIMOLS	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.11707396	pyrazinamide	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
FKBP5	hgnc:3721	FKBP5	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	S-166659	chembl:CHEMBL252417	CHEMBL:CHEMBL252417	FALSE	FALSE	FALSE
CYP17A1	hgnc:2593	CYP17A1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	DNDI1417560	chembl:CHEMBL1373255	CHEMBL:CHEMBL1373255	FALSE	FALSE	FALSE
KLB	hgnc:15527	KLB	PharmGKB	4/5/24	NULL	0.3323270331373069	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.051731696	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
ZMAT4	hgnc:25844	ZMAT4	PharmGKB	4/5/24	NULL	1.458546423213736	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.2651902587661338	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	PharmGKB	4/5/24	NULL	0.076263865	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NQO2	hgnc:7856	NQO2	PharmGKB	4/5/24	NULL	0.076263865	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.3409589041278864	sildenafil	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.018081154	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
CBR3	hgnc:1549	CBR3	PharmGKB	4/5/24	NULL	0.1440539677248134	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
LAG3	hgnc:6476	LAG3	PharmGKB	4/5/24	NULL	NULL	nivolumab / relatlimab	NULL	NULL	NULL	NULL	NULL
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	1.810609352954982	TENOVIN-6	chembl:CHEMBL1945130	CHEMBL:CHEMBL1945130	FALSE	FALSE	FALSE
ANKS1B	hgnc:24600	ANKS1B	PharmGKB	4/5/24	NULL	0.3323270331373069	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	PharmGKB	4/5/24	NULL	0.1389091831632129	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	PharmGKB	4/5/24	NULL	0.4947116523181093	gilteritinib	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
HTR3B	hgnc:5298	HTR3B	PharmGKB	4/5/24	NULL	0.078194596	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.04593847	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
GLCCI1	hgnc:18713	GLCCI1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.048083948	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.1107756777124356	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
EPHX1	hgnc:3401	EPHX1	PharmGKB	4/5/24	NULL	0.1035654265003836	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.007390242	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	NULL	desmethyl olanzapine	NULL	NULL	NULL	NULL	NULL
HSD3B1	hgnc:5217	HSD3B1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
FGFR4	hgnc:3691	FGFR4	PharmGKB	4/5/24	NULL	0.063839114	everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
ABCC1	hgnc:51	ABCC1	PharmGKB	4/5/24	NULL	0.1912847768149162	conjugated estrogens	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.014757637	propranolol	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.005483257	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
NPHS1	hgnc:7908	NPHS1	PharmGKB	4/5/24	NULL	19.09369863116163	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	NULL	propionic acid derivatives	NULL	NULL	NULL	NULL	NULL
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.01090502	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.1363127498330594	conjugated estrogens	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.1058622403945453	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.1101693521639275	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.092606122	XL647	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	TALC	12-May-16	inhibitor	0.1162317016838838	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	2.972132334095915	CIXUTUMUMAB	ncit:C79828	CIXUTUMUMAB	FALSE	TRUE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	1.981421556063943	R1507	ncit:C95797	TEPROTUMUMAB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	NULL	ENMD-0276	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00202529	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
KIF11	hgnc:6388	KIF11	TALC	12-May-16	inhibitor	13.12691780892362	ISPINESIB	ncit:C38131	ISPINESIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.018305561	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.2641230947469542	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	0.525076712	ALOGLIPTIN	rxcui:1368001	ALOGLIPTIN	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	NULL	AN-2898	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.045898314	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P45984	hgnc:6886	MAPK9	TdgClinicalTrial	Jan-14	NULL	0.4102161815288632	AM-111	iuphar.ligand:9101	BRIMAPITIDE	FALSE	FALSE	FALSE
UNIPROT:P13945	hgnc:288	ADRB3	TdgClinicalTrial	Jan-14	NULL	1.500219178	AMIBEGRON	ncit:C77932	AMIBEGRON	FALSE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	NULL	AN-2898	NULL	NULL	NULL	NULL	NULL
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.025244073	PLX-4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
UNIPROT:P08648	hgnc:6141	ITGA5	TdgClinicalTrial	Jan-14	NULL	NULL	F200	NULL	NULL	NULL	NULL	NULL
UNIPROT:P05556	hgnc:6153	ITGB1	TdgClinicalTrial	Jan-14	NULL	NULL	F200	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.00258837	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
UNIPROT:Q9Y5N1	hgnc:5184	HRH3	TdgClinicalTrial	Jan-14	NULL	NULL	APD916	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.068637479	ANG1005	drugbank:DB18167	ANG1005	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.5048814541893701	APD791	drugbank:DB05227	APD791	FALSE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	NULL	ARC100	NULL	NULL	NULL	NULL	NULL
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
UNIPROT:P25445	hgnc:11920	FAS	TdgClinicalTrial	Jan-14	NULL	NULL	ARG098	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8TDS4	hgnc:24827	HCAR2	TdgClinicalTrial	Jan-14	NULL	NULL	ARI-3037MO	NULL	NULL	NULL	NULL	NULL
UNIPROT:P49019	hgnc:16824	HCAR3	TdgClinicalTrial	Jan-14	NULL	NULL	ARI-3037MO	NULL	NULL	NULL	NULL	NULL
UNIPROT:P40261	hgnc:7861	NNMT	TdgClinicalTrial	Jan-14	NULL	NULL	ARI-3037MO	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	AMINOHIPPURIC ACID	rxcui:42837	P-AMINOHIPPURATE	TRUE	FALSE	FALSE
UNIPROT:Q15274	hgnc:9755	QPRT	TdgClinicalTrial	Jan-14	NULL	NULL	ARI-3037MO	NULL	NULL	NULL	NULL	NULL
UNIPROT:P19235	hgnc:3416	EPOR	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	EPOETIN ALFA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P35557	hgnc:4195	GCK	TdgClinicalTrial	Jan-14	NULL	NULL	ARRY-403	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.020542907	ARRY-614	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TRIFLOXYSTROBIN	chembl:CHEMBL1897483	TRIFLOXYSTROBIN	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	NULL	ASC-J9	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01106	hgnc:7553	MYC	TdgClinicalTrial	Jan-14	NULL	NULL	AVI-5126	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08709	hgnc:3544	F7	TdgClinicalTrial	Jan-14	NULL	0.069454592	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TdgClinicalTrial	Jan-14	NULL	NULL	FILGRAMSTIM	NULL	NULL	NULL	NULL	NULL
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	PIRENZEPINE	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
UNIPROT:P20839	hgnc:6052	IMPDH1	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	AVN-944	drugbank:DB05500	AVN-944	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	BALSALAZIDE	rxcui:18747	BALSALAZIDE	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	0.3889457128569963	INTERFERON BETA-1A	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	0.1374032518317239	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.1312691780892362	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CHLORALIN	chembl:CHEMBL144530	CHLORALIN	FALSE	FALSE	FALSE
UNIPROT:P14151	hgnc:10720	SELL	TdgClinicalTrial	Jan-14	NULL	11.66837138570988	BIMOSIAMOSE	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	0.1465330360065893	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.596678082	BUCINDOLOL	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.5016656487486736	CALCIPOTRIENE	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
UNIPROT:P41597	hgnc:1603	CCR2	TdgClinicalTrial	Jan-14	NULL	NULL	CCL2-LPM	NULL	NULL	NULL	NULL	NULL
UNIPROT:P51686	hgnc:1610	CCR9	TdgClinicalTrial	Jan-14	NULL	NULL	CCX025	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	NARINGENIN	rxcui:1368173	NARINGENIN	FALSE	FALSE	FALSE
UNIPROT:O14788	hgnc:11926	TNFSF11	TdgClinicalTrial	Jan-14	NULL	NULL	CEP-37251	NULL	NULL	NULL	NULL	NULL
UNIPROT:P49069	hgnc:1471	CAMLG	TdgClinicalTrial	Jan-14	NULL	0.6035364509849942	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
UNIPROT:A1Z199	NULL	NULL	TdgClinicalTrial	Jan-14	NULL	NULL	CMLVAX100	drugbank:DB05164	CMLVAX100	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	TRIS(2,3-DIBROMOPROPYL)PHOSPHATE	chembl:CHEMBL1904600	TRIS(2,3-DIBROMOPROPYL)PHOSPHATE	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.087318744	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.078682824	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1835932560688619	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TdgClinicalTrial	Jan-14	NULL	0.1704794520639432	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	SEMAPIMOD	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
UNIPROT:O15264	hgnc:6875	MAPK13	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	SEMAPIMOD	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.050246575	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
UNIPROT:Q9UM73	hgnc:427	ALK	TdgClinicalTrial	Jan-14	NULL	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.090064616	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	SEMAPIMOD	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
UNIPROT:P11362	hgnc:3688	FGFR1	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141B	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21802	hgnc:3689	FGFR2	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141B	NULL	NULL	NULL	NULL	NULL
UNIPROT:P22607	hgnc:3690	FGFR3	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141B	NULL	NULL	NULL	NULL	NULL
UNIPROT:P22455	hgnc:3691	FGFR4	TdgClinicalTrial	Jan-14	NULL	NULL	CVBT-141B	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.2027323213733378	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
UNIPROT:P29460	hgnc:5970	IL12B	TdgClinicalTrial	Jan-14	NULL	NULL	DNA IL-12	NULL	NULL	NULL	NULL	NULL
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	SJ000236197	chembl:CHEMBL582496	CHEMBL:CHEMBL582496	FALSE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TdgClinicalTrial	Jan-14	NULL	NULL	EVT-302	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q16665	hgnc:4910	HIF1A	TdgClinicalTrial	Jan-14	NULL	NULL	SPC/ENZ2968	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.07182992	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	S-ETOMIDATE	chembl:CHEMBL279678	S-ETOMIDATE	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	FISPEMIFENE	ncit:C65687	FISPEMIFENE	FALSE	FALSE	FALSE
UNIPROT:P06493	hgnc:1722	CDK1	TdgClinicalTrial	Jan-14	NULL	0.1544343271638073	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DI-TERT-BUTYLHYDROQUINONE	chembl:CHEMBL480626	CHEMBL:CHEMBL480626	FALSE	FALSE	FALSE
UNIPROT:Q00534	hgnc:1777	CDK6	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.2419708351875322	TOFACITINIB	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
UNIPROT:P24941	hgnc:1771	CDK2	TdgClinicalTrial	Jan-14	NULL	0.1022876712383659	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.1835932560688619	FOSPHENYTOIN	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	TCMDC-124557	chembl:CHEMBL530682	CHEMBL:CHEMBL530682	FALSE	FALSE	FALSE
UNIPROT:Q15131	hgnc:1770	CDK10	TdgClinicalTrial	Jan-14	NULL	0.5250767123569451	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
UNIPROT:O14836	hgnc:18153	TNFRSF13B	TdgClinicalTrial	Jan-14	NULL	NULL	LYMPHORAD	NULL	NULL	NULL	NULL	NULL
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE	chembl:CHEMBL1255936	CHEMBL:CHEMBL1255936	FALSE	FALSE	FALSE
UNIPROT:Q96RJ3	hgnc:17755	TNFRSF13C	TdgClinicalTrial	Jan-14	NULL	NULL	LYMPHORAD	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
UNIPROT:Q02223	hgnc:11913	TNFRSF17	TdgClinicalTrial	Jan-14	NULL	NULL	LYMPHORAD	NULL	NULL	NULL	NULL	NULL
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.056097939	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
UNIPROT:P48546	hgnc:4271	GIPR	TdgClinicalTrial	Jan-14	NULL	NULL	MAR701	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	MAR701	NULL	NULL	NULL	NULL	NULL
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	4.375639269641208	6-METHOXYCOMAPARVIN 5-METHYL ETHER	chembl:CHEMBL256967	CHEMBL:CHEMBL256967	FALSE	FALSE	FALSE
UNIPROT:P46976	hgnc:4699	GYG1	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.038187397	MESALAZINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	3-((2,4-DICHLOROPHENYLTHIO)METHYL)BENZOATE	chembl:CHEMBL1923999	CHEMBL:CHEMBL1923999	FALSE	FALSE	FALSE
UNIPROT:P47989	hgnc:12805	XDH	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	OXYPURINOL	ncit:C87294	OXYPURINOL	TRUE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.007624172	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.038187397	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	QUINOXALINE	chembl:CHEMBL39444	QUINOXALINE	FALSE	FALSE	FALSE
UNIPROT:Q683C9	NULL	NULL	TdgClinicalTrial	Jan-14	NULL	NULL	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.8140724222588294	MILVETEROL	ncit:C77935	MILVETEROL	FALSE	FALSE	FALSE
UNIPROT:P09874	hgnc:270	PARP1	TdgClinicalTrial	Jan-14	NULL	0.900131507	MK-4827	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1215455352678113	TCMDC-124544	chembl:CHEMBL531322	CHEMBL:CHEMBL531322	FALSE	FALSE	FALSE
UNIPROT:P15328	hgnc:3791	FOLR1	TdgClinicalTrial	Jan-14	NULL	8.751278539282417	FARLETUZUMAB	ncit:C61503	FARLETUZUMAB	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	GUAIFENESIN	rxcui:5032	GUAIFENESIN	TRUE	FALSE	FALSE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	MT-103	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.2014360789093139	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.021422958	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.179119736	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.03140411	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:P04049	hgnc:9829	RAF1	TdgClinicalTrial	Jan-14	NULL	0.159436249	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.076765601	GINGKOLIC ACID	chembl:CHEMBL445177	GINGKOLIC ACID	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.063331621	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.035430277	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.106290832	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:P00519	hgnc:76	ABL1	TdgClinicalTrial	Jan-14	NULL	0.637458239	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	NULL	PEG-DOCETAXEL	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	NULL	PEG-DOCETAXEL	NULL	NULL	NULL	NULL	NULL
UNIPROT:P06213	hgnc:6091	INSR	TdgClinicalTrial	Jan-14	NULL	NULL	NN1952	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10827	hgnc:11796	THRA	TdgClinicalTrial	Jan-14	NULL	NULL	TRIIODOTHYRONINE (T3)	NULL	NULL	NULL	NULL	NULL
UNIPROT:P10828	hgnc:11799	THRB	TdgClinicalTrial	Jan-14	NULL	NULL	TRIIODOTHYRONINE (T3)	NULL	NULL	NULL	NULL	NULL
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.021733308	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
UNIPROT:P47989	hgnc:12805	XDH	TdgClinicalTrial	Jan-14	NULL	0.31414846	ALLOPURINOL	rxcui:519	ALLOPURINOL	TRUE	FALSE	FALSE
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	0.7001022831425933	OTELIXIZUMAB	ncit:C95790	OTELIXIZUMAB	FALSE	FALSE	FALSE
UNIPROT:P42345	hgnc:3942	MTOR	TdgClinicalTrial	Jan-14	NULL	0.3697723326457359	PALOMID 529	drugbank:DB12812	PALOMID 529	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TdgClinicalTrial	Jan-14	NULL	0.087222045	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.3846715841442821	CRA-024781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.2027323213733378	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
UNIPROT:Q05655	hgnc:9399	PRKCD	TdgClinicalTrial	Jan-14	NULL	0.1025540453822158	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
UNIPROT:P24723	hgnc:9403	PRKCH	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
UNIPROT:Q9Y251	hgnc:5164	HPSE	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	2-O, 3-O DESULFATED HEPARIN	drugbank:DB17569	2-O, 3-O DESULFATED HEPARIN	FALSE	FALSE	FALSE
UNIPROT:P78348	hgnc:100	ASIC1	TdgClinicalTrial	Jan-14	NULL	NULL	PPC-5650	NULL	NULL	NULL	NULL	NULL
UNIPROT:P12259	hgnc:3542	F5	TdgClinicalTrial	Jan-14	NULL	0.024582243	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT PEGYLATED ACETYLCHOLINESTERASE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	NULL	PSN602	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	NULL	PSN602	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	NULL	PSN602	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	NULL	PSN602	NULL	NULL	NULL	NULL	NULL
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	PRX-08066	drugbank:DB05607	PRX-08066	FALSE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.081407242	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.085378327	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.2333674277141978	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P25024	hgnc:6026	CXCR1	TdgClinicalTrial	Jan-14	NULL	3.000438356	SCH-527123	iuphar.ligand:8497	NAVARIXIN	FALSE	FALSE	FALSE
UNIPROT:Q04609	hgnc:3788	FOLH1	TdgClinicalTrial	Jan-14	NULL	0.2160809515872201	CLAVULANIC ACID	rxcui:21216	CLAVULANIC ACID	TRUE	FALSE	FALSE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.076098074	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.1029562181092049	SOLIFENACIN	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	NULL	GONADOTROPIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P05412	hgnc:6204	JUN	TdgClinicalTrial	Jan-14	NULL	NULL	T-5224	NULL	NULL	NULL	NULL	NULL
UNIPROT:O00206	hgnc:11850	TLR4	TdgClinicalTrial	Jan-14	NULL	4.565884455277782	TAK-242	iuphar.ligand:9036	RESATORVID	FALSE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	SULODEXIDE	ncit:C152467	SULODEXIDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.054695491	SULFASALAZINE	rxcui:9524	SULFASALAZINE	TRUE	FALSE	FALSE
UNIPROT:P24462	hgnc:2640	CYP3A7	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	TESMILIFENE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
UNIPROT:P20815	hgnc:2638	CYP3A5	TdgClinicalTrial	Jan-14	NULL	0.072927321	TESMILIFENE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
UNIPROT:P35499	hgnc:10591	SCN4A	TdgClinicalTrial	Jan-14	NULL	0.080781033	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
UNIPROT:Q9UI33	hgnc:10583	SCN11A	TdgClinicalTrial	Jan-14	NULL	0.084689792	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	2.423430980108977	HOMOTAURINE	rxcui:1374845	TRAMIPROSATE	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.054695491	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:Q8N0U8	hgnc:21492	VKORC1L1	TdgClinicalTrial	Jan-14	NULL	1.810609352954982	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:Q14416	hgnc:4594	GRM2	TdgClinicalTrial	Jan-14	NULL	NULL	TS-032, PF-4802540	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14832	hgnc:4595	GRM3	TdgClinicalTrial	Jan-14	NULL	NULL	TS-032, PF-4802540	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00749	hgnc:9052	PLAU	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
UNIPROT:Q9H2X6	hgnc:14402	HIPK2	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	VADIMEZAN	ncit:C2504	VADIMEZAN	FALSE	FALSE	TRUE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.2465148884304905	VADIMEZAN	ncit:C2504	VADIMEZAN	FALSE	FALSE	TRUE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.071439008	MELEVODOPA	ncit:C83927	MELEVODOPA	TRUE	FALSE	FALSE
UNIPROT:P05120	hgnc:8584	SERPINB2	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
UNIPROT:P01133	hgnc:3229	EGF	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	NIMOTUZUMAB	ncit:C2733	NIMOTUZUMAB	FALSE	TRUE	TRUE
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	NULL	VEGF-121	NULL	NULL	NULL	NULL	NULL
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	NULL	VEGF GENE THERAPY	NULL	NULL	NULL	NULL	NULL
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.1458546423213736	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
UNIPROT:Q03431	hgnc:9608	PTH1R	TdgClinicalTrial	Jan-14	NULL	NULL	H-PTH 1-34	NULL	NULL	NULL	NULL	NULL
UNIPROT:P49190	hgnc:9609	PTH2R	TdgClinicalTrial	Jan-14	NULL	NULL	H-PTH 1-34	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q03181	hgnc:9235	PPARD	TdgClinicalTrial	Jan-14	NULL	NULL	ETHYL EICOSAPENTAENOIC ACID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P51681	hgnc:1606	CCR5	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	VICRIVIROC	ncit:C73589	VICRIVIROC	FALSE	FALSE	FALSE
UNIPROT:Q8NER1	hgnc:12716	TRPV1	TdgClinicalTrial	Jan-14	NULL	NULL	TRPV1 ANTAGONIST	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	VRS-859	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	NULL	XEN2174	NULL	NULL	NULL	NULL	NULL
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
UNIPROT:P30536	hgnc:1158	TSPO	TdgClinicalTrial	Jan-14	NULL	4.145342465975881	CHLORMEZANONE	rxcui:2373	CHLORMEZANONE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.091583148	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.100976291	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.2019525816757481	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1363127498330594	CONJUGATED ESTROGENS	rxcui:4099	ESTROGENS, CONJUGATED (USP)	TRUE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	CROMOGLICATE	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.133607306	DESOXIMETASONE	rxcui:3255	DESOXIMETASONE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.04724037	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	1.790034246671403	ENPROFYLLINE	ncit:C74327	ENPROFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P06870	hgnc:6357	KLK1	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	ECALLANTIDE	rxcui:658708	ECALLANTIDE	TRUE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TdgClinicalTrial	Jan-14	NULL	2.812910959055062	EPOPROSTENOL	rxcui:8814	EPOPROSTENOL	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.039390601	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.080225625	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.3006164383722967	FLUOROMETHOLONE	rxcui:4491	FLUOROMETHOLONE	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	GLIPIZIDE	rxcui:4821	GLIPIZIDE	TRUE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	0.9376369863516874	INTERFERON ALFA-2B, RECOMBINANT	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.7143900848393808	IBUTILIDE	rxcui:41289	IBUTILIDE	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TdgClinicalTrial	Jan-14	NULL	16.40864726115453	LUTROPIN ALFA	rxcui:388084	LUTROPIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.4817217544559128	METHADYL ACETATE	rxcui:6814	METHADYL ACETATE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1479089330582944	MEPERIDINE	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.693795846312725	METHDILAZINE	rxcui:29648	METHDILAZINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.2734774543525755	METHOXAMINE	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.048083948	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TdgClinicalTrial	Jan-14	NULL	0.053361455	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.050879526	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.056097939	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.052090944	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.049723174	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.035083077	NILUTAMIDE	rxcui:31805	NILUTAMIDE	TRUE	FALSE	TRUE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	1.166837138570988	OUABAIN	rxcui:7762	OUABAIN	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.1591141552596803	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.088945801	SULPIRIDE	rxcui:10239	SULPIRIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.1049104320393496	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.1164249916534246	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	0.2892984641085096	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1396480617970598	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:Q92887	hgnc:53	ABCC2	TEND	1-Aug-11	NULL	0.1562728310586145	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	2-HYDROXY-NAPHTHALDEHYDE THIOSEMICARBAZONE	chembl:CHEMBL505209	CHEMBL:CHEMBL505209	FALSE	FALSE	FALSE
UNIPROT:P14060	hgnc:5217	HSD3B1	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.2206204673768676	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.078194596	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.087318744	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.078682824	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:Q06432	hgnc:1405	CACNG1	TEND	1-Aug-11	NULL	0.4688184931758437	CLEVIDIPINE	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TEND	1-Aug-11	NULL	1.458546423213736	CROMOGLICATE	rxcui:2921	CROMOGLYCATE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.2631963470460877	DIPHENIDOL	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.07458476	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TEND	1-Aug-11	NULL	0.1092771513750145	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.039390601	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TEND	1-Aug-11	NULL	0.8468979231563629	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TEND	1-Aug-11	NULL	1.640864726115453	EPINASTINE	rxcui:39684	EPINASTINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.054695491	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.8607814956671229	ETHYNODIOL DIACETATE	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.1408971500063358	ERGOLOID MESYLATE	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
UNIPROT:Q14500	hgnc:6258	KCNJ12	TEND	1-Aug-11	NULL	8.078103267029924	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1436598392221464	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.145753425	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
NOD2	hgnc:5331	NOD2	DTC	9/2/20	NULL	0.3409589041278864	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.067839369	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TEND	1-Aug-11	NULL	0.1875273972703375	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	1.334940794127826	FOSINOPRIL	rxcui:50166	FOSINOPRIL	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1505380482674727	HYDROCODONE	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.046221542	HYDROCODONE	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.4817217544559128	ALFENTANIL	rxcui:203203	ALFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.066297565	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW832467X	chembl:CHEMBL188247	GW832467X	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	DTC	9/2/20	NULL	0.3271505995993426	IOBENGUANE	ncit:C87757	IOBENGUANE	FALSE	FALSE	FALSE
UNIPROT:Q08499	hgnc:8783	PDE4D	TEND	1-Aug-11	NULL	0.5357925636295358	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.3211478363039418	LEVALLORPHAN	rxcui:6370	LEVALLORPHAN	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TEND	1-Aug-11	NULL	0.074690855	LISURIDE	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.032769506	LISURIDE	rxcui:6446	LISURIDE	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.8334550989792776	METOCURINE IODIDE	rxcui:203206	METOCURINE IODIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.048083948	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.052090944	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.048618214	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TEND	1-Aug-11	NULL	0.9723642821424908	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TEND	1-Aug-11	NULL	0.09745299	NANDROLONE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.3889457128569962	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.078136416	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.085239726	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.4070362111294147	PROGABIDE	rxcui:34568	PROGABIDE	FALSE	FALSE	FALSE
UNIPROT:P60880	hgnc:11132	SNAP25	TEND	1-Aug-11	NULL	17.50255707856483	BOTULINUM TOXIN TYPE A	rxcui:1000104	INCOBOTULINUMTOXINA	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1193356164447602	SERTRALINE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.010024374	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
UNIPROT:P27487	hgnc:3009	DPP4	TEND	1-Aug-11	NULL	0.630092055	SITAGLIPTIN	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
UNIPROT:P27338	hgnc:6834	MAOB	TEND	1-Aug-11	NULL	0.7740688634254718	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	NULL	TZP-202	NULL	NULL	NULL	NULL	NULL
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.051680779	GW3965	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
E2F TRANSCRIPTION FACTOR 1	hgnc:3113	E2F1	TTD	2020.06.01	NULL	NULL	ARQ-171	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	NULL	AP-761	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	SEP-228432	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	NULL	ERB-257	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Lu-AE04621	NULL	NULL	NULL	NULL	NULL
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FENCHLORAZOL-ETHYL	chembl:CHEMBL2229892	FENCHLORAZOL-ETHYL	FALSE	FALSE	FALSE
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	NULL	ND-0801	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tipelukast	ncit:C74581	TIPELUKAST	FALSE	FALSE	FALSE
PANCREATIC TRIACYLGLYCEROL LIPASE	hgnc:9155	PNLIP	TTD	2020.06.01	NULL	2.187819634820604	Liprotamase	chembl:CHEMBL2108703	LIPROTAMASE	FALSE	FALSE	FALSE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	B-cell lymphoma vaccine	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	IODOMELATONIN	drugbank:DB08190	N-[2-(2-IODO-5-METHOXY-1H-INDOL-3-YL)ETHYL]ACETAMIDE	FALSE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	HuM-195-Ac-225	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-V/BETA-3	NULL	NULL	TTD	2020.06.01	NULL	NULL	VLTS-589	drugbank:DB05430	VLTS-589	FALSE	FALSE	FALSE
ION CHANNEL UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lu-AA39959	NULL	NULL	NULL	NULL	NULL
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	NULL	PF-2413873	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	Hepapoietin	NULL	NULL	NULL	NULL	NULL
CARBOXYPEPTIDASE B2	hgnc:2300	CPB2	TTD	2020.06.01	NULL	NULL	SAR-104772	NULL	NULL	NULL	NULL	NULL
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	8.078103267029922	MDX-1203	ncit:C84855	ANTI-CD70 ANTIBODY-DRUG CONJUGATE MDX-1203	FALSE	FALSE	FALSE
VASOPRESSIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BR6819	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL O-ACYLTRANSFERASE 2	hgnc:16940	DGAT2	TTD	2020.06.01	NULL	NULL	PF-06427878	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	REC-01	NULL	NULL	NULL	NULL	NULL
TRAIL RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABBV-621	ncit:C146854	EFTOZANERMIN ALFA	FALSE	FALSE	FALSE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	7.501095891	Ralinepag	ncit:C152148	RALINEPAG	FALSE	FALSE	FALSE
EGFR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AC0010	ncit:C147125	ABIVERTINIB	FALSE	FALSE	FALSE
INHIBITOR OF APOPTOSIS PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	APG-1387	drugbank:DB16095	APG-1387	FALSE	FALSE	FALSE
POSITIVE TRANSCRIPTION ELONGATION FACTOR B	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY1251152	ncit:C128266	ENITOCICLIB	FALSE	FALSE	FALSE
MUTATED OXALOSUCCINATE DECARBOXYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY1436032	chembl:CHEMBL4206033	BAY1436032	FALSE	FALSE	FALSE
S-ADENOSYLMETHIONINE SYNTHASE TYPE-2	hgnc:6904	MAT2A	TTD	2020.06.01	NULL	52.50767123569449	AG-270	chembl:CHEMBL4802164	AG-270	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	DFP 13318	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	MENTHOFURAN	chembl:CHEMBL1522900	MENTHOFURAN	FALSE	FALSE	FALSE
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	8.751278539282415	CC-90011	iuphar.ligand:11284	CC-90011	FALSE	FALSE	FALSE
RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	LXH254	chembl:CHEMBL4583691	LXH254	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	0.6105543166941221	KA2507	iuphar.ligand:12269	KA2507	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.364636606	M2698	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-06873600	ncit:C151988	EBVACICLIB	FALSE	FALSE	FALSE
GERANYLGERANYL TRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PTX-100	drugbank:DB18125	PTX-100	FALSE	FALSE	FALSE
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	RGX-104	ncit:C131910	ABEQUOLIXRON	FALSE	FALSE	FALSE
DNA SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAR-200	ncit:C150807	GEMCITABINE-RELEASING INTRAVESICAL SYSTEM	FALSE	FALSE	FALSE
ANGIOGENESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRX-818	ncit:C123824	FOSLINANIB	FALSE	FALSE	FALSE
FGFR4 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	FGF401	chembl:CHEMBL3545293	FGF401	FALSE	FALSE	FALSE
MAMMALIAN TARGET OF RAPAMYCIN COMPLEX 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD2014	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
TARGET OF RAPAMYCIN COMPLEX 2 MAPKAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD2014	ncit:C88329	VISTUSERTIB	FALSE	FALSE	TRUE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	BGB-3112	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PHOSPHATIDYLINOSITOL-3-PHOSPHATE 5-KINASE	hgnc:23785	PIKFYVE	TTD	2020.06.01	NULL	52.50767123569449	Apilimod dimesylate	ncit:C90809	APILIMOD MESYLATE	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	NULL	PTX-200	NULL	NULL	NULL	NULL	NULL
FREE RADICAL	NULL	NULL	TTD	2020.06.01	NULL	NULL	SM-88	ncit:C74152	RACEMETYROSINE	FALSE	FALSE	FALSE
DNA REPLICATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAS-109	chembl:CHEMBL337450	TAS-109	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	FLX-787	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	1.514644363	APD371	ncit:C166825	OLORINAB	FALSE	FALSE	FALSE
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	0.9053046764774912	SEP-363856	drugbank:DB15665	SEP-363856	FALSE	FALSE	FALSE
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	NULL	852	NULL	NULL	NULL	NULL	NULL
NUCLEAR RECEPTOR ROR-GAMMA	hgnc:10260	RORC	TTD	2020.06.01	NULL	NULL	BBI-6000	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ruxolitinib cream	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ruxolitinib cream	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	ATI-502 topical	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	INCB54707	NULL	NULL	NULL	NULL	NULL
HEDGEHOG SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	Patidegib	ncit:C80063	PATIDEGIB	FALSE	FALSE	TRUE
ARYL HYDROCARBON RECEPTOR	hgnc:348	AHR	TTD	2020.06.01	NULL	NULL	RVT-505	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	IBI-20089	NULL	NULL	NULL	NULL	NULL
PROTEIN-TYROSINE PHOSPHATASE 1B	hgnc:9642	PTPN1	TTD	2020.06.01	NULL	NULL	KQ-791	NULL	NULL	NULL	NULL	NULL
GASTRIC INHIBITORY POLYPEPTIDE RECEPTOR	hgnc:4271	GIPR	TTD	2020.06.01	NULL	NULL	SAR438335	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	SAR438335	NULL	NULL	NULL	NULL	NULL
GLUCAGON	hgnc:4191	GCG	TTD	2020.06.01	NULL	NULL	ZP2929	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	NULL	Galnobax	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	IONIS-GCGRRX	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	0.6364566210387211	Efpeglenatide	ncit:C166682	EFPEGLENATIDE	FALSE	FALSE	FALSE
CASPASE-1	hgnc:1499	CASP1	TTD	2020.06.01	NULL	0.2243917574174978	AC-201	rxcui:22759	DIACETYLRHEIN	TRUE	FALSE	FALSE
INTERLEUKIN-22	hgnc:14900	IL22	TTD	2020.06.01	NULL	26.25383561784724	RG7880	ncit:C174771	EFMARODOCOKIN ALFA	FALSE	FALSE	FALSE
SLC5A2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bexagliflozin	rxcui:2627044	BEXAGLIFLOZIN	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	NBXT-001+Nobilis inhalation device	NULL	NULL	NULL	NULL	NULL
ACETOACETYL-COA THIOLASE	hgnc:93	ACAT1	TTD	2020.06.01	NULL	NULL	ATR-01	NULL	NULL	NULL	NULL	NULL
MUTATED TYROSINE-PROTEIN KINASE KIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	BLU-285	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
MAMMALIAN TARGET OF RAPAMYCIN COMPLEX 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
TARGET OF RAPAMYCIN COMPLEX 2 MAPKAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.8468979231563628	TCMDC-125548	chembl:CHEMBL528045	CHEMBL:CHEMBL528045	FALSE	FALSE	FALSE
RYANODINE RECEPTOR	hgnc:10483	RYR1	TTD	2020.06.01	NULL	3.750547945	ARM210	chembl:CHEMBL4594418	ARM-210	FALSE	FALSE	FALSE
FARNESYL PROTEIN TRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GGTI-2418	chembl:CHEMBL3218390	GGTI-2418	FALSE	FALSE	FALSE
BCL-2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PNT-2258	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PUR0200	NULL	NULL	NULL	NULL	NULL
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	GSK-2130579A	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE	NULL	NULL	TTD	2020.06.01	NULL	NULL	IPL 550,260	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AD-529	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	DA-727	chembl:CHEMBL41194	PRATOSARTAN	FALSE	FALSE	FALSE
MUCIN	hgnc:7515	MUC5AC	TTD	2020.06.01	NULL	NULL	KLS-0611	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	AC-262271	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	NULL	AMT-060	NULL	NULL	NULL	NULL	NULL
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	NULL	K-828-AB	NULL	NULL	NULL	NULL	NULL
UBIQUITIN-PROTEIN LIGASE E3 MDM2	hgnc:6973	MDM2	TTD	2020.06.01	NULL	NULL	RG7775	NULL	NULL	NULL	NULL	NULL
APOPTOSIS MEDIATING SURFACE ANTIGEN FAS	hgnc:11920	FAS	TTD	2020.06.01	NULL	NULL	DE-098	NULL	NULL	NULL	NULL	NULL
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BIT225	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	NULL	DV-1179	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	DV-1179	NULL	NULL	NULL	NULL	NULL
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
CHOLESTEROL SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	ETC-1002	rxcui:2282403	BEMPEDOIC ACID	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	TGWOOAA	NULL	NULL	NULL	NULL	NULL
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	TGWOOAA	NULL	NULL	NULL	NULL	NULL
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	TGOF02N	NULL	NULL	NULL	NULL	NULL
BETA-ADRENERGIC RECEPTOR KINASE 1	hgnc:289	GRK2	TTD	2020.06.01	NULL	NULL	BDBM50173306	NULL	NULL	NULL	NULL	NULL
ACTIVIN RECEPTOR TYPE IB	hgnc:172	ACVR1B	TTD	2020.06.01	NULL	NULL	US10030004, Compound 11a	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US10034861, Example 164	NULL	NULL	NULL	NULL	NULL
INTEGRIN BETA-8	hgnc:6163	ITGB8	TTD	2020.06.01	NULL	NULL	US10035778, Example 1	NULL	NULL	NULL	NULL	NULL
INTEGRIN BETA-8	hgnc:6163	ITGB8	TTD	2020.06.01	NULL	NULL	US10035778, Example 16	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	BDBM50158794	NULL	NULL	NULL	NULL	NULL
LEUCYL-CYSTEINYL AMINOPEPTIDASE	hgnc:6656	LNPEP	TTD	2020.06.01	NULL	NULL	US10059720, Example 80	NULL	NULL	NULL	NULL	NULL
LEUCYL-CYSTEINYL AMINOPEPTIDASE	hgnc:6656	LNPEP	TTD	2020.06.01	NULL	NULL	US10059720, Example 82	NULL	NULL	NULL	NULL	NULL
CYTOMEGALOVIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Adefovir	rxcui:16521	ADEFOVIR	TRUE	FALSE	FALSE
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US9434727, 93	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10087167, Compound 4001	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10149841, Compound 1	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US10149841, Compound 9	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10150740, Example 1	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9522888, 412	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	US10174026, Example 2	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US10179791, Compound 171	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US10179791, Compound 176	NULL	NULL	NULL	NULL	NULL
UBIQUITIN-ACTIVATING ENZYME E1	NULL	NULL	TTD	2020.06.01	NULL	NULL	QCPOIDRINIAUKU-SRBBEKPSSA-N	NULL	NULL	NULL	NULL	NULL
UBIQUITIN-ACTIVATING ENZYME E1	NULL	NULL	TTD	2020.06.01	NULL	NULL	SCHEMBL15198146	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL-PEPTIDASE 7	hgnc:14892	DPP7	TTD	2020.06.01	NULL	NULL	US8470836, 5	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8481586, 40	NULL	NULL	NULL	NULL	NULL
ACTIVATED CDC42 KINASE 1	hgnc:19297	TNK2	TTD	2020.06.01	NULL	NULL	US8481733, 95	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US8524917, 60	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US8524917, 12	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US8563594, 152	NULL	NULL	NULL	NULL	NULL
SUPPRESSOR OF TUMORIGENICITY 14 PROTEIN	hgnc:11344	ST14	TTD	2020.06.01	NULL	NULL	US8569313, Inhibitor 14	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 2	hgnc:3169	S1PR2	TTD	2020.06.01	NULL	NULL	US8975409, Comparative compound B	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8987457, 117	NULL	NULL	NULL	NULL	NULL
ENDOPLASMIC RETICULUM TO NUCLEUS SIGNALING 1	hgnc:3449	ERN1	TTD	2020.06.01	NULL	NULL	US9040714, 155	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE D1	hgnc:9067	PLD1	TTD	2020.06.01	NULL	NULL	US9127005, P0L	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE D1	hgnc:9067	PLD1	TTD	2020.06.01	NULL	NULL	US9127005, P2C	NULL	NULL	NULL	NULL	NULL
PC4 AND SFRS1-INTERACTING PROTEIN	hgnc:9527	PSIP1	TTD	2020.06.01	NULL	NULL	US9132129, Cpd002	NULL	NULL	NULL	NULL	NULL
PC4 AND SFRS1-INTERACTING PROTEIN	hgnc:9527	PSIP1	TTD	2020.06.01	NULL	NULL	US9132129, Cpd047	NULL	NULL	NULL	NULL	NULL
DISCOIDIN DOMAIN-CONTAINING RECEPTOR 2	hgnc:2731	DDR2	TTD	2020.06.01	NULL	NULL	US9156852, 38	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	B7673	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9181182, 34	NULL	NULL	NULL	NULL	NULL
SERINE PROTEASE HEPSIN	hgnc:5155	HPN	TTD	2020.06.01	NULL	NULL	AC1LFXA6	NULL	NULL	NULL	NULL	NULL
PLASMODIUM HYPOXANTHINE-GUANINE PHOSPHORIBOSYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9200020, Table 3, Compound 1B	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9216972, 61	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9216972, 67	NULL	NULL	NULL	NULL	NULL
DIBASIC-PROCESSING ENZYME	hgnc:8568	FURIN	TTD	2020.06.01	NULL	NULL	US9266828, B	NULL	NULL	NULL	NULL	NULL
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE CSK	hgnc:2444	CSK	TTD	2020.06.01	NULL	NULL	936563-93-8	NULL	NULL	NULL	NULL	NULL
PLASMODIUM PLASMEPSIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9353089, 327	NULL	NULL	NULL	NULL	NULL
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	3.621218705909965	ALTISSIMACOUMARIN E	chembl:CHEMBL2071527	ALTISSIMACOUMARIN E	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	US9359293, TM	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN-2	hgnc:10886	SIRT2	TTD	2020.06.01	NULL	NULL	BDBM50363782	NULL	NULL	NULL	NULL	NULL
SCN1A MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9694002, 495	NULL	NULL	NULL	NULL	NULL
SCN1A MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9694002, 59	NULL	NULL	NULL	NULL	NULL
SRSF PROTEIN KINASE 1	hgnc:11305	SRPK1	TTD	2020.06.01	NULL	NULL	Sphinx	NULL	NULL	NULL	NULL	NULL
SRSF PROTEIN KINASE 1	hgnc:11305	SRPK1	TTD	2020.06.01	NULL	NULL	SPHINX scaffold, 3	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004961042	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8921389, 2	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8921389, 210	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9340511, 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	BDBM50158791	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	NCGC00381656-01	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	3-(6-allyloxy-2-naphthyl)-1-(4-piperidylmethyl)pyrazolo[3,4-d]pyrimidin-4-amine	NULL	NULL	NULL	NULL	NULL
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.015407181	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE ALPHA-6	NULL	NULL	TTD	2020.06.01	NULL	NULL	CID 138805970	NULL	NULL	NULL	NULL	NULL
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.3684748858645227	CHRYSOERIOL	drugbank:DB17283	CHRYSOERIOL	FALSE	FALSE	FALSE
CYTOMEGALOVIRUS GLYCOPROTEIN B	NULL	NULL	TTD	2020.06.01	NULL	NULL	CMV glycoprotein B subunit vaccine	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003720782	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
JAK-STAT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	WP-1066	drugbank:DB12679	WP-1066	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.7095631248066824	Apadenoson	ncit:C74246	APADENOSON	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.004645052	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.2333674277141978	Pracinostat	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
GLUCOSE-DEPENDENT INSULINOTROPIC RECEPTOR	hgnc:19060	GPR119	TTD	2020.06.01	NULL	NULL	Guanfacine extended release	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	DM-99	NULL	NULL	NULL	NULL	NULL
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pacritinib	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	HM-5016504	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	RG3638	NULL	NULL	NULL	NULL	NULL
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	NULL	HPP-607	NULL	NULL	NULL	NULL	NULL
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.050781113	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	NULL	HPP-607	NULL	NULL	NULL	NULL	NULL
AURORA KINASE C	hgnc:11391	AURKC	TTD	2020.06.01	NULL	NULL	HPP-607	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE CHK2	hgnc:16627	CHEK2	TTD	2020.06.01	NULL	NULL	E7850	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.5147810905460245	ACP-319	ncit:C95891	PI3K-DELTA INHIBITOR AMG 319	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	NULL	P-7170	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	VBY- 891	NULL	NULL	NULL	NULL	NULL
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	2-PYRIDYLKETONE BENZOYL HYDRAZONE	chembl:CHEMBL252151	CHEMBL:CHEMBL252151	FALSE	FALSE	FALSE
INSULIN-DEGRADING ENZYME	hgnc:5381	IDE	TTD	2020.06.01	NULL	NULL	PRO-001	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	AAB-003/PF-05236812	NULL	NULL	NULL	NULL	NULL
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	MER-5101	NULL	NULL	NULL	NULL	NULL
PROSTATE SPECIFIC ANTIGEN	hgnc:6364	KLK3	TTD	2020.06.01	NULL	0.8751278539282416	ADXS-PSA	ncit:C120103	LISTERIA MONOCYTOGENES-LLO-PSA VACCINE ADXS31-142	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	NN-818	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	CM3.1-AC100	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	GSK2661380	NULL	NULL	NULL	NULL	NULL
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	NULL	ADMVA	NULL	NULL	NULL	NULL	NULL
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1562728310586145	DNDI1417560	chembl:CHEMBL1373255	CHEMBL:CHEMBL1373255	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	MK-3328	NULL	NULL	NULL	NULL	NULL
BOMBESIN RECEPTOR	hgnc:1058	BLM	TTD	2020.06.01	NULL	NULL	Demobesin	NULL	NULL	NULL	NULL	NULL
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	0.252440727	AM-251	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	Nerenone	NULL	NULL	NULL	NULL	NULL
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.029443554	Raloxifene	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydrotestosterone	ncit:C29619	DIHYDROTESTOSTERONE	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	MCT-125	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	NULL	ST-1141	NULL	NULL	NULL	NULL	NULL
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.03292017	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
BACTERIAL PROTECTIVE ANTIGEN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Valortim	chembl:CHEMBL2109304	MDX-1303	FALSE	FALSE	FALSE
GLUCOSE METABOLISM	NULL	NULL	TTD	2020.06.01	NULL	NULL	INS-1	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	NULL	AVN 211	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004829624	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	TNF alpha kinoid	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	EVT 401	NULL	NULL	NULL	NULL	NULL
APOB MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TKM-ApoB	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	SAR-21609	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP120	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-821385	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.004684003	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	NULL	11C-AZD-2184	NULL	NULL	NULL	NULL	NULL
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ARRY-162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
SCLEROSTIN	hgnc:13771	SOST	TTD	2020.06.01	NULL	NULL	AMG 167	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	ON-01135	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	CNSB-001	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	DIPHENHYDRAMINE	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	APD-209	NULL	NULL	NULL	NULL	NULL
GROWTH/DIFFERENTIATION FACTOR 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Stamulumab	ncit:C95795	STAMULUMAB	FALSE	FALSE	FALSE
GROWTH/DIFFERENTIATION FACTOR 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	LY2495655	ncit:C99640	LANDOGROZUMAB	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	EXO-230	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	ATryn antithrombin	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	DERRUBONE	chembl:CHEMBL412010	DERRUBONE	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	NULL	CM2489	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	THVD-201	NULL	NULL	NULL	NULL	NULL
CONNECTIVE TISSUE GROWTH FACTOR	hgnc:2500	CCN2	TTD	2020.06.01	NULL	NULL	RXI-109	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mibampator	ncit:C174617	MIBAMPATOR	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.043629141	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 40 MEMBER 1	hgnc:10909	SLC40A1	TTD	2020.06.01	NULL	NULL	Ferroportin mab	NULL	NULL	NULL	NULL	NULL
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
TAU PROTEIN AGGREGATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	LMT-X	NULL	NULL	NULL	NULL	NULL
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.043109746	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	LFG-316	ncit:C129315	TESIDOLUMAB	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	BETULINIC ACID	ncit:C38126	BETULINIC ACID	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acriflavine	rxcui:249	ACRIFLAVINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
T(H2) CYTOKINE PRODUCTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Suplatast tosilate	ncit:C152475	SUPLATAST TOSILATE	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	NULL	S-2150	NULL	NULL	NULL	NULL	NULL
PLATELET GLYCOPROTEIN IB ALPHA	hgnc:4439	GP1BA	TTD	2020.06.01	NULL	NULL	TGX-6B4	NULL	NULL	NULL	NULL	NULL
DYRK1B	hgnc:3092	DYRK1B	DTC	9/2/20	NULL	0.040452751	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	111In-hEGF	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV1.5	hgnc:6224	KCNA5	TTD	2020.06.01	NULL	NULL	IQB-9302	NULL	NULL	NULL	NULL	NULL
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	0.024309107	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PMN APOPTOSIS AND CHEMOTAXIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Synthetic neutrophil inhibitor peptide	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.021805511	Sodium chloride	rxcui:9863	SODIUM CHLORIDE	TRUE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	0.760980743	APOMINE	ncit:C1873	APOMINE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.008562895	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
STRESS-ACTIVATED PROTEIN KINASE 2B	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-745	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Suprofen	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	Bevacizumab + Trastuzumab	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	TRYPTAMINE	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006967578	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.4321619031744403	Pravastatin	rxcui:203144	PRAVASTATIN SODIUM	TRUE	FALSE	FALSE
STERYL-SULFATASE	hgnc:11425	STS	TTD	2020.06.01	NULL	0.3182283105193606	Tranilast	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	EMD 55900	ncit:C2714	ANTI-EGFR MONOCLONAL ANTIBODY EMD 55900	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004972317	FLUPHENAZINE HYDROCHLORIDE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.4150804050252529	Quinagolide	rxcui:76887	QUINAGOLIDE	FALSE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	CNI-1493	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Insulin Lyspro recombinant	NULL	NULL	NULL	NULL	NULL
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	Insulin recombinant	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	NULL	PDC-41	NULL	NULL	NULL	NULL	NULL
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.2586584789935689	NAPHAZOLINE HYDROCHLORIDE	rxcui:82054	NAPHAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.073643298	Riluzole	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	DLX-105	NULL	NULL	NULL	NULL	NULL
TRYPANOSOMA TRYPANOTHIONE REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bivalirudin	rxcui:60819	BIVALIRUDIN	TRUE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	NULL	NCX-1015	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	MUC-1 dendritic cancer vaccine	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mozavaptan	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.2465148884304905	IDAZOXAN HYDROCHLORIDE	chembl:CHEMBL543467	IDAZOXAN HYDROCHLORIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009115915	DOXAZOSIN MESYLATE	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.2	hgnc:6256	KCNJ10	TTD	2020.06.01	NULL	3.750547945	Glycodiazine	rxcui:102848	GLYMIDINE	FALSE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ketanserin	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	Thiopilocarpine	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR RECEPTOR TYPE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVX-470	drugbank:DB18455	AVX-470	FALSE	FALSE	FALSE
GABA TRANSPORTER GAT-1	hgnc:11042	SLC6A1	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.055271233	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperacillin	rxcui:1546000	PIPERACILLIN ANHYDROUS	TRUE	FALSE	FALSE
SODIUM/POTASSIUM-TRANSPORTING ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Digoxin	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	NULL	E-4716	NULL	NULL	NULL	NULL	NULL
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tioconazole	rxcui:38298	TIOCONAZOLE	TRUE	FALSE	FALSE
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	5-hydroxymethyl-2-furfural (sickle cell disease), AesRx LLC	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	GUAIFENESIN	rxcui:5032	GUAIFENESIN	TRUE	FALSE	FALSE
CHARYBDOTOXIN RECEPTOR BETA-4	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-223131	chembl:CHEMBL222460	BMS-223131	FALSE	FALSE	FALSE
PLG	hgnc:9071	PLG	DTC	9/2/20	NULL	2.500365296937833	RADIOSUMIN B	chembl:CHEMBL478092	RADIOSUMIN B	FALSE	FALSE	FALSE
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	Synthetic hypericin	ncit:C122400	SYNTHETIC HYPERICIN	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Apratastat	ncit:C76767	APRATASTAT	FALSE	FALSE	FALSE
SODIUM/POTASSIUM-TRANSPORTING ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rostafuroxin	ncit:C90733	ROSTAFUROXIN	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PPL-100	drugbank:DB05961	PPL-100	FALSE	FALSE	FALSE
THROMBOPOIETIN RECEPTOR	hgnc:7217	MPL	TTD	2020.06.01	NULL	NULL	NIP-004	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	0.3365876361262467	R-flurbiprofen	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR	hgnc:18284	RAB40B	TTD	2020.06.01	NULL	NULL	Velac Gel	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	NULL	IC-485	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Otilonium bromide	rxcui:54216	OTILONIUM BROMIDE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.212581665	GNF-PF-211	chembl:CHEMBL582699	CHEMBL:CHEMBL582699	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dextofisopam	ncit:C76460	DEXTOFISOPAM	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	GTP-010	NULL	NULL	NULL	NULL	NULL
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	NULL	ATI-17000	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	NULL	EP-51216	NULL	NULL	NULL	NULL	NULL
BRDT	hgnc:1105	BRDT	DTC	9/2/20	NULL	0.2273059360852576	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
ESTROGEN-RELATED RECEPTOR-ALPHA	hgnc:3471	ESRRA	TTD	2020.06.01	NULL	4.375639269641208	Pregnenolone	rxcui:114052	PREGNENOLONE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Mebeverine	rxcui:29410	MEBEVERINE	FALSE	FALSE	FALSE
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	NULL	EP-51389	NULL	NULL	NULL	NULL	NULL
PTH1R	hgnc:9608	PTH1R	DTC	9/2/20	NULL	3.750547945	TCMDC-123778	chembl:CHEMBL586870	CHEMBL:CHEMBL586870	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 1	hgnc:4584	GRIN1	TTD	2020.06.01	NULL	NULL	H-Gly-PMe-Glu-OH	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2A	hgnc:4585	GRIN2A	TTD	2020.06.01	NULL	NULL	H-Gly-PMe-Glu-OH	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	NULL	H-Gly-PMe-Glu-OH	NULL	NULL	NULL	NULL	NULL
SUPEROXIDE ANION	hgnc:10798	SFTPA1	TTD	2020.06.01	NULL	NULL	OPC-14117	NULL	NULL	NULL	NULL	NULL
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.00809055	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
CALCIUM-ACTIVATED POTASSIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Charybdotoxin	iuphar.ligand:2328	CHARYBDOTOXIN	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	CO-101	chembl:CHEMBL3039516	GEMCITABINE ELAIDATE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclacillin	rxcui:2968	CYCLACILLIN	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pivampicillin	rxcui:8372	PIVAMPICILLIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	2,4-DIACETYL PHLOROGLUCINOL	chembl:CHEMBL276139	2,4-DIACETYLPHLOROGLUCINOL	FALSE	FALSE	FALSE
INTEGRIN ALPHA-5/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-alpha5Beta1-integrin antibody	drugbank:DB05870	ANTI-ALPHA5BETA1-INTEGRIN ANTIBODY	FALSE	FALSE	FALSE
INTEGRIN ALPHA-5/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Volociximab	ncit:C48426	VOLOCIXIMAB	FALSE	FALSE	TRUE
RIBOSOMAL PROTEIN S6 KINASE ALPHA-6	NULL	NULL	TTD	2020.06.01	NULL	NULL	BI-D1870	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	DERRUBONE	chembl:CHEMBL412010	DERRUBONE	FALSE	FALSE	FALSE
BACTERIAL LETHAL FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
LUTEINIZING HORMONE RECEPTOR	hgnc:6585	LHCGR	TTD	2020.06.01	NULL	NULL	ML-04	NULL	NULL	NULL	NULL	NULL
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.012015485	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
SODIUM/CALCIUM EXCHANGER	hgnc:10620	CCL21	TTD	2020.06.01	NULL	NULL	CALDARET HYDRATE	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	0.3070624048871023	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.1259176768242074	SKI-758	chembl:CHEMBL219557	CHEMBL:CHEMBL219557	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DNDI1416975	chembl:CHEMBL1415851	CHEMBL:CHEMBL1415851	FALSE	FALSE	FALSE
MUCOSAL ADDRESSIN CELL ADHESION MOLECULE 1	hgnc:6765	MADCAM1	TTD	2020.06.01	NULL	3.500511415712967	SCH-527123	iuphar.ligand:8497	NAVARIXIN	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.8	hgnc:10582	SCN10A	TTD	2020.06.01	NULL	0.2302968036653267	Tiapride	rxcui:10588	TIAPRIDE	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.1290114772375786	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	SKF-105809	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Halothane	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clofarabine	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	NULL	Guanfacine extended release	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE PROTEINASE-3	hgnc:9495	PRTN3	TTD	2020.06.01	NULL	NULL	Combined PR1/WT1 vaccine	NULL	NULL	NULL	NULL	NULL
WILMS TUMOR PROTEIN	hgnc:12796	WT1	TTD	2020.06.01	NULL	NULL	Combined PR1/WT1 vaccine	NULL	NULL	NULL	NULL	NULL
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	ETHYL VANILLIN	rxcui:1311571	ETHYL VANILLIN	TRUE	FALSE	FALSE
G-PROTEIN COUPLED RECEPTOR 55	hgnc:4511	GPR55	TTD	2020.06.01	NULL	NULL	Guanfacine extended release	NULL	NULL	NULL	NULL	NULL
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	DESMOSDUMOTIN C	chembl:CHEMBL53628	DESMOSDUMOTIN C	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	SC-75416	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	SB-639	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	SB-623	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.081407242	Butalbital	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.028444026	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
FACTOR XI MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	alpha-ketothiazole analogue 36	iuphar.ligand:6549	ALPHA-KETOTHIAZOLE ANALOGUE 36	FALSE	FALSE	FALSE
LEUKOTRIENE B4 RECEPTOR 1	hgnc:6713	LTB4R	TTD	2020.06.01	NULL	NULL	LTB 019	NULL	NULL	NULL	NULL	NULL
ERBB2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	HKI-272	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
LIPASE UNSPECIFIC	hgnc:30045	SMG1	TTD	2020.06.01	NULL	NULL	ApoC-III	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clomocycline	rxcui:21272	CLOMOCYCLINE	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.1857035233799982	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	NULL	Artemisinin SP	NULL	NULL	NULL	NULL	NULL
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1	hgnc:2357	CRHR1	TTD	2020.06.01	NULL	2.917092846427472	Pexacerfont	ncit:C76508	PEXACERFONT	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Coluracetam	ncit:C77391	COLURACETAM	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.011850072	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
MITOCHONDRIAL 10KDA HEAT SHOCK PROTEIN	hgnc:5269	HSPE1	TTD	2020.06.01	NULL	NULL	XToll	NULL	NULL	NULL	NULL	NULL
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PACHYRRIZINE	chembl:CHEMBL479689	PACHYRRIZINE	FALSE	FALSE	FALSE
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	NULL	Bupropion+naltrexone	NULL	NULL	NULL	NULL	NULL
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	Bupropion+naltrexone	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.038159645	Etazolate	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.6250913242344582	MK-0873	drugbank:DB13029	MK-0873	FALSE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bupropion+naltrexone	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 2	hgnc:11848	TLR2	TTD	2020.06.01	NULL	NULL	MCS-18	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Guanfacine extended release	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-693571	chembl:CHEMBL1287983	CHEMBL:CHEMBL1287983	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenelzine	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Desoxypeganine	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Desoxypeganine	NULL	NULL	NULL	NULL	NULL
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.078136416	GNF-PF-3756	chembl:CHEMBL597035	CHEMBL:CHEMBL597035	FALSE	FALSE	FALSE
CATALASE	hgnc:1516	CAT	TTD	2020.06.01	NULL	NULL	EUK-189	NULL	NULL	NULL	NULL	NULL
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	EUK-189	NULL	NULL	NULL	NULL	NULL
CARBOXYPEPTIDASE B2	hgnc:2300	CPB2	TTD	2020.06.01	NULL	NULL	SAR-126119	NULL	NULL	NULL	NULL	NULL
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ecallantide	rxcui:658708	ECALLANTIDE	TRUE	FALSE	FALSE
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiamphenicol	rxcui:10463	THIAMPHENICOL	FALSE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Econazole	rxcui:142434	ECONAZOLE NITRATE	TRUE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	0.3029288725136221	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.2187819634820604	Trapidil	rxcui:10735	TRAPIDIL	FALSE	FALSE	FALSE
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Iron Dextran	rxcui:5992	IRON-DEXTRAN COMPLEX	TRUE	FALSE	FALSE
PARATHYROID HORMONE RECEPTOR	hgnc:9609	PTH2R	TTD	2020.06.01	NULL	NULL	PTH(7-34) liposomal cream	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lindane	rxcui:1388	LINDANE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.729273212	HMG-CoA reductase inhibitor	ncit:C1655	HMG-COA REDUCTASE INHIBITOR	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	0.084012274	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	V-24343	NULL	NULL	NULL	NULL	NULL
GAP JUNCTION PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Danegaptide	ncit:C83647	DANEGAPTIDE	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.145753425	Flunisolide	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Vinpocetine	rxcui:24506	VINPOCETINE	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	IMRECOXIB	drugbank:DB12354	IMRECOXIB	FALSE	FALSE	FALSE
INTERFERON-ALPHA 5	hgnc:5426	IFNA5	TTD	2020.06.01	NULL	NULL	NAHE-001	NULL	NULL	NULL	NULL	NULL
AURKA	hgnc:11393	AURKA	DTC	9/2/20	inhibitor	0.060956201	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
INTERFERON-OMEGA	hgnc:5448	IFNW1	TTD	2020.06.01	NULL	NULL	ITCA-638	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Amprenavir	rxcui:228656	AMPRENAVIR	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REV PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	ATI-0917	NULL	NULL	NULL	NULL	NULL
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pemetrexed	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
INTERLEUKIN 7 RECEPTOR ALPHA	hgnc:6024	IL7R	TTD	2020.06.01	NULL	NULL	CYT 99007	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	0.089298761	Albendazole	rxcui:430	ALBENDAZOLE	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MBX-2044	chembl:CHEMBL3545020	MBX-2044	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MBX-102	ncit:C83536	ARHALOFENATE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Didanosine	rxcui:3364	DIDANOSINE	TRUE	FALSE	FALSE
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Epalrestat	ncit:C72762	EPALRESTAT	FALSE	FALSE	FALSE
MEASLES VIRUS FUSION GLYCOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	TTP889	drugbank:DB05131	TTP889	FALSE	FALSE	FALSE
FATTY ACID SYNTHASE	hgnc:3594	FASN	TTD	2020.06.01	NULL	NULL	FAS1	NULL	NULL	NULL	NULL	NULL
FATTY ACID SYNTHASE	hgnc:3594	FASN	TTD	2020.06.01	NULL	NULL	FSA2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rasagiline	rxcui:134748	RASAGILINE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2A	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	NULL	Connexyn	NULL	NULL	NULL	NULL	NULL
INTERFERON ALPHA/BETA RECEPTOR 2	hgnc:5433	IFNAR2	TTD	2020.06.01	NULL	1.312691780892362	Interferon beta-1b	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.2273059360852575	AG-024322	ncit:C52182	CDK1/2/4 INHIBITOR AG-024322	FALSE	FALSE	FALSE
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	FX-107	NULL	NULL	NULL	NULL	NULL
FOLATE RECEPTOR ALPHA	hgnc:3791	FOLR1	TTD	2020.06.01	NULL	NULL	FolateImmune	NULL	NULL	NULL	NULL	NULL
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	1.270346884734544	Azatadine	rxcui:18600	AZATADINE	TRUE	FALSE	FALSE
VON WILLEBRAND FACTOR	hgnc:12726	VWF	TTD	2020.06.01	NULL	NULL	DA-697b	NULL	NULL	NULL	NULL	NULL
KINESIN SPINDLE MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	EMD-534085	chembl:CHEMBL1077204	CHEMBL:CHEMBL1077204	FALSE	FALSE	FALSE
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	3.500511415712966	LU AE58054	ncit:C166835	IDALOPIRDINE	FALSE	FALSE	FALSE
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	NULL	MK-6302	NULL	NULL	NULL	NULL	NULL
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	EcoNail	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-29	hgnc:18363	IFNL1	TTD	2020.06.01	NULL	NULL	PEG-Interferon lambda (IL-29)	NULL	NULL	NULL	NULL	NULL
CATECHOL-O-METHYL-TRANSFERASE	hgnc:2228	COMT	TTD	2020.06.01	NULL	NULL	PGX-200097	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PGX-200097	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE XIV	NULL	NULL	TTD	2020.06.01	NULL	NULL	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
CHYMOTRYPSIN	hgnc:1440	CALCR	TTD	2020.06.01	NULL	NULL	CM-AT	NULL	NULL	NULL	NULL	NULL
RETINAL PIGMENT EPITHELIUM PROTEIN	hgnc:10294	RPE65	TTD	2020.06.01	NULL	7.501095891	TgAAG76	drugbank:DB18421	TGAAG-76	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.5048814541893701	PHENOL	rxcui:33290	PHENOL	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	NULL	Neu-2000	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	BM-ca	NULL	NULL	NULL	NULL	NULL
POTASSIUM	NULL	NULL	TTD	2020.06.01	NULL	NULL	Patiromer calcium	chembl:CHEMBL2107840	PATIROMER CALCIUM	TRUE	FALSE	FALSE
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	0.1159109740302306	ALT-801	drugbank:DB15386	ALT-801	FALSE	FALSE	FALSE
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	5.250767123569449	SCH-721015	hemonc:111273	NADOFARAGENE FIRADENOVEC	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	NULL	GDC-0980/RG7422	NULL	NULL	NULL	NULL	NULL
MITOCHONDRIAL ALDEHYDE DEHYDROGENASE	hgnc:404	ALDH2	TTD	2020.06.01	NULL	NULL	ALD-401	NULL	NULL	NULL	NULL	NULL
PROSTATE STEM CELL ANTIGEN	hgnc:9500	PSCA	TTD	2020.06.01	NULL	NULL	Anti-PSCA mab	NULL	NULL	NULL	NULL	NULL
MYC MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-5126	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	APD-916	NULL	NULL	NULL	NULL	NULL
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	NULL	SPP-600	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAR-110894	NULL	NULL	NULL	NULL	NULL
FREE RADICAL	NULL	NULL	TTD	2020.06.01	NULL	NULL	RRx-001	drugbank:DB12060	RRX-001	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	NULL	MSDC-0602	NULL	NULL	NULL	NULL	NULL
ENDOSTATIN	hgnc:2195	COL18A1	TTD	2020.06.01	NULL	NULL	RetinoStat	NULL	NULL	NULL	NULL	NULL
PLASMINOGEN	hgnc:9071	PLG	TTD	2020.06.01	NULL	NULL	RetinoStat	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	OBP-601	chembl:CHEMBL124363	CENSAVUDINE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.3453256329104173	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	EP-101	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE	hgnc:4341	GLUL	TTD	2020.06.01	NULL	NULL	SPI-014	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS ENVELOPE GLYCOPROTEIN E2	NULL	NULL	TTD	2020.06.01	NULL	NULL	MBL-HCV1	drugbank:DB17776	MBL-HCV1	FALSE	FALSE	FALSE
ANGIOTENSINOGENASE RENIN	hgnc:9958	REN	TTD	2020.06.01	NULL	NULL	ACT-178882	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GAG PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bevirimat	ncit:C78044	BEVIRIMAT	FALSE	FALSE	FALSE
STAPHYLOCOCCUS ENOYL ACP REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AFN-1252	drugbank:DB12658	AFN-1252	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tiotropium	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
TOXIC METHOTREXATE	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	0.1339481409073839	Glucarpidase	rxcui:1242127	GLUCARPIDASE	TRUE	FALSE	FALSE
PROTEASOME	hgnc:9338	PRB2	TTD	2020.06.01	NULL	0.1250182648468916	Carfilzomib	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
UROKINASE-TYPE PLASMINOGEN ACTIVATOR	hgnc:9052	PLAU	TTD	2020.06.01	NULL	2.500365296937833	Upamostat	ncit:C73985	UPAMOSTAT	FALSE	FALSE	FALSE
GLUCOSYLCERAMIDASE	hgnc:4177	GBA1	TTD	2020.06.01	NULL	1.500219178	Taliglucerase alfa	rxcui:1291609	TALIGLUCERASE ALFA	TRUE	FALSE	FALSE
INDUCIBLE T-CELL COSTIMULATOR	hgnc:5351	ICOS	TTD	2020.06.01	NULL	35.00511415712966	MEDI-570	chembl:CHEMBL2109449	MEDI-570	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nafcillin	rxcui:7233	NAFCILLIN	TRUE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	AMG 747	NULL	NULL	NULL	NULL	NULL
FREE FATTY ACID RECEPTOR 1	hgnc:4498	FFAR1	TTD	2020.06.01	NULL	NULL	P-1736	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	I.V. carbamazepine	NULL	NULL	NULL	NULL	NULL
CYTOCHROME P450 3A	ncbigene:1574	CYP3A	TTD	2020.06.01	NULL	NULL	Cobicistat/darunavir	NULL	NULL	NULL	NULL	NULL
BONE MORPHOGENETIC PROTEIN 2	hgnc:1069	BMP2	TTD	2020.06.01	NULL	NULL	DWP-431	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	NS-018	chembl:CHEMBL3545217	NS-018	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMA-76	NULL	NULL	NULL	NULL	NULL
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	AZD-7009	NULL	NULL	NULL	NULL	NULL
GTPASE NRAS	hgnc:7989	NRAS	TTD	2020.06.01	NULL	NULL	Mutant ras vaccine	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	2.917092846427472	EPZ-6438	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	1.712206670729168	EVP-6124	ncit:C166844	ENCENICLINE	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,2,4,5-tetra-substituted imidazole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	1,2,4-triazole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 5	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Aminoazetidine derivative 8	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Azetidine-1-carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Azetidine-1-carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diphenyl purine derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diphenyl purine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Diphenyl purine derivative 5	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Furopyridine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Heterocyclic-substituted 3-alkyl azetidine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Imidazole derivative 4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	N-phenyl-5-phenyl-pyrazolin-3-yl amide derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 13	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 14	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 15	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 17	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 24	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 25	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 26	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 28	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 29	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 31	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 32	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 36	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 38	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 4	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 40	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 57	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 60	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 11	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 12	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 13	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrido[2,3-d]pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 3	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Sulfonylated piperazine derivative 5	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	AZD-9819	NULL	NULL	NULL	NULL	NULL
TISSUE FACTOR	hgnc:3541	F3	TTD	2020.06.01	NULL	NULL	TT-173	NULL	NULL	NULL	NULL	NULL
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	0.1657439117288336	BAY 80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	NULL	BMS-986189	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	1.280674908	LZM009	ncit:C153149	LIPUSTOBART	FALSE	FALSE	FALSE
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	0.5250767123569451	ARRY-162	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
T-CELL SURFACE GLYCOPROTEIN CD4	hgnc:1678	CD4	TTD	2020.06.01	NULL	3.281729452230906	Ibalizumab	rxcui:2043283	IBALIZUMAB	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	1.790034246671403	Enprofylline	ncit:C74327	ENPROFYLLINE	FALSE	FALSE	FALSE
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clevidipine butyrate	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	NULL	ABBV-2451	NULL	NULL	NULL	NULL	NULL
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	NULL	ABBV-2737	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	DSP-3905	NULL	NULL	NULL	NULL	NULL
SHORT TRANSIENT RECEPTOR POTENTIAL CHANNEL 4	hgnc:12336	TRPC4	TTD	2020.06.01	NULL	NULL	TRPC4 and TRPC5 inhibitor	NULL	NULL	NULL	NULL	NULL
SHORT TRANSIENT RECEPTOR POTENTIAL CHANNEL 5	hgnc:12337	TRPC5	TTD	2020.06.01	NULL	NULL	TRPC4 and TRPC5 inhibitor	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	NULL	PD-145065	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN B RECEPTOR	hgnc:3180	EDNRB	TTD	2020.06.01	NULL	NULL	PD-145065	NULL	NULL	NULL	NULL	NULL
ADENOSINE A2B RECEPTOR	hgnc:264	ADORA2B	TTD	2020.06.01	NULL	NULL	YT-146	NULL	NULL	NULL	NULL	NULL
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Turosteride	ncit:C99549	TUROSTERIDE	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ticarcillin	rxcui:10591	TICARCILLIN	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	TETRAPLATIN TETRANITRATE	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PT-302	chembl:CHEMBL253996	CHEMBL:CHEMBL253996	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Doxacurium	rxcui:23651	DOXACURIUM	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Brompheniramine	rxcui:1767	BROMPHENIRAMINE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	VEGF-2 gene therapy	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PT-112	ncit:C121375	IMIFOPLATIN	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Darifenacin	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Filibuvir	ncit:C83717	FILIBUVIR	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	TZTX-001	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PSI-938	chembl:CHEMBL2160007	PSI-352938	FALSE	FALSE	FALSE
ERYTHROPOIETIN	hgnc:3415	EPO	TTD	2020.06.01	NULL	NULL	Long-acting erythropoietin conjugate	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	T3D-959	chembl:CHEMBL3545176	DB959	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	GSK311739	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	QLT-091568	NULL	NULL	NULL	NULL	NULL
P53 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	OPI-1002	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Bevacizumab + Trastuzumab	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Bevacizumab + Trastuzumab	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	R1678	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	NULL	CCX872	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PPI-383	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-8	hgnc:7175	MMP8	TTD	2020.06.01	NULL	0.300043836	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
INTERLEUKIN-12 BETA	hgnc:5970	IL12B	TTD	2020.06.01	NULL	NULL	SFV IL-12 gene therapy	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	NULL	TZP-301	NULL	NULL	NULL	NULL	NULL
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	TVI-Kidney-1	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-916	NULL	NULL	NULL	NULL	NULL
IMMUNOGLOBULIN E	hgnc:5522	IGHE	TTD	2020.06.01	NULL	NULL	Xmab-7195	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	ZP2929	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	ZP2929	NULL	NULL	NULL	NULL	NULL
CORTICOSTEROID 11-BETA-DEHYDROGENASE 2	hgnc:5209	HSD11B2	TTD	2020.06.01	NULL	NULL	RG-7234	NULL	NULL	NULL	NULL	NULL
TENASCIN	hgnc:5318	TNC	TTD	2020.06.01	NULL	NULL	F-16-131I	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19- CAR	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Anti-CD20-CAR vector-transduced autologous T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	19-28z T CELLS	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	0.7095631248066824	MSC2363318A	ncit:C112004	P70S6K/AKT INHIBITOR M-2698	FALSE	FALSE	FALSE
CO-STIMULATORY MOLECULE 4-1BB	hgnc:11924	TNFRSF9	TTD	2020.06.01	NULL	NULL	CD28 and CD137 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19 CAR transduced T cells	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	CD33-specific gene-engineered T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-UCART	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD19/CD22 Chimeric Antigen Receptor T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19/CD22 Chimeric Antigen Receptor T Cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD22-specific CAR T-cells also expressing an EGFRt	NULL	NULL	NULL	NULL	NULL
PROSTATE STEM CELL ANTIGEN	hgnc:9500	PSCA	TTD	2020.06.01	NULL	NULL	CAR-T Cells targeting PSCA	NULL	NULL	NULL	NULL	NULL
MUCIN-1	hgnc:7508	MUC1	TTD	2020.06.01	NULL	NULL	CART-Muc1 cells	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	CAR-GPC3 T cell	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CAR-20/19-T Cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CAR-20/19-T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	ICAR19 CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 and CD20 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CD19 and CD20 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19-targeted CART cells	NULL	NULL	NULL	NULL	NULL
NKG2 D ACTIVATING NK RECEPTOR	hgnc:18788	KLRK1	TTD	2020.06.01	NULL	NULL	NKR-2 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CART-19/22	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART-19/22	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CART22-65s cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CART22-65s cells and huCART19 Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART22-65s cells and huCART19 Cells	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	CD123/CLL1 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
MYELOID INHIBITORY C-TYPE LECTIN-LIKE RECEPTOR	hgnc:31713	CLEC12A	TTD	2020.06.01	NULL	NULL	CD123/CLL1 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
MYELOID INHIBITORY C-TYPE LECTIN-LIKE RECEPTOR	hgnc:31713	CLEC12A	TTD	2020.06.01	NULL	NULL	CLL1 CAR-T Cell	NULL	NULL	NULL	NULL	NULL
TRAIL RECEPTOR 2	hgnc:11905	TNFRSF10B	TTD	2020.06.01	NULL	NULL	Anti-DR5 cells	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	NULL	C-Met/PD-L1 CAR-T Cell	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	NULL	C-Met/PD-L1 CAR-T Cell	NULL	NULL	NULL	NULL	NULL
T-CELL ANTIGEN CD7	hgnc:1695	CD7	TTD	2020.06.01	NULL	NULL	CD7.CAR/28zeta CAR T cells	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HER2-CAR T Cells	NULL	NULL	NULL	NULL	NULL
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.1544343271638073	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
SLAM FAMILY MEMBER 7 SLAMF7	hgnc:21394	SLAMF7	TTD	2020.06.01	NULL	NULL	CS1-CAR T Therapy	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	IM21 CART	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	Anti-BCMA CART Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19 CART Cells	NULL	NULL	NULL	NULL	NULL
MYCOBACTERIUM PROTON PUMP	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bedaquiline	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
BACTERIAL RNA POLYMERASE SWITCH REGION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fidaxomicin	rxcui:1111103	FIDAXOMICIN	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.026748686	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
5-HT RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nafronyl	rxcui:7236	NAFRONYL	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	NULL	Ovine corticotropin-releasing hormone	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TAK-137	chembl:CHEMBL4594501	TAK-137	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PIKAMILONE	NULL	NULL	NULL	NULL	NULL
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.027010119	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	0.1375060601009582	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.9460841664089098	Regadenoson	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
ENDOTHELIN A RECEPTOR	hgnc:3179	EDNRA	TTD	2020.06.01	NULL	2.282942227638891	Bosentan	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.2917092846427472	Bepridil	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.988926940746003	Abarelix	rxcui:301739	ABARELIX	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010093747	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	Anileridine Hydrochloride	rxcui:235413	ANILERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PROTEASOME	hgnc:9338	PRB2	TTD	2020.06.01	NULL	0.087222045	Bortezomib	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cortisone Acetate	rxcui:21655	CORTISONE ACETATE	TRUE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	1.193356164447602	Chlorphentermine Hydrochloride	ncit:C65324	CHLORPHENTERMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
INTERLEUKIN 2 RECEPTOR ALPHA	hgnc:6008	IL2RA	TTD	2020.06.01	NULL	NULL	RFT-5.dgA	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.1232574442152452	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
HAEMATIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ferroquine	ncit:C171721	FERROQUINE	FALSE	FALSE	FALSE
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	ABT-957	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.011906501	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	3.281729452230906	PIRITREXIM	ncit:C1031	PIRITREXIM	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	NSC-175743	chembl:CHEMBL1609016	CHEMBL:CHEMBL1609016	FALSE	FALSE	FALSE
VOLTAGE-DEPENDENT ANION-SELECTIVE CHANNEL 3	hgnc:12674	VDAC3	TTD	2020.06.01	NULL	NULL	PRLX93936	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	13-DEOXYADRIAMYCIN HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	13-DEOXYADRIAMYCIN HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	ACH-3102	chembl:CHEMBL3544977	ODALASVIR	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	CAP-7.1	NULL	NULL	NULL	NULL	NULL
PSEUDOMONAS PCRV PROTEIN TYPE III	NULL	NULL	TTD	2020.06.01	NULL	NULL	KB-001	chembl:CHEMBL2109536	KB-001	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	NHS-IL2-LT	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	ONO-5129	NULL	NULL	NULL	NULL	NULL
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	CID 650707	chembl:CHEMBL408653	CHEMBL:CHEMBL408653	FALSE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	0.900131507	MK-4827	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	0.2381300282797936	Phenoxodiol	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Doxorubicin-eluting beads	ncit:C82419	DOXORUBICIN-ELUTING BEADS	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	DDP-225	drugbank:DB05642	DDP-225	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ONO-5129	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PPI-668	chembl:CHEMBL3545312	RAVIDASVIR HYDROCHLORIDE	FALSE	FALSE	FALSE
CHLORIDE CHANNEL PROTEIN 2	hgnc:2020	CLCN2	TTD	2020.06.01	NULL	NULL	RK-023	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Dronabinol oral solution	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Dronabinol oral solution	NULL	NULL	NULL	NULL	NULL
HUMAN PAPILLOMAVIRUS PROTEIN E6	NULL	NULL	TTD	2020.06.01	NULL	NULL	VGX-3100	ncit:C77909	BIZALIMOGENE RALAPLASMID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
HUMAN PAPILLOMAVIRUS PROTEIN E7	NULL	NULL	TTD	2020.06.01	NULL	NULL	VGX-3100	ncit:C77909	BIZALIMOGENE RALAPLASMID	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BIIR-777	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.1131630845596864	Tirapazamine	ncit:C1464	TIRAPAZAMINE	FALSE	FALSE	FALSE
ATP-BINDING CASSETTE TRANSPORTER C8	hgnc:59	ABCC8	TTD	2020.06.01	NULL	1.750255707856483	Acetohexamide	rxcui:173	ACETOHEXAMIDE	TRUE	FALSE	FALSE
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	0.2333674277141978	BMN-673	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
MHC CLASS II ANTIGEN DR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Apolizumab	ncit:C2228	APOLIZUMAB	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.052090944	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alovudine	ncit:C65226	ALOVUDINE	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR B	hgnc:8800	PDGFB	TTD	2020.06.01	NULL	NULL	CR-002	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	NULL	PH-794428	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	TC-2216	chembl:CHEMBL504652	TC-2216	FALSE	FALSE	FALSE
BACTERIAL LETHAL FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IQ-DAA	NULL	NULL	NULL	NULL	NULL
BACTERIAL PROTECTIVE ANTIGEN	NULL	NULL	TTD	2020.06.01	NULL	NULL	IQ-DAA	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-5	hgnc:6016	IL5	TTD	2020.06.01	NULL	5.834185692854944	Mepolizumab	rxcui:1720597	MEPOLIZUMAB	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.03729238	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
CELL CYCLE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BZL-101	NULL	NULL	NULL	NULL	NULL
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Viquidacin	ncit:C152895	VIQUIDACIN	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	BGC-20-1259	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Melphalan	rxcui:6718	MELPHALAN	TRUE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	F-14512	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	TESAGLITAZAR	ncit:C75985	TESAGLITAZAR	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.1162317016838838	AZD0530	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Balaglitazone	ncit:C78125	BALAGLITAZONE	FALSE	FALSE	FALSE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2013059594(IV)	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	CGS-15943	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Heteroaryl-pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	N-substituted pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-10	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-20	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-20	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-45	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-47	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	PMID25435285-Compound-53	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 76	NULL	NULL	NULL	NULL	NULL
ME3	hgnc:6985	ME3	DTC	9/2/20	NULL	8.751278539282415	MALEIC ACID	rxcui:1426330	MALEIC ACID	TRUE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 79	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 6	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Tetra-hydro-imidazo[1,5-d][1,4]oxazepin-3-yl derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	Tetra-hydro-imidazo[1,5-d][1,4]oxazepin-3-yl derivative 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	2,2-bipyridyl derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	2,2-bipyridyl derivative 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	2,2-bipyridyl derivative 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hydroxamate analog 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hydroxamate analog 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	Hydroxyqunoline analog 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 5	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4E	hgnc:37098	KDM4E	TTD	2020.06.01	NULL	NULL	N-oxalyl-D-tyrosine derivative 6	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-50	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25468267-Compound-51	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridine-2,4-dicarboxylic acid derivative 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Pyrido[1,2-a]indole-1.-carboxylic acid analog 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Pyrido[1,2-a]indole-1.-carboxylic acid analog 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Pyrido[1,2-a]indole-1.-carboxylic acid analog 5	NULL	NULL	NULL	NULL	NULL
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1019566431761058	TCMDC-124585	chembl:CHEMBL587856	CHEMBL:CHEMBL587856	FALSE	FALSE	FALSE
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Pyrido[1,2-a]indole-1.-carboxylic acid analog 6	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4C	hgnc:17071	KDM4C	TTD	2020.06.01	NULL	NULL	Pyrido[1,2-a]indole-1.-carboxylic acid analog 7	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Azole derivative 6	NULL	NULL	NULL	NULL	NULL
MANNOSIDE ACETYLGLUCOSAMINYLTRANSFERASE 2	hgnc:7045	MGAT2	TTD	2020.06.01	NULL	NULL	Bicyclic pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
MANNOSIDE ACETYLGLUCOSAMINYLTRANSFERASE 2	hgnc:7045	MGAT2	TTD	2020.06.01	NULL	NULL	Dihydropyrimidinone derivative 4	NULL	NULL	NULL	NULL	NULL
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.2051080907644316	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Lactam derivative 2	NULL	NULL	NULL	NULL	NULL
MANNOSIDE ACETYLGLUCOSAMINYLTRANSFERASE 2	hgnc:7045	MGAT2	TTD	2020.06.01	NULL	NULL	Phenylmethanesulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL O-ACYLTRANSFERASE 2	hgnc:16940	DGAT2	TTD	2020.06.01	NULL	NULL	PMID25470667-Compound-roselipins	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	Pyridine-carboximide derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-phe compound 3	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo cyclohexylamine derivative 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 48	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 50	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 51	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-14	NULL	NULL	NULL	NULL	NULL
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.046059361	TRYPTAMINE	drugbank:DB08653	TRYPTAMINE	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-15	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-34	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-50	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-52	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-70	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25482888-Compound-72	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 1	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GNF-PF-2713	chembl:CHEMBL578719	CHEMBL:CHEMBL578719	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiomorpholine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiomorpholine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiomorpholine derivative 1	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiomorpholine derivative 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiomorpholine derivative 2	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiomorpholine derivative 2	NULL	NULL	NULL	NULL	NULL
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-12	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-13	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-8	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-9	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-Figure2-3	NULL	NULL	NULL	NULL	NULL
CHOLESTEROL 24-HYDROXYLASE	hgnc:2641	CYP46A1	TTD	2020.06.01	NULL	NULL	PMID25514969-Compound-Figure2-4	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-11	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-14	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-115	NULL	NULL	NULL	NULL	NULL
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-116	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-129	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-13	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-132	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-136	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-139	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-141	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-147	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-154	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-159	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-16	NULL	NULL	NULL	NULL	NULL
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.012573676	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-160	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-161	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-162	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-23	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-26	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-27	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-29	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-32	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-34	NULL	NULL	NULL	NULL	NULL
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-35	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-4	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-52	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-53	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-58	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-6	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-61	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-67	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-72	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-73	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-78	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-89	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2-dihydroindazolo[4,3-bc][1,5]benzoxazepine derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 10	NULL	NULL	NULL	NULL	NULL
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004207345	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 4	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-carboxamide derivative 7	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Aromatic ring compound 4	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Picolinamido propanoic acid derivative 1	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Picolinamido propanoic acid derivative 2	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Spiroimidazolone derivative 3	NULL	NULL	NULL	NULL	NULL
GLUCAGON RECEPTOR	hgnc:4192	GCGR	TTD	2020.06.01	NULL	NULL	Spiroimidazolone derivative 5	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-1	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 2	hgnc:591	BIRC3	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-1	NULL	NULL	NULL	NULL	NULL
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.014369915	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-1	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-10	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-26	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-3	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-3	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-32	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-36	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-36	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-38	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-38	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-40	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-41	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-41	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-43	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 2	hgnc:591	BIRC3	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-43	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-43	NULL	NULL	NULL	NULL	NULL
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-7	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	PMID25980951-Compound-7	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 6	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A11	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A11	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-A5	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-C2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-E5	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-F1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-G2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-G5	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-H1	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-H2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-H3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK2	hgnc:6886	MAPK9	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK3	hgnc:6872	MAPK10	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-J2	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-K2	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	N-(pyridin-2-yl)pyridine methylsulfone derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 5	hgnc:1774	CDK5	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-18	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-18	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	PMID26161698-Compound-32	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 1	hgnc:1722	CDK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 10	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 10	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	NULL	(R)-mequitazine (incontinence/respiratory disease), Pierre Fabre	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 5	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	NULL	Aromatic bicyclic compound 5	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Flavonoid derivative 5	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 1	hgnc:11362	STAT1	TTD	2020.06.01	NULL	NULL	Peptide analog 8	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-12	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-20	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-22	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-43	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-53	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	PMID26394986-Compound-Figure16	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 64	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 66	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Salicylic acid derivative 7	NULL	NULL	NULL	NULL	NULL
SIGNAL TRANSDUCER AND ACTIVATOR OF TRANSCRIPTION 3	hgnc:11364	STAT3	TTD	2020.06.01	NULL	NULL	Tri-substituted purine derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Aryl urea derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Aryl urea derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azetidine urea derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azole derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Azole derivative 4	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Benzyl pyrrolyloxoacetamide derivative 2	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-33	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-35	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-5	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-7	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	Ampicidin analog 1	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 14	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 14	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 17	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 17	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 11	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 15	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 2	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 21	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl mannoside derivative 23	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-cyclodextrin conjugate derivative 2	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Beta-cyclodextrin conjugate derivative 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 1	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 11	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 12	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 19	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 2	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 20	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 21	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 24	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 25	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 29	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl mannoside derivative 7	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 10	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 11	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 18	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 19	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 20	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 22	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 25	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 27	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 28	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 30	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biphenyl mannoside derivative 9	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-47	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-48	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-49	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5c	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-5f	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-7a	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-7b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-7e	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-9a	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 1	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzoic acid linked peptide analog 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzoic acid linked peptide analog 6	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzothiazole analog 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Benzothiazole analog 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Beta-phenyl-alpha,beta-unsaturated carbonyl derivative 7	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Cyclohexyl carbamate derivative 7	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-3	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	PMID26882240-Compound-4	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Steroid derivative 2	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Triptolidenol analog 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Dihydropyrido pyrazinone compound 1	NULL	NULL	NULL	NULL	NULL
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.010368813	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	NULL	Dihydropyrido pyrazinone compound 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-50	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-52	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrazole and thiophene derivative 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	Pyrazole and thiophene derivative 4	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Quinazolinone derivative 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Quinazolinone derivative 5	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Tetra-hydro-quinoline derivative 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Tetra-hydro-quinoline derivative 3	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 10	NULL	NULL	NULL	NULL	NULL
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	DOCONEXENT	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 8	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzothiazine-carboxamide compound 2	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Benzothiazine-carboxamide compound 5	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Heteroaryl-cyclopropylamine derivative 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 1	NULL	NULL	NULL	NULL	NULL
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.008562895	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-(2-phenylcyclopropyl) amino acid derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 4A	hgnc:22978	KDM4A	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-21c	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-21c	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-31a	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-31b	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-37b	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-41	NULL	NULL	NULL	NULL	NULL
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.035719504	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID27019002-Compound-43b	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-24	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-24	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-25	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-25	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-3	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-4	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-5	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 1	NULL	NULL	NULL	NULL	NULL
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.024309107	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 1	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 1	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Isoxazoles and isoxazoline derivative 6	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	N,N-methylenebis-2-phenylacetamide and benzenesulfonamide derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	N,N-methylenebis-2-phenylacetamide and benzenesulfonamide derivative 2	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	Phytocannabinoid/aminoalkylindole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	Phytocannabinoid/aminoalkylindole derivative 1	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-13	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.013622434	TICLOPIDINE	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-27	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c][1,2,4]benzotriazine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 6	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 6	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 8	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 8	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Oxindole derivative 1	NULL	NULL	NULL	NULL	NULL
PSEN1	hgnc:9508	PSEN1	DTC	9/2/20	NULL	1.154014752432846	IC261	drugbank:DB03083	IC261	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-427	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3A	hgnc:2978	DNMT3A	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-427	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 3B	hgnc:2979	DNMT3B	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-427	NULL	NULL	NULL	NULL	NULL
DNA [CYTOSINE-5]-METHYLTRANSFERASE 1	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-MTC-433	NULL	NULL	NULL	NULL	NULL
PSEN2	hgnc:9509	PSEN2	DTC	9/2/20	NULL	1.363835616511545	IC261	drugbank:DB03083	IC261	FALSE	FALSE	FALSE
DNA [CYTOSINE-5]-METHYLTRANSFERASE	hgnc:2976	DNMT1	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-PG-11047	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID27376512-Compound-PG-11047	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-1	hgnc:10430	RPS6KA1	TTD	2020.06.01	NULL	NULL	1,6-diazanaphthalenes and pyrido[2,3-d] pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-3	hgnc:10431	RPS6KA2	TTD	2020.06.01	NULL	NULL	PMID27410995-Compound-Figure3j	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE CHK2	hgnc:16627	CHEK2	TTD	2020.06.01	NULL	NULL	PMID27410995-Compound-Figure3j	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	NULL	PMID27410995-Compound-Figure3k	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-78	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-79	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-81	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 10	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 2	NULL	NULL	NULL	NULL	NULL
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	NSC-26699	chembl:CHEMBL221721	CHEMBL:CHEMBL221721	FALSE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 7	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Tricyclic indole compound 8	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Aryl oxyanilide derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzimidazolone acetamide derivative 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzodiazepine derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Benzothiazepine analog 6	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Bidentate pyrazolopyrimidine acetamide analog 4	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine acetamide derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine acetamide derivative 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine acetamide derivative 7	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 3	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 6	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Phenylpyrrolidinone derivative 2	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Phenylpyrrolidinone derivative 3	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Dihydropyridine compound 3	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Dihydropyridine compound 5	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Fused triazoloamino-phenyl analog 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Heterocyclic-fused piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Imidazolidine derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Piperazine derivative 6	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	PMID27724045-Compound-19	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Quinoline derivative 10	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Quinoline derivative 11	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 11	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Quinoline derivative 13	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Quinoline derivative 13	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Tetrazole derivative 1	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Triazole derivative 2	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	Indole-based analog 2	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	NULL	Indole-based analog 2	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	Indole-based analog 2	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-10	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-10	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-10	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-13	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 7	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrrole derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrazine derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrazine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrazine derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrazine derivative 4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridone derivative 3	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridone derivative 3	NULL	NULL	NULL	NULL	NULL
JAK-STAT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	Imidazo[4,5-c]pyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-(cyanomethyl)-4-(2-(phenylamino)pyrimidin-4-yl)benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-(cyanomethyl)-4-(2-(phenylamino)pyrimidin-4-yl)benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	N-(cyanomethyl)-4-(2-(phenylamino)pyrimidin-4-yl)benzamide derivative 1	NULL	NULL	NULL	NULL	NULL
JAK-STAT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure11Example1up	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure11Example1up	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure11Example1up	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure11Example1up	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure11Example1up	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure11Example1up	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure12Example61	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure12Example61	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure2Example4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure2Example4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure2Example4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure3Example7	NULL	NULL	NULL	NULL	NULL
T-CELL-SPECIFIC KINASE	hgnc:6171	ITK	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure3Example7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure6Example6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure6Example6	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure7Example10	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure7Example10	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure8Example22	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2up	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2up	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2up	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2up	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID27774824-Compound-Figure9Example2up	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrazolopyridine derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidopyridazinone derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidopyridazinone derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Pyrimidopyridazinone derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	NULL	Pyrimidopyridazinone derivative 2	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-134	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-155	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	PMID27841045-Compound-157	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	2-PAM derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	4-PAM derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Fluorinated donepezil derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Galantamine analog 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Lycorine dimer salt derivative 1	NULL	NULL	NULL	NULL	NULL
HORMONE SENSITIVE LIPASE	hgnc:6621	LIPE	TTD	2020.06.01	NULL	13.12691780892362	BENZYL BENZOATE	rxcui:19044	BENZYL BENZOATE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-47	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-49	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-51	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-52	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID27967267-Compound-stenine	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine-caffeic acid hybrid derivative 2	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-45	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-5	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-6	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Triazole gold complexe 1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	Dimethoxybenzylidene-2-thio-imidazole-4-one derivative 1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	Phenylalanine derivative 1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	Phenylalanine derivative 1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-10	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-17	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-17	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-17	NULL	NULL	NULL	NULL	NULL
CATHEPSIN B	hgnc:2527	CTSB	TTD	2020.06.01	NULL	NULL	PMID27998201-Compound-24	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoquinoline derivative 4	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoquinoline sulfonamide derivative 1	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoquinoline sulfonamide derivative 2	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoquinoline sulfonyl derivative 2	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-11	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-20	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-7	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	PMID28048944-Compound-7	NULL	NULL	NULL	NULL	NULL
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	NULL	Tricyclic compound 6	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Aryl alkanolamine derivative 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 4	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	N-substituted 9-azabicyclo[3.3.1]nonan-3alpha-yl-phenylcarbamate analog 2	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Phenylpropylamine derivative 3	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Phenylpropylamine derivative 5	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID28051882-Compound-XI	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Bicarboxylic and tricarboxylic ethynyl derivative 1	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33d	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33d	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33g	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33g	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33o	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33o	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33p	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33p	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-34b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-34b	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Bidentate ligands of Markush derivative 2	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bidentate ligands of Markush derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 7	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N,N-bis(5-pyrazoyl)urea derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure17-1	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure24-b	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure24-b	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure24-b	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-2	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270010-Compound-Figure5-2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 16	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 19	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyrimidine derivative 25	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 11	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 12	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolidinyl urea derivative 7	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Thiadiazolyl carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Thiazole derivative 4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Ureido-phenyl-substituted triazine derivative 2	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	Azaindazole amide derivative 1	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	Azaindazole amide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Azaindazole amide derivative 1	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl benzamide derivative 6	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpiperidine ether derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpiperidine ether derivative 6	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	N-acylpiperidine ether derivative 7	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2010077680 109	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2010077680 811	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2015042088Example4	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2015042088Example4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2015042088Example4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	PMID28270021-Compound-WO2016054807Example80	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrazolo[1,5-a]pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-b]pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
BDNF/NT-3 GROWTH FACTORS RECEPTOR	hgnc:8032	NTRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
NT-3 GROWTH FACTOR RECEPTOR	hgnc:8033	NTRK3	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Six-membered heterocyclic benzamide derivative 2	NULL	NULL	NULL	NULL	NULL
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Tri-substituted urea derivative 1	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-13	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-19	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-36	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	PMID28350212-Compound-7	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-16	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-20	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-21	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-25	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-26	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-32	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE	hgnc:6847	MAP2K7	TTD	2020.06.01	NULL	NULL	PMID28594589-Compound-TABLE3C2	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 2	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 3	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Antibodie derivative 9	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 15	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 16	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 17	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 18	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 19	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Carbamide derivative 20	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Conjugated 3-(indolyl)-and 3-(azaindolyl)-4-arylmaleimide compound 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 12	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 19	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Indoline derivative 21	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Oxetane 3,3-dicarboxamide compound 1	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	PMID28621580-Compound-WO2014079545C69	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 2	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 9	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 10	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 10	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 3	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	Quinoline and quinazoline derivative 8	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Alpha-substituted pirinixic acid and pirinixic acid ester derivative 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	PMID28627961-Compound-32	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	PMID28627961-Compound-33	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	PMID28627961-Compound-41	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Polycyclic compound 1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E SYNTHASE	hgnc:9599	PTGES	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Piperidinyl triazole derivative 6	NULL	NULL	NULL	NULL	NULL
PROLYLCARBOXYPEPTIDASE	hgnc:9344	PRCP	TTD	2020.06.01	NULL	NULL	Proline amide derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 12	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 14	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 15	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 20	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 27	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme11	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme12-1	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme12-3	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme12-4	NULL	NULL	NULL	NULL	NULL
GELATINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure15(7)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure16(9b)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure16(9b)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure18(14)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure18(14)	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-LonimacranthoideVI	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-LonimacranthoideVII	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-9	hgnc:7176	MMP9	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-LonimacranthoideVII	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29324067-Compound-38	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Schiff base compound 2	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Secondary and tertiary (hetero)arylamide derivative 2	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Acrylamide compound 3	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazol-2(3H)-one derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzo[d]oxazol-2(3H)-one derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylsulfonyl derivative 2	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piperazine carbamate/urea derivative 5	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-22	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-23	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29334795-Compound-24	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyridazin-3(2H)-one derivative 1	NULL	NULL	NULL	NULL	NULL
HISTAMINE H3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Steroidal carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-19	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-21	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-30	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-34	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-38	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-39	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-41	NULL	NULL	NULL	NULL	NULL
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	PMID29338548-Compound-45	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Aryl 1,2-diamine derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Azetidine derivative 5	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Biphenyl derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Cyclic hydroxamate derivative 1	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Five-membered heteroaromatic compound 3	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	Indazole derivative 4	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-11	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-15	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-73	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-73	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 9	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-73	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-8	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 10	hgnc:18128	HDAC10	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-8	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-8	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-8	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-8	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Decyle nelycorine dibromo salt derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Decyle nelycorine dibromo salt derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Di-substituted piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Oxime derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-10	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-10	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-2a	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-2a	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8d	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	PMID29757691-Compound-8d	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Quinazoline alkaloid derivative 1	NULL	NULL	NULL	NULL	NULL
CHOLINESTERASE	hgnc:983	BCHE	TTD	2020.06.01	NULL	NULL	Quinazoline alkaloid derivative 1	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 14	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 15	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 18	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 19	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 19	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 21	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 21	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 21	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 21	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 21	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 21	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 23	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 23	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 23	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 23	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 23	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 23	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 25	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 25	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 26	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 27	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 27	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 29	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	Peptide analog 35	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 39	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 39	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 39	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-40	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-43	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-43	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-44	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-44	NULL	NULL	NULL	NULL	NULL
IMMUNOPROTEASOME COMPLEX	hgnc:871	ATP5IF1	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-47	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-48	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-5	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-48	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-48	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-9	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-48	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	Cyclic compound 2	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 3	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 3	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Peptide analog 3	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example13	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2013148427	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO2015091734	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	L-697,661	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TROVIRDINE HYDROCHLORIDE	chembl:CHEMBL543611	TROVIRDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
ACETYLCHOLINE RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Abobotulinum toxin A	NULL	NULL	NULL	NULL	NULL
INTERFERON ALPHA	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	Alfaferone	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alogliptin	rxcui:1368001	ALOGLIPTIN	TRUE	FALSE	FALSE
SODIUM PUMP SUBUNIT ALPHA-1	hgnc:799	ATP1A1	TTD	2020.06.01	NULL	3.500511415712966	Aluminium	rxcui:1311504	ALUMINUM	TRUE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	0.5048814541893701	Abilify Maintena	wikidata:Q29003613	ABILIFY MAINTENA	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	1.193356164447602	Acebutolol	rxcui:149	ACEBUTOLOL	TRUE	FALSE	FALSE
INFLUENZA HEMAGGLUTININ	NULL	NULL	TTD	2020.06.01	NULL	NULL	Arbidol	ncit:C152799	UMIFENOVIR	FALSE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Baclofen	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Baquting	NULL	NULL	NULL	NULL	NULL
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.1534190540122556	Caffeine	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
ENZYME UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Desoxyribonuclease	rxcui:3210	DEOXYRIBONUCLEASES	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.2031244535229961	Dicyclomine	rxcui:152021	DICYCLOMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.086861325	Etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.2453629496995069	Esterified estrogens	rxcui:214549	ESTROGENS, ESTERIFIED (USP)	TRUE	FALSE	FALSE
BACTERIAL UDP-N-ACETYLGLUCOSAMINE CARBOXYVINYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fosfomycin	rxcui:4550	FOSFOMYCIN	TRUE	FALSE	FALSE
PLASMODIUM DOXP REDUCTOISOMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fosmidomycin	ncit:C65764	FOSMIDOMYCIN	FALSE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Framycetin	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
ENZYME UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glutathione	rxcui:4890	GLUTATHIONE	TRUE	FALSE	FALSE
FUNGAL MICROTUBULE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Griseofulvin	rxcui:5021	GRISEOFULVIN	TRUE	FALSE	FALSE
ADRENERGIC NEURON	NULL	NULL	TTD	2020.06.01	NULL	NULL	Guanethidine	rxcui:5036	GUANETHIDINE	TRUE	FALSE	FALSE
HYALURONIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hylenex	wikidata:Q47521698	HYLENEX	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.061055432	Meperidine	rxcui:103755	MEPERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TYROSINE 3-MONOOXYGENASE	hgnc:11782	TH	TTD	2020.06.01	NULL	2.500365296937833	L-Tyrosine	rxcui:10962	TYROSINE	TRUE	FALSE	FALSE
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nalmefene	rxcui:31479	NALMEFENE	TRUE	FALSE	FALSE
OXIDOREDUCTASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Olsalazine	rxcui:32385	OLSALAZINE	TRUE	FALSE	FALSE
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	0.027577558	Nefazodone	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
PROTEASOME	hgnc:9338	PRB2	TTD	2020.06.01	NULL	0.192335792	MLN9708	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
ENDOPEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Racecadotril	rxcui:16738	RACECADOTRIL	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ritonavir	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Safinamide	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.09055649	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thrombin/fibrinogen matrix patch	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Troglitazone	rxcui:72610	TROGLITAZONE	TRUE	FALSE	FALSE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Tyverb/Tykerb	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Unoprostone	rxcui:1546408	UNOPROSTONE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.2128689374420047	Tiotropium	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	0.7292732116068681	Trimetrexate	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	IZONSTERIDE	ncit:C99548	IZONSTERIDE	FALSE	FALSE	FALSE
PROSTATE SPECIFIC ANTIGEN	hgnc:6364	KLK3	TTD	2020.06.01	NULL	NULL	MVA-BN Breast	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PF-4418948	NULL	NULL	NULL	NULL	NULL
NICOTINIC ACETYLCHOLINE RECEPTOR	hgnc:1958	CHRNA4	TTD	2020.06.01	NULL	NULL	RPI-78M injectable	NULL	NULL	NULL	NULL	NULL
NOCICEPTIN RECEPTOR	hgnc:8155	OPRL1	TTD	2020.06.01	NULL	2.187819634820604	NOCICEPTIN	iuphar.ligand:1681	NOCICEPTIN/ORPHANIN FQ	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-265744 LAP	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	SA-5845	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	SB-1578	drugbank:DB15294	SB-1578	FALSE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	NULL	TAK-058	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.9723642821424906	Sonepcizumab	ncit:C78195	SONEPCIZUMAB	FALSE	FALSE	TRUE
CILIARY NEUROTROPHIC FACTOR	hgnc:2169	CNTF	TTD	2020.06.01	NULL	NULL	CNTF, Syntex-Synergen, cell therapy	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	0.2083637747448194	Birinapant	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
C-C CHEMOKINE RECEPTOR TYPE 2	hgnc:1603	CCR2	TTD	2020.06.01	NULL	2.282942227638891	BMS-813160	drugbank:DB16240	BMS-813160	FALSE	FALSE	FALSE
CELLULAR INHIBITOR OF APOPTOSIS 1	hgnc:590	BIRC2	TTD	2020.06.01	NULL	1.312691780892362	Birinapant	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
NITRIC-OXIDE SYNTHASE INDUCIBLE	hgnc:7873	NOS2	TTD	2020.06.01	NULL	NULL	CR-3294	NULL	NULL	NULL	NULL	NULL
TRACE AMINE-ASSOCIATED RECEPTOR-1	hgnc:17734	TAAR1	TTD	2020.06.01	NULL	NULL	D-amphetamine transdermal	NULL	NULL	NULL	NULL	NULL
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	NULL	DTI-0009 (oral)	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	LY2090314	iuphar.ligand:7958	LY2090314	FALSE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	LY2090314	iuphar.ligand:7958	LY2090314	FALSE	FALSE	FALSE
PROTEIN KINASE C BETA	hgnc:9395	PRKCB	TTD	2020.06.01	NULL	NULL	LY333531	NULL	NULL	NULL	NULL	NULL
DOPAMINE TRANSPORTER	hgnc:11049	SLC6A3	TTD	2020.06.01	NULL	NULL	NS 2359	NULL	NULL	NULL	NULL	NULL
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	NS 2359	NULL	NULL	NULL	NULL	NULL
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	NULL	NS 2359	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	NU-172	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	NULL	ONO-4641	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	1.875273972703375	Oleoyl-estrone	drugbank:DB04870	OLEOYL-ESTRONE	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	2.625383561784724	Oleoyl-estrone	drugbank:DB04870	OLEOYL-ESTRONE	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.1801292323694494	MGCD-0103	hemonc:337	MOCETINOSTAT	FALSE	FALSE	FALSE
MITOCHONDRIAL PROTEIN UNSPECIFIC	hgnc:9282	PPP1CB	TTD	2020.06.01	NULL	8.751278539282415	Mitoglitazone	drugbank:DB11721	MITOGLITAZONE	FALSE	FALSE	FALSE
TUBULIN BETA-1 CHAIN	hgnc:16257	TUBB1	TTD	2020.06.01	NULL	NULL	PI-88/Taxotere	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RALURIDINE	ncit:C152150	RALURIDINE	FALSE	FALSE	FALSE
MYC MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Resten-NG	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	S-1360	chembl:CHEMBL218227	S-1360	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	NULL	SEN-196	NULL	NULL	NULL	NULL	NULL
INSULIN-LIKE GROWTH FACTOR I RECEPTOR	hgnc:5465	IGF1R	TTD	2020.06.01	NULL	1.981421556063943	R1507	ncit:C95797	TEPROTUMUMAB	FALSE	FALSE	TRUE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	1.166837138570988	Remetinostat	ncit:C97513	REMETINOSTAT	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.075732218	SAR245409	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
HYPERPOLARIZATION CYCLIC NUCLEOTIDE-GATED CHANNEL	hgnc:29665	MALAT1	TTD	2020.06.01	NULL	NULL	SKL-NP	NULL	NULL	NULL	NULL	NULL
HUMAN PAPILLOMAVIRUS PROTEIN E6	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tipapkinogene sovacivec	ncit:C88326	TIPAPKINOGENE SOVACIVEC	FALSE	FALSE	FALSE
HUMAN PAPILLOMAVIRUS PROTEIN E7	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tipapkinogene sovacivec	ncit:C88326	TIPAPKINOGENE SOVACIVEC	FALSE	FALSE	FALSE
GLUCOCORTICOID RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	VBP15	rxcui:2669799	VAMOROLONE	TRUE	FALSE	FALSE
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	1.141471113819445	VX-509	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3	hgnc:3767	FLT4	TTD	2020.06.01	NULL	0.039068208	ABT-869	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY 86-9766	NULL	NULL	NULL	NULL	NULL
HAEMOPHILUS INFLUENZAE DNA GYRASE A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cetraxal Otic	NULL	NULL	NULL	NULL	NULL
STREPTOCOCCUS TOPOISOMERASE IV A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cetraxal Otic	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED L-TYPE CALCIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cilnidipine	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
MITOCHONDRIAL FUNCTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Creatine ALS-08	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CS-038	iuphar.ligand:12287	CHIGLITAZAR	FALSE	FALSE	FALSE
DYSTROPHIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK2402968	chembl:CHEMBL2108735	DRISAPERSEN	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imiglitazar	ncit:C83791	IMIGLITAZAR	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	Liposomal encapsulated paclitaxel (LEP)	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	Liposomal encapsulated paclitaxel (LEP)	NULL	NULL	NULL	NULL	NULL
MICROTUBULE-ASSOCIATED PROTEIN TAU	hgnc:6893	MAPT	TTD	2020.06.01	NULL	NULL	LMT-X	NULL	NULL	NULL	NULL	NULL
TAR DNA BINDING PROTEIN 43	hgnc:11571	TARDBP	TTD	2020.06.01	NULL	NULL	LMT-X	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Marimastat	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	SU5614	NULL	NULL	NULL	NULL	NULL
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.031631127	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.042174836	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	inhibitor	0.1396480617970598	IUPHAR.LIGAND:136	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:152	iuphar.ligand:152	&ALPHA;-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:40	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:153	iuphar.ligand:153	(+)-DOI	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.037884323	IUPHAR.LIGAND:150	rxcui:6883	METHYLERGONOVINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:9880	iuphar.ligand:9880	H05	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:181	iuphar.ligand:181	LY314228	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.041672755	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.016669102	IUPHAR.LIGAND:22	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:176	iuphar.ligand:176	EGIS-7625	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:8427	ncit:C152177	RELENOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.042898424	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1447821817160693	IUPHAR.LIGAND:198	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613069	IUPHAR.LIGAND:3233	iuphar.ligand:3233	SB269970	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613069	IUPHAR.LIGAND:3237	iuphar.ligand:3237	SB656104	FALSE	FALSE	FALSE
NCBIGENE:768	hgnc:1383	CA9	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11786	iuphar.ligand:11786	WS-898	FALSE	FALSE	FALSE
NCBIGENE:756	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.7573221812840553	IUPHAR.LIGAND:7277	rxcui:8699	PROBUCOL	TRUE	FALSE	FALSE
NCBIGENE:783	hgnc:1402	CACNB2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8829	iuphar.ligand:8829	COMPOUND 2 [PMID: 22380603]	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1259176768242074	IUPHAR.LIGAND:10630	ncit:C165549	OLVEREMBATINIB	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:6598	rxcui:8299	PHYSOSTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12084	iuphar.ligand:12084	PIFUSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.1539814405738841	IUPHAR.LIGAND:10316	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.2561349816375342	IUPHAR.LIGAND:515	ncit:C77294	CIRAZOLINE	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:507	iuphar.ligand:507	RHO-TIA	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.066047385	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	agonist	0.2386712328895204	IUPHAR.LIGAND:515	ncit:C77294	CIRAZOLINE	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.085378327	IUPHAR.LIGAND:5385	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.094438258	IUPHAR.LIGAND:12577	iuphar.ligand:12577	MK-912	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.025183535	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.053964719	IUPHAR.LIGAND:499	iuphar.ligand:499	WB 4101	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:136	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:10182	iuphar.ligand:10182	ARD-69	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.1810609352954983	IUPHAR.LIGAND:2863	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	0.093931433	IUPHAR.LIGAND:5158	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
NCBIGENE:1614	hgnc:13557	ACE2	GuideToPharmacology	2024.1	NULL	5.250767123569449	IUPHAR.LIGAND:11603	iuphar.ligand:11603	CPS4	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:405	drugbank:DB08770	4-{2-[(7-AMINO-2-FURAN-2-YL[1,2,4]TRIAZOLO[1,5-A][1,3,5]TRIAZIN-5-YL)AMINO]ETHYL}PHENOL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	6-METHOXY-HARMALAN	chembl:CHEMBL338115	CHEMBL:CHEMBL338115	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:5603	iuphar.ligand:5603	CPFPX	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:5593	iuphar.ligand:5593	GS9667	FALSE	FALSE	FALSE
NCBIGENE:937	hgnc:1648	CD24P3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:4693	iuphar.ligand:4693	&ALPHA;-METHYL-D,L-TRYPTOPHAN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.036212187	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.5413161983061289	IUPHAR.LIGAND:468	iuphar.ligand:468	MRS1177	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.1215455352678113	IUPHAR.LIGAND:7949	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.3387591692625452	IUPHAR.LIGAND:8448	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
NCBIGENE:35	hgnc:90	ACADS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:11930	iuphar.ligand:11930	COMPOUND 1 [PMID: 28379944]	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:11259	iuphar.ligand:11259	[LEU14]BOMBESIN	FALSE	FALSE	FALSE
NCBIGENE:2845	hgnc:4477	GPR22	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8320	iuphar.ligand:8320	ABT-737	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.064347636	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8505	iuphar.ligand:8505	ML-18	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:10569	iuphar.ligand:10569	NMU (104-114)	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:6191	iuphar.ligand:6191	AC-PHE-TRP-ALA-HIS(&TAU;BZL)-NIP-GLY-ARG-NH2	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:11775	iuphar.ligand:11775	COMPOUND 6 [PMID: 34553947]	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.1875273972703375	IUPHAR.LIGAND:557	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:543	iuphar.ligand:543	ICI 118551	FALSE	FALSE	FALSE
NCBIGENE:1786	hgnc:2976	DNMT1	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:11888	ncit:C175551	ZILURGISERTIB	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2019525816757481	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:5703	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:10388	iuphar.ligand:10388	SZM594	FALSE	FALSE	FALSE
NCBIGENE:1944	hgnc:3223	EFNA3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7807	iuphar.ligand:7807	ME BROMODOMAIN INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7528	iuphar.ligand:7528	COMPOUND 15 [HAY ET AL., 2013]	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:10072	iuphar.ligand:10072	DUAL BRD4/PLK1 INHIBITOR 23	FALSE	FALSE	FALSE
NCBIGENE:1947	hgnc:3226	EFNB1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8215	iuphar.ligand:8215	CCT244747	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7523	iuphar.ligand:7523	PFI-1	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:11671	ncit:C162573	LUXEPTINIB	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.030598876	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:661	iuphar.ligand:661	R-715	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:673	iuphar.ligand:673	FR167344	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:10226	iuphar.ligand:10226	ALBUTENSIN A	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:576	iuphar.ligand:576	N-METHYL-PHE-LYS-PRO-D-CHA-TRP-D-ARG-CO2H	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:581	iuphar.ligand:581	W54011	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:11286	iuphar.ligand:11286	EU-DTPA-HC3A	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	0.2419708351875322	IUPHAR.LIGAND:579	iuphar.ligand:579	PMX53	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.020226376	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:2337	ncbigene:2337	FNL1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8569	iuphar.ligand:8569	COMPOUND 19 [PMID: 8831774]	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.061773731	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
NCBIGENE:1556	hgnc:2616	CYP2B7P	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2597	hgnc:4141	GAPDH	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:10434	iuphar.ligand:10434	COMPOUND 5B  [PMID: 31287314]	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	0.2524407270946851	IUPHAR.LIGAND:2439	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002657809	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:573	iuphar.ligand:573	C5A	FALSE	FALSE	FALSE
NCBIGENE:1998	hgnc:3317	ELF2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8916	rxcui:2478439	UMBRALISIB	TRUE	FALSE	FALSE
NCBIGENE:389	hgnc:669	RHOC	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:5412	iuphar.ligand:5412	PGF1&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:2351	ncbigene:2351	FOLR2L	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:6533	iuphar.ligand:6533	KGP94	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
NCBIGENE:388	hgnc:668	RHOB	GuideToPharmacology	2024.1	activator	0.2536602475154323	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
NCBIGENE:2353	hgnc:3796	FOS	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:11515	iuphar.ligand:11515	K777	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:10178	iuphar.ligand:10178	MDMB-FUBINACA	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:12754	iuphar.ligand:12754	AZD1940	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	0.6731752722524935	IUPHAR.LIGAND:764	iuphar.ligand:764	[125I]CCL5 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:778	iuphar.ligand:778	MC148R	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	CYSTEAMINE HYDROCHLORIDE	rxcui:1426886	CYSTEAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:781	iuphar.ligand:781	RS-504393	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:9045	iuphar.ligand:9045	INCB3284	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:754	iuphar.ligand:754	CCL15	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	0.5000730593875666	IUPHAR.LIGAND:764	iuphar.ligand:764	[125I]CCL5 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:780	iuphar.ligand:780	RS-136270	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:787	iuphar.ligand:787	CCL11	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	DNDI1416988	chembl:CHEMBL1389794	CHEMBL:CHEMBL1389794	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:805	ncit:C78043	APLAVIROC	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	1.458546423213736	IUPHAR.LIGAND:12409	iuphar.ligand:12409	AK-2292	FALSE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8113	iuphar.ligand:8113	XL413	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:10241	iuphar.ligand:10241	FK-881	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:10494	iuphar.ligand:10494	SWE101	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
NCBIGENE:726	hgnc:1482	CAPN5	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:723	hgnc:4283	GJB1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8499	ncit:C174724	ELUBRIXIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002796829	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
NCBIGENE:72	hgnc:145	ACTG2	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:3645	iuphar.ligand:3645	CXCL13	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	8-AZAGUANINE	ncit:C28788	8-AZAGUANINE	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:607	iuphar.ligand:607	ALX40-4C	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:10146	iuphar.ligand:10146	CXCR4 ANTAGONIST 22	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:5948	iuphar.ligand:5948	CDK2 INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:5946	drugbank:DB07664	K-00546	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:5945	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:6035	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1442518440541057	IUPHAR.LIGAND:10357	iuphar.ligand:10357	CDK INHIBITOR 4.35	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:5950	iuphar.ligand:5950	CDK4 INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:12074	iuphar.ligand:12074	ASNUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:5948	iuphar.ligand:5948	CDK2 INHIBITOR III	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:11409	iuphar.ligand:11409	CIMPUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:10531	iuphar.ligand:10531	BSJ-04-132	FALSE	FALSE	FALSE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:5945	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
NCBIGENE:1360	hgnc:2299	CPB1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12362	ncit:C184908	BAXDROSTAT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.009838424	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:11841	iuphar.ligand:11841	SY-5609	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:6035	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
NCBIGENE:1359	hgnc:2298	CPA3	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:5224	rxcui:6923	METYRAPONE	TRUE	FALSE	FALSE
NCBIGENE:1325	hgnc:2257	CORT	GuideToPharmacology	2024.1	inhibitor	0.8751278539282417	IUPHAR.LIGAND:7266	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
NCBIGENE:1329	hgnc:2269	COX5B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9882	iuphar.ligand:9882	TIQ-15	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.014369915	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
NCBIGENE:1353	hgnc:2261	COX11	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8795	iuphar.ligand:8795	COMPOUND 7P [PMID: 7861416]	FALSE	FALSE	FALSE
NCBIGENE:3002	hgnc:4709	GZMB	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9931	iuphar.ligand:9931	COMPOUND 7C [PMID: 22041175]	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	1,3-DIPHENYLTHIOUREA	chembl:CHEMBL275260	CHEMBL:CHEMBL275260	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:3634	ncit:C96712	PRANLUKAST	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	0.2019525816757481	HONOKIOL	rxcui:2562546	HONOKIOL	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:3334	ncit:C96710	POBILUKAST	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.019361236	IUPHAR.LIGAND:8286	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1603	iuphar.ligand:1603	(-)-BREMAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:2004	hgnc:3325	ELK3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8126	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.1842374429322614	IUPHAR.LIGAND:7266	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.01223955	DULOXETINE HYDROCHLORIDE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.013666755	IUPHAR.LIGAND:1605	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1397	hgnc:2361	CRIP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10246	iuphar.ligand:10246	LEI105	FALSE	FALSE	FALSE
NCBIGENE:2603	hgnc:2861	DHFR	GuideToPharmacology	2024.1	inhibitor	0.1904575128526865	IUPHAR.LIGAND:4815	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NCBIGENE:1396	hgnc:2360	CRIP1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10245	iuphar.ligand:10245	KT-109	FALSE	FALSE	FALSE
NCBIGENE:3211	hgnc:5111	HOXB1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:13010	iuphar.ligand:13010	PF-07202954	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:7002	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
NCBIGENE:2009	hgnc:3330	EML1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:10688	iuphar.ligand:10688	GNF4877	FALSE	FALSE	FALSE
NCBIGENE:218	hgnc:405	ALDH3A1	GuideToPharmacology	2024.1	inhibitor	0.051731696	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
NCBIGENE:1616	hgnc:2681	DAXX	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8673	iuphar.ligand:8673	COMPOUND 1 [PMID: 18507370]	FALSE	FALSE	FALSE
NCBIGENE:1249	hgnc:7876	NOS3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9849	iuphar.ligand:9849	GW274150	FALSE	FALSE	FALSE
CASP1	hgnc:1499	CASP1	DTC	9/2/20	NULL	0.100976291	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
NCBIGENE:1833	hgnc:3053	EPYC	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:7944	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10516	iuphar.ligand:10516	PF-06821497	FALSE	FALSE	FALSE
NCBIGENE:1828	hgnc:3048	DSG1	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
NCBIGENE:1822	hgnc:3033	ATN1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:9248	ncit:C115110	NAQUOTINIB	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:10628	iuphar.ligand:10628	REZIVERTINIB	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:10635	iuphar.ligand:10635	MS154	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:3167	iuphar.ligand:3167	NE21650	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	DIMETHYL GAMBOGATE	chembl:CHEMBL1436860	DIMETHYL GAMBOGATE	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:6483	iuphar.ligand:6483	TUG-770	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	modulator	3.750547945	IUPHAR.LIGAND:5803	iuphar.ligand:5803	AMG7703	FALSE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:5588	iuphar.ligand:5588	GRIFOLIC ACID	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.016449772	PROPRANOLOL HYDROCHLORIDE	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:5587	iuphar.ligand:5587	NCG21	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:5712	iuphar.ligand:5712	SU-14813	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:11546	iuphar.ligand:11546	ALDAFERMIN	FALSE	FALSE	FALSE
NCBIGENE:3177	hgnc:11004	SLC29A2	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:11484	iuphar.ligand:11484	DM-CHX	FALSE	FALSE	FALSE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:8104	iuphar.ligand:8104	LY2874455	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.004715129	IUPHAR.LIGAND:5698	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:1811	hgnc:3018	SLC26A3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:9788	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.043180651	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.002909335	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.2051080907644316	IUPHAR.LIGAND:5973	iuphar.ligand:5973	G&OUML; 6976	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.02646556	IUPHAR.LIGAND:7885	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:12911	iuphar.ligand:12911	COMPOUND 34F [PMID: 37535845]	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.008728004	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:1606	hgnc:2849	DGKA	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:6878	rxcui:136300	CAPROMAB PENDETIDE	TRUE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.010205573	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:11024	iuphar.ligand:11024	BMS-986235	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:10138	iuphar.ligand:10138	1R-11	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.092118721	IUPHAR.LIGAND:9404	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.1017590527823536	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.054243462	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:3594	iuphar.ligand:3594	GALANIN-LIKE PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:11417	iuphar.ligand:11417	SPEXIN-1	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	modulator	1.544343271638073	IUPHAR.LIGAND:9574	iuphar.ligand:9574	NNC0640	FALSE	FALSE	FALSE
NCBIGENE:450	hgnc:768	ASS1P5	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:4333	iuphar.ligand:4333	UBP302	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4168	iuphar.ligand:4168	D-AP5	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:11720	iuphar.ligand:11720	S-DESCHLOROKETAMINE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.084689792	IUPHAR.LIGAND:3309	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4170	iuphar.ligand:4170	D-CCPENE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:4161	iuphar.ligand:4161	CONANTOKIN-G	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.1539814405738841	IUPHAR.LIGAND:6511	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:935	hgnc:1646	CD24P1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4712	iuphar.ligand:4712	LY2365109	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1177	rxcui:38782	TRIPTORELIN	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:1164	iuphar.ligand:1164	GNRH II	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:3320	iuphar.ligand:3320	G15	FALSE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:10198	iuphar.ligand:10198	INT-767	FALSE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:11696	iuphar.ligand:11696	XYT528B	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:5017	rxcui:1307404	LINACLOTIDE	TRUE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:5053	iuphar.ligand:5053	SANP	FALSE	FALSE	FALSE
NCBIGENE:2905	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:9260	iuphar.ligand:9260	SNX0723	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:5798	drugbank:DB03225	D-TRYPTOPHAN	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:1598	iuphar.ligand:1598	COMPOUND 5B [PMID: 17358052]	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.050294704	IUPHAR.LIGAND:1059	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.051327147	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.1223004764806549	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.3201687270469177	IUPHAR.LIGAND:7498	rxcui:1796	BUFEXAMAC	TRUE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.023284998	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.04573839	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.073437302	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:1381	hgnc:2338	CRABP1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6662	drugbank:DB07917	4-(BENZHYDRYLOXY)-1-[3-(1H-TETRAAZOL-5-YL)PROPYL]PIPERIDINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.060353645	IUPHAR.LIGAND:7427	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1384	hgnc:2342	CRAT	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8745	iuphar.ligand:8745	COMPOUND 3 [PMID: 21650226]	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.013411921	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.013716738	IUPHAR.LIGAND:1225	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:1212	iuphar.ligand:1212	(-)-TRANS-H2-PAT	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.013716738	IUPHAR.LIGAND:3958	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:1224	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:1207	iuphar.ligand:1207	(&PLUSMN;)-TRANS-H2-PAT	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:1227	rxcui:9009	PYRILAMINE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:1199	iuphar.ligand:1199	OXO-ARPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:8985	iuphar.ligand:8985	ADRIFORANT	FALSE	FALSE	FALSE
NCBIGENE:3194	hgnc:9476	HTRA1	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:11759	iuphar.ligand:11759	GALEGENIMAB	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2991	iuphar.ligand:2991	COMPOUND 1E [PMID: 2153213]	FALSE	FALSE	FALSE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:9742	iuphar.ligand:9742	COMPOUND 83 [PMID: 23888932]	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.093763699	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5565	iuphar.ligand:5565	CID2440433	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1966	iuphar.ligand:1966	[3H]ILOPROST	FALSE	FALSE	FALSE
NCBIGENE:1448	hgnc:2446	CSN3	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9548	iuphar.ligand:9548	GNF362	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:5215	iuphar.ligand:5215	LUTEOLIN	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:10631	iuphar.ligand:10631	LORPUCITINIB	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.020320306	IUPHAR.LIGAND:1605	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.017295017	IUPHAR.LIGAND:7944	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
NCBIGENE:266	hgnc:462	AMELY	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4012	iuphar.ligand:4012	PEPTIDE 234	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12066	iuphar.ligand:12066	LY3499446	FALSE	FALSE	FALSE
NCBIGENE:520	hgnc:844	ATP5MC2P1	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:515	hgnc:840	ATP5PB	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:2506	iuphar.ligand:2506	R-(+)-METHANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	0.1141471113819445	IUPHAR.LIGAND:2326	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	activator	1.250182648468916	IUPHAR.LIGAND:2323	iuphar.ligand:2323	CYPPA	FALSE	FALSE	FALSE
NCBIGENE:386	hgnc:18866	KCNT2	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:2507	iuphar.ligand:2507	CLOFILIUM	FALSE	FALSE	FALSE
NCBIGENE:543	hgnc:880	ALDH7A1P3	GuideToPharmacology	2024.1	blocker	13.12691780892362	IUPHAR.LIGAND:2548	iuphar.ligand:2548	MAST CELL DEGRANULATING PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:546	hgnc:886	ATRX	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11478	iuphar.ligand:11478	RY785	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:2592	iuphar.ligand:2592	L735821	FALSE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	activator	0.729273212	IUPHAR.LIGAND:2307	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	activator	0.5048814541893701	IUPHAR.LIGAND:2307	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
NCBIGENE:560	ncbigene:560	AZF1	GuideToPharmacology	2024.1	activator	0.3365876361262468	IUPHAR.LIGAND:2439	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:564	hgnc:6299	KCNQ5	GuideToPharmacology	2024.1	activator	1.250182648468916	IUPHAR.LIGAND:2601	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2601	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6713	iuphar.ligand:6713	COMPOUND 7 [PMID: 22533316]	FALSE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	0.3431873936973497	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:6003	iuphar.ligand:6003	LCK INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8054	iuphar.ligand:8054	PF-06447475	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:2750	iuphar.ligand:2750	24(S)-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:2750	iuphar.ligand:2750	24(S)-HYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:6580	iuphar.ligand:6580	GRI977143	FALSE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	0.760980743	IUPHAR.LIGAND:11315	iuphar.ligand:11315	SAR100842	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:8074	iuphar.ligand:8074	NG-25	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1306	iuphar.ligand:1306	COMPOUND 17 [PMID: 17125263]	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:7755	iuphar.ligand:7755	COMPOUND 4B [PMID: 19683441]	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6219	iuphar.ligand:6219	MNI-135	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:10009	iuphar.ligand:10009	VU0483605	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.3860858179095183	IUPHAR.LIGAND:8946	iuphar.ligand:8946	JNJ-40411813	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:1409	iuphar.ligand:1409	FP0429	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:295	iuphar.ligand:295	ARECAIDINE PROPARGYL ESTER	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:6937	iuphar.ligand:6937	IPEROXO	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:289	iuphar.ligand:289	AC-42	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:289	iuphar.ligand:289	AC-42	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:8549	iuphar.ligand:8549	BENZOQUINAZOLINONE 12	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:3272	iuphar.ligand:3272	[3H]PIRENZEPINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:8584	iuphar.ligand:8584	AQ-RA 741	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.035098711	IUPHAR.LIGAND:320	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:313	iuphar.ligand:313	MUSCARINIC TOXIN 3	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:3264	iuphar.ligand:3264	AFDX384	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:7459	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1491695205559502	IUPHAR.LIGAND:301	ncit:C132273	MILAMELINE	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	agonist	0.1591141552596803	IUPHAR.LIGAND:6937	iuphar.ligand:6937	IPEROXO	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:7257	rxcui:7818	OXYPHENONIUM	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.099446347	IUPHAR.LIGAND:7459	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:8584	iuphar.ligand:8584	AQ-RA 741	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:7770	iuphar.ligand:7770	[125I]SD6	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1354	iuphar.ligand:1354	S24773	FALSE	FALSE	FALSE
NCBIGENE:3004	hgnc:4712	GZMM	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:9931	iuphar.ligand:9931	COMPOUND 7C [PMID: 22041175]	FALSE	FALSE	FALSE
NCBIGENE:3001	hgnc:4708	GZMA	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9931	iuphar.ligand:9931	COMPOUND 7C [PMID: 22041175]	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:10003	iuphar.ligand:10003	GNE-131	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:9858	iuphar.ligand:9858	GS-458967	FALSE	FALSE	FALSE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	blocker	0.1000146118775133	IUPHAR.LIGAND:10355	iuphar.ligand:10355	GNE-616	FALSE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	blocker	0.6563458904461813	IUPHAR.LIGAND:7602	rxcui:35780	ROPIVACAINE	TRUE	FALSE	FALSE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	blocker	0.1750255707856483	IUPHAR.LIGAND:2629	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:12644	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	blocker	0.7501095890813498	IUPHAR.LIGAND:10355	iuphar.ligand:10355	GNE-616	FALSE	FALSE	FALSE
NCBIGENE:1749	hgnc:2918	DLX5	GuideToPharmacology	2024.1	agonist	8.751278539282415	IUPHAR.LIGAND:4892	iuphar.ligand:4892	CANF4-23	FALSE	FALSE	FALSE
NCBIGENE:585	hgnc:969	BBS4	GuideToPharmacology	2024.1	blocker	3.750547945	IUPHAR.LIGAND:8521	iuphar.ligand:8521	PF-01247324	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	blocker	0.5357925636295356	IUPHAR.LIGAND:10355	iuphar.ligand:10355	GNE-616	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:12644	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	0.3621218705909966	IUPHAR.LIGAND:3969	ncit:C169814	BRADANICLINE	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2099	iuphar.ligand:2099	SUBSTANCE P-(4-11)	FALSE	FALSE	FALSE
NCBIGENE:2117	hgnc:3492	ETV3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8150	iuphar.ligand:8150	GSK579289A	FALSE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:3981	iuphar.ligand:3981	[3H]&ALPHA;-BUNGAROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:2087	iuphar.ligand:2087	HEMOKININ 1	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:3473	iuphar.ligand:3473	[18F]SPA-RQ	FALSE	FALSE	FALSE
NCBIGENE:1770	hgnc:2953	DNAH9	GuideToPharmacology	2024.1	modulator	5.834185692854944	IUPHAR.LIGAND:12280	iuphar.ligand:12280	GDC-2394	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5773	iuphar.ligand:5773	GSK 172981	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:8864	iuphar.ligand:8864	(R)-RO65-6570	FALSE	FALSE	FALSE
NCBIGENE:1220	hgnc:10959	SLCO1B1	GuideToPharmacology	2024.1	inhibitor	0.027177884	IUPHAR.LIGAND:2765	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
NCBIGENE:1219	hgnc:10956	SLCO1A2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:4570	rxcui:35616	RIFAMYCIN SV	TRUE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	inhibitor	0.075010959	IUPHAR.LIGAND:2765	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NCBIGENE:2964	hgnc:4654	GTF2F2P1	GuideToPharmacology	2024.1	blocker	5.250767123569449	IUPHAR.LIGAND:10087	iuphar.ligand:10087	CM4620	FALSE	FALSE	FALSE
NCBIGENE:2965	hgnc:4655	GTF2H1	GuideToPharmacology	2024.1	blocker	13.12691780892362	IUPHAR.LIGAND:10087	iuphar.ligand:10087	CM4620	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	agonist	0.036718651	IUPHAR.LIGAND:2176	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:9998	iuphar.ligand:9998	MRS4458	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.03729238	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2269	iuphar.ligand:2269	BAY 55-9837	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1830	iuphar.ligand:1830	2-O-METHYL-PAF C-18	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1839	iuphar.ligand:1839	RP-52770	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:3842	iuphar.ligand:3842	[LYS15,ARG16,LEU27]VIP-(1-7)/GRF-(8-27)-NH2	FALSE	FALSE	FALSE
NCBIGENE:2751	hgnc:4340	GLUD1P5	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11612	ncit:C184910	RENCOFILSTAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	0.577007376	IUPHAR.LIGAND:2691	drugbank:DB08078	{4-[3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPOXY]PHENOXY}ACETIC ACID	FALSE	FALSE	FALSE
NCBIGENE:594	hgnc:987	BCKDHB	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:2673	iuphar.ligand:2673	GW9578	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:3440	iuphar.ligand:3440	GW6471	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:2672	ncit:C81693	FARGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.5303805175322676	IUPHAR.LIGAND:2673	iuphar.ligand:2673	GW9578	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:8907	ncit:C75189	EDAGLITAZONE	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:6691	iuphar.ligand:6691	CP-775146	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003077463	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.1250182648468916	IUPHAR.LIGAND:12287	iuphar.ligand:12287	CHIGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:2672	ncit:C81693	FARGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	inhibitor	0.012756966	IUPHAR.LIGAND:8741	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.023598953	IUPHAR.LIGAND:7878	ncit:C90565	BUPARLISIB	FALSE	FALSE	TRUE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.015627283	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
NCBIGENE:2496	hgnc:3979	FTH1P1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6631	iuphar.ligand:6631	LY134046	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.045461187	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
NCBIGENE:2698	hgnc:4275	GJA1P1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:7025	iuphar.ligand:7025	DAMINOZIDE	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.053633985	IUPHAR.LIGAND:10097	ncit:C116877	PAXALISIB	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.026045472	PRASTERONE	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:12119	iuphar.ligand:12119	NVP-CLR457	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	PROROXAN	ncit:C84119	PROROXAN	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.026816992	IUPHAR.LIGAND:7875	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.073746729	IUPHAR.LIGAND:8793	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.046303061	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:7743	iuphar.ligand:7743	IZORLISIB	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:12487	iuphar.ligand:12487	ROGINOLISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.035098711	IUPHAR.LIGAND:7875	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NCBIGENE:1297	hgnc:2217	COL9A1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:5179	iuphar.ligand:5179	EHNA	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9374	iuphar.ligand:9374	CX-5279	FALSE	FALSE	FALSE
NCBIGENE:2170	hgnc:3557	FABP3	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:7918	ncit:C143162	ONVANSERTIB	FALSE	FALSE	TRUE
NCBIGENE:2171	hgnc:3560	FABP5	GuideToPharmacology	2024.1	inhibitor	0.1117184494376478	IUPHAR.LIGAND:10361	iuphar.ligand:10361	RG-1530	FALSE	FALSE	FALSE
NCBIGENE:2169	hgnc:3556	FABP2	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:7918	ncit:C143162	ONVANSERTIB	FALSE	FALSE	TRUE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.1067229090156392	IUPHAR.LIGAND:2878	rxcui:3706	DYDROGESTERONE	TRUE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:10734	iuphar.ligand:10734	GARCINOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2385	hgnc:8747	PCSK5	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:6564	iuphar.ligand:6564	PHENYLACETYL-ARG-VAL-ARG-4-AMIDINOBENZYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.1067229090156392	IUPHAR.LIGAND:2882	ncit:C170255	ONAPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:1504	iuphar.ligand:1504	NEUROPEPTIDE Y	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:5573	iuphar.ligand:5573	[ALA1,12,AIB3,GLN10,HARG11,TRP14,ARG19]PTH-(1-34)-NH2	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	NSC-747265	chembl:CHEMBL595682	CHEMBL:CHEMBL595682	FALSE	FALSE	FALSE
NCBIGENE:2915	hgnc:4597	GRM5	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:9362	iuphar.ligand:9362	AZD7545	FALSE	FALSE	FALSE
NCBIGENE:3006	hgnc:4716	H1-2	GuideToPharmacology	2024.1	activator	7.501095891	IUPHAR.LIGAND:9936	iuphar.ligand:9936	DMAMCL	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:7880	iuphar.ligand:7880	AGERAFENIB	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
PARG	hgnc:8605	PARG	DTC	9/2/20	NULL	105.0153424713889	BENZAMIDE	chembl:CHEMBL267373	BENZAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:11867	drugbank:DB15254	AVUTOMETINIB	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:11711	iuphar.ligand:11711	AZD0284	FALSE	FALSE	FALSE
NCBIGENE:1527	hgnc:2563	TEX28	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
NCBIGENE:2630	hgnc:4178	GBA1LP	GuideToPharmacology	2024.1	inhibitor	0.112919723	IUPHAR.LIGAND:4793	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:1851	hgnc:9665	PTPRB	GuideToPharmacology	2024.1	inhibitor	19.69037671338543	IUPHAR.LIGAND:11336	ncit:C152161	RAZUPROTAFIB	FALSE	FALSE	FALSE
NCBIGENE:1530	hgnc:10435	RPS6KA6	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:7949	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:9321	iuphar.ligand:9321	(B7-33)H2	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.4039051633514961	IUPHAR.LIGAND:1991	iuphar.ligand:1991	[33P]RELAXIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:1518	hgnc:39084	CTSLP8	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8210	iuphar.ligand:8210	COMPOUND 27 [PMID: 21123062]	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.081407242	IUPHAR.LIGAND:7266	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
NCBIGENE:1535	hgnc:2577	CYBA	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:9423	iuphar.ligand:9423	COMPOUND 14N [PMID: 25589934]	FALSE	FALSE	FALSE
NCBIGENE:2553	hgnc:4074	GABPB1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:6682	iuphar.ligand:6682	SM 21	FALSE	FALSE	FALSE
NCBIGENE:833	hgnc:1493	CARS1	GuideToPharmacology	2024.1	inhibitor	0.3860858179095184	IUPHAR.LIGAND:4726	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3110	iuphar.ligand:3110	J-104123	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:7997	iuphar.ligand:7997	SQ-109	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:2050	iuphar.ligand:2050	L-779,976	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:2035	iuphar.ligand:2035	BIM 23034	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.2234368988752957	IUPHAR.LIGAND:2004	iuphar.ligand:2004	BIM 23052	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	inhibitor	0.2763561643983921	IUPHAR.LIGAND:2026	iuphar.ligand:2026	BIM 23454	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	4'-METHOXYCHALCONE	chembl:CHEMBL34398	4'-METHOXYCHALCONE	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2053	iuphar.ligand:2053	NOC-ATE	FALSE	FALSE	FALSE
NCBIGENE:2237	hgnc:3650	FEN1	GuideToPharmacology	2024.1	inhibitor	0.1244257612220248	IUPHAR.LIGAND:9580	iuphar.ligand:9580	MPI-0485520	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:5514	iuphar.ligand:5514	COMPOUND 5G [PMID: 21571530]	FALSE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.8078103267029924	IUPHAR.LIGAND:8148	iuphar.ligand:8148	COMPOUND 31 [PMID: 24915291]	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	AG-528	chembl:CHEMBL56542	CHEMBL:CHEMBL56542	FALSE	FALSE	FALSE
NCBIGENE:2526	hgnc:4015	FUT4	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:6650	rxcui:8794	PROPYLTHIOURACIL	TRUE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.6482428547616604	IUPHAR.LIGAND:10662	iuphar.ligand:10662	BMS-986260	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:9783	iuphar.ligand:9783	MK6-83	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	4.773424657790408	IUPHAR.LIGAND:12551	iuphar.ligand:12551	TRPVICIN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.021036727	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	0.2592971419046642	IUPHAR.LIGAND:2341	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	0.3723948314588262	IUPHAR.LIGAND:12705	iuphar.ligand:12705	BAY1217389	FALSE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.2822993077187876	IUPHAR.LIGAND:10744	iuphar.ligand:10744	GOLIDOCITINIB	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.002378065	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2277	iuphar.ligand:2277	[125I]VIP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:2193	iuphar.ligand:2193	3-N3-PHPA-LVA	FALSE	FALSE	FALSE
NCBIGENE:2284	hgnc:3716	FKBP1AP3	GuideToPharmacology	2024.1	inhibitor	0.1988926940746004	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:1522	iuphar.ligand:1522	[ALA31,AIB32]NPY (PIG)	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.020936073	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1554	iuphar.ligand:1554	PYY-(3-36)	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	0.5250767123569451	IUPHAR.LIGAND:1504	iuphar.ligand:1504	NEUROPEPTIDE Y	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	NULL	VEGF/VEGFR INHIBITORS	NULL	NULL	NULL	NULL	NULL
PDGFRB	hgnc:8804	PDGFRB	CIViC	10-Apr-24	NULL	0.059667808	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	1.250182648468916	FACT COMPLEX-TARGETING CURAXIN CBL0137	ncit:C107239	FACT COMPLEX-TARGETING CURAXIN CBL0137	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.179119736	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.019114551	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	CIViC	10-Apr-24	NULL	0.070129236	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	0.1108075556053025	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CIViC	10-Apr-24	NULL	0.1766118064547324	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.003186532	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
NPM1	hgnc:7910	NPM1	CIViC	10-Apr-24	NULL	0.082429625	TRETINOIN	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	CIViC	10-Apr-24	NULL	NULL	9F7-F11	NULL	NULL	NULL	NULL	NULL
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.011762471	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CRLF2	hgnc:14281	CRLF2	CIViC	10-Apr-24	NULL	2.917092846427472	JAK INHIBITOR I	drugbank:DB04716	2-TERT-BUTYL-9-FLUORO-1,6-DIHYDROBENZO[H]IMIDAZO[4,5-F]ISOQUINOLIN-7-ONE	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	RMC-4550	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	NULL	R406	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	DIGOXIGENIN	drugbank:DB03671	DIGOXIGENIN	FALSE	FALSE	FALSE
NUDT15	hgnc:23063	NUDT15	CIViC	10-Apr-24	NULL	0.5834185692854944	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
BARD1	hgnc:952	BARD1	CIViC	10-Apr-24	NULL	0.1084869240406911	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.020002922	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
CCND3	hgnc:1585	CCND3	CIViC	10-Apr-24	NULL	0.4286340509036285	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
SMARCA4	hgnc:11100	SMARCA4	CIViC	10-Apr-24	NULL	0.1339481409073839	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
KDM4D	hgnc:25498	KDM4D	DTC	9/2/20	NULL	8.751278539282415	N-OXALYLGLYCINE	chembl:CHEMBL90852	N-OXALYLGLYCINE	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.020056406	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.1215455352678113	ANTI-EGFR MONOCLONAL ANTIBODY	ncit:C133878	ANTI-EGFR MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.091159151	SCH772984	iuphar.ligand:8056	SCH772984	FALSE	FALSE	TRUE
RB1	hgnc:9884	RB1	CIViC	10-Apr-24	NULL	0.6035364509849942	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.036212187	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.005943143	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.011435427	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.015475294	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
FANCA	hgnc:3582	FANCA	CIViC	10-Apr-24	NULL	0.1207072901969988	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
TCF3	hgnc:11633	TCF3	CIViC	10-Apr-24	NULL	NULL	HYPERCVAD REGIMEN	NULL	NULL	NULL	NULL	NULL
TCF3	hgnc:11633	TCF3	CIViC	10-Apr-24	NULL	NULL	NCT00137111	NULL	NULL	NULL	NULL	NULL
NTRK1	hgnc:8031	NTRK1	CIViC	10-Apr-24	NULL	NULL	LAROTRECTINIB REGIMEN	NULL	NULL	NULL	NULL	NULL
RRM1	hgnc:10451	RRM1	CIViC	10-Apr-24	NULL	0.2324817828272369	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SMARCA4	hgnc:11100	SMARCA4	CIViC	10-Apr-24	NULL	0.045265234	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GNAS	hgnc:4392	GNAS	CIViC	10-Apr-24	NULL	0.010346339	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	CIViC	10-Apr-24	NULL	0.03409589	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.3547815624033412	MEK INHIBITOR CI-1040	ncit:C2670	MEK INHIBITOR CI-1040	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	BUTYL 2-AMINOBENZOATE	chembl:CHEMBL1558498	BUTYL 2-AMINOBENZOATE	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DoCM	10-Apr-24	NULL	2.212697851403848	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DoCM	10-Apr-24	NULL	1.184383561707394	AFATINIB	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DoCM	10-Apr-24	NULL	0.637458239	NILOTINIB	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	DoCM	10-Apr-24	NULL	0.4278402841426959	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	4-HYDROXYESTRADIOL	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DoCM	10-Apr-24	NULL	0.6050266644442165	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.009996701	Cediranib	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	EBI-907	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	DS03090629	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	PHI-501	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	SJ-C1044	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	JSI-1187	ncit:C174203	ERK1/2 INHIBITOR JSI-1187	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	BGB3290	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	PET-16	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	ST-162	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	SYM004	ncit:C91381	FUTUXIMAB/MODOTUXIMAB MIXTURE	FALSE	TRUE	TRUE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	GSK8062	chembl:CHEMBL476302	CHEMBL:CHEMBL476302	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	DCC-3084	NULL	NULL	NULL	NULL	NULL
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.7955707762984014	NMS-P715	iuphar.ligand:9401	NMS-P715	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.1223955040459079	Temsirolimus	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
DNMT3A	hgnc:2978	DNMT3A	JAX-CKB	10-Apr-24	NULL	0.088396753	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.036262204	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	1.842374429322613	PLX8394	drugbank:DB16038	PLX8394	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	NULL	NGI-1	NULL	NULL	NULL	NULL	NULL
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.029740964	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1356787370431382	RO5126766	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.2035181055647073	Trabectedin	rxcui:1716278	TRABECTEDIN	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	NULL	AZ8010	NULL	NULL	NULL	NULL	NULL
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	NULL	AZ8010	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.6105543166941221	GSK3052230	ncit:C77970	FGF RECEPTOR ANTAGONIST HGS1036	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.7369497717290455	Pemigatinib	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.1744440904840348	LY3214996	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	NULL	BPR1J373	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.6326225450083675	Flumatinib	hemonc:38662	FLUMATINIB	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	0.027047221	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.4735540335109532	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	JAX-CKB	10-Apr-24	NULL	1.640864726115453	Pinometostat	ncit:C103179	PINOMETOSTAT	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.010505737	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	NULL	DS03090629	NULL	NULL	NULL	NULL	NULL
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	NULL	RO4927350	NULL	NULL	NULL	NULL	NULL
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	NULL	YX-02-030	NULL	NULL	NULL	NULL	NULL
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.03378872	Leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
MSH3	hgnc:7326	MSH3	JAX-CKB	10-Apr-24	NULL	1.193356164447602	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	SBI-0640726	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	BI-69A11	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	Belvarafenib	ncit:C121646	BELVARAFENIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	LY3009120	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.0343337	Leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1154860804304131	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	PLX7904	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	UCM-1336	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	DS03090629	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	JDQ443	ncit:C177916	OPNURASIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	ABT-737	drugbank:DB17023	ABT-737	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.030386384	GSK690693	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	A-1210477	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.037398626	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.088695391	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	A-1210477	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	OP449	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	DETD-35	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.7095631248066824	CX-5461	chembl:CHEMBL4303309	CX-5461	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	BI-69A11	NULL	NULL	NULL	NULL	NULL
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	NULL	ST-162	NULL	NULL	NULL	NULL	NULL
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.1270603054705251	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	0.2715914029432474	Trichostatin A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	NULL	ELR510444	NULL	NULL	NULL	NULL	NULL
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1767935058440892	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.1166837138570989	AMINOPHYLLINE	rxcui:689	AMINOPHYLLINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.2442217266776488	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
CDK13	hgnc:1733	CDK13	ChEMBL	33	inhibitor	0.5000730593875666	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.085937269	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.005618798	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.024773612	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	PharmGKB	4/5/24	NULL	0.08914715	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.018106094	IUPHAR.LIGAND:22	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:10584	iuphar.ligand:10584	DONECOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:609	rxcui:1440856	CHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	agonist	0.1280674908187671	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:3484	iuphar.ligand:3484	[35S]NON-PEPTIDE OT ANTAGONIST	FALSE	FALSE	FALSE
NCBIGENE:597	hgnc:991	BCL2A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8902	drugbank:DB02110	PROTOPORPHYRIN IX CONTAINING CO	FALSE	FALSE	FALSE
ABL2	hgnc:77	ABL2	DTC	9/2/20	inhibitor	0.027664737	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006113363	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	TCMDC-124544	chembl:CHEMBL531322	CHEMBL:CHEMBL531322	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.039899446	NSC-693571	chembl:CHEMBL1287983	CHEMBL:CHEMBL1287983	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.01555322	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
PA	hgnc:8549	BLOC1S6	ChEMBL	33	inhibitor	17.50255707856483	BALOXAVIR MARBOXIL	rxcui:2099995	BALOXAVIR MARBOXIL	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	PharmGKB	4/5/24	NULL	0.015702055	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.088248187	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
UNIPROT:P29371	hgnc:11528	TACR3	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	TALNETANT	ncit:C76464	TALNETANT	FALSE	FALSE	FALSE
UNIPROT:P98194	hgnc:13211	ATP2C1	TdgClinicalTrial	Jan-14	NULL	0.8468979231563629	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	AT13387	ncit:C85454	ONALESPIB	FALSE	FALSE	TRUE
SOLUTE CARRIER FAMILY 12 MEMBER 3	hgnc:10912	SLC12A3	TTD	2020.06.01	NULL	2.917092846427472	Metolazone	rxcui:6916	METOLAZONE	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.06714536	HYDROCHLOROTHIAZIDE	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	2.500365296937833	IUPHAR.LIGAND:2333	iuphar.ligand:2333	COMPOUND RAC-16 [PMID: 15603962]	FALSE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.039068208	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
PRKCE	hgnc:9401	PRKCE	DTC	9/2/20	NULL	1.050153425	[3H]-PHORBOL 12,13-DIBUTYRATE	chembl:CHEMBL27768	CHEMBL:CHEMBL27768	FALSE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	0.5966780822238011	RUCAPARIB	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.024479101	ALBUTEROL	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PROPARGITE	chembl:CHEMBL1416084	PROPARGITE	FALSE	FALSE	FALSE
PTK6	hgnc:9617	PTK6	DTC	9/2/20	NULL	0.2734774543525755	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ISOPIMPINELLIN	ncit:C63673	ISOPIMPINELLIN	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.054355767	CEP-11981	iuphar.ligand:8189	CEP-11981	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.024130364	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.041672755	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.008854582	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	AM-404	iuphar.ligand:12556	AM404	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	CID 752709	chembl:CHEMBL429335	CHEMBL:CHEMBL429335	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.016206071	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	2.333674277141977	CNTO-95	ncit:C61070	INTETUMUMAB	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.029301156	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
UNIPROT:Q70Z44	hgnc:24004	HTR3D	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	DDP225	chembl:CHEMBL5095232	DDP-225	FALSE	FALSE	FALSE
UNIPROT:P15941	hgnc:7508	MUC1	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	GO-203-2C	drugbank:DB15008	GO-203-2C	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	RS-39604	drugbank:DB17050	RS-39604	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1185944014357865	DOMPERIDONE	rxcui:3626	DOMPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:845	iuphar.ligand:845	CXCL12&BETA;	FALSE	FALSE	FALSE
NCBIGENE:313	hgnc:548	AOAH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:5801	iuphar.ligand:5801	4-(N-PROPYL)AMINO-3-NITROBENZOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1243	ncbigene:1243	CMM	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:5094	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.04573839	IUPHAR.LIGAND:2805	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.04573839	IUPHAR.LIGAND:2805	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:1522	iuphar.ligand:1522	[ALA31,AIB32]NPY (PIG)	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.1296485709523321	Selinexor	rxcui:2178390	SELINEXOR	TRUE	FALSE	TRUE
UNIPROT:P10912	hgnc:4263	GHR	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	ARX201	drugbank:DB05082	ARX201	FALSE	FALSE	FALSE
UNIPROT:P15538	hgnc:2591	CYP11B1	TEND	1-Aug-11	NULL	5.250767123569449	METYRAPONE	rxcui:6923	METYRAPONE	TRUE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:3877	rxcui:259264	GANIRELIX ACETATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	3,5 DIBROMOTYROSINE	chembl:CHEMBL1232132	DIBROMOTYROSINE	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.095468493	FLUPHENAZINE HYDROCHLORIDE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.02896176	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.2302968036653267	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1750255707856483	2-BROMO-HEXADECANOIC ACID	chembl:CHEMBL118417	CHEMBL:CHEMBL118417	FALSE	FALSE	FALSE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	0.076765601	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
INTERLEUKIN-12 BETA	hgnc:5970	IL12B	TTD	2020.06.01	NULL	0.1172046232939609	Isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	TICLOPIDINE	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:6033	iuphar.ligand:6033	RHO KINASE INHIBITOR IV	FALSE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.3580068493342807	SUPROFEN	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	AZAMETHIPHOS	chembl:CHEMBL1867031	AZAMETHIPHOS	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.030996264	METARAMINOL	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
NCBIGENE:2957	hgnc:4646	GTF2A1	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:9671	iuphar.ligand:9671	COMPOUND 8C [PMID: 28760529]	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.036718651	BGT-226	iuphar.ligand:7951	BGT-226	FALSE	FALSE	FALSE
NCBIGENE:2429	hgnc:3939	FRA9E	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:9413	iuphar.ligand:9413	VLX1570	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.048618214	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.042619863	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	DTC	9/2/20	NULL	0.029833904	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.079197091	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
MC1R	hgnc:6929	MC1R	PharmGKB	4/5/24	NULL	0.4839416703750645	isoflurane	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.020218587	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
PTGER4	hgnc:9596	PTGER4	PharmGKB	4/5/24	NULL	0.187193124	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.055271233	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TEND	1-Aug-11	NULL	1.312691780892362	CARPHENAZINE	ncit:C73285	CARPHENAZINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.065226921	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:3977	iuphar.ligand:3976	[125I]EPIBATIDINE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.038187397	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.039184829	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.03140411	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.3241214273808303	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.015475294	lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	SILVER SULFADIAZINE	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	TALC	12-May-16	inhibitor	0.1108075556053025	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.04464938	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	1.544343271638073	Tipelukast	ncit:C74581	TIPELUKAST	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.015930725	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.026319635	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.9546849315580818	ARRY-382	iuphar.ligand:9108	ARRY-382	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.3500511415712966	NSC-339578	chembl:CHEMBL353764	CHEMBL:CHEMBL353764	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
MYELIN-ASSOCIATED GLYCOPROTEIN	hgnc:6783	MAG	TTD	2020.06.01	NULL	17.50255707856483	GSK249320	chembl:CHEMBL3545317	REFANEZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:9788	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:4165	iuphar.ligand:4165	CX516	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.2075402025126264	IUPHAR.LIGAND:6056	drugbank:DB07288	N-(4-CHLOROPHENYL)-2-[(PYRIDIN-4-YLMETHYL)AMINO]BENZAMIDE	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	agonist	0.5147810905460244	IUPHAR.LIGAND:8709	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.045304289	abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	DNDI1417722	chembl:CHEMBL1503190	CHEMBL:CHEMBL1503190	FALSE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	inhibitor	0.1041818873724097	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.1651184630053286	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	BRL-50481	iuphar.ligand:5154	BRL50481	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	1.875273972703375	LY-2300559	drugbank:DB13016	LY-2300559	FALSE	FALSE	FALSE
NCBIGENE:1328	hgnc:2621	CYP2C19	GuideToPharmacology	2024.1	inhibitor	0.036162308	IUPHAR.LIGAND:12037	iuphar.ligand:12037	UE2343	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.2476776945079929	DPPE	ncit:C75196	TESMILIFENE	FALSE	FALSE	FALSE
MSH2	hgnc:7325	MSH2	PharmGKB	4/5/24	NULL	0.040235763	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P56524	hgnc:14063	HDAC4	TdgClinicalTrial	Jan-14	NULL	0.1630673019742065	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.089501712	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
NCBIGENE:1617	hgnc:2682	DAZ1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8654	iuphar.ligand:8654	M826	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:5959	iuphar.ligand:5959	NU-7026	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.026136223	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.03337352	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ADRM1	hgnc:15759	ADRM1	DTC	9/2/20	NULL	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
GRIA4	hgnc:4574	GRIA4	ChEMBL	33	positive modulator	0.596678082	CX1739	chembl:CHEMBL3707399	CX1739	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.02339914	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.1581556362520918	IUPHAR.LIGAND:7110	rxcui:279645	ALMOTRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:1480	iuphar.ligand:1480	PANCREATIC POLYPEPTIDE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.019079822	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.011162345	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.3860858179095183	mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.005955952	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.073437302	PIROXICAM	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	0.1092771513750145	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.3125456621172291	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
SMAD2	hgnc:6768	SMAD2	NCI	14-Sep-17	NULL	0.1442518440541057	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.4070362111294147	THIABENDAZOLE	rxcui:10450	THIABENDAZOLE	TRUE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	0.025244073	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:1414	iuphar.ligand:1414	MAP4	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.1479089330582944	GW559768X	chembl:CHEMBL237347	GW559768X	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.016501468	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PREGNENOLONE	rxcui:114052	PREGNENOLONE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.010388507	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	0.6908904109959803	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.021431703	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.061055432	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.025123288	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.068191781	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.1875273972703375	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
NCBIGENE:59	hgnc:130	ACTA2	GuideToPharmacology	2024.1	modulator	1.591141552596803	IUPHAR.LIGAND:9431	iuphar.ligand:9431	CCR2-RA-[R]	FALSE	FALSE	FALSE
NCBIGENE:2534	hgnc:4037	FYN	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:8797	iuphar.ligand:8797	COMPOUND 13 [PMID: 17502136]	FALSE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.042619863	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.090452491	DIPIVEFRIN HYDROCHLORIDE	rxcui:203156	DIPIVEFRIN HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	PharmGKB	4/5/24	NULL	0.029540181	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
NCBIGENE:2904	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.6731752722524935	IUPHAR.LIGAND:9227	iuphar.ligand:9227	COMPOUND 18C [PMID: 25901531]	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	1.184383561707394	BIBW 2992	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.016429184	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.079557078	9-AMINOCAMPTOTHECIN	drugbank:DB12515	9-AMINOCAMPTOTHECIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	GARCINOLIC ACID	chembl:CHEMBL1456870	GARCINOLIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	NCI	14-Sep-17	NULL	0.094099769	N-METHYL-N-NITROSOUREA	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
UNIPROT:P50750	hgnc:1780	CDK9	TdgClinicalTrial	Jan-14	NULL	0.6806549974997433	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
NCBIGENE:1972	hgnc:19338	CDK19	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8945	iuphar.ligand:8945	CCT251545	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.1389091831632129	LY3009120	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.02804897	CUDC-907	ncit:C104008	FIMEPINOSTAT	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.037081689	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	5.527123287967842	IUPHAR.LIGAND:11421	ncit:C91100	EMVODODSTAT	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1025540453822158	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:11716	iuphar.ligand:11716	LONDAMOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2084	hgnc:6861	MAP3K9	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	GNF-PF-3537	chembl:CHEMBL601110	CHEMBL:CHEMBL601110	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.019676849	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00899412	SOFALCONE	ncit:C81118	SOFALCONE	FALSE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.5385402178019949	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	PEMIROLAST	rxcui:19551	PEMIROLAST	TRUE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	0.2966535098061835	ACE-011	ncit:C80038	SOTATERCEPT	FALSE	FALSE	TRUE
CHRNE	hgnc:1966	CHRNE	ChEMBL	33	inhibitor	0.5527123287967842	PIPECURONIUM BROMIDE	rxcui:66983	PIPECURONIUM BROMIDE	TRUE	FALSE	FALSE
KCNJ5	hgnc:6266	KCNJ5	ChEMBL	33	blocker	0.9723642821424906	VERNAKALANT HYDROCHLORIDE	ncit:C152865	VERNAKALANT HYDROCHLORIDE	FALSE	FALSE	FALSE
CATIONIC TRYPSINOGEN	hgnc:9475	PRSS1	TTD	2020.06.01	NULL	0.305277158	Bortezomib	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PROLYL 4-HYDROXYLASESUBUNIT ALPHA-1	hgnc:8546	P4HA1	TTD	2020.06.01	NULL	17.50255707856483	Lufironil	ncit:C97361	LUFIRONIL	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.5000730593875666	AMG-208	drugbank:DB08079	AMG-208	FALSE	FALSE	FALSE
RPL7A	hgnc:10364	RPL7A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.1000146118775133	NINGETINIB	drugbank:DB16256	NINGETINIB	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.046343929	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:9588	iuphar.ligand:9588	PEPTIDE 5 [PMID: 28562585]	FALSE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	TALC	12-May-16	inhibitor	1.640864726115453	OSI 027	chembl:CHEMBL3120215	OSI-027	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.012154554	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.7955707762984014	TESAGLITAZAR	ncit:C75985	TESAGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	modulator	0.3163112725041837	IUPHAR.LIGAND:137	iuphar.ligand:137	5-HT-MODULINE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.094864808	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.039390601	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011806109	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	PHOSALONE	chembl:CHEMBL1528531	PHOSALONE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.010271454	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	4'-EPICHAETOVIRIDIN A	chembl:CHEMBL1306556	CHEMBL:CHEMBL1306556	FALSE	FALSE	FALSE
UNIPROT:P31749	hgnc:391	AKT1	TdgClinicalTrial	Jan-14	NULL	0.4930297768609811	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	2.351089756822142	BI-811283	chembl:CHEMBL3545395	BI-811283	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.004227671	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
RPS6KA3	hgnc:10432	RPS6KA3	NCI	14-Sep-17	NULL	0.1875273972703375	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:2764	iuphar.ligand:2764	HYPERFORIN	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	BMS-599626	drugbank:DB12318	BMS-599626	FALSE	FALSE	TRUE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:9915	ncit:C90996	PAMAPIMOD	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.027333509	pioglitazone	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1527273741585063	RO5126766	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
OR4D6	hgnc:15175	OR4D6	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	ZINC 00035263	chembl:CHEMBL2059068	CHEMBL:CHEMBL2059068	FALSE	FALSE	FALSE
STAT5B	hgnc:11367	STAT5B	CIViC	10-Apr-24	NULL	10.50153424713889	MULTI-SUBTYPE NATURAL HUMAN LEUKOCYTE INTERFERON ALPHA	ncit:C97509	MULTI-SUBTYPE NATURAL HUMAN LEUKOCYTE INTERFERON ALPHA	FALSE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.002429898	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.041672755	FLAVOPIRIDOL	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.005036707	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.3571950424196904	NELFINAVIR	rxcui:134527	NELFINAVIR	TRUE	FALSE	TRUE
EPM2A	hgnc:3413	EPM2A	PharmGKB	4/5/24	NULL	0.2239133101735373	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P08473	hgnc:7154	MME	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	CANDOXATRIL	ncit:C171870	CANDOXATRIL	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR 4	hgnc:11850	TLR4	TTD	2020.06.01	NULL	1.521961485092594	Cadi-05	ncit:C77884	TLR AGONIST CADI-05	FALSE	FALSE	FALSE
NCBIGENE:3024	hgnc:4715	H1-1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:2919	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	DTC	9/2/20	NULL	0.023274677	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:P20839	hgnc:6052	IMPDH1	TEND	1-Aug-11	NULL	0.6563458904461812	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
FGFR1	hgnc:3688	FGFR1	TALC	12-May-16	antibody	0.4907258993990139	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.099446347	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.026227608	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
SSTR2	hgnc:11331	SSTR2	NCI	14-Sep-17	NULL	0.1100789753368857	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.061055432	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.014883127	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	agonist	0.035430277	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
CSNK1G1	hgnc:2454	CSNK1G1	DTC	9/2/20	NULL	0.065634589	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.068191781	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	TEBUFENPYRAD	chembl:CHEMBL1897070	TEBUFENPYRAD	FALSE	FALSE	FALSE
HTR7	hgnc:5302	HTR7	PharmGKB	4/5/24	NULL	0.2917092846427472	venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	0.3750547945406749	MELEVODOPA	ncit:C83927	MELEVODOPA	TRUE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	JAX-CKB	10-Apr-24	NULL	0.251232877	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	1.040600372117402	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.8468979231563628	Dimethindene	rxcui:3449	DIMETHINDENE	TRUE	FALSE	FALSE
NCBIGENE:674	ncbigene:674	BRAFPS1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:7074	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.4134462302023188	CHLORISONDAMINE	ncit:C83619	CHLORISONDAMINE	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.045579576	IUPHAR.LIGAND:6057	iuphar.ligand:6057	VEGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	1.312691780892362	ALRN-6924	ncit:C118669	SULANEMADLIN	FALSE	FALSE	FALSE
IGHE	hgnc:5522	IGHE	ChEMBL	33	inhibitor	8.751278539282415	TALIZUMAB	ncit:C95796	TALIZUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.5223276196220918	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004428038	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	2.333674277141977	IL-17	ncit:C1684	RECOMBINANT INTERLEUKIN-17	FALSE	FALSE	FALSE
UNIPROT:P23458	hgnc:6190	JAK1	TdgClinicalTrial	Jan-14	NULL	1.494525746746522	INCB18424	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.085239726	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	CNV2197944	chembl:CHEMBL3545172	CNV2197944	FALSE	FALSE	FALSE
NCBIGENE:2114	hgnc:3489	ETS2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:8180	iuphar.ligand:8180	COMPOUND 31 [PMID: 20936789]	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.037081689	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
POLE2	hgnc:9178	POLE2	ChEMBL	33	inhibitor	0.094099769	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.1902451856365742	SEMAPIMOD	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:5263	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2032	iuphar.ligand:2032	BIM 23023	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.014464923	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
BCL2	hgnc:990	BCL2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.023716202	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	GNF-PF-4832	chembl:CHEMBL601137	CHEMBL:CHEMBL601137	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001085497	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	2.187819634820604	N-OXALYLGLYCINE	chembl:CHEMBL90852	N-OXALYLGLYCINE	FALSE	FALSE	FALSE
ISG15	hgnc:4053	ISG15	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.8334550989792777	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UGT1A10	hgnc:12531	UGT1A10	NCI	14-Sep-17	NULL	0.3768493150887165	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.085332077	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.016634776	Etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.052507671	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006349558	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002657809	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	GNF-PF-2298	chembl:CHEMBL578905	CHEMBL:CHEMBL578905	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 1	hgnc:4584	GRIN1	TTD	2020.06.01	NULL	0.5357925636295356	D-Serine	ncit:C61739	D-SERINE	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2335	iuphar.ligand:2335	SKA-31	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:2107	iuphar.ligand:2107	NOLPITANTIUM	FALSE	FALSE	FALSE
NCBIGENE:2800	hgnc:4424	GOLGA1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:8011	iuphar.ligand:8011	KU-0060648	FALSE	FALSE	TRUE
SV2A	hgnc:20566	SV2A	ChEMBL	33	modulator	0.5527123287967842	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	DTC	9/2/20	NULL	0.013905633	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.030670369	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.093346971	TREPROSTINIL	rxcui:343048	TREPROSTINIL	TRUE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:9008	iuphar.ligand:9008	COMPOUND 5D [PMID: 25815150]	FALSE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	0.1881995384791917	IUPHAR.LIGAND:7885	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.010537361	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	0.7778914257139926	ISTAROXIME	ncit:C83849	ISTAROXIME	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	DTC	9/2/20	NULL	2.500365296937833	GERONTOXANTHONE B	chembl:CHEMBL478938	GERONTOXANTHONE B	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	Fleroxacin	rxcui:42322	FLEROXACIN	FALSE	FALSE	FALSE
NCBIGENE:2225	hgnc:11408	STK4	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:11811	iuphar.ligand:11811	SBP-3264	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.04440395	Cediranib	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
ATR	hgnc:882	ATR	NCI	14-Sep-17	NULL	0.048282916	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.081092929	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1041818873724097	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	chembl:CHEMBL1449651	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	FALSE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	1.193356164447602	FILOREXANT	ncit:C169980	FILOREXANT	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.061773731	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1310	iuphar.ligand:1310	S36541	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	1.544343271638073	IUPHAR.LIGAND:4101	iuphar.ligand:4101	HYP 9	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.077273983	MPI-0479605	iuphar.ligand:9399	MPI-0479605	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	ChEMBL	33	inhibitor	0.9376369863516875	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	LIPIDYL PSEUDOPTERANE D	chembl:CHEMBL449388	LIPIDYL PSEUDOPTERANE D	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:6687	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	agonist	0.036062961	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
NCBIGENE:2366	hgnc:3874	FRA1G	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:6564	iuphar.ligand:6564	PHENYLACETYL-ARG-VAL-ARG-4-AMIDINOBENZYLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:698	ncbigene:698	BTS1	GuideToPharmacology	2024.1	blocker	7.501095891	IUPHAR.LIGAND:4097	iuphar.ligand:4097	S-(-)CPB	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.01274458	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
CERS6	hgnc:23826	CERS6	PharmGKB	4/5/24	NULL	0.7955707762984016	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.4907258993990139	4-TRIETHYLSILYLPHENOL	chembl:CHEMBL2313445	CHEMBL:CHEMBL2313445	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.063034419	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.050488145	GW559768X	chembl:CHEMBL237347	GW559768X	FALSE	FALSE	FALSE
FBXW7	hgnc:16712	FBXW7	JAX-CKB	10-Apr-24	NULL	0.4251633298436802	Temsirolimus	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
HTR3A	hgnc:5297	HTR3A	PharmGKB	4/5/24	NULL	0.03070624	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.4475085616678508	PROCAINAMIDE	rxcui:8700	PROCAINAMIDE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.025003653	IUPHAR.LIGAND:22	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.008854582	PIRENZEPINE	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
NCBIGENE:2763	ncbigene:2763	GMFA	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:12037	iuphar.ligand:12037	UE2343	FALSE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	antibody	2.917092846427472	IUPHAR.LIGAND:11125	iuphar.ligand:11125	PF-07062119	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	SULISOBENZONE	rxcui:1311567	SULISOBENZONE	TRUE	FALSE	FALSE
UNIPROT:RNA-SEQUENCE	hgnc:11727	TERC	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	IMETELSTAT	ncit:C49084	IMETELSTAT	FALSE	FALSE	TRUE
CACNA1I	hgnc:1396	CACNA1I	ChEMBL	33	blocker	0.8334550989792776	PHENSUXIMIDE	rxcui:33309	PHENSUXIMIDE	TRUE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.3906820776465364	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	3,3',4,4',5'-PENTAMETHOXYCHALCONE	chembl:CHEMBL190474	CHEMBL:CHEMBL190474	FALSE	FALSE	FALSE
UNIPROT:P00740	hgnc:3551	F9	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	FACTOR VIII	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TdgClinicalTrial	Jan-14	NULL	6.848826682916673	FELYPRESSIN	rxcui:4319	FELYPRESSIN	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:1326	iuphar.ligand:1326	[125I]NDP-MSH	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.061412481	L-755507	iuphar.ligand:3931	L 755507	FALSE	FALSE	FALSE
NCBIGENE:599	hgnc:995	BCL2L2	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:2740	iuphar.ligand:2740	ALRT 1550	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2218	iuphar.ligand:2218	D(CH2)5[TYR(ME)2,THR4,PHE(3125I,4N3)-NH29]OVT	FALSE	FALSE	FALSE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.1136529680426287	Sulindac	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	FLAZALONE	ncit:C80552	FLAZALONE	FALSE	FALSE	FALSE
ARHGAP28	hgnc:25509	ARHGAP28	PharmGKB	4/5/24	NULL	7.001022831425933	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.034727296	METARAMINOL	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.044498026	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
SLC22A1	hgnc:10963	SLC22A1	DTC	9/2/20	NULL	0.364636606	TETRYLAMMONIUM	drugbank:DB03095	TETRAMETHYLAMMONIUM	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	CANTHARIDIC_ACID	chembl:CHEMBL275516	CANTHARIDIC_ACID	FALSE	FALSE	FALSE
TSHB	hgnc:12372	TSHB	NCI	14-Sep-17	NULL	2.763561643983921	OESTROGENS	ncit:C483	THERAPEUTIC ESTROGEN	FALSE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.054581779	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.014977128	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	inhibitor	0.039068208	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
CHEK1	hgnc:1925	CHEK1	DTC	9/2/20	NULL	0.032899543	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	0.9376369863516874	INTERFERON ALPHA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
UNIPROT:P49190	hgnc:9609	PTH2R	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	OSTABOLIN-C	chembl:CHEMBL4802222	OSTABOLIN-C	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:387	iuphar.ligand:387	FR194921	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.028004091	IUPHAR.LIGAND:22	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.029665351	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:7501	iuphar.ligand:7501	RGFP109	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.016970805	IUPHAR.LIGAND:1605	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.009443826	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.01514062	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	CLEMIZOLE	ncit:C81139	CLEMIZOLE	FALSE	FALSE	FALSE
MBNL1	hgnc:6923	MBNL1	DTC	9/2/20	NULL	0.6250913242344582	RAMATROBAN	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	3,7-DIMETHOXYFLAVONE	chembl:CHEMBL1449187	3,7-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.063331621	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	2.763561643983921	TTP889	drugbank:DB05131	TTP889	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009875432	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
UNIPROT:O15111	hgnc:1974	CHUK	TdgClinicalTrial	Jan-14	NULL	0.1704794520639432	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	RS-39604	drugbank:DB17050	RS-39604	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	NSC-32984	chembl:CHEMBL1339015	CHEMBL:CHEMBL1339015	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.024309107	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	CLOCORTOLONE PIVALATE	rxcui:21249	CLOCORTOLONE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.013935157	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2892984641085096	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1250182648468916	SJ000114740	chembl:CHEMBL592068	CHEMBL:CHEMBL592068	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2246	iuphar.ligand:2246	L-367,773	FALSE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	1.193356164447602	HISTRELIN ACETATE	rxcui:1294622	HISTRELIN ACETATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	(+)-THALIPORPHINE	chembl:CHEMBL1397308	CHEMBL:CHEMBL1397308	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	L-755507	iuphar.ligand:3931	L 755507	FALSE	FALSE	FALSE
IL13RA1	hgnc:5974	IL13RA1	ChEMBL	33	binder	17.50255707856483	CINTREDEKIN BESUDOTOX	ncit:C2599	CINTREDEKIN BESUDOTOX	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.9634435089118256	CLOCINNAMOX	chembl:CHEMBL386492	CLOCINNAMOX	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	0.096123883	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
UNIPROT:P30049	hgnc:837	ATP5F1D	TdgClinicalTrial	Jan-14	NULL	0.6775183385250904	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
NCBIGENE:63	hgnc:136	ACTBP3	GuideToPharmacology	2024.1	agonist	10.50153424713889	IUPHAR.LIGAND:3654	iuphar.ligand:3654	[125I]CCL20 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4161	iuphar.ligand:4161	CONANTOKIN-G	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8113	iuphar.ligand:8113	XL413	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.020226376	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:10366	iuphar.ligand:10366	XY101	FALSE	FALSE	FALSE
SREBF1	hgnc:11289	SREBF1	NCI	14-Sep-17	NULL	1.981421556063943	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
HSPB2	hgnc:5247	HSPB2	NCI	14-Sep-17	NULL	0.072125922	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
AMH	hgnc:464	AMH	NCI	14-Sep-17	NULL	0.280789686	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005864158	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.035418328	LEUPRORELIN ACETATE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.04593847	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.056826484	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.024108205	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.4039051633514962	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.003422925	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.044198376	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
MT3	hgnc:7408	MT3	NCI	14-Sep-17	NULL	5.527123287967842	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 1	hgnc:6026	CXCR1	TTD	2020.06.01	NULL	3.000438356	SCH-527123	iuphar.ligand:8497	NAVARIXIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007063179	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.1721562991334246	TAK-593	drugbank:DB13093	TAK-593	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.067839369	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.045579576	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	CIPROFLOXACIN HYDROCHLORIDE	rxcui:81981	CIPROFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.280789686	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000290256	chembl:CHEMBL590666	CHEMBL:CHEMBL590666	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.017649637	MIBEFRADIL	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.027650169	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.013087655	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003139923	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.086361301	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.07699072	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.018867291	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008558708	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.1535312024435511	IUPHAR.LIGAND:743	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:6239	iuphar.ligand:6239	ASPIRIN-TRIGGERED RESOLVIN D1	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	NCI	14-Sep-17	NULL	0.105015342	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.038608582	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
POMC	hgnc:9201	POMC	PharmGKB	4/5/24	NULL	52.50767123569449	alpha-MSH	drugbank:DB17612	INTERMEDINE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.729273212	4-METHYLUMBELLIFERYL ACETATE	chembl:CHEMBL12019	CHEMBL:CHEMBL12019	FALSE	FALSE	FALSE
PSMD3	hgnc:9560	PSMD3	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GNF-PF-3955	chembl:CHEMBL605747	CHEMBL:CHEMBL605747	FALSE	FALSE	FALSE
SMARCA2	hgnc:11098	SMARCA2	DTC	9/2/20	NULL	2.187819634820604	TCMDC-125813	chembl:CHEMBL580076	CHEMBL:CHEMBL580076	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
MSTN	hgnc:4223	MSTN	ChEMBL	33	inhibitor	2.187819634820604	RAMATERCEPT	ncit:C152151	RAMATERCEPT	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	agonist	0.041540879	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.8899605294185507	IUPHAR.LIGAND:3245	iuphar.ligand:3245	[125I]SB258585	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.091583148	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	modulator	0.210030685	NETOGLITAZONE	ncit:C72822	NETOGLITAZONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	GNF-PF-2383	chembl:CHEMBL578915	CHEMBL:CHEMBL578915	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	ChEMBL	33	inhibitor	0.2567612285364034	OLUTASIDENIB	rxcui:2623641	OLUTASIDENIB	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.005359019	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PIRITREXIM ISETHIONATE	ncit:C91407	PIRITREXIM ISETHIONATE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004517955	RAUWOLFIA SERPENTINA	rxcui:17205	AJMALICINE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.1419126249613365	PROPANTHELINE BROMIDE	rxcui:8762	PROPANTHELINE BROMIDE	TRUE	FALSE	FALSE
UNIPROT:P34998	hgnc:2357	CRHR1	TdgClinicalTrial	Jan-14	NULL	0.729273212	CORTICOTROPIN-RELEASING FACTOR	iuphar.ligand:913	CORTICOTROPIN-RELEASING FACTOR	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	BERGAPTEN	rxcui:15842	5-METHOXYPSORALEN	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.8607814956671229	ETHYNODIOL DIACETATE	rxcui:4170	ETHYNODIOL DIACETATE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:343	iuphar.ligand:343	BRUCINE N-OXIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.6563458904461812	GNF-PF-1859	chembl:CHEMBL1520837	CHEMBL:CHEMBL1520837	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.018699313	FLUVOXAMINE	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.022249013	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.2822993077187876	TV-45070	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.016780975	METARAMINOL	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.012504804	MIBEFRADIL	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
AKAP13	hgnc:371	AKAP13	PharmGKB	4/5/24	NULL	1.381780822	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
EXTRACELLULAR CALCIUM-SENSING RECEPTOR	hgnc:1514	CASR	TTD	2020.06.01	NULL	1.640864726115453	AXT-914	iuphar.ligand:10696	AXT914	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.03223307	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.025672984	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.1744440904840348	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:433	iuphar.ligand:433	VISNAGIN	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.030368809	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3558	iuphar.ligand:3558	DESULFATED GASTRIN-14	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	FLAVONE	rxcui:1536070	FLAVONE	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.055978328	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.2573905452730122	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
UNIPROT:P01584	hgnc:5992	IL1B	TEND	1-Aug-11	NULL	2.573905452730122	CANAKINUMAB	rxcui:853491	CANAKINUMAB	TRUE	TRUE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TRIFLUPERIDOL HYDROCHLORIDE	rxcui:236140	TRIFLUPERIDOL HYDROCHLORIDE	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.8468979231563628	evinacumab	rxcui:2478335	EVINACUMAB	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006434764	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	0.1682938180631233	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NCBIGENE:2035	hgnc:3377	EPB41	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8126	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	1.544343271638073	IUPHAR.LIGAND:2442	iuphar.ligand:2442	SLG	FALSE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.084146909	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.5000730593875666	APRATOXIN F	chembl:CHEMBL2022560	APRATOXIN F	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	TCMDC-124755	chembl:CHEMBL580207	CHEMBL:CHEMBL580207	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	TCMDC-124544	chembl:CHEMBL531322	CHEMBL:CHEMBL531322	FALSE	FALSE	FALSE
NCBIGENE:2411	hgnc:3922	FRA7D	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8356	iuphar.ligand:8356	PBD150	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.077273983	Bendamustine	rxcui:134547	BENDAMUSTINE	TRUE	FALSE	TRUE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.1077080435603989	Myo-inositol	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.007905401	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	1.193356164447602	DARIDOREXANT	rxcui:2591497	DARIDOREXANT	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	ChEMBL	33	inhibitor	0.1500219178162699	ASN007	chembl:CHEMBL4650280	ASN007	FALSE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:9073	rxcui:1546421	EDROPHONIUM CATION	TRUE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:754	iuphar.ligand:754	CCL15	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10379	ncit:C76508	PEXACERFONT	FALSE	FALSE	FALSE
NCBIGENE:1831	hgnc:3051	TSC22D3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	inhibitor	0.305277158	IUPHAR.LIGAND:2882	ncit:C170255	ONAPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:3318	iuphar.ligand:3318	PSN375963	FALSE	FALSE	FALSE
NCBIGENE:2964	hgnc:4654	GTF2F2P1	GuideToPharmacology	2024.1	blocker	10.50153424713889	IUPHAR.LIGAND:12713	iuphar.ligand:12713	COMPOUND 36 [PMID: 34843241]	FALSE	FALSE	FALSE
TH	hgnc:11782	TH	NCI	14-Sep-17	NULL	0.1470803115845784	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010122936	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	THIOCYCLAM HYDROGEN OXALATE	chembl:CHEMBL2270412	THIOCYCLAM HYDROGEN OXALATE	FALSE	FALSE	FALSE
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	0.09003373	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.000552271	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE ALPHA-3	hgnc:10431	RPS6KA2	TTD	2020.06.01	NULL	3.750547945406749	BI-D1870	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	DTC	9/2/20	NULL	1.458546423213736	CYROMAZINE	chembl:CHEMBL1231107	CYROMAZINE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.010148371	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
CSNK1G2	hgnc:2455	CSNK1G2	DTC	9/2/20	NULL	0.1562728310586145	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.151464436	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
UNIPROT:P12236	hgnc:10992	SLC25A6	TdgClinicalTrial	Jan-14	NULL	0.09741683	CLODRONATE	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
NCBIGENE:2159	hgnc:3528	F10	GuideToPharmacology	2024.1	inhibitor	0.1339481409073839	IUPHAR.LIGAND:5263	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(+)-VENTILOQUINONE L METHYL ETHER	chembl:CHEMBL594259	CHEMBL:CHEMBL594259	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 2	hgnc:3689	FGFR2	TTD	2020.06.01	NULL	0.305277158	Palifermin	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001580319	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	0.3236220106976548	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	1.842374429322613	AM-461	iuphar.ligand:10170	AM-461	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HTR1D	hgnc:5289	HTR1D	ChEMBL	33	inhibitor	1.009762908	ELZASONAN HYDROCHLORIDE	ncit:C73806	ELZASONAN HYDROCHLORIDE	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
CA13	hgnc:14914	CA13	ChEMBL	33	inhibitor	2.187819634820604	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.085239726	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.2	hgnc:1395	CACNA1H	TTD	2020.06.01	NULL	2.442217266776488	ABT-639	drugbank:DB15055	ABT-639	FALSE	FALSE	FALSE
CDH17	hgnc:1756	CDH17	NCI	14-Sep-17	NULL	0.7001022831425933	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.1988926940746003	PHENFORMIN HYDROCHLORIDE	rxcui:235288	PHENFORMIN HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	DTC	9/2/20	NULL	1.640864726115453	NSC-39249	chembl:CHEMBL482792	CHEMBL:CHEMBL482792	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.001915989	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	GINGKOLIC ACID	chembl:CHEMBL445177	GINGKOLIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	HEXYLRESORCINOL	rxcui:5321	HEXYLRESORCINOL	TRUE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	ChEMBL	33	agonist	1.514644363	OLORINAB	ncit:C166825	OLORINAB	FALSE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:9230	iuphar.ligand:9230	COMPOUND 6J [PMID: 27219676]	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:8297	iuphar.ligand:8297	SERIBANTUMAB	FALSE	FALSE	FALSE
NCBIGENE:455	hgnc:760	ASS1P10	GuideToPharmacology	2024.1	agonist	0.3281729452230906	IUPHAR.LIGAND:3309	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.03223307	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
NCBIGENE:1516	hgnc:6515	LATS2	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:5655	iuphar.ligand:5655	A-674563	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.5303805175322676	PROSTAGLANDIN D2	drugbank:DB02056	PROSTAGLANDIN D2	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.00725645	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.082300425	CGS-15943	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	4,5,6,7-TETRABROMOBENZIMIDAZOLE	chembl:CHEMBL373937	CHEMBL:CHEMBL373937	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.4930297768609811	RX-0201	ncit:C88335	ARCHEXIN	FALSE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.092118721	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.076263865	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.6250913242344582	FISPEMIFENE	ncit:C65687	FISPEMIFENE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	ChEMBL	33	inhibitor	0.058733413	TABIMORELIN	ncit:C76887	TABIMORELIN	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	ChEMBL	33	inhibitor	3.281729452230906	FORIGERIMOD ACETATE	ncit:C170004	FORIGERIMOD ACETATE	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.1595977849109255	CILNIDIPINE	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:183	iuphar.ligand:183	LY53857	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1902451856365742	TRITON X	chembl:CHEMBL39763	TRITON X	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DEXBUDESONIDE	ncit:C80814	DEXBUDESONIDE	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.035964158	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	0.212581665	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
APH1A	hgnc:29509	APH1A	ChEMBL	33	inhibitor	0.6250913242344582	RG-4733	drugbank:DB11870	RG-4733	FALSE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	2.917092846427472	DARIDOREXANT HYDROCHLORIDE	rxcui:2591496	DARIDOREXANT HYDROCHLORIDE	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	DTC	9/2/20	NULL	4.773424657790408	TETRA-IODOPHENOLPHTHALEIN	chembl:CHEMBL2324200	TETRA-IODOPHENOLPHTHALEIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.002103673	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.015521038	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.3059887601147698	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6414	iuphar.ligand:6414	5PAM523	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.4773424657790409	DULAGLUTIDE	rxcui:1551291	DULAGLUTIDE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	agonist	0.036463661	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.041672755	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	0.9460841664089098	ETRUMADENANT	ncit:C159564	ETRUMADENANT	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.01864619	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	agonist	0.1422972120208523	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.018106094	IUPHAR.LIGAND:5698	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:252	hgnc:10608	SCTR	GuideToPharmacology	2024.1	agonist	31.50460274141669	IUPHAR.LIGAND:3643	rxcui:606396	SECRETIN HUMAN, SYNTHETIC	TRUE	FALSE	FALSE
RABEP1	hgnc:17677	RABEP1	PharmGKB	4/5/24	NULL	0.142490288	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.1835932560688619	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
TGFB2	hgnc:11768	TGFB2	ChEMBL	33	inhibitor	1.875273972703375	LUSPATERCEPT	rxcui:2262543	LUSPATERCEPT-AAMT	TRUE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:8408	iuphar.ligand:8408	DESULFATED GASTRIN-17	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.050488145	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	ChEMBL	33	inhibitor	0.7544205637312429	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	KP201	chembl:CHEMBL3137310	BENZHYDROCODONE HYDROCHLORIDE	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.048764961	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CIViC	10-Apr-24	NULL	0.1535312024435511	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	NSC-21588	chembl:CHEMBL1611308	CHEMBL:CHEMBL1611308	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1060761035064535	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	0.2763561643983921	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.7955707762984013	(-)-ROLIPRAM	chembl:CHEMBL430893	(-)-ROLIPRAM	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	ATOVAQUONE	rxcui:60212	ATOVAQUONE	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	NCI	14-Sep-17	NULL	0.08914715	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
SMPD1	hgnc:11120	SMPD1	DTC	9/2/20	NULL	0.5048814541893702	AMIODARONE HYDROCHLORIDE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.063858524	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.3409589041278863	WX-554	chembl:CHEMBL3545145	WX-554	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	agonist	0.035890411	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.012573676	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.00777661	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
OX40L RECEPTOR	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	3.500511415712966	MEDI0562	ncit:C120041	TAVOLIMAB	FALSE	FALSE	FALSE
ALPP	hgnc:439	ALPP	NCI	14-Sep-17	NULL	2.333674277141978	BETA-ADRENERGIC ANTAGONIST	ncit:C29576	BETA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
LOH19CR1	hgnc:10402	RPS19	NCI	14-Sep-17	NULL	0.1408971500063358	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.005483257	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	3.088686543276147	IUPHAR.LIGAND:4135	iuphar.ligand:4135	APETX2	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:7058	iuphar.ligand:7058	NQN-1	FALSE	FALSE	FALSE
NCBIGENE:2042	hgnc:3387	EPHA3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8084	iuphar.ligand:8084	COMPOUND 1 [WO2012007375]	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:6069	iuphar.ligand:6069	10,10-DIFLUORO TXA2	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.049723174	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.087952548	CNQX DISODIUM	chembl:CHEMBL1255647	CHEMBL:CHEMBL1255647	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.6563458904461813	XANTHOANGELOL B	chembl:CHEMBL494082	XANTHOANGELOL B	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.024861587	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.1816874437221262	NOCARDAMINE	chembl:CHEMBL505734	NOCARDAMINE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.021554873	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
PROTEIN CEREBLON	hgnc:30185	CRBN	TTD	2020.06.01	NULL	1.458546423213736	CC-220	ncit:C129048	IBERDOMIDE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.4375639269641208	PYRAZOLOACRIDINE	ncit:C1564	PYRAZOLOACRIDINE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.2778183663264259	CO 1686	hemonc:449	ROCILETINIB	FALSE	FALSE	TRUE
GRIK1	hgnc:4579	GRIK1	ChEMBL	33	inhibitor	2.100306849	DASOLAMPANEL	ncit:C166510	DASOLAMPANEL	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.007132256	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.07182992	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	GNF-PF-3955	chembl:CHEMBL605747	CHEMBL:CHEMBL605747	FALSE	FALSE	FALSE
SRD5A1	hgnc:11284	SRD5A1	DTC	9/2/20	NULL	8.751278539282415	LY-266111	chembl:CHEMBL29166	CHEMBL:CHEMBL29166	FALSE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	DTC	9/2/20	NULL	0.1842374429322614	PIPERTRAMINE	chembl:CHEMBL127273	PIPERTRAMINE	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	other/unknown	1.193356164447602	CHLORPHENTERMINE HYDROCHLORIDE	ncit:C65324	CHLORPHENTERMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2763	ncbigene:2763	GMFA	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:7715	iuphar.ligand:7715	AZD8329	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:9812	iuphar.ligand:9812	AZD9567	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	0.1400204566285186	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:11144	iuphar.ligand:11144	COMPOUND 49 [PMID: 30889352]	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2199274187882492	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.021933029	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	DTC	9/2/20	NULL	0.012588749	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.034727296	gliquidone	rxcui:25793	GLIQUIDONE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.045265234	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.035418328	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.028184472	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.098884503	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.375054795	INSULIN ZINC SUSP RECOMBINANT HUMAN	chembl:CHEMBL1201644	INSULIN ZINC SUSP RECOMBINANT HUMAN	TRUE	FALSE	FALSE
SELE	hgnc:10718	SELE	ChEMBL	33	inhibitor	6.364566210387211	RIVIPANSEL	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.159436249	CHLOROPROCAINE	rxcui:20859	CHLOROPROCAINE	TRUE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.030796288	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	MEBEVERINE HYDROCHLORIDE	rxcui:235827	MEBEVERINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.041639708	CLOZAPINE	rxcui:2626	CLOZAPINE	TRUE	FALSE	FALSE
PSMD6	hgnc:9564	PSMD6	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.031273181	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.077789143	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.028078969	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.4102161815288632	PEFLOXACIN	rxcui:7960	PEFLOXACIN	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.2917092846427472	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.5645986154375752	FDG	rxcui:1362737	FLUORODEOXYGLUCOSE F18	TRUE	FALSE	FALSE
UNIPROT:P41594	hgnc:4597	GRM5	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	AZD2066	drugbank:DB17078	AZD2066	FALSE	FALSE	FALSE
UNIPROT:Q08499	hgnc:8783	PDE4D	TdgClinicalTrial	Jan-14	NULL	0.5357925636295358	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:12371	iuphar.ligand:12371	MILREBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1629	iuphar.ligand:1629	NALORPHINE	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	PharmGKB	4/5/24	NULL	0.3365876361262468	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.2243917574174978	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.031301145	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.003091232	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.2692701089009974	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
VCAM1	hgnc:12663	VCAM1	NCI	14-Sep-17	NULL	0.2035181055647073	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003313623	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.062808219	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.093931433	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
TLR3	hgnc:11849	TLR3	ChEMBL	33	activator	5.250767123569449	BEVASIRANIB SODIUM	ncit:C142953	BEVASIRANIB SODIUM	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.11707396	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:1094	iuphar.ligand:1094	[125I][HIS9]GHRELIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1965	iuphar.ligand:1965	TEI-9063	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:8125	iuphar.ligand:8125	COMPOUND 12 [PMID: 22521646]	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.032252869	IUPHAR.LIGAND:1225	rxcui:203179	DOXEPIN HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:4191	iuphar.ligand:4191	FLUFENAMATE	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.5250767123569451	XANTHOANGELOL B	chembl:CHEMBL494082	XANTHOANGELOL B	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.072125922	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.039068208	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	ENPIROLINE	ncit:C75267	ENPIROLINE	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	PharmGKB	4/5/24	NULL	1.810609352954982	crizanlizumab-tmca	rxcui:2262279	CRIZANLIZUMAB	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.084146909	LOXAPINE SUCCINATE	rxcui:6476	LOXAPINE SUCCINATE	TRUE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	ChEMBL	33	inhibitor	0.09003373	PF-00562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.1389091831632129	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.1215455352678113	ACECLOFENAC	rxcui:16689	ACECLOFENAC	TRUE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	NCI	14-Sep-17	NULL	0.2447910080918158	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.027855529	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.030945115	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NCBIGENE:2719	hgnc:4451	GPC3	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:9521	iuphar.ligand:9521	GSK8814	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:10590	iuphar.ligand:10590	(R)-2H [PMID:19625189]	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2990	iuphar.ligand:2990	COMPOUND 1F [PMID: 2153213]	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.015806042	Sapanisertib	rxcui:2395271	SAPANISERTIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	GW3965	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
SLCO1B3	hgnc:10961	SLCO1B3	DTC	9/2/20	NULL	1.400204566285186	DIOSCIN	iuphar.ligand:840	DIOSCIN	FALSE	FALSE	FALSE
EPM2A	hgnc:3413	EPM2A	PharmGKB	4/5/24	NULL	0.1973972602845657	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.089298761	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1346350544504987	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.017363648	ZUCAPSAICIN	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2117244807890907	8-GERANYLOXY PSORALEN	chembl:CHEMBL1412710	CHEMBL:CHEMBL1412710	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:7773	iuphar.ligand:7773	UCM 724	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	0.6403374540938354	IUPHAR.LIGAND:9462	iuphar.ligand:9462	LY2940094	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.2763561643983921	SR9011	iuphar.ligand:8900	SR9011	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.009842113	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005059761	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	NCI	14-Sep-17	NULL	0.081030357	HERBIMYCIN A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	TCMDC-123868	chembl:CHEMBL548615	CHEMBL:CHEMBL548615	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.07614901	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	(S)-NIMODIPINE	chembl:CHEMBL255033	(S)-NIMODIPINE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.007083666	CLONAZEPAM	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	TALC	12-May-16	inhibitor	0.192335792	SARACATINIB	ncit:C48378	SARACATINIB	FALSE	FALSE	TRUE
AKT2	hgnc:392	AKT2	CGI	2/1/22	NULL	0.364636606	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.637458239	Nilotinib	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	CancerCommons	25-Jul-13	inhibitor	0.1704794520639432	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CancerCommons	25-Jul-13	inhibitor	0.1725334213659184	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	CancerCommons	25-Jul-13	antibody	2.972132334095915	CIXUTUMUMAB	ncit:C79828	CIXUTUMUMAB	FALSE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.029244039	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	0.1481697953740938	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
MET	hgnc:7029	MET	CGI	2/1/22	NULL	0.066676408	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
NOTCH1	hgnc:7881	NOTCH1	CGI	2/1/22	NULL	19.69037671338543	OMP-52M51	ncit:C103274	BRONTICTUZUMAB	FALSE	FALSE	TRUE
RAD50	hgnc:9816	RAD50	CGI	2/1/22	NULL	NULL	CHK1	NULL	NULL	NULL	NULL	NULL
ATM	hgnc:795	ATM	CGI	2/1/22	NULL	NULL	CHK1	NULL	NULL	NULL	NULL	NULL
SMO	hgnc:11119	SMO	CGI	2/1/22	NULL	15.31473744374422	Vismodegib	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
ATM	hgnc:795	ATM	CGI	2/1/22	NULL	0.045668773	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PML	hgnc:9113	PML	CGI	2/1/22	NULL	0.384671584	Tretinoin	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
STK11	hgnc:11389	STK11	CGI	2/1/22	NULL	0.9053046764774912	Phenformin	rxcui:8129	PHENFORMIN	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.2917092846427472	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.086861325	ETANERCEPT	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.022286787	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	agonist	0.047049885	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.2075402025126264	THIETHYLPERAZINE MALEATE	rxcui:71529	THIETHYLPERAZINE MALEATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.069180068	THIOTHIXENE HYDROCHLORIDE	rxcui:91135	THIOTHIXENE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	1.693795846312725	BEPOTASTINE BESYLATE	rxcui:658552	BEPOTASTINE BESILATE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	DIPHENYLPYRALINE HYDROCHLORIDE	rxcui:203155	DIPHENYLPYRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	1.186614039224734	VALSARTAN	rxcui:69749	VALSARTAN	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	inhibitor	0.7955707762984014	CETRORELIX ACETATE	rxcui:259338	CETRORELIX ACETATE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	inhibitor	0.2792961235941196	HEXOCYCLIUM METHYLSULFATE	rxcui:235430	HEXOCYCLIUM METHYLSULFATE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1108075556053025	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1988926940746003	PROTRIPTYLINE HYDROCHLORIDE	rxcui:203199	PROTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP BEEF	chembl:CHEMBL1201639	INSULIN ZINC SUSP BEEF	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN SUSP ISOPHANE PURIFIED PORK	chembl:CHEMBL1201656	INSULIN SUSP ISOPHANE PURIFIED PORK	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN ZINC SUSP EXTENDED RECOMBINANT HUMAN	chembl:CHEMBL1201641	INSULIN ZINC SUSP EXTENDED RECOMBINANT HUMAN	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.750109589	INSULIN SUSP ISOPHANE BEEF	chembl:CHEMBL1201545	INSULIN SUSP ISOPHANE BEEF	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.059397818	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.084146909	THIOTHIXENE	rxcui:10510	THIOTHIXENE	TRUE	FALSE	FALSE
HTR2C	hgnc:5295	HTR2C	ChEMBL	33	inhibitor	0.064347636	METHYSERGIDE MALEATE	rxcui:203190	METHYSERGIDE MALEATE	TRUE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	agonist	0.9460841664089098	REGADENOSON	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	ALFENTANIL HYDROCHLORIDE	rxcui:203203	ALFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.358239472	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	MORPHINE SULFATE	rxcui:30236	MORPHINE SULFATE	TRUE	FALSE	FALSE
DDL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CYCLOSERINE	rxcui:3007	CYCLOSERINE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.2408608772279564	ANILERIDINE PHOSPHATE	ncit:C87352	ANILERIDINE PHOSPHATE	TRUE	FALSE	FALSE
SSTR3	hgnc:11332	SSTR3	ChEMBL	33	agonist	1.458546423213736	PASIREOTIDE DIASPARTATE	rxcui:1364104	PASIREOTIDE DIASPARTATE	TRUE	FALSE	FALSE
CYP11A1	hgnc:2590	CYP11A1	ChEMBL	33	inhibitor	4.375639269641208	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.3860858179095183	PYRIDOSTIGMINE BROMIDE	rxcui:9001	PYRIDOSTIGMINE BROMIDE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.400821918	HYDROCORTISONE CYPIONATE	rxcui:163524	HYDROCORTISONE CYPIONATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.080164384	CLOBETASOL PROPIONATE	rxcui:21245	CLOBETASOL PROPIONATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.3006164383722967	FLUMETHASONE PIVALATE	rxcui:25113	FLUMETHASONE PIVALATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.2386712328895204	EMTRICITABINE	rxcui:276237	EMTRICITABINE	TRUE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	ChEMBL	33	inhibitor	0.7740688634254718	SELEGILINE	rxcui:9639	SELEGILINE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	agonist	0.04907259	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.267214612	FLURANDRENOLIDE	rxcui:4500	FLURANDRENOLIDE	TRUE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	ChEMBL	33	inhibitor	3.500511415712966	EPTIFIBATIDE	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
GRIN1	hgnc:4584	GRIN1	ChEMBL	33	inhibitor	0.056399217	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.040051618	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	1.591141552596802	ANAGRELIDE HYDROCHLORIDE	rxcui:236612	ANAGRELIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	1.458546423213736	ANAGRELIDE HYDROCHLORIDE	rxcui:236612	ANAGRELIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.201952582	ALFUZOSIN HYDROCHLORIDE	rxcui:46043	ALFUZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	inhibitor	0.076098074	PRAZOSIN HYDROCHLORIDE	rxcui:203210	PRAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.1902451856365742	PHENYLEPHRINE HYDROCHLORIDE	rxcui:8164	PHENYLEPHRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.1367387271762877	PHENYLEPHRINE HYDROCHLORIDE	rxcui:8164	PHENYLEPHRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1178056726441863	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	BISMUTH SUBSALICYLATE	rxcui:19478	BISMUTH SUBSALICYLATE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	inhibitor	0.082171629	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	blocker	0.5173169579871378	REPAGLINIDE	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.4773424657790409	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2628669398532891	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	ANILERIDINE HYDROCHLORIDE	rxcui:235413	ANILERIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMAD2	hgnc:6768	SMAD2	DTC	9/2/20	NULL	13.12691780892362	GERANIIN	chembl:CHEMBL506069	GERANIIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.1017590527823536	DOBUTAMINE HYDROCHLORIDE	rxcui:203121	DOBUTAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	2.838252499226729	APREPITANT	rxcui:358255	APREPITANT	TRUE	FALSE	FALSE
UREA	NULL	NULL	ChEMBL	33	inhibitor	NULL	ACETOHYDROXAMIC ACID	rxcui:16728	ACETOHYDROXAMIC ACID	TRUE	FALSE	FALSE
UREB	NULL	NULL	ChEMBL	33	inhibitor	NULL	ACETOHYDROXAMIC ACID	rxcui:16728	ACETOHYDROXAMIC ACID	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	GNF-PF-372	chembl:CHEMBL580155	CHEMBL:CHEMBL580155	FALSE	FALSE	FALSE
UREC	NULL	NULL	ChEMBL	33	inhibitor	NULL	ACETOHYDROXAMIC ACID	rxcui:16728	ACETOHYDROXAMIC ACID	TRUE	FALSE	FALSE
PBP4	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLOXACILLIN SODIUM	rxcui:9864	CLOXACILLIN SODIUM	TRUE	FALSE	FALSE
PBPF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLOXACILLIN SODIUM	rxcui:9864	CLOXACILLIN SODIUM	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.076765601	FLUMEQUINE	rxcui:25112	FLUMEQUINE	FALSE	FALSE	FALSE
MECA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLOXACILLIN SODIUM	rxcui:9864	CLOXACILLIN SODIUM	TRUE	FALSE	FALSE
PBP2	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLOXACILLIN SODIUM	rxcui:9864	CLOXACILLIN SODIUM	TRUE	FALSE	FALSE
PBPA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLOXACILLIN SODIUM	rxcui:9864	CLOXACILLIN SODIUM	TRUE	FALSE	FALSE
ERG11	NULL	NULL	ChEMBL	33	inhibitor	NULL	ITRACONAZOLE	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
SLC18A2	hgnc:10935	SLC18A2	ChEMBL	33	inhibitor	0.8751278539282416	DEXTROAMPHETAMINE SACCHARATE	rxcui:221088	DEXTROAMPHETAMINE SACCHARATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.1060761035064535	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.08178765	SIBUTRAMINE HYDROCHLORIDE	rxcui:1294535	SIBUTRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	ECADOTRIL	ncit:C75238	ECADOTRIL	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.1944728564284981	MAZINDOL	rxcui:6664	MAZINDOL	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.099446347	SIBUTRAMINE HYDROCHLORIDE	rxcui:1294535	SIBUTRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE9A	hgnc:8795	PDE9A	ChEMBL	33	inhibitor	0.1875273972703375	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE8A	hgnc:8793	PDE8A	ChEMBL	33	inhibitor	0.5000730593875666	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PTGER2	hgnc:9594	PTGER2	ChEMBL	33	agonist	0.6563458904461813	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.019304291	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
PDE1B	hgnc:8775	PDE1B	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.051731696	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE8A	hgnc:8793	PDE8A	ChEMBL	33	inhibitor	2.187819634820604	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.039598545	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.037666909	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.01311053	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.079557078	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.088396753	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.083257407	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.021715331	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.033232703	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.031254566	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.033658764	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.025439763	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.027914764	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.036770078	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.017306418	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.039598545	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.032016873	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAMETHAZINE	rxcui:10178	SULFAMETHAZINE	TRUE	FALSE	FALSE
FOLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
SRD5A2	hgnc:11285	SRD5A2	ChEMBL	33	inhibitor	13.12691780892362	DUTASTERIDE	rxcui:228790	DUTASTERIDE	TRUE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TRIMETHOPRIM	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	8-GERANYLOXY PSORALEN	chembl:CHEMBL1412710	CHEMBL:CHEMBL1412710	FALSE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TRIMETHOPRIM HYDROCHLORIDE	rxcui:259281	TRIMETHOPRIM HYDROCHLORIDE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.037857009	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEPHAPIRIN SODIUM	rxcui:42562	CEPHAPIRIN SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN INDANYL SODIUM	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN INDANYL SODIUM	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN INDANYL SODIUM	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN INDANYL SODIUM	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN INDANYL SODIUM	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN INDANYL SODIUM	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CARBENICILLIN INDANYL SODIUM	rxcui:56461	CARBENICILLIN INDANYL SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.079077818	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFACLOR	rxcui:1450910	CEFACLOR ANHYDROUS	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTETAN DISODIUM	rxcui:203141	CEFOTETAN DISODIUM	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTETAN DISODIUM	rxcui:203141	CEFOTETAN DISODIUM	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTETAN DISODIUM	rxcui:203141	CEFOTETAN DISODIUM	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTETAN DISODIUM	rxcui:203141	CEFOTETAN DISODIUM	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTETAN DISODIUM	rxcui:203141	CEFOTETAN DISODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFOTETAN DISODIUM	rxcui:203141	CEFOTETAN DISODIUM	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMDINOCILLIN	rxcui:626	AMDINOCILLIN	TRUE	FALSE	FALSE
PBP4	NULL	NULL	ChEMBL	33	inhibitor	NULL	DICLOXACILLIN SODIUM	rxcui:267257	DICLOXACILLIN SODIUM	TRUE	FALSE	FALSE
PBPF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DICLOXACILLIN SODIUM	rxcui:267257	DICLOXACILLIN SODIUM	TRUE	FALSE	FALSE
MECA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DICLOXACILLIN SODIUM	rxcui:267257	DICLOXACILLIN SODIUM	TRUE	FALSE	FALSE
PBP2	NULL	NULL	ChEMBL	33	inhibitor	NULL	DICLOXACILLIN SODIUM	rxcui:267257	DICLOXACILLIN SODIUM	TRUE	FALSE	FALSE
PBPA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DICLOXACILLIN SODIUM	rxcui:267257	DICLOXACILLIN SODIUM	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
VSSC	NULL	NULL	ChEMBL	33	blocker	NULL	PERMETHRIN	rxcui:33199	PERMETHRIN	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.041021618	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
ABCA1	hgnc:29	ABCA1	ChEMBL	33	inhibitor	0.7573221812840553	PROBUCOL	rxcui:8699	PROBUCOL	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.012573676	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMIKACIN SULFATE	rxcui:641	AMIKACIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	FLUOXETINE HYDROCHLORIDE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	0.1023541349623674	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN PHOSPHATE	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CHLORAMPHENICOL SODIUM SUCCINATE	rxcui:47998	CHLORAMPHENICOL SODIUM SUCCINATE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLINDAMYCIN HYDROCHLORIDE	rxcui:81982	CLINDAMYCIN HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.1750255707856483	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	MINOCYCLINE HYDROCHLORIDE	rxcui:6979	MINOCYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	ERYTHROMYCIN ESTOLATE	rxcui:4055	ERYTHROMYCIN ESTOLATE	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
ATPG	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
ATPD	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
ATPA	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
ATPF	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
ATPC	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
ATPB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
ATPFH	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CIPROFLOXACIN HYDROCHLORIDE	rxcui:81981	CIPROFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CIPROFLOXACIN HYDROCHLORIDE	rxcui:81981	CIPROFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NALIDIXIC ACID	rxcui:7240	NALIDIXIC ACID	TRUE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NALIDIXIC ACID	rxcui:7240	NALIDIXIC ACID	TRUE	FALSE	FALSE
ATPE	hgnc:838	ATP5F1E	ChEMBL	33	inhibitor	3.750547945	BEDAQUILINE FUMARATE	rxcui:1364503	BEDAQUILINE FUMARATE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.043866058	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.07458476	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.070860555	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.073437302	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.080905503	PRILOCAINE HYDROCHLORIDE	rxcui:2557	PRILOCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.058602312	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.021189536	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.1835932560688619	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.062139256	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.027121731	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.03140411	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
SCN2A	hgnc:10588	SCN2A	ChEMBL	33	blocker	0.151537291	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.045461187	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.1810609352954983	APREMILAST	rxcui:1492727	APREMILAST	TRUE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	DASABUVIR SODIUM	chembl:CHEMBL3544985	DASABUVIR SODIUM	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOLOZANE SULFATE	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOLOZANE SULFATE	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOLOZANE SULFATE	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOLOZANE SULFATE	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOLOZANE SULFATE	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOLOZANE SULFATE	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFTOLOZANE SULFATE	rxcui:1597608	CEFTOLOZANE SULFATE	TRUE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	ChEMBL	33	inhibitor	5.000730593875666	IMD-0354	chembl:CHEMBL3545089	IMD-0354	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.093763699	SU-014813	chembl:CHEMBL1721885	SU-014813	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	1.322135606654178	ASCIMINIB	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.1620607136904151	AS-602868	chembl:CHEMBL129857	AS-602868	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.007905401	AST-487	iuphar.ligand:5661	AST-487	FALSE	FALSE	TRUE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.4487835148349957	AT-13148	chembl:CHEMBL3544960	AT-13148	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.4861821410712453	AZD-0424	drugbank:DB13088	AZD-0424	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.030386384	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	ChEMBL	33	inhibitor	1.944728564284981	CEP-37440	drugbank:DB13060	CEP-37440	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	1.175544878411071	PF-03814735	drugbank:DB13059	PF-03814735	FALSE	FALSE	TRUE
CDK19	hgnc:19338	CDK19	ChEMBL	33	inhibitor	0.1666910197958555	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1666910197958555	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.005342661	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	inhibitor	0.9907107780319716	PL-225B	chembl:CHEMBL3545004	PL-225B	FALSE	FALSE	FALSE
MAPK11	hgnc:6873	MAPK11	ChEMBL	33	inhibitor	0.7955707762984013	RWJ-67657	chembl:CHEMBL190333	RWJ-67657	FALSE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	potentiator	0.6563458904461812	SARAKALIM	ncit:C72978	SARAKALIM	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	agonist	0.3125456621172291	CR 1447	chembl:CHEMBL3545092	CR 1447	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	ChEMBL	33	inhibitor	0.3431873936973496	BENTAMAPIMOD	ncit:C87441	BENTAMAPIMOD	FALSE	FALSE	FALSE
CDK14	hgnc:8883	CDK14	ChEMBL	33	inhibitor	0.6250913242344582	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.1389091831632129	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
CDK19	hgnc:19338	CDK19	ChEMBL	33	inhibitor	0.1666910197958555	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.090374649	ANLOTINIB	ncit:C138997	ANLOTINIB	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.089298761	ANLOTINIB	ncit:C138997	ANLOTINIB	FALSE	FALSE	FALSE
CDK17	hgnc:8750	CDK17	ChEMBL	33	inhibitor	0.4688184931758437	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK13	hgnc:1733	CDK13	ChEMBL	33	inhibitor	0.3750547945406749	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK11B	hgnc:1729	CDK11B	ChEMBL	33	inhibitor	0.1103102336884338	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.4735540335109532	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	KC-706	chembl:CHEMBL3545282	KC-706	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.1389091831632129	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
GSK3A	hgnc:4616	GSK3A	ChEMBL	33	inhibitor	0.07767407	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
ACVRL1	hgnc:175	ACVRL1	ChEMBL	33	inhibitor	17.50255707856483	ASCRINVACUMAB	ncit:C91073	ASCRINVACUMAB	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.095122593	PAMAPIMOD	ncit:C90996	PAMAPIMOD	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.055504938	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.044611445	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	ChEMBL	33	inhibitor	0.028850369	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.059532507	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	inhibitor	6.177373086552294	EPELSIBAN	ncit:C99151	EPELSIBAN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.8140724222588294	MILVETEROL	ncit:C77935	MILVETEROL	FALSE	FALSE	FALSE
PTGIR	hgnc:9602	PTGIR	ChEMBL	33	agonist	7.501095891	RALINEPAG	ncit:C152148	RALINEPAG	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	inhibitor	0.7721716358190367	ABT-288	drugbank:DB15192	ABT-288	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.2365210416022274	BATEFENTEROL	ncit:C166503	BATEFENTEROL	FALSE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	5.834185692854944	SB-649868	drugbank:DB14822	SB-649868	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	ChEMBL	33	agonist	1.166837138570988	PONESIMOD	rxcui:2532300	PONESIMOD	TRUE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.2778183663264259	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	0.3387591692625452	DASOLAMPANEL	ncit:C166510	DASOLAMPANEL	FALSE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.040515178	ETAZOLATE	ncit:C73334	ETAZOLATE	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.1860654544142257	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.233887177	ENOBOSARM	rxcui:2168587	ENOBOSARM	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	agonist	0.042073455	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.028360625	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
TLR9	hgnc:15633	TLR9	ChEMBL	33	agonist	1.544343271638073	AGATOLIMOD SODIUM	rxcui:2665621	AGATOLIMOD SODIUM	TRUE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	modulator	0.035719504	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.038894571	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
FNTB	hgnc:3785	FNTB	ChEMBL	33	inhibitor	3.500511415712966	LONAFARNIB	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
MPL	hgnc:7217	MPL	ChEMBL	33	agonist	2.045753424767318	AVATROMBOPAG	rxcui:2045726	AVATROMBOPAG	TRUE	FALSE	FALSE
SELL	hgnc:10720	SELL	ChEMBL	33	inhibitor	11.66837138570988	BIMOSIAMOSE	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
SELP	hgnc:10721	SELP	ChEMBL	33	inhibitor	8.751278539282417	RIVIPANSEL	ncit:C102786	RIVIPANSEL	FALSE	FALSE	FALSE
TNNT3	hgnc:11950	TNNT3	ChEMBL	33	activator	8.751278539282415	TIRASEMTIV	ncit:C152657	TIRASEMTIV	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	ChEMBL	33	inhibitor	0.3365876361262467	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
HDAC3	hgnc:4854	HDAC3	ChEMBL	33	inhibitor	0.3201687270469177	MOCETINOSTAT	ncit:C62521	MOCETINOSTAT	FALSE	FALSE	TRUE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.033919684	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.075768645	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.064111931	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.037398626	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
POLD1	hgnc:9175	POLD1	ChEMBL	33	inhibitor	0.364636606	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
POLE	hgnc:9177	POLE	ChEMBL	33	inhibitor	0.4375639269641208	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
PDK4	hgnc:8812	PDK4	ChEMBL	33	inhibitor	4.375639269641208	SODIUM DICHLOROACETATE	rxcui:1366930	SODIUM DICHLOROACETATE	TRUE	FALSE	FALSE
POLE3	hgnc:13546	POLE3	ChEMBL	33	inhibitor	0.729273212	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
POLE2	hgnc:9178	POLE2	ChEMBL	33	inhibitor	0.729273212	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	ChEMBL	33	inhibitor	0.5834185692854944	TREBANANIB	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
ANGPT1	hgnc:484	ANGPT1	ChEMBL	33	inhibitor	1.312691780892362	TREBANANIB	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
ITGB6	hgnc:6161	ITGB6	ChEMBL	33	inhibitor	2.187819634820604	ABITUZUMAB	ncit:C82422	ABITUZUMAB	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	1.009762908	BROLUCIZUMAB	rxcui:2204915	BROLUCIZUMAB	TRUE	FALSE	FALSE
ITGB1	hgnc:6153	ITGB1	ChEMBL	33	inhibitor	0.729273212	ABITUZUMAB	ncit:C82422	ABITUZUMAB	FALSE	FALSE	FALSE
TNFRSF9	hgnc:11924	TNFRSF9	ChEMBL	33	agonist	78.76150685354175	URELUMAB	ncit:C62449	URELUMAB	FALSE	FALSE	TRUE
CCL11	hgnc:10610	CCL11	ChEMBL	33	inhibitor	17.50255707856483	BERTILIMUMAB	ncit:C166879	BERTILIMUMAB	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.6563458904461812	CDP-860	chembl:CHEMBL2109544	CDP-860	FALSE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	ChEMBL	33	inhibitor	4.773424657790408	BENFLUOREX	rxcui:18880	BENFLUOREX	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.3182283105193605	LIXISENATIDE	rxcui:1440051	LIXISENATIDE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.1562728310586145	CYCLOFENIL	rxcui:2983	CYCLOFENIL	TRUE	FALSE	FALSE
CALCB	hgnc:1438	CALCB	ChEMBL	33	inhibitor	5.834185692854944	GALCANEZUMAB	rxcui:2058846	GALCANEZUMAB	TRUE	FALSE	FALSE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	1.250182648468916	ANISTREPLASE	rxcui:40028	ANISTREPLASE	TRUE	FALSE	FALSE
DACB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
FTSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
MRCA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
MRCB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
DACA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
MRDA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
DACC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
MMP1	hgnc:7155	MMP1	ChEMBL	33	inhibitor	0.1750255707856483	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
MMP7	hgnc:7174	MMP7	ChEMBL	33	inhibitor	1.500219178	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
IDH2	hgnc:5383	IDH2	ChEMBL	33	inhibitor	1.093909817410302	ENASIDENIB MESYLATE	rxcui:1940331	ENASIDENIB MESYLATE	TRUE	FALSE	FALSE
TPH1	hgnc:12008	TPH1	ChEMBL	33	inhibitor	3.281729452230906	TELOTRISTAT ETIPRATE	rxcui:1872448	TELOTRISTAT ETIPRATE	TRUE	FALSE	FALSE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	inhibitor	4.039051633514961	HUMIK-BETA-1	chembl:CHEMBL2109610	HUMIK-BETA-1	FALSE	FALSE	FALSE
CCR5	hgnc:1606	CCR5	ChEMBL	33	inhibitor	2.625383561784724	CCR5MAB004	chembl:CHEMBL2109341	CCR5MAB004	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	inhibitor	6.300920548	ULOCUPLUMAB	ncit:C95755	ULOCUPLUMAB	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	ChEMBL	33	inhibitor	1.458546423213736	MLN-01	chembl:CHEMBL2109496	MLN-01	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	ChEMBL	33	inhibitor	1.400204566285186	GIMSILUMAB	ncit:C172615	GIMSILUMAB	FALSE	FALSE	FALSE
TFR2	hgnc:11762	TFR2	ChEMBL	33	inhibitor	13.12691780892362	E2.3	chembl:CHEMBL2109495	E2.3	FALSE	FALSE	FALSE
C5	hgnc:1331	C5	ChEMBL	33	inhibitor	0.3889457128569963	RAVULIZUMAB	rxcui:2107301	RAVULIZUMAB	TRUE	FALSE	FALSE
RPOB	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMYCIN SODIUM	rxcui:236475	RIFAMYCIN SODIUM	TRUE	FALSE	FALSE
RPOA	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMYCIN SODIUM	rxcui:236475	RIFAMYCIN SODIUM	TRUE	FALSE	FALSE
RPOC	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMYCIN SODIUM	rxcui:236475	RIFAMYCIN SODIUM	TRUE	FALSE	FALSE
RPOZ	NULL	NULL	ChEMBL	33	inhibitor	NULL	RIFAMYCIN SODIUM	rxcui:236475	RIFAMYCIN SODIUM	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMINOSALICYLATE SODIUM	ncit:C47958	AMINOSALICYLATE SODIUM	TRUE	FALSE	FALSE
FOLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	AMINOSALICYLATE POTASSIUM	chembl:CHEMBL1200584	AMINOSALICYLATE POTASSIUM	TRUE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
TGFB3	hgnc:11769	TGFB3	ChEMBL	33	inhibitor	3.281729452230906	LUSPATERCEPT	rxcui:2262543	LUSPATERCEPT-AAMT	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	ASUNAPREVIR	rxcui:1652103	ASUNAPREVIR	FALSE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	VANIPREVIR	ncit:C152828	VANIPREVIR	FALSE	FALSE	FALSE
NS4A	NULL	NULL	ChEMBL	33	inhibitor	NULL	DANOPREVIR	ncit:C171872	DANOPREVIR	FALSE	FALSE	FALSE
HA	NULL	NULL	ChEMBL	33	negative modulator	NULL	UMIFENOVIR	ncit:C152799	UMIFENOVIR	FALSE	FALSE	FALSE
EPOR	hgnc:3416	EPOR	ChEMBL	33	agonist	0.6177373086552295	EPOETIN ZETA	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
P2RY6	hgnc:8543	P2RY6	ChEMBL	33	agonist	6.563458904461812	DIQUAFOSOL TETRASODIUM	ncit:C65437	DIQUAFOSOL TETRASODIUM	FALSE	FALSE	FALSE
P2RY4	hgnc:8542	P2RY4	ChEMBL	33	agonist	4.375639269641208	DIQUAFOSOL TETRASODIUM	ncit:C65437	DIQUAFOSOL TETRASODIUM	FALSE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	inhibitor	0.042619863	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	ChEMBL	33	blocker	0.2792961235941196	AMLODIPINE BENZOATE	rxcui:2184116	AMLODIPINE BENZOATE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	inhibitor	0.040021091	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	inhibitor	0.025439763	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	inhibitor	0.042073455	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	inhibitor	0.041540879	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
GYRB	NULL	NULL	ChEMBL	33	inhibitor	NULL	PRULIFLOXACIN	ncit:C72637	PRULIFLOXACIN	FALSE	FALSE	FALSE
GYRA	NULL	NULL	ChEMBL	33	inhibitor	NULL	PRULIFLOXACIN	ncit:C72637	PRULIFLOXACIN	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	ChEMBL	33	inhibitor	0.42006137	MONOMETHYL FUMARATE	rxcui:1546433	MONOMETHYL FUMARATE	TRUE	FALSE	FALSE
TBXAS1	hgnc:11609	TBXAS1	ChEMBL	33	inhibitor	3.281729452230906	OZAGREL	ncit:C66288	OZAGREL	FALSE	FALSE	FALSE
ENV	hgnc:39031	ERVK-20	ChEMBL	33	inhibitor	5.250767123569449	FOSTEMSAVIR	rxcui:2380373	FOSTEMSAVIR	TRUE	FALSE	FALSE
TRHR	hgnc:12299	TRHR	ChEMBL	33	agonist	4.375639269641208	TALTIRELIN	ncit:C77011	TALTIRELIN	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	ChEMBL	33	binder	0.2778183663264259	CETUXIMAB SAROTALOCAN	ncit:C190488	CETUXIMAB SAROTALOCAN	FALSE	FALSE	FALSE
SLC10A1	hgnc:10905	SLC10A1	ChEMBL	33	inhibitor	8.751278539282415	BULEVIRTIDE	ncit:C169819	BULEVIRTIDE	TRUE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	PRULIFLOXACIN	ncit:C72637	PRULIFLOXACIN	FALSE	FALSE	FALSE
PSMA3	hgnc:9532	PSMA3	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMB2	hgnc:9539	PSMB2	ChEMBL	33	inhibitor	0.1562728310586145	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMD2	hgnc:9559	PSMD2	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMB3	hgnc:9540	PSMB3	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMB5	hgnc:9542	PSMB5	ChEMBL	33	inhibitor	0.1250182648468916	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	ChEMBL	33	inhibitor	0.096167896	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMC5	hgnc:9552	PSMC5	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
HELI	NULL	NULL	ChEMBL	33	inhibitor	NULL	PRITELIVIR	ncit:C136516	PRITELIVIR	FALSE	FALSE	FALSE
PB2	NULL	NULL	ChEMBL	33	inhibitor	NULL	PIMODIVIR	ncit:C158086	PIMODIVIR	FALSE	FALSE	FALSE
RPS16	hgnc:10396	RPS16	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPS24	hgnc:10411	RPS24	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL17	hgnc:10307	RPL17	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL18A	hgnc:10311	RPL18A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL14	hgnc:10305	RPL14	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL22	hgnc:10315	RPL22	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL23A	hgnc:10317	RPL23A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL18	hgnc:10310	RPL18	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	ChEMBL	33	inhibitor	2.917092846427472	XENTUZUMAB	ncit:C106118	XENTUZUMAB	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	DELPAZOLID	ncit:C166717	DELPAZOLID	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	BEKANAMYCIN	ncit:C65248	BEKANAMYCIN	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.8751278539282416	TLC-388	chembl:CHEMBL4594352	TLC-388	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	APRICITABINE	ncit:C79871	APRICITABINE	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	GSK-364735	drugbank:DB13119	GSK-364735	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
E2F4	hgnc:3118	E2F4	ChEMBL	33	inhibitor	1.640864726115453	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
E2F3	hgnc:3115	E2F3	ChEMBL	33	inhibitor	1.640864726115453	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.4907258993990139	AMPRELOXETINE	ncit:C166483	AMPRELOXETINE	FALSE	FALSE	FALSE
NS5B	NULL	NULL	ChEMBL	33	inhibitor	NULL	BMS-986094	drugbank:DB11966	BMS-986094	FALSE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.4234489615781814	GSK-1004723	drugbank:DB12806	GSK-1004723	FALSE	FALSE	FALSE
P	hgnc:8101	OCA2	ChEMBL	33	inhibitor	2.386712328895204	ELVUCITABINE	ncit:C73201	ELVUCITABINE	FALSE	FALSE	FALSE
EZH2	hgnc:3527	EZH2	ChEMBL	33	inhibitor	2.333674277141978	GSK2816126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
PARE	NULL	NULL	ChEMBL	33	inhibitor	NULL	CIPROFLOXACIN HYDROCHLORIDE	rxcui:81981	CIPROFLOXACIN HYDROCHLORIDE	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	1.250182648468916	NILOTINIB HYDROCHLORIDE MONOHYDRATE	ncit:C95229	NILOTINIB HYDROCHLORIDE MONOHYDRATE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
APCS	hgnc:584	APCS	ChEMBL	33	modulator	13.12691780892362	MIRIDESAP	ncit:C153209	MIRIDESAP	FALSE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	ChEMBL	33	inhibitor	4.773424657790408	NEVANIMIBE	ncit:C170216	NEVANIMIBE	FALSE	FALSE	FALSE
CA3	hgnc:1374	CA3	ChEMBL	33	inhibitor	1.093909817410302	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	agonist	0.030368809	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	agonist	0.034981793	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
F	NULL	NULL	ChEMBL	33	inhibitor	NULL	NIRSEVIMAB	rxcui:2642401	NIRSEVIMAB	TRUE	FALSE	FALSE
IMPDH2	hgnc:6053	IMPDH2	ChEMBL	33	inhibitor	1.312691780892362	MIZORIBINE	ncit:C66172	MIZORIBINE	FALSE	FALSE	FALSE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	1.750255707856483	MIZORIBINE	ncit:C66172	MIZORIBINE	FALSE	FALSE	FALSE
POLR1A	hgnc:17264	POLR1A	ChEMBL	33	inhibitor	17.50255707856483	TAS-106	drugbank:DB06656	TAS-106	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	ChEMBL	33	inhibitor	0.2500365296937833	AMIVANTAMAB	rxcui:2549198	AMIVANTAMAB-VMJW	TRUE	FALSE	TRUE
CD3D	hgnc:1673	CD3D	ChEMBL	33	binder	0.4102161815288632	TALQUETAMAB	rxcui:2644447	TALQUETAMAB	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.1312691780892362	TIVOZANIB HYDROCHLORIDE	rxcui:2534245	TIVOZANIB HYDROCHLORIDE	TRUE	FALSE	FALSE
ATP1A4	hgnc:14073	ATP1A4	ChEMBL	33	inhibitor	0.1750255707856483	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
FXYD2	hgnc:4026	FXYD2	ChEMBL	33	inhibitor	0.2917092846427472	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
ATP1B1	hgnc:804	ATP1B1	ChEMBL	33	inhibitor	0.1842374429322614	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.1666910197958555	MOSAPRIDE	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
GCK	hgnc:4195	GCK	ChEMBL	33	activator	3.500511415712966	MK-0941	chembl:CHEMBL3580737	MK-0941	FALSE	FALSE	FALSE
ATP1B3	hgnc:806	ATP1B3	ChEMBL	33	inhibitor	0.5834185692854944	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
FUSA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FUSIDIC ACID	rxcui:113608	FUSIDATE	TRUE	FALSE	FALSE
FUSA	NULL	NULL	ChEMBL	33	inhibitor	NULL	FUSIDATE SODIUM	rxcui:9874	FUSIDATE SODIUM	TRUE	FALSE	FALSE
HDAC6	hgnc:14064	HDAC6	ChEMBL	33	inhibitor	0.055504938	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLR	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLS	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLT	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLU	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLV	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLW	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLX	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLY	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMA	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLB	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMD	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	NAFITHROMYCIN	ncit:C166991	NAFITHROMYCIN	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	IMDEVIMAB	rxcui:2465249	IMDEVIMAB	TRUE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	ADINTREVIMAB	ncit:C182620	ADINTREVIMAB	FALSE	FALSE	FALSE
S	NULL	NULL	ChEMBL	33	inhibitor	NULL	ROMLUSEVIMAB	ncit:C175226	ROMLUSEVIMAB	FALSE	FALSE	FALSE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	1.640864726115453	PF-03049423	chembl:CHEMBL591501	PF-03049423	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
SSTR4	hgnc:11333	SSTR4	ChEMBL	33	agonist	1.750255707856483	SOMATOSTATIN	rxcui:9939	SOMATOSTATIN	FALSE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.4667348554283956	REVAMILAST	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
SSTR3	hgnc:11332	SSTR3	ChEMBL	33	agonist	3.500511415712966	SOMATOSTATIN	rxcui:9939	SOMATOSTATIN	FALSE	FALSE	FALSE
YKGM	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPME	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPMF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPMG	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPMH	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPMI	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
YKGO	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLC	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLE	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLF	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
RPLL	NULL	NULL	ChEMBL	33	inhibitor	NULL	LINCOMYCIN	rxcui:6398	LINCOMYCIN	TRUE	FALSE	FALSE
FGG	hgnc:3694	FGG	ChEMBL	33	cleavage	1.640864726115453	ANCROD	rxcui:772	ANCROD	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	0.1591141552596802	SERALUTINIB	ncit:C175203	SERALUTINIB	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	ChEMBL	33	agonist	1.875273972703375	SETOGEPRAM	drugbank:DB15447	SETOGEPRAM	FALSE	FALSE	FALSE
FGB	hgnc:3662	FGB	ChEMBL	33	cleavage	1.166837138570988	PLASMINOGEN	rxcui:2557200	PLASMINOGEN	TRUE	FALSE	FALSE
FGA	hgnc:3661	FGA	ChEMBL	33	cleavage	1.193356164447602	ANCROD	rxcui:772	ANCROD	FALSE	FALSE	FALSE
RPSB	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLD	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSK	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSL	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSM	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSN	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSO	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSP	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSR	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSS	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPST	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSU	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSC	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSD	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSE	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSF	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSG	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSH	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPSI	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLJ	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLK	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLM	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLN	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLO	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLP	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
RPLQ	NULL	NULL	ChEMBL	33	inhibitor	NULL	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	ChEMBL	33	inhibitor	0.6177373086552294	DANBURSTOTUG	ncit:C172819	DANBURSTOTUG	FALSE	FALSE	FALSE
SIRT1	hgnc:14929	SIRT1	ChEMBL	33	inhibitor	1.810609352954982	EX-527	chembl:CHEMBL382277	EX-527	FALSE	FALSE	FALSE
HBCAG	NULL	NULL	ChEMBL	33	modulator	NULL	BERSACAPAVIR	ncit:C175058	BERSACAPAVIR	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.2083637747448194	ENSIFENTRINE	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
PDE3A	hgnc:8778	PDE3A	ChEMBL	33	inhibitor	0.7955707762984013	ENSIFENTRINE	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.297662535	CID 5330286	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
BIRC2	hgnc:590	BIRC2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.312691780892362	BIRINAPANT	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
APH1B	hgnc:24080	APH1B	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.8078103267029924	MK-0752	drugbank:DB12852	MK-0752	FALSE	FALSE	TRUE
ANGPT1	hgnc:484	ANGPT1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	1.312691780892362	TREBANINIB	ncit:C91711	TREBANANIB	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.024756092	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NFKB1	hgnc:7794	NFKB1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.006426888	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.063331621	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	COSMIC	4-Sep-20	NULL	0.1481697953740938	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	COSMIC	4-Sep-20	NULL	1.040600372117402	Quizartinib	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	GRAMINE	ncit:C64181	GRAMINE	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	DTC	9/2/20	NULL	0.482607272	DONEPEZIL	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-46080	chembl:CHEMBL1331754	CHEMBL:CHEMBL1331754	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00149902	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.347732922	GNF-PF-4829	chembl:CHEMBL526034	CHEMBL:CHEMBL526034	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.005409816	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	0.8751278539282418	[3H]-PHORBOL 12,13-DIBUTYRATE	chembl:CHEMBL27768	CHEMBL:CHEMBL27768	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.020470827	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.072424374	CLEMIZOLE	ncit:C81139	CLEMIZOLE	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.082043236	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	NSC-74859	chembl:CHEMBL477936	CHEMBL:CHEMBL477936	FALSE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.1274458039701322	GNF-PF-186	chembl:CHEMBL601140	CHEMBL:CHEMBL601140	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.003622218	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.009796207	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	ESREBOXETINE	rxcui:60842	REBOXETINE	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.3070624048871023	CHAULMOOGRIC ACID, ETHYL ESTER	chembl:CHEMBL1329881	CHAULMOOGRIC ACID, ETHYL ESTER	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005953251	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
BRD3	hgnc:1104	BRD3	DTC	9/2/20	NULL	0.1446492320542548	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.4134462302023188	TRIMETHIDINIUM	chembl:CHEMBL1708232	TRIMETHIDINIUM	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.058602312	FLAVANONE	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.2224901323546377	NORHARMANE	iuphar.ligand:8222	BETA-CARBOLINE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.045579576	ENOXIMONE	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.016181101	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	SJ000069305	chembl:CHEMBL603739	CHEMBL:CHEMBL603739	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.016181101	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.012087401	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	TCMDC-123770	chembl:CHEMBL533529	CHEMBL:CHEMBL533529	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.026766867	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	5.000730593875666	R-RUGULACTONE	chembl:CHEMBL1253688	R-RUGULACTONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006193403	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.008857569	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.075010959	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.037721028	GW3965	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.048618214	ENDO-ATROPINE	chembl:CHEMBL2449003	ENDO-ATROPINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010058941	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.043466615	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	chembl:CHEMBL1322879	2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.1033615575505797	GARCINOLIC ACID	chembl:CHEMBL1456870	GARCINOLIC ACID	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01495945	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.036212187	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.025955349	NSC-402083	chembl:CHEMBL1546228	CHEMBL:CHEMBL1546228	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001526652	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TOMATINE	chembl:CHEMBL525778	TOMATINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005873341	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	RESOKAEMPFEROL	chembl:CHEMBL242383	RESOKAEMPFEROL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	SJ000147784	chembl:CHEMBL590186	CHEMBL:CHEMBL590186	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.003890322	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	SOPHORIDINE	chembl:CHEMBL1824581	SOPHORIDINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	ARISTOLOCHIC ACID	iuphar.ligand:12438	ARISTOLOCHIC ACID	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.086818239	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	DIGOXIGENIN	drugbank:DB03671	DIGOXIGENIN	FALSE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	DTC	9/2/20	NULL	0.151537291	WIN-552122	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.003217382	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	inhibitor	0.064413418	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	DTC	9/2/20	NULL	0.2991890098899971	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.023620185	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.007749066	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	NSC-135810	chembl:CHEMBL1605629	CHEMBL:CHEMBL1605629	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.015806042	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2243917574174979	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	TECHTOCHRYSIN	chembl:CHEMBL164841	TECHTOCHRYSIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	MINOCYCLINE	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	TUBERCIDIN	ncit:C911	TUBERCIDIN	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GSK-319347A	chembl:CHEMBL373751	GSK-319347A	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.063645662	TCMDC-125142	chembl:CHEMBL528791	CHEMBL:CHEMBL528791	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.2224901323546377	CEPHALOSPORIN C ZINC SALT	chembl:CHEMBL1326149	CEPHALOSPORIN C ZINC SALT	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.01305187	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	U-73122	iuphar.ligand:5283	U73122	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.017357908	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2907401508067248	NADOLOL	rxcui:7226	NADOLOL	TRUE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	GANODERIOL F	chembl:CHEMBL1915761	GANODERIOL F	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.2625383561784725	DNDI1417006	chembl:CHEMBL1415258	CHEMBL:CHEMBL1415258	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	TINORIDINE	ncit:C76821	TINORIDINE	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.014249029	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL201761	SALINAZID	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.019724895	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	MMV667491	chembl:CHEMBL1437888	CHEMBL:CHEMBL1437888	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.008382451	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	DSM-106	chembl:CHEMBL444928	CHEMBL:CHEMBL444928	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.021697385	RACLOPRIDE	ncit:C152139	RACLOPRIDE	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.040640612	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1117184494376478	LONIDAMINE	ncit:C1146	LONIDAMINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.09745299	NANDROLONE DECANOATE	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.036162308	BRL-52537	chembl:CHEMBL1256835	CHEMBL:CHEMBL1256835	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002623285	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.05853698	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	DEVAZEPIDE	ncit:C98235	DEVAZEPIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	METHANANDAMIDE	iuphar.ligand:2506	R-(+)-METHANANDAMIDE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	LEAD DIACETATE TRIHYDRATE	chembl:CHEMBL1350036	LEAD DIACETATE TRIHYDRATE	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.091317689	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.2917092846427472	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
CFLAR	hgnc:1876	CFLAR	DTC	9/2/20	NULL	1.093909817410302	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	RUFLOXACIN	ncit:C72638	RUFLOXACIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003405608	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.077444943	METHYLBENZETHONIUM CHLORIDE	rxcui:1796444	METHYLBENZETHONIUM CHLORIDE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.018619742	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1981421556063943	NSC-645827	chembl:CHEMBL95704	CHEMBL:CHEMBL95704	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007866318	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	PHOSMET	drugbank:DB11448	PHOSMET	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	CID 2056784	chembl:CHEMBL261123	CHEMBL:CHEMBL261123	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.02617531	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.008621949	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.030386384	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	SJ000120515	chembl:CHEMBL592314	CHEMBL:CHEMBL592314	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.004011894	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	DTC	9/2/20	NULL	0.2792961235941196	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.002236844	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	SJ000150791	chembl:CHEMBL600572	CHEMBL:CHEMBL600572	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005534114	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.019534104	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.1598407039138341	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.072826174	SOFALCONE	ncit:C81118	SOFALCONE	FALSE	FALSE	FALSE
GAK	hgnc:4113	GAK	DTC	9/2/20	inhibitor	10.50153425	HTS-466284	drugbank:DB03921	4-(3-PYRIDIN-2-YL-1H-PYRAZOL-4-YL)QUINOLINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.06697407	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.028977744	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.062509132	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.09869863	N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE	chembl:CHEMBL201761	SALINAZID	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	DNDI1417420	chembl:CHEMBL1546223	CHEMBL:CHEMBL1546223	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	MEPIVACAINE	rxcui:203185	MEPIVACAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.009192519	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
SIRT1	hgnc:14929	SIRT1	DTC	9/2/20	NULL	0.2785552850699974	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	CINALUKAST	ncit:C96709	CINALUKAST	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	LINURON	chembl:CHEMBL448213	LINURON	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005953251	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
FYN	hgnc:4037	FYN	DTC	9/2/20	NULL	0.012360563	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.009853194	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	MINOCYCLINE	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.021697385	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	NSC-209931	chembl:CHEMBL472656	CHEMBL:CHEMBL472656	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.013022736	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.015263858	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
SLC22A7	hgnc:10971	SLC22A7	DTC	9/2/20	NULL	4.375639269641208	GS-9256	drugbank:DB12876	GS-9256	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	DESIPRAMINE HYDROCHLORIDE	rxcui:203174	DESIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	S-166659	chembl:CHEMBL252417	CHEMBL:CHEMBL252417	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	S(+)-RACLOPRIDE L-TARTRATE	chembl:CHEMBL1369632	CHEMBL:CHEMBL1369632	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.3409589041278863	DINACICLIB	ncit:C78854	DINACICLIB	FALSE	FALSE	TRUE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.043902735	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.069824031	NSC-628113	chembl:CHEMBL176599	CHEMBL:CHEMBL176599	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.043866058	AM-404	iuphar.ligand:12556	AM404	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003262967	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
PRKG1	hgnc:9414	PRKG1	DTC	9/2/20	NULL	0.059667808	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.002778184	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	2-METHOXYESTRADIOL	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006557721	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.0135995	OXYBUTYNIN CHLORIDE	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
EP300	hgnc:3373	EP300	DTC	9/2/20	NULL	4.375639269641208	GARCINOL	iuphar.ligand:7001	GARCINOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.039331589	CEFDITORIN PIVOXIL	chembl:CHEMBL1514735	CEFDITORIN PIVOXIL	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.6563458904461812	EVODIAMINE	rxcui:2199291	EVODIAMINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.028739831	DAPHNORIN	chembl:CHEMBL1209491	DAPHNORIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	FLUNARIZINE	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	GNF-PF-1878	chembl:CHEMBL1500740	CHEMBL:CHEMBL1500740	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.048935388	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005835482	FLUPHENAZINE HYDROCHLORIDE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	GNF-PF-1477	chembl:CHEMBL582675	CHEMBL:CHEMBL582675	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.012588749	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.012838061	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.1779921058837101	8-PHENOXYCAFFEINE	chembl:CHEMBL1529697	CHEMBL:CHEMBL1529697	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.022249013	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.009767052	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	PD-160170	chembl:CHEMBL422942	CHEMBL:CHEMBL422942	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.006250913	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.1875273972703375	TDR77578	chembl:CHEMBL1364172	CHEMBL:CHEMBL1364172	FALSE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	DTC	9/2/20	NULL	1.060761035064535	BETA-NAPHTHOFLAVONE	ncit:C29812	BETA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.5357925636295356	WR-243246	chembl:CHEMBL117217	CHEMBL:CHEMBL117217	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.5834185692854944	N-(3-METHOXYPHENYL)ANTHRANILIC ACID	chembl:CHEMBL1328677	CHEMBL:CHEMBL1328677	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1750255707856483	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.01535312	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
GPR12	hgnc:4466	GPR12	DTC	9/2/20	NULL	15.00219178	24-EPI-CYCLOCITRINOL	chembl:CHEMBL496266	CHEMBL:CHEMBL496266	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.029106248	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.022108493	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	MENTHOFURAN	chembl:CHEMBL1522900	MENTHOFURAN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002397282	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	DIPHENHYDRAMINE	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	MAKALUVAMINE C TFA SALT	chembl:CHEMBL450970	MAKALUVAMINE C TFA SALT	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.010777437	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.003720782	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.026519026	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006909813	MIBEFRADIL	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	DTC	9/2/20	NULL	0.010128795	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.037884323	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	2-PYRIDYLKETONE BENZOYL HYDRAZONE	chembl:CHEMBL252151	CHEMBL:CHEMBL252151	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.292250489	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.1108075556053025	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.2500365296937833	GNF-PF-2936	chembl:CHEMBL582503	CHEMBL:CHEMBL582503	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01514062	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.038636991	ARTEMISIN	rxcui:2367409	ARTEMISININ	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.010629083	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.043611023	DAPHNORIN	chembl:CHEMBL1209491	DAPHNORIN	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.033148782	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.079557078	AMORFRUTIN A	chembl:CHEMBL491820	AMORFRUTIN A	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.035287413	DNDI1417221	chembl:CHEMBL1459280	CHEMBL:CHEMBL1459280	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	5'-FORMYLGLABRIDIN	chembl:CHEMBL599165	CHEMBL:CHEMBL599165	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	2-BROMO-HEXADECANOIC ACID	chembl:CHEMBL118417	CHEMBL:CHEMBL118417	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.011906501	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	1,5-ISOQUINOLINEDIOL	chembl:CHEMBL338314	CHEMBL:CHEMBL338314	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003844181	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.2381300282797936	4,6-BIS(4-MORPHOLINOSTYRYL)PYRIMIDINE	chembl:CHEMBL2181046	CHEMBL:CHEMBL2181046	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001049314	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.009539911	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004842988	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	FIPEXIDE	ncit:C65685	FIPEXIDE	TRUE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.1544343271638073	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	U-37883A	iuphar.ligand:13269	PNU-37883	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	METHYL ALCOHOL	chembl:CHEMBL14688	METHYL ALCOHOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	HTS-05056	chembl:CHEMBL196814	CHEMBL:CHEMBL196814	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.031842129	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.027433475	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.025489161	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.052824619	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	4-BENZYLOXYANILINE	chembl:CHEMBL1351571	4-BENZYLOXYANILINE	FALSE	FALSE	FALSE
NCOA2	hgnc:7669	NCOA2	DTC	9/2/20	NULL	2.187819634820604	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	8-(3-CHLOROBENZYLOXY)CAFFEINE	chembl:CHEMBL602260	CHEMBL:CHEMBL602260	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	NONIVAMIDE	rxcui:31945	NONIVAMIDE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	GARCINOLIC ACID	chembl:CHEMBL1456870	GARCINOLIC ACID	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.029317516	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	DNDI1417221	chembl:CHEMBL1459280	CHEMBL:CHEMBL1459280	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.006100578	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.012154554	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.052455216	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.034251579	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
GALR3	hgnc:4134	GALR3	DTC	9/2/20	NULL	1.750255707856483	CHLORMIDAZOLE	ncit:C78032	CHLORMIDAZOLE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.004172574	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.057955487	TCMDC-123868	chembl:CHEMBL548615	CHEMBL:CHEMBL548615	FALSE	FALSE	FALSE
PTPN11	hgnc:9644	PTPN11	DTC	9/2/20	NULL	7.501095891	4-HYDRAZINYLBENZENESULFONIC ACID	chembl:CHEMBL510966	CHEMBL:CHEMBL510966	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	DANTHRON	rxcui:22293	DANTHRON	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	MEZLOCILLIN	rxcui:6927	MEZLOCILLIN	FALSE	FALSE	FALSE
MARK4	hgnc:13538	MARK4	DTC	9/2/20	NULL	0.081030357	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
BLK	hgnc:1057	BLK	DTC	9/2/20	NULL	0.018385039	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.5000730593875666	TCMDC-124353	chembl:CHEMBL529918	CHEMBL:CHEMBL529918	FALSE	FALSE	FALSE
ESRRA	hgnc:3471	ESRRA	DTC	9/2/20	NULL	0.729273212	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PARAMETHASONE ACETATE	rxcui:32895	PARAMETHASONE ACETATE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003405608	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-601364	chembl:CHEMBL1270061	CHEMBL:CHEMBL1270061	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.047432404	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.097236428	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.006521882	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.028977744	MUNDULONE	chembl:CHEMBL465339	MUNDULONE	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.2287915957982331	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	EMETINE	rxcui:3820	EMETINE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.045579576	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.051277023	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
HKDC1	hgnc:23302	HKDC1	DTC	9/2/20	NULL	2.019525817	SJ000032153	chembl:CHEMBL600862	CHEMBL:CHEMBL600862	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	REV-5901	chembl:CHEMBL8747	REV-5901	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.42006137	TECNAZENE	chembl:CHEMBL1420059	TECNAZENE	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.035098711	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	(-)-ROLIPRAM	chembl:CHEMBL430893	(-)-ROLIPRAM	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665980	chembl:CHEMBL601325	CHEMBL:CHEMBL601325	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.04321619	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.01651704	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.060562481	PROTOCATECHUALDEHYDE	rxcui:1362689	PROTOCATECHUALDEHYDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	METHYL ABIETATE	rxcui:2465733	METHYL ABIETATE	FALSE	FALSE	FALSE
PIM2	hgnc:8987	PIM2	DTC	9/2/20	NULL	0.1600843635234588	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.039214094	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	GUAIFENESIN	rxcui:5032	GUAIFENESIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002016269	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.022622866	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	APRINDINE HYDROCHLORIDE	rxcui:236158	APRINDINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	CLEBOPRIDE MALEATE	rxcui:236701	CLEBOPRIDE MALEATE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	DNDI1416934	chembl:CHEMBL1989750	CHEMBL:CHEMBL1989750	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	WIN-552122	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	(R,S)-AMPA	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.009673484	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.029009763	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.01037701	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
PIN1	hgnc:8988	PIN1	DTC	9/2/20	NULL	0.2169738480813822	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.033615667	CGS-15943	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.032817295	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	SJ000133784	chembl:CHEMBL589670	CHEMBL:CHEMBL589670	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.01823183	AZELNIDIPINE	ncit:C73023	AZELNIDIPINE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	ECADOTRIL	ncit:C75238	ECADOTRIL	FALSE	FALSE	FALSE
APOBEC3F	hgnc:17356	APOBEC3F	DTC	9/2/20	NULL	0.4861821410712453	GNF-PF-1477	chembl:CHEMBL582675	CHEMBL:CHEMBL582675	FALSE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	0.2430910705356226	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	PF-228	chembl:CHEMBL514554	CHEMBL:CHEMBL514554	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.031803556	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	FLUPHENAZINE DIHYDROCHLORIDE	chembl:CHEMBL1448187	FLUPHENAZINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	TCMDC-124356	chembl:CHEMBL22062	CHEMBL:CHEMBL22062	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	DTC	9/2/20	NULL	0.016605842	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.012977675	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.025739055	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
RPS6KA1	hgnc:10430	RPS6KA1	DTC	9/2/20	NULL	0.9723642821424908	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.024174803	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
ALPPL2	hgnc:441	ALPG	DTC	9/2/20	NULL	0.1286952726365061	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	DTC	9/2/20	NULL	0.6482428547616604	HINOKININ	chembl:CHEMBL242011	HINOKININ	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.009603891	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	DTC	9/2/20	NULL	1.721562991334245	(R)-VERAPAMIL	ncit:C1563	DEXVERAPAMIL	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1750255707856483	CHLORFENAPYR	chembl:CHEMBL1869551	CHLORFENAPYR	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1041818873724097	GEDUNIN	chembl:CHEMBL465226	GEDUNIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.029918901	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	HYDROCORTISONE HEMISUCCINATE	ncit:C61786	HYDROCORTISONE HEMISUCCINATE	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	DTC	9/2/20	NULL	1.944728564284981	GNF-PF-2262	chembl:CHEMBL577862	CHEMBL:CHEMBL577862	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	0.6250913242344582	GW3965	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	DTC	9/2/20	NULL	0.1495945049449985	MIANSERIN	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
MC4R	hgnc:6932	MC4R	DTC	9/2/20	NULL	0.021933029	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.027276712	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	NITROFEN	chembl:CHEMBL561004	NITROFEN	FALSE	FALSE	FALSE
SLC2A3	hgnc:11007	SLC2A3	DTC	9/2/20	NULL	0.4286340509036285	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.009290105	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	ENOXIMONE	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011049594	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.2734774543525755	OPIPRAMOL	rxcui:7674	OPIPRAMOL	FALSE	FALSE	FALSE
IDE	hgnc:5381	IDE	DTC	9/2/20	NULL	0.5834185692854945	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
SIK2	hgnc:21680	SIK2	DTC	9/2/20	NULL	0.1060761035064535	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
PRKCZ	hgnc:9412	PRKCZ	DTC	9/2/20	NULL	0.037081689	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.035358701	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	1.381780822	TCMDC-125385	chembl:CHEMBL586628	CHEMBL:CHEMBL586628	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.2333674277141978	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.017363648	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	U-50488 METHANE SULFONATE	iuphar.ligand:1652	U50488	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.084146909	GW806742X	iuphar.ligand:9513	MLKL COMPOUND 1	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.009430257	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.027524552	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.043756393	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009875432	A-443654	drugbank:DB08073	(2S)-1-(1H-INDOL-3-YL)-3-{[5-(3-METHYL-1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}PROPAN-2-AMINE	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	RIMCAZOLE	ncit:C152218	RIMCAZOLE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	DNDI1417024	chembl:CHEMBL1462710	CHEMBL:CHEMBL1462710	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	GLABRANIN	chembl:CHEMBL253998	GLABRANIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.025298806	METARAMINOL	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	TCMDC-125142	chembl:CHEMBL528791	CHEMBL:CHEMBL528791	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.030796288	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009832897	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.3889457128569962	HISPIDULIN	drugbank:DB14008	HISPIDULIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	HYDRAMETHYLNON	chembl:CHEMBL464812	HYDRAMETHYLNON	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.033529803	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	5-DEMETHYLNOBILETIN	chembl:CHEMBL75978	5-DEMETHYLNOBILETIN	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.014634245	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	ORSELLINIC ACID, ETHYL ESTER	chembl:CHEMBL1601166	ORSELLINIC ACID, ETHYL ESTER	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	OSAJIN	chembl:CHEMBL238188	OSAJIN	FALSE	FALSE	FALSE
CDK5R1	hgnc:1775	CDK5R1	DTC	9/2/20	NULL	1.875273972703375	HTS-05058	chembl:CHEMBL261692	CHEMBL:CHEMBL261692	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	BIPHENYL	chembl:CHEMBL1231413	BIPHENYL	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.112919723	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.006286838	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
P2RY2	hgnc:8541	P2RY2	DTC	9/2/20	NULL	1.050153425	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.022969235	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-4276	chembl:CHEMBL605753	CHEMBL:CHEMBL605753	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	THIOTHIXENE HYDROCHLORIDE	rxcui:91135	THIOTHIXENE HYDROCHLORIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.016992774	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	TRIBUTYLTIN-OXIDE	chembl:CHEMBL511667	TRIBUTYLTIN-OXIDE	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.4234489615781814	SJ000032154	chembl:CHEMBL591876	CHEMBL:CHEMBL591876	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.3804903712731485	RHODOMYRTOXIN B	chembl:CHEMBL1552997	RHODOMYRTOXIN B	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	AMBUNOL	chembl:CHEMBL454893	AMBUNOL	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.056826484	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1215455352678113	2-HYDROXYESTRADIOL	ncit:C120474	2-HYDROXYESTRADIOL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	CIS-2,4,3',5'-TETRAMETHOXYSTILBENE	chembl:CHEMBL221300	CHEMBL:CHEMBL221300	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.076765601	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	METHYLPREDNISOLONE SODIUM SUCCINATE	rxcui:203189	METHYLPREDNISOLONE SODIUM SUCCINATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	BENZO[E]PYRENE	chembl:CHEMBL1371125	BENZO[E]PYRENE	FALSE	FALSE	FALSE
RPS6KA5	hgnc:10434	RPS6KA5	DTC	9/2/20	NULL	0.093763699	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002669701	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.042741287	CISAPRIDE	rxcui:35255	CISAPRIDE	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	1.141471113819445	(-)-CAMPHOR	chembl:CHEMBL2252949	(-)-CAMPHOR	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	FAGARONINE	chembl:CHEMBL282622	FAGARONINE	FALSE	FALSE	FALSE
FOXO3	hgnc:3821	FOXO3	DTC	9/2/20	NULL	1.071585127259071	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.1100789753368857	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.157680694	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.005787883	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
FES	hgnc:3657	FES	DTC	9/2/20	NULL	0.1640864726115453	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.021652648	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-4522	chembl:CHEMBL585417	CHEMBL:CHEMBL585417	FALSE	FALSE	FALSE
GLI1	hgnc:4317	GLI1	DTC	9/2/20	NULL	0.4861821410712453	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
NR0B1	hgnc:7960	NR0B1	DTC	9/2/20	NULL	0.2187819634820604	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	CARMUSTINE	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.086789539	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.9053046764774912	TCMDC-123747	chembl:CHEMBL530698	CHEMBL:CHEMBL530698	FALSE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.02926849	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.3500511415712966	METHYLBENZETHONIUM CHLORIDE	rxcui:1796444	METHYLBENZETHONIUM CHLORIDE	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.027177884	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	CEPHALOTHIN SODIUM	rxcui:9860	CEPHALOTHIN SODIUM	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.069824031	GNF-PF-4992	chembl:CHEMBL275177	CHEMBL:CHEMBL275177	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.033148782	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	CHLORFENAPYR	chembl:CHEMBL1869551	CHLORFENAPYR	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	MMV396678	chembl:CHEMBL1459149	CHEMBL:CHEMBL1459149	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.005562253	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	0.03297185	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.150021918	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.013299815	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.01816246	DIHYDREXIDINE	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	4'-HYDROXY-FLAVANONE	chembl:CHEMBL73933	4'-HYDROXY-FLAVANONE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.069089041	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.2800409132570373	ISOSILYBIN A	chembl:CHEMBL592676	ISOSILYBIN A	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.022201975	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	RELCOVAPTAN	ncit:C1497	RELCOVAPTAN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.026572708	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.069824031	ATOMOXETINE	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	FPL-55712	chembl:CHEMBL267475	FPL-55712	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.029833904	FENOLDOPAM MESYLATE	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006381584	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.009171646	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00194906	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	4'-HYDROXYCHALCONE	chembl:CHEMBL276473	4'-HYDROXYCHALCONE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.3684748858645227	TAMARIXETIN	chembl:CHEMBL226034	TAMARIXETIN	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	1.750255707856483	DEMETHYLWEDELOLACTONE	chembl:CHEMBL2089002	DEMETHYLWEDELOLACTONE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	FAMOTIDINE	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.078136416	FAGARONINE	chembl:CHEMBL282622	FAGARONINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	NSC-747270	chembl:CHEMBL594772	CHEMBL:CHEMBL594772	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.050007306	PH-011685	chembl:CHEMBL126804	CHEMBL:CHEMBL126804	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	4.039051633514961	DEOXY CHOLATE	chembl:CHEMBL412272	TAURODEOXYCHOLIC ACID	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.01535312	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	DIPHENHYDRAMINE	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	GARCINOLIC ACID	chembl:CHEMBL1456870	GARCINOLIC ACID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	GF-109203	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	IMAZODAN	ncit:C83787	IMAZODAN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.014264513	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005787883	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.005867434	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.1875273972703374	SB-242235	chembl:CHEMBL95692	SB-242235	FALSE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.2917092846427472	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	GF-109203	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	BERBAMINE	ncit:C162341	BERBAMINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002936671	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.7721716358190367	GLAUCINE METHIODIDE	chembl:CHEMBL225852	GLAUCINE METHIODIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003454907	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.074797252	S(+)-RACLOPRIDE L-TARTRATE	chembl:CHEMBL1369632	CHEMBL:CHEMBL1369632	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.05010274	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	DEXBUDESONIDE	ncit:C80814	DEXBUDESONIDE	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.1715936968486748	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.0191914	2-AMINOETHOXYDIPHENYL BORATE	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.03292017	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.1035654265003836	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	NAPHTHALEN-1-YLAMINE	chembl:CHEMBL57394	CHEMBL:CHEMBL57394	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	4-HYDROXYFLAVONOL	chembl:CHEMBL272682	CHEMBL:CHEMBL272682	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	IOPANOIC ACID	rxcui:5967	IOPANOIC ACID	FALSE	FALSE	FALSE
MELK	hgnc:16870	MELK	DTC	9/2/20	NULL	0.024309107	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	TCMDC-124585	chembl:CHEMBL587856	CHEMBL:CHEMBL587856	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.4773424657790409	NODAKENIN	chembl:CHEMBL459825	NODAKENIN	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	RESOKAEMPFEROL	chembl:CHEMBL242383	RESOKAEMPFEROL	FALSE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.1363835616511545	GS 6201	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.017009288	NSC-402083	chembl:CHEMBL1546228	CHEMBL:CHEMBL1546228	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.027347745	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GARDENIN B	chembl:CHEMBL226512	GARDENIN B	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	BUFEXAMAC	rxcui:1796	BUFEXAMAC	TRUE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.045461187	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	TRIACETYLRESVERATROL	chembl:CHEMBL597744	TRIACETYLRESVERATROL	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.019447286	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.013588942	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	EPITIOSTANOL	ncit:C1089	EPITIOSTANOL	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	0.4434769530041765	SAFINAMIDE	rxcui:1922448	SAFINAMIDE	TRUE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.024479101	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.016856395	ZUCAPSAICIN	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	1.346350544504987	8-(3-CHLOROBENZYLOXY)CAFFEINE	chembl:CHEMBL602260	CHEMBL:CHEMBL602260	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.007416338	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	AMINOCARB	ncit:C163585	AMINOCARB	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.082043236	DNDI1416988	chembl:CHEMBL1389794	CHEMBL:CHEMBL1389794	FALSE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	5.000730593875666	RICCARDI C	chembl:CHEMBL411317	RICCARDI C	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.015921065	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	CITICOLINE SODIUM	rxcui:1099914	CITICOLINE SODIUM	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.017608206	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	GNF-PF-3446	chembl:CHEMBL582486	CHEMBL:CHEMBL582486	FALSE	FALSE	FALSE
CHEK2	hgnc:16627	CHEK2	DTC	9/2/20	NULL	0.014299475	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.078136416	JNJ-1661010	iuphar.ligand:5206	JNJ1661010	FALSE	FALSE	FALSE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.087512785	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	CALCIPOTRIENE	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
RNASEL	hgnc:10050	RNASEL	DTC	9/2/20	NULL	52.50767123569449	C-5950331	chembl:CHEMBL259633	CHEMBL:CHEMBL259633	FALSE	FALSE	FALSE
CA1	hgnc:1368	CA1	DTC	9/2/20	NULL	1.312691780892362	MEDRONIC ACID	rxcui:1314368	MEDRONIC ACID	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.058602312	DNDI1417195	chembl:CHEMBL1303948	CHEMBL:CHEMBL1303948	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004972317	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	BERGAPTEN	rxcui:15842	5-METHOXYPSORALEN	FALSE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.016916131	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.036162308	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.030246354	SOFALCONE	ncit:C81118	SOFALCONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.025390557	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.007946076	FLUPIRTINE	rxcui:25193	FLUPIRTINE	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	GNF-PF-3756	chembl:CHEMBL597035	CHEMBL:CHEMBL597035	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.011786234	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.028598949	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	TCMDC-125821	chembl:CHEMBL547977	CHEMBL:CHEMBL547977	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00224853	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	PD-123319	iuphar.ligand:597	PD123319	FALSE	FALSE	FALSE
PBRM1	hgnc:30064	PBRM1	DTC	9/2/20	NULL	0.167488584	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	MUNDULONE	chembl:CHEMBL465339	MUNDULONE	FALSE	FALSE	FALSE
PTGES3	hgnc:16049	PTGES3	DTC	9/2/20	NULL	5.834185692854944	GEDUNIN	chembl:CHEMBL465226	GEDUNIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124555	chembl:CHEMBL547488	CHEMBL:CHEMBL547488	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	DIHYDRO-OBLIQUIN	chembl:CHEMBL1610638	DIHYDRO-OBLIQUIN	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	METHIXENE HYDROCHLORIDE	rxcui:258230	METHIXENE HYDROCHLORIDE	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.024479101	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
ARNT	hgnc:700	ARNT	DTC	9/2/20	NULL	1.193356164447602	FUROSPONGOLIDE	chembl:CHEMBL1077108	FUROSPONGOLIDE	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.1848861663228679	NU-6027	chembl:CHEMBL303958	CHEMBL:CHEMBL303958	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	DTC	9/2/20	NULL	0.8401227397711121	DEMETHYLWEDELOLACTONE	chembl:CHEMBL2089002	DEMETHYLWEDELOLACTONE	FALSE	FALSE	FALSE
MAPK13	hgnc:6875	MAPK13	DTC	9/2/20	NULL	0.6482428547616604	N-(3-OXODODECANOYL)HOMOSERINELACTONE	chembl:CHEMBL8483	CHEMBL:CHEMBL8483	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.022305723	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001198641	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.019534104	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.030959712	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	GALLAMINE TRIETHIODIDE	rxcui:4639	GALLAMINE TRIETHIODIDE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	DTC	9/2/20	NULL	0.5073204950308646	ISOSILYBIN A	chembl:CHEMBL592676	ISOSILYBIN A	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.091159151	CID2350207	chembl:CHEMBL259615	CHEMBL:CHEMBL259615	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	DI-TERT-BUTYLHYDROQUINONE	chembl:CHEMBL480626	CHEMBL:CHEMBL480626	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	1.591141552596803	4-PHENOXY-BENZOIC ACID	chembl:CHEMBL107518	CHEMBL:CHEMBL107518	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002657809	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001124458	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.009532983	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.014630168	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	PROPENTOFYLLINE	rxcui:34644	PROPENTOFYLLINE	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.072927321	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.099446347	2-(PHENOXYMETHYL)BENZOTHIAZOLE	chembl:CHEMBL233302	2-(PHENOXYMETHYL)BENZOTHIAZOLE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.006811217	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.040452751	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.044955198	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.030281241	TERAZOSIN HYDROCHLORIDE	rxcui:235224	TERAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
ARSA	hgnc:713	ARSA	DTC	9/2/20	NULL	1.093909817410302	BENZOXATHIAN	chembl:CHEMBL191044	BENZOXATHIAN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.011464557	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.056157937	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.019607047	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	VITAMIN B2	chembl:CHEMBL1397833	VITAMIN B2	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.03378872	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005953251	FENOLDOPAM MESYLATE	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	1.029562181092048	GNF-PF-3314	chembl:CHEMBL582287	CHEMBL:CHEMBL582287	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.0148243	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	JNJ-1661010	iuphar.ligand:5206	JNJ1661010	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.024861587	CGS-15943	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.009922085	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.066297565	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.051478109	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.058019526	ROEMERINE	chembl:CHEMBL36654	ROEMERINE	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.016206071	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.009170044	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.011767743	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2853677784548614	CRIDANIMOD	ncit:C77948	CRIDANIMOD	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	(R)-EDELFOSINE	chembl:CHEMBL107514	(R)-EDELFOSINE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.063568609	TCMDC-124570	chembl:CHEMBL546475	CHEMBL:CHEMBL546475	FALSE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	inhibitor	0.9546849315580819	HTS-466284	drugbank:DB03921	4-(3-PYRIDIN-2-YL-1H-PYRAZOL-4-YL)QUINOLINE	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	DTC	9/2/20	NULL	0.2035181055647073	GNF-PF-5576	chembl:CHEMBL599896	CHEMBL:CHEMBL599896	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003091232	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-390527	chembl:CHEMBL160937	CHEMBL:CHEMBL160937	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01150727	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
EGLN1	hgnc:1232	EGLN1	DTC	9/2/20	NULL	2.386712328895204	N-OXALYLGLYCINE	chembl:CHEMBL90852	N-OXALYLGLYCINE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-123798	chembl:CHEMBL532510	CHEMBL:CHEMBL532510	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.5097832158805291	4-METHOXYCINNAMIC ACID	chembl:CHEMBL95770	4-METHOXYCINNAMIC ACID	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.026519026	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.013206155	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.040328473	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	ETODOLAC	rxcui:24605	ETODOLAC	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	BERGAPTEN	rxcui:15842	5-METHOXYPSORALEN	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.02232469	STAUROSPORINE	ncit:C1237	STAUROSPORINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.019447286	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.801643836	REL-BENDIGOLE F	chembl:CHEMBL1915271	CHEMBL:CHEMBL1915271	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.023976106	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	GNF-PF-134	chembl:CHEMBL578896	CHEMBL:CHEMBL578896	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	CGS-12066B	iuphar.ligand:109	CGS-12066	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.007658645	LYCOPENE	rxcui:29008	LYCOPENE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.013905633	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.035358701	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.017461813	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.089910396	GW632580X	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.013890918	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.040452751	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	0.212581665	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.038636991	RS-39604	drugbank:DB17050	RS-39604	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	DTC	9/2/20	NULL	0.3271505995993426	HINOKININ	chembl:CHEMBL242011	HINOKININ	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	DUP-697	chembl:CHEMBL42485	DUP-697	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.009922085	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	DNDI1417195	chembl:CHEMBL1303948	CHEMBL:CHEMBL1303948	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.090530468	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.016161179	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.1500219178162699	MADOLIN U	chembl:CHEMBL2333546	MADOLIN U	FALSE	FALSE	FALSE
BACE1	hgnc:933	BACE1	DTC	9/2/20	NULL	4.039051633514961	(2S)-2'-METHOXYKURARINONE	chembl:CHEMBL496451	CHEMBL:CHEMBL496451	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	NORETHYNODREL	rxcui:7515	NORETHYNODREL	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.020844649	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006780433	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	SJ000040549	chembl:CHEMBL589421	CHEMBL:CHEMBL589421	FALSE	FALSE	FALSE
ALB	hgnc:399	ALB	DTC	9/2/20	NULL	0.4773424657790409	EPICATECHIN GALLATE	iuphar.ligand:12462	EPICATECHIN GALLATE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	NSC-402083	chembl:CHEMBL1546228	CHEMBL:CHEMBL1546228	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	PK-11195	iuphar.ligand:8703	PK 11195	FALSE	FALSE	FALSE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.094608417	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.034184682	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.060353645	DEOXIEPINEPHRINE	chembl:CHEMBL31088	DEOXIEPINEPHRINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.010678802	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.6035364509849942	CLENBUTEROL HYDROCHLORIDE	rxcui:235955	CLENBUTEROL HYDROCHLORIDE	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.050246575	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.035418328	ENDO-ATROPINE	chembl:CHEMBL2449003	ENDO-ATROPINE	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.017945205	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	PROROXAN	ncit:C84119	PROROXAN	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.013126918	Epinephrine	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.1324279224103266	Anastrozole	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.1312691780892362	Binimetinib	rxcui:2049122	BINIMETINIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.525076712	Sodium Sulfate	rxcui:1299926	SODIUM SULFATE ANHYDROUS	TRUE	FALSE	FALSE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	2.100306849	Ombitasvir	rxcui:1597371	OMBITASVIR	TRUE	FALSE	FALSE
FGFR	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
SERPINC1	hgnc:775	SERPINC1	FDA	10-Apr-24	NULL	0.024721126	Progesterone	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
PROC	hgnc:9451	PROC	FDA	10-Apr-24	NULL	0.088996053	Progesterone	rxcui:8727	PROGESTERONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.002529881	Escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.016273039	Ethinyl Estradiol	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.006199253	Escitalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.012649403	Nefazodone	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
RAS	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
BRCA	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Rucaparib	rxcui:1862579	RUCAPARIB	TRUE	FALSE	TRUE
BRCA	NULL	NULL	FDA	10-Apr-24	NULL	NULL	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.3500511415712966	Sodium Nitrite	rxcui:9894	SODIUM NITRITE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	2.100306849	Voxilaprevir	rxcui:1939323	VOXILAPREVIR	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	FDA	10-Apr-24	NULL	0.1852122442176172	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
PROC	hgnc:9451	PROC	FDA	10-Apr-24	NULL	0.1591141552596803	Warfarin	rxcui:11289	WARFARIN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.022136455	Umeclidinium	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.035418328	Upadacitinib	rxcui:2196092	UPADACITINIB	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	MyCancerGenome	20-Jun-17	inhibitor	0.4930297768609811	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	MyCancerGenome	20-Jun-17	inhibitor	4.702860988936115	CH5424802	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	inhibitor	0.1101693521639275	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
ERBB4	hgnc:3432	ERBB4	MyCancerGenome	20-Jun-17	inhibitor	0.3017682254924971	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	MyCancerGenome	20-Jun-17	inhibitor	0.292250489	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.172722603	BMS-690514	drugbank:DB11665	BMS-690514	FALSE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.036925226	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PRKCZ	hgnc:9412	PRKCZ	MyCancerGenome	20-Jun-17	inhibitor	0.055387839	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.075732218	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.015825097	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.1875273972703375	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PRKCB	hgnc:9395	PRKCB	MyCancerGenome	20-Jun-17	inhibitor	0.041540879	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3R3	hgnc:8981	PIK3R3	MyCancerGenome	20-Jun-17	inhibitor	0.018990116	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.1041818873724097	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
PIK3C2G	hgnc:8973	PIK3C2G	MyCancerGenome	20-Jun-17	inhibitor	0.041540879	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PRKD3	hgnc:9408	PRKD3	MyCancerGenome	20-Jun-17	inhibitor	0.016616352	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.09055649	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.2641230947469542	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
CD274	hgnc:17635	CD274	MyCancerGenome	20-Jun-17	immunotherapy	0.6471533709721451	MPDL3280A	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
CD274	hgnc:17635	CD274	MyCancerGenome	20-Jun-17	antibody	0.6471533709721451	MPDL3280A	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
PSEN1	hgnc:9508	PSEN1	MyCancerGenome	20-Jun-17	other/unknown	0.4039051633514962	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	MyCancerGenome	20-Jun-17	antibody	11.66837138570988	APOMAB	ncit:C71693	APOMAB	FALSE	TRUE	TRUE
HGF	hgnc:4893	HGF	MyCancerGenome	20-Jun-17	antibody	7.778914257139925	RILOTUMUMAB	ncit:C67079	RILOTUMUMAB	FALSE	TRUE	TRUE
PDGFRA	hgnc:8803	PDGFRA	MyCancerGenome	20-Jun-17	antibody	0.2869271652223742	RAMUCIRUMAB	rxcui:1535922	RAMUCIRUMAB	TRUE	TRUE	TRUE
HSP90AA2	hgnc:5256	HSP90AA2P	MyCancerGenome	20-Jun-17	other/unknown	7.001022831425932	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
NOTCH3	hgnc:7883	NOTCH3	MyCancerGenome	20-Jun-17	other/unknown	1.050153425	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
HSP90AA2	hgnc:5256	HSP90AA2P	MyCancerGenome	20-Jun-17	other/unknown	7.001022831425932	RETASPIMYCIN	ncit:C80378	RETASPIMYCIN	FALSE	FALSE	TRUE
PSMA1	hgnc:9530	PSMA1	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA2	hgnc:9531	PSMA2	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
NOTCH2	hgnc:7882	NOTCH2	MyCancerGenome	20-Jun-17	other/unknown	0.7501095890813501	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
NOTCH4	hgnc:7884	NOTCH4	MyCancerGenome	20-Jun-17	other/unknown	0.8751278539282418	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
PSMA5	hgnc:9534	PSMA5	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMC3	hgnc:9549	PSMC3	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMC2	hgnc:9548	PSMC2	MyCancerGenome	20-Jun-17	other/unknown	0.5087952639117684	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD1	hgnc:9554	PSMD1	MyCancerGenome	20-Jun-17	other/unknown	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD2	hgnc:9559	PSMD2	MyCancerGenome	20-Jun-17	other/unknown	0.7326651800329465	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMF1	hgnc:9571	PSMF1	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD10P1	hgnc:16602	PSMD10P1	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD4P1	hgnc:9562	PSMD4P1	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.064824285	AZACITIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.443726799	PERIFOSINE	ncit:C1727	PERIFOSINE	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.4735540335109532	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	1.721562991334245	ANNAMYCIN	ncit:C2632	ANNAMYCIN	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	2.540693769469088	PMEA	rxcui:16521	ADEFOVIR	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.546954909	OSI-774	rxcui:477320	ERLOTINIB HYDROCHLORIDE	TRUE	FALSE	TRUE
ABP1	hgnc:80	AOC1	NCI	14-Sep-17	NULL	0.053038052	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADK	hgnc:257	ADK	NCI	14-Sep-17	NULL	2.625383561784724	LOMUSTINE	rxcui:6466	LOMUSTINE	TRUE	FALSE	TRUE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.2685814385457519	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.5147810905460244	CEFADROXIL	rxcui:1545975	CEFADROXIL ANHYDROUS	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	NCI	14-Sep-17	NULL	0.027774489	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
ATP7A	hgnc:869	ATP7A	NCI	14-Sep-17	NULL	0.8751278539282416	PLATINUM	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.041182487	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.1000146118775133	INTERFERON ALFA-2B	rxcui:5880	INTERFERON ALFA-2B	TRUE	TRUE	TRUE
BCHE	hgnc:983	BCHE	NCI	14-Sep-17	NULL	0.3281729452230906	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.017664481	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CCK	hgnc:1569	CCK	NCI	14-Sep-17	NULL	2.692701089009974	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
CCL3	hgnc:10627	CCL3	NCI	14-Sep-17	NULL	2.333674277141977	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
CCL22	hgnc:10621	CCL22	NCI	14-Sep-17	NULL	8.751278539282415	CC CHEMOKINES	ncit:C1591	RECOMBINANT BETA CHEMOKINE	FALSE	FALSE	FALSE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	0.1329308132549227	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	1.750255707856483	FDG	rxcui:1362737	FLUORODEOXYGLUCOSE F18	TRUE	FALSE	FALSE
CD28	hgnc:1653	CD28	NCI	14-Sep-17	NULL	0.2282942227638891	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
CD163	hgnc:1631	CD163	NCI	14-Sep-17	NULL	2.763561643983921	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
CD52	hgnc:1804	CD52	NCI	14-Sep-17	NULL	3.088686543276147	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
CDC25C	hgnc:1727	CDC25C	NCI	14-Sep-17	NULL	0.3323270331373069	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CDA	hgnc:1712	CDA	NCI	14-Sep-17	NULL	0.3704244884352345	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
CDH17	hgnc:1756	CDH17	NCI	14-Sep-17	NULL	1.750255707856483	HGF/SF	ncit:C1122	RECOMBINANT HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.1948336595016493	TOMUDEX	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.4234489615781814	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	1.693795846312725	AZQ	ncit:C1363	DIAZIQUONE	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.1693795846312726	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1272913242077442	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.077789143	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	NCI	14-Sep-17	NULL	0.3500511415712966	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	0.7955707762984016	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.013622434	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	0.1389091831632129	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.3292017005372696	PRIMAQUINE	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	0.3889457128569963	CANDESARTAN CILEXETIL	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
EEF1A1	hgnc:3189	EEF1A1	NCI	14-Sep-17	NULL	1.141471113819445	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.024973922	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
EPHB1	hgnc:3392	EPHB1	NCI	14-Sep-17	NULL	0.1591141552596803	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.069089041	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.016449772	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.031765076	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.1651184630053286	ANGIOGENESIS INHIBITOR	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	1.981421556063943	MMP INHIBITOR	ncit:C1970	MATRIX METALLOPROTEINASE INHIBITOR	FALSE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.076709527	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.037843367	STI 571	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
FKBP4	hgnc:3720	FKBP4	NCI	14-Sep-17	NULL	1.944728564284981	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
FST	hgnc:3971	FST	NCI	14-Sep-17	NULL	0.5834185692854944	BRDU	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.42006137	IMMUNOMODULATORS	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
FXN	hgnc:3951	FXN	NCI	14-Sep-17	NULL	0.1448487482363986	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.007242437	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GAL	hgnc:4114	GAL	NCI	14-Sep-17	NULL	1.312691780892362	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.079376676	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
HDGF	hgnc:4856	HDGF	NCI	14-Sep-17	NULL	2.917092846427472	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
HCK	hgnc:4840	HCK	NCI	14-Sep-17	NULL	0.6250913242344582	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
HIST3H2A	hgnc:20507	H2AC25	NCI	14-Sep-17	NULL	0.1448487482363986	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HEXB	hgnc:4879	HEXB	NCI	14-Sep-17	NULL	1.166837138570989	AMINOGLYCOSIDES	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	NCI	14-Sep-17	NULL	0.1857582708809946	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	5.527123287967842	INTERCALATING AGENT	ncit:C582	DNA INTERCALATING AGENT	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.1256164383629055	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.09869863	ANTINEOPLASTIC	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.07631929	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	1.221108633388244	GDNF	iuphar.ligand:4940	GDNF	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.067839369	PKC412	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.8140724222588294	PHOTOSENSITIZERS	ncit:C1420	PHOTOSENSITIZING AGENT	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.128537751	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	2.442217266776488	PHOTOFRIN	wikidata:Q47521991	PHOTOFRIN	FALSE	FALSE	FALSE
HSPA8	hgnc:5241	HSPA8	NCI	14-Sep-17	NULL	0.07631929	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
HTR4	hgnc:5299	HTR4	NCI	14-Sep-17	NULL	0.018570352	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HYAL2	hgnc:5321	HYAL2	NCI	14-Sep-17	NULL	0.4070362111294147	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.025865848	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.2941606231691568	MAPK INHIBITORS	ncit:C2149	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	NCI	14-Sep-17	NULL	5.000730593875666	IL-17	ncit:C1684	RECOMBINANT INTERLEUKIN-17	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.5357925636295356	CHINESE HERBS	ncit:C2663	CHINESE HERBS	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.1260688385010672	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.2381300282797936	LINEZOLID	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.076263865	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.06823609	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
LIPA	hgnc:6617	LIPA	NCI	14-Sep-17	NULL	0.4487835148349957	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.1875273972703375	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.1165542091802319	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.108374966	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.025081286	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.02262774	ALL-TRANS-RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.212152207	DTIC	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.2243917574174978	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.1750255707856483	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
MTAP	hgnc:7413	MTAP	NCI	14-Sep-17	NULL	10.50153425	DIFLUOROMETHYLORNITHINE	ncit:C226	EFLORNITHINE	FALSE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	NCI	14-Sep-17	NULL	0.4730420832044549	ZINC SULFATE	rxcui:1299928	ZINC SULFATE ANHYDROUS	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	1.500219178	AN-9	drugbank:DB05103	AN-9	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.045461187	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	NULL	LIGNAN	NULL	NULL	NULL	NULL	NULL
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.5000730593875666	POH	ncit:C1461	PERILLYL ALCOHOL	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	NULL	CAROTENOID	NULL	NULL	NULL	NULL	NULL
NAT1	hgnc:7645	NAT1	NCI	14-Sep-17	NULL	0.020688602	ACETYLSALICYLIC ACID	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.1056492378987816	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.5303805175322677	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.087005255	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2465148884304905	SOY PROTEIN	ncit:C1803	SOY PROTEIN ISOLATE	FALSE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	1.193356164447602	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
NR4A1	hgnc:7980	NR4A1	NCI	14-Sep-17	NULL	0.5834185692854944	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
NRIP1	hgnc:8001	NRIP1	NCI	14-Sep-17	NULL	1.693795846312725	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	0.3365876361262467	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
OGG1	hgnc:8125	OGG1	NCI	14-Sep-17	NULL	3.088686543276147	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
NTS	hgnc:8038	NTS	NCI	14-Sep-17	NULL	0.1741547968016401	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
NTRK3	hgnc:8033	NTRK3	NCI	14-Sep-17	NULL	0.2035181055647073	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
OGG1	hgnc:8125	OGG1	NCI	14-Sep-17	NULL	1.419126249613364	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
P2RX1	hgnc:8533	P2RX1	NCI	14-Sep-17	NULL	NULL	DIPHOSPHONATE	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.081030357	ZINC SULFATE	rxcui:1299928	ZINC SULFATE ANHYDROUS	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.040515178	17-AAG	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	NULL	ANTI-INFLAMMATORY DRUGS	NULL	NULL	NULL	NULL	NULL
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.1389091831632129	ZINC SULFATE	rxcui:1299928	ZINC SULFATE ANHYDROUS	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.015825097	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.055563673	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.052090944	GNF-PF-5061	chembl:CHEMBL601385	CHEMBL:CHEMBL601385	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.3125456621172291	HERBIMYCIN A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.1666910197958555	PAPAVERINE	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
PLTP	hgnc:9093	PLTP	NCI	14-Sep-17	NULL	4.375639269641208	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.2917092846427472	BETA-BLOCKER	ncit:C29576	BETA-ADRENERGIC ANTAGONIST	FALSE	FALSE	FALSE
PRKAA1	hgnc:9376	PRKAA1	NCI	14-Sep-17	NULL	0.071341945	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1325951293830669	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.060772768	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.364636606	PHOSPHODIESTERASE INHIBITOR	ncit:C744	PHOSPHODIESTERASE INHIBITOR	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	DTC	9/2/20	NULL	1.544343271638073	SEN-12333	chembl:CHEMBL565540	CHEMBL:CHEMBL565540	FALSE	FALSE	FALSE
PSEN1	hgnc:9508	PSEN1	NCI	14-Sep-17	NULL	0.175610941	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1041818873724097	VASCULAR ENDOTHELIAL GROWTH FACTOR	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
PTGER3	hgnc:9595	PTGER3	NCI	14-Sep-17	NULL	2.187819634820604	MISOPROSTOL	rxcui:42331	MISOPROSTOL	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	SB-218795	iuphar.ligand:5764	SB 218795	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.2243917574174978	ANTHRACYCLINE ANTIBIOTIC	ncit:C1594	ANTHRACYCLINE ANTINEOPLASTIC ANTIBIOTIC	FALSE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.6731752722524935	CLOMIPHENE	rxcui:2596	CLOMIPHENE	TRUE	FALSE	FALSE
PZP	hgnc:9750	PZP	NCI	14-Sep-17	NULL	0.2035181055647073	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PZP	hgnc:9750	PZP	NCI	14-Sep-17	NULL	2.500365296937833	PPD	rxcui:1362740	4-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
SERPINA5	hgnc:8723	SERPINA5	NCI	14-Sep-17	NULL	0.8204323630577265	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.1470803115845784	9-CIS RETINOIC ACID	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.014299475	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
SLC29A2	hgnc:11004	SLC29A2	NCI	14-Sep-17	NULL	0.4667348554283955	6-MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.020117882	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.047647615	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
TACSTD1	hgnc:11529	EPCAM	NCI	14-Sep-17	NULL	0.3818739726232327	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.789589041	HEPARIN SODIUM	rxcui:104466	TINZAPARIN SODIUM	TRUE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.2966535098061835	RAMIPRIL	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.063722902	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
TGFBR3	hgnc:11774	TGFBR3	NCI	14-Sep-17	NULL	0.1526385791735305	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.2243917574174978	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.1121958787087489	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	NULL	CAROTENOID	NULL	NULL	NULL	NULL	NULL
TNFRSF11B	hgnc:11909	TNFRSF11B	NCI	14-Sep-17	NULL	3.000438356	RISEDRONATE	rxcui:55685	RISEDRONIC ACID	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.024838066	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
TP73	hgnc:12003	TP73	NCI	14-Sep-17	NULL	0.6819178082557726	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	NCI	14-Sep-17	NULL	0.023182195	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
TSC22D3	hgnc:3051	TSC22D3	NCI	14-Sep-17	NULL	0.305277158	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	1.166837138570989	AMINOGLYCOSIDES	ncit:C2363	AMINOGLYCOSIDE ANTIBIOTIC	FALSE	FALSE	FALSE
TPM3	hgnc:12012	TPM3	NCI	14-Sep-17	NULL	0.2917092846427472	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
ERG	hgnc:3446	ERG	DTC	9/2/20	NULL	4.039051633514961	N-ACETYLASPARTIC ACID	chembl:CHEMBL1162494	N-ACETYLASPARTIC ACID	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.027347745	DICHLORVOS	drugbank:DB11397	DICHLORVOS	FALSE	FALSE	FALSE
TRIT1	hgnc:20286	TRIT1	NCI	14-Sep-17	NULL	2.625383561784725	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.015409441	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.049652644	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	FDA	10-Apr-24	NULL	0.4375639269641208	Indacaterol	rxcui:1114326	INDACATEROL	TRUE	FALSE	FALSE
UGT1A4	hgnc:12536	UGT1A4	NCI	14-Sep-17	NULL	0.3750547945406749	ANTINEOPLASTIC AGENT	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	FDA	10-Apr-24	NULL	0.2639729920045843	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	NCI	14-Sep-17	NULL	0.5048814541893701	PEITC	ncit:C2233	PHENETHYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.172722603	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	6.563458904461812	IL-7	iuphar.ligand:4999	IL-7	FALSE	FALSE	FALSE
VIP	hgnc:12693	VIP	NCI	14-Sep-17	NULL	0.6563458904461813	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.3500511415712966	sodium nitrite	rxcui:9894	SODIUM NITRITE	TRUE	FALSE	FALSE
CHRNE	hgnc:1966	CHRNE	PharmGKB	4/5/24	NULL	0.251232877	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
FIP1L1	hgnc:19124	FIP1L1	FDA	10-Apr-24	NULL	0.7001022831425933	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.015702055	olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.040021091	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
OTC	hgnc:8512	OTC	PharmGKB	4/5/24	NULL	NULL	sodium benzoate / sodium phenylacetate	NULL	NULL	NULL	NULL	NULL
ALDH5A1	hgnc:408	ALDH5A1	PharmGKB	4/5/24	NULL	0.4412409347537353	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.1770916399180253	mephedrone	drugbank:DB13108	MEPHEDRONE	FALSE	FALSE	FALSE
C9ORF72	hgnc:28337	C9orf72	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	1.875273972703375	morphine-6-glucuronide	ncit:C166899	MORPHINE GLUCURONIDE	FALSE	FALSE	FALSE
NELFCD	hgnc:15934	NELFCD	PharmGKB	4/5/24	NULL	4.375639269641208	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.038722471	bexarotene	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.092933931	cephalexin	rxcui:1299782	CEPHALEXIN ANHYDROUS	TRUE	FALSE	FALSE
CLCN6	hgnc:2024	CLCN6	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CYB5R1	hgnc:13397	CYB5R1	PharmGKB	4/5/24	NULL	0.7501095890813498	metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	3.150460274	daclatasvir	rxcui:1606218	DACLATASVIR	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	NULL	Angiotensin II Antagonists	NULL	NULL	NULL	NULL	NULL
ERCC2	hgnc:3434	ERCC2	PharmGKB	4/5/24	NULL	0.6819178082557726	ifosfamide	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
KCNE1	hgnc:6240	KCNE1	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.6563458904461813	amantadine	rxcui:282415	AMANTADINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	NULL	Other general anesthetics	NULL	NULL	NULL	NULL	NULL
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	NULL	volatile anesthetics	NULL	NULL	NULL	NULL	NULL
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.3125456621172291	trihexyphenidyl	rxcui:10811	TRIHEXYPHENIDYL	TRUE	FALSE	FALSE
MIR1264	hgnc:35246	MIR1264	PharmGKB	4/5/24	NULL	0.7292732116068681	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NT5C1A	hgnc:17819	NT5C1A	PharmGKB	4/5/24	NULL	2.333674277141977	cladribine	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	NULL	Antiemetics And Antinauseants	NULL	NULL	NULL	NULL	NULL
ZNF804A	hgnc:21711	ZNF804A	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
KLRD1	hgnc:6378	KLRD1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
ATP5F1E	hgnc:838	ATP5F1E	PharmGKB	4/5/24	NULL	1.071585127259071	certolizumab pegol	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	PharmGKB	4/5/24	NULL	0.020158043	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
RRM2B	hgnc:17296	RRM2B	PharmGKB	4/5/24	NULL	0.7001022831425934	cladribine	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	FDA	10-Apr-24	NULL	0.071731791	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
MED19	hgnc:29600	MED19	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.032899543	abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.4167275494896388	Ergot alkaloids	rxcui:4023	ERGOT ALKALOIDS	FALSE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	FDA	10-Apr-24	NULL	0.5672124979164529	Midostaurin	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
GABRG3	hgnc:4088	GABRG3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
GRIK3	hgnc:4581	GRIK3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
GRM3	hgnc:4595	GRM3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
HSPG2	hgnc:5273	HSPG2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.005534114	Nortriptyline	rxcui:7531	NORTRIPTYLINE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
MC4R	hgnc:6932	MC4R	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
NRG1	hgnc:7997	NRG1	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
NRXN1	hgnc:8008	NRXN1	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
SLC18A2	hgnc:10935	SLC18A2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
PRKAA2	hgnc:9377	PRKAA2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
PRKAB2	hgnc:9379	PRKAB2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
RGS2	hgnc:9998	RGS2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
SLC1A3	hgnc:10941	SLC1A3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CDK4	hgnc:1773	CDK4	MyCancerGenome	20-Jun-17	inhibitor	0.3704244884352345	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
SLC1A4	hgnc:10942	SLC1A4	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
SNAP25	hgnc:11132	SNAP25	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
SMYD3	hgnc:15513	SMYD3	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
CACNB2	hgnc:1402	CACNB2	PharmGKB	4/5/24	NULL	NULL	antipsychotics	NULL	NULL	NULL	NULL	NULL
IL18	hgnc:5986	IL18	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
RBX1	hgnc:9928	RBX1	PharmGKB	4/5/24	NULL	0.1829535583125243	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.8290684931951763	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
LRRC15	hgnc:20818	LRRC15	PharmGKB	4/5/24	NULL	0.9723642821424908	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
SUGCT	hgnc:16001	SUGCT	PharmGKB	4/5/24	NULL	NULL	hormonal contraceptives for systemic use	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	PharmGKB	4/5/24	NULL	0.0026791	estradiol	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
AGT	hgnc:333	AGT	PharmGKB	4/5/24	NULL	0.3889457128569963	amlodipine	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	benzodiazepine derivatives	NULL	NULL	NULL	NULL	NULL
GAL	hgnc:4114	GAL	PharmGKB	4/5/24	NULL	NULL	benzodiazepine derivatives	NULL	NULL	NULL	NULL	NULL
FCGR2B	hgnc:3618	FCGR2B	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	0.075496292	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
TAP1	hgnc:43	TAP1	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
TNFRSF10A	hgnc:11904	TNFRSF10A	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.029918901	testosterone	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00903591	testosterone	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
FBXL19	hgnc:25300	FBXL19	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.4906052389860809	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	1.521961485092594	sulfamethoxazole / trimethoprim	wikidata:Q48566821	SULFAMETHOXAZOLE / TRIMETHOPRIM	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	NULL	3-cyano-7-ethoxycoumarin	NULL	NULL	NULL	NULL	NULL
RYR1	hgnc:10483	RYR1	PharmGKB	4/5/24	NULL	NULL	volatile anesthetics	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	Quinolone Antibacterials	NULL	NULL	NULL	NULL	NULL
FHIT	hgnc:3701	FHIT	PharmGKB	4/5/24	NULL	1.750255707856483	interferon beta-1b	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
FHIT	hgnc:3701	FHIT	PharmGKB	4/5/24	NULL	1.166837138570988	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	0.546954909	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
HMGCS2	hgnc:5008	HMGCS2	PharmGKB	4/5/24	NULL	7.501095890813499	chlorothiazide	rxcui:2396	CHLOROTHIAZIDE	TRUE	FALSE	FALSE
SLC22A6	hgnc:10970	SLC22A6	PharmGKB	4/5/24	NULL	0.4526523382387457	lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
FAAH	hgnc:3553	FAAH	PharmGKB	4/5/24	NULL	0.2187819634820604	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
FGB	hgnc:3662	FGB	PharmGKB	4/5/24	NULL	1.400204566285186	eptifibatide	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.049864835	droperidol	rxcui:3648	DROPERIDOL	TRUE	FALSE	FALSE
FGA	hgnc:3661	FGA	PharmGKB	4/5/24	NULL	1.909369863116163	eptifibatide	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
ITGB3	hgnc:6156	ITGB3	PharmGKB	4/5/24	NULL	3.500511415712966	eptifibatide	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
NEDD4L	hgnc:7728	NEDD4L	PharmGKB	4/5/24	NULL	NULL	Beta blocking agents, selective	NULL	NULL	NULL	NULL	NULL
NR3C1	hgnc:7978	NR3C1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
CYP2A7P1	hgnc:2612	CYP2A7P1	PharmGKB	4/5/24	NULL	0.7721716358190368	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CYP4X1	hgnc:20244	CYP4X1	PharmGKB	4/5/24	NULL	NULL	taxanes	NULL	NULL	NULL	NULL	NULL
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.3906820776465364	PIMASERTIB	ncit:C84864	PIMASERTIB	FALSE	FALSE	TRUE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.1209854175937661	isoflurane	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
ACSS2	hgnc:15814	ACSS2	PharmGKB	4/5/24	NULL	0.1448487482363986	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ACSS2	hgnc:15814	ACSS2	PharmGKB	4/5/24	NULL	0.2386712328895204	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CYP2E1	hgnc:2631	CYP2E1	PharmGKB	4/5/24	NULL	0.046303061	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
MECP2	hgnc:6990	MECP2	PharmGKB	4/5/24	NULL	0.5966780822238011	mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
ZNF816	hgnc:26995	ZNF816	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CDKAL1	hgnc:21050	CDKAL1	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
MOB3B	hgnc:23825	MOB3B	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
MAP2K2	hgnc:6842	MAP2K2	MyCancerGenome	20-Jun-17	inhibitor	0.596678082	AZD8330	iuphar.ligand:8474	AZD8330	FALSE	FALSE	TRUE
LY96	hgnc:17156	LY96	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CERS6	hgnc:23826	CERS6	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
IL23R	hgnc:19100	IL23R	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
GBP6	hgnc:25395	GBP6	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	MyCancerGenome	20-Jun-17	inhibitor	0.062509132	MK-2461	iuphar.ligand:7962	MK-2461	FALSE	FALSE	TRUE
CNPY4	hgnc:28631	CNPY4	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
ARAP2	hgnc:16924	ARAP2	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
ALPL	hgnc:438	ALPL	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CD14	hgnc:1628	CD14	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.069332312	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
CHUK	hgnc:1974	CHUK	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CNTN5	hgnc:2175	CNTN5	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
CST5	hgnc:2477	CST5	PharmGKB	4/5/24	NULL	NULL	Tumor necrosis factor alpha (TNF-alpha) inhibitors	NULL	NULL	NULL	NULL	NULL
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.210030685	raloxifene	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
ASS1	hgnc:758	ASS1	PharmGKB	4/5/24	NULL	NULL	sodium benzoate / sodium phenylacetate	NULL	NULL	NULL	NULL	NULL
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.8153365098710326	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
CES2	hgnc:1864	CES2	PharmGKB	4/5/24	NULL	0.9376369863516874	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.1630673019742065	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	NULL	low density lipoprotein	NULL	NULL	NULL	NULL	NULL
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.7395446652914718	RIDAFOROLIMUS	ncit:C49061	RIDAFOROLIMUS	FALSE	FALSE	TRUE
OR10P1	hgnc:15378	OR10P1	PharmGKB	4/5/24	NULL	1.458546423213736	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
SH2B1	hgnc:30417	SH2B1	PharmGKB	4/5/24	NULL	0.2917092846427472	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.004698673	clonazepam	rxcui:2598	CLONAZEPAM	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006349558	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.00301197	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.005339401	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.05293112	tucatinib	rxcui:2361285	TUCATINIB	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	PharmGKB	4/5/24	NULL	0.025588534	dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	PharmGKB	4/5/24	NULL	NULL	nivolumab / relatlimab	NULL	NULL	NULL	NULL	NULL
DRD4	hgnc:3025	DRD4	PharmGKB	4/5/24	NULL	0.00781946	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
SDK1	hgnc:19307	SDK1	PharmGKB	4/5/24	NULL	NULL	Antiemetics And Antinauseants	NULL	NULL	NULL	NULL	NULL
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.1323722804261206	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	PharmGKB	4/5/24	NULL	0.044198376	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenome	20-Jun-17	inhibitor	0.015434354	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
HTR1B	hgnc:5287	HTR1B	PharmGKB	4/5/24	NULL	0.1654653505326507	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	Ascorbic acid (vitamin C), combinations	NULL	NULL	NULL	NULL	NULL
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	NULL	Antithyroid Preparations	NULL	NULL	NULL	NULL	NULL
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	NULL	Rubella vaccines	NULL	NULL	NULL	NULL	NULL
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	NULL	diclofenac acyl glucuronide	NULL	NULL	NULL	NULL	NULL
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	NULL	diclofenac acyl glucuronide	NULL	NULL	NULL	NULL	NULL
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	NULL	etoposide catechol	NULL	NULL	NULL	NULL	NULL
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.058341857	Vitamin K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	NULL	Opium derivatives and expectorants	NULL	NULL	NULL	NULL	NULL
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.012150335	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
IL27	hgnc:19157	IL27	PharmGKB	4/5/24	NULL	1.591141552596803	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NFATC2	hgnc:7776	NFATC2	PharmGKB	4/5/24	NULL	0.5303805175322677	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	PharmGKB	4/5/24	NULL	0.1627303860610366	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	0.012831787	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NOS2	hgnc:7873	NOS2	PharmGKB	4/5/24	NULL	0.1520492410300034	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NRG3	hgnc:7999	NRG3	PharmGKB	4/5/24	NULL	0.2386712328895204	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
SLC31A1	hgnc:11016	SLC31A1	PharmGKB	4/5/24	NULL	1.193356164447602	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
GSR	hgnc:4623	GSR	PharmGKB	4/5/24	NULL	0.054243462	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
LIG3	hgnc:6600	LIG3	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.013259513	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PIK3C2B	hgnc:8972	PIK3C2B	MyCancerGenome	20-Jun-17	inhibitor	0.1215455352678113	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
C6ORF15	hgnc:13927	C6orf15	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
DSCAM	hgnc:3039	DSCAM	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PSORS1C1	hgnc:17202	PSORS1C1	PharmGKB	4/5/24	NULL	0.2386712328895204	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
TIGD1	hgnc:14523	TIGD1	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
XYLT2	hgnc:15517	XYLT2	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ALDH3A1	hgnc:405	ALDH3A1	PharmGKB	4/5/24	NULL	0.03409589	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	NULL	Antithyroid Preparations	NULL	NULL	NULL	NULL	NULL
NLRP1	hgnc:14374	NLRP1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
PRKCI	hgnc:9404	PRKCI	MyCancerGenome	20-Jun-17	inhibitor	0.066465407	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.4773424657790409	tocilizumab	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
SCNN1B	hgnc:10600	SCNN1B	PharmGKB	4/5/24	NULL	NULL	Insulins And Analogues	NULL	NULL	NULL	NULL	NULL
VEGFC	hgnc:12682	VEGFC	PharmGKB	4/5/24	NULL	2.333674277141978	aflibercept	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
MIR1912	hgnc:35396	MIR1912	PharmGKB	4/5/24	NULL	0.7292732116068681	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
COQ8B	hgnc:19041	COQ8B	PharmGKB	4/5/24	NULL	NULL	Immunoglobulins	NULL	NULL	NULL	NULL	NULL
PRIMPOL	hgnc:26575	PRIMPOL	PharmGKB	4/5/24	NULL	NULL	Immunoglobulins	NULL	NULL	NULL	NULL	NULL
CASP3	hgnc:1504	CASP3	PharmGKB	4/5/24	NULL	NULL	Immunoglobulins	NULL	NULL	NULL	NULL	NULL
ITPKC	hgnc:14897	ITPKC	PharmGKB	4/5/24	NULL	NULL	Immunoglobulins	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.060772768	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
TNF	hgnc:11892	TNF	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
GSTT1	hgnc:4641	GSTT1	PharmGKB	4/5/24	NULL	0.098513454	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
GRIK2	hgnc:4580	GRIK2	PharmGKB	4/5/24	NULL	0.05853698	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	3.889457128569962	sulfamethoxazole / trimethoprim	wikidata:Q48566821	SULFAMETHOXAZOLE / TRIMETHOPRIM	FALSE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.3409589041278864	dapsone	rxcui:3108	DAPSONE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	PharmGKB	4/5/24	NULL	0.6471533709721451	atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
MAOB	hgnc:6834	MAOB	PharmGKB	4/5/24	NULL	NULL	5-hydroxyindole-3-acetic acid	NULL	NULL	NULL	NULL	NULL
HTR3B	hgnc:5298	HTR3B	PharmGKB	4/5/24	NULL	0.1342907192728759	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
CES2	hgnc:1864	CES2	PharmGKB	4/5/24	NULL	1.640864726115453	mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
MAOA	hgnc:6833	MAOA	PharmGKB	4/5/24	NULL	0.05853698	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	PharmGKB	4/5/24	NULL	NULL	Antiemetics And Antinauseants	NULL	NULL	NULL	NULL	NULL
HTR3B	hgnc:5298	HTR3B	PharmGKB	4/5/24	NULL	NULL	Antiemetics And Antinauseants	NULL	NULL	NULL	NULL	NULL
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	NULL	Antiemetics And Antinauseants	NULL	NULL	NULL	NULL	NULL
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	NULL	Other general anesthetics	NULL	NULL	NULL	NULL	NULL
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	NULL	volatile anesthetics	NULL	NULL	NULL	NULL	NULL
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1930429089547591	XL-765	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
AGAP1	hgnc:16922	AGAP1	PharmGKB	4/5/24	NULL	1.567393171214761	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	MyCancerGenome	20-Jun-17	antibody	0.2778183663264259	SYM004	ncit:C91381	FUTUXIMAB/MODOTUXIMAB MIXTURE	FALSE	TRUE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.08334551	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1346350544504987	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.033348791	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	0.2239133101735373	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
TNFRSF11A	hgnc:11908	TNFRSF11A	PharmGKB	4/5/24	NULL	NULL	Pyrazolones	NULL	NULL	NULL	NULL	NULL
AKT3	hgnc:393	AKT3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3076621361466474	MK2206	ncit:C90581	AKT INHIBITOR MK2206	FALSE	FALSE	TRUE
THSD7B	hgnc:29348	THSD7B	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.057073556	GANETESPIB	ncit:C77872	GANETESPIB	FALSE	FALSE	TRUE
MAP2K3	hgnc:6843	MAP2K3	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.3241214273808303	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.458240639	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCF4	hgnc:7662	NCF4	PharmGKB	4/5/24	NULL	0.2561349816375341	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
ALDH3A1	hgnc:405	ALDH3A1	PharmGKB	4/5/24	NULL	0.073181423	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	PharmGKB	4/5/24	NULL	0.018295356	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.128067491	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
F11	hgnc:3529	F11	PharmGKB	4/5/24	NULL	NULL	hormonal contraceptives for systemic use	NULL	NULL	NULL	NULL	NULL
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.1372151687343933	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.2734774543525755	tipiracil / trifluridine	drugbank:DB08937	TAS-102	FALSE	FALSE	FALSE
CXCL12	hgnc:10672	CXCL12	PharmGKB	4/5/24	NULL	0.1600843635234588	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.020257589	dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.044878351	CMA-676	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.017260904	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	PharmGKB	4/5/24	NULL	1.166837138570988	belzutifan	rxcui:2567226	BELZUTIFAN	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	PharmGKB	4/5/24	NULL	0.03292017	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
CHRNA5	hgnc:1959	CHRNA5	PharmGKB	4/5/24	NULL	NULL	combination nicotine replacement therapy	NULL	NULL	NULL	NULL	NULL
HLA-DQB1	hgnc:4944	HLA-DQB1	PharmGKB	4/5/24	NULL	NULL	Antithyroid Preparations	NULL	NULL	NULL	NULL	NULL
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.093680056	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
DCK	hgnc:2704	DCK	PharmGKB	4/5/24	NULL	0.1037701012563132	mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
UGT1A4	hgnc:12536	UGT1A4	PharmGKB	4/5/24	NULL	0.2625383561784725	imipramine	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	PharmGKB	4/5/24	NULL	NULL	fluorouracil / salicylic acid	NULL	NULL	NULL	NULL	NULL
AGTR1	hgnc:336	AGTR1	NCI	14-Sep-17	NULL	0.020696756	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	NULL	erythromycin ethylsuccinate / sulfisoxazole acetyl	NULL	NULL	NULL	NULL	NULL
AHRR	hgnc:346	AHRR	NCI	14-Sep-17	NULL	2.100306849	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.150021918	zonisamide	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.051885051	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	3.182283105193605	artesunate	rxcui:18346	ARTESUNATE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	PharmGKB	4/5/24	NULL	NULL	dasabuvir / ombitasvir / paritaprevir / ritonavir	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	NCI	14-Sep-17	NULL	0.4773424657790409	DIFLUOROMETHYLORNITHINE	ncit:C226	EFLORNITHINE	FALSE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.6731752722524935	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	NULL	Fibrates	NULL	NULL	NULL	NULL	NULL
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.1241316104862754	hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	PharmGKB	4/5/24	NULL	NULL	Antithyroid Preparations	NULL	NULL	NULL	NULL	NULL
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.1187956362798518	EPIGALLOCATECHIN GALLATE	rxcui:24246	EPIGALLOCATECHIN GALLATE	TRUE	FALSE	FALSE
FOXF2	hgnc:3810	FOXF2	PharmGKB	4/5/24	NULL	NULL	Antithyroid Preparations	NULL	NULL	NULL	NULL	NULL
SOD2	hgnc:11180	SOD2	PharmGKB	4/5/24	NULL	NULL	Antithyroid Preparations	NULL	NULL	NULL	NULL	NULL
ASL	hgnc:746	ASL	PharmGKB	4/5/24	NULL	NULL	sodium benzoate / sodium phenylacetate	NULL	NULL	NULL	NULL	NULL
CPS1	hgnc:2323	CPS1	PharmGKB	4/5/24	NULL	NULL	sodium benzoate / sodium phenylacetate	NULL	NULL	NULL	NULL	NULL
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.032412143	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
AQP1	hgnc:633	AQP1	NCI	14-Sep-17	NULL	0.095295229	GLYBURIDE	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	PharmGKB	4/5/24	NULL	0.1107756777124356	venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	NULL	volatile anesthetics	NULL	NULL	NULL	NULL	NULL
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	NULL	Alkylating Agents	NULL	NULL	NULL	NULL	NULL
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1130007271930297	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
BST1	hgnc:1118	BST1	PharmGKB	4/5/24	NULL	NULL	Beta blocking agents, selective	NULL	NULL	NULL	NULL	NULL
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1458546423213736	arteether	ncit:C73002	ARTEMOTIL	TRUE	FALSE	FALSE
CACNA1S	hgnc:1397	CACNA1S	PharmGKB	4/5/24	NULL	0.3195841219457973	isoflurane	rxcui:6026	ISOFLURANE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	PharmGKB	4/5/24	NULL	0.064347636	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CDH2	hgnc:1759	CDH2	PharmGKB	4/5/24	NULL	1.029562181092049	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BDNF-AS	hgnc:20608	BDNF-AS	PharmGKB	4/5/24	NULL	1.544343271638073	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
DCBLD1	hgnc:21479	DCBLD1	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.217423069	rocuronium	rxcui:68139	ROCURONIUM	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	PharmGKB	4/5/24	NULL	0.037398626	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
RARS	hgnc:9870	RARS1	PharmGKB	4/5/24	NULL	0.7242437411819931	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
RAF1	hgnc:9829	RAF1	PharmGKB	4/5/24	NULL	0.027855529	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
TBX2	hgnc:11597	TBX2	PharmGKB	4/5/24	NULL	2.917092846427472	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
MED12L	hgnc:16050	MED12L	PharmGKB	4/5/24	NULL	0.6482428547616604	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NUDT1	hgnc:8048	NUDT1	PharmGKB	4/5/24	NULL	NULL	8-oxo-dGTP	NULL	NULL	NULL	NULL	NULL
KNG1	hgnc:6383	KNG1	PharmGKB	4/5/24	NULL	NULL	hormonal contraceptives for systemic use	NULL	NULL	NULL	NULL	NULL
ABO	hgnc:79	ABO	PharmGKB	4/5/24	NULL	NULL	hormonal contraceptives for systemic use	NULL	NULL	NULL	NULL	NULL
CHRNA1	hgnc:1955	CHRNA1	PharmGKB	4/5/24	NULL	0.2273059360852575	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
ABL1	hgnc:76	ABL1	PharmGKB	4/5/24	NULL	1.322135606654178	asciminib	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	4.773424657790408	arteether	ncit:C73002	ARTEMOTIL	TRUE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	PharmGKB	4/5/24	NULL	0.071439008	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.1041818873724097	codeine	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
C5	hgnc:1331	C5	PharmGKB	4/5/24	NULL	1.591141552596803	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	0.076765601	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	0.1973972602845657	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	2.212697851403848	crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.093098708	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
ORMDL3	hgnc:16038	ORMDL3	PharmGKB	4/5/24	NULL	5.527123287967842	fluticasone propionate	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
CRHR1	hgnc:2357	CRHR1	PharmGKB	4/5/24	NULL	NULL	glucocorticoids	NULL	NULL	NULL	NULL	NULL
ERBB3	hgnc:3431	ERBB3	TALC	12-May-16	inhibitor	0.5147810905460245	MM121	chembl:CHEMBL3545071	SERIBANTUMAB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	0.1110098757625676	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
AKT1	hgnc:391	AKT1	TALC	12-May-16	inhibitor	0.1232574442152452	NELFINAVIR	rxcui:134527	NELFINAVIR	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	inhibitor	NULL	ENMD-0276	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	TALC	12-May-16	inhibitor	NULL	ENMD-0276	NULL	NULL	NULL	NULL	NULL
ANPEP	hgnc:500	ANPEP	TALC	12-May-16	NULL	0.7721716358190367	NGR-HTNF	ncit:C48383	CNGRC PEPTIDE-TNF ALPHA CONJUGATE	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	TALC	12-May-16	inhibitor	1.831662950082366	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	TALC	12-May-16	inhibitor	0.075768645	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	TALC	12-May-16	inhibitor	0.179119736	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FN1	hgnc:3778	FN1	TALC	12-May-16	antibody	NULL	1311-L19SIP	NULL	NULL	NULL	NULL	NULL
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	NULL	ENMD-0276	NULL	NULL	NULL	NULL	NULL
HDAC2	hgnc:4853	HDAC2	TALC	12-May-16	inhibitor	0.3846715841442821	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.2071308530007672	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
ITGAV	hgnc:6150	ITGAV	TALC	12-May-16	inhibitor	NULL	L-000845704	NULL	NULL	NULL	NULL	NULL
ITGB3	hgnc:6156	ITGB3	TALC	12-May-16	inhibitor	NULL	L-000845704	NULL	NULL	NULL	NULL	NULL
ITGB1	hgnc:6153	ITGB1	TALC	12-May-16	antibody	2.187819634820604	PF-04605412	chembl:CHEMBL2109622	PF-04605412	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.3163112725041837	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.4735540335109532	SELUMETINIB	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	TALC	12-May-16	inhibitor	1.312691780892362	AMG900	iuphar.ligand:8060	AMG-900	FALSE	FALSE	TRUE
MET	hgnc:7029	MET	TALC	12-May-16	inhibitor	3.000438356	METMAB	ncit:C82348	ONARTUZUMAB	FALSE	TRUE	TRUE
MERTK	hgnc:7027	MERTK	TALC	12-May-16	inhibitor	0.9546849315580819	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
MUC1	hgnc:7508	MUC1	TALC	12-May-16	vaccine	NULL	BLP25 LIPOSOME VACCINE STIMUVAX	NULL	NULL	NULL	NULL	NULL
PARP1	hgnc:270	PARP1	TALC	12-May-16	inhibitor	4.200613699	INIPARIB	ncit:C62526	INIPARIB	FALSE	FALSE	TRUE
NAIP	hgnc:7634	NAIP	TALC	12-May-16	inhibitor	3.281729452230906	TL 32711	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.058931169	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	TALC	12-May-16	inhibitor	0.1375060601009582	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
SMO	hgnc:11119	SMO	TALC	12-May-16	inhibitor	NULL	BMS-33923	NULL	NULL	NULL	NULL	NULL
TNFRSF10B	hgnc:11905	TNFRSF10B	TALC	12-May-16	agonist	11.66837138570988	DROZITUMAB	ncit:C95784	DROZITUMAB	FALSE	FALSE	TRUE
SMO	hgnc:11119	SMO	TALC	12-May-16	inhibitor	5.104912481248077	LDE 225	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
BIRC2	hgnc:590	BIRC2	TALC	12-May-16	inhibitor	1.312691780892362	TL 32711	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	TALC	12-May-16	vaccine	NULL	MUTANT P53 PEPTIDE PULSED DENDRITIC CELL	NULL	NULL	NULL	NULL	NULL
WT1	hgnc:12796	WT1	TALC	12-May-16	vaccine	NULL	WT-1 (WILMS TUMOR) ANALOG PEPTIDE VACCINE	NULL	NULL	NULL	NULL	NULL
XIAP	hgnc:592	XIAP	TALC	12-May-16	inhibitor	0.2083637747448194	TL 32711	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	NULL	AMAP102	NULL	NULL	NULL	NULL	NULL
CHEK1	hgnc:1925	CHEK1	TALC	12-May-16	inhibitor	NULL	SCH900776	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	NULL	MEHD7945	NULL	NULL	NULL	NULL	NULL
MTOR	hgnc:3942	MTOR	TALC	12-May-16	inhibitor	NULL	BEZ 235	NULL	NULL	NULL	NULL	NULL
EGFR	hgnc:3236	EGFR	TALC	12-May-16	inhibitor	0.6945459158160648	NECITUMUMAB	rxcui:1723738	NECITUMUMAB	TRUE	TRUE	TRUE
UNIPROT:P56817	hgnc:933	BACE1	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	POSIPHEN	drugbank:DB15317	POSIPHEN	FALSE	FALSE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	ABCIXIMAB	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TdgClinicalTrial	Jan-14	NULL	NULL	AC-100,DENTONIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43116	hgnc:9594	PTGER2	TdgClinicalTrial	Jan-14	NULL	NULL	AC-100,DENTONIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43115	hgnc:9595	PTGER3	TdgClinicalTrial	Jan-14	NULL	NULL	AC-100,DENTONIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35408	hgnc:9596	PTGER4	TdgClinicalTrial	Jan-14	NULL	NULL	AC-100,DENTONIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	NULL	AMAP102	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	NULL	AD 337	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	NULL	AD 337	NULL	NULL	NULL	NULL	NULL
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	NULL	AD01	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	ACLIDINIUM	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
UNIPROT:GLOBOTRIAOSYLCERAMIDE (GB3)	NULL	NULL	TdgClinicalTrial	Jan-14	NULL	NULL	AGALSIDASE ALFA	rxcui:338817	AGALSIDASE BETA	TRUE	FALSE	FALSE
UNIPROT:P08107	hgnc:5232	HSPA1A	TdgClinicalTrial	Jan-14	NULL	NULL	AIMPILA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.04907259	ETHINYL ESTRADIOL	rxcui:4124	ETHINYL ESTRADIOL	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.1447821817160693	AGOMELATINE	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
UNIPROT:Q99720	hgnc:8157	SIGMAR1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	DEXTROMETHORPHAN	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
UNIPROT:P43088	hgnc:9600	PTGFR	TdgClinicalTrial	Jan-14	NULL	NULL	NCX116	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q96BI3	hgnc:29509	APH1A	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	BMS-708163	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2442217266776488	TIMOLOL	rxcui:10600	TIMOLOL	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	NULL	BVT.28949	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01584	hgnc:5992	IL1B	TdgClinicalTrial	Jan-14	NULL	2.573905452730122	CANAKINUMAB	rxcui:853491	CANAKINUMAB	TRUE	TRUE	TRUE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.087512785	C-1311	chembl:CHEMBL338604	C-1311	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.085378327	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.01123399	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.024163678	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.4730420832044549	BDNF	iuphar.ligand:4872	BDNF	FALSE	FALSE	FALSE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.9460841664089098	BIOCHANIN A	ncit:C28201	BIOCHANIN A	FALSE	FALSE	FALSE
UNIPROT:Q16853	hgnc:550	AOC3	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	BTT-1023	ncit:C131541	TIMOLUMAB	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.1422972120208522	ZINC SULFATE	rxcui:1299928	ZINC SULFATE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.1810609352954983	C-1311	chembl:CHEMBL338604	C-1311	FALSE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	0.2373228078449469	CANDESARTAN	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.070197421	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.023274677	ACETYLSALICYLIC ACID	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.096758608	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P18084	hgnc:6160	ITGB5	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	CNTO-95	ncit:C61070	INTETUMUMAB	FALSE	FALSE	FALSE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.1785975212098452	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
UNIPROT:P42261	hgnc:4571	GRIA1	TdgClinicalTrial	Jan-14	NULL	NULL	CX1632/S 47445	NULL	NULL	NULL	NULL	NULL
UNIPROT:P42262	hgnc:4572	GRIA2	TdgClinicalTrial	Jan-14	NULL	NULL	CX1632/S 47445	NULL	NULL	NULL	NULL	NULL
UNIPROT:P42263	hgnc:4573	GRIA3	TdgClinicalTrial	Jan-14	NULL	NULL	CX1632/S 47445	NULL	NULL	NULL	NULL	NULL
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.4268916360625568	TYROSINE HYDROXYLASE INHIBITOR	ncit:C2155	TYROSINE HYDROXYLASE INHIBITOR	FALSE	FALSE	FALSE
UNIPROT:P48058	hgnc:4574	GRIA4	TdgClinicalTrial	Jan-14	NULL	NULL	CX1632/S 47445	NULL	NULL	NULL	NULL	NULL
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.021309932	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UNIPROT:Q04609	hgnc:3788	FOLH1	TdgClinicalTrial	Jan-14	NULL	NULL	DCVAX-PROSTATE	NULL	NULL	NULL	NULL	NULL
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.3977853881492006	VALDECOXIB	rxcui:278567	VALDECOXIB	TRUE	FALSE	FALSE
CARTPT	hgnc:24323	CARTPT	NCI	14-Sep-17	NULL	0.2442217266776488	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.3241214273808303	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.064111931	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
CGB5	hgnc:16452	CGB5	NCI	14-Sep-17	NULL	0.6141248097742047	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q8WXA8	hgnc:24003	HTR3C	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	DDP225	chembl:CHEMBL5095232	DDP-225	FALSE	FALSE	FALSE
UNIPROT:P54289	hgnc:1399	CACNA2D1	TdgClinicalTrial	Jan-14	NULL	0.1875273972703375	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	DDP225	chembl:CHEMBL5095232	DDP-225	FALSE	FALSE	FALSE
UNIPROT:P11177	hgnc:8808	PDHB	TdgClinicalTrial	Jan-14	NULL	NULL	DEXLIPOTAM	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	DESLORATADINE	rxcui:275635	DESLORATADINE	TRUE	FALSE	FALSE
UNIPROT:P10613	NULL	NULL	TdgClinicalTrial	Jan-14	NULL	NULL	DIO-902	rxcui:2588846	LEVOKETOCONAZOLE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	NULL	DOV 216,303	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	NULL	DOV 216,303	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31645	hgnc:11050	SLC6A4	TdgClinicalTrial	Jan-14	NULL	NULL	DOV 216,303	NULL	NULL	NULL	NULL	NULL
UNIPROT:P46098	hgnc:5297	HTR3A	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	DOLASETRON	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
UNIPROT:Q70Z44	hgnc:24004	HTR3D	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	DOLASETRON	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	NULL	DSC-103	NULL	NULL	NULL	NULL	NULL
COL1A2	hgnc:2198	COL1A2	NCI	14-Sep-17	NULL	0.4861821410712453	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
UNIPROT:P49768	hgnc:9508	PSEN1	TdgClinicalTrial	Jan-14	NULL	2.019525817	E2012	iuphar.ligand:7358	E2012	FALSE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TdgClinicalTrial	Jan-14	NULL	0.1672218829162245	DOXERCALCIFEROL	rxcui:11516	DOXERCALCIFEROL	TRUE	FALSE	FALSE
UNIPROT:P29459	hgnc:5969	IL12A	TdgClinicalTrial	Jan-14	NULL	NULL	DNA IL-12	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01375	hgnc:11892	TNF	TdgClinicalTrial	Jan-14	NULL	0.086861325	ETANERCEPT	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
UNIPROT:P24158	hgnc:9495	PRTN3	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	ELAFIN	drugbank:DB05161	ELAFIN	FALSE	FALSE	FALSE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.3659071166250487	ENTINOSTAT	ncit:C1863	ENTINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	0.7955707762984014	EP-100	chembl:CHEMBL4297748	EP-100	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	1.400204566285186	HALS	ncit:C29771	HORSE ANTI-MOUSE ANTI-LYMPHOCYTE SERUM	FALSE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.01715937	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
UNIPROT:Q13224	hgnc:4586	GRIN2B	TdgClinicalTrial	Jan-14	NULL	NULL	EVT-103	NULL	NULL	NULL	NULL	NULL
UNIPROT:P33681	hgnc:1700	CD80	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	GALIXIMAB	ncit:C26447	GALIXIMAB	FALSE	FALSE	FALSE
UNIPROT:Q9Y243	hgnc:393	AKT3	TdgClinicalTrial	Jan-14	NULL	0.546954909	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
CXCL2	hgnc:4603	CXCL2	NCI	14-Sep-17	NULL	0.5147810905460245	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
UNIPROT:P43490	hgnc:30092	NAMPT	TdgClinicalTrial	Jan-14	NULL	21.00306849427779	GMX1777	drugbank:DB05217	GMX1777	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	NULL	GSK-961081	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	NULL	GSK-961081	NULL	NULL	NULL	NULL	NULL
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.325124899	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	1.166837138570988	BIOCHANIN A	ncit:C28201	BIOCHANIN A	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.6250913242344582	4-HYDROXYANDROSTENEDIONE	rxcui:15070	FORMESTANE	FALSE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	GTP-010	NULL	NULL	NULL	NULL	NULL
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.011352028	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:Q92847	hgnc:4267	GHSR	TdgClinicalTrial	Jan-14	NULL	NULL	GTP-200	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.2917092846427472	TRASTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
UNIPROT:P14151	hgnc:10720	SELL	TdgClinicalTrial	Jan-14	NULL	NULL	SMART ANTI-L-SELECTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	NULL	HYDROXYTAMOXIFEN	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	NULL	HYDROXYTAMOXIFEN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P98170	hgnc:592	XIAP	TdgClinicalTrial	Jan-14	NULL	0.2083637747448194	HGS1029	ncit:C78484	IAP INHIBITOR HGS1029	FALSE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	NCI	14-Sep-17	NULL	1.640864726115453	TROFOSFAMIDE	rxcui:38865	TROFOSFAMIDE	FALSE	FALSE	FALSE
UNIPROT:Q13490	hgnc:590	BIRC2	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	HGS1029	ncit:C78484	IAP INHIBITOR HGS1029	FALSE	FALSE	FALSE
UNIPROT:P22304	hgnc:5389	IDS	TdgClinicalTrial	Jan-14	NULL	NULL	IDURONATE-2 SULFATASE	NULL	NULL	NULL	NULL	NULL
CYP27A1	hgnc:2605	CYP27A1	NCI	14-Sep-17	NULL	0.8204323630577265	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	NULL	MODIFIED IFN-ALPHA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	NULL	MODIFIED IFN-ALPHA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	NULL	MODIFIED IFN-BETA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	NULL	MODIFIED IFN-BETA	NULL	NULL	NULL	NULL	NULL
UNIPROT:P01589	hgnc:6008	IL2RA	TdgClinicalTrial	Jan-14	NULL	NULL	INTERLEUKIN-2 EXPRESSING PLASMID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14784	hgnc:6009	IL2RB	TdgClinicalTrial	Jan-14	NULL	NULL	INTERLEUKIN-2 EXPRESSING PLASMID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P31785	hgnc:6010	IL2RG	TdgClinicalTrial	Jan-14	NULL	NULL	INTERLEUKIN-2 EXPRESSING PLASMID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	1.009762908	IFERANSERIN	ncit:C90945	IFERANSERIN	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.072125922	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
UNIPROT:Q13464	hgnc:10251	ROCK1	TdgClinicalTrial	Jan-14	NULL	NULL	INS117548	NULL	NULL	NULL	NULL	NULL
UNIPROT:O75116	hgnc:10252	ROCK2	TdgClinicalTrial	Jan-14	NULL	NULL	INS117548	NULL	NULL	NULL	NULL	NULL
UNIPROT:O00519	hgnc:3553	FAAH	TdgClinicalTrial	Jan-14	NULL	NULL	IPI-940	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	NULL	IPL455	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	NULL	IPL455	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	NULL	MECASERMIN RINFIBATE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P48551	hgnc:5433	IFNAR2	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	INTERFERON ALFA-N3	rxcui:612937	INTERFERON ALFA-N3	TRUE	TRUE	TRUE
UNIPROT:P17181	hgnc:5432	IFNAR1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	INTERFERON ALFA-N3	rxcui:612937	INTERFERON ALFA-N3	TRUE	TRUE	TRUE
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	NULL	JVS-100	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.172950169	ROPINIROLE	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.6226206075378794	JNJ-37822681	drugbank:DB12579	JNJ-37822681	FALSE	FALSE	FALSE
UNIPROT:Q99835	hgnc:11119	SMO	TdgClinicalTrial	Jan-14	NULL	5.104912481248077	ERISMODEGIB	rxcui:1659191	SONIDEGIB	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	NULL	LU 02-750	NULL	NULL	NULL	NULL	NULL
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	NULL	LU 02-750	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	NULL	LU 02-750	NULL	NULL	NULL	NULL	NULL
UNIPROT:P20138	hgnc:1659	CD33	TdgClinicalTrial	Jan-14	NULL	8.078103267029922	LINTUZUMAB	ncit:C1716	LINTUZUMAB	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	LURTOTECAN	ncit:C1610	LURTOTECAN	FALSE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	NULL	LU 02-750	NULL	NULL	NULL	NULL	NULL
UNIPROT:P21918	hgnc:3026	DRD5	TdgClinicalTrial	Jan-14	NULL	NULL	LU 02-750	NULL	NULL	NULL	NULL	NULL
UNIPROT:P15692	hgnc:12680	VEGFA	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	RANIBIZUMAB	rxcui:595060	RANIBIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	VISILIZUMAB	ncit:C2229	VISILIZUMAB	FALSE	FALSE	FALSE
CYP2E1	hgnc:2631	CYP2E1	NCI	14-Sep-17	NULL	3.750547945	PERFLUOROOCTYLBROMIDE	ncit:C1422	PERFLUBRON	FALSE	FALSE	FALSE
UNIPROT:RIBOSOME A-SITE	NULL	NULL	TdgClinicalTrial	Jan-14	NULL	NULL	OMACETAXINE MEPESUCCINATE	rxcui:27100	OMACETAXINE MEPESUCCINATE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	NULL	ESTRIOL E3	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	NULL	ESTRIOL E3	NULL	NULL	NULL	NULL	NULL
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	NULL	ORMD-0901	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	ORTATAXEL	ncit:C1867	ORTATAXEL	FALSE	FALSE	FALSE
UNIPROT:P06858	hgnc:6677	LPL	TdgClinicalTrial	Jan-14	NULL	0.1442518440541058	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	NULL	OX914	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	NULL	OX914	NULL	NULL	NULL	NULL	NULL
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	NULL	PW2101	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q15761	hgnc:7958	NPY5R	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	PYY3-36	drugbank:DB05004	PEPTIDE YY (3-36)	FALSE	FALSE	FALSE
UNIPROT:P24941	hgnc:1771	CDK2	TdgClinicalTrial	Jan-14	NULL	NULL	TG02, SB1317	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.2892984641085096	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
UNIPROT:O15379	hgnc:4854	HDAC3	TdgClinicalTrial	Jan-14	NULL	0.2910624791335615	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P08311	hgnc:2532	CTSG	TdgClinicalTrial	Jan-14	NULL	NULL	DERMOLASTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08246	hgnc:3309	ELANE	TdgClinicalTrial	Jan-14	NULL	NULL	DERMOLASTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	NULL	DERMOLASTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P07477	hgnc:9475	PRSS1	TdgClinicalTrial	Jan-14	NULL	NULL	DERMOLASTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P07478	hgnc:9483	PRSS2	TdgClinicalTrial	Jan-14	NULL	NULL	DERMOLASTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35030	hgnc:9486	PRSS3	TdgClinicalTrial	Jan-14	NULL	NULL	DERMOLASTIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT ANTIHEMOPHILIC FACTOR	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00740	hgnc:3551	F9	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT ANTIHEMOPHILIC FACTOR	NULL	NULL	NULL	NULL	NULL
UNIPROT:P04275	hgnc:12726	VWF	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT ANTIHEMOPHILIC FACTOR	NULL	NULL	NULL	NULL	NULL
UNIPROT:P49286	hgnc:7464	MTNR1B	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	RAMELTEON	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT FACTOR IX FC FUSION PROTEIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	RETEPLASE	rxcui:76895	RETEPLASE	TRUE	FALSE	FALSE
UNIPROT:P63261	hgnc:144	ACTG1	TdgClinicalTrial	Jan-14	NULL	0.375054795	THYMOSIN BETA-4	drugbank:DB12003	THYMOSIN BETA-4	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.004698673	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
UNIPROT:Q96C86	hgnc:29812	DCPS	TdgClinicalTrial	Jan-14	NULL	105.0153424713889	RG3039	drugbank:DB16938	D-157495	FALSE	FALSE	FALSE
UNIPROT:P02671	hgnc:3661	FGA	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	RETEPLASE	rxcui:76895	RETEPLASE	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
UNIPROT:P09884	hgnc:9173	POLA1	TdgClinicalTrial	Jan-14	NULL	NULL	BROMOVINYL DEOXYURIDINE	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q14432	hgnc:8778	PDE3A	TdgClinicalTrial	Jan-14	NULL	0.7955707762984013	RPL-554	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
UNIPROT:Q13370	hgnc:8779	PDE3B	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	RPL-554	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
UNIPROT:P40238	hgnc:7217	MPL	TdgClinicalTrial	Jan-14	NULL	2.983390411119005	ROMIPLOSTIM	rxcui:805452	ROMIPLOSTIM	TRUE	FALSE	FALSE
UNIPROT:P21554	hgnc:2159	CNR1	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	RIMONABANT	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	0.1077080435603989	SCYLLO-INOSITOL	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	NULL	SLX-2101	NULL	NULL	NULL	NULL	NULL
UNIPROT:P27487	hgnc:3009	DPP4	TdgClinicalTrial	Jan-14	NULL	0.630092055	SITAGLIPTIN	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT THROMBOMODULIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	NULL	SOU-001	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	NULL	SOU-001	NULL	NULL	NULL	NULL	NULL
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	NULL	SOU-001	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q8NBP7	hgnc:20001	PCSK9	TdgClinicalTrial	Jan-14	NULL	NULL	SPC5001	NULL	NULL	NULL	NULL	NULL
CYP3A43	hgnc:17450	CYP3A43	NCI	14-Sep-17	NULL	3.750547945	GINKGO	ncit:C29072	GINKGO	FALSE	FALSE	FALSE
UNIPROT:P01031	hgnc:1331	C5	TdgClinicalTrial	Jan-14	NULL	1.591141552596803	ECULIZUMAB	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.5585922471882393	TC-6499	chembl:CHEMBL4594254	SIMPINICLINE	FALSE	FALSE	FALSE
UNIPROT:Q13164	hgnc:6880	MAPK7	TdgClinicalTrial	Jan-14	NULL	NULL	TG02, SB1317	NULL	NULL	NULL	NULL	NULL
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	NULL	TG02, SB1317	NULL	NULL	NULL	NULL	NULL
UNIPROT:O60674	hgnc:6192	JAK2	TdgClinicalTrial	Jan-14	NULL	NULL	TG02, SB1317	NULL	NULL	NULL	NULL	NULL
CYP3A7	hgnc:2640	CYP3A7	NCI	14-Sep-17	NULL	0.375054795	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
UNIPROT:P10747	hgnc:1653	CD28	TdgClinicalTrial	Jan-14	NULL	NULL	TGN 1412	NULL	NULL	NULL	NULL	NULL
UNIPROT:P51677	hgnc:1604	CCR3	TdgClinicalTrial	Jan-14	NULL	NULL	TPI-ASM8	NULL	NULL	NULL	NULL	NULL
UNIPROT:P32927	hgnc:2436	CSF2RB	TdgClinicalTrial	Jan-14	NULL	NULL	TPI-ASM8	NULL	NULL	NULL	NULL	NULL
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	1.221108633388244	6-DIAZO-5-OXO-L-NORLEUCINE	drugbank:DB17537	6-DIAZO-5-OXO-L-NORLEUCINE	FALSE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	NULL	LUTEINIZING HORMONE-RELEASING HORMONE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.07458476	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.1535312024435511	TRASTUZUMAB EMTANSINE	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
UNIPROT:P01730	hgnc:1678	CD4	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	TRX1	drugbank:DB05863	TRX1	FALSE	FALSE	FALSE
UNIPROT:P00740	hgnc:3551	F9	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	TTP889	drugbank:DB05131	TTP889	FALSE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TdgClinicalTrial	Jan-14	NULL	NULL	LUTEINIZING HORMONE-RELEASING HORMONE	NULL	NULL	NULL	NULL	NULL
UNIPROT:P37288	hgnc:895	AVPR1A	TdgClinicalTrial	Jan-14	NULL	NULL	VA111913	NULL	NULL	NULL	NULL	NULL
UNIPROT:P47901	hgnc:896	AVPR1B	TdgClinicalTrial	Jan-14	NULL	NULL	VA111913	NULL	NULL	NULL	NULL	NULL
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	NULL	VA111913	NULL	NULL	NULL	NULL	NULL
UNIPROT:P52333	hgnc:6193	JAK3	TdgClinicalTrial	Jan-14	NULL	1.141471113819445	VX-509	ncit:C132740	DECERNOTINIB	FALSE	FALSE	FALSE
UNIPROT:Q15858	hgnc:10597	SCN9A	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	XEN402	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	NULL	ETHYL EICOSAPENTAENOIC ACID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	6.848826682916673	YM-598	chembl:CHEMBL2107760	NEBENTAN	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.1101693521639275	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
UNIPROT:P12319	hgnc:3609	FCER1A	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	OMALIZUMAB	rxcui:302379	OMALIZUMAB	TRUE	FALSE	FALSE
UNIPROT:Q01362	hgnc:7316	MS4A2	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	OMALIZUMAB	rxcui:302379	OMALIZUMAB	TRUE	FALSE	FALSE
UNIPROT:P02671	hgnc:3661	FGA	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT FACTOR IX FC FUSION PROTEIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P02675	hgnc:3662	FGB	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT FACTOR IX FC FUSION PROTEIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P02679	hgnc:3694	FGG	TdgClinicalTrial	Jan-14	NULL	NULL	RECOMBINANT FACTOR IX FC FUSION PROTEIN	NULL	NULL	NULL	NULL	NULL
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	NULL	AZD1419	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	NULL	SAMIDOPRHAN	NULL	NULL	NULL	NULL	NULL
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	NULL	ETHYL EICOSAPENTAENOIC ACID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	NULL	ETHYL EICOSAPENTAENOIC ACID	NULL	NULL	NULL	NULL	NULL
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.6177373086552295	ZOLMITRIPTAN	rxcui:135775	ZOLMITRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	ACETOHEXAMIDE	rxcui:173	ACETOHEXAMIDE	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TdgClinicalTrial	Jan-14	NULL	4.200613698855561	ACENOCOUMAROL	rxcui:154	ACENOCOUMAROL	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.5427149481725528	ARFORMOTEROL	rxcui:304962	ARFORMOTEROL	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.1773907812016706	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	ANISTREPLASE	rxcui:40028	ANISTREPLASE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.2573905452730122	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P51787	hgnc:6294	KCNQ1	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.1643432589536604	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.1595977849109255	CEVIMELINE	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.8140724222588294	CARTEOLOL	rxcui:2116	CARTEOLOL	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.151464436	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TdgClinicalTrial	Jan-14	NULL	0.9376369863516874	CIMETIDINE	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1500219178162699	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:P43116	hgnc:9594	PTGER2	TdgClinicalTrial	Jan-14	NULL	0.6563458904461813	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:Q9NP56	hgnc:8792	PDE7B	TdgClinicalTrial	Jan-14	NULL	3.750547945406749	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.070197421	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.07182992	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.2386712328895204	ETHOTOIN	rxcui:4136	ETHOTOIN	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.267214612	FLURANDRENOLIDE	rxcui:4500	FLURANDRENOLIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	1.270346884734544	PEMIROLAST	rxcui:19551	PEMIROLAST	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.042619863	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TdgClinicalTrial	Jan-14	NULL	0.058602312	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.099446347	PHENOXYBENZAMINE	rxcui:8149	PHENOXYBENZAMINE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.5427149481725528	PROCATEROL	rxcui:34530	PROCATEROL	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.4475085616678508	PROCAINAMIDE	rxcui:8700	PROCAINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2004109589148645	PREDNICARBATE	rxcui:34369	PREDNICARBATE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	PROPERICIAZINE	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.1767935058440892	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.021846337	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08912	hgnc:1954	CHRM5	TdgClinicalTrial	Jan-14	NULL	0.093596562	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P37288	hgnc:895	AVPR1A	TEND	1-Aug-11	NULL	1.712206670729168	CONIVAPTAN	rxcui:302285	CONIVAPTAN	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TEND	1-Aug-11	NULL	0.2373228078449469	CANDESARTAN	rxcui:135481	CANDESARTAN CILEXETIL	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.2890330526735477	ALVIMOPAN	rxcui:1516803	ALVIMOPAN ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	2.500365296937833	ATRACURIUM	rxcui:1218	ATRACURIUM	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TEND	1-Aug-11	NULL	0.9376369863516875	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.099446347	BECLOMETHASONE	rxcui:1347	BECLOMETHASONE	TRUE	FALSE	FALSE
UNIPROT:P20711	hgnc:2719	DDC	TEND	1-Aug-11	NULL	5.250767123569449	CARBIDOPA	rxcui:1545982	CARBIDOPA ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.068637479	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
UNIPROT:P08246	hgnc:3309	ELANE	TEND	1-Aug-11	NULL	1.521961485092594	ALPHA-1-PROTEINASE INHIBITOR	rxcui:535	ALPHA 1-ANTITRYPSIN	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.201952582	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.1902451856365742	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.081407242	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.086551106	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.3182283105193606	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	0.7778914257139926	SAQUINAVIR	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.1221108633388244	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.1280674908187671	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.2282942227638891	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.8140724222588294	CARTEOLOL	rxcui:2116	CARTEOLOL	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.151464436	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TEND	1-Aug-11	NULL	0.1500219178162699	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:Q02643	hgnc:4266	GHRHR	TEND	1-Aug-11	NULL	19.69037671338543	SERMORELIN	rxcui:56188	SERMORELIN	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.096758608	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P24046	hgnc:4090	GABRR1	TEND	1-Aug-11	NULL	0.1704794520639432	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1835932560688619	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P05981	hgnc:5155	HPN	TEND	1-Aug-11	NULL	52.50767123569449	BENTIROMIDE	rxcui:18896	BENTIROMIDE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	DEXBROMPHENIRAMINE	rxcui:1767	BROMPHENIRAMINE	TRUE	FALSE	FALSE
CYP7B1	hgnc:2652	CYP7B1	NCI	14-Sep-17	NULL	3.500511415712966	GINKGO	ncit:C29072	GINKGO	FALSE	FALSE	FALSE
UNIPROT:P27930	hgnc:5994	IL1R2	TEND	1-Aug-11	NULL	5.834185692854945	ANAKINRA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	0.482607272	DONEPEZIL	rxcui:135447	DONEPEZIL	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	2.500365296937833	DOXACURIUM	rxcui:23651	DOXACURIUM	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.596678082	DISOPYRAMIDE	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.3488881809680697	MAPK INHIBITORS	ncit:C2149	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
UNIPROT:P01375	hgnc:11892	TNF	TEND	1-Aug-11	NULL	2.258394462	GOLIMUMAB	rxcui:819300	GOLIMUMAB	TRUE	TRUE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.091583148	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.091583148	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P41143	hgnc:8153	OPRD1	TEND	1-Aug-11	NULL	0.1458546423213736	HYDROCODONE	rxcui:5489	HYDROCODONE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.1178056726441863	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
UNIPROT:P48551	hgnc:5433	IFNAR2	TEND	1-Aug-11	NULL	1.312691780892362	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
UNIPROT:P08235	hgnc:7979	NR3C2	TEND	1-Aug-11	NULL	2.763561643983921	DESOXYCORTICOSTERONE PIVALATE	rxcui:22537	DESOXYCORTICOSTERONE PIVALATE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.093098708	IPRATROPIUM	rxcui:1546373	IPRATROPIUM CATION	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.060772768	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
UNIPROT:P10828	hgnc:11799	THRB	TEND	1-Aug-11	NULL	0.061791905	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.063858524	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.1356787370431382	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
UNIPROT:Q9NP56	hgnc:8792	PDE7B	TEND	1-Aug-11	NULL	3.750547945406749	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P22888	hgnc:6585	LHCGR	TEND	1-Aug-11	NULL	2.461297089173179	MENOTROPINS	rxcui:134404	UROFOLLITROPIN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.693795846312725	METHDILAZINE	rxcui:29648	METHDILAZINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.693795846312725	MEQUITAZINE	rxcui:29528	MEQUITAZINE	TRUE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.056097939	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.053361455	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.050879526	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.049723174	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.074797252	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.072125922	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TEND	1-Aug-11	NULL	0.060077427	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.6482428547616604	PHENTERMINE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	PHENIRAMINE	rxcui:8132	PHENIRAMINE	TRUE	FALSE	FALSE
UNIPROT:P08185	hgnc:1540	SERPINA6	TEND	1-Aug-11	NULL	3.281729452230906	ALCLOMETASONE	rxcui:108088	ALCLOMETASONE	TRUE	FALSE	FALSE
UNIPROT:P49286	hgnc:7464	MTNR1B	TEND	1-Aug-11	NULL	10.50153424713889	RAMELTEON	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TEND	1-Aug-11	NULL	0.2864054794674245	ROSIGLITAZONE	rxcui:84108	ROSIGLITAZONE	TRUE	FALSE	FALSE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TEND	1-Aug-11	NULL	0.358239472	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
UNIPROT:P10912	hgnc:4263	GHR	TEND	1-Aug-11	NULL	1.400204566285186	SOMATROPIN RECOMBINANT	rxcui:314845	SOMATROPIN (RECOMBINANT DNA ORIGIN)	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.3580068493342807	SUPROFEN	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TEND	1-Aug-11	NULL	2.187819634820604	SULODEXIDE	ncit:C152467	SULODEXIDE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.1123158743009508	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:Q14432	hgnc:8778	PDE3A	TEND	1-Aug-11	NULL	0.2651902587661338	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.4375639269641208	TOLMETIN	rxcui:10636	TOLMETIN	TRUE	FALSE	FALSE
UNIPROT:P08514	hgnc:6138	ITGA2B	TEND	1-Aug-11	NULL	3.500511415712967	TIROFIBAN	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.2792961235941196	TRIDIHEXETHYL	rxcui:38617	TRIDIHEXETHYL	TRUE	FALSE	FALSE
UNIPROT:P80404	hgnc:23	ABAT	TEND	1-Aug-11	NULL	0.08470687	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
HEPATITIS B VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pradefovir	ncit:C66453	PRADEFOVIR	FALSE	FALSE	FALSE
TRANSFERRIN	hgnc:11740	TF	TTD	2020.06.01	NULL	NULL	EP-2167	NULL	NULL	NULL	NULL	NULL
TUMOR SUPPRESSOR CANDIDATE 2	hgnc:17034	TUSC2	TTD	2020.06.01	NULL	NULL	CNVN-202	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	N-8295	NULL	NULL	NULL	NULL	NULL
UNIPROT:O43497	hgnc:1394	CACNA1G	TEND	1-Aug-11	NULL	0.1750255707856483	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	NULL	TV-1390	NULL	NULL	NULL	NULL	NULL
DIACYLGLYCEROL ACYLTRANSFERASE 1	hgnc:2843	DGAT1	TTD	2020.06.01	NULL	NULL	P-7435	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 9	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASP-4901	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	PF-05230905	NULL	NULL	NULL	NULL	NULL
NA-K-CL COTRANSPORTER	NULL	NULL	TTD	2020.06.01	NULL	NULL	CLP-1001	NULL	NULL	NULL	NULL	NULL
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	NULL	BI 655064	NULL	NULL	NULL	NULL	NULL
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.062620956	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
GLYCOSIDE HYDROLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MNLP-18	NULL	NULL	NULL	NULL	NULL
DIABLO	hgnc:21528	DIABLO	NCI	14-Sep-17	NULL	4.773424657790408	CASPASE INHIBITOR	ncit:C38461	CASPASE INHIBITOR	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 2	hgnc:6027	CXCR2	TTD	2020.06.01	NULL	2.917092846427472	AZD4721	iuphar.ligand:12100	VIMNERIXIN	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	NULL	ABI-013	NULL	NULL	NULL	NULL	NULL
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	NULL	PF-4554878	NULL	NULL	NULL	NULL	NULL
GTPASE NRAS	hgnc:7989	NRAS	TTD	2020.06.01	NULL	NULL	Reovirus	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAY1163877	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Embeconazole	ncit:C98011	EMBECONAZOLE	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	CT-200	NULL	NULL	NULL	NULL	NULL
FK506-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	FK-505	NULL	NULL	NULL	NULL	NULL
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	SAR-161271	NULL	NULL	NULL	NULL	NULL
DHFR	hgnc:2861	DHFR	NCI	14-Sep-17	NULL	0.546954909	4-HYDROPEROXYCYCLOPHOSPHAMIDE	ncit:C1423	PERFOSFAMIDE	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	SSR411298	NULL	NULL	NULL	NULL	NULL
PYRUVATE KINASE	hgnc:17797	MAP3K20	TTD	2020.06.01	NULL	NULL	AGS-348	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	Ublituximab + umbralisib	NULL	NULL	NULL	NULL	NULL
ERK ACTIVATOR KINASE 1	hgnc:6840	MAP2K1	TTD	2020.06.01	NULL	0.4735540335109532	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.8334550989792777	INCB50465	ncit:C113434	PARSACLISIB	FALSE	FALSE	FALSE
DPYS	hgnc:3013	DPYS	NCI	14-Sep-17	NULL	0.3281729452230906	DEXRAZOXANE	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	4.375639269641208	IMG-7289	ncit:C131827	BOMEDEMSTAT	FALSE	FALSE	FALSE
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	AX-024	iuphar.ligand:11253	AX-024	FALSE	FALSE	FALSE
CD40L RECEPTOR	hgnc:11919	CD40	TTD	2020.06.01	NULL	NULL	BI 655064	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 9	hgnc:1610	CCR9	TTD	2020.06.01	NULL	NULL	CCX507	NULL	NULL	NULL	NULL	NULL
NCK ADAPTOR PROTEIN 1	hgnc:7664	NCK1	TTD	2020.06.01	NULL	26.25383561784724	AX-024	iuphar.ligand:11253	AX-024	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.5147810905460245	BGB-3111	rxcui:2262435	ZANUBRUTINIB	TRUE	FALSE	FALSE
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IMO-9200	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C1S COMPONENT	hgnc:1247	C1S	TTD	2020.06.01	NULL	NULL	SHP616	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CHS-131	chembl:CHEMBL1236924	INT131	FALSE	FALSE	FALSE
INTERLEUKIN 17 RECEPTOR	hgnc:5985	IL17RA	TTD	2020.06.01	NULL	NULL	CNTO-6785	NULL	NULL	NULL	NULL	NULL
MELANOMA ANTIGEN GP75	hgnc:12450	TYRP1	TTD	2020.06.01	NULL	NULL	FLX-787	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAN-300	chembl:CHEMBL4297822	SAN-300	FALSE	FALSE	FALSE
DPEP1	hgnc:3002	DPEP1	NCI	14-Sep-17	NULL	0.1017590527823536	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
STEROID HORMONE RECEPTOR ERR	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDP-122	chembl:CHEMBL1200908	HALOBETASOL PROPIONATE	FALSE	FALSE	FALSE
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	NULL	AFP TCR	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	JCAR018	NULL	NULL	NULL	NULL	NULL
OVARIAN CARCINOMA ANTIGEN CA125	hgnc:15582	MUC16	TTD	2020.06.01	NULL	NULL	JCAR020	NULL	NULL	NULL	NULL	NULL
T-CELL-SPECIFIC SURFACE GLYCOPROTEIN CD28	hgnc:1653	CD28	TTD	2020.06.01	NULL	NULL	AU101	NULL	NULL	NULL	NULL	NULL
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Baltaleucel-T	ncit:C129374	BALTALEUCEL-T	FALSE	FALSE	FALSE
PLACENTAL CADHERIN	hgnc:1762	CDH3	TTD	2020.06.01	NULL	26.25383561784724	PF-06671008	chembl:CHEMBL4297805	PF-06671008	FALSE	FALSE	FALSE
DTYMK	hgnc:3061	DTYMK	NCI	14-Sep-17	NULL	1.009762908	D4T	rxcui:59763	STAVUDINE	TRUE	FALSE	FALSE
MELANOMA-ASSOCIATED ANTIGEN 3	hgnc:6801	MAGEA3	TTD	2020.06.01	NULL	8.751278539282415	KITE-718	ncit:C135534	AUTOLOGOUS MAGE-A3/A6-SPECIFIC TCR GENE-ENGINEERED LYMPHOCYTES KITE-718	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	DSP-1200	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-2A	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	NULL	DSP-1200	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	DSP-1200	NULL	NULL	NULL	NULL	NULL
CHEMOSENSORY RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PH10 nasal spray	NULL	NULL	NULL	NULL	NULL
G-PROTEIN-COUPLED RECEPTOR PGR3	hgnc:19995	GPR139	TTD	2020.06.01	NULL	26.25383561784724	TAK-041	iuphar.ligand:11685	ZELATRIAZIN (TAK-041)	FALSE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 4	hgnc:11333	SSTR4	TTD	2020.06.01	NULL	NULL	CNTX-0290	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	DNL151	NULL	NULL	NULL	NULL	NULL
ELAVL1	hgnc:3312	ELAVL1	NCI	14-Sep-17	NULL	1.105424657593568	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
SYNAPTIC TRANSMISSION	NULL	NULL	TTD	2020.06.01	NULL	NULL	E2730	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	GDC0310	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.6	hgnc:10596	SCN8A	TTD	2020.06.01	NULL	NULL	PRAX-330	NULL	NULL	NULL	NULL	NULL
SUPEROXIDE DISMUTASE CU-ZN	NULL	NULL	TTD	2020.06.01	NULL	NULL	BIIB067	chembl:CHEMBL3833346	TOFERSEN	FALSE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMO-02	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID B RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ASP8062	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	BTD-001	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CX1789	NULL	NULL	NULL	NULL	NULL
GROWTH/DIFFERENTIATION FACTOR 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	Domagrozumab	ncit:C166800	DOMAGROZUMAB	FALSE	FALSE	FALSE
QUINONE REDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	EPI 589	NULL	NULL	NULL	NULL	NULL
MEASLES VIRUS FUSION GLYCOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AC 165198	NULL	NULL	NULL	NULL	NULL
MHC CLASS II ANTIGEN DR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AEA-35p	NULL	NULL	NULL	NULL	NULL
CELLULAR TUMOR ANTIGEN P53	hgnc:11998	TP53	TTD	2020.06.01	NULL	NULL	ISA-P53-01	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-072	drugbank:DB15156	ABT-072	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	ABT-450	rxcui:1597373	PARITAPREVIR	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	APD-515	NULL	NULL	NULL	NULL	NULL
X-LINKED INHIBITOR OF APOPTOSIS PROTEIN	hgnc:592	XIAP	TTD	2020.06.01	NULL	NULL	HGS-1029	NULL	NULL	NULL	NULL	NULL
TRANSTHYRETIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALN-TTR01	NULL	NULL	NULL	NULL	NULL
MEASLES VIRUS FUSION GLYCOPROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	AMG 876	NULL	NULL	NULL	NULL	NULL
DIHYDROOROTATE DEHYDROGENASE	hgnc:2867	DHODH	TTD	2020.06.01	NULL	NULL	LAS-186323	NULL	NULL	NULL	NULL	NULL
GASTRIC H(+)/K(+) ATPASE ALPHA	hgnc:819	ATP4A	TTD	2020.06.01	NULL	NULL	Esomeprazole magnesium + Aspirin	NULL	NULL	NULL	NULL	NULL
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	ATL101	NULL	NULL	NULL	NULL	NULL
COLONY STIMULATING FACTOR-1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.9546849315580818	ARRY-382	iuphar.ligand:9108	ARRY-382	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	PF-06439535	NULL	NULL	NULL	NULL	NULL
INTERCELLULAR ADHESION MOLECULE ICAM-1	hgnc:5344	ICAM1	TTD	2020.06.01	NULL	NULL	APC-8015F	NULL	NULL	NULL	NULL	NULL
PLACENTAL CADHERIN	hgnc:1762	CDH3	TTD	2020.06.01	NULL	NULL	PF-3732010	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C3	hgnc:7422	MT-CO3	TTD	2020.06.01	NULL	NULL	Imprime PGG immunotherapeutic	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pacritinib	rxcui:2595243	PACRITINIB	TRUE	FALSE	TRUE
TENASCIN	hgnc:5318	TNC	TTD	2020.06.01	NULL	NULL	F-16-IL-2 fusion protein	NULL	NULL	NULL	NULL	NULL
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.2381300282797936	GS-9820	ncit:C103277	ACALISIB	FALSE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	DFP-11207	ncit:C116720	THYMIDYLATE SYNTHASE INHIBITOR DFP-11207	FALSE	FALSE	FALSE
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	NULL	CF602	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	URC102	NULL	NULL	NULL	NULL	NULL
DOPAMINE D5 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	DS-8273	chembl:CHEMBL4594356	DS-8273A	FALSE	FALSE	FALSE
B-CELL-ACTIVATING FACTOR RECEPTOR	hgnc:17755	TNFRSF13C	TTD	2020.06.01	NULL	35.00511415712966	VAY736	ncit:C116788	IANALUMAB	FALSE	FALSE	FALSE
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	US8586571, 12	NULL	NULL	NULL	NULL	NULL
POLO-LIKE KINASE 2	hgnc:19699	PLK2	TTD	2020.06.01	NULL	NULL	US8598172, 1	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8598210, Table XV, 1	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US8598210, Table XV, 4	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-10	NULL	NULL	TTD	2020.06.01	NULL	NULL	3ts4	NULL	NULL	NULL	NULL	NULL
CARBOXYPEPTIDASE B1	hgnc:2299	CPB1	TTD	2020.06.01	NULL	NULL	US8710232, 1	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8759338, 1	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8759338, 12	NULL	NULL	NULL	NULL	NULL
ADAM METALLOPEPTIDASE 33	hgnc:15478	ADAM33	TTD	2020.06.01	NULL	NULL	US8772478, 2	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8829193, 3	NULL	NULL	NULL	NULL	NULL
PRKACA MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AGGGWZCOULSEER-PYUWXLGESA-N	NULL	NULL	NULL	NULL	NULL
PLASMA RETINOL-BINDING PROTEIN	hgnc:9922	RBP4	TTD	2020.06.01	NULL	NULL	A1-10436	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS CORE PROTEIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	US8877733, 27	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C ZETA	hgnc:9412	PRKCZ	TTD	2020.06.01	NULL	NULL	Methyl 2-amino-4-phenylthiophene-3-carboxylate	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C ZETA	hgnc:9412	PRKCZ	TTD	2020.06.01	NULL	NULL	Y-9680	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US8889696, Staurosporine	NULL	NULL	NULL	NULL	NULL
ROTAMASE D	hgnc:9257	PPID	TTD	2020.06.01	NULL	NULL	US8901295, F673	NULL	NULL	NULL	NULL	NULL
HEMATOPOIETIC CELL KINASE	hgnc:4840	HCK	TTD	2020.06.01	NULL	NULL	US8933228, 3	NULL	NULL	NULL	NULL	NULL
BCL-2-RELATED PROTEIN A1	hgnc:991	BCL2A1	TTD	2020.06.01	NULL	NULL	US8937193-compound-7	NULL	NULL	NULL	NULL	NULL
CASEIN KINASE II ALPHA PRIME	hgnc:2459	CSNK2A2	TTD	2020.06.01	NULL	NULL	US8940736, 23	NULL	NULL	NULL	NULL	NULL
ACTIVATED CDC42 KINASE 1	hgnc:19297	TNK2	TTD	2020.06.01	NULL	NULL	BDBM50379214	NULL	NULL	NULL	NULL	NULL
HIF-PROLYL HYDROXYLASE 2	hgnc:1232	EGLN1	TTD	2020.06.01	NULL	NULL	US9422240, 1-297	NULL	NULL	NULL	NULL	NULL
PIM-3 PROTEIN KINASE	hgnc:19310	PIM3	TTD	2020.06.01	NULL	NULL	US9434725, 315	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9493447, 1001	NULL	NULL	NULL	NULL	NULL
BETA-ADRENERGIC RECEPTOR KINASE 1	hgnc:289	GRK2	TTD	2020.06.01	NULL	NULL	US9493490, C	NULL	NULL	NULL	NULL	NULL
BETA-ADRENERGIC RECEPTOR KINASE 1	hgnc:289	GRK2	TTD	2020.06.01	NULL	NULL	US9493490, L	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9586942, 2	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9586942, 3*	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9586945, 1	NULL	NULL	NULL	NULL	NULL
MEK KINASE KINASE 4	hgnc:6866	MAP4K4	TTD	2020.06.01	NULL	NULL	BDBM50011552	NULL	NULL	NULL	NULL	NULL
MEK KINASE KINASE 4	hgnc:6866	MAP4K4	TTD	2020.06.01	NULL	NULL	BDBM50011553	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4C	hgnc:8782	PDE4C	TTD	2020.06.01	NULL	NULL	CS-W011402	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US9073936, 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 1B	hgnc:8775	PDE1B	TTD	2020.06.01	NULL	NULL	US9073936, 2	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	AKOS020330481	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC DEMETHYLASE 5A	hgnc:9886	KDM5A	TTD	2020.06.01	NULL	NULL	BDBM50158803	NULL	NULL	NULL	NULL	NULL
CALMODULIN-DEPENDENT KINASE II	hgnc:1470	CAMKK2	TTD	2020.06.01	NULL	NULL	US9623028, Compound 101	NULL	NULL	NULL	NULL	NULL
TYRO3 TYROSINE KINASE RECEPTOR	hgnc:12446	TYRO3	TTD	2020.06.01	NULL	NULL	BDBM50444058	NULL	NULL	NULL	NULL	NULL
N-ACETYLGLUCOSAMINYLTRANSFERASE I	NULL	NULL	TTD	2020.06.01	NULL	NULL	US9656955, Example 652	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 2	hgnc:3169	S1PR2	TTD	2020.06.01	NULL	NULL	SCHEMBL15295829	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9670220, 33	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 3	hgnc:3167	S1PR3	TTD	2020.06.01	NULL	NULL	US9670220, 77	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-6	NULL	NULL	TTD	2020.06.01	NULL	NULL	US10081632, Compound 25	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	NULL	Anti-FGFR3	NULL	NULL	NULL	NULL	NULL
M1-PRIME SEGMENT OF MEMBRANE-EXPRESSED IGE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-M1 prime	chembl:CHEMBL2109456	QUILIZUMAB	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-9256	drugbank:DB12876	GS-9256	FALSE	FALSE	FALSE
LATE INWARD SODIUM CURRENT	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-6615	ncit:C174857	ELECLAZINE	FALSE	FALSE	FALSE
HEPATITIS C VIRUS NS3 HELICASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-9857	rxcui:1939323	VOXILAPREVIR	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	NULL	KOS-2484	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	JB991	drugbank:DB05081	JB991	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MSH-372	NULL	NULL	NULL	NULL	NULL
SODIUM/POTASSIUM TRANSPORT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alilusem	ncit:C74249	ALILUSEM	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	Tyverb/Tykerb	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Tyverb/Tykerb	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	B7-2/GM-CSF	NULL	NULL	NULL	NULL	NULL
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1	hgnc:2357	CRHR1	TTD	2020.06.01	NULL	NULL	GSK586529	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK610677	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dilmapimod	ncit:C96531	DILMAPIMOD	FALSE	FALSE	FALSE
HIF-PROLYL HYDROXYLASE 1	hgnc:44465	RAB4B-EGLN2	TTD	2020.06.01	NULL	3.500511415712967	GSK1278863	rxcui:2628210	DAPRODUSTAT	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	NULL	Darotropium + 642444	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Losmapimod	ncit:C96532	LOSMAPIMOD	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	IPI-940	NULL	NULL	NULL	NULL	NULL
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Kombiglyze XR/Komboglyze FDC	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-8683	NULL	NULL	NULL	NULL	NULL
ACETYL-COA CARBOXYLASE 2	hgnc:85	ACACB	TTD	2020.06.01	NULL	1.693795846312725	PF-05175157	drugbank:DB12096	PF-05175157	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	DE-766	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 7	hgnc:15631	TLR7	TTD	2020.06.01	NULL	NULL	IM0-8400	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 8	hgnc:15632	TLR8	TTD	2020.06.01	NULL	NULL	IM0-8400	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	IM0-8400	NULL	NULL	NULL	NULL	NULL
TERT MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
APOC-III MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-APOCIII	NULL	NULL	NULL	NULL	NULL
SLC5A2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-SGLT2	NULL	NULL	NULL	NULL	NULL
PCSK9 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	BMS-PCSK9	NULL	NULL	NULL	NULL	NULL
GLUCOCORTICOID RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-GCCR	NULL	NULL	NULL	NULL	NULL
STAT3 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-STAT3	NULL	NULL	NULL	NULL	NULL
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lopinavir	rxcui:195088	LOPINAVIR	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	0.8751278539282416	JD-5037	iuphar.ligand:10690	JD5037	FALSE	FALSE	FALSE
PROSTATIC ACID PHOSPHATASE	hgnc:125	ACP3	TTD	2020.06.01	NULL	NULL	MVI-816	NULL	NULL	NULL	NULL	NULL
PHOSPHORYLATED PROTEIN KINASE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	MNX-100	NULL	NULL	NULL	NULL	NULL
HEAT SHOCK PROTEIN 70	hgnc:5232	HSPA1A	TTD	2020.06.01	NULL	NULL	Enkastim-ev	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	SDZ-MAR-327	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	SDZ-MAR-327	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GLYCOPROTEIN 41	NULL	NULL	TTD	2020.06.01	NULL	NULL	MaC46/M87o	NULL	NULL	NULL	NULL	NULL
APOLIPOPROTEIN E	hgnc:613	APOE	TTD	2020.06.01	NULL	0.9053046764774912	AEM-28	drugbank:DB17642	AEM-28	FALSE	FALSE	FALSE
PROTEIN-TYROSINE PHOSPHATASE 1B	hgnc:9642	PTPN1	TTD	2020.06.01	NULL	NULL	TTP-814	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG7203	NULL	NULL	NULL	NULL	NULL
CARCINOEMBRYONIC ANTIGEN CEA	hgnc:1817	CEACAM5	TTD	2020.06.01	NULL	NULL	123-Iodine-labeled MFE-23	NULL	NULL	NULL	NULL	NULL
TRIGEMINAL GANGLION STIMULATION-INDUCED RESPONSE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Carabersat	ncit:C77999	CARABERSAT	FALSE	FALSE	FALSE
F2R	hgnc:3537	F2R	NCI	14-Sep-17	NULL	1.346350544504987	ARGATROBAN	rxcui:15202	ARGATROBAN	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	NULL	AG-013958	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	NULL	GTP-200	NULL	NULL	NULL	NULL	NULL
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	RANBEZOLID HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	SBI-087	NULL	NULL	NULL	NULL	NULL
RESPIRATORY SYNCYTIAL VIRUS PROTEIN F	NULL	NULL	TTD	2020.06.01	NULL	NULL	Motavizumab	ncit:C88584	MOTAVIZUMAB	FALSE	FALSE	FALSE
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	SKL-10406	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	SKL-10406	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XIII	hgnc:3534	F13B	TTD	2020.06.01	NULL	NULL	NN8717	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV7.2	hgnc:6296	KCNQ2	TTD	2020.06.01	NULL	NULL	ICA-69673	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV7.3	hgnc:6297	KCNQ3	TTD	2020.06.01	NULL	NULL	ICA-69673	NULL	NULL	NULL	NULL	NULL
FCGR2B	hgnc:3618	FCGR2B	NCI	14-Sep-17	NULL	0.2734774543525755	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
SODIUM/IODIDE COTRANSPORTER	hgnc:11040	SLC5A5	TTD	2020.06.01	NULL	NULL	Ad5CMV-NIS	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.9376369863516875	Oglemilast	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS TRANSMISSION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ushercell	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pafuramidine	rxcui:718967	PAFURAMIDINE	FALSE	FALSE	FALSE
T-CELLS	NULL	NULL	TTD	2020.06.01	NULL	NULL	RTL-1000	drugbank:DB17946	RTL-1000	FALSE	FALSE	FALSE
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	IW-6118	NULL	NULL	NULL	NULL	NULL
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.2651902587661338	ANGIOGENESIS INHIBITOR	ncit:C1742	ANGIOGENESIS INHIBITOR	FALSE	FALSE	FALSE
RING FINGER PROTEIN 43	hgnc:18505	RNF43	TTD	2020.06.01	NULL	NULL	RNF43-721	NULL	NULL	NULL	NULL	NULL
FDFT1	hgnc:3629	FDFT1	NCI	14-Sep-17	NULL	1.346350544504987	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	NULL	CSL-654	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NS3 HELICASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-9451	chembl:CHEMBL2013174	VEDROPREVIR	FALSE	FALSE	FALSE
TUMOR ANTIGEN NGCGM3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Racotumomab	ncit:C95024	RACOTUMOMAB	FALSE	FALSE	FALSE
EBOLA VIRUS VP24 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-6002	NULL	NULL	NULL	NULL	NULL
EBOLA VIRUS VP35 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	AVI-6002	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-22	hgnc:14900	IL22	TTD	2020.06.01	NULL	NULL	ILV-095	NULL	NULL	NULL	NULL	NULL
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.045226246	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
THYROID HORMONE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	3,5-diiodothyropropionic acid (Allan-Herndon-Dudley syndrome), Zarion Pharmaceuticals	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	PWT-33597	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-7295	drugbank:DB12724	AZD-7295	FALSE	FALSE	FALSE
TNF RELATED ACTIVATION PROTEIN	hgnc:11935	CD40LG	TTD	2020.06.01	NULL	NULL	UltraCD40L	NULL	NULL	NULL	NULL	NULL
GHRH	hgnc:4265	GHRH	NCI	14-Sep-17	NULL	1.207072901969988	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	4.375639269641208	RG-7090	ncit:C166619	BASIMGLURANT	FALSE	FALSE	FALSE
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.6471533709721451	MPDL-3280A	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
B-CELL-SPECIFIC GLYCOPROTEIN B29	hgnc:1699	CD79B	TTD	2020.06.01	NULL	26.25383561784724	DCDS-4501A	chembl:CHEMBL3301582	POLATUZUMAB VEDOTIN	FALSE	FALSE	FALSE
NUCLEOLIN	hgnc:7667	NCL	TTD	2020.06.01	NULL	NULL	ACT-GRO-777	NULL	NULL	NULL	NULL	NULL
SURVIVAL MOTOR NEURON PROTEIN	hgnc:11117	SMN1	TTD	2020.06.01	NULL	NULL	RG7800	NULL	NULL	NULL	NULL	NULL
QUINONE REDUCTASE 1	hgnc:2874	NQO1	TTD	2020.06.01	NULL	NULL	Coenzyme Q10 analog	NULL	NULL	NULL	NULL	NULL
GRIA4	hgnc:4574	GRIA4	NCI	14-Sep-17	NULL	0.2386712328895204	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD3	NULL	NULL	TTD	2020.06.01	NULL	NULL	MGD006	ncit:C117238	FLOTETUZUMAB	FALSE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK-1399686	NULL	NULL	NULL	NULL	NULL
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nolatrexed	ncit:C143088	NOLATREXED	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydroergotoxine	rxcui:3419	DIHYDROERGOTOXINE	FALSE	FALSE	FALSE
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	Netivudine	ncit:C96547	NETIVUDINE	FALSE	FALSE	FALSE
LYASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	YM-116	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	ZD7114	NULL	NULL	NULL	NULL	NULL
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	0.6177373086552295	Darbepoetin alfa	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Floxuridine	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
GPI	hgnc:4458	GPI	NCI	14-Sep-17	NULL	2.187819634820604	FDG	rxcui:1362737	FLUORODEOXYGLUCOSE F18	TRUE	FALSE	FALSE
HAEMOPHILUS INFLUENZAE CRM197	NULL	NULL	TTD	2020.06.01	NULL	NULL	HibTITER	rxcui:221105	HAEMOPHILUS CAPSULAR OLIGOSACCHARIDE	FALSE	FALSE	FALSE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	NULL	LY333531	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
STRESS-ACTIVATED PROTEIN KINASE 2B	NULL	NULL	TTD	2020.06.01	NULL	NULL	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
BACTERIAL 16S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Framycetin	rxcui:4556	FRAMYCETIN	TRUE	FALSE	FALSE
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	RGD-891	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	0.057197899	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
RIBOSOMAL PROTEIN S6 KINASE BETA-1	hgnc:10436	RPS6KB1	TTD	2020.06.01	NULL	0.078840347	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.596678082	Disopyramide	rxcui:3541	DISOPYRAMIDE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	XR-5944	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	Anti-CD3 and anti-Her2/neu bispecific antibody-armed activated T cells	NULL	NULL	NULL	NULL	NULL
GNRH1	hgnc:4419	GNRH1	NCI	14-Sep-17	NULL	0.9211872146613068	DDC	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
INTERLEUKIN-4	hgnc:6014	IL4	TTD	2020.06.01	NULL	NULL	IL-4R	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	CL-316,243	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mitomycin A	ncit:C1164	MITOMYCIN A	FALSE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	CMI-392	NULL	NULL	NULL	NULL	NULL
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	NULL	CMI-392	NULL	NULL	NULL	NULL	NULL
GRIA4	hgnc:4574	GRIA4	NCI	14-Sep-17	NULL	0.4339476961627644	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gramicidin D	rxcui:5011	GRAMICIDIN	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clarithromycin	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
BACTERIAL 50S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clindamycin	rxcui:2582	CLINDAMYCIN	TRUE	FALSE	FALSE
BACTERIAL 23S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Spiramycin	rxcui:9991	SPIRAMYCIN	TRUE	FALSE	FALSE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Adaphostin	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	L-694,458	NULL	NULL	NULL	NULL	NULL
GRM1	hgnc:4593	GRM1	NCI	14-Sep-17	NULL	0.3547815624033412	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	DP-VPA	drugbank:DB05821	DP-VPA	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Artemisinin SP	NULL	NULL	NULL	NULL	NULL
NITRIC-OXIDE SYNTHASE ENDOTHELIAL	hgnc:7876	NOS3	TTD	2020.06.01	NULL	NULL	Autologous cell based gene therapy	NULL	NULL	NULL	NULL	NULL
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.1226814748497534	FGF-1	iuphar.ligand:4923	FGF-1	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.043756393	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
GROUP IIA PHOSPHOLIPASE A2	NULL	NULL	TTD	2020.06.01	NULL	NULL	KH064	drugbank:DB04287	KH064	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	5-FP	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	NULL	ELND-004	NULL	NULL	NULL	NULL	NULL
CANDIDA THYMIDYLATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	NB1011	ncit:C1882	BRIVUDINE PHOSPHORAMIDATE	FALSE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	NCI	14-Sep-17	NULL	0.7895890411382631	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.2	hgnc:6256	KCNJ10	TTD	2020.06.01	NULL	1.071585127259071	Gliquidone	rxcui:25793	GLIQUIDONE	FALSE	FALSE	FALSE
PLASMODIUM DOXP REDUCTOISOMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Fosclin	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	Irofulven/Taxotere	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-4/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	HMR-1031	NULL	NULL	NULL	NULL	NULL
TENASCIN	hgnc:5318	TNC	TTD	2020.06.01	NULL	6.563458904461812	8H9	ncit:C170251	OMBURTAMAB	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS TAT PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-HIV ribozyme therapy	NULL	NULL	NULL	NULL	NULL
MOTILIN RECEPTOR	hgnc:4495	MLNR	TTD	2020.06.01	NULL	NULL	RWJ-68023	NULL	NULL	NULL	NULL	NULL
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.2573905452730122	Procyclidine	rxcui:8718	PROCYCLIDINE	TRUE	FALSE	FALSE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.729273212	AMP-579	chembl:CHEMBL1950650	CHEMBL:CHEMBL1950650	FALSE	FALSE	FALSE
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Efaproxyn	ncit:C1435	EFAPROXIRAL	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.546954909	BACILLUS CALMETTE-GUERIN	hemonc:59	BCG VACCINE	TRUE	FALSE	FALSE
HEME OXYGENASE 1	hgnc:5013	HMOX1	TTD	2020.06.01	NULL	5.834185692854944	Stannsoporfin	ncit:C152424	STANNSOPORFIN	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GS-7340	rxcui:1721603	TENOFOVIR ALAFENAMIDE	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.1715936968486748	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
NATURAL KILLER CELL ACTIVATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Virulizin	ncit:C26677	VIRULIZIN	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TRICIRIBINE	ncit:C142998	TRICIRIBINE	FALSE	FALSE	TRUE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Doripenem	rxcui:119771	DORIPENEM	TRUE	FALSE	FALSE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	2.059124362184098	PENTAMIDINE	rxcui:7994	PENTAMIDINE	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.1132444383228493	Maprotiline	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV1.5	hgnc:6224	KCNA5	TTD	2020.06.01	NULL	0.3889457128569963	Dronedarone	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	Pancreatic cancer vaccine	NULL	NULL	NULL	NULL	NULL
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.045758319	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	LADIRUBICIN	ncit:C83861	LADIRUBICIN	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	CX-516	iuphar.ligand:4165	CX516	FALSE	FALSE	FALSE
CILIARY NEUROTROPHIC FACTOR RECEPTOR ALPHA	hgnc:2170	CNTFR	TTD	2020.06.01	NULL	NULL	PegCNTF	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	NULL	CB1 antagonist, Bayer	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE SECRETAGOGUE RECEPTOR 1	hgnc:4267	GHSR	TTD	2020.06.01	NULL	NULL	EP-01492	NULL	NULL	NULL	NULL	NULL
IL1RN	hgnc:6000	IL1RN	NCI	14-Sep-17	NULL	0.2344092465879218	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	MCH antagonist	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	T-226293	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	FK-614	drugbank:DB12557	FK-614	FALSE	FALSE	FALSE
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	0.8607814956671229	Tosagestin	ncit:C77017	TOSAGESTIN	FALSE	FALSE	FALSE
TNF RELATED APOPTOSIS INDUCING LIGAND	hgnc:11925	TNFSF10	TTD	2020.06.01	NULL	NULL	DA-3607	NULL	NULL	NULL	NULL	NULL
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	NULL	T83193	NULL	NULL	NULL	NULL	NULL
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	1.640864726115453	CELL DIFFERENTIATING AGENT	ncit:C2122	CELL DIFFERENTIATING AGENT	FALSE	FALSE	FALSE
SUCCINATE-SEMIALDEHYDE DEHYDROGENASE	hgnc:408	ALDH5A1	TTD	2020.06.01	NULL	NULL	T83193	NULL	NULL	NULL	NULL	NULL
CCR5 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Maraviroc	rxcui:620216	MARAVIROC	TRUE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1367387271762877	OFLOXACIN	rxcui:7623	OFLOXACIN	TRUE	FALSE	FALSE
ADENOSINE KINASE	hgnc:257	ADK	TTD	2020.06.01	NULL	NULL	GP-3269	NULL	NULL	NULL	NULL	NULL
INTERFERON-ALPHA 2	hgnc:5423	IFNA2	TTD	2020.06.01	NULL	NULL	Hebergel	NULL	NULL	NULL	NULL	NULL
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	4.039051633514961	CO-101	chembl:CHEMBL3039516	GEMCITABINE ELAIDATE	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.014650578	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bromfenac	rxcui:19737	BROMFENAC	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALLOPREGNANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.045758319	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
CALCIUM-ACTIVATED POTASSIUM CHANNEL	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chlorzoxazone	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tigecycline	rxcui:384455	TIGECYCLINE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR BETA-2	hgnc:4082	GABRB2	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR GAMMA-2	hgnc:4087	GABRG2	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.5147810905460245	CHINESE HERBS	ncit:C2663	CHINESE HERBS	FALSE	FALSE	FALSE
RIBOSOMAL PROTEIN S6 KINASE ALPHA-1	hgnc:10430	RPS6KA1	TTD	2020.06.01	NULL	1.250182648468916	BI-D1870	iuphar.ligand:8038	BI-D1870	FALSE	FALSE	FALSE
BACTERIAL GLUCOSAMINE-6-PHOSPHATE SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glucose-6-Phosphate	rxcui:1541246	GLUCOSE-6-PHOSPHATE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.108374966	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	0.4167275494896389	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID MAJOR GROOVE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Carzinophilin	ncit:C1040	CARZINOPHILIN	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.6584034010745392	ATG	ncit:C278	ANTI-THYMOCYTE GLOBULIN	TRUE	TRUE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pirarubicin	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Zinostatin stimalamer	ncit:C162544	ZINOSTATIN STIMALAMER	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Decitabine	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	NULL	MRX-6	NULL	NULL	NULL	NULL	NULL
INTEGRIN ALPHA-4	hgnc:6140	ITGA4	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	NULL	Dextromethorphan+quinidine	NULL	NULL	NULL	NULL	NULL
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dextromethorphan+quinidine	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefdinir	rxcui:25037	CEFDINIR	TRUE	FALSE	FALSE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	NULL	AIR-insulin	NULL	NULL	NULL	NULL	NULL
GMCSFR-ALPHA	hgnc:2435	CSF2RA	TTD	2020.06.01	NULL	NULL	KH-901	NULL	NULL	NULL	NULL	NULL
ITGA2B	hgnc:6138	ITGA2B	NCI	14-Sep-17	NULL	2.187819634820604	ENOXAPARIN	rxcui:221095	ENOXAPARIN SODIUM	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	NULL	FK-3311	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lomustine	rxcui:6466	LOMUSTINE	TRUE	FALSE	TRUE
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	0.2625383561784725	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.112919723	Celastrol	iuphar.ligand:10386	CELASTROL	FALSE	FALSE	FALSE
INTERLEUKIN-1 BETA	hgnc:5992	IL1B	TTD	2020.06.01	NULL	0.2059124362184098	Celastrol	iuphar.ligand:10386	CELASTROL	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.1981421556063943	Phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	1.500219178	BMS-196085	chembl:CHEMBL322862	CHEMBL:CHEMBL322862	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 1	hgnc:4593	GRM1	TTD	2020.06.01	NULL	3.281729452230906	A-841720	iuphar.ligand:3953	A-841720	FALSE	FALSE	FALSE
IRS2	hgnc:6126	IRS2	NCI	14-Sep-17	NULL	0.305277158	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	2.386712328895204	Ganirelix	rxcui:259264	GANIRELIX ACETATE	TRUE	FALSE	FALSE
GLYCINE TRANSPORTER GLYT-1	hgnc:11056	SLC6A9	TTD	2020.06.01	NULL	NULL	Organon-2	NULL	NULL	NULL	NULL	NULL
DOPAMINE D4 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	U-99363E	NULL	NULL	NULL	NULL	NULL
PLASMODIUM DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Primaquine	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
KCNA1	hgnc:6218	KCNA1	NCI	14-Sep-17	NULL	0.06697407	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	1.166837138570988	Tetrandrine	ncit:C28952	TETRANDRINE	FALSE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	NULL	PegCNTF	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-13	hgnc:7159	MMP13	TTD	2020.06.01	NULL	NULL	PMID17935984C1	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	NNC-0151-0000-0000	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cefluprenam	ncit:C76034	CEFLUPRENAM	FALSE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.9907107780319716	HC-Toxin	ncit:C1121	HC-TOXIN	FALSE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Methacycline	rxcui:6812	METHACYCLINE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	NULL	Sphingosomal topotecan	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR DELTA	hgnc:9235	PPARD	TTD	2020.06.01	NULL	NULL	KD-3020	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.596678082	MK-0873	drugbank:DB13029	MK-0873	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.5645986154375752	Certolizumab	ncit:C97947	CERTOLIZUMAB	FALSE	FALSE	FALSE
THYROID HORMONE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	B7-2/GM-CSF	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dextropropoxyphene	rxcui:8785	PROPOXYPHENE	TRUE	FALSE	FALSE
C-C CHEMOKINE RECEPTOR TYPE 3	hgnc:1604	CCR3	TTD	2020.06.01	NULL	NULL	YM-344031	NULL	NULL	NULL	NULL	NULL
KCNJ11	hgnc:6257	KCNJ11	NCI	14-Sep-17	NULL	0.3621218705909966	FLECAINIDE	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
LEUTINIZING-HORMONE-RELEASING HORMONE	hgnc:4419	GNRH1	TTD	2020.06.01	NULL	0.2763561643983921	Leuprolide	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	NULL	SKF-105809	NULL	NULL	NULL	NULL	NULL
HEAT SHOCK PROTEIN 70	hgnc:5232	HSPA1A	TTD	2020.06.01	NULL	NULL	H-103	NULL	NULL	NULL	NULL	NULL
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bromazepam	rxcui:1749	BROMAZEPAM	TRUE	FALSE	FALSE
FIBRIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Adhexil	NULL	NULL	NULL	NULL	NULL
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	0.6035364509849942	4-hydroxybenzaldehyde	chembl:CHEMBL14193	4-HYDROXYBENZALDEHYDE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Etravirine	rxcui:475969	ETRAVIRINE	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	NULL	BUTYLATEDHYDROXYTOLUENE	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Reformulated raltegravir	NULL	NULL	NULL	NULL	NULL
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.4861821410712453	RANTES	ncit:C1211	RECOMBINANT RANTES	FALSE	FALSE	FALSE
LONG TRANSIENT RECEPTOR POTENTIAL CHANNEL 8	hgnc:17961	TRPM8	TTD	2020.06.01	NULL	4.836232876971861	Menthol	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	2.019525817	S-777469	drugbank:DB16321	S-777469	FALSE	FALSE	FALSE
GLUTAMATE RECEPTOR AMPA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sevoflurane	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dexanabinol	ncit:C99381	DEXANABINOL	FALSE	FALSE	FALSE
N-METHYL-D-ASPARTATE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Magnesium	rxcui:6574	MAGNESIUM	TRUE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.1268301237577161	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
SERINE PROTEASE UNSPECIFIC	hgnc:11756	TFF2	TTD	2020.06.01	NULL	0.7955707762984016	Nafamostat	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
JUNB	hgnc:6205	JUNB	NCI	14-Sep-17	NULL	0.6604738520213144	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
MANNOSE-6-PHOSPHATE RECEPTOR	hgnc:6752	M6PR	TTD	2020.06.01	NULL	17.50255707856483	Alglucosidase alfa	rxcui:2475360	LYSOSOMAL ALPHA-GLUCOSIDASE	TRUE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Streptozocin	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tazobactam	rxcui:37617	TAZOBACTAM	TRUE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfamerazine	rxcui:10176	SULFAMERAZINE	TRUE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclobenzaprine	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	0.1093909817410302	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	0.375054795	AEW-541	chembl:CHEMBL551064	AEW-541	FALSE	FALSE	FALSE
CATECHOL-O-METHYL-TRANSFERASE	hgnc:2228	COMT	TTD	2020.06.01	NULL	NULL	CGP-28014	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS INTEGRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	C-2507	NULL	NULL	NULL	NULL	NULL
PROTEIN KINASE C	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAFINGOL	ncit:C1568	SAFINGOL	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	NULL	PI-88/Taxotere	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS ENVELOPE GLYCOPROTEIN GP160	NULL	NULL	TTD	2020.06.01	NULL	NULL	TBC-M4	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS GAG PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	TBC-M4	NULL	NULL	NULL	NULL	NULL
KLK3	hgnc:6364	KLK3	NCI	14-Sep-17	NULL	2.625383561784724	IMMUNOCONJUGATE	ncit:C1512	IMMUNOCONJUGATE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE XIV	NULL	NULL	TTD	2020.06.01	NULL	NULL	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
LCT	hgnc:6530	LCT	NCI	14-Sep-17	NULL	105.0153424713889	DMM	ncit:C1073	DIMETHYLMYLERAN	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE XIV	NULL	NULL	TTD	2020.06.01	NULL	NULL	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
GROWTH/DIFFERENTIATION FACTOR 8	NULL	NULL	TTD	2020.06.01	NULL	NULL	SAR391786	iuphar.ligand:8929	TREVOGRUMAB	FALSE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	BL-22	NULL	NULL	NULL	NULL	NULL
ANDROGEN RECEPTOR MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	EUGENOL	rxcui:4186	EUGENOL	TRUE	FALSE	FALSE
PLATELET-ACTIVATING FACTOR RECEPTOR	hgnc:9582	PTAFR	TTD	2020.06.01	NULL	NULL	YM-264	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	NULL	Sphingosine-1-phosphate	NULL	NULL	NULL	NULL	NULL
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	0.3454452054979901	Tonapofylline	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE VI	hgnc:1380	CA6	TTD	2020.06.01	NULL	1.875273972703375	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.1773907812016706	Tonapofylline	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	0.5250767123569451	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE XII	hgnc:1371	CA12	TTD	2020.06.01	NULL	0.7501095890813501	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.075279815	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
BACTERIAL PROTEIN SYNTHESIS	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sutezolid	ncit:C152482	SUTEZOLID	FALSE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV7	NULL	NULL	TTD	2020.06.01	NULL	NULL	CNSB-001	NULL	NULL	NULL	NULL	NULL
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	HB-AS02V	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	ABY-025	NULL	NULL	NULL	NULL	NULL
C-C CHEMOKINE RECEPTOR TYPE 9	hgnc:1610	CCR9	TTD	2020.06.01	NULL	39.38075342677087	Vercirnon	ncit:C152858	VERCIRNON	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.044573575	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.037748146	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.6945459158160648	Necitumumab	rxcui:1723738	NECITUMUMAB	TRUE	TRUE	TRUE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.1254663589861278	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
CORYNEBACTERIUM MUTATED CRM197	NULL	NULL	TTD	2020.06.01	NULL	NULL	Meningococcal groups A, C, Y and W-135 conjugate vaccine	NULL	NULL	NULL	NULL	NULL
URIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pegloticase	rxcui:1011650	PEGLOTICASE	TRUE	FALSE	FALSE
CORYNEBACTERIUM MUTATED CRM197	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pneumococcal 13-valent conjugate vaccine	ncit:C97121	PNEUMOCOCCAL 13-VALENT CONJUGATE VACCINE	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	PM-00104	chembl:CHEMBL4297453	PM-00104	FALSE	FALSE	FALSE
CARBAMOYL-PHOSPHATE SYNTHETASE I	hgnc:2323	CPS1	TTD	2020.06.01	NULL	7.501095891	Carglumic acid	rxcui:401713	CARGLUMIC ACID	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Rivoglitazone	ncit:C72841	RIVOGLITAZONE	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.2573905452730122	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
N-ACETYLMANNOSAMINE KINASE	hgnc:23657	GNE	TTD	2020.06.01	NULL	NULL	GNE Lipoplex	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 8	hgnc:15632	TLR8	TTD	2020.06.01	NULL	NULL	VTX-1463	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	NPB-001-056	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	NULL	Solulin	NULL	NULL	NULL	NULL	NULL
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.3000438356325399	GDNF	iuphar.ligand:4940	GDNF	FALSE	FALSE	FALSE
GLUTAMATE CARBOXYPEPTIDASE II	hgnc:3788	FOLH1	TTD	2020.06.01	NULL	NULL	IRX-4	NULL	NULL	NULL	NULL	NULL
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	4.702860988936115	Alectinib	rxcui:1727455	ALECTINIB	TRUE	FALSE	TRUE
P53 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cenersen	ncit:C37454	CENERSEN	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	A-366833	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN D2 RECEPTOR 2	hgnc:4502	PTGDR2	TTD	2020.06.01	NULL	1.842374429322613	AM-461	iuphar.ligand:10170	AM-461	FALSE	FALSE	FALSE
HEPATITIS C VIRUS SERINE PROTEASE NS3/4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	BOCEPREVIR	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
MAP2	hgnc:6839	MAP2	NCI	14-Sep-17	NULL	1.810609352954982	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
PROTEIN BACTERICIDAL PERMEABILITY-INCREASING	hgnc:1095	BPI	TTD	2020.06.01	NULL	NULL	XOMA-629	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	XZK-monascus	NULL	NULL	NULL	NULL	NULL
ENDOTHELIN-CONVERTING ENZYME	hgnc:3146	ECE1	TTD	2020.06.01	NULL	5.250767123569449	SLV 306	ncit:C73039	DAGLUTRIL	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN	hgnc:12099	HSP90B2P	TTD	2020.06.01	NULL	NULL	Heat shock protein vaccine	NULL	NULL	NULL	NULL	NULL
HEMOGLOBIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	FBS-0701	chembl:CHEMBL487465	DEFERITAZOLE	FALSE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	NULL	BAY 794980	NULL	NULL	NULL	NULL	NULL
AURORA KINASE C	hgnc:11391	AURKC	TTD	2020.06.01	NULL	0.060353645	ABT-348	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
FUNGAL 1,3-BETA-GLUCAN SYNTHASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-3118	rxcui:2560213	IBREXAFUNGERP	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.061340737	Danazol	rxcui:3102	DANAZOL	TRUE	FALSE	TRUE
B-CELL-ACTIVATING FACTOR	hgnc:11929	TNFSF13B	TTD	2020.06.01	NULL	19.69037671338543	Tabalumab	ncit:C91727	TABALUMAB	FALSE	FALSE	FALSE
INTEGRIN ALPHA-4/BETA-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	AJM-300	iuphar.ligand:10510	CAROTEGRAST METHYL	FALSE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	NULL	18F-LMI-1195	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	2.282942227638891	SRX-246	drugbank:DB16968	SRX-246	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.8751278539282416	EMD-1214063	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.058471794	GLPG-0492	drugbank:DB12461	GLPG-0492	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	NULL	LY3012212	NULL	NULL	NULL	NULL	NULL
GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR	hgnc:2439	CSF3R	TTD	2020.06.01	NULL	NULL	AX-200	NULL	NULL	NULL	NULL	NULL
ADRB2 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	SYL-040012	chembl:CHEMBL4298113	BAMOSIRAN	FALSE	FALSE	FALSE
SYNAPTIC VESICLE AMINE TRANSPORTER	hgnc:10935	SLC18A2	TTD	2020.06.01	NULL	NULL	AV 133	NULL	NULL	NULL	NULL	NULL
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	NULL	PF-06438179	NULL	NULL	NULL	NULL	NULL
ALPHA-KETOGLUTARATE DEHYDROGENASE	hgnc:8124	OGDH	TTD	2020.06.01	NULL	3.281729452230906	CPI-613	ncit:C80039	DEVIMISTAT	FALSE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	NULL	BAY 94-9027	NULL	NULL	NULL	NULL	NULL
SODIUM/POTASSIUM-TRANSPORTING ATPASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PBI-05204	ncit:C90586	OLEANDRIN	FALSE	FALSE	FALSE
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	Bydureon Dual Chamber Pen	NULL	NULL	NULL	NULL	NULL
BACTERIAL CELL MEMBRANE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Brilacidin	ncit:C169816	BRILACIDIN	FALSE	FALSE	FALSE
INFLUENZA POLYMERASE BASIC PROTEIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-787	ncit:C158086	PIMODIVIR	FALSE	FALSE	FALSE
BETA-HEMATIN FORMATION	NULL	NULL	TTD	2020.06.01	NULL	NULL	KAE609	ncit:C169853	CIPARGAMIN	FALSE	FALSE	FALSE
B1 BRADYKININ RECEPTOR	hgnc:1029	BDKRB1	TTD	2020.06.01	NULL	NULL	BI 113823	NULL	NULL	NULL	NULL	NULL
PROTEASE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	ONO-3307	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	NULL	JNJ-42491293	NULL	NULL	NULL	NULL	NULL
MULTIDRUG RESISTANCE PROTEIN 1	hgnc:40	ABCB1	TTD	2020.06.01	NULL	NULL	EDP-322	NULL	NULL	NULL	NULL	NULL
PROGESTERONE RECEPTOR	hgnc:8910	PGR	TTD	2020.06.01	NULL	NULL	Nestorone transdermal spray	NULL	NULL	NULL	NULL	NULL
GLUCOSE-DEPENDENT INSULINOTROPIC RECEPTOR	hgnc:19060	GPR119	TTD	2020.06.01	NULL	8.751278539282415	BMS-903452	drugbank:DB11773	BMS-903452	FALSE	FALSE	FALSE
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	REV-576	chembl:CHEMBL4297928	NOMACOPAN	FALSE	FALSE	FALSE
CASEIN KINASE II	NULL	NULL	TTD	2020.06.01	NULL	NULL	CIGB-300	ncit:C102849	CK2-TARGETING SYNTHETIC PEPTIDE CIGB-300	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	KM-023	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	0.8537832721251137	MOR-208	rxcui:2387211	TAFASITAMAB	TRUE	FALSE	FALSE
HEMOGLOBIN SUBUNIT BETA	hgnc:4827	HBB	TTD	2020.06.01	NULL	NULL	LentiGlobin	NULL	NULL	NULL	NULL	NULL
OXYSTEROLS RECEPTOR LXR	NULL	NULL	TTD	2020.06.01	NULL	NULL	XL-041	chembl:CHEMBL3545047	BMS-852927	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pennvax-B	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-17	hgnc:5981	IL17A	TTD	2020.06.01	NULL	NULL	CNTO-6785	NULL	NULL	NULL	NULL	NULL
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	NULL	BLY719	NULL	NULL	NULL	NULL	NULL
5-HT 6 RECEPTOR	hgnc:5301	HTR6	TTD	2020.06.01	NULL	7.001022831425932	PRX-07034	drugbank:DB05993	PRX-07034	FALSE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	NULL	HPP-854	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	NULL	OBI-1	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS BETA-LACTAMASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ceftolozane/tazobactam	ncit:C156396	CEFTOLOZANE-TAZOBACTAM	FALSE	FALSE	FALSE
HYALURONIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Hyqvia	wikidata:Q29005941	HYQVIA	FALSE	FALSE	FALSE
COMPLEMENT FACTOR H	hgnc:4883	CFH	TTD	2020.06.01	NULL	26.25383561784724	Trumenba	rxcui:1593128	MENINGOCOCCAL GROUP B VACCINE	TRUE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	NULL	PF-446687	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	CQA 206-291	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	BI 655066	rxcui:2166040	RISANKIZUMAB	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS GAG PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	LIPO-5	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS NEGATIVE FACTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	LIPO-5	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR 9	hgnc:15633	TLR9	TTD	2020.06.01	NULL	NULL	CYT003	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN-23	NULL	NULL	TTD	2020.06.01	NULL	NULL	MK-3222	rxcui:2053436	TILDRAKIZUMAB	TRUE	FALSE	FALSE
HEPATITIS C VIRUS NON-STRUCTURAL 5A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glecaprevir; pibrentasvir	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS SERINE PROTEASE NS3/4A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Glecaprevir; pibrentasvir	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH 1 LIGAND 1	hgnc:17635	CD274	TTD	2020.06.01	NULL	0.6471533709721451	Atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	NULL	Palonosetron and fosnetupitant	NULL	NULL	NULL	NULL	NULL
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	NULL	Palonosetron and fosnetupitant	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 3	hgnc:8534	P2RX3	TTD	2020.06.01	NULL	NULL	BAY-1902607a	NULL	NULL	NULL	NULL	NULL
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	GALAMUSTINE HYDROCHLORIDE	NULL	NULL	NULL	NULL	NULL
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.1508841127462485	Enoxacin	rxcui:3925	ENOXACIN	TRUE	FALSE	FALSE
GABA TRANSPORTER-3	hgnc:11044	SLC6A11	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dicloxacillin	rxcui:3356	DICLOXACILLIN	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flucloxacillin	rxcui:4448	FLOXACILLIN	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-2	hgnc:4076	GABRA2	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR ALPHA-3	hgnc:4077	GABRA3	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
GABA(A) RECEPTOR ALPHA-5	hgnc:4079	GABRA5	TTD	2020.06.01	NULL	NULL	GSK683699	NULL	NULL	NULL	NULL	NULL
HISTAMINE/PEPTIDE LEUKOTRIENE RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinotolast	ncit:C73052	QUINOTOLAST	FALSE	FALSE	FALSE
5-HT 2 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nexopamil	ncit:C66239	NEXOPAMIL	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	2.763561643983921	Desoxycorticosterone Pivalate	rxcui:22537	DESOXYCORTICOSTERONE PIVALATE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	NCI	14-Sep-17	NULL	0.037505479	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
CYTOCHROME P450 2A6	hgnc:2610	CYP2A6	TTD	2020.06.01	NULL	0.2651902587661338	Methoxsalen	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	0.4039051633514962	Clocortolone	rxcui:21249	CLOCORTOLONE	TRUE	FALSE	FALSE
INTERLEUKIN-4	hgnc:6014	IL4	TTD	2020.06.01	NULL	5.250767123569449	Tepoxalin	ncit:C76817	TEPOXALIN	FALSE	FALSE	FALSE
MC2R	hgnc:6930	MC2R	NCI	14-Sep-17	NULL	0.2302968036653267	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
DELTA(24)-STEROL REDUCTASE	hgnc:2859	DHCR24	TTD	2020.06.01	NULL	NULL	T-226293	NULL	NULL	NULL	NULL	NULL
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bortezomib	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
IL-1 SYNTHESIS/RELEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Flezelastine	ncit:C65692	FLEZELASTINE	FALSE	FALSE	FALSE
MARCKSL1	hgnc:7142	MARCKSL1	NCI	14-Sep-17	NULL	0.3804903712731485	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
MITOCHONDRIAL UNCOUPLING PROTEIN 1	hgnc:12517	UCP1	TTD	2020.06.01	NULL	NULL	CL-316,243	NULL	NULL	NULL	NULL	NULL
MITOCHONDRIAL UNCOUPLING PROTEIN 2	hgnc:12518	UCP2	TTD	2020.06.01	NULL	NULL	CL-316,243	NULL	NULL	NULL	NULL	NULL
MBP	hgnc:6925	MBP	NCI	14-Sep-17	NULL	0.1899011617927468	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
MITOCHONDRIAL UNCOUPLING PROTEIN 3	hgnc:12519	UCP3	TTD	2020.06.01	NULL	NULL	CL-316,243	NULL	NULL	NULL	NULL	NULL
MARCKSL1	hgnc:7142	MARCKSL1	NCI	14-Sep-17	NULL	2.187819634820604	HERBIMYCIN A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
MYCOBACTERIUM D-ALANINE-D-ALANINE LIGASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	BAM-002	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	NULL	Flobufen	NULL	NULL	NULL	NULL	NULL
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	NULL	1954U89	NULL	NULL	NULL	NULL	NULL
DOPAMINE BETA HYDROXYLASE	hgnc:2689	DBH	TTD	2020.06.01	NULL	NULL	Nepicastat oral	NULL	NULL	NULL	NULL	NULL
MCL1	hgnc:32041	ADAMTSL4-AS1	NCI	14-Sep-17	NULL	0.035382528	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	ALPIDEM	ncit:C80669	ALPIDEM	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	NULL	R-salbutamol sulphate	NULL	NULL	NULL	NULL	NULL
PHOSPHOLIPASE A2	hgnc:9030	PLA2G1B	TTD	2020.06.01	NULL	NULL	AllerB	NULL	NULL	NULL	NULL	NULL
GROWTH HORMONE RECEPTOR	hgnc:4263	GHR	TTD	2020.06.01	NULL	NULL	Syntropin	NULL	NULL	NULL	NULL	NULL
MATK	hgnc:6906	MATK	NCI	14-Sep-17	NULL	3.000438356	C-KIT LIGAND	ncit:C1410	RECOMBINANT HUMAN STEM CELL FACTOR	FALSE	FALSE	FALSE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	NULL	YM-57158	NULL	NULL	NULL	NULL	NULL
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	NULL	YM-57158	NULL	NULL	NULL	NULL	NULL
DIHYDROFOLATE REDUCTASE	hgnc:2861	DHFR	TTD	2020.06.01	NULL	NULL	L-MDAM	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.2169738480813822	Prilocaine	rxcui:8686	PRILOCAINE	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Latamoxef	rxcui:7069	MOXALACTAM	FALSE	FALSE	FALSE
MYCOBACTERIUM CDP-DIACYLGLYCEROL-INOSITOL PHOSPHATIDYLTRANSFERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Myo-inositol	rxcui:5833	INOSITOL	TRUE	FALSE	FALSE
GLYCOGEN SYNTHASE KINASE-3 BETA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Neu-120	NULL	NULL	NULL	NULL	NULL
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.079557078	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Neu-120	NULL	NULL	NULL	NULL	NULL
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	NULL	SNN-0029	NULL	NULL	NULL	NULL	NULL
CILIARY NEUROTROPHIC FACTOR	hgnc:2169	CNTF	TTD	2020.06.01	NULL	NULL	NT-501 CNTF	NULL	NULL	NULL	NULL	NULL
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	NULL	OI287GT	NULL	NULL	NULL	NULL	NULL
GLUCAGON-LIKE PEPTIDE 1 RECEPTOR	hgnc:4324	GLP1R	TTD	2020.06.01	NULL	NULL	OG987SC	NULL	NULL	NULL	NULL	NULL
MMP1	hgnc:7155	MMP1	NCI	14-Sep-17	NULL	0.4922594178346359	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.2365210416022274	Neu-P11	chembl:CHEMBL4297523	PIROMELATINE	FALSE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	AZD-3161	NULL	NULL	NULL	NULL	NULL
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	1.060761035064535	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	TMC-310911	drugbank:DB15623	TMC-310911	FALSE	FALSE	FALSE
CHOLESTEROL ABSORPTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	MD-0727	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	2.386712328895204	EMA-401	iuphar.ligand:8374	OLODANRIGAN	FALSE	FALSE	FALSE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	NULL	TAK-128	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Anti-CD19-CAR PBL	NULL	NULL	NULL	NULL	NULL
COMPLEMENT C5	NULL	NULL	TTD	2020.06.01	NULL	NULL	ARC-1905	iuphar.ligand:12857	AVACINCAPTAD PEGOL	FALSE	FALSE	FALSE
SOD1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-SOD1Rx	chembl:CHEMBL3833346	TOFERSEN	FALSE	FALSE	FALSE
MT1F	hgnc:7398	MT1F	NCI	14-Sep-17	NULL	0.3621218705909965	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
LEUKOTRIENE CYSLT1 RECEPTOR	hgnc:17451	CYSLTR1	TTD	2020.06.01	NULL	2.386712328895204	LY-2300559	drugbank:DB13016	LY-2300559	FALSE	FALSE	FALSE
T-CELL-SPECIFIC SURFACE GLYCOPROTEIN CD28	hgnc:1653	CD28	TTD	2020.06.01	NULL	NULL	CD28 and CD137 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
NEUROTROPHIC TYROSINE KINASE ROR1	hgnc:10256	ROR1	TTD	2020.06.01	NULL	NULL	ROR1R-CAR-T Cell	NULL	NULL	NULL	NULL	NULL
NEURAL CELL ADHESION MOLECULE L1	hgnc:6470	L1CAM	TTD	2020.06.01	NULL	NULL	CD171 specific CAR T cells expressing EGFRt	NULL	NULL	NULL	NULL	NULL
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.002196239	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	Anti-EGFR CAR T	NULL	NULL	NULL	NULL	NULL
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	NULL	HER-2-targeting CAR T Cells	NULL	NULL	NULL	NULL	NULL
EPHRIN TYPE-A RECEPTOR 2	hgnc:3386	EPHA2	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting EphA2	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART19 cells	NULL	NULL	NULL	NULL	NULL
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	NULL	Meso-CART	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-GD2 T-cells (1RG-CART)	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Anti-GD2 CART	NULL	NULL	NULL	NULL	NULL
NLRP3	hgnc:16400	NLRP3	NCI	14-Sep-17	NULL	1.944728564284981	ANAKINRA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	CD30 CAR T Cells	NULL	NULL	NULL	NULL	NULL
GANGLIOSIDE GD2	NULL	NULL	TTD	2020.06.01	NULL	NULL	GD2-targeted CAR-T cells	NULL	NULL	NULL	NULL	NULL
GLYPICAN-3	hgnc:4451	GPC3	TTD	2020.06.01	NULL	NULL	GAP T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19CAT-41BBZ CAR T-cells	NULL	NULL	NULL	NULL	NULL
LYMPHOCYTE ACTIVATION ANTIGEN CD30	hgnc:11923	TNFRSF8	TTD	2020.06.01	NULL	NULL	Anti-CD30-CAR-transduced T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.921012362281506	CART-19	rxcui:1986438	TISAGENLECLEUCEL	TRUE	FALSE	TRUE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Autologous CD19-targeting CAR T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	EGFRt/19-28z/4-1BBL CAR T cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	4SCAR19/22 T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	4SCAR19/22 T cells	NULL	NULL	NULL	NULL	NULL
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	NULL	CD33-CAR-T Cell	NULL	NULL	NULL	NULL	NULL
NKX6-1	hgnc:7839	NKX6-1	NCI	14-Sep-17	NULL	0.9907107780319716	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	5.250767123569449	Anti-CD123 CAR-T cells	ncit:C201493	ANTI-CD123 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CART	NULL	NULL	NULL	NULL	NULL
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	NULL	EGFR CART	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	UCART019	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	CD19 and CD22 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 and CD22 CAR-T Cells	NULL	NULL	NULL	NULL	NULL
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	NULL	Donor-derived CD19/22 bispecific CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	Donor-derived CD19/22 bispecific CAR-T cells	NULL	NULL	NULL	NULL	NULL
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	NULL	BCMA-specific CAR-expressing T Lymphocytes	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CD19 CAR T	NULL	NULL	NULL	NULL	NULL
LEUKOCYTE SURFACE ANTIGEN LEU-16	hgnc:7315	MS4A1	TTD	2020.06.01	NULL	NULL	CD20-CAR-T Cells	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	NULL	IM23	NULL	NULL	NULL	NULL	NULL
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Efavirenz	rxcui:195085	EFAVIRENZ	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2958178661165888	RESINIFERATOXIN	ncit:C1214	RESINIFERATOXIN	FALSE	FALSE	FALSE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	0.6563458904461812	Dextromethorphan Polistirex	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	0.7001022831425934	Ethoxzolamide	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
BACTERIAL 30S RIBOSOMAL RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Gentamicin	rxcui:1596450	GENTAMICIN	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lamivudine	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
ANTITHROMBIN-III	hgnc:775	SERPINC1	TTD	2020.06.01	NULL	1.458546423213736	Heparin Calcium	rxcui:20044	HEPARIN CALCIUM	TRUE	FALSE	FALSE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	0.9546849315580819	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
SYNAPTIC VESICLE GLYCOPROTEIN 2A	hgnc:20566	SV2A	TTD	2020.06.01	NULL	4.500657534	Levetiracetam	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
INSULIN	hgnc:6081	INS	TTD	2020.06.01	NULL	8.751278539282415	Inulin	rxcui:5924	INULIN	TRUE	FALSE	FALSE
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	0.130291988	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.2917092846427472	Isradipine	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.2273059360852576	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Moxifloxacin	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Moxifloxacin	rxcui:139462	MOXIFLOXACIN	TRUE	FALSE	FALSE
CRYPTOSPORIDIUM PYRUVATE:FERREDOXIN OXIDOREDUCTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Nitazoxanide	rxcui:31819	NITAZOXANIDE	TRUE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.1630673019742065	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
SCHISTOSOMA DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxamniquine	rxcui:7778	OXAMNIQUINE	TRUE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.1238388472539964	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Piroxicam	rxcui:68115	PIROXICAM-BETA-CYCLODEXTRIN	TRUE	FALSE	FALSE
OXO-5-ALPHA-STEROID 4-DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Polyestradiol Phosphate	rxcui:34120	POLYESTRADIOL PHOSPHATE	TRUE	FALSE	FALSE
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pramipexole	rxcui:746741	PRAMIPEXOLE	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.182318303	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Ropinirole	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
SAMARIUM	NULL	NULL	TTD	2020.06.01	NULL	NULL	Samarium Sm-153 Lexidronam Pentasodium	rxcui:317675	SAMARIUM SM-153 LEXIDRONAM PENTASODIUM	FALSE	FALSE	FALSE
BACTERIAL DIHYDROPTEROATE SYNTHETASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfanilamide	rxcui:10184	SULFANILAMIDE	TRUE	FALSE	FALSE
PAX5	hgnc:8619	PAX5	NCI	14-Sep-17	NULL	4.200613699	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
HUMAN DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Temozolomide	rxcui:37776	TEMOZOLOMIDE	TRUE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.1988926940746003	Sibutramine	rxcui:36514	SIBUTRAMINE	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.172950169	Ropinirole	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
E3 UBIQUITIN-PROTEIN LIGASE COP1	hgnc:17440	COP1	TTD	2020.06.01	NULL	0.9546849315580819	Propafenone	rxcui:8754	PROPAFENONE	TRUE	FALSE	FALSE
GLYCOPROTEIN IIB/IIIA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tirofiban	rxcui:73137	TIROFIBAN	TRUE	FALSE	FALSE
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Trovafloxacin	rxcui:115552	TROVAFLOXACIN	FALSE	FALSE	FALSE
PEBP1	hgnc:8630	PEBP1	NCI	14-Sep-17	NULL	2.625383561784725	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
MYCOBACTERIUM FUSION PROTEIN RV2608-RV3619-RV3620-RV1813	NULL	NULL	TTD	2020.06.01	NULL	NULL	ID-93/GLA-SE	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	NULL	CP-331684	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	CS-00028	NULL	NULL	NULL	NULL	NULL
INTERLEUKIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PF-04236921	chembl:CHEMBL2109613	PF-04236921	FALSE	FALSE	FALSE
HORMONE UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	NV-04	NULL	NULL	NULL	NULL	NULL
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	NULL	P-552-02	NULL	NULL	NULL	NULL	NULL
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1346350544504987	FDG	rxcui:1362737	FLUORODEOXYGLUCOSE F18	TRUE	FALSE	FALSE
HEPATITIS B VIRUS MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-HBV	NULL	NULL	NULL	NULL	NULL
PLASMA KALLIKREIN MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS-PKK	NULL	NULL	NULL	NULL	NULL
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	2.187819634820604	CORTISONE	rxcui:2878	CORTISONE	TRUE	FALSE	FALSE
HEPATITIS C VIRUS MICRORNA MIR-122	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG-101	chembl:CHEMBL3990019	TEMAVIRSEN SODIUM	FALSE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Penicillin G Procaine	rxcui:7983	PENICILLIN G PROCAINE	TRUE	FALSE	FALSE
CANDIDA CYTOCHROME P450 51	NULL	NULL	TTD	2020.06.01	NULL	NULL	Luliconazole 10%	NULL	NULL	NULL	NULL	NULL
BACTERIAL DEOXYRIBONUCLEIC ACID	NULL	NULL	TTD	2020.06.01	NULL	NULL	Metronidazole	rxcui:6922	METRONIDAZOLE	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS PROTEASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	KNI-272	ncit:C29140	KNI-272	FALSE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.017243899	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.546954909	ARQ 092	ncit:C99172	MIRANSERTIB	FALSE	FALSE	TRUE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	1.193356164447602	Luvox	rxcui:203143	FLUVOXAMINE MALEATE	TRUE	FALSE	FALSE
PVT1	hgnc:9709	PVT1	NCI	14-Sep-17	NULL	0.7001022831425933	GLIVEC	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
MICRORNA HSA-MIR-34	NULL	NULL	TTD	2020.06.01	NULL	NULL	MRX34	ncit:C105802	LIPOSOME-ENCAPSULATED MIR-34 MIMIC MRX34	FALSE	FALSE	FALSE
PI3-KINASE ALPHA	hgnc:8975	PIK3CA	TTD	2020.06.01	NULL	NULL	PWT-33597	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS RNA-DIRECTED RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RG-7348	NULL	NULL	NULL	NULL	NULL
THYMIDINE KINASE 1	hgnc:11830	TK1	TTD	2020.06.01	NULL	NULL	Thymidine kinase-expressing adenovirus and ganciclovir suicide gene therapy	NULL	NULL	NULL	NULL	NULL
MELANOCORTIN RECEPTOR 1	hgnc:6929	MC1R	TTD	2020.06.01	NULL	NULL	AP-1030	NULL	NULL	NULL	NULL	NULL
RBP3	hgnc:9921	RBP3	NCI	14-Sep-17	NULL	8.751278539282415	RETINYL PALMITATE	rxcui:35406	VITAMIN A PALMITATE	TRUE	FALSE	FALSE
MELANOCORTIN RECEPTOR 4	hgnc:6932	MC4R	TTD	2020.06.01	NULL	NULL	AP-1030	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Avrina	NULL	NULL	NULL	NULL	NULL
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-4/BETA-2	NULL	NULL	TTD	2020.06.01	NULL	NULL	AZD-1446	chembl:CHEMBL2179529	AZD1446	FALSE	FALSE	FALSE
MYCOBACTERIUM RNA POLYMERASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	T-705	ncit:C81605	FAVIPIRAVIR	FALSE	FALSE	FALSE
TGF-BETA RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	GC-1008	chembl:CHEMBL1743022	FRESOLIMUMAB	FALSE	FALSE	TRUE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	AVE0118	NULL	NULL	NULL	NULL	NULL
T-CELL SURFACE GLYCOPROTEIN CD3	NULL	NULL	TTD	2020.06.01	NULL	NULL	Otelixizumab	ncit:C95790	OTELIXIZUMAB	FALSE	FALSE	FALSE
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	5-azolone derivative 1	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 11	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Carboxamide derivative 7	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	Epoxysuccinate derivative 4	NULL	NULL	NULL	NULL	NULL
CALPAIN-2	hgnc:1479	CAPN2	TTD	2020.06.01	NULL	NULL	PMID25399719-Compound-17	NULL	NULL	NULL	NULL	NULL
CATHEPSIN K	hgnc:2536	CTSK	TTD	2020.06.01	NULL	NULL	PMID25399719-Compound-17	NULL	NULL	NULL	NULL	NULL
CATHEPSIN L	hgnc:2537	CTSL	TTD	2020.06.01	NULL	NULL	PMID25399719-Compound-17	NULL	NULL	NULL	NULL	NULL
CATHEPSIN S	hgnc:2545	CTSS	TTD	2020.06.01	NULL	NULL	PMID25399719-Compound-17	NULL	NULL	NULL	NULL	NULL
CALPAIN-1	hgnc:1476	CAPN1	TTD	2020.06.01	NULL	NULL	Undecylenic acid derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenelzine	rxcui:8123	PHENELZINE	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	4-hydroxybenzaldehyde	chembl:CHEMBL14193	4-HYDROXYBENZALDEHYDE	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	4-Methoxybenzaldehyde	chembl:CHEMBL161598	ANISALDEHYDE	FALSE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	EUGENOL	rxcui:4186	EUGENOL	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	FERULIC ACID	rxcui:1368647	FERULIC ACID	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure1-Chukrasone B	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure1-Eryngiolide A	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure1-Sarcaboside A	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure2-Spirooliganone B	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure3-Fluevirosine A	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Figure3-Lycojaponicumin C	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-13	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table 6-13	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C10	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C18	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C22	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C23	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C6	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25399762-Compound-Table1-C8	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	T83193	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	3-phenyl acrylic acid derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	A-substituted phenylpropionic acid derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	MRL24	iuphar.ligand:6743	MRL24	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	NULL	Phenylpyridine derivative 3	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenylpyridine derivative 3	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-A	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-A	NULL	NULL	NULL	NULL	NULL
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-E	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25416646-Compound-Figure5-E	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Spirolaxine derivative 1	NULL	NULL	NULL	NULL	NULL
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 18	NULL	NULL	NULL	NULL	NULL
MAPK/ERK KINASE KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	RO-5126766	drugbank:DB15254	AVUTOMETINIB	FALSE	FALSE	FALSE
NAD-DEPENDENT DEACETYLASE SIRTUIN-1	hgnc:14929	SIRT1	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2012106509Salermide	NULL	NULL	NULL	NULL	NULL
NAD-DEPENDENT DEACETYLASE SIRTUIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25435179-Compound-WO2013059587(V, 1st set)	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-16	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-18	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-2	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-23	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-26	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-27	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-31	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-33	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-35	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-36	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-37	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-38	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-42	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-44	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-46	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-48	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-49	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-50	NULL	NULL	NULL	NULL	NULL
MELANIN-CONCENTRATING HORMONE RECEPTOR 1	hgnc:4479	MCHR1	TTD	2020.06.01	NULL	NULL	PMID25522065-Compound-8	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.3	hgnc:10590	SCN3A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Aryl carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 11	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 12	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Cyclopropyl-spiro piperidine derivative 2	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.3	hgnc:10590	SCN3A	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 5	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyridinone derivative 5	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	NULL	Tarizine derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 2	NULL	NULL	NULL	NULL	NULL
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydrothieno [2,3-e]indazole derivative 1	NULL	NULL	NULL	NULL	NULL
INHIBITOR OF NUCLEAR FACTOR KAPPA-B KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Dihydrothieno [2,3-e]indazole derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-quinolin-benzene sulphonamide derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	N-quinolin-benzene sulphonamide derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2011799419010	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2012820715110	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US2012830453910	NULL	NULL	NULL	NULL	NULL
POLYUBIQUITIN-C	hgnc:12468	UBC	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-US20130237529 36	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2013082253 31	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25553724-Compound-WO2013082253 33	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoxaline derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoxaline derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR NF-KAPPA-B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinoxaline derivative 5	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	PMID25623274-Compound-WO2014132220C1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Indol-5-ol derivative 1	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-15a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-18	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-19a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-19a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-20b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-21b	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR BETA	hgnc:8804	PDGFRB	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-21b	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-21b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-26c	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-28a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-31c	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-34a	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-34b	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-36c	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-37a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-37a	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	PMID25656651-Compound-38	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	NULL	Pyridoindole derivative 3	NULL	NULL	NULL	NULL	NULL
FUSION PROTEIN BCR-ABL T315I MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-b]pyridine derivative 4	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-101	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-11	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-111	NULL	NULL	NULL	NULL	NULL
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	NULL	PMID25666693-Compound-112	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indazole derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Indolinone derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-EP20041486488	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20120277229 41(1.3)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20130053382 36(3-5)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-US20130053382 37(4-6)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2008005457	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25684022-Compound-WO2012135799 43(1.5)	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 61	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 2	NULL	NULL	NULL	NULL	NULL
PYRUVATE DEHYDROGENASE KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiazole carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-14	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-16	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-19	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-21	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-28	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-36	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-39	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-46	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-57	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-58	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	PMID25726713-Compound-61	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 19	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 20	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750M1	NULL	NULL	NULL	NULL	NULL
PROSTAGLANDIN E2 RECEPTOR EP2	hgnc:9594	PTGER2	TTD	2020.06.01	NULL	NULL	PMID25772215-Compound-US02014179750TG7-76	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	PMID25776143-Compound-2	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	PMID25776143-Compound-4	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	PMID25776143-Compound-7	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	NULL	PMID25776143-Compound-8	NULL	NULL	NULL	NULL	NULL
JNK-INTERACTING PROTEIN PEPTIDE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-N3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE JNK1	hgnc:6881	MAPK8	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-N3	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-O2	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P2	NULL	NULL	NULL	NULL	NULL
MITOGEN-ACTIVATED PROTEIN KINASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID25991433-Compound-P3	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-U2014S0288042C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140142115C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140275020D	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-US20140275020E	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2012058134A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2012058134C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013039802B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013062892D	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013062900A	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013062900B	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2013062900C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014085210C	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014099633E	NULL	NULL	NULL	NULL	NULL
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.1	hgnc:6255	KCNJ1	TTD	2020.06.01	NULL	NULL	PMID26004420-Compound-WO2014126944A	NULL	NULL	NULL	NULL	NULL
ZINC FINGER-CONTAINING UBIQUITIN PEPTIDASE 1	hgnc:21224	ZUP1	TTD	2020.06.01	NULL	NULL	Azepan-4-one derivative 2	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	4-pyridone derivative 2	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Hypersulfated disaccharide compound 1	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 56	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 56	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 59	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 59	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 65	NULL	NULL	NULL	NULL	NULL
CATHEPSIN G	hgnc:2532	CTSG	TTD	2020.06.01	NULL	NULL	Peptide analog 70	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Peptide analog 70	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Tetra-hydro-pyrrolopyrimidinedione derivative 1	NULL	NULL	NULL	NULL	NULL
NEUTROPHIL ELASTASE	hgnc:3309	ELANE	TTD	2020.06.01	NULL	NULL	Uracil derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 9	hgnc:1780	CDK9	TTD	2020.06.01	NULL	NULL	Benzothiazine derivative 1	NULL	NULL	NULL	NULL	NULL
SERINE/THREONINE-PROTEIN KINASE PIM-1	hgnc:8986	PIM1	TTD	2020.06.01	NULL	NULL	Benzothiazine derivative 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	Fluorinated compound 1	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	NULL	Imidazo pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 8	hgnc:1779	CDK8	TTD	2020.06.01	NULL	NULL	Macrocycle derivative 14	NULL	NULL	NULL	NULL	NULL
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	NULL	N-(pyridin-2-yl)pyridine methylsulfone derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY-ACID AMIDE HYDROLASE 1	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 6	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 8	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Heteroaryl-substituted urea derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Imidazolyl urea derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Isoxazoline derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Isoxazoline derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	N-alkyl-4-oxazolecar boxamide derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	N-alkyl-4-oxazolecar boxamide derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Spirocyclic diamine urea derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Tetra-hydro-naphthalene derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Tetra-hydro-naphthalene derivative 2	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Tetra-substituted urea derivative 1	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Tetra-substituted urea derivative 2	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	PMID26560362-Compound-90	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	Triazole derivative 3	NULL	NULL	NULL	NULL	NULL
ARACHIDONATE 15-LIPOXYGENASE	hgnc:433	ALOX15	TTD	2020.06.01	NULL	NULL	Tri-substituted benzene derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	2-alkyloxy-3-phenylethynyl-4a,5-dihydropyrido[2,3-b]pyrazine derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	3-acylidene-2-oxoindole derivative 2	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Dihydroisoxazole derivative 1	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	Dipeptide analog 4	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XIIIA	hgnc:3531	F13A1	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-13	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-13	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-15	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-18	NULL	NULL	NULL	NULL	NULL
TISSUE TRANSGLUTAMINASE	hgnc:11778	TGM2	TTD	2020.06.01	NULL	NULL	PMID26560530-Compound-3	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 21	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 21	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 22	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 22	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 23	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 23	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 24	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 24	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 27	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 27	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 29	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 29	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 1	hgnc:4848	HCRTR1	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 9	NULL	NULL	NULL	NULL	NULL
OREXIN RECEPTOR TYPE 2	hgnc:4849	HCRTR2	TTD	2020.06.01	NULL	NULL	1,2-diamino cyclopentane-based derivative 9	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	3-phenyl pyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Benzazepine derivative 2	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Diarylamine and arylheteroarylamine pyrazole derivative 2	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 14	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 2	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 4	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 7	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Heteroaryl-azepine derivative 9	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	PMID26609882-Compound-35	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 67	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 72	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrazole-3-carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 26	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 26	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 26	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 28	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 28	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 28	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 29	NULL	NULL	NULL	NULL	NULL
5-HT 2B RECEPTOR	hgnc:5294	HTR2B	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 29	NULL	NULL	NULL	NULL	NULL
5-HT 2C RECEPTOR	hgnc:5295	HTR2C	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 29	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 10	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 3	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Alkyl mannoside derivative 6	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	C-linked disaccharide biphenyl mannoside derivative 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 4	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Mannoside derivative 6	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-10a	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-10b	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-10c	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-118	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-120	NULL	NULL	NULL	NULL	NULL
BACTERIAL FIMBRIN D-MANNOSE ADHESIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26651364-Compound-125	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 6	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 6	NULL	NULL	NULL	NULL	NULL
SMOOTHENED HOMOLOG	hgnc:11119	SMO	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 7	NULL	NULL	NULL	NULL	NULL
ZINC FINGER PROTEIN GLI1	hgnc:4317	GLI1	TTD	2020.06.01	NULL	NULL	Isoflavone derivative 7	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure12bottomright	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure12left	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9bottomright	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9left01	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle01	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9middle02	NULL	NULL	NULL	NULL	NULL
GLYCOGEN PHOSPHORYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID26666989-Compound-Figure9toprightR02	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Diamine derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Monoamine derivative 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Monoamine derivative 4	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	P-coumaric acid derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	P-coumaric acid derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	P-coumaric acid derivative 5	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-114	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-118	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-31	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-48	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-64	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	PMID26815044-Compound-I	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Polyhydroxy benzamide derivative 3	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 12	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 13	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 2	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 21	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 25	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 32	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Resorcinol compound 33	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Thiazole derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	NULL	Thiazoline derivative 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Alkaloid derivative 4	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Aromatic and heteroaryl compound 1	NULL	NULL	NULL	NULL	NULL
HYPOXIA-INDUCIBLE FACTOR 1	hgnc:18420	SETD2	TTD	2020.06.01	NULL	NULL	Aryl carbamate analog 1	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 14	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 19	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 2	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 3	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	NULL	Isoxazole-based bicyclic compound 6	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN TESTIS-SPECIFIC PROTEIN	hgnc:1105	BRDT	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-103	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-103	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 3	hgnc:1104	BRD3	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-103	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-103	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN TESTIS-SPECIFIC PROTEIN	hgnc:1105	BRDT	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-104	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-104	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 3	hgnc:1104	BRD3	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-104	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-104	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN TESTIS-SPECIFIC PROTEIN	hgnc:1105	BRDT	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-105	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-105	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 3	hgnc:1104	BRD3	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-105	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-105	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 2	hgnc:1103	BRD2	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-106	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-21	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-25	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-30	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR SIGNAL-REGULATED KINASE 5	hgnc:6880	MAPK7	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-30	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-32	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR SIGNAL-REGULATED KINASE 5	hgnc:6880	MAPK7	TTD	2020.06.01	NULL	NULL	PMID26924192-Compound-32	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Imidazopyridazine derivative 7	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Peptidomimetic analog 6	NULL	NULL	NULL	NULL	NULL
PROTEINASE ACTIVATED RECEPTOR 2	hgnc:30225	SLC52A1	TTD	2020.06.01	NULL	NULL	Quinazoline derivative 10	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Benzenamine derivative 4	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclic peptide derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Cyclic peptide derivative 1	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclic peptide derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 1	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 10	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 10	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 6	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Cyclopropylamine derivative 7	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Pyrimidine derivative 16	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1	hgnc:2959	DNASE1L3	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 3	NULL	NULL	NULL	NULL	NULL
LYSINE-SPECIFIC HISTONE DEMETHYLASE 1B	hgnc:21577	KDM1B	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE A	hgnc:6833	MAOA	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 3	NULL	NULL	NULL	NULL	NULL
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tarnylcypromine derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-11	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-2	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 4	hgnc:3559	FABP4	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-21	NULL	NULL	NULL	NULL	NULL
FATTY ACID-BINDING PROTEIN 5	hgnc:3560	FABP5	TTD	2020.06.01	NULL	NULL	PMID27109571-Compound-21	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 7	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 2	hgnc:27269	IDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 7	NULL	NULL	NULL	NULL	NULL
TRYPTOPHAN 2,3-DIOXYGENASE	hgnc:11708	TDO2	TTD	2020.06.01	NULL	NULL	2,3-diamino-benzo[b]thiophene derivative 7	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 5	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 7	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Aryl pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 4	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 5	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Benzene sulfonamide derivative 7	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 2	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 4	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 5	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 6	NULL	NULL	NULL	NULL	NULL
KYNURENINE 3-HYDROXYLASE	hgnc:6381	KMO	TTD	2020.06.01	NULL	NULL	Cyclopropane 1-carboxylic acid derivative 8	NULL	NULL	NULL	NULL	NULL
CANNABINOID RECEPTOR 2	hgnc:2160	CNR2	TTD	2020.06.01	NULL	NULL	PMID27215781-Compound-29	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Amidopyrazole derivative 2	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Amidopyrazole derivative 5	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Diaminopyridine analog 4	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Diaminopyridine analog 5	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Fused benzoheterocycle amide derivative 1	NULL	NULL	NULL	NULL	NULL
IL-1 RECEPTOR-ASSOCIATED KINASE 1	hgnc:6112	IRAK1	TTD	2020.06.01	NULL	NULL	Indazoletriazolephenyl derivative 2	NULL	NULL	NULL	NULL	NULL
RENAL CARCINOMA ANTIGEN NY-REN-64	hgnc:17967	IRAK4	TTD	2020.06.01	NULL	NULL	Indazoletriazolephenyl derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [4,3-a]quinoxaline derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	1,2,4-triazole [4,3-a]quinoxaline derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	PMID27321640-Compound-74	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrazolo[3,4-d]pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrido[2,3-d]pyrimidine-2,4-diamine derivative 1	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 2	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 3	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 4	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 5	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 10A	NULL	NULL	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 6	NULL	NULL	NULL	NULL	NULL
PHOSPHODIESTERASE 2A	hgnc:8777	PDE2A	TTD	2020.06.01	NULL	NULL	Triazolo-pyridine derivative 6	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR BETA	hgnc:9865	RARB	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-10	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR ALPHA	hgnc:9864	RARA	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-4	NULL	NULL	NULL	NULL	NULL
RETINOIC ACID RECEPTOR BETA	hgnc:9865	RARB	TTD	2020.06.01	NULL	NULL	PMID27336223-Compound-8	NULL	NULL	NULL	NULL	NULL
RIBOSOMAL PROTEIN S6 KINASE ALPHA-3	hgnc:10431	RPS6KA2	TTD	2020.06.01	NULL	NULL	Pyrrolo[2,3-d]pyrimidine derivative 35	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	2-ethyl-3-(4-hydroxy) benzoyl benzofuran derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	PMID27414413-Compound-Figure8right	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Succinamide derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Tihoacetate derivative 1	NULL	NULL	NULL	NULL	NULL
URATE ANION EXCHANGER 1	hgnc:17989	SLC22A12	TTD	2020.06.01	NULL	NULL	Triazole propanedioic acid derivative 1	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-102	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-91	NULL	NULL	NULL	NULL	NULL
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	NULL	PMID27454349-Compound-92	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Atorvastatin lactole derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Hexahydro naphthalene derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Hexahydro naphthalene derivative 2	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Hexahydro naphthalene derivative 3	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Pitavastatin derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	PMID27537201-Compound-Figure11	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	PMID27537201-Compound-Figure15b	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Poly-substituted azoles statin lactone derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Poly-substituted azoles statin lactone derivative 2	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Pravastatin derivative 1	NULL	NULL	NULL	NULL	NULL
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	NULL	Quinoline derivative 16	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	2-piperidine thiazole derivative 2	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-12	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-16	NULL	NULL	NULL	NULL	NULL
SPHINGOSINE KINASE	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	NULL	PMID27539678-Compound-8	NULL	NULL	NULL	NULL	NULL
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	NULL	PMID27551786-Compound-II	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27599163-Compound-75	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine acetamide analog 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine acetamide analog 3	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine acetamide analog 6	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Imidazopyridine derivative 2	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivative 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-58	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-63	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	PMID27607364-Compound-64	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine acetamide analog 1	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 6	NULL	NULL	NULL	NULL	NULL
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	NULL	Quinoline carboxamide derivative 9	NULL	NULL	NULL	NULL	NULL
PRKR-LIKE ENDOPLASMIC RETICULUM KINASE	hgnc:3255	EIF2AK3	TTD	2020.06.01	NULL	NULL	Indoline derivative 2	NULL	NULL	NULL	NULL	NULL
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	NULL	Pyridine derivative 22	NULL	NULL	NULL	NULL	NULL
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	NULL	Pyridine derivative 22	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyridine derivative 22	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	NULL	Pyridine derivative 22	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 4	NULL	NULL	NULL	NULL	NULL
PLATELET-ACTIVATING FACTOR ACETYLHYDROLASE	hgnc:9040	PLA2G7	TTD	2020.06.01	NULL	NULL	Bicyclic pyrimidine derivative 2	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Chlorobenzamide derivative 2	NULL	NULL	NULL	NULL	NULL
P2X PURINOCEPTOR 7	hgnc:8537	P2RX7	TTD	2020.06.01	NULL	NULL	Fluorophenyl-substituted heterocyclic amide analog 1	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-20	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-23	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-26	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-26	NULL	NULL	NULL	NULL	NULL
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-27	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-27	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-28	NULL	NULL	NULL	NULL	NULL
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	NULL	PMID27744724-Compound-29	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloalkyl nitrile pyrazolo pyridone derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cycloalkyl nitrile pyrazolo pyridone derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoxazole derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isoxazole derivative 2	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Isoxazole derivative 2	NULL	NULL	NULL	NULL	NULL
ACTIVIN RECEPTOR-LIKE KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Compound12	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Compound12	NULL	NULL	NULL	NULL	NULL
ACTIVIN RECEPTOR-LIKE KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Compound4	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10Compound4	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure10CompoundA	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure11Example5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure11Example5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure11Example5	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure11Example5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure1Example20	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure1Example20	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure1Example20	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure8Example5	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	PMID27774822-Compound-Figure8Example5	NULL	NULL	NULL	NULL	NULL
JAK-STAT SIGNALING PATHWAY	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminotriazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminotriazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aminotriazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Aminotriazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Aminotriazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	NULL	Aminotriazolopyridine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 7	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Benzimidazole derivative 7	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bipyrazole derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
JANUS KINASE 3	hgnc:6193	JAK3	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	NULL	Bis-aminopyrimidine derivative 3	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	4,5,6,7-tetrahydrofuro[3,4-c]pyridine-1(3H)-one derivative 4	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Imidazo pyridine derivative 5	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Indanone and indandione derivative 1	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	Oxazolo[3,4-a]pyrazine derivative 7	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-5c	NULL	NULL	NULL	NULL	NULL
NEUROPEPTIDE S RECEPTOR	hgnc:23631	NPSR1	TTD	2020.06.01	NULL	NULL	PMID27788040-Compound-6b	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-16	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-17	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-18	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-21	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID27828716-Compound-BIO-acetoxime	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Quinolinyl pyrazinyl urea derivative 2	NULL	NULL	NULL	NULL	NULL
GLYCOGEN SYNTHASE KINASE-3 ALPHA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Thiadiazolidindione derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 3	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	4-Carboxamido-isoindolinone derivative 5	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	7-azaindole derivative 9	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Dihydropyrido phthalazinone derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Phthalazine derivative 1	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE 1	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	Phthalazine ketone derivative 2	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-24	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-XI	NULL	NULL	NULL	NULL	NULL
POLY [ADP-RIBOSE] POLYMERASE	hgnc:270	PARP1	TTD	2020.06.01	NULL	NULL	PMID27841036-Compound-XVII	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azaindole derivative 3	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azaindole derivative 4	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Azole benzene derivative 1	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 1	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 5	NULL	NULL	NULL	NULL	NULL
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	NULL	Fused heterocyclic compound 8	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine-indole hybrid derivative 1	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine-indole hybrid derivative 2	NULL	NULL	NULL	NULL	NULL
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	NULL	Tacrine-phenothiazine hybrid derivative 1	NULL	NULL	NULL	NULL	NULL
THIOREDOXIN REDUCTASE	hgnc:9355	PRDX5	TTD	2020.06.01	NULL	NULL	Diterpene triepoxide derivative 1	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	Palmarumycin derivative 3	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-27	NULL	NULL	NULL	NULL	NULL
CYTOPLASMIC THIOREDOXIN REDUCTASE	hgnc:12437	TXNRD1	TTD	2020.06.01	NULL	NULL	PMID27977313-Compound-39	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Bicyclic heteroaryl carboxamide analog 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Central azetidine derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Ethynyl compound 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Ethynyl compound 4	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Imidazopyridine and triazolopyridine compound 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	N-alkylamide derivative 2	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	PMID28067079-Compound-97	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	PMID28067079-Compound-98	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyrazolopyrimidine derivative 1	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyridine derivative 13	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Pyridine derivative 14	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-oxazolopyridine derivative 3	NULL	NULL	NULL	NULL	NULL
METABOTROPIC GLUTAMATE RECEPTOR 5	hgnc:4597	GRM5	TTD	2020.06.01	NULL	NULL	Tetra-hydro-pyrazolopyrazine derivative 4	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Carbamide derivative 6	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 6	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Mycophenolic acid/nucleotide derivative 8	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-US20120264760C81	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	PMID28074661-Compound-WO2009018344C78	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Quinazolinone derivative 1	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Quinazolinone derivative 2	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Quinolone derivative 1	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 10	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 14	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 3	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 6	NULL	NULL	NULL	NULL	NULL
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE 1	hgnc:6052	IMPDH1	TTD	2020.06.01	NULL	NULL	Urea and carbamate bioisostere derivative 7	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32i	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32i	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32k	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32k	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32l	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32l	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32o	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32o	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32s	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32s	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32u	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-32u	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID28092474-Compound-33	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Hydrazide derivative 4	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Oxindole derivative 2	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Oxindole derivative 4	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2 G2019S MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Oxindole derivative 4	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	PMID28117607-Compound-4	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	PMID28117607-Compound-7	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyridopyrimidinone derivative 1	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyridopyrimidinone derivative 3	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 10	NULL	NULL	NULL	NULL	NULL
LEUCINE-RICH REPEAT KINASE 2	hgnc:18618	LRRK2	TTD	2020.06.01	NULL	NULL	Pyrrolo-pyrimidine derivative 8	NULL	NULL	NULL	NULL	NULL
SMN1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	nusinersen	rxcui:1863556	NUSINERSEN	TRUE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	NULL	Imidazo[1,2-b]pyridazine derivative 5	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-46	NULL	NULL	NULL	NULL	NULL
EZH2 Y641N MUTANT	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-46	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-47	NULL	NULL	NULL	NULL	NULL
ENHANCER OF ZESTE HOMOLOG 2	hgnc:3527	EZH2	TTD	2020.06.01	NULL	NULL	PMID28394193-Compound-52	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaromatic ring derivative 2	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Heteroaromatic ring derivative 3	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-21	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-26	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28447479-Compound-4	NULL	NULL	NULL	NULL	NULL
EXTRACELLULAR LYSOPHOSPHOLIPASE D	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tetra-hydro-carboline derivative 2	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DUAL DLG AND ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	1,2,3,4-tetrahydroisoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	1,2,3,4-tetrahydroisoquinoline derivative 1	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DLG] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	1-phenyl-1,3,4-triazole derivative 3	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	1-phenyl-1,3,4-triazole derivative 3	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	2-hydroxybenzamide derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	2-hydroxybenzamide derivative 1	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	2-hydroxybenzamide derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	2-hydroxybenzamide derivative 2	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	3-phenyl propanoic derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	3-phenyl propanoic derivative 1	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	3-phenyl propanoic derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	3-phenyl propanoic derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	4-(2-cyclohexylethoxy) aniline derivative 3	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chalcone derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Chalcone derivative 1	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Chalcone derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Chalcone derivative 2	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Diterpenoid derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Diterpenoid derivative 1	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Diterpenoid derivative 2	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Diterpenoid derivative 2	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-10	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-10	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-11	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-11	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-34	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-34	NULL	NULL	NULL	NULL	NULL
KEAP1-NRF2[DUAL DLG AND ETGE] PPI	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-60	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-60	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-92	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-95	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	PMID28454500-Compound-96	NULL	NULL	NULL	NULL	NULL
CYSTEINES OF KEAP1	NULL	NULL	TTD	2020.06.01	NULL	NULL	Trepenoid derivative 1	NULL	NULL	NULL	NULL	NULL
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	NULL	Trepenoid derivative 1	NULL	NULL	NULL	NULL	NULL
GAMMA-SECRETASE SUBUNIT APH-1A/1B	hgnc:29509	APH1A	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 15	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme23MPPDerivatives	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme25-2	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme25-2	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme2WO2012/098065bottom	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme2WO2012/098065bottom	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme4Upper	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme4Upper	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme5	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme5	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme8NCGC-00189310	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1A	hgnc:3091	DYRK1A	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT3356	NULL	NULL	NULL	NULL	NULL
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 1B	hgnc:3092	DYRK1B	TTD	2020.06.01	NULL	NULL	PMID28766366-Compound-Scheme9EHT3356	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-36	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-42	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-49	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-51	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-54	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-61	NULL	NULL	NULL	NULL	NULL
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	NULL	PMID28870136-Compound-65	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	Indomethacin analog 2	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	Indomethacin analog 3	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	N-(benzimidazolylcarbonyl)-piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
DIHYDRODIOL DEHYDROGENASE TYPE I	hgnc:386	AKR1C3	TTD	2020.06.01	NULL	NULL	N-(pyridinepyrroylylcarbonyl)-piperidine derivative 1	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidine-benzoxazin-3(4H)-one derivative 2	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidine-benzoxazin-3(4H)-one derivative 3	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidinyl-piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidinyl-piperidine derivative 2	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Azetidinyl-piperidine derivative 3	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 10	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 10	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 11	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Carbamate derivative 16	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Carbamate derivative 16	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 5	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Piperazine carbamic compound 5	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-11c	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-11c	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-7b	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	PMID29053063-Compound-7e	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 82	NULL	NULL	NULL	NULL	NULL
MONOACYLGLYCEROL LIPASE ABHD6	hgnc:21398	ABHD6	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 82	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 82	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 83	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 83	NULL	NULL	NULL	NULL	NULL
FATTY ACID AMIDE HYDROLASE	hgnc:3553	FAAH	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 84	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 84	NULL	NULL	NULL	NULL	NULL
MONOGLYCERIDE LIPASE	hgnc:17038	MGLL	TTD	2020.06.01	NULL	NULL	Pyrazole derivative 85	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-1	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure10(2a)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure10(2a)	NULL	NULL	NULL	NULL	NULL
MATRIX METALLOPROTEINASE-3	hgnc:7173	MMP3	TTD	2020.06.01	NULL	NULL	PMID29130358-Compound-Figure10(2a)	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-22	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-34	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-43	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-48	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-59	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-60	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-71	NULL	NULL	NULL	NULL	NULL
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	NULL	PMID29473428-Compound-80	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-1	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-13	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-23	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-26	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-27	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-28	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-34	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-35	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID29649907-Compound-37	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-12	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-15	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-16	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-18	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-18	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-26	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-26	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-27	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-27	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-37	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-38b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-38b	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-39	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-39	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-42	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-45a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 5	hgnc:14068	HDAC5	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-45a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-45a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 9	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-45a	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-47c	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-47d	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-50	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 10	hgnc:18128	HDAC10	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 6	hgnc:14064	HDAC6	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 7	hgnc:14067	HDAC7	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 8	hgnc:13315	HDAC8	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-56	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-57	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-57	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-59	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 2	hgnc:4853	HDAC2	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-59	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 3	hgnc:4854	HDAC3	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-59	NULL	NULL	NULL	NULL	NULL
HISTONE DEACETYLASE 4	hgnc:14063	HDAC4	TTD	2020.06.01	NULL	NULL	PMID29671355-Compound-70	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-63	NULL	NULL	NULL	NULL	NULL
PROTEASOME BETA-8	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID29865878-Compound-64	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30074415-Compound-20	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfonamide derivative 12	NULL	NULL	NULL	NULL	NULL
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sulfonamide-thiadiazole derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic acetylene derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aromatic ethylene derivative 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Benzyl phenyl ether derivative 1	NULL	NULL	NULL	NULL	NULL
CD80-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl compound 1	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	Biaryl compound 1	NULL	NULL	NULL	NULL	NULL
PROGRAMMED CELL DEATH PROTEIN 1	hgnc:8760	PDCD1	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example16	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example4	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example42	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example48	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example50	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example51	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example53	NULL	NULL	NULL	NULL	NULL
PD-1-PD-L1 INTERACTION	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30107136-Compound-Example7	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 2A RECEPTOR	hgnc:5293	HTR2A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
DOPAMINE D3 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 1	NULL	NULL	NULL	NULL	NULL
5-HT 1 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 14	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	Aryl piperazine derivative 14	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-60TABLE5	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR	hgnc:3642	FDXR	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-60TABLE5	NULL	NULL	NULL	NULL	NULL
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-60TABLE5	NULL	NULL	NULL	NULL	NULL
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-LDT66	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-1A	hgnc:277	ADRA1A	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-LDT66	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	NULL	PMID30124346-Compound-LDT66	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Aryl azepine derivative 1	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Benzamide derivative 7	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Benzamide derivative 7	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 1	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 1	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 1	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 2	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 2	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	NULL	Isoindoline derivative 2	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazinyl methyl quinazolinone derivative 3	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	Piperazinyl norbenzomorphane compound 3	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-27	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-54	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-55	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-57	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-57	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-64	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	PMID30185082-Compound-64	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID30259754-Compound-Px-102	NULL	NULL	NULL	NULL	NULL
FARNESOID X-ACTIVATED RECEPTOR	hgnc:7967	NR1H4	TTD	2020.06.01	NULL	NULL	PMID30259754-Compound-pyrrole[2,3-d]azepines	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-15	NULL	NULL	NULL	NULL	NULL
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	NULL	PMID30273516-Compound-39	NULL	NULL	NULL	NULL	NULL
TOLL-LIKE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	PMID30280939-Compound-WO200606195	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.596678082	Bretylium	rxcui:19685	BRETYLIUM	TRUE	FALSE	FALSE
KALLIKREIN-RELATED PEPTIDASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Cetraxate	ncit:C79885	CETRAXATE	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Conjugated estrogens b	NULL	NULL	NULL	NULL	NULL
CALCIUM-DEPENDENT CHLORIDE CHANNEL ANOCTAMIN	NULL	NULL	TTD	2020.06.01	NULL	NULL	Crofelemer	rxcui:1364449	CROFELEMER	TRUE	FALSE	FALSE
HISTAMINE H2 RECEPTOR	hgnc:5183	HRH2	TTD	2020.06.01	NULL	0.9376369863516874	Cimetidine	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
LCK TYROSINE PROTEIN KINASE	hgnc:6524	LCK	TTD	2020.06.01	NULL	0.05348375	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	1.193356164447602	Dapagliflozin	rxcui:1486966	DAPAGLIFLOZIN PROPANEDIOL	TRUE	FALSE	FALSE
FUSION PROTEIN BCR-ABL	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.1766118064547324	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Enteric-coated mycophenolate sodium	NULL	NULL	NULL	NULL	NULL
BACTERIAL DNA GYRASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Finafloxacin	rxcui:1598641	FINAFLOXACIN	TRUE	FALSE	FALSE
STAPHYLOCOCCUS TOPOISOMERASE IV	NULL	NULL	TTD	2020.06.01	NULL	NULL	Finafloxacin	rxcui:1598641	FINAFLOXACIN	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Emepronium	rxcui:3816	EMEPRONIUM	FALSE	FALSE	FALSE
ERYTHROPOIETIN RECEPTOR	hgnc:3416	EPOR	TTD	2020.06.01	NULL	0.6177373086552295	Epoetin alfa	rxcui:105694	EPOETIN ALFA	TRUE	FALSE	FALSE
BACTERIAL PENICILLIN BINDING PROTEIN 2	NULL	NULL	TTD	2020.06.01	NULL	NULL	Imipenem	rxcui:1545986	IMIPENEM ANHYDROUS	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Isopropamide iodide	rxcui:6051	ISOPROPAMIDE IODIDE	TRUE	FALSE	FALSE
PLASMODIUM DIHYDROOROTATE DEHYDROGENASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Leflunomide	rxcui:27169	LEFLUNOMIDE	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	NULL	Levormeloxifene non-steroidal	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V1 RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Lypressin	rxcui:6531	LYPRESSIN	TRUE	FALSE	FALSE
SQUALENE MONOOXYGENASE	hgnc:11279	SQLE	TTD	2020.06.01	NULL	6.563458904461812	Naftifine	rxcui:31476	NAFTIFINE	TRUE	FALSE	FALSE
GAMMA-AMINOBUTYRIC ACID RECEPTOR	NULL	NULL	TTD	2020.06.01	NULL	NULL	Phenobarbital	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Pioglitazone	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CELL MEDIATED IMMUNITY RESPONSE	hgnc:23356	MARCHF8	TTD	2020.06.01	NULL	NULL	Polyoxidonium	NULL	NULL	NULL	NULL	NULL
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.4070362111294147	Pirbuterol	rxcui:33767	PIRBUTEROL	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Saxagliptin	rxcui:1546030	SAXAGLIPTIN ANHYDROUS	TRUE	FALSE	FALSE
MONOAMINE OXIDASE TYPE B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Selegiline Hydrochloride	rxcui:203137	SELEGILINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sitagliptin	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sorivudine	ncit:C1460	SORIVUDINE	TRUE	FALSE	FALSE
STAPHYLOCOCCUS 30S RIBOSOMAL SUBUNIT	NULL	NULL	TTD	2020.06.01	NULL	NULL	Streptomycin	rxcui:10109	STREPTOMYCIN	TRUE	FALSE	FALSE
HUMAN IMMUNODEFICIENCY VIRUS REVERSE TRANSCRIPTASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	Tenofovir disoproxil fumarate	rxcui:322248	TENOFOVIR DISOPROXIL FUMARATE	TRUE	FALSE	FALSE
SOLUTE CARRIER FAMILY 23 MEMBER 2	hgnc:10973	SLC23A2	TTD	2020.06.01	NULL	1.640864726115453	Ursodeoxycholic acid	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	NULL	BMY-43748	NULL	NULL	NULL	NULL	NULL
HEPATITIS C VIRUS NON-STRUCTURAL 4B	NULL	NULL	TTD	2020.06.01	NULL	NULL	Clemizole	ncit:C81139	CLEMIZOLE	FALSE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	NULL	CS-0777	NULL	NULL	NULL	NULL	NULL
SIGMA INTRACELLULAR RECEPTOR 2	hgnc:28106	TMEM97	TTD	2020.06.01	NULL	NULL	CT1812	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA	hgnc:20778	TUBB	TTD	2020.06.01	NULL	NULL	DAVLB-HYDRAZIDE	NULL	NULL	NULL	NULL	NULL
LEUKOTRIENE B4 RECEPTOR 1	hgnc:6713	LTB4R	TTD	2020.06.01	NULL	1.640864726115453	Biomed 101	ncit:C2206	BIOMED 101	FALSE	FALSE	FALSE
LOW-AFFINITY NERVE GROWTH FACTOR RECEPTOR	hgnc:7809	NGFR	TTD	2020.06.01	NULL	NULL	LM11A-31	NULL	NULL	NULL	NULL	NULL
P2Y PURINOCEPTOR 6	hgnc:8543	P2RY6	TTD	2020.06.01	NULL	NULL	GC021109	NULL	NULL	NULL	NULL	NULL
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	NULL	GCC-4401	NULL	NULL	NULL	NULL	NULL
MITOCHONDRIAL ALDEHYDE DEHYDROGENASE	hgnc:404	ALDH2	TTD	2020.06.01	NULL	NULL	GS-6637	NULL	NULL	NULL	NULL	NULL
CAMBRIDGE PATHOLOGY 1 ANTIGEN	hgnc:1804	CD52	TTD	2020.06.01	NULL	NULL	GZ402668	NULL	NULL	NULL	NULL	NULL
RAF MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ICo-007	drugbank:DB05268	ICO-007	FALSE	FALSE	FALSE
IMMUNOGLOBULIN UNSPECIFIC	NULL	NULL	TTD	2020.06.01	NULL	NULL	Immune globulin	ncit:C2701	THERAPEUTIC IMMUNE GLOBULIN	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	NULL	Iptakalim hydrochloride	NULL	NULL	NULL	NULL	NULL
TUBULIN BETA-1 CHAIN	hgnc:16257	TUBB1	TTD	2020.06.01	NULL	NULL	Irofulven/Taxotere	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	0.9211872146613068	GSK525762	ncit:C101538	MOLIBRESIB	FALSE	FALSE	FALSE
B7 HOMOLOG 3	hgnc:19137	CD276	TTD	2020.06.01	NULL	NULL	Omburtamab I-124	NULL	NULL	NULL	NULL	NULL
VEGFR1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	Sirna-027	drugbank:DB05896	SIRNA-027	FALSE	FALSE	FALSE
LEUKOCYTE COMMON ANTIGEN	hgnc:9666	PTPRC	TTD	2020.06.01	NULL	NULL	[131I]-BC8	NULL	NULL	NULL	NULL	NULL
BROMODOMAIN-CONTAINING PROTEIN 4	hgnc:13575	BRD4	TTD	2020.06.01	NULL	1.105424657593568	CPI-0610	ncit:C188265	PELABRESIB	FALSE	FALSE	FALSE
THROMBOSPONDIN-1	hgnc:11785	THBS1	TTD	2020.06.01	NULL	0.9376369863516875	ABT-510	drugbank:DB05434	ABT-510	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	NULL	GDC-0980/RG7422	NULL	NULL	NULL	NULL	NULL
STAPHYLOCOCCUS PEPTIDE DEFORMYLASE	NULL	NULL	TTD	2020.06.01	NULL	NULL	GSK1322322	chembl:CHEMBL3301608	LANOPEPDEN	FALSE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 1	hgnc:10251	ROCK1	TTD	2020.06.01	NULL	NULL	H-1152	NULL	NULL	NULL	NULL	NULL
VOLTAGE-GATED POTASSIUM CHANNEL KV11.1	hgnc:6251	KCNH2	TTD	2020.06.01	NULL	0.1495945049449985	Desmethylastemizole	chembl:CHEMBL60796	DESMETHEYLASTEMIZOLE	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE IX	NULL	NULL	TTD	2020.06.01	NULL	NULL	INDISULAM	ncit:C25797	INDISULAM	FALSE	FALSE	FALSE
PTPN1 MESSENGER RNA	NULL	NULL	TTD	2020.06.01	NULL	NULL	ISIS 113715	drugbank:DB05506	ISIS 113715	FALSE	FALSE	FALSE
GUANYLATE CYCLASE SOLUBLE BETA-1	hgnc:4687	GUCY1B1	TTD	2020.06.01	NULL	NULL	Vericigiuat	NULL	NULL	NULL	NULL	NULL
STRESS-ACTIVATED PROTEIN KINASE 2A	NULL	NULL	TTD	2020.06.01	NULL	NULL	VX-745	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
FMS-LIKE TYROSINE KINASE 3	NULL	NULL	TTD	2020.06.01	NULL	NULL	AC220	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
MATRIX METALLOPROTEINASE-7	hgnc:7174	MMP7	TTD	2020.06.01	NULL	1.500219178	Marimastat	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.5303805175322676	Imiglitazar	ncit:C83791	IMIGLITAZAR	FALSE	FALSE	FALSE
HYPOXIA-INDUCIBLE FACTOR 1 ALPHA	hgnc:4910	HIF1A	TTD	2020.06.01	NULL	0.3621218705909965	IT-101	ncit:C62600	DAVAMOTECAN PEGADEXAMER	FALSE	FALSE	FALSE
DIPEPTIDYL PEPTIDASE 4	NULL	NULL	TTD	2020.06.01	NULL	NULL	SYR-472	chembl:CHEMBL1650443	TRELAGLIPTIN	FALSE	FALSE	FALSE
TRANSFORMING GROWTH FACTOR BETA 1	hgnc:11766	TGFB1	TTD	2020.06.01	NULL	NULL	TG-C	NULL	NULL	NULL	NULL	NULL
NOCICEPTIN RECEPTOR	hgnc:8155	OPRL1	TTD	2020.06.01	NULL	NULL	ATI-17000	NULL	NULL	NULL	NULL	NULL
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	NULL	CART 19	NULL	NULL	NULL	NULL	NULL
NEURAL CELL ADHESION MOLECULE 1	hgnc:7656	NCAM1	TTD	2020.06.01	NULL	NULL	CAR-T cells targeting CD56	NULL	NULL	NULL	NULL	NULL
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	1.193356164447602	Satavaptan	ncit:C80380	SATAVAPTAN	FALSE	FALSE	FALSE
HMG-COA REDUCTASE	hgnc:5006	HMGCR	TTD	2020.06.01	NULL	0.3241214273808303	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.1535312024435511	Trastuzumab-DM1	rxcui:1371041	ADO-TRASTUZUMAB EMTANSINE	TRUE	FALSE	TRUE
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	NULL	EPCAM-targeted CAR-T cells	NULL	NULL	NULL	NULL	NULL
HERPES SIMPLEX VIRUS DNA POLYMERASE UL30	NULL	NULL	TTD	2020.06.01	NULL	NULL	IDX136	NULL	NULL	NULL	NULL	NULL
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	LY-25582	chembl:CHEMBL300662	CHEMBL:CHEMBL300662	FALSE	FALSE	FALSE
NCBIGENE:1519	hgnc:2542	CTSO	GuideToPharmacology	2024.1	inhibitor	0.5770073762164232	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.3163112725041837	IUPHAR.LIGAND:120	ncit:C77255	ALNIDITAN	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.042174836	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.1250182648468916	IUPHAR.LIGAND:7191	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.079077818	IUPHAR.LIGAND:136	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:46	ncit:C76441	OCAPERIDONE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:119	iuphar.ligand:119	[3H]SUMATRIPTAN	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1595977849109255	IUPHAR.LIGAND:152	iuphar.ligand:152	&ALPHA;-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.023151531	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:198	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.036847489	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:169	iuphar.ligand:169	[125I]DOI	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.025739055	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:152	iuphar.ligand:152	&ALPHA;-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.4861821410712453	IUPHAR.LIGAND:233	iuphar.ligand:233	BIMU 1	FALSE	FALSE	FALSE
NCBIGENE:10	hgnc:7646	NAT2	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:261	iuphar.ligand:261	[125I]LSD	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	agonist	0.083744292	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.3777530304726222	IUPHAR.LIGAND:12126	iuphar.ligand:12126	COMPOUND 33A [PMID: 35944901]	FALSE	FALSE	FALSE
NCBIGENE:1263	hgnc:2154	PLK3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8884	iuphar.ligand:8884	COMPOUND 21 [PMID: 23981033]	FALSE	FALSE	FALSE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.637458239	IUPHAR.LIGAND:5697	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
NCBIGENE:1923	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.1108075556053025	IUPHAR.LIGAND:5687	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:1657	hgnc:2937	DMXL1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:9	iuphar.ligand:9	BMY-7378	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	agonist	0.049535539	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6352	rxcui:1546359	QUINAPRILAT	TRUE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:11836	iuphar.ligand:11836	COMPOUND 21 [PMID: 34855405]	FALSE	FALSE	FALSE
NCBIGENE:687	hgnc:1123	KLF9	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:603	iuphar.ligand:603	[125I][NLE75,TYR77]APELIN-36 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:689	hgnc:1125	BTF3	GuideToPharmacology	2024.1	inhibitor	5.250767124	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	0.3860858179095183	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	activator	0.2375912725597036	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:686	hgnc:1122	BTD	GuideToPharmacology	2024.1	blocker	0.1403948428761885	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.201178817	IUPHAR.LIGAND:378	iuphar.ligand:378	PENECA	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:9813	iuphar.ligand:9813	LUF5962	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:5590	iuphar.ligand:5590	TCPA	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:5612	ncit:C152892	VIPADENANT	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1363835616511545	IUPHAR.LIGAND:5593	iuphar.ligand:5593	GS9667	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:447	iuphar.ligand:447	3-ISOBUTYL-8-PYRROLIDINOXANTHINE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1363835616511545	IUPHAR.LIGAND:5601	iuphar.ligand:5601	MRS3558	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278863	IUPHAR.LIGAND:381	iuphar.ligand:381	AS100	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.2273059360852575	IUPHAR.LIGAND:3285	iuphar.ligand:3285	PSB36	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.5413161983061289	IUPHAR.LIGAND:8421	iuphar.ligand:8421	MRS5698	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1804387327687096	IUPHAR.LIGAND:378	iuphar.ligand:378	PENECA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.067664525	IUPHAR.LIGAND:410	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
NCBIGENE:849	ncbigene:849	CATHL1L	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:5488	rxcui:1294569	ESOMEPRAZOLE SODIUM	TRUE	FALSE	FALSE
NCBIGENE:849	ncbigene:849	CATHL1L	GuideToPharmacology	2024.1	inhibitor	0.4730420832044549	IUPHAR.LIGAND:4279	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:1935	hgnc:882	ATR	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12073	iuphar.ligand:12073	CAMONSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:7937	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:6033	iuphar.ligand:6033	RHO KINASE INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:7937	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:8355	iuphar.ligand:8355	COMPOUND 46 [PMID: 16451062]	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:12070	iuphar.ligand:12070	VIC 1911	FALSE	FALSE	FALSE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9397	iuphar.ligand:9397	SNS-314	FALSE	FALSE	FALSE
NCBIGENE:2901	hgnc:4583	GRIK5	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9144	iuphar.ligand:9144	EXAMPLE 2 [WO2013054185]	FALSE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:6189	iuphar.ligand:6189	BAG-2	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11260	iuphar.ligand:11260	BAY86-7548	FALSE	FALSE	FALSE
NCBIGENE:2846	hgnc:4478	LPAR4	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:8318	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:631	iuphar.ligand:631	[125I][D-TYR6,&BETA;-ALA11,PHE13,NLE14]BOMBESIN-(6-14)	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7854	iuphar.ligand:7854	COMPOUND J [PMID: 21907142]	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:6936	iuphar.ligand:6936	LY2811376	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:484	iuphar.ligand:484	NORADRENALINE	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	modulator	0.045898314	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.07767407	IUPHAR.LIGAND:553	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	agonist	0.3387591692625452	IUPHAR.LIGAND:557	rxcui:4333	FENOTEROL	TRUE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:6155	iuphar.ligand:6155	CP-195543	FALSE	FALSE	FALSE
NCBIGENE:1942	hgnc:3221	EFNA1	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:8148	iuphar.ligand:8148	COMPOUND 31 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:1593	hgnc:2605	CYP27A1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8623	iuphar.ligand:8623	COMPOUND 4 [PMID: 19954973]	FALSE	FALSE	FALSE
NCBIGENE:54	hgnc:124	ACP5	GuideToPharmacology	2024.1	modulator	2.019525817	IUPHAR.LIGAND:9474	iuphar.ligand:9474	ENCALERET	FALSE	FALSE	FALSE
NCBIGENE:1623	hgnc:2691	DBIP2	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:8654	iuphar.ligand:8654	M826	FALSE	FALSE	FALSE
NCBIGENE:530	hgnc:1391	CACNA1D	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:2334	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7721	iuphar.ligand:7721	ABT-639	FALSE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7721	iuphar.ligand:7721	ABT-639	FALSE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	0.3281729452230906	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	modulator	0.1535312024435511	IUPHAR.LIGAND:4150	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:9612	iuphar.ligand:9612	AM11542	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:10178	iuphar.ligand:10178	MDMB-FUBINACA	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:735	iuphar.ligand:735	[3H]HU-243	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:9257	iuphar.ligand:9257	AM7499	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.514644363	IUPHAR.LIGAND:10058	ncit:C166825	OLORINAB	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:6665	iuphar.ligand:6665	JNJ-26070109	FALSE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:901	iuphar.ligand:901	AG-041R	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:9055	iuphar.ligand:9055	CE-326597	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:804	iuphar.ligand:802	[3H]ANCRIVIROC	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:796	iuphar.ligand:795	[3H]BANYU (I)	FALSE	FALSE	FALSE
NCBIGENE:2764	hgnc:4373	GMFB	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:11521	iuphar.ligand:11521	LONCASTUXIMAB TESIRINE	FALSE	FALSE	FALSE
NCBIGENE:65	ncbigene:65	ACTBP5	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:814	iuphar.ligand:814	[125I]CCL1 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:66	hgnc:139	ACTBP6	GuideToPharmacology	2024.1	modulator	6.563458904461812	IUPHAR.LIGAND:9046	ncit:C152858	VERCIRNON	FALSE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:11125	iuphar.ligand:11125	PF-07062119	FALSE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	0.6563458904461813	IUPHAR.LIGAND:7385	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:12252	iuphar.ligand:12252	TEPLIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1960	hgnc:3240	EGR3	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8219	iuphar.ligand:8219	COMPOUND 74 [PMID: 24793884]	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4284	iuphar.ligand:4284	PHENYLGLYCINE-01	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:9549	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	NULL	2.386712328895204	IUPHAR.LIGAND:11547	ncit:C174620	ICENTICAFTOR	FALSE	FALSE	FALSE
NCBIGENE:1987	hgnc:3304	EIF5AP3	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:8043	iuphar.ligand:8043	PF-477736	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:8043	iuphar.ligand:8043	PF-477736	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.1187956362798518	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2341	hgnc:3784	FNTAP2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8555	iuphar.ligand:8555	COMPOUND 20 [PMID: 12372533]	FALSE	FALSE	FALSE
NCBIGENE:700	hgnc:1153	BVR1	GuideToPharmacology	2024.1	blocker	8.751278539282415	IUPHAR.LIGAND:4104	iuphar.ligand:4104	3-PHENYL-CPP	FALSE	FALSE	FALSE
NCBIGENE:698	ncbigene:698	BTS1	GuideToPharmacology	2024.1	blocker	7.501095891	IUPHAR.LIGAND:2662	iuphar.ligand:2662	FENOFIBRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:703	hgnc:2022	CLCN4	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:698	ncbigene:698	BTS1	GuideToPharmacology	2024.1	blocker	0.5770073762164232	IUPHAR.LIGAND:2439	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:3248	hgnc:5154	HPGD	GuideToPharmacology	2024.1	inhibitor	0.1058622403945453	IUPHAR.LIGAND:12205	ncit:C175167	OBICETRAPIB	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:6498	iuphar.ligand:6498	WX-UK1	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.082559232	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	antibody	0.9907107780319716	IUPHAR.LIGAND:9109	iuphar.ligand:9109	LY3022855	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.01708122	IUPHAR.LIGAND:5698	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:2361	hgnc:3869	FRA1B	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:6553	iuphar.ligand:6553	METHYL 5-[(4-TERT-BUTYLBENZOYL)AMINO]-2H-1,2,4-TRIAZOLE-3-CARBOXYLATE	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:12375	iuphar.ligand:12375	ADRIXETINIB	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:11190	ncit:C175876	VIMSELTINIB	FALSE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	inhibitor	0.1981421556063943	IUPHAR.LIGAND:5982	iuphar.ligand:5982	GTP-14564	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:4194	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
NCBIGENE:1806	hgnc:3012	DPYD	GuideToPharmacology	2024.1	NULL	0.2476776945079929	IUPHAR.LIGAND:4905	iuphar.ligand:4905	M-CSF	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:7131	rxcui:19737	BROMFENAC	TRUE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10376	iuphar.ligand:10376	ONO-2333MS	FALSE	FALSE	FALSE
NCBIGENE:212	hgnc:397	ALAS2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:920	iuphar.ligand:920	UROCORTIN 1	FALSE	FALSE	FALSE
NCBIGENE:213	hgnc:399	ALB	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:930	iuphar.ligand:930	[125I]ANTISAUVAGINE	FALSE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:10683	iuphar.ligand:10683	KBP-088	FALSE	FALSE	FALSE
NCBIGENE:1840	hgnc:3060	DTX1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306535	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:729	hgnc:1339	C6	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:732	hgnc:1353	C8B	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:730	hgnc:1346	C7	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:8536	iuphar.ligand:8536	SDF1 P2G	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:5924	drugbank:DB07364	6-PHENYL[5H]PYRROLO[2,3-B]PYRAZINE	FALSE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:9701	iuphar.ligand:9701	CX549	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:3634	ncit:C96712	PRANLUKAST	FALSE	FALSE	FALSE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	0.3750547945406749	IUPHAR.LIGAND:7247	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
NCBIGENE:642	hgnc:1059	BLMH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:3206	iuphar.ligand:3206	DIPHOSPHOGLYCOLYL PROLINE	FALSE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12943	iuphar.ligand:12943	TOMINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9354	iuphar.ligand:9354	DDR-IN-1	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.5048814541893701	IUPHAR.LIGAND:1877	iuphar.ligand:1877	15-DEOXY-&DELTA;12,14-PGJ2	FALSE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:5697	rxcui:662281	NILOTINIB	TRUE	FALSE	TRUE
NCBIGENE:2486	ncbigene:2486	FRV3	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:6630	ncit:C84003	NEPICASTAT	FALSE	FALSE	FALSE
NCBIGENE:338	hgnc:603	APOB	GuideToPharmacology	2024.1	agonist	0.063110182	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:7652	iuphar.ligand:7652	UNC9994	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.1166837138570988	IUPHAR.LIGAND:7295	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.2333674277141977	IUPHAR.LIGAND:8370	iuphar.ligand:8370	(-)-STEPHOLIDINE	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	0.1620607136904151	IUPHAR.LIGAND:7002	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7004	iuphar.ligand:7004	C646	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	antibody	0.1666910197958555	IUPHAR.LIGAND:9125	iuphar.ligand:9125	MM-151	FALSE	TRUE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.026319635	IUPHAR.LIGAND:5667	rxcui:1430438	AFATINIB	TRUE	FALSE	TRUE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:1912	iuphar.ligand:1912	17-PHENYL-&OMEGA;-TRINOR-PGE2	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:11889	iuphar.ligand:11889	ZIPALERTINIB	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.1215455352678113	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.3977853881492006	IUPHAR.LIGAND:1892	iuphar.ligand:1892	BUTAPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.055681518	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:5844	iuphar.ligand:5844	L-826266	FALSE	FALSE	FALSE
NCBIGENE:1117	hgnc:1933	CHI3L2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:4717	ncit:C65389	DILAZEP	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:12965	iuphar.ligand:12965	16&ALPHA;-HYDROXYESTRONE	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	NULL	0.4526523382387456	IUPHAR.LIGAND:5027	iuphar.ligand:5027	NEUREGULIN-1	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.7544205637312429	IUPHAR.LIGAND:7422	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.1325951293830669	IUPHAR.LIGAND:2819	iuphar.ligand:2819	PROPYLPYRAZOLETRIOL	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.024479101	IUPHAR.LIGAND:1016	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.024479101	IUPHAR.LIGAND:1016	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2825	iuphar.ligand:2825	DIARYLPROPIONITRILE	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.375054795	IUPHAR.LIGAND:8448	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:994	iuphar.ligand:994	[18F]ET-1 (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:1000	iuphar.ligand:1000	SB234551	FALSE	FALSE	FALSE
NCBIGENE:220	hgnc:409	ALDH1A3	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:1011	iuphar.ligand:1011	RO 46-8443	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:3183	ncit:C66420	PIRIDRONIC ACID	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.062808219	IUPHAR.LIGAND:4360	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:4156	iuphar.ligand:4156	CGS8216	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.054243462	IUPHAR.LIGAND:4277	ncit:C81614	OCINAPLON	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.2134458180312784	IUPHAR.LIGAND:4146	ncit:C72111	BRETAZENIL	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	blocker	0.055681518	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	1.810609352954982	IUPHAR.LIGAND:12404	iuphar.ligand:12404	LAU159	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:4328	iuphar.ligand:4328	TPMPA	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:4099	iuphar.ligand:4099	TRANS-3-ACPBPA	FALSE	FALSE	FALSE
NCBIGENE:422	hgnc:17969	GABRR3	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:419	hgnc:725	ART3	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6103	iuphar.ligand:6103	M1152	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:6119	iuphar.ligand:6119	GALMIC	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:6095	iuphar.ligand:6095	GALANIN(D-TRP2) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:245	hgnc:432	ALOX12P2	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:3861	iuphar.ligand:3861	C7	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3192	iuphar.ligand:3192	COMPOUND 12  [PMID: 12014956]	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	modulator	0.3070624048871023	IUPHAR.LIGAND:5868	iuphar.ligand:5868	L-692,429	FALSE	FALSE	FALSE
NCBIGENE:246	hgnc:433	ALOX15	GuideToPharmacology	2024.1	agonist	0.3070624048871023	IUPHAR.LIGAND:5868	iuphar.ligand:5868	L-692,429	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:4210	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:3784	iuphar.ligand:3784	[125I]GLP-1-(7-37) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:249	hgnc:438	ALPL	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:12175	iuphar.ligand:12175	ORFORGLIPRON	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.6563458904461812	IUPHAR.LIGAND:4165	iuphar.ligand:4165	CX516	FALSE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:4165	iuphar.ligand:4165	CX516	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	modulator	0.6563458904461812	IUPHAR.LIGAND:4248	iuphar.ligand:4248	LY392098	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.028397875	IUPHAR.LIGAND:7096	rxcui:8640	PREDNISONE	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1521961485092594	IUPHAR.LIGAND:4079	iuphar.ligand:4079	[3H]CGP61594	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	inhibitor	0.1902451856365742	IUPHAR.LIGAND:4161	iuphar.ligand:4161	CONANTOKIN-G	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4161	iuphar.ligand:4161	CONANTOKIN-G	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4170	iuphar.ligand:4170	D-CCPENE	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	blocker	0.3977853881492007	IUPHAR.LIGAND:4286	iuphar.ligand:4286	PICROTIN	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	blocker	0.4234489615781814	IUPHAR.LIGAND:4260	iuphar.ligand:4260	N1-DANSYL-SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	blocker	0.069180068	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4332	iuphar.ligand:4332	UBP141	FALSE	FALSE	FALSE
NCBIGENE:423	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	modulator	0.1223955040459079	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	modulator	0.2386712328895204	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:425	ncbigene:425	ARVD4	GuideToPharmacology	2024.1	blocker	1.009762908	IUPHAR.LIGAND:4286	iuphar.ligand:4286	PICROTIN	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:3884	rxcui:1294622	HISTRELIN ACETATE	TRUE	FALSE	FALSE
NCBIGENE:1750	hgnc:2919	DLX6	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:8718	iuphar.ligand:8718	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
NCBIGENE:403	hgnc:694	ARL3	GuideToPharmacology	2024.1	blocker	1.500219178	IUPHAR.LIGAND:2359	iuphar.ligand:2359	ZD7288	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3000	iuphar.ligand:3000	COMPOUND 17 [PMID: 15686906]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5739	iuphar.ligand:5739	COMPOUND 8G [PMID: 21444206]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5740	iuphar.ligand:5740	COMPOUND 23 [PMID: 21444206]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:12151	iuphar.ligand:12151	APD668	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:10166	iuphar.ligand:10166	MBX-2982	FALSE	FALSE	FALSE
NCBIGENE:86	hgnc:24124	ACTL6A	GuideToPharmacology	2024.1	agonist	13.12691780892362	IUPHAR.LIGAND:4032	iuphar.ligand:4032	SPHINGOSYLPHOSPHORYLCHOLINE	FALSE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:8766	iuphar.ligand:8766	JNJ-63533054	FALSE	FALSE	FALSE
NCBIGENE:81	hgnc:166	ACTN4	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:4355	iuphar.ligand:4355	7&BETA;, 25-DIHYDROXYCHOLESTEROL	FALSE	FALSE	FALSE
NCBIGENE:88	hgnc:164	ACTN2	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:5518	iuphar.ligand:5518	ASN04421891	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	0.6482428547616605	IUPHAR.LIGAND:4150	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
NCBIGENE:103	hgnc:225	ADAR	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:2496	iuphar.ligand:2496	NEUROPEPTIDE HEAD ACTIVATOR	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5568	iuphar.ligand:5568	CP55,244	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:745	iuphar.ligand:745	[3H]RIMONABANT	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:10043	iuphar.ligand:10043	SETOGEPRAM	FALSE	FALSE	FALSE
NCBIGENE:148	hgnc:277	ADRA1A	GuideToPharmacology	2024.1	agonist	0.182318303	IUPHAR.LIGAND:3697	iuphar.ligand:3697	R-SPONDIN-1	FALSE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	1.419126249613364	IUPHAR.LIGAND:5246	iuphar.ligand:5246	PIBTU	FALSE	FALSE	FALSE
NCBIGENE:1801	hgnc:3003	DPH1	GuideToPharmacology	2024.1	antibody	2.763561643983921	IUPHAR.LIGAND:10612	iuphar.ligand:10612	TEPROTUMUMAB	FALSE	FALSE	FALSE
NCBIGENE:2457	hgnc:3854	FRA14B	GuideToPharmacology	2024.1	inhibitor	10.50153425	IUPHAR.LIGAND:10450	iuphar.ligand:10450	COMPOUND 7 [PMID: 31381331]	FALSE	FALSE	FALSE
NCBIGENE:2042	hgnc:3387	EPHA3	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8085	iuphar.ligand:8085	COMPOUND 7 [WO2012007375]	FALSE	FALSE	FALSE
NCBIGENE:1738	hgnc:2898	DLD	GuideToPharmacology	2024.1	antibody	17.50255707856483	IUPHAR.LIGAND:7540	rxcui:1872251	BRODALUMAB	TRUE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8085	iuphar.ligand:8085	COMPOUND 7 [WO2012007375]	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.081533651	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:1892	iuphar.ligand:1892	BUTAPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
NCBIGENE:165	hgnc:303	AEBP1	GuideToPharmacology	2024.1	agonist	1.875273972703374	IUPHAR.LIGAND:2906	iuphar.ligand:2906	LPA	FALSE	FALSE	FALSE
NCBIGENE:744	hgnc:1180	MPPED2	GuideToPharmacology	2024.1	activator	5.250767123569449	IUPHAR.LIGAND:4223	iuphar.ligand:4223	INOSITOL 2,4,5-TRISPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1963	iuphar.ligand:1963	BMY 45778	FALSE	FALSE	FALSE
NCBIGENE:2884	hgnc:4561	GPX1P2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11884	iuphar.ligand:11884	SAFUSIDENIB	FALSE	FALSE	FALSE
NCBIGENE:671	hgnc:1095	BPI	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:10930	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
NCBIGENE:682	hgnc:1116	BSG	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:12495	iuphar.ligand:12495	GOITRIN	FALSE	FALSE	FALSE
NCBIGENE:675	hgnc:1101	BRCA2	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:12463	iuphar.ligand:12463	SCUTELLAREIN	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.051478109	IUPHAR.LIGAND:5688	rxcui:1193326	RUXOLITINIB	TRUE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:7909	ncit:C116857	GANDOTINIB	FALSE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:5992	drugbank:DB04716	2-TERT-BUTYL-9-FLUORO-1,6-DIHYDROBENZO[H]IMIDAZO[4,5-F]ISOQUINOLIN-7-ONE	FALSE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.057574201	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:12621	iuphar.ligand:12621	WXFL10203614	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:10744	iuphar.ligand:10744	GOLIDOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.3454452054979901	IUPHAR.LIGAND:9044	rxcui:2569089	DIFELIKEFALIN	TRUE	FALSE	FALSE
NCBIGENE:2379	hgnc:3891	FRA2G	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11584	ncit:C169799	AVORALSTAT	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.138178082	IUPHAR.LIGAND:1642	iuphar.ligand:1642	NOR-BINALTORPHIMINE	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.003578279	IUPHAR.LIGAND:5698	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.003578279	IUPHAR.LIGAND:5717	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.051885051	IUPHAR.LIGAND:7648	drugbank:DB14765	RIVOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	activator	0.1630673019742065	IUPHAR.LIGAND:2326	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
NCBIGENE:514	hgnc:838	ATP5F1E	GuideToPharmacology	2024.1	activator	1.875273972703375	IUPHAR.LIGAND:10336	iuphar.ligand:10336	BL-1249	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	0.2500365296937833	IUPHAR.LIGAND:2334	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:2507	iuphar.ligand:2507	CLOFILIUM	FALSE	FALSE	FALSE
NCBIGENE:385	hgnc:18865	KCNT1	GuideToPharmacology	2024.1	blocker	2.625383561784724	IUPHAR.LIGAND:2507	iuphar.ligand:2507	CLOFILIUM	FALSE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:5240	ncit:C81112	FENCLONINE	FALSE	FALSE	FALSE
NCBIGENE:1242	hgnc:20692	TPH2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:4613	rxcui:3268	DEXFENFLURAMINE	TRUE	FALSE	FALSE
NCBIGENE:1243	ncbigene:1243	CMM	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:6956	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
NCBIGENE:1242	hgnc:20692	TPH2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:5095	iuphar.ligand:5095	&ALPHA;-PROPYLDOPACETAMIDE	FALSE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:1326	iuphar.ligand:1326	[125I]NDP-MSH	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:1337	iuphar.ligand:1337	RY764	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.055504938	IUPHAR.LIGAND:7875	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.045226246	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	0.1842374429322614	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6343	iuphar.ligand:6343	COMPOUND 11C [PMID: 17929793]	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:3050	drugbank:DB07780	FARNESYL DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	agonist	0.1750255707856483	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.7721716358190367	IUPHAR.LIGAND:6253	iuphar.ligand:6253	GSK1331268	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6237	iuphar.ligand:6237	LU AF21934	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6233	iuphar.ligand:6233	VU0400195	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	inhibitor	0.1530835896084387	IUPHAR.LIGAND:1378	iuphar.ligand:1378	LY341495	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6706	iuphar.ligand:6706	LSP4-2022	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	0.3500511415712967	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:296	hgnc:4600	GRM8	GuideToPharmacology	2024.1	agonist	0.3500511415712967	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:1378	iuphar.ligand:1378	LY341495	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9894	ncit:C174741	ESAXERENONE	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	4.145342465975881	IUPHAR.LIGAND:8678	rxcui:2562811	FINERENONE	TRUE	FALSE	FALSE
NCBIGENE:1502	hgnc:6875	MAPK13	GuideToPharmacology	2024.1	inhibitor	0.6482428547616604	IUPHAR.LIGAND:8179	iuphar.ligand:8179	PF-03715455	FALSE	FALSE	FALSE
NCBIGENE:1499	hgnc:2514	CTNNB1	GuideToPharmacology	2024.1	inhibitor	0.061197752	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2093	ncbigene:2093	ERVT3	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:8057	iuphar.ligand:8057	XMD8-92	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:9989	iuphar.ligand:9989	COMPOUND 11 [PMID: 26431428]	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9915	ncit:C90996	PAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:2067	hgnc:3433	ERCC1	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2074	hgnc:3438	ERCC6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9965	iuphar.ligand:9965	COMPOUND 3A [PIPIONNE ET AL, 2018]	FALSE	FALSE	FALSE
NCBIGENE:2072	hgnc:3436	ERCC4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12909	iuphar.ligand:12909	IACS-52825	FALSE	FALSE	FALSE
NCBIGENE:1631	hgnc:7174	MMP7	GuideToPharmacology	2024.1	inhibitor	0.300043836	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1631	hgnc:7174	MMP7	GuideToPharmacology	2024.1	inhibitor	0.6522692078968261	IUPHAR.LIGAND:6464	rxcui:1545992	DOXYCYCLINE ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:1638	hgnc:2709	DCT	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6638	ncit:C66428	PIRLINDOLE	FALSE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:6544	iuphar.ligand:6544	ONO-4817	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:10062	iuphar.ligand:10062	ABX-1431	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:1444	ncit:C81349	ALEMCINAL	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1458	iuphar.ligand:1458	MOTILIN	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:6640	ncit:C80964	LAZABEMIDE	FALSE	FALSE	FALSE
NCBIGENE:2490	ncbigene:2490	FSHMD1B	GuideToPharmacology	2024.1	inhibitor	0.6482428547616605	IUPHAR.LIGAND:10827	rxcui:190376	LINEZOLID	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.252440727	IUPHAR.LIGAND:337	iuphar.ligand:337	KT 5720	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:324	iuphar.ligand:324	HIMBACINE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:312	iuphar.ligand:312	MUSCARINIC TOXIN 2	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	agonist	0.138178082	IUPHAR.LIGAND:295	iuphar.ligand:295	ARECAIDINE PROPARGYL ESTER	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.1105424657593568	IUPHAR.LIGAND:324	iuphar.ligand:324	HIMBACINE	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.03251249	IUPHAR.LIGAND:320	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
NCBIGENE:1818	hgnc:3028	DRD5P2	GuideToPharmacology	2024.1	inhibitor	0.3409589041278864	IUPHAR.LIGAND:10316	rxcui:2670644	REPOTRECTINIB	TRUE	FALSE	TRUE
NCBIGENE:462	hgnc:775	SERPINC1	GuideToPharmacology	2024.1	blocker	0.1215455352678113	IUPHAR.LIGAND:3990	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
NCBIGENE:466	hgnc:783	ATF1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:3970	iuphar.ligand:3970	&ALPHA;-CONOTOXIN MII	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:2087	iuphar.ligand:2087	HEMOKININ 1	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:2103	iuphar.ligand:2103	FK 224	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	0.4268916360625568	IUPHAR.LIGAND:1692	iuphar.ligand:1692	JTC-801	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:10500	iuphar.ligand:10500	NIK-21273	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	inhibitor	1.280674908	IUPHAR.LIGAND:1691	iuphar.ligand:1691	J-113397	FALSE	FALSE	FALSE
NCBIGENE:2859	hgnc:4492	GPR35	GuideToPharmacology	2024.1	antibody	2.019525817	IUPHAR.LIGAND:8453	iuphar.ligand:8453	TAREXTUMAB	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:3797	iuphar.ligand:3797	[125I]NPFF	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	NULL	0.9546849315580818	IUPHAR.LIGAND:3756	iuphar.ligand:3756	[111IN]DOTA-DLVT	FALSE	FALSE	FALSE
NCBIGENE:271	hgnc:469	AMPD2	GuideToPharmacology	2024.1	modulator	4.773424657790408	IUPHAR.LIGAND:6173	iuphar.ligand:6173	GUE1654	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:9122	iuphar.ligand:9122	ACT-335827	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:11448	iuphar.ligand:11448	DANAVOREXTON	FALSE	FALSE	FALSE
NCBIGENE:1873	hgnc:11918	TNFRSF4	GuideToPharmacology	2024.1	NULL	3.500511415712966	IUPHAR.LIGAND:9092	iuphar.ligand:9092	COMPOUND 1 [PMID: 24930776]	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:11403	iuphar.ligand:11403	JH112	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:10277	iuphar.ligand:10277	YNT-185	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:9307	iuphar.ligand:9307	MK-3697	FALSE	FALSE	FALSE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:8132	iuphar.ligand:8132	IL-94	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:8941	iuphar.ligand:8941	COMPOUND 4 [PMID: 24432870]	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9304	iuphar.ligand:9304	TCS 1102	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	inhibitor	0.5527123287967842	IUPHAR.LIGAND:1725	iuphar.ligand:1725	PPADS	FALSE	FALSE	FALSE
NCBIGENE:481	hgnc:804	ATP1B1	GuideToPharmacology	2024.1	modulator	0.1842374429322614	IUPHAR.LIGAND:6981	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1734	drugbank:DB04005	URIDINE 5'-TRIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:2450	iuphar.ligand:2450	NAADP	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:6202	iuphar.ligand:6202	2-THIO-UDP	FALSE	FALSE	FALSE
NCBIGENE:330	hgnc:591	BIRC3	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:1782	iuphar.ligand:1782	UDP-GALACTOSE	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1745	iuphar.ligand:1745	3-PHENACYL-UDP	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:1734	drugbank:DB04005	URIDINE 5'-TRIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:325	hgnc:584	APCS	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:4044	iuphar.ligand:4044	MRS4062	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	agonist	1.193356164447602	IUPHAR.LIGAND:5902	iuphar.ligand:5902	PSB1114	FALSE	FALSE	FALSE
NCBIGENE:370	hgnc:242	ADCYAP1R1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2277	iuphar.ligand:2277	[125I]VIP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:9455	iuphar.ligand:9455	AY77	FALSE	FALSE	FALSE
NCBIGENE:2877	hgnc:4554	GPX2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12481	iuphar.ligand:12481	JBI-589	FALSE	FALSE	FALSE
NCBIGENE:3179	hgnc:9257	PPID	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11612	ncit:C184910	RENCOFILSTAT	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:12119	iuphar.ligand:12119	NVP-CLR457	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.089298761	IUPHAR.LIGAND:8011	iuphar.ligand:8011	KU-0060648	FALSE	FALSE	TRUE
NCBIGENE:2498	hgnc:3990	FTH1P3	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:2844	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:12119	iuphar.ligand:12119	NVP-CLR457	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:12075	iuphar.ligand:12075	VULOLISIB	FALSE	FALSE	FALSE
NCBIGENE:2857	hgnc:4490	GPR34	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9859	ncit:C90808	APILIMOD	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8518	iuphar.ligand:8518	IS20	FALSE	FALSE	FALSE
NCBIGENE:2147	hgnc:3535	F2	GuideToPharmacology	2024.1	inhibitor	0.081281225	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1867	iuphar.ligand:1867	PROKINETICIN-2	FALSE	FALSE	FALSE
NCBIGENE:2393	hgnc:3905	FRA5A	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:6543	iuphar.ligand:6543	UK-356202	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:1865	iuphar.ligand:1865	MIT1	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:12357	ncit:C180833	ELENESTINIB	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:9691	iuphar.ligand:9691	KBP-7018	FALSE	FALSE	FALSE
NCBIGENE:1803	hgnc:3009	DPP4	GuideToPharmacology	2024.1	inhibitor	0.033875917	IUPHAR.LIGAND:7885	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:5712	iuphar.ligand:5712	SU-14813	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:12085	ncit:C162375	PLOGOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:8150	iuphar.ligand:8150	GSK579289A	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:8646	iuphar.ligand:8646	COMPOUND 2 [PMID: 19097784]	FALSE	FALSE	FALSE
NCBIGENE:2771	hgnc:4385	GNAI2	GuideToPharmacology	2024.1	inhibitor	0.1023541349623674	IUPHAR.LIGAND:8313	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
NCBIGENE:938	hgnc:1649	CD24P4	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8520	iuphar.ligand:8520	COMPOUND 58 [PMID: 25037917]	FALSE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11321	iuphar.ligand:11321	WLL-VS	FALSE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:12174	iuphar.ligand:12174	NIC-0102	FALSE	FALSE	FALSE
NCBIGENE:2408	hgnc:9545	PSMB8	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:10409	iuphar.ligand:10409	ZETOMIPZOMIB	FALSE	FALSE	FALSE
NCBIGENE:1485	hgnc:2491	CTAG1B	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:11659	iuphar.ligand:11659	CC-90005	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6025	iuphar.ligand:6025	PKCBETA INHIBITOR	FALSE	FALSE	FALSE
NCBIGENE:1488	hgnc:2495	CTBP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11659	iuphar.ligand:11659	CC-90005	FALSE	FALSE	FALSE
NCBIGENE:1484	ncbigene:1484	CTAA2	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5192	iuphar.ligand:5192	G&OUML; 6983	FALSE	FALSE	FALSE
NCBIGENE:1488	hgnc:2495	CTBP2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9452	iuphar.ligand:9452	PKC&THETA; INHIBITOR 14	FALSE	FALSE	FALSE
NCBIGENE:3084	hgnc:7997	NRG1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:10373	iuphar.ligand:10373	NC1	FALSE	FALSE	FALSE
NCBIGENE:1520	hgnc:2545	CTSS	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
NCBIGENE:1521	hgnc:2546	CTSW	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:5290	iuphar.ligand:5290	Y27632	FALSE	FALSE	FALSE
NCBIGENE:1520	hgnc:2545	CTSS	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:9750	iuphar.ligand:9750	NECROSTATIN-1	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:2642	iuphar.ligand:2642	RO 41-5253	FALSE	FALSE	FALSE
NCBIGENE:591	ncbigene:591	BCHEL1	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:9962	rxcui:2205637	TRIFAROTENE	TRUE	FALSE	FALSE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.3804903712731485	IUPHAR.LIGAND:9691	iuphar.ligand:9691	KBP-7018	FALSE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:2807	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NCBIGENE:592	ncbigene:592	BCHEL3	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:3431	iuphar.ligand:3431	AHPN	FALSE	FALSE	FALSE
NCBIGENE:2549	hgnc:4066	GAB1	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8792	iuphar.ligand:8792	A1120	FALSE	FALSE	FALSE
NCBIGENE:612	hgnc:10479	RXRG	GuideToPharmacology	2024.1	agonist	1.988926940746004	IUPHAR.LIGAND:2807	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NCBIGENE:2185	hgnc:9612	PTK2B	GuideToPharmacology	2024.1	inhibitor	0.023295329	IUPHAR.LIGAND:5713	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
NCBIGENE:2631	hgnc:4179	NIPSNAP2	GuideToPharmacology	2024.1	inhibitor	0.1411496538593938	IUPHAR.LIGAND:4793	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.5000730593875667	IUPHAR.LIGAND:10423	ncit:C152226	RIPASUDIL	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:11910	iuphar.ligand:11910	H3 14S18 STAPLED B-CHAIN	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8330	iuphar.ligand:8330	A(10-24)INSL3	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:11906	iuphar.ligand:11906	COMPOUND 10D [PMID: 34855388]	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:9824	iuphar.ligand:9824	CENERIMOD	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:8709	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.1221108633388244	IUPHAR.LIGAND:7427	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	agonist	0.6563458904461812	IUPHAR.LIGAND:6953	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	NULL	0.1615620653405984	IUPHAR.LIGAND:7189	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
NCBIGENE:922	hgnc:1690	CD5L	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:2713	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:11979	iuphar.ligand:11979	COMPOUND 6F [PMID: 35476936]	FALSE	FALSE	FALSE
NCBIGENE:960	hgnc:1681	CD44	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:9996	ncit:C171820	ELOBIXIBAT	FALSE	FALSE	FALSE
NCBIGENE:1172	hgnc:18044	SLC38A3	GuideToPharmacology	2024.1	NULL	6.563458904461812	IUPHAR.LIGAND:4633	rxcui:4885	GLUTAMINE	TRUE	FALSE	FALSE
NCBIGENE:2204	hgnc:3608	FCAR	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:6622	iuphar.ligand:6622	SK1-I	FALSE	FALSE	FALSE
NCBIGENE:2205	hgnc:3609	FCER1A	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:6625	iuphar.ligand:6625	ROME	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.086361301	IUPHAR.LIGAND:2020	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5633	iuphar.ligand:5633	SIFA-ASN(ACNH-&BETA;-GLC)-TYR3-OCTREOTATE	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2063	iuphar.ligand:2063	[111IN]DOTA-BOC-ATE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.1500219178162699	IUPHAR.LIGAND:2031	rxcui:236167	LANREOTIDE ACETATE	TRUE	FALSE	FALSE
NCBIGENE:2200	hgnc:3603	FBN1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7937	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
NCBIGENE:588	ncbigene:588	BCGF1	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:2638	drugbank:DB03176	KB-141	FALSE	FALSE	FALSE
NCBIGENE:2247	hgnc:3676	FGF2	GuideToPharmacology	2024.1	inhibitor	0.7095631248066824	IUPHAR.LIGAND:11806	iuphar.ligand:11806	GSK329	FALSE	FALSE	FALSE
NCBIGENE:1754	hgnc:11850	TLR4	GuideToPharmacology	2024.1	inhibitor	4.565884455277782	IUPHAR.LIGAND:9036	iuphar.ligand:9036	RESATORVID	FALSE	FALSE	FALSE
NCBIGENE:1755	hgnc:2926	DMBT1	GuideToPharmacology	2024.1	agonist	52.50767123569449	IUPHAR.LIGAND:4931	iuphar.ligand:4931	FLAGELLIN	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.1151484018326633	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	agonist	0.086361301	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:393	hgnc:674	ARHGAP4	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11857	iuphar.ligand:11857	MT-8	FALSE	FALSE	FALSE
NCBIGENE:2420	ncbigene:2420	FRDA2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8624	iuphar.ligand:8624	INHIBITOR 1 [COLOMBO ET AL., 2012]	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	1.544343271638073	IUPHAR.LIGAND:2437	iuphar.ligand:2437	SAG	FALSE	FALSE	FALSE
NCBIGENE:492	hgnc:816	ATP2B3	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:12530	iuphar.ligand:12530	BI 749327	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	2.763561643983921	IUPHAR.LIGAND:2444	iuphar.ligand:2444	ADP RIBOSE	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.7721716358190367	IUPHAR.LIGAND:12530	iuphar.ligand:12530	BI 749327	FALSE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	blocker	0.2125816649218401	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:495	hgnc:819	ATP4A	GuideToPharmacology	2024.1	blocker	0.182318303	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	activator	3.281729452230906	IUPHAR.LIGAND:6405	iuphar.ligand:6405	SF-21	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
NCBIGENE:503	hgnc:13358	MCOLN3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11860	iuphar.ligand:11860	ESTRADIOL 3-METHYL ETHER	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	inhibitor	0.062733179	IUPHAR.LIGAND:5464	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
NCBIGENE:2269	hgnc:12440	TYK2	GuideToPharmacology	2024.1	inhibitor	0.1411496538593938	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:2165	iuphar.ligand:2165	SB-706375	FALSE	FALSE	FALSE
NCBIGENE:1012	hgnc:1753	CDH13	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:4608	iuphar.ligand:4608	[11C]DTBZ	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:2161	iuphar.ligand:2161	4-CL-CINNAMOYL-C[DCYS-4PAL-DTRP-ORN-VAL-CYS]-HIS-AMIDE	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2269	iuphar.ligand:2269	BAY 55-9837	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2222	iuphar.ligand:2222	D(CH2)5[TYR(ME)2,THR4]OVT	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.019490598	IUPHAR.LIGAND:2183	iuphar.ligand:2183	DVDAVP	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:10444	iuphar.ligand:10444	LIT-001	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:2183	iuphar.ligand:2183	DVDAVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2212	iuphar.ligand:2212	[TBAA1,D-TYR(ET)2,VAL4,LYS6,ARG-NH28,DES-GLY9]AVP	FALSE	FALSE	FALSE
NCBIGENE:2790	hgnc:4402	GNG10	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:7732	iuphar.ligand:7732	SM-337	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:2199	ncit:C80380	SATAVAPTAN	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2204	iuphar.ligand:2204	YM 218	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2233	iuphar.ligand:2233	[125I]D(CH2)5[D-TYR(ET)2,VAL4,TYR-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:1510	iuphar.ligand:1510	NPY-(3-36) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	0.7001022831425934	IUPHAR.LIGAND:1504	iuphar.ligand:1504	NEUROPEPTIDE Y	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	FOLFOX-4 REGIMEN	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.2500365296937833	ANTI-EGFR MONOCLONAL ANTIBODY	ncit:C133878	ANTI-EGFR MONOCLONAL ANTIBODY	FALSE	FALSE	TRUE
BAP1	hgnc:950	BAP1	CIViC	10-Apr-24	NULL	0.1491695205559502	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	JNJ38877605	NULL	NULL	NULL	NULL	NULL
FGFR2	hgnc:3689	FGFR2	CIViC	10-Apr-24	NULL	1.831662950082366	FGFR INHIBITOR AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.6050266644442165	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.3090959307472817	REBEMADLIN	ncit:C74594	REBEMADLIN	FALSE	FALSE	TRUE
IKZF1	hgnc:13176	IKZF1	CIViC	10-Apr-24	NULL	0.1400204566285186	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	1.040600372117402	QUIZARTINIB	rxcui:2643048	QUIZARTINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	NULL	RADIATION IONIZING RADIOTHERAPY	NULL	NULL	NULL	NULL	NULL
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	NULL	2,4-PYRIMIDINEDIAMINE	NULL	NULL	NULL	NULL	NULL
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	0.8751278539282416	TEPOTINIB	rxcui:2477103	TEPOTINIB	TRUE	FALSE	TRUE
HLA-DRA	hgnc:4947	HLA-DRA	CIViC	10-Apr-24	NULL	0.3571950424196904	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
MET	hgnc:7029	MET	CIViC	10-Apr-24	NULL	NULL	CARBOPLATIN/PEMETREXED REGIMEN	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.063517344	OMIPALISIB	ncit:C88270	OMIPALISIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.00799386	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
BRCA1	hgnc:1100	BRCA1	CIViC	10-Apr-24	NULL	0.010156223	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.011591097	DOXORUBICIN	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	NULL	G-573	NULL	NULL	NULL	NULL	NULL
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.007103311	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
CCNE1	hgnc:1589	CCNE1	CIViC	10-Apr-24	NULL	5.250767123569449	CDK INHIBITOR SNS-032	ncit:C62523	CDK INHIBITOR SNS-032	FALSE	FALSE	TRUE
IGF2	hgnc:5466	IGF2	CIViC	10-Apr-24	NULL	0.4861821410712453	GANITUMAB	ncit:C71531	GANITUMAB	FALSE	TRUE	TRUE
SGK1	hgnc:10810	SGK1	CIViC	10-Apr-24	NULL	NULL	SGK1-INH	NULL	NULL	NULL	NULL	NULL
CDK9	hgnc:1780	CDK9	CIViC	10-Apr-24	NULL	NULL	CAN508	NULL	NULL	NULL	NULL	NULL
STAT1	hgnc:11362	STAT1	CIViC	10-Apr-24	NULL	8.751278539282415	PICOPLATIN	ncit:C48416	PICOPLATIN	FALSE	FALSE	TRUE
IL6	hgnc:6018	IL6	CIViC	10-Apr-24	NULL	0.007390242	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	CIViC	10-Apr-24	NULL	0.017047945	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	CIViC	10-Apr-24	NULL	0.002914179	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
STAT1	hgnc:11362	STAT1	CIViC	10-Apr-24	NULL	0.060353645	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
MYC	hgnc:7553	MYC	CIViC	10-Apr-24	NULL	0.00517317	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NAPRT	hgnc:30450	NAPRT	CIViC	10-Apr-24	NULL	NULL	GNE-617	NULL	NULL	NULL	NULL	NULL
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.1785975212098452	NIRAPARIB	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
RAC1	hgnc:9801	RAC1	CIViC	10-Apr-24	NULL	0.5834185692854945	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.2282942227638891	NUV-655	ncit:C188054	ALK INHIBITOR NVL-655	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	NULL	TQ-B3101	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	CCT070535	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	iCRT-5	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	IWR-1	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	JW67	NULL	NULL	NULL	NULL	NULL
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	NULL	K-756	NULL	NULL	NULL	NULL	NULL
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.5303805175322676	Berzosertib	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.5303805175322676	Molibresib	ncit:C101538	MOLIBRESIB	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.041101895	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	PLX7904	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1546364663354877	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	RXDX-105	ncit:C107245	AGERAFENIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2290910612377596	RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	S3I-201	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	SBI-0640726	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	BI-69A11	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	DETD-35	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	INU-152	NULL	NULL	NULL	NULL	NULL
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	NULL	BGB659	NULL	NULL	NULL	NULL	NULL
CBL	hgnc:1541	CBL	JAX-CKB	10-Apr-24	NULL	1.312691780892362	Entospletinib	ncit:C105402	ENTOSPLETINIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	Denosumab	rxcui:993449	DENOSUMAB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.015573209	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.3671865121377238	Milciclib	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	JAX-CKB	10-Apr-24	NULL	0.070860555	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
CTNNB1	hgnc:2514	CTNNB1	JAX-CKB	10-Apr-24	NULL	0.072324616	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.020029629	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.736088849	GSK3052230	ncit:C77970	FGF RECEPTOR ANTAGONIST HGS1036	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.026766867	Cediranib	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.1962903597596056	PHA-665752	iuphar.ligand:5700	PHA-665752	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.017218453	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.064824285	Azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.033497717	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.092606122	E6201	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.1842374429322613	LY294002	ncit:C148229	PI3K/BET INHIBITOR LY294002	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	PLM-101	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.081030357	Danusertib	ncit:C61587	DANUSERTIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	Ki23819	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	UNC1666	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	A-1210477	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	IACS-13909	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	NULL	HC-7366	NULL	NULL	NULL	NULL	NULL
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	TP-0184	ncit:C156729	ITACNOSERTIB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.014732792	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.040515178	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	Pz-1	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	AZ8010	NULL	NULL	NULL	NULL	NULL
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.6908904109959803	JDQ443	ncit:C177916	OPNURASIB	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	NULL	PLX7904	NULL	NULL	NULL	NULL	NULL
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.012838061	Trichostatin A	ncit:C1261	TRICHOSTATIN A	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.2567612285364034	Olutasidenib	rxcui:2623641	OLUTASIDENIB	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.022466607	Azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.036680176	Tazemetostat	rxcui:2274378	TAZEMETOSTAT	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	0.055020263	Pamiparib	ncit:C120553	PAMIPARIB	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	JAX-CKB	10-Apr-24	NULL	NULL	TETi76	NULL	NULL	NULL	NULL	NULL
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	NULL	TETi76	NULL	NULL	NULL	NULL	NULL
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	0.8468979231563628	ASP015K	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.048083948	Daunorubicin	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
JAK1	hgnc:6190	JAK1	JAX-CKB	10-Apr-24	NULL	NULL	VSV-delta51	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	NULL	Ropeginterferon	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	NULL	HSV1-dICP0	NULL	NULL	NULL	NULL	NULL
JAK2	hgnc:6192	JAK2	JAX-CKB	10-Apr-24	NULL	NULL	VSV-delta51	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	BGB659	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	PHI-501	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	NULL	NST-628	NULL	NULL	NULL	NULL	NULL
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.07699072	Futibatinib	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.205692444	Temsirolimus	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.2430910705356226	CYH33	ncit:C178401	RISOVALISIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	Carboxyamidotriazole Orotate	ncit:C91090	CARBOXYAMIDOTRIAZOLE OROTATE	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	NULL	WYE-125132	NULL	NULL	NULL	NULL	NULL
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.013140058	Leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.081030357	LY294002	ncit:C148229	PI3K/BET INHIBITOR LY294002	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	Pz-1	NULL	NULL	NULL	NULL	NULL
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	NULL	Y078-DM4	NULL	NULL	NULL	NULL	NULL
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	3.621218705909965	Dalpiciclib	ncit:C125899	DALPICICLIB	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	TPX-0046	ncit:C167210	ENBEZOTINIB	FALSE	FALSE	FALSE
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	NULL	NPS-1034	NULL	NULL	NULL	NULL	NULL
ROS1	hgnc:10261	ROS1	JAX-CKB	10-Apr-24	NULL	NULL	TQ-B3101	NULL	NULL	NULL	NULL	NULL
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.9053046764774912	Camrelizumab	ncit:C123816	CAMRELIZUMAB	FALSE	FALSE	FALSE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	NULL	TETi76	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	MI-63	NULL	NULL	NULL	NULL	NULL
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	1.750255707856483	Selinexor	rxcui:2178390	SELINEXOR	TRUE	FALSE	TRUE
TET2	hgnc:25941	TET2	JAX-CKB	10-Apr-24	NULL	0.2187819634820604	Azacitidine	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.3090959307472817	Nutlin-3a	ncit:C74594	REBEMADLIN	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	NSC59984	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	PK11007	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.005893778	Etoposide	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	p53-SLP vaccine	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	NSC319726	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	YX-02-030	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	Ezabenlimab	ncit:C132252	EZABENLIMAB	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.04636439	TAE684	ncit:C171615	ALK INHIBITOR TAE684	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.077273983	PF-04217903	drugbank:DB12848	PF-04217903	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	Ad5CMV-p53 gene	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	CP-31398	NULL	NULL	NULL	NULL	NULL
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	NULL	NU6027	NULL	NULL	NULL	NULL	NULL
APH1B	hgnc:24080	APH1B	ChEMBL	33	modulator	0.3365876361262467	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	modulator	0.042689164	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1250182648468916	TIVOZANIB HYDROCHLORIDE	rxcui:2534245	TIVOZANIB HYDROCHLORIDE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.093346971	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.09963505	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	FUMAGILLIN	rxcui:1926480	FUMAGILLIN	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.019304291	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	TOXAPHENE	iuphar.ligand:2830	TOXAPHENE	FALSE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	2.386712328895204	DIETHYL-2-TRIDECYLMALONATE	chembl:CHEMBL1797711	CHEMBL:CHEMBL1797711	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.016352436	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.033985548	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.06375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.8140724222588294	POH	ncit:C1461	PERILLYL ALCOHOL	FALSE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	ALMITRINE	rxcui:528	ALMITRINE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.1363835616511545	IUPHAR.LIGAND:5604	ncit:C96195	ROLOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7036	iuphar.ligand:7036	LYS-COA	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.019636377	Rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	ChEMBL	33	inhibitor	0.1151484018326633	ENTRECTINIB	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
MAPK3	hgnc:6877	MAPK3	NCI	14-Sep-17	NULL	0.1524170427741495	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.003608031	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
LTK	hgnc:6721	LTK	DTC	9/2/20	NULL	0.054355767	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
IGH	hgnc:5477	IGH	FDA	10-Apr-24	NULL	1.250182648468916	Venetoclax	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.08914715	IUPHAR.LIGAND:8708	rxcui:2105806	GILTERITINIB	TRUE	FALSE	TRUE
NCBIGENE:2734	hgnc:4316	GLG1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8824	iuphar.ligand:8824	COMPOUND 50 [PMID: 24313754]	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.011152861	olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:9874	iuphar.ligand:9874	VUF14862	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	1.346350544504987	IUPHAR.LIGAND:1273	iuphar.ligand:1273	HTMT	FALSE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8742	iuphar.ligand:8742	VS-4718	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.029698909	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.100589408	STALLIMYCIN	ncit:C1517	STALLIMYCIN	FALSE	FALSE	FALSE
HIPK4	hgnc:19007	HIPK4	DTC	9/2/20	NULL	0.051478109	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.1215455352678113	N-(3,4-DICHLOROPHENYL)BENZAMIDE	chembl:CHEMBL560296	CHEMBL:CHEMBL560296	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	1.458546423213736	OESTROGENS	ncit:C483	THERAPEUTIC ESTROGEN	FALSE	FALSE	FALSE
DTNBP1	hgnc:17328	DTNBP1	PharmGKB	4/5/24	NULL	0.600087671	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
ACY3	hgnc:24104	ACY3	PharmGKB	4/5/24	NULL	1.458546423213736	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:11973	iuphar.ligand:11973	HR1405-01	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	FAMPROFAZONE	ncit:C65616	FAMPROFAZONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.033338204	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
NECTIN4	hgnc:19688	NECTIN4	FDA	10-Apr-24	NULL	4.118248724368196	Enfortumab Vedotin-ejfv	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
CACNG7	hgnc:13626	CACNG7	ChEMBL	33	modulator	0.2243917574174979	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	FLAVANONE	iuphar.ligand:408	FLAVANONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.027929612	GUANIDINONALTRINDOLE	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.071148606	VENLAFAXINE	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.068191781	GLAFENINE	ncit:C72119	GLAFENINE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DIMETHYLAMINOETHANOL	chembl:CHEMBL1135	DIMETHYLAMINOETHANOL	FALSE	FALSE	FALSE
CYBA	hgnc:2577	CYBA	PharmGKB	4/5/24	NULL	0.1746374874801369	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.016690296	lacosamide	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.071780822	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	1.009762908	PYRAZOLE	drugbank:DB02757	PYRAZOLE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.042689164	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.023274677	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.108711535	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
MLLT3	hgnc:7136	MLLT3	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:7709	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	modulator	0.760980743	IUPHAR.LIGAND:12051	iuphar.ligand:12051	PLAZINEMDOR	FALSE	FALSE	FALSE
NCBIGENE:2620	hgnc:4167	GAS2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:2083	ncbigene:2083	ERPL2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6007	iuphar.ligand:6007	MEK INHIBITOR II	FALSE	FALSE	FALSE
PSMB10	hgnc:9538	PSMB10	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
VASOPRESSIN V1B RECEPTOR	hgnc:896	AVPR1B	TTD	2020.06.01	NULL	0.5770073762164232	Oxytocin	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1840222122746302	Clomifene	rxcui:2596	CLOMIPHENE	TRUE	FALSE	FALSE
COAGULATION FACTOR VIII	hgnc:3546	F8	TTD	2020.06.01	NULL	3.088686543276147	Turoctocog alfa	rxcui:1737557	TUROCTOCOG ALFA	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 2	hgnc:1771	CDK2	TTD	2020.06.01	NULL	0.2479701120930082	PHA848125	ncit:C148410	MILCICLIB	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:3444	iuphar.ligand:3444	T0070907	FALSE	FALSE	FALSE
NCBIGENE:2552	hgnc:8157	SIGMAR1	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:10431	iuphar.ligand:10431	E-52862	FALSE	FALSE	FALSE
PDPK1	hgnc:8816	PDPK1	DTC	9/2/20	NULL	0.022099188	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	DTC	9/2/20	NULL	0.008240375	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.2711239478607289	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
NPY	hgnc:7955	NPY	NCI	14-Sep-17	NULL	0.8678953923255289	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
SUBSTANCE-P RECEPTOR	hgnc:11526	TACR1	TTD	2020.06.01	NULL	0.7095631248066824	Rolapitant	rxcui:1665496	ROLAPITANT	TRUE	FALSE	FALSE
NCBIGENE:2443	hgnc:3841	FRA11F	GuideToPharmacology	2024.1	antibody	2.500365296937833	IUPHAR.LIGAND:11531	ncit:C139025	ABRILUMAB	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.1640864726115453	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
NCBIGENE:38	hgnc:93	ACAT1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3871	iuphar.ligand:3871	DNAL-CYC(CYS-TYR-DTRP-ORN-VAL)-NAL-NH2	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.011049594	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002657809	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.019325606	DNDI1417548	chembl:CHEMBL2094789	CHEMBL:CHEMBL2094789	FALSE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	0.6213925590023018	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	1.193356164447602	Oglemilast	ncit:C87376	OGLEMILAST	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.210030685	AVE0847	chembl:CHEMBL3545295	AVE0847	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PHENYL SALICYLATE	rxcui:36122	PHENYL SALICYLATE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.004889893	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.016221091	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	1.810609352954982	EDELFOSINE	ncit:C956	EDELFOSINE	FALSE	FALSE	FALSE
RPL27A	hgnc:10329	RPL27A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
APOLIPOPROTEIN E	hgnc:613	APOE	TTD	2020.06.01	NULL	0.9053046764774912	CN-105	drugbank:DB18345	CN-105	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:8427	ncit:C152177	RELENOPRIDE	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.1187956362798518	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.4167275494896388	IUPHAR.LIGAND:1799	iuphar.ligand:1799	[ILE5,TRP23]PTHRP-(2-36) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:364	hgnc:640	AQP7	GuideToPharmacology	2024.1	agonist	4.773424657790408	IUPHAR.LIGAND:2144	iuphar.ligand:2144	&BETA;-PHENYLETHYLAMINE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.2453629496995069	MONOETHANOLAMINE	ncit:C61756	MONOETHANOLAMINE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	CP-339818	iuphar.ligand:2558	CP-339818	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	ZUCAPSAICIN	ncit:C75078	ZUCAPSAICIN	FALSE	FALSE	FALSE
LUTEINIZING HORMONE RECEPTOR	hgnc:6585	LHCGR	TTD	2020.06.01	NULL	6.563458904461812	Choriogonadotropin alfa	rxcui:283550	CHORIOGONADOTROPIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:255	iuphar.ligand:255	SB 203186	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:743	ncit:C73244	RIMONABANT	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	1.186614039224734	Perindopril	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:5693	ncit:C77392	ENZASTAURIN	FALSE	FALSE	TRUE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.100976291	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	ALVERINE CITRATE	rxcui:71767	ALVERINE CITRATE	FALSE	FALSE	FALSE
SODIUM/GLUCOSE COTRANSPORTER 2	hgnc:11039	SLC5A4	TTD	2020.06.01	NULL	1.193356164447602	Canagliflozin	rxcui:1373458	CANAGLIFLOZIN	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:9003	iuphar.ligand:9003	ADL5747	TRUE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.072927321	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
NCBIGENE:2230	hgnc:3638	FDX1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
CA9	hgnc:1383	CA9	ChEMBL	33	inhibitor	0.3125456621172291	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
PRKCH	hgnc:9403	PRKCH	MyCancerGenome	20-Jun-17	inhibitor	0.060423097	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
SERINE PROTEASE HEPSIN	hgnc:5155	HPN	TTD	2020.06.01	NULL	3.750547945406749	Meclizine	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:5605	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	0.729273212	IUPHAR.LIGAND:3317	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.056157937	TRIFLUOPERAZINE HYDROCHLORIDE	rxcui:91130	TRIFLUOPERAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:420	hgnc:726	ART4	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:4328	iuphar.ligand:4328	TPMPA	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.012495876	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.018521224	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
MMP8	hgnc:7175	MMP8	ChEMBL	33	inhibitor	1.250182648468916	REBIMASTAT	ncit:C1875	REBIMASTAT	FALSE	FALSE	FALSE
CXCR5	hgnc:1060	CXCR5	NCI	14-Sep-17	NULL	0.4167275494896388	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:11898	iuphar.ligand:11898	COMPOUND 54	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.009349657	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
NCBIGENE:43	hgnc:108	ACHE	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:681	iuphar.ligand:681	&ALPHA;-CGRP	FALSE	FALSE	FALSE
CALCB	hgnc:1438	CALCB	ChEMBL	33	inhibitor	4.375639269641208	FREMANEZUMAB	rxcui:2056691	FREMANEZUMAB	TRUE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	0.089756703	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	CD19-CAR-T2 Cells	ncit:C179281	CD19-TARGETED CAR T2 CELLS	FALSE	FALSE	FALSE
CD3G	hgnc:1675	CD3G	ChEMBL	33	modulator	0.42006137	BLINATUMOMAB	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.2792961235941196	LEVOSALBUTAMOL	rxcui:237159	LEVALBUTEROL	TRUE	FALSE	FALSE
EIF2AK4	hgnc:19687	EIF2AK4	PharmGKB	4/5/24	NULL	0.4861821410712454	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
UNIPROT:P06213	hgnc:6091	INSR	TEND	1-Aug-11	NULL	0.042459033	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.016161179	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
TMSB10	hgnc:11879	TMSB10	NCI	14-Sep-17	NULL	3.182283105193606	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.037666909	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:2180	hgnc:3569	ACSL1	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:7864	iuphar.ligand:7864	COMPOUND 30 [PMID: 23414845]	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.4167275494896388	COPANLISIB HYDROCHLORIDE	ncit:C138994	COPANLISIB HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.097236428	TAK-733	drugbank:DB12241	TAK-733	FALSE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.1646008502686348	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.001864751	SORAFENIB TOSYLATE	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	LAMELLARIN D	chembl:CHEMBL373114	LAMELLARIN D	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	3.500511415712966	HMS5552	ncit:C169919	DORZAGLIATIN	FALSE	FALSE	FALSE
NCBIGENE:2599	hgnc:1375	CA4	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:10434	iuphar.ligand:10434	COMPOUND 5B  [PMID: 31287314]	FALSE	FALSE	FALSE
CCND3	hgnc:1585	CCND3	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.5834185692854945	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	METOCHALCONE	chembl:CHEMBL36584	METOCHALCONE	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.042073455	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.038159645	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	1.312691780892362	IMMUNOMODULATORS	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
S100A8	hgnc:10498	S100A8	NCI	14-Sep-17	NULL	0.9376369863516874	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.2128689374420047	SOLIFENACIN	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.099220845	NVP-BEZ239	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	GNF-PF-4992	chembl:CHEMBL275177	CHEMBL:CHEMBL275177	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	TUBERCIDIN	ncit:C911	TUBERCIDIN	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.1286952726365061	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.3241214273808302	IMC-EB10	chembl:CHEMBL2109328	IMC-EB10	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	binder	3.889457128569962	LUTETIUM LU 177 VIPIVOTIDE TETRAXETAN	rxcui:2597053	LUTETIUM LU 177 VIPIVOTIDE TETRAXETAN	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.06375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1875273972703374	MECLOFENAMIC ACID	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	OncoKB	23-Jul-20	NULL	0.1151484018326633	Entrectinib	rxcui:2197862	ENTRECTINIB	TRUE	FALSE	TRUE
VOLTAGE-GATED POTASSIUM CHANNEL KV7.3	hgnc:6297	KCNQ3	TTD	2020.06.01	NULL	0.5357925636295356	Linopirdine	ncit:C82306	LINOPIRDINE	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	DTC	9/2/20	NULL	0.032817295	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1458546423213736	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.092443083	CANTHARIDIC_ACID	chembl:CHEMBL275516	CANTHARIDIC_ACID	FALSE	FALSE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TEND	1-Aug-11	NULL	10.50153424713889	ALMITRINE	rxcui:528	ALMITRINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	DEOXIEPINEPHRINE	chembl:CHEMBL31088	DEOXIEPINEPHRINE	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1708122031089606	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.108040476	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
UNIPROT:P16581	hgnc:10718	SELE	TdgClinicalTrial	Jan-14	NULL	4.773424657790408	BIMOSIAMOSE	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
UNIPROT:P00740	hgnc:3551	F9	TdgClinicalTrial	Jan-14	NULL	0.1535312024435511	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2041114528112516	CID 5330286	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	GNF-PF-1008	chembl:CHEMBL602424	CHEMBL:CHEMBL602424	FALSE	FALSE	FALSE
SENP7	hgnc:30402	SENP7	DTC	9/2/20	NULL	0.2734774543525755	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
CD5	hgnc:1685	CD5	NCI	14-Sep-17	NULL	0.6563458904461812	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.5000730593875666	PSORALEN	ncit:C2586	PSORALEN	FALSE	FALSE	FALSE
NCBIGENE:496	hgnc:820	ATP4B	GuideToPharmacology	2024.1	blocker	0.1250182648468916	IUPHAR.LIGAND:2844	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
NCBIGENE:507	hgnc:831	ATP5F1BP1	GuideToPharmacology	2024.1	blocker	0.750109589	IUPHAR.LIGAND:2419	iuphar.ligand:2419	ALLICIN	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	inhibitor	0.078276194	CARVEDILOL PHOSPHATE	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.009076521	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
KLKB1	hgnc:6371	KLKB1	ChEMBL	33	inhibitor	7.501095891	BEROTRALSTAT HYDROCHLORIDE	rxcui:2467541	BEROTRALSTAT HYDROCHLORIDE	TRUE	FALSE	FALSE
PSMA1	hgnc:9530	PSMA1	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.3351553483129436	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.1591141552596803	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
CRABP2	hgnc:2339	CRABP2	DTC	9/2/20	NULL	7.001022831425932	BESTATIN METHYL ESTER	chembl:CHEMBL457092	BESTATIN METHYL ESTER	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	MEDI-551	rxcui:2373950	INEBILIZUMAB-CDON	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8469	iuphar.ligand:8469	SCH 900271	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.053445395	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	1-HEXYLPYRIDINIUM IODIDE	chembl:CHEMBL555242	CHEMBL:CHEMBL555242	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.3500511415712966	BIPHENYL	chembl:CHEMBL1231413	BIPHENYL	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.047176704	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005105763	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.019318496	CID 2056784	chembl:CHEMBL261123	CHEMBL:CHEMBL261123	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	OncoKB	23-Jul-20	NULL	1.831662950082366	Debio1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.00679975	RITANSERIN	ncit:C95217	RITANSERIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	DNDI1417420	chembl:CHEMBL1546223	CHEMBL:CHEMBL1546223	FALSE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.7095631248066824	IMIDAFENACIN	ncit:C83789	IMIDAFENACIN	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	ChEMBL	33	inhibitor	0.4487835148349957	BENTAMAPIMOD	ncit:C87441	BENTAMAPIMOD	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007330402	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	ILOPROST	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
UNIPROT:P00451	hgnc:3546	F8	TdgClinicalTrial	Jan-14	NULL	0.1286952726365061	THROMBIN	rxcui:10528	THROMBIN	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.059532507	IUPHAR.LIGAND:152	iuphar.ligand:152	&ALPHA;-METHYL-5-HT	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	DTC	9/2/20	NULL	0.008301608	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:Q8WUI4	hgnc:14067	HDAC7	TdgClinicalTrial	Jan-14	NULL	0.094608417	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:1120	hgnc:1938	CHKB	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:1231	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	CARBETAPENTANE CITRATE	rxcui:283547	CARBETAPENTANE CITRATE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.025304902	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	CLORGYLINE HYDROCHLORIDE	chembl:CHEMBL539507	CLORGYLINE HYDROCHLORIDE	FALSE	FALSE	FALSE
DTNBP1	hgnc:17328	DTNBP1	PharmGKB	4/5/24	NULL	0.4145342465975881	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
POLYPEPTIDE DEFORMYLASE	hgnc:30012	PDF	TTD	2020.06.01	NULL	6.563458904461812	Chlorproguanil	ncit:C79941	CHLORPROGUANIL	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.1190650141398968	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	inhibitor	0.036062961	ETIFOXINE	rxcui:24441	ETIFOXINE	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1988926940746003	DIGOXIGENIN	drugbank:DB03671	DIGOXIGENIN	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1172046232939609	DIHYDREXIDINE	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
NOTCH2	hgnc:7882	NOTCH2	MyCancerGenome	20-Jun-17	other/unknown	1.500219178	REGN421	ncit:C82367	ENOTICUMAB	FALSE	FALSE	TRUE
UNIPROT:P29320	hgnc:3387	EPHA3	TdgClinicalTrial	Jan-14	NULL	11.66837138570988	KB004	ncit:C116629	IFABOTUZUMAB	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.6674703970639131	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
NCBIGENE:939	hgnc:11922	CD27	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11229	iuphar.ligand:11229	INHIBITOR CB3	FALSE	FALSE	FALSE
ARID1A	hgnc:11110	ARID1A	JAX-CKB	10-Apr-24	NULL	0.1446492320542548	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.079557078	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
CYB5R2	hgnc:24376	CYB5R2	PharmGKB	4/5/24	NULL	2.100306849	rasburicase	rxcui:283821	RASBURICASE	TRUE	FALSE	FALSE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.1440539677248134	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:12165	iuphar.ligand:12165	CHF-6366	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.091636424	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
SRD5A2	hgnc:11285	SRD5A2	ChEMBL	33	inhibitor	3.750547945	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.011810092	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.008922289	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.042379073	CIS-2,4,3',5'-TETRAMETHOXYSTILBENE	chembl:CHEMBL221300	CHEMBL:CHEMBL221300	FALSE	FALSE	FALSE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	MT110	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
NCBIGENE:372	hgnc:649	ARCN1	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2276	iuphar.ligand:2276	RO 25-1392	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.4167275494896388	MECAMYLAMINE	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	DTC	9/2/20	NULL	1.666910197958555	GSK-4112	iuphar.ligand:2903	GSK4112	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.070860555	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.039598545	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002936671	OXYMETAZOLINE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIM1	hgnc:8986	PIM1	DTC	9/2/20	NULL	1.500219178	BAS-8770954	chembl:CHEMBL478324	CHEMBL:CHEMBL478324	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	LEFAMULIN ACETATE	rxcui:2198943	LEFAMULIN ACETATE	TRUE	FALSE	FALSE
RPL24	hgnc:10325	RPL24	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	MUSCARINE	iuphar.ligand:3996	MUSCARINE	FALSE	FALSE	FALSE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TEND	1-Aug-11	NULL	2.625383561784724	BACLOFEN	rxcui:1292	BACLOFEN	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TEND	1-Aug-11	NULL	0.091796628	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-RET	hgnc:9967	RET	TTD	2020.06.01	NULL	4.699760697022038	LOXO-292	rxcui:2370147	SELPERCATINIB	TRUE	FALSE	TRUE
IBSP	hgnc:5341	IBSP	NCI	14-Sep-17	NULL	0.3962843112127886	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	0.750109589	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
ECTO-5'-NUCLEOTIDASE	hgnc:8021	NT5E	TTD	2020.06.01	NULL	2.763561643983921	CPI-006	ncit:C156061	MUPADOLIMAB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	2,3,4-TRIHYDROXYBENZALDEHYDE	chembl:CHEMBL254077	CHEMBL:CHEMBL254077	FALSE	FALSE	FALSE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.060423097	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006182465	enalapril	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.071439008	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
PLASMA KALLIKREIN	hgnc:6371	KLKB1	TTD	2020.06.01	NULL	11.25164383622025	Ecallantide	rxcui:658708	ECALLANTIDE	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.041475254	FAGARONINE	chembl:CHEMBL282622	FAGARONINE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.012070729	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	4-IMIDAZOLEACRYLIC ACID	chembl:CHEMBL1236602	CHEMBL:CHEMBL1236602	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
SCN7A	hgnc:10594	SCN7A	ChEMBL	33	blocker	0.076765601	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:10185	iuphar.ligand:10185	NFP	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:5906	iuphar.ligand:5906	COMPOUND 20O [PMID: 22984835]	FALSE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.023151531	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:224	hgnc:403	ALDH3A2	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:3935	iuphar.ligand:3935	F2L	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.030176823	DOXORUBICIN HYDROCHLORIDE	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
PSEN1	hgnc:9508	PSEN1	ChEMBL	33	inhibitor	0.6731752722524935	RG-4733	drugbank:DB11870	RG-4733	FALSE	FALSE	FALSE
RPL21	hgnc:10313	RPL21	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	ENPIROLINE	ncit:C75267	ENPIROLINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.058341857	AMBUNOL	chembl:CHEMBL454893	AMBUNOL	FALSE	FALSE	FALSE
UNIPROT:P51170	hgnc:10602	SCNN1G	TEND	1-Aug-11	NULL	1.372749574789398	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	TCMDC-124557	chembl:CHEMBL530682	CHEMBL:CHEMBL530682	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.021484317	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PROROXAN	ncit:C84119	PROROXAN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	4'-METHOXYCHALCONE	chembl:CHEMBL34398	4'-METHOXYCHALCONE	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.1161674142382621	griseofulvin	rxcui:5021	GRISEOFULVIN	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.029665351	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.2711239478607289	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	0.5707355569097228	ALCURONIUM	rxcui:460	ALCURONIUM	TRUE	FALSE	FALSE
ISOCITRATE DEHYDROGENASE	hgnc:5382	IDH1	TTD	2020.06.01	NULL	0.1604757678352521	AG-881	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.034727296	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	ChEMBL	33	inhibitor	0.1227531764715242	MLN-8054	iuphar.ligand:5696	MLN-8054	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.5903640284436551	COBIMETINIB	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.011757204	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	NSC-402083	chembl:CHEMBL1546228	CHEMBL:CHEMBL1546228	FALSE	FALSE	FALSE
UNIPROT:P14778	hgnc:5993	IL1R1	TEND	1-Aug-11	NULL	3.141484604	ANAKINRA	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
PTK2	hgnc:9611	PTK2	DTC	9/2/20	NULL	3.889457128569962	TPKI-48	chembl:CHEMBL2333445	CHEMBL:CHEMBL2333445	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.016992774	FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
UNIPROT:Q9Y275	hgnc:11929	TNFSF13B	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	TACI-IG	ncit:C81166	ATACICEPT	FALSE	FALSE	FALSE
NCBIGENE:2360	hgnc:3868	FRA1A	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11990	iuphar.ligand:11990	EP-7041	FALSE	FALSE	FALSE
NCBIGENE:214	hgnc:400	ALCAM	GuideToPharmacology	2024.1	modulator	1.346350544504987	IUPHAR.LIGAND:10506	iuphar.ligand:10506	MEVIDALEN	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:11695	iuphar.ligand:11695	HTL6641	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.097236428	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	PharmGKB	4/5/24	NULL	0.026519026	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR	hgnc:2434	CSF2	TTD	2020.06.01	NULL	0.7001022831425933	CGTG-102	ncit:C98287	GM-CSF-ENCODING ONCOLYTIC ADENOVIRUS CGTG-102	FALSE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	activator	1.093909817410302	IUPHAR.LIGAND:2626	iuphar.ligand:2626	VERATRIDINE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.063415062	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
TRPC5	hgnc:12337	TRPC5	DTC	9/2/20	NULL	21.00306849427779	5,5'-DITHIOBIS(2-NITROBENZOIC ACID)	chembl:CHEMBL395814	CHEMBL:CHEMBL395814	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.024479101	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.086219493	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.00804962	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
CACNA1C	hgnc:1390	CACNA1C	PharmGKB	4/5/24	NULL	0.063839114	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
UNIPROT:P30939	hgnc:5292	HTR1F	TdgClinicalTrial	Jan-14	NULL	0.4150804050252529	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.076765601	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	OncoKB	23-Jul-20	NULL	1.105424657593568	Debio1347	ncit:C174762	ZOLIGRATINIB	FALSE	FALSE	TRUE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.037884323	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.025298806	METARAMINOL	rxcui:6805	METARAMINOL	TRUE	FALSE	FALSE
HLA-C	hgnc:4933	HLA-C	PharmGKB	4/5/24	NULL	0.066297565	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.037398626	DOXAZOSIN MESYLATE	rxcui:39173	DOXAZOSIN MESYLATE	TRUE	FALSE	FALSE
TSSK2	hgnc:11401	TSSK2	DTC	9/2/20	NULL	0.2692701089009974	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	1.640864726115453	EMPAGLIFLOZIN	rxcui:1545653	EMPAGLIFLOZIN	TRUE	FALSE	FALSE
PSMC1	hgnc:9547	PSMC1	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:8074	iuphar.ligand:8074	NG-25	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.010199625	mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.011190893	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.064347636	AM-251	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:12716	ncit:C160603	CAMIZESTRANT	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:8584	iuphar.ligand:8584	AQ-RA 741	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.007903021	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
MAOB	hgnc:6834	MAOB	NCI	14-Sep-17	NULL	0.097870776	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006756874	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
STAT1	hgnc:11362	STAT1	DTC	9/2/20	NULL	2.187819634820604	GARCINOL	iuphar.ligand:7001	GARCINOL	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	TENATOPRAZOLE	ncit:C90934	TENATOPRAZOLE	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	CHLORPHENIRAMINE	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
HSPB1	hgnc:5246	HSPB1	NCI	14-Sep-17	NULL	0.3241214273808303	PROTEIN KINASE C INHIBITOR	ncit:C2089	PROTEIN KINASE C INHIBITOR	FALSE	FALSE	FALSE
CHRM4	hgnc:1953	CHRM4	DTC	9/2/20	NULL	0.3889457128569963	PIPERTRAMINE	chembl:CHEMBL127273	PIPERTRAMINE	FALSE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.072927321	Rigosertib	ncit:C152216	RIGOSERTIB	FALSE	FALSE	TRUE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.012756966	palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
GRK5	hgnc:4544	GRK5	DTC	9/2/20	NULL	0.034727296	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	0.1666910197958555	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	BROMOXYNIL	chembl:CHEMBL453905	BROMOXYNIL	FALSE	FALSE	FALSE
UNIPROT:P22102	hgnc:4163	GART	TEND	1-Aug-11	NULL	0.1536809889825205	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
UNIPROT:P78334	hgnc:4085	GABRE	TEND	1-Aug-11	NULL	0.100976291	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:2600	hgnc:1639	CD2	GuideToPharmacology	2024.1	NULL	11.66837138570988	IUPHAR.LIGAND:6787	rxcui:299635	ALEFACEPT	TRUE	TRUE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:2087	iuphar.ligand:2087	HEMOKININ 1	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	(S)-WILLARDIINE	chembl:CHEMBL122005	(S)-WILLARDIINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.00903591	FLUVOXAMINE	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002861765	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.2917092846427472	CID 752709	chembl:CHEMBL429335	CHEMBL:CHEMBL429335	FALSE	FALSE	FALSE
ATP7B	hgnc:870	ATP7B	PharmGKB	4/5/24	NULL	0.1988926940746004	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1346350544504987	IUPHAR.LIGAND:4079	iuphar.ligand:4079	[3H]CGP61594	FALSE	FALSE	FALSE
NCBIGENE:2071	hgnc:3435	ERCC3	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:8173	iuphar.ligand:8173	CEP-1347	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124620	chembl:CHEMBL524930	CHEMBL:CHEMBL524930	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.032055965	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
FOCAL ADHESION KINASE 1	hgnc:9611	PTK2	TTD	2020.06.01	NULL	3.889457128569962	GSK-2256098	chembl:CHEMBL4742157	GSK-2256098	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.1640864726115453	OLSALAZINE SODIUM	rxcui:104123	OLSALAZINE SODIUM	TRUE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:7453	rxcui:1364449	CROFELEMER	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CIViC	10-Apr-24	NULL	0.3509871071904712	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	OncoKB	23-Jul-20	NULL	0.5903640284436551	Cobimetinib	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	1.544343271638073	Demecarium bromide	rxcui:22482	DEMECARIUM BROMIDE	TRUE	FALSE	FALSE
RPS4X	hgnc:10424	RPS4X	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
PROS1	hgnc:9456	PROS1	PharmGKB	4/5/24	NULL	1.875273972703375	synthetic conjugated estrogens, A	rxcui:253166	SYNTHETIC CONJUGATED ESTROGENS, A	FALSE	FALSE	FALSE
VCAM1	hgnc:12663	VCAM1	NCI	14-Sep-17	NULL	0.3889457128569962	6-MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
GATA4	hgnc:4173	GATA4	DTC	9/2/20	NULL	17.50255707856483	RIBAVIRIN MONOPHOSPHATE	drugbank:DB14663	RIBAVIRIN MONOPHOSPHATE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.027276712	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.044310271	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.1400204566285186	MURAGLITAZAR	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
UNIPROT:P10826	hgnc:9865	RARB	TdgClinicalTrial	Jan-14	NULL	0.8423690572571311	TAZAROTENE	rxcui:83947	TAZAROTENE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:170	iuphar.ligand:170	ORG 12962	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.057700738	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	11.66837138570988	BAY 94-9343	ncit:C98293	ANETUMAB RAVTANSINE	FALSE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	1.078924751	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005835482	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	TCMDC-124585	chembl:CHEMBL587856	CHEMBL:CHEMBL587856	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.4565884455277783	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV2.1	hgnc:1388	CACNA1A	TTD	2020.06.01	NULL	0.3182283105193606	Flunarizine	rxcui:4459	FLUNARIZINE	FALSE	FALSE	FALSE
RIPK2	hgnc:10020	RIPK2	DTC	9/2/20	NULL	0.8751278539282416	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.058799184	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	DICHLORVOS	drugbank:DB11397	DICHLORVOS	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	PROMAZINE HYDROCHLORIDE	rxcui:142444	PROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PADI4	hgnc:18368	PADI4	DTC	9/2/20	NULL	1.312691780892362	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.2206204673768676	VX-702	drugbank:DB05470	VX-702	FALSE	FALSE	FALSE
NCBIGENE:1936	hgnc:3211	EEF1D	GuideToPharmacology	2024.1	inhibitor	0.047049885	IUPHAR.LIGAND:7885	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:6478	iuphar.ligand:6478	ODANACATIB	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
IL2	hgnc:6001	IL2	NCI	14-Sep-17	NULL	0.1491695205559502	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1470803115845784	THC	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	DNDI1417032	chembl:CHEMBL1523974	CHEMBL:CHEMBL1523974	FALSE	FALSE	FALSE
P4HB	hgnc:8548	P4HB	DTC	9/2/20	NULL	4.773424657790408	LIQUIRITIN	chembl:CHEMBL511995	LIQUIRITIN	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.8607814956671229	DYDROGESTERONE	rxcui:3706	DYDROGESTERONE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.057574201	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.055740628	U-74389G MALEATE	chembl:CHEMBL1256186	CHEMBL:CHEMBL1256186	FALSE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.015193192	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.05890913	Neratinib	rxcui:1940643	NERATINIB	TRUE	FALSE	TRUE
STK11	hgnc:11389	STK11	JAX-CKB	10-Apr-24	NULL	0.9053046764774912	Rivoceranib	ncit:C152237	RIVOCERANIB	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.1158257453728555	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.3409589041278864	PMSG	ncit:C29773	PREGNANT MARE SERUM GONADOTROPIN	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.172722603	tipiracil / trifluridine	drugbank:DB08937	TAS-102	FALSE	FALSE	FALSE
UNIPROT:P33527	hgnc:51	ABCC1	TEND	1-Aug-11	NULL	0.1844531776429549	SULFINPYRAZONE	rxcui:10205	SULFINPYRAZONE	TRUE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.2117244807890907	IUPHAR.LIGAND:6908	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
ALB	hgnc:399	ALB	NCI	14-Sep-17	NULL	0.3409589041278863	RALTITREXED	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	ADIPHENINE	rxcui:333	ADIPHENINE	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.017775109	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
NCBIGENE:268	hgnc:464	AMH	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:3351	iuphar.ligand:3351	LY255283	FALSE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.1653584607713247	ISOPROTERENOL HYDROCHLORIDE	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	agonist	0.064033745	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:7074	rxcui:4278	FAMOTIDINE	TRUE	FALSE	FALSE
NCBIGENE:540	hgnc:870	ATP7B	GuideToPharmacology	2024.1	blocker	1.458546423213736	IUPHAR.LIGAND:2547	iuphar.ligand:2547	MARGATOXIN	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.006723133	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	MyCancerGenome	20-Jun-17	inhibitor	1.165474011072658	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.010417155	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.5339763176511304	sparsentan	rxcui:2630535	SPARSENTAN	TRUE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.024721126	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	THIOPHENE	rxcui:154876	THIOPHENE	FALSE	FALSE	FALSE
KHK	hgnc:6315	KHK	PharmGKB	4/5/24	NULL	52.50767123569449	fructose	rxcui:4570	FRUCTOSE	TRUE	FALSE	FALSE
TSSK1B	hgnc:14968	TSSK1B	DTC	9/2/20	NULL	0.055622533	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.060492709	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1875273972703375	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.5527123287967841	DEHYDROXYMETHYLEPOXYQUINOMICIN	chembl:CHEMBL169300	DEHYDROXYMETHYLEPOXYQUINOMICIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	PARATHION	ncit:C163685	PARATHION	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.305277158	IUPHAR.LIGAND:7469	rxcui:274964	CICLESONIDE	TRUE	FALSE	FALSE
NCBIGENE:676	hgnc:1105	BRDT	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:12422	iuphar.ligand:12422	COHUMULONE	FALSE	FALSE	FALSE
PROSTAGLANDIN F2-ALPHA RECEPTOR	hgnc:9600	PTGFR	TTD	2020.06.01	NULL	3.750547945	BOL-303259-X	rxcui:1988390	LATANOPROSTENE BUNOD	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	ACETANILIDE	rxcui:162	ACETANILIDE	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.1161674142382621	GNF-PF-4576	chembl:CHEMBL527336	CHEMBL:CHEMBL527336	FALSE	FALSE	FALSE
PKN3	hgnc:17999	PKN3	MyCancerGenome	20-Jun-17	inhibitor	0.2215513554248712	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1400204566285186	TRIBUTYLTIN-OXIDE	chembl:CHEMBL511667	TRIBUTYLTIN-OXIDE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006574965	LIOTHYRONINE	rxcui:10814	LIOTHYRONINE	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.042898424	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
GUANYLYL CYCLASE C	hgnc:4688	GUCY2C	TTD	2020.06.01	NULL	19.69037671338543	Guanilib	rxcui:1873752	PLECANATIDE	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.2991890098899971	DARUISOLINE	chembl:CHEMBL2216904	DARUISOLINE	FALSE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.087222045	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
UNIPROT:P47712	hgnc:9035	PLA2G4A	TEND	1-Aug-11	NULL	0.3977853881492008	FLUNISOLIDE	rxcui:1546428	FLUNISOLIDE ANHYDROUS	TRUE	FALSE	FALSE
SLC47A1	hgnc:25588	SLC47A1	PharmGKB	4/5/24	NULL	1.500219178162699	trimethoprim	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-125110	chembl:CHEMBL580816	CHEMBL:CHEMBL580816	FALSE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	inhibitor	0.2059124362184098	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.01689436	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:1017	iuphar.ligand:1017	[125I]CATHEPSIN G (HUMAN)	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.029515273	S-ETOMIDATE	chembl:CHEMBL279678	S-ETOMIDATE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	OXAZEPAM	rxcui:7781	OXAZEPAM	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002421494	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.092443083	Sulfatinib	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:12717	iuphar.ligand:12717	I-BET282	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	inhibitor	0.027433475	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
PXN	hgnc:9718	PXN	NCI	14-Sep-17	NULL	0.6731752722524935	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	DIMETHYL GAMBOGATE	chembl:CHEMBL1436860	DIMETHYL GAMBOGATE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.021258166	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.3125456621172291	MP0112	iuphar.ligand:8371	ABICIPAR PEGOL	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.035098711	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	1.897867635025102	AVAPRITINIB	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.010588359	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
TNK2	hgnc:19297	TNK2	DTC	9/2/20	NULL	0.030073122	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	OncoKB	23-Jul-20	NULL	0.2025758921130189	Serabelisib	ncit:C98844	SERABELISIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	(S)-ROSCOVITINE	chembl:CHEMBL133342	(S)-ROSCOVITINE	FALSE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	0.6674703970639131	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.045898314	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.042516333	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.056826484	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
RPS26	hgnc:10414	RPS26	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	1.381780822	AZD-8165	drugbank:DB15132	AZD-8165	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	DNDI1417777	chembl:CHEMBL1412002	CHEMBL:CHEMBL1412002	FALSE	FALSE	FALSE
NOS2	hgnc:7873	NOS2	ChEMBL	33	inhibitor	1.419126249613364	GW-274150	drugbank:DB12237	GW-274150	FALSE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.08334551	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
NCBIGENE:1241	hgnc:6713	LTB4R	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5095	iuphar.ligand:5095	&ALPHA;-PROPYLDOPACETAMIDE	FALSE	FALSE	FALSE
NCBIGENE:597	hgnc:991	BCL2A1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8903	iuphar.ligand:8903	ZINC PROTOPORPHYRIN IX	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	DoCM	10-Apr-24	NULL	0.089103927	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.067897851	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:10579	iuphar.ligand:10579	ARD-266	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:440	iuphar.ligand:440	AS94	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1179947668217854	IUPHAR.LIGAND:10598	iuphar.ligand:10598	COMPOUND 41 [PMID: 31855425]	FALSE	FALSE	FALSE
NCBIGENE:2645	hgnc:4195	GCK	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:6838	rxcui:8130	PHENINDIONE	TRUE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.463302981	Rivoceranib	ncit:C152237	RIVOCERANIB	FALSE	FALSE	FALSE
CERAMIDE GLUCOSYLTRANSFERASE	hgnc:12524	UGCG	TTD	2020.06.01	NULL	5.250767123569449	Genz-682452	ncit:C152852	VENGLUSTAT	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	CIViC	10-Apr-24	NULL	0.099071078	PLX4720	drugbank:DB06999	PLX-4720	FALSE	FALSE	TRUE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.054695491	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
GABA(A) RECEPTOR GAMMA-3	hgnc:4088	GABRG3	TTD	2020.06.01	NULL	0.05814803	ALLOPREGNANOLONE	rxcui:2121777	BREXANOLONE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.017951341	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.4861821410712453	KX-02	iuphar.ligand:10004	KX2-361	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	PharmGKB	4/5/24	NULL	0.049723174	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
PKN2	hgnc:9406	PKN2	DTC	9/2/20	NULL	0.060984519	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.068847471	CARVEDILOL PHOSPHATE	rxcui:20352	CARVEDILOL	TRUE	FALSE	FALSE
NCBIGENE:467	hgnc:785	ATF3	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:3975	iuphar.ligand:3975	[125I]&ALPHA;-CONOTOXIN MII	FALSE	FALSE	FALSE
CD247	hgnc:1677	CD247	NCI	14-Sep-17	NULL	0.8751278539282418	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.012558639	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2063	iuphar.ligand:2063	[111IN]DOTA-BOC-ATE	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.2083637747448194	BESTATIN	ncit:C1015	UBENIMEX	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.1111273465305703	DIMETHYLCURCUMIN	drugbank:DB06133	DIMETHYLCURCUMIN	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.5707355569097228	ACTEIN	chembl:CHEMBL3391990	ACTEIN	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	4.375639269641208	(+)-TUBERIFERIN	chembl:CHEMBL1940084	CHEMBL:CHEMBL1940084	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	DTC	9/2/20	NULL	0.036770078	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.018443158	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
EYA4	hgnc:3522	EYA4	PharmGKB	4/5/24	NULL	0.5303805175322677	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	0.258658479	lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
NCBIGENE:1398	hgnc:2362	CRK	GuideToPharmacology	2024.1	inhibitor	0.3201687270469177	IUPHAR.LIGAND:11069	rxcui:5293	HEXACHLOROPHENE	TRUE	FALSE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8084	iuphar.ligand:8084	COMPOUND 1 [WO2012007375]	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	0.8078103267029924	IUPHAR.LIGAND:1514	iuphar.ligand:1514	PEPTIDE YY	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	3.850562557284263	PLERIXAFOR	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.038665443	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.2573905452730122	Oxyphencyclimine	rxcui:32698	OXYPHENCYCLIMINE	TRUE	FALSE	FALSE
SAE1	hgnc:30660	SAE1	DTC	9/2/20	NULL	3.281729452230906	GINGKOLIC ACID	chembl:CHEMBL445177	GINGKOLIC ACID	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	0.3571950424196904	Vecuronium	rxcui:11153	VECURONIUM BROMIDE	TRUE	FALSE	FALSE
NCBIGENE:71	hgnc:144	ACTG1	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:10679	rxcui:2664896	MOTIXAFORTIDE	TRUE	FALSE	FALSE
NCBIGENE:1362	hgnc:2301	CPD	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:10204	iuphar.ligand:10204	NORENDOXIFEN	FALSE	FALSE	FALSE
UNIPROT:P07766	hgnc:1674	CD3E	TdgClinicalTrial	Jan-14	NULL	0.729273212	MT110	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
UNIPROT:P04234	hgnc:1673	CD3D	TdgClinicalTrial	Jan-14	NULL	0.3281729452230906	VISILIZUMAB	ncit:C2229	VISILIZUMAB	FALSE	FALSE	FALSE
UNIPROT:Q16513	hgnc:9406	PKN2	TdgClinicalTrial	Jan-14	NULL	0.1562728310586145	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.5147810905460245	SIGNAL TRANSDUCTION INHIBITORS	ncit:C2189	SIGNAL TRANSDUCTION INHIBITOR	FALSE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.6455861217503421	DROSPIRENONE	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.1438566335224507	ENPIROLINE	ncit:C75267	ENPIROLINE	FALSE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	MyCancerGenome	20-Jun-17	other/unknown	0.760980743	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.016480751	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PHETA2	hgnc:27161	PHETA2	PharmGKB	4/5/24	NULL	6.563458904461812	dextromethorphan	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.040390516	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.1093909817410302	osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	CancerCommons	25-Jul-13	inhibitor	0.058471794	ODM-201	rxcui:2180325	DAROLUTAMIDE	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CGI	2/1/22	NULL	0.043636393	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
CCND2	hgnc:1583	CCND2	CGI	2/1/22	NULL	0.4286340509036285	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
FANCC	hgnc:3584	FANCC	CGI	2/1/22	NULL	0.1448487482363986	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ERCC6	hgnc:3438	ERCC6	CGI	2/1/22	NULL	0.036212187	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	CGI	2/1/22	NULL	0.8643238063488805	Lestaurtinib	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	CGI	2/1/22	NULL	0.1461794856227575	Arn-509	rxcui:1999574	APALUTAMIDE	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	NCI	14-Sep-17	NULL	0.108040476	17-AAG	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	CGI	2/1/22	NULL	0.009053047	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CGI	2/1/22	NULL	0.1520492410300034	BYL719	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	CGI	2/1/22	NULL	1.078924751	Larotrectinib	rxcui:2105628	LAROTRECTINIB	TRUE	FALSE	TRUE
TPMT	hgnc:12014	TPMT	CGI	2/1/22	NULL	0.2273059360852576	Thioguanine	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	agonist	0.7955707762984013	VASOPRESSIN TANNATE	chembl:CHEMBL1201528	VASOPRESSIN TANNATE	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.6364566210387211	EXENATIDE	rxcui:60548	EXENATIDE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	agonist	0.2365210416022274	METHACHOLINE CHLORIDE	rxcui:40165	METHACHOLINE CHLORIDE	TRUE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.097236428	IRINOTECAN HYDROCHLORIDE	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PLG	hgnc:9071	PLG	ChEMBL	33	activator	0.4688184931758437	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	ChEMBL	33	inhibitor	0.4526523382387456	DAUNORUBICIN CITRATE	rxcui:1364321	DAUNORUBICIN CITRATE	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	ChEMBL	33	inhibitor	1.186614039224734	PERINDOPRIL ERBUMINE	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
SSTR2	hgnc:11331	SSTR2	ChEMBL	33	agonist	0.729273212	PASIREOTIDE DIASPARTATE	rxcui:1364104	PASIREOTIDE DIASPARTATE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.2117244807890907	DEXBROMPHENIRAMINE MALEATE	rxcui:48936	DEXBROMPHENIRAMINE MALEATE	TRUE	FALSE	FALSE
GNRHR	hgnc:4421	GNRHR	ChEMBL	33	agonist	0.3977853881492007	LEUPROLIDE ACETATE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.1888765152363111	NILOTINIB HYDROCHLORIDE MONOHYDRATE	ncit:C95229	NILOTINIB HYDROCHLORIDE MONOHYDRATE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	0.596678082	ACEBUTOLOL HYDROCHLORIDE	rxcui:142130	ACEBUTOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.3977853881492006	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	agonist	0.1491695205559502	DOBUTAMINE HYDROCHLORIDE	rxcui:203121	DOBUTAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.091796628	DULOXETINE HYDROCHLORIDE	rxcui:476250	DULOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HRH2	hgnc:5183	HRH2	ChEMBL	33	inhibitor	0.8204323630577265	RANITIDINE HYDROCHLORIDE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PPIA	hgnc:9253	PPIA	ChEMBL	33	modulator	0.4310974649892816	CYCLOSPORINE	rxcui:3008	CYCLOSPORINE	TRUE	TRUE	FALSE
TSHR	hgnc:12373	TSHR	ChEMBL	33	agonist	0.2234368988752957	THYROTROPIN	rxcui:10579	THYROTROPIN	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	ChEMBL	33	activator	1.458546423213736	ENOXAPARIN SODIUM	rxcui:221095	ENOXAPARIN SODIUM	TRUE	FALSE	FALSE
TYR	hgnc:12442	TYR	ChEMBL	33	inhibitor	3.182283105193605	MONOBENZONE	rxcui:17145	MONOBENZONE	TRUE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	1.500219178	INSULIN PORK	rxcui:221109	INSULIN, REGULAR, PORK	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1635752997996713	DESIPRAMINE HYDROCHLORIDE	rxcui:203174	DESIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.051655358	AMPHETAMINE	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.6543011991986852	PHENTERMINE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.13086024	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
KCNJ8	hgnc:6269	KCNJ8	ChEMBL	33	potentiator	0.5048814541893702	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	0.5834185692854945	VARENICLINE TARTRATE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	agonist	0.8607814956671229	DYDROGESTERONE	rxcui:3706	DYDROGESTERONE	TRUE	FALSE	FALSE
GRIA1	hgnc:4571	GRIA1	ChEMBL	33	inhibitor	1.270346884734544	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	ChEMBL	33	inhibitor	0.9376369863516875	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	agonist	0.3351553483129436	VARENICLINE TARTRATE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	1.193356164447602	PERAMPANEL	rxcui:1356552	PERAMPANEL	TRUE	FALSE	FALSE
PDE4B	hgnc:8781	PDE4B	ChEMBL	33	inhibitor	0.1458546423213736	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	inhibitor	0.1305078821102597	NALTREXONE	rxcui:7243	NALTREXONE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.069454592	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.025613498	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.023336743	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
ABL1	hgnc:76	ABL1	ChEMBL	33	inhibitor	0.8008364246019593	PONATINIB HYDROCHLORIDE	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
GRIN3A	hgnc:16767	GRIN3A	ChEMBL	33	inhibitor	0.095295229	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.015964631	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.013836014	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
DRD5	hgnc:3026	DRD5	ChEMBL	33	inhibitor	0.1750255707856483	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.047518255	ERGOLOID MESYLATES	rxcui:4024	ERGOLOID MESYLATES, USP	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	inhibitor	0.018168744	PIMOZIDE	rxcui:8331	PIMOZIDE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	agonist	0.039068208	PERGOLIDE MESYLATE	rxcui:8048	PERGOLIDE MESYLATE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.4922594178346359	SUPROFEN	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
ADORA3	hgnc:268	ADORA3	ChEMBL	33	inhibitor	0.6908904109959803	CAFFEINE, CITRATED	rxcui:20033	CAFFEINE CITRATE	TRUE	FALSE	FALSE
EEF2	hgnc:3214	EEF2	ChEMBL	33	inhibitor	0.4861821410712453	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.2302968036653267	TROSPIUM CHLORIDE	rxcui:236778	TROSPIUM	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	agonist	0.3070624048871023	BETHANECHOL CHLORIDE	rxcui:47088	BETHANECHOL CHLORIDE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	DARUNAVIR ETHANOLATE	rxcui:644682	DARUNAVIR ETHANOLATE	TRUE	FALSE	FALSE
ADH1B	hgnc:250	ADH1B	ChEMBL	33	inhibitor	13.12691780892362	FOMEPIZOLE	rxcui:15226	FOMEPIZOLE	TRUE	FALSE	FALSE
PDE10A	hgnc:21160	LINC00473	ChEMBL	33	inhibitor	0.2500365296937833	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE6A	hgnc:8785	PDE6A	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE3B	hgnc:8779	PDE3B	ChEMBL	33	inhibitor	0.1250182648468916	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	ChEMBL	33	inhibitor	0.035719504	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.091796628	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.021997349	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.081407242	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.096050618	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.018430211	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.093763699	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.037666909	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.1562728310586145	ZALEPLON	rxcui:74667	ZALEPLON	TRUE	FALSE	FALSE
CACNG1	hgnc:1405	CACNG1	ChEMBL	33	modulator	0.1262203635473425	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNA1G	hgnc:1394	CACNA1G	ChEMBL	33	modulator	0.084146909	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNG6	hgnc:13625	CACNG6	ChEMBL	33	modulator	0.2243917574174979	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNB3	hgnc:1403	CACNB3	ChEMBL	33	modulator	0.1553481397505754	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNA1A	hgnc:1388	CACNA1A	ChEMBL	33	modulator	0.4039051633514961	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNG5	hgnc:1409	CACNG5	ChEMBL	33	modulator	0.2243917574174979	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CACNA1E	hgnc:1392	CACNA1E	ChEMBL	33	modulator	0.2019525816757481	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.054243462	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.056826484	BENOXINATE HYDROCHLORIDE	rxcui:235398	BENOXINATE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN4A	hgnc:10591	SCN4A	ChEMBL	33	blocker	0.080781033	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.082043236	HEXYLCAINE HYDROCHLORIDE	rxcui:1546032	HEXYLCAINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.040703621	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.076098074	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.029416062	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.012208247	CHLORPROMAZINE HYDROCHLORIDE	rxcui:104728	CHLORPROMAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	0.150021918	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	ChEMBL	33	agonist	0.073954467	HYDROXYAMPHETAMINE HYDROBROMIDE	rxcui:82066	HYDROXYAMPHETAMINE HYDROBROMIDE	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	ChEMBL	33	inhibitor	0.08334551	LOXAPINE SUCCINATE	rxcui:6476	LOXAPINE SUCCINATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.034590034	LOXAPINE SUCCINATE	rxcui:6476	LOXAPINE SUCCINATE	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	ChEMBL	33	agonist	0.1544343271638073	ROPINIROLE HYDROCHLORIDE	rxcui:236553	ROPINIROLE HYDROCHLORIDE	TRUE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.2573905452730122	TOBRAMYCIN SULFATE	rxcui:10627	TOBRAMYCIN	TRUE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	ChEMBL	33	blocker	0.4070362111294147	PHENSUXIMIDE	rxcui:33309	PHENSUXIMIDE	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	ChEMBL	33	agonist	0.112036283	ARIPIPRAZOLE LAUROXIL	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.5233322714521047	ROGARATINIB	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.069089041	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.1396480617970598	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.092443083	SURUFATINIB	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	ChEMBL	33	inhibitor	0.750109589	SOVLEPLENIB	ncit:C123912	SOVLEPLENIB	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.1562728310586145	SURUFATINIB	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.364636606	INK-1117	chembl:CHEMBL3545055	INK-1117	FALSE	FALSE	TRUE
PTK2	hgnc:9611	PTK2	ChEMBL	33	inhibitor	3.889457128569962	GSK-2256098	chembl:CHEMBL4742157	GSK-2256098	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	ChEMBL	33	inhibitor	0.3302369260106572	MK-8353	iuphar.ligand:9974	MK-8353	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	ChEMBL	33	inhibitor	0.098053541	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.092606122	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
CDK14	hgnc:8883	CDK14	ChEMBL	33	inhibitor	0.6250913242344582	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.1250182648468916	TAK-593	drugbank:DB13093	TAK-593	FALSE	FALSE	FALSE
HRH3	hgnc:5184	HRH3	ChEMBL	33	agonist	0.7721716358190367	CIPRALISANT MALEATE	ncit:C76885	CIPRALISANT MALEATE	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	0.6403374540938354	AMG-517	iuphar.ligand:4129	AMG517	FALSE	FALSE	FALSE
CDK3	hgnc:1772	CDK3	ChEMBL	33	inhibitor	0.3125456621172291	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.7143900848393808	REFAMETINIB	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.047712559	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
MAPK9	hgnc:6886	MAPK9	ChEMBL	33	inhibitor	0.2734774543525755	TANZISERTIB	ncit:C152510	TANZISERTIB	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	ChEMBL	33	inhibitor	0.025280535	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.05348829	ENMD-2076	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.097308509	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
TRPV1	hgnc:12716	TRPV1	ChEMBL	33	inhibitor	1.280674908	JTS-653	chembl:CHEMBL3545228	JTS-653	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	ChEMBL	33	inhibitor	3.150460274	MOTIXAFORTIDE	rxcui:2664896	MOTIXAFORTIDE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	agonist	0.108711535	RAPASTINEL	ncit:C152156	RAPASTINEL	FALSE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	ChEMBL	33	inhibitor	0.108711535	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.1209854175937661	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.2885036881082115	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	positive modulator	0.1209854175937661	NEBOGLAMINE	ncit:C66222	NEBOGLAMINE	FALSE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.2778183663264258	AV-101	drugbank:DB12878	AV-101	FALSE	FALSE	FALSE
CHRNB4	hgnc:1964	CHRNB4	ChEMBL	33	agonist	1.093909817410302	SIMPINICLINE	ncit:C179121	SIMPINICLINE	FALSE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	ChEMBL	33	inhibitor	0.4167275494896389	SELURAMPANEL	ncit:C152327	SELURAMPANEL	FALSE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	ChEMBL	33	inhibitor	0.8334550989792778	TEZAMPANEL	ncit:C77316	TEZAMPANEL	FALSE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	agonist	0.039068208	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.031254566	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.0701037	BRIVANIB ALANINATE	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.1579178082276526	BRIVANIB ALANINATE	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.089298761	BRIVANIB ALANINATE	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	inhibitor	0.4605936073306534	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.042516333	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.031317948	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ChEMBL	33	inhibitor	0.032492371	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ADORA2A	hgnc:263	ADORA2A	ChEMBL	33	inhibitor	2.128689374420047	TOZADENANT	ncit:C152704	TOZADENANT	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.2557191780959147	LUMATEPERONE	rxcui:2275602	LUMATEPERONE	TRUE	FALSE	FALSE
ITGA5	hgnc:6141	ITGA5	ChEMBL	33	inhibitor	4.375639269641208	VOLOCIXIMAB	ncit:C48426	VOLOCIXIMAB	FALSE	FALSE	TRUE
CA9	hgnc:1383	CA9	ChEMBL	33	other/unknown	1.250182648468916	GIRENTUXIMAB	ncit:C1960	GIRENTUXIMAB	FALSE	FALSE	FALSE
APP	hgnc:620	APP	ChEMBL	33	binder	2.423430980108977	SOLANEZUMAB	ncit:C88585	SOLANEZUMAB	FALSE	FALSE	FALSE
ITGB1	hgnc:6153	ITGB1	ChEMBL	33	inhibitor	4.375639269641208	VOLOCIXIMAB	ncit:C48426	VOLOCIXIMAB	FALSE	FALSE	TRUE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.042174836	LEXIBULIN	ncit:C77882	LEXIBULIN	FALSE	FALSE	FALSE
TNFRSF10B	hgnc:11905	TNFRSF10B	ChEMBL	33	agonist	5.834185692854944	CONATUMUMAB	ncit:C71015	CONATUMUMAB	FALSE	TRUE	TRUE
TGFB1	hgnc:11766	TGFB1	ChEMBL	33	inhibitor	0.4449802647092754	METELIMUMAB	ncit:C166745	METELIMUMAB	FALSE	FALSE	FALSE
IGF1	hgnc:5464	IGF1	ChEMBL	33	inhibitor	13.12691780892362	DUSIGITUMAB	ncit:C82683	DUSIGITUMAB	FALSE	FALSE	FALSE
IGF2	hgnc:5466	IGF2	ChEMBL	33	inhibitor	2.917092846427472	DUSIGITUMAB	ncit:C82683	DUSIGITUMAB	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	ChEMBL	33	inhibitor	0.4449802647092754	LY-2382770	chembl:CHEMBL2109585	LY-2382770	FALSE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	ChEMBL	33	inhibitor	6.563458904461812	ICM3	chembl:CHEMBL2109481	ICM3	FALSE	FALSE	FALSE
TNC	hgnc:5318	TNC	ChEMBL	33	binder	6.563458904461812	F16SIP 131I	chembl:CHEMBL2109584	F16SIP 131I	FALSE	FALSE	FALSE
CD4	hgnc:1678	CD4	ChEMBL	33	inhibitor	3.281729452230906	TRX-1	chembl:CHEMBL2109474	TRX-1	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	modulator	0.2869271652223742	CHLORMADINONE ACETATE	rxcui:2369	CHLORMADINONE ACETATE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.596678082	INDALPINE	ncit:C170063	INDALPINE	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.054695491	INDOPROFEN	ncit:C83801	INDOPROFEN	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.036463661	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
GABRE	hgnc:4085	GABRE	ChEMBL	33	positive modulator	0.042073455	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	METHAQUALONE	rxcui:6823	METHAQUALONE	TRUE	FALSE	FALSE
SCN5A	hgnc:10593	SCN5A	ChEMBL	33	blocker	0.1988926940746003	PRENYLAMINE	rxcui:8674	PRENYLAMINE	TRUE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	ChEMBL	33	binder	0.5469549087051511	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.072125922	SERTINDOLE	rxcui:41996	SERTINDOLE	TRUE	FALSE	FALSE
EPCAM	hgnc:11529	EPCAM	ChEMBL	33	modulator	1.260184109656668	CATUMAXOMAB	ncit:C62445	CATUMAXOMAB	TRUE	FALSE	TRUE
TNFRSF10B	hgnc:11905	TNFRSF10B	ChEMBL	33	agonist	17.50255707856483	LBY-135	chembl:CHEMBL2109247	LBY-135	FALSE	TRUE	TRUE
EPHA3	hgnc:3387	EPHA3	ChEMBL	33	inhibitor	11.66837138570988	KB-004	chembl:CHEMBL2109398	KB-004	FALSE	FALSE	FALSE
FN1	hgnc:3778	FN1	ChEMBL	33	binder	4.039051633514961	AS-1409	chembl:CHEMBL2109413	AS-1409	FALSE	FALSE	FALSE
CD3D	hgnc:1673	CD3D	ChEMBL	33	modulator	0.4102161815288632	FBT-A05	chembl:CHEMBL2109351	FBT-A05	FALSE	FALSE	FALSE
CD3E	hgnc:1674	CD3E	ChEMBL	33	modulator	0.364636606	FBT-A05	chembl:CHEMBL2109351	FBT-A05	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	ChEMBL	33	inhibitor	0.4688184931758437	CAPIVASERTIB	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	OMADACYCLINE TOSYLATE	rxcui:2059268	OMADACYCLINE TOSYLATE	TRUE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.9546849315580818	DAPIVIRINE	ncit:C73205	DAPIVIRINE	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	ChEMBL	33	inhibitor	0.3125456621172291	SELUMETINIB SULFATE	rxcui:2361596	SELUMETINIB SULFATE	TRUE	FALSE	FALSE
PSMC4	hgnc:9551	PSMC4	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
GCGR	hgnc:4192	GCGR	ChEMBL	33	agonist	1.312691780892362	COTADUTIDE	ncit:C174890	COTADUTIDE	FALSE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.2386712328895204	DIFAMILAST	ncit:C169909	DIFAMILAST	FALSE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	ChEMBL	33	inhibitor	3.088686543276147	MK-0736	drugbank:DB15209	MK-0736	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.3621218705909966	DIFAMILAST	ncit:C169909	DIFAMILAST	FALSE	FALSE	FALSE
RPS27	hgnc:10416	RPS27	ChEMBL	33	inhibitor	0.092606122	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPS9	hgnc:10442	RPS9	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL3	hgnc:10332	RPL3	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL9P7	hgnc:30335	RPL9P7	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL36A	hgnc:10359	RPL36A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL35A	hgnc:10345	RPL35A	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	ChEMBL	33	agonist	0.1591141552596802	COTADUTIDE	ncit:C174890	COTADUTIDE	FALSE	FALSE	FALSE
HCRTR1	hgnc:4848	HCRTR1	ChEMBL	33	inhibitor	2.917092846427472	ALMOREXANT	ncit:C87423	ALMOREXANT	FALSE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	NCI	14-Sep-17	NULL	0.06390386	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HCRTR2	hgnc:4849	HCRTR2	ChEMBL	33	inhibitor	2.386712328895204	ALMOREXANT	ncit:C87423	ALMOREXANT	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	modulator	0.039068208	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.042174836	KOS-1584	drugbank:DB05903	KOS-1584	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	modulator	0.039538909	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
PRIM1	hgnc:9369	PRIM1	ChEMBL	33	inhibitor	0.6819178082557728	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	CETHROMYCIN	ncit:C83613	CETHROMYCIN	FALSE	FALSE	FALSE
PRIM2	hgnc:9370	PRIM2	ChEMBL	33	inhibitor	0.7955707762984016	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.1367387271762877	GS-9256	drugbank:DB12876	GS-9256	FALSE	FALSE	FALSE
ELANE	hgnc:3309	ELANE	ChEMBL	33	inhibitor	2.282942227638891	.ALPHA.1-PROTEINASE INHIBITOR HUMAN	chembl:CHEMBL4297879	.ALPHA.1-PROTEINASE INHIBITOR HUMAN	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	agonist	0.039068208	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.4861821410712453	INAVOLISIB	ncit:C132166	INAVOLISIB	FALSE	FALSE	TRUE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	agonist	0.03729238	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	agonist	0.044347695	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
SI	hgnc:10856	SI	NCI	14-Sep-17	NULL	0.1526385791735305	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PTGER4	hgnc:9596	PTGER4	ChEMBL	33	inhibitor	1.544343271638073	GRAPIPRANT	rxcui:1862951	GRAPIPRANT	FALSE	FALSE	FALSE
APCS	hgnc:584	APCS	ChEMBL	33	inhibitor	6.563458904461812	DEZAMIZUMAB	ncit:C153210	DEZAMIZUMAB	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	positive modulator	1.117184494376478	TAK-071	iuphar.ligand:12302	TAK-071	FALSE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	ChEMBL	33	inhibitor	0.5357925636295356	TILARGININE	ncit:C1178	TILARGININE	FALSE	FALSE	FALSE
HTR3A	hgnc:5297	HTR3A	ChEMBL	33	inhibitor	0.1555782851427985	TROPISETRON	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
ACACB	hgnc:85	ACACB	ChEMBL	33	inhibitor	0.8468979231563628	OLUMACOSTAT GLASARETIL	ncit:C166791	OLUMACOSTAT GLASARETIL	FALSE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	ChEMBL	33	inhibitor	0.5048814541893701	FARICIMAB	rxcui:2591519	FARICIMAB	TRUE	FALSE	FALSE
SI	hgnc:10856	SI	NCI	14-Sep-17	NULL	0.2476776945079929	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
GHSR	hgnc:4267	GHSR	ChEMBL	33	inverse agonist	2.917092846427472	PF-5190457	drugbank:DB14870	PF-5190457	FALSE	FALSE	FALSE
ADRB1	hgnc:285	ADRB1	ChEMBL	33	inhibitor	1.790034246671403	PRACTOLOL	rxcui:8620	PRACTOLOL	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	ChEMBL	33	inhibitor	0.5585922471882393	NOLATREXED	ncit:C143088	NOLATREXED	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.064824285	NINGETINIB	drugbank:DB16256	NINGETINIB	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.073954467	NINGETINIB	drugbank:DB16256	NINGETINIB	FALSE	FALSE	FALSE
JAK1	hgnc:6190	JAK1	ChEMBL	33	inhibitor	1.693795846312725	AZD4205	chembl:CHEMBL4577523	AZD4205	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	1.463203610631835	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.1842374429322613	FGFR INHIBITOR DEBIO 1347	chembl:CHEMBL3907479	FGFR INHIBITOR DEBIO 1347	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	ChEMBL	33	inhibitor	0.039538909	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
TYR	hgnc:12442	TYR	ChEMBL	33	inhibitor	4.773424657790408	ARBUTIN	rxcui:1367175	ARBUTIN	TRUE	FALSE	FALSE
FGG	hgnc:3694	FGG	ChEMBL	33	cleavage	4.375639269641208	ALFIMEPRASE	ncit:C79877	ALFIMEPRASE	FALSE	FALSE	FALSE
NAMPT	hgnc:30092	NAMPT	ChEMBL	33	inhibitor	21.00306849427779	DAPORINAD	ncit:C67043	DAPORINAD	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.035902681	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
IL2RB	hgnc:6009	IL2RB	ChEMBL	33	binder	1.346350544504987	SIMLUKAFUSP ALFA	ncit:C129383	SIMLUKAFUSP ALFA	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.04907259	DOTHIEPIN	rxcui:3634	DOTHIEPIN	TRUE	FALSE	FALSE
SNAP25	hgnc:11132	SNAP25	NCI	14-Sep-17	NULL	1.346350544504987	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
PNP	hgnc:7892	PNP	ChEMBL	33	inhibitor	17.50255707856483	ULODESINE	ncit:C152793	ULODESINE	FALSE	FALSE	FALSE
HDAC2	hgnc:4853	HDAC2	ChEMBL	33	inhibitor	0.056826484	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	NCI	14-Sep-17	NULL	0.1110098757625676	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
TNNI2	hgnc:11946	TNNI2	ChEMBL	33	activator	8.751278539282415	RELDESEMTIV	ncit:C166781	RELDESEMTIV	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
P2RX3	hgnc:8534	P2RX3	ChEMBL	33	inhibitor	26.25383561784724	CAMLIPIXANT	ncit:C190487	CAMLIPIXANT	FALSE	FALSE	FALSE
CALCRL	hgnc:16709	CALCRL	ChEMBL	33	inhibitor	1.750255707856483	ZAVEGEPANT	rxcui:2637955	ZAVEGEPANT	TRUE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	NCI	14-Sep-17	NULL	0.2210849315187136	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
IL10RA	hgnc:5964	IL10RA	ChEMBL	33	agonist	13.12691780892362	PEGILODECAKIN	ncit:C113295	PEGILODECAKIN	FALSE	FALSE	FALSE
CDKN2A	hgnc:1787	CDKN2A	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.5609793935437446	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.016086909	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.1143957978991165	XL-147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.2375912725597036	XL-147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	ClearityFoundationBiomarkers	26-Jul-13	NULL	0.062608511	XL-147	ncit:C71705	PILARALISIB	FALSE	FALSE	TRUE
SLPI	hgnc:11092	SLPI	NCI	14-Sep-17	NULL	1.640864726115453	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
SPARC	hgnc:11219	SPARC	ClearityFoundationBiomarkers	26-Jul-13	NULL	13.12691780892362	NAB-PACLITAXEL	ncit:C2688	NAB-PACLITAXEL	FALSE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2545826484154885	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
RPS6KB1	hgnc:10436	RPS6KB1	DTC	9/2/20	NULL	0.2027323213733378	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	AUSTOCYSTIN D	chembl:CHEMBL1966436	AUSTOCYSTIN D	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.061628722	CEFUROXIME SODIUM	rxcui:204144	CEFUROXIME SODIUM	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.015777545	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.060772768	2-AMINO-ANTHRAQUINONE	chembl:CHEMBL84685	CHEMBL:CHEMBL84685	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.005339401	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
S1PR4	hgnc:3170	S1PR4	DTC	9/2/20	NULL	0.5834185692854945	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	DTC	9/2/20	NULL	0.1302273592155121	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	D,L-ARMEPAVINE	chembl:CHEMBL451722	CHEMBL:CHEMBL451722	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	CRYPTOCHINONE A	chembl:CHEMBL1223740	CRYPTOCHINONE A	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	NSC-693571	chembl:CHEMBL1287983	CHEMBL:CHEMBL1287983	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	METIPRANOLOL	rxcui:10824	METIPRANOLOL	TRUE	FALSE	FALSE
SOAT1	hgnc:11177	SOAT1	NCI	14-Sep-17	NULL	0.596678082	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
SST	hgnc:11329	SST	NCI	14-Sep-17	NULL	0.057291513	ACETYLSALICYLIC ACID	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
EIF2AK1	hgnc:24921	EIF2AK1	DTC	9/2/20	NULL	105.0153424713889	TCMDC-123956	chembl:CHEMBL534675	CHEMBL:CHEMBL534675	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.076765601	LY-255283	chembl:CHEMBL15766	LY-255283	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	3,5 DIBROMOTYROSINE	chembl:CHEMBL1232132	DIBROMOTYROSINE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.016829382	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.01186614	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004919212	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.0136917	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.005847179	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1060761035064535	TCMDC-137788	chembl:CHEMBL587564	CHEMBL:CHEMBL587564	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.021590325	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
PSMB7	hgnc:9544	PSMB7	DTC	9/2/20	NULL	0.5834185692854944	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMC6	hgnc:9553	PSMC6	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD2	hgnc:9559	PSMD2	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB1	hgnc:9537	PSMB1	DTC	9/2/20	NULL	0.6250913242344582	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB11	hgnc:31963	PSMB11	DTC	9/2/20	NULL	0.4375639269641209	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMD12	hgnc:9557	PSMD12	DTC	9/2/20	NULL	0.7001022831425934	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB5	hgnc:9542	PSMB5	DTC	9/2/20	NULL	0.5250767123569451	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
PSMB8	hgnc:9545	PSMB8	DTC	9/2/20	NULL	0.3182283105193606	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.050978322	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
PIM3	hgnc:19310	PIM3	DTC	9/2/20	NULL	0.02617531	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.017799211	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1988926940746003	NSC-339578	chembl:CHEMBL353764	CHEMBL:CHEMBL353764	FALSE	FALSE	FALSE
TFPI2	hgnc:11761	TFPI2	NCI	14-Sep-17	NULL	1.640864726115453	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.042516333	(S)-ROSCOVITINE	chembl:CHEMBL133342	(S)-ROSCOVITINE	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.009003373	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
ENPP2	hgnc:3357	ENPP2	DTC	9/2/20	NULL	17.50255707856483	NSC-34937	chembl:CHEMBL1092743	CHEMBL:CHEMBL1092743	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.004373453	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.1067229090156392	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006258861	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1810609352954982	DIETHYLSTILBESTROL DIPROPIONATE	ncit:C74557	DIETHYLSTILBESTROL DIPROPIONATE	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008503267	PAROXETINE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	THIOINOSINE	ncit:C877	THIOINOSINE	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003497713	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
TERT	hgnc:11730	TERT	NCI	14-Sep-17	NULL	0.2143170254518142	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
PKM	hgnc:9021	PKM	DTC	9/2/20	NULL	0.1121958787087489	AMLEXANOX	rxcui:46307	AMLEXANOX	TRUE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	DTC	9/2/20	NULL	0.005787883	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GANAB	hgnc:4138	GANAB	DTC	9/2/20	NULL	35.00511415712966	MIGLUSTAT	rxcui:402316	MIGLUSTAT	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.3804903712731485	AMINEPTINE	rxcui:17698	AMINEPTIN	TRUE	FALSE	FALSE
CLK1	hgnc:2068	CLK1	DTC	9/2/20	NULL	1.400204566285186	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.5645986154375752	BISPECIFIC ANTIBODY	ncit:C1454	BISPECIFIC ANTIBODY	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	TCMDC-123868	chembl:CHEMBL548615	CHEMBL:CHEMBL548615	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.015193192	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.061773731	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	DTC	9/2/20	NULL	0.008240375	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
HDAC4	hgnc:14063	HDAC4	DTC	9/2/20	NULL	0.175610941	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.008651783	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	CEPHALOSPORIN C ZINC SALT	chembl:CHEMBL1326149	CEPHALOSPORIN C ZINC SALT	FALSE	FALSE	FALSE
STK3	hgnc:11406	STK3	DTC	9/2/20	NULL	0.051226996	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.071196842	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
TLR7	hgnc:15631	TLR7	DTC	9/2/20	NULL	1.969037671338543	RESIQUIMOD	ncit:C63958	RESIQUIMOD	FALSE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	DTC	9/2/20	NULL	1.400204566285186	ISOSILYBIN A	chembl:CHEMBL592676	ISOSILYBIN A	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-123811	chembl:CHEMBL587433	CHEMBL:CHEMBL587433	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	(-)-THALIPORPHINE	chembl:CHEMBL1394328	CHEMBL:CHEMBL1394328	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.019776901	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.018540844	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.375054795	ROEMERINE	chembl:CHEMBL36654	ROEMERINE	FALSE	FALSE	FALSE
XPO1	hgnc:12825	XPO1	DTC	9/2/20	NULL	17.50255707856483	LEPTOMYCIN B	chembl:CHEMBL486133	LEPTOMYCIN B	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.010537361	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.086861325	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SCARLET RED	rxcui:36224	SCARLET RED	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.016916131	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.729273212	CEFAMANDOLE	rxcui:2178	CEFAMANDOLE	TRUE	FALSE	FALSE
OPN1LW	hgnc:9936	OPN1LW	DTC	9/2/20	NULL	21.00306849427779	RHODOPSIN	iuphar.ligand:6669	11-CIS-RETINAL	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.120017534	DEMETHYLWEDELOLACTONE	chembl:CHEMBL2089002	DEMETHYLWEDELOLACTONE	FALSE	FALSE	FALSE
CNR2	hgnc:2160	CNR2	DTC	9/2/20	NULL	0.1442518440541057	WIN-552122	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
NCOA3	hgnc:7670	NCOA3	DTC	9/2/20	NULL	0.2187819634820604	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	CP-55940	iuphar.ligand:730	CP55940	FALSE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	MOROLIC ACID	chembl:CHEMBL463665	MOROLIC ACID	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.009349657	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	DIPHENOXYLATE HYDROCHLORIDE	rxcui:82005	DIPHENOXYLATE HYDROCHLORIDE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.057322785	DNDI1417147	chembl:CHEMBL2094484	CHEMBL:CHEMBL2094484	FALSE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	NCI	14-Sep-17	NULL	0.1691068316769549	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
MAPK9	hgnc:6886	MAPK9	DTC	9/2/20	NULL	0.013905633	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	BROMOXYNIL	chembl:CHEMBL453905	BROMOXYNIL	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002594637	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.015407181	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	CHLORZOXAZONE	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.028661393	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	PHENFORMIN HYDROCHLORIDE	rxcui:235288	PHENFORMIN HYDROCHLORIDE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.014504882	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006570029	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
TK2	hgnc:11831	TK2	NCI	14-Sep-17	NULL	17.50255707856483	DDC	rxcui:3363	ZALCITABINE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	OXIBENDAZOLE	rxcui:1009342	OXIBENDAZOLE	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.022632617	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1635752997996713	PUERARIN	drugbank:DB12290	PUERARIN	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	DTC	9/2/20	NULL	0.007818295	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	GNF-PF-4370	chembl:CHEMBL600971	CHEMBL:CHEMBL600971	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1640864726115453	CETRIMONIUM BROMIDE	rxcui:288999	CETRIMONIUM BROMIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003053304	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.3182283105193606	CETRIMONIUM BROMIDE	rxcui:288999	CETRIMONIUM BROMIDE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.01535312	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
P4HA1	hgnc:8546	P4HA1	DTC	9/2/20	NULL	35.00511415712966	PYRIDINE-2,5-DICARBOXYLIC ACID	chembl:CHEMBL88972	PYRIDINE-2,5-DICARBOXYLIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	chembl:CHEMBL1449651	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	FALSE	FALSE	FALSE
ACVR1	hgnc:171	ACVR1	DTC	9/2/20	NULL	0.021189536	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.055859225	AMBUNOL	chembl:CHEMBL454893	AMBUNOL	FALSE	FALSE	FALSE
TMSB10	hgnc:11879	TMSB10	NCI	14-Sep-17	NULL	2.822993077187876	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	BETAXOLOL HYDROCHLORIDE	rxcui:142144	BETAXOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.033148782	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	HERACLENOL	chembl:CHEMBL1173444	HERACLENOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	NSC-11437	chembl:CHEMBL1814509	CHEMBL:CHEMBL1814509	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.150021918	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.010128795	(S)-ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	NAPHTHALEN-1-YLAMINE	chembl:CHEMBL57394	CHEMBL:CHEMBL57394	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.01609924	CHLORPROPAMIDE	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
TJP1	hgnc:11827	TJP1	NCI	14-Sep-17	NULL	0.305277158	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	AP-7	chembl:CHEMBL274440	AP-7	FALSE	FALSE	FALSE
SYK	hgnc:11491	SYK	DTC	9/2/20	NULL	0.012713722	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.029170928	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.005778964	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007937668	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
PLIN1	hgnc:9076	PLIN1	DTC	9/2/20	NULL	1.458546423213736	SUFENTANIL CITRATE	rxcui:58964	SUFENTANIL CITRATE	TRUE	FALSE	FALSE
MARK2	hgnc:3332	MARK2	DTC	9/2/20	NULL	0.031254566	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.026385764	SHIKONIN	chembl:CHEMBL9470	SHIKONIN	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1154014752432846	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	NSC-11437	chembl:CHEMBL1814509	CHEMBL:CHEMBL1814509	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.212581665	ALPHA-SOLANINE	chembl:CHEMBL1392894	CHEMBL:CHEMBL1392894	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	SULFAPHENAZOLE	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.150021918	3,3'-DIMETHOXYBENZIDINE	chembl:CHEMBL398363	CHEMBL:CHEMBL398363	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.010824092	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
RUNX1	hgnc:10471	RUNX1	DTC	9/2/20	NULL	0.1154014752432846	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.0135995	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.021805511	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
THRSP	hgnc:11800	THRSP	NCI	14-Sep-17	NULL	0.305277158	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CDC25C	hgnc:1727	CDC25C	DTC	9/2/20	NULL	2.187819634820604	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	0.082364974	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.029515273	IOBENGUANE	ncit:C87757	IOBENGUANE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.08178765	TRIS(2,3-DIBROMOPROPYL)PHOSPHATE	chembl:CHEMBL1904600	TRIS(2,3-DIBROMOPROPYL)PHOSPHATE	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.068169648	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.069454592	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.092933931	ROEMERINE	chembl:CHEMBL36654	ROEMERINE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.015416228	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW819077X	chembl:CHEMBL189415	GW819077X	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.192335792	AZITHROMYCIN	rxcui:18631	AZITHROMYCIN	TRUE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.02534154	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	MRS-2179	iuphar.ligand:1720	MRS2179	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.028413242	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.005065374	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.028490326	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
SHH	hgnc:10848	SHH	DTC	9/2/20	NULL	6.563458904461812	VISMODEGIB	rxcui:1242987	VISMODEGIB	TRUE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	CP-339818	iuphar.ligand:2558	CP-339818	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.3387591692625452	NSC-645827	chembl:CHEMBL95704	CHEMBL:CHEMBL95704	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.089756703	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1315981735230438	BAZEDOXIFENE ACETATE	rxcui:1442171	BAZEDOXIFENE ACETATE	TRUE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.020869504	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.2651902587661338	RAFOXANIDE	ncit:C152146	RAFOXANIDE	FALSE	FALSE	FALSE
S1PR1	hgnc:3165	S1PR1	DTC	9/2/20	NULL	0.1620607136904151	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	CALCIPOTRIENE	rxcui:29365	CALCIPOTRIENE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.210030685	AMORFRUTIN A	chembl:CHEMBL491820	AMORFRUTIN A	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.004068785	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	SILVER SULFADIAZINE	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
XRCC5	hgnc:12833	XRCC5	NCI	14-Sep-17	NULL	0.1034633915974275	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	DNDI1417032	chembl:CHEMBL1523974	CHEMBL:CHEMBL1523974	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.040452751	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	LUZINDOLE	iuphar.ligand:1363	LUZINDOLE	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.003057215	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.011575765	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.021172448	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.2853677784548614	1,3-DIPHENYLTHIOUREA	chembl:CHEMBL275260	CHEMBL:CHEMBL275260	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.063415062	MITOTANE	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.017243899	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	3-HYDROXYCOUMARIN	chembl:CHEMBL150372	3-HYDROXYCOUMARIN	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	DTC	9/2/20	NULL	0.546954909	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	CYSTEAMINE HYDROCHLORIDE	rxcui:1426886	CYSTEAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00808059	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
XIAP	hgnc:592	XIAP	NCI	14-Sep-17	NULL	0.1666910197958555	FLAVOPIRIDOL	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.1902451856365742	OPHIOBOLIN O	chembl:CHEMBL1934283	OPHIOBOLIN O	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.012454381	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001851731	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.059667808	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
KRAS	hgnc:6407	KRAS	OncoKB	23-Jul-20	NULL	0.9845188356692719	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
GRIA1	hgnc:4571	GRIA1	DTC	9/2/20	NULL	0.6775183385250904	PIRACETAM	rxcui:8351	PIRACETAM	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	OncoKB	23-Jul-20	NULL	0.8649519486500064	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.2051080907644316	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.1396480617970598	CP-339818	iuphar.ligand:2558	CP-339818	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.020117882	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	OSAJIN	chembl:CHEMBL238188	OSAJIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004660306	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.061628722	ISOORIENTIN	chembl:CHEMBL239559	ISOORIENTIN	FALSE	FALSE	FALSE
APOBEC3A	hgnc:17343	APOBEC3A	DTC	9/2/20	NULL	0.7721716358190367	SJ000040549	chembl:CHEMBL589421	CHEMBL:CHEMBL589421	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	RAFOXANIDE	ncit:C152146	RAFOXANIDE	FALSE	FALSE	FALSE
PSMD14	hgnc:16889	PSMD14	DTC	9/2/20	NULL	0.6731752722524935	AG-528	chembl:CHEMBL56542	CHEMBL:CHEMBL56542	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004207345	AMIODARONE HYDROCHLORIDE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	ARBACLOFEN	ncit:C90890	ARBACLOFEN	FALSE	FALSE	FALSE
RNASEL	hgnc:10050	RNASEL	DTC	9/2/20	NULL	52.50767123569449	C-5966451	chembl:CHEMBL259819	CHEMBL:CHEMBL259819	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.008118069	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	TCMDC-124468	chembl:CHEMBL1376851	CHEMBL:CHEMBL1376851	FALSE	FALSE	FALSE
XPA	hgnc:12814	XPA	NCI	14-Sep-17	NULL	5.834185692854945	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
ACP1	hgnc:122	ACP1	DTC	9/2/20	NULL	0.9546849315580819	GNF-PF-3542	chembl:CHEMBL598477	CHEMBL:CHEMBL598477	FALSE	FALSE	FALSE
GABRA1	hgnc:4075	GABRA1	DTC	9/2/20	NULL	0.4070362111294147	ISOPIMARIC ACID	chembl:CHEMBL512164	ISOPIMARIC ACID	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.002565104	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	NSC-209931	chembl:CHEMBL472656	CHEMBL:CHEMBL472656	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.009562497	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	NSC-326757	chembl:CHEMBL1368535	CHEMBL:CHEMBL1368535	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	METIZOLINE	ncit:C99577	METIZOLINE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.095122593	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	(S)-NIMODIPINE	chembl:CHEMBL255033	(S)-NIMODIPINE	FALSE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	NCI	14-Sep-17	NULL	1.193356164447602	PLATINUM	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
HSD11B1	hgnc:5208	HSD11B1	DTC	9/2/20	NULL	6.177373086552294	3-EPICOROSOLIC ACID METHYL ESTER	chembl:CHEMBL604538	CHEMBL:CHEMBL604538	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.2792961235941196	NSC-21588	chembl:CHEMBL1611308	CHEMBL:CHEMBL1611308	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.01759051	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	DTC	9/2/20	NULL	0.1715936968486748	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	PYRIPROXYFEN	chembl:CHEMBL1883234	PYRIPROXYFEN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.011124507	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007292732	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	GRAMINE	ncit:C64181	GRAMINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001914661	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.072324616	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.03821519	DITHIAZANINE	ncit:C72743	DITHIAZANINE	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	OncoKB	23-Jul-20	NULL	0.7369497717290455	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	0.1000146118775133	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
HDAC10	hgnc:18128	HDAC10	DTC	9/2/20	NULL	0.2651902587661338	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
GPR17	hgnc:4471	GPR17	DTC	9/2/20	NULL	26.25383561784724	9BETA-D-ARABINOFURANOSYLGUANOSINE 5'-TRIPHOSPHATE	chembl:CHEMBL1201369	GTP	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.026385764	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.023440925	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.014993624	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	DTC	9/2/20	NULL	0.2328499833068492	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	OncoKB	23-Jul-20	NULL	0.2778183663264258	Alpelisib	rxcui:2169285	ALPELISIB	TRUE	FALSE	TRUE
DPP4	hgnc:3009	DPP4	DTC	9/2/20	NULL	2.100306849	VALACYCLOVIR	rxcui:73645	VALACYCLOVIR	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	DTC	9/2/20	NULL	0.009173248	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.2580229544751573	BML-210	chembl:CHEMBL324053	CHEMBL:CHEMBL324053	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004195244	PROPAFENONE HYDROCHLORIDE	rxcui:203135	PROPAFENONE HYDROCHLORIDE	TRUE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.210030685	SJ000114961	chembl:CHEMBL590168	CHEMBL:CHEMBL590168	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.017799211	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.017859752	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.014883127	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.09972967	OMARIGLIPTIN	ncit:C174662	OMARIGLIPTIN	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	OncoKB	23-Jul-20	NULL	0.2540693769469088	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.062212881	GNF-PF-2713	chembl:CHEMBL578719	CHEMBL:CHEMBL578719	FALSE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.012974468	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	HYDROCORTISONE ACETATE	rxcui:27197	HYDROCORTISONE ACETATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.018619742	3,4-DICHLOROISOCOUMARIN	drugbank:DB04459	3,4-DICHLOROISOCOUMARIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	GNF-PF-3266	chembl:CHEMBL581869	CHEMBL:CHEMBL581869	FALSE	FALSE	FALSE
HEXA	hgnc:4878	HEXA	DTC	9/2/20	NULL	10.50153424713889	TCMDC-124296	chembl:CHEMBL22148	CHEMBL:CHEMBL22148	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.030038714	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	DTC	9/2/20	NULL	0.020510809	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.025439763	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.1367387271762877	GW632580X	iuphar.ligand:5685	GW-2580	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	TCMDC-124340	chembl:CHEMBL580516	CHEMBL:CHEMBL580516	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	6-HYDROXYMELATONIN	iuphar.ligand:1347	6-HYDROXYMELATONIN	FALSE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.040112812	MIBEFRADIL	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.014114965	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-630812	chembl:CHEMBL237570	CHEMBL:CHEMBL237570	FALSE	FALSE	FALSE
CACNA1H	hgnc:1395	CACNA1H	DTC	9/2/20	NULL	1.221108633388244	DNDI1417957	chembl:CHEMBL1570199	CHEMBL:CHEMBL1570199	FALSE	FALSE	FALSE
ELANE	hgnc:3309	ELANE	DTC	9/2/20	NULL	3.804903712731485	SIVELESTAT	ncit:C66539	SIVELESTAT	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005208578	DIGOXIN	rxcui:3407	DIGOXIN	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.031032903	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.02926849	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	CID 650707	chembl:CHEMBL408653	CHEMBL:CHEMBL408653	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.016286499	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	DNDI1417097	chembl:CHEMBL1531222	CHEMBL:CHEMBL1531222	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.007548544	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	GNF-PF-1083	chembl:CHEMBL530361	CHEMBL:CHEMBL530361	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.019844169	2-HYDROXYESTRADIOL	ncit:C120474	2-HYDROXYESTRADIOL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.001608691	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.3621218705909965	DNDI1417171	chembl:CHEMBL1438389	CHEMBL:CHEMBL1438389	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	SJ000059269	chembl:CHEMBL590686	CHEMBL:CHEMBL590686	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	GNF-PF-2713	chembl:CHEMBL578719	CHEMBL:CHEMBL578719	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	(1R)-TRANS-TETRAMETHRIN	chembl:CHEMBL1892154	(1R)-TRANS-TETRAMETHRIN	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.018006746	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.1325951293830669	XANTHYLETIN	chembl:CHEMBL303846	XANTHYLETIN	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.048083948	TCMDC-123764	chembl:CHEMBL533226	CHEMBL:CHEMBL533226	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.027577558	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	DTC	9/2/20	NULL	0.6250913242344582	RO-5068760	chembl:CHEMBL1956073	CHEMBL:CHEMBL1956073	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.013727496	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.069546584	GNF-PF-1083	chembl:CHEMBL530361	CHEMBL:CHEMBL530361	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.070197421	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.023440925	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.017541538	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	TCMDC-124353	chembl:CHEMBL529918	CHEMBL:CHEMBL529918	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.3125456621172291	ZINC 02849675	chembl:CHEMBL605959	CHEMBL:CHEMBL605959	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.012067955	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.9293393139060973	SOLOMONSTEROL B	chembl:CHEMBL1649713	SOLOMONSTEROL B	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.012713722	ANDROSTENEDIONE	rxcui:784	ANDROSTENEDIONE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	CL-976	chembl:CHEMBL22373	CL-976	FALSE	FALSE	FALSE
ALOX12	hgnc:429	ALOX12	DTC	9/2/20	NULL	0.067751834	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.007955708	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.064824285	CID 650707	chembl:CHEMBL408653	CHEMBL:CHEMBL408653	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.1479089330582944	U-50488 METHANE SULFONATE	iuphar.ligand:1652	U50488	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	TUBERCIDIN	ncit:C911	TUBERCIDIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	TETRAPHENYL-UREA	chembl:CHEMBL169335	CHEMBL:CHEMBL169335	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	PITTSBURGH COMPOUND B	drugbank:DB15161	PITTSBURGH COMPOUND B	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	BENZAMIL	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
SENP8	hgnc:22992	SENP8	DTC	9/2/20	NULL	0.2187819634820604	IPRIFLAVONE	rxcui:51487	IPRIFLAVONE	FALSE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.026319635	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.021484317	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.065964411	AVOBENZONE	rxcui:45045	AVOBENZONE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001012645	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.1367387271762877	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	3.281729452230906	STROBOPININ	chembl:CHEMBL1556958	STROBOPININ	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003439517	EXEMESTANE	rxcui:258494	EXEMESTANE	TRUE	FALSE	TRUE
EPHA2	hgnc:3386	EPHA2	DTC	9/2/20	NULL	0.039960176	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	1,2-BENZANTHRACENE	chembl:CHEMBL1873684	CHEMBL:CHEMBL1873684	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.017643707	BRIMONIDINE	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.014126358	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.1029562181092048	AG-528	chembl:CHEMBL56542	CHEMBL:CHEMBL56542	FALSE	FALSE	FALSE
STK11	hgnc:11389	STK11	DTC	9/2/20	inhibitor	0.049605736	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.007592202	FLUOXETINE HYDROCHLORIDE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	PREDNISOLONE SODIUM SUCCINATE	rxcui:55063	PREDNISOLONE SODIUM SUCCINATE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.021733308	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.011694359	ENDOSULFAN	chembl:CHEMBL194399	ENDOSULFAN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.012649403	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.1367387271762877	NSC-26699	chembl:CHEMBL221721	CHEMBL:CHEMBL221721	FALSE	FALSE	FALSE
CAMK2D	hgnc:1462	CAMK2D	DTC	9/2/20	NULL	0.051478109	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	DTC	9/2/20	NULL	0.089103927	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.098884503	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	TETRAIDOFLUORESCEIN	chembl:CHEMBL1160028	TETRAIDOFLUORESCEIN	FALSE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	DTC	9/2/20	NULL	0.7501095890813501	ETRAVIRINE	rxcui:475969	ETRAVIRINE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	DTC	9/2/20	NULL	0.1881995384791917	BENZO[E]PYRENE	chembl:CHEMBL1371125	BENZO[E]PYRENE	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	(+)-ISOBICYCLOGERMACRENAL	chembl:CHEMBL2333548	CHEMBL:CHEMBL2333548	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.041279616	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.009838424	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
PTPN1	hgnc:9642	PTPN1	DTC	9/2/20	NULL	4.200613699	2-CARBOPEROXYBENZOATE	chembl:CHEMBL1162414	CHEMBL:CHEMBL1162414	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.051629962	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	3.088686543276147	NSC-640559	chembl:CHEMBL1287866	CHEMBL:CHEMBL1287866	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002450766	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	N-PHENETHYLCINNAMAMIDE	chembl:CHEMBL1305393	CHEMBL:CHEMBL1305393	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.013673873	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.08854582	(R)-PROCYCLIDINE	chembl:CHEMBL400598	(R)-PROCYCLIDINE	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.1041818873724097	2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE	chembl:CHEMBL1255936	CHEMBL:CHEMBL1255936	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	DTC	9/2/20	NULL	0.1988926940746003	TCMDC-125813	chembl:CHEMBL580076	CHEMBL:CHEMBL580076	FALSE	FALSE	FALSE
NCOA1	hgnc:7668	NCOA1	DTC	9/2/20	NULL	0.2224901323546377	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
DCLK1	hgnc:2700	DCLK1	DTC	9/2/20	NULL	0.2224901323546377	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.057955487	DNDI1417485	chembl:CHEMBL1346468	CHEMBL:CHEMBL1346468	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	INDINAVIR SULFATE	rxcui:203153	INDINAVIR SULFATE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.1174668260306364	GSK369796	iuphar.ligand:10411	GSK369796	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002248915	AMIODARONE HYDROCHLORIDE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.007318142	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	THIOINOSINE	ncit:C877	THIOINOSINE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.1750255707856483	DOCONEXENT	rxcui:1006469	DOCONEXENT	TRUE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.023171964	PRIMAQUINE PHOSPHATE	rxcui:8687	PRIMAQUINE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.052507671	PHENOLPHTHALEIN	rxcui:155122	PHENOLPHTHALEIN	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	1.394008970859145	MENATETRENONE	rxcui:29495	MENATETRENONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.032095154	GNF-PF-3792	chembl:CHEMBL582983	CHEMBL:CHEMBL582983	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00097453	CARFILZOMIB	rxcui:1302966	CARFILZOMIB	TRUE	FALSE	TRUE
TUBB4B	hgnc:20771	TUBB4B	DTC	9/2/20	NULL	0.043629141	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	DTC	9/2/20	NULL	0.040235763	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.044161204	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	DTC	9/2/20	NULL	0.2734774543525755	CEFOXITIN	rxcui:203118	CEFOXITIN SODIUM	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.051731696	NSC-693571	chembl:CHEMBL1287983	CHEMBL:CHEMBL1287983	FALSE	FALSE	FALSE
NEK4	hgnc:11399	NEK4	DTC	9/2/20	NULL	0.049210563	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.012054103	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.030814361	TCMDC-123723	chembl:CHEMBL525103	CHEMBL:CHEMBL525103	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.003133664	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.008899605	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	BISACODYL	rxcui:1596	BISACODYL	TRUE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.046881849	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	TDR78026	chembl:CHEMBL1483413	CHEMBL:CHEMBL1483413	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002784962	FLUPHENAZINE HYDROCHLORIDE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001990963	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ITK	hgnc:6171	ITK	DTC	9/2/20	NULL	0.028598949	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	GNF-PF-2936	chembl:CHEMBL582503	CHEMBL:CHEMBL582503	FALSE	FALSE	FALSE
CFL1	hgnc:1874	CFL1	DTC	9/2/20	NULL	1.458546423213736	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	ERGOSTEROL PEROXIDE	chembl:CHEMBL434750	ERGOSTEROL PEROXIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.042793538	TCMDC-137788	chembl:CHEMBL587564	CHEMBL:CHEMBL587564	FALSE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.014222013	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFKB1	hgnc:7794	NFKB1	DTC	9/2/20	NULL	0.050246575	SJ000128325	chembl:CHEMBL602718	CHEMBL:CHEMBL602718	FALSE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.033832262	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	DTC	9/2/20	NULL	0.023110771	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.00410569	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
HDAC5	hgnc:14068	HDAC5	DTC	9/2/20	NULL	0.1957415516708089	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.1957415516708089	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.010594768	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.05486695	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.012302641	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	GLIQUIDONE	rxcui:25793	GLIQUIDONE	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	N-(4-CHLOROBENZOYL)EVODIAMINE	chembl:CHEMBL1277315	CHEMBL:CHEMBL1277315	FALSE	FALSE	FALSE
HEXA	hgnc:4878	HEXA	DTC	9/2/20	NULL	10.50153424713889	ECHINOMYCIN	ncit:C462	ECHINOMYCIN	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.020226376	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.003053304	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	BROMUCONAZOLE	chembl:CHEMBL271579	BROMUCONAZOLE	FALSE	FALSE	FALSE
TERT	hgnc:11730	TERT	DTC	9/2/20	NULL	3.000438356	2,7-BIS[3-(DIMETHYLAMINO)PROPIONAMIDO]ANTHRAQUINONE	chembl:CHEMBL89977	CHEMBL:CHEMBL89977	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.01495945	DAPH	chembl:CHEMBL268868	DAPH	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	N6-METHYLADENOSINE	chembl:CHEMBL383144	CHEMBL:CHEMBL383144	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.010726797	5,7-DIHYDROXYISOFLAVONE	chembl:CHEMBL1488393	5,7-DIHYDROXYISOFLAVONE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	BTCP	chembl:CHEMBL279556	CHEMBL:CHEMBL279556	FALSE	FALSE	FALSE
WRN	hgnc:12791	WRN	DTC	9/2/20	NULL	0.030886865	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.006836936	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.03219848	CIPROFLOXACIN	rxcui:2551	CIPROFLOXACIN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	CID 2056784	chembl:CHEMBL261123	CHEMBL:CHEMBL261123	FALSE	FALSE	FALSE
DAO	hgnc:2671	DAO	DTC	9/2/20	NULL	21.00306849427779	THIOPHENE-3-CARBOXYLIC ACID	chembl:CHEMBL164585	CHEMBL:CHEMBL164585	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.067231333	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005953251	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.008390488	5-(4-PHENYLBUTOXY)PSORALEN	iuphar.ligand:9583	PSORA-4	FALSE	FALSE	FALSE
SRMS	hgnc:11298	SRMS	DTC	9/2/20	NULL	0.082043236	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.049723174	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	SJ000156747	chembl:CHEMBL592786	CHEMBL:CHEMBL592786	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.1591141552596803	ENPIROLINE	ncit:C75267	ENPIROLINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.116943588	ZINC 02058890	chembl:CHEMBL1738936	CHEMBL:CHEMBL1738936	FALSE	FALSE	FALSE
HSPA5	hgnc:5238	HSPA5	DTC	9/2/20	NULL	0.6563458904461813	4-METHYLDAPHNETIN	chembl:CHEMBL276618	4-METHYLDAPHNETIN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	DESMETHOXYYANGONIN	chembl:CHEMBL254218	DESMETHOXYYANGONIN	FALSE	FALSE	FALSE
ARNT	hgnc:700	ARNT	DTC	9/2/20	NULL	0.4773424657790409	EPICATECHIN GALLATE	iuphar.ligand:12462	EPICATECHIN GALLATE	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	DTC	9/2/20	NULL	0.006280822	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	CHLORAMPHENICOL PALMITATE	rxcui:20767	CHLORAMPHENICOL PALMITATE	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.053038052	PROMETHAZINE HYDROCHLORIDE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	DTC	9/2/20	NULL	0.1419126249613365	PIPERTRAMINE	chembl:CHEMBL127273	PIPERTRAMINE	FALSE	FALSE	FALSE
GBA	hgnc:4177	GBA1	DTC	9/2/20	NULL	0.025865848	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	DNDI1417420	chembl:CHEMBL1546223	CHEMBL:CHEMBL1546223	FALSE	FALSE	FALSE
BRD2	hgnc:1103	BRD2	DTC	9/2/20	NULL	0.2447910080918158	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.1591141552596802	SJ000072878	chembl:CHEMBL601400	CHEMBL:CHEMBL601400	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.2917092846427472	1,2-BENZANTHRACENE	chembl:CHEMBL1873684	CHEMBL:CHEMBL1873684	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	3-METHOXY-MORPHANIN HCL	chembl:CHEMBL1257022	CHEMBL:CHEMBL1257022	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.006027051	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.029170928	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.066297565	2-AMINO-ANTHRAQUINONE	chembl:CHEMBL84685	CHEMBL:CHEMBL84685	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	ONONIN	chembl:CHEMBL465980	ONONIN	FALSE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.3500511415712966	GNF-PF-3286	chembl:CHEMBL581880	CHEMBL:CHEMBL581880	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003670838	2-AMINOETHOXYDIPHENYL BORATE	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	DTC	9/2/20	NULL	1.419126249613364	5-(2-PHENYLETHYL)ISATIN	chembl:CHEMBL1642672	CHEMBL:CHEMBL1642672	FALSE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.2386712328895204	5-CHLORO-[1,10]PHENANTHROLINE	chembl:CHEMBL317115	CHEMBL:CHEMBL317115	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.034612835	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
PSENEN	hgnc:30100	PSENEN	DTC	9/2/20	NULL	1.250182648468916	IC261	drugbank:DB03083	IC261	FALSE	FALSE	FALSE
APH1B	hgnc:24080	APH1B	DTC	9/2/20	NULL	1.154014752432846	IC261	drugbank:DB03083	IC261	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.006570029	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.015193192	CID 663143	chembl:CHEMBL1342336	CHEMBL:CHEMBL1342336	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	ALLO-OCIMENE	chembl:CHEMBL2268552	ALLO-OCIMENE	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.051177067	PH-011685	chembl:CHEMBL126804	CHEMBL:CHEMBL126804	FALSE	FALSE	FALSE
KDM4C	hgnc:17071	KDM4C	DTC	9/2/20	NULL	4.375639269641208	N-METHOXYCARBONYLMETHYL-OXALAMIC ACID METHYL ESTER	chembl:CHEMBL92309	CHEMBL:CHEMBL92309	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001210998	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
BTK	hgnc:1133	BTK	DTC	9/2/20	NULL	0.014103592	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.1131630845596864	GNF-PF-4659	chembl:CHEMBL584442	CHEMBL:CHEMBL584442	FALSE	FALSE	FALSE
AKT3	hgnc:393	AKT3	DTC	9/2/20	NULL	0.056581542	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.023182195	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.04636439	PIFITHRIN-ALPHA	chembl:CHEMBL198759	CHEMBL:CHEMBL198759	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.065145994	ZIRAM	chembl:CHEMBL1519327	ZIRAM	FALSE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.061773731	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.008504644	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.02075402	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
ALPL	hgnc:438	ALPL	DTC	9/2/20	NULL	0.1100789753368857	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.025476793	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	CHLORMIDAZOLE	ncit:C78032	CHLORMIDAZOLE	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.042968634	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	2',3,4-TRIHYDROXYCHALCONE	chembl:CHEMBL339587	CHEMBL:CHEMBL339587	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.016558711	PROPACHLOR	chembl:CHEMBL1394829	PROPACHLOR	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	1.657092009619794	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
KCNQ2	hgnc:6296	KCNQ2	DTC	9/2/20	NULL	3.000438356325399	EZOGABINE	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.017799211	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.3000438356325399	SPINASAPONIN A METHYL ESTER	chembl:CHEMBL1288830	SPINASAPONIN A METHYL ESTER	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	LEAD DIACETATE TRIHYDRATE	chembl:CHEMBL1350036	LEAD DIACETATE TRIHYDRATE	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
HSP90AB1	hgnc:5258	HSP90AB1	DTC	9/2/20	NULL	0.024814589	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.1535312024435511	DALBERGIONE, 4-METHOXY-4'-HYDROXY-	chembl:CHEMBL1374504	DALBERGIONE, 4-METHOXY-4'-HYDROXY-	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.3542686252046857	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.013229446	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	AMODIAQUINE DIHYDROCHLORIDE	chembl:CHEMBL1521739	AMODIAQUINE DIHYDROCHLORIDE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	OncoKB	23-Jul-20	NULL	0.4907258993990139	AZD9496	ncit:C122834	SELECTIVE ESTROGEN RECEPTOR DEGRADER AZD9496	FALSE	FALSE	TRUE
NPY2R	hgnc:7957	NPY2R	DTC	9/2/20	NULL	0.9376369863516874	N6-PHENYLADENOSINE	chembl:CHEMBL262083	N6-PHENYLADENOSINE	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.016764901	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.025588534	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.036162308	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	BERGAPTEN	rxcui:15842	5-METHOXYPSORALEN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	(-)-ASARININ	chembl:CHEMBL1572261	CHEMBL:CHEMBL1572261	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.6563458904461813	[3H]-PHORBOL 12,13-DIBUTYRATE	chembl:CHEMBL27768	CHEMBL:CHEMBL27768	FALSE	FALSE	FALSE
AGTR2	hgnc:338	AGTR2	DTC	9/2/20	NULL	2.386712328895204	PD-123319	iuphar.ligand:597	PD123319	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	ETHOPROPAZINE	rxcui:4134	PROFENAMINE	TRUE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.032412143	GNF-PF-2812	chembl:CHEMBL125044	CHEMBL:CHEMBL125044	FALSE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	DTC	9/2/20	NULL	0.3547815624033412	COLFORSIN	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.035982643	ENZALUTAMIDE	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
ABCG2	hgnc:74	ABCG2	DTC	9/2/20	NULL	0.3281729452230906	ETRAVIRINE	rxcui:475969	ETRAVIRINE	TRUE	FALSE	FALSE
ZAK	hgnc:17797	MAP3K20	DTC	9/2/20	NULL	0.027347745	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.024309107	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
CTNNB1	hgnc:2514	CTNNB1	DTC	9/2/20	NULL	1.591141552596803	FLUORESCEIN SODIUM	rxcui:57789	FLUORESCEIN SODIUM	TRUE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	METHYLBENZETHONIUM CHLORIDE	rxcui:1796444	METHYLBENZETHONIUM CHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006909813	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006995426	MITOTANE	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	GRAMINE	ncit:C64181	GRAMINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.001670623	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.014749346	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.022315202	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.097236428	2-(PHENOXYMETHYL)BENZOTHIAZOLE	chembl:CHEMBL233302	2-(PHENOXYMETHYL)BENZOTHIAZOLE	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.017502557	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.7395446652914718	CEFAMANDOLE NAFATE	rxcui:20473	CEFAMANDOLE NAFATE	TRUE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.025390557	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
MCHR1	hgnc:4479	MCHR1	DTC	9/2/20	NULL	5.000730593875666	SB-568849	iuphar.ligand:1312	SB-568849	FALSE	FALSE	FALSE
STAT3	hgnc:11364	STAT3	DTC	9/2/20	NULL	3.500511415712966	REL-8ALPHA-TIGLOYLOXYHIRSUTINOLIDE	chembl:CHEMBL2062862	CHEMBL:CHEMBL2062862	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	OncoKB	23-Jul-20	NULL	0.6241137025199848	Bosutinib	rxcui:1307619	BOSUTINIB	TRUE	FALSE	TRUE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	2.282942227638891	GO-Y015	chembl:CHEMBL477052	CHEMBL:CHEMBL477052	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PHOSALONE	chembl:CHEMBL1528531	PHOSALONE	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.039778539	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.1535312024435511	NSC-71097	chembl:CHEMBL1939687	CHEMBL:CHEMBL1939687	FALSE	FALSE	FALSE
NCOA1	hgnc:7668	NCOA1	DTC	9/2/20	NULL	0.546954909	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008558708	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	ACETYLSEROTONIN	iuphar.ligand:5451	N-ACETYLSEROTONIN	FALSE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	DTC	9/2/20	NULL	0.1339481409073839	GEDATOLISIB	ncit:C91732	GEDATOLISIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	ESTRIOL	rxcui:4094	ESTRIOL	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1491695205559502	(+/-)-OCTOCLOTHEPIN MALEATE	chembl:CHEMBL1256660	CHEMBL:CHEMBL1256660	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00292359	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.010211527	DEOXIEPINEPHRINE	chembl:CHEMBL31088	DEOXIEPINEPHRINE	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	OncoKB	23-Jul-20	NULL	0.3697723326457359	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	NITROFEN	chembl:CHEMBL561004	NITROFEN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	MINOCYCLINE	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.012466209	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.011799477	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.01654306	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.061773731	PICTILISIB	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
MAPK8	hgnc:6881	MAPK8	DTC	9/2/20	NULL	0.008725103	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
ALPI	hgnc:437	ALPI	DTC	9/2/20	NULL	0.1750255707856483	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002436325	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.1207072901969988	ETHAMSYLATE	rxcui:4112	ETHAMSYLATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.005709838	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
DUSP3	hgnc:3069	DUSP3	DTC	9/2/20	NULL	0.7501095890813501	1,4-DIMETHOXYANTHRAQUINONE	chembl:CHEMBL570408	1,4-DIMETHOXYANTHRAQUINONE	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.016669102	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
EPHX2	hgnc:3402	EPHX2	DTC	9/2/20	NULL	0.1250182648468916	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
RPS6KA5	hgnc:10434	RPS6KA5	DTC	9/2/20	NULL	0.192335792	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.018168744	ALTENUSIN	chembl:CHEMBL483531	ALTENUSIN	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	2-ETHOXYCARBONYL-2-ETHOXYOXALOYLOXYDIHYDROCHRYSIN DIMETHYL ETHER	chembl:CHEMBL1414316	2-ETHOXYCARBONYL-2-ETHOXYOXALOYLOXYDIHYDROCHRYSIN DIMETHYL ETHER	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.003013007	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.040452751	CGS-15943	iuphar.ligand:384	CGS 15943	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00389812	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005534114	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.015429818	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.020672312	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
SPHK1	hgnc:11240	SPHK1	DTC	9/2/20	NULL	26.25383561784724	VPC45129	chembl:CHEMBL554130	CHEMBL:CHEMBL554130	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	OncoKB	23-Jul-20	NULL	0.1900426678745596	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
TNK1	hgnc:11940	TNK1	DTC	9/2/20	inhibitor	1.438566335224506	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.050978322	DIMETHYL GAMBOGATE	chembl:CHEMBL1436860	DIMETHYL GAMBOGATE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	OXYQUINOLINE	rxcui:110	OXYQUINOLINE	TRUE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.1446492320542548	TRIAZOLAM	rxcui:10767	TRIAZOLAM	TRUE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	DTC	9/2/20	NULL	0.729273212	ENCLOMIPHENE CITRATE	ncit:C61745	ENCLOMIPHENE CITRATE	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.011399842	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	NOSCAPINE	rxcui:7533	NOSCAPINE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.099446347	PANCURONIUM BROMIDE	rxcui:7884	PANCURONIUM BROMIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	METHYL YELLOW	chembl:CHEMBL1090440	METHYL YELLOW	FALSE	FALSE	FALSE
PAK4	hgnc:16059	PAK4	DTC	9/2/20	NULL	0.022554842	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	MOMETASONE FUROATE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	OncoKB	23-Jul-20	NULL	0.4906052389860809	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.036413087	GNF-PF-2298	chembl:CHEMBL578905	CHEMBL:CHEMBL578905	FALSE	FALSE	FALSE
ATG4B	hgnc:20790	ATG4B	DTC	9/2/20	NULL	1.346350544504987	SJ000196127	chembl:CHEMBL605084	CHEMBL:CHEMBL605084	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.034184682	BENZAMIL	iuphar.ligand:4145	BENZAMIL	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	SERATRODAST	ncit:C90671	SERATRODAST	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.022583945	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002450766	PAROXETINE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
CACNA1B	hgnc:1389	CACNA1B	DTC	9/2/20	NULL	0.4102161815288632	PHENAZINE-2,3-DIAMINE	chembl:CHEMBL274921	CHEMBL:CHEMBL274921	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	PATULIN	drugbank:DB15586	PATULIN	FALSE	FALSE	FALSE
PTPN6	hgnc:9658	PTPN6	DTC	9/2/20	NULL	8.751278539282415	4-HYDRAZINYLBENZENESULFONIC ACID	chembl:CHEMBL510966	CHEMBL:CHEMBL510966	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003262967	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.013927764	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.017009288	NORSTICTIC ACID	chembl:CHEMBL228281	NORSTICTIC ACID	FALSE	FALSE	FALSE
ABCC4	hgnc:55	ABCC4	PharmGKB	4/5/24	NULL	0.046725403	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FENHEXAMID	chembl:CHEMBL1688541	FENHEXAMID	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.006525935	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
GLA	hgnc:4296	GLA	DTC	9/2/20	NULL	0.08780547	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
MTOR	hgnc:3942	MTOR	DTC	9/2/20	NULL	0.020542907	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	DNDI1416934	chembl:CHEMBL1989750	CHEMBL:CHEMBL1989750	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.04427291	SULMAZOLE	ncit:C84188	SULMAZOLE	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.027347745	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.018043873	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.008681824	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.012442576	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.4375639269641208	6,4'-DIHYDROXYFLAVONE	chembl:CHEMBL484663	CHEMBL:CHEMBL484663	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	GNF-PF-2374	chembl:CHEMBL600298	CHEMBL:CHEMBL600298	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.031784305	3,6-DIMETHOXYFLAVONE	chembl:CHEMBL1331521	3,6-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.1226814748497534	4-(7-METHYLOCTYL)PHENOL	chembl:CHEMBL503990	CHEMBL:CHEMBL503990	FALSE	FALSE	FALSE
KAT2B	hgnc:8638	KAT2B	DTC	9/2/20	NULL	5.834185692854944	DIETHYL-2-TRIDECYLMALONATE	chembl:CHEMBL1797711	CHEMBL:CHEMBL1797711	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.042344896	PHOSMET	drugbank:DB11448	PHOSMET	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.004252322	MIFEPRISTONE	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.00804962	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
MAPK3	hgnc:6877	MAPK3	DTC	9/2/20	NULL	0.4953553890159858	MADOLIN U	chembl:CHEMBL2333546	MADOLIN U	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.021933029	GNF-PF-5061	chembl:CHEMBL601385	CHEMBL:CHEMBL601385	FALSE	FALSE	FALSE
CYBB	hgnc:2578	CYBB	DTC	9/2/20	NULL	1.009762908	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	DTC	9/2/20	NULL	0.078136416	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	CYCLOSTREPTIN	chembl:CHEMBL1242194	CYCLOSTREPTIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.005208578	LEVOBUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
MEN1	hgnc:7010	MEN1	DTC	9/2/20	NULL	0.093596562	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.001284874	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	ASTEMIZOLE	rxcui:42328	ASTEMIZOLE	TRUE	FALSE	FALSE
BIRC3	hgnc:591	BIRC3	DTC	9/2/20	NULL	1.666910197958555	BESTATIN METHYL ESTER	chembl:CHEMBL457092	BESTATIN METHYL ESTER	FALSE	FALSE	FALSE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	0.5834185692854944	2-ARACHIDONOYLGLYCEROL	iuphar.ligand:729	2-ARACHIDONOYLGLYCEROL	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001856641	THIOGUANINE	rxcui:10485	THIOGUANINE	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.035598421	PIFITHRIN-ALPHA	chembl:CHEMBL198759	CHEMBL:CHEMBL198759	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	NOMIFENSINE	rxcui:7500	NOMIFENSINE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.027347745	PIRENZEPINE	rxcui:8352	PIRENZEPINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.015892152	NAN-190	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	SJ000143975	iuphar.ligand:2827	HPTE	FALSE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.033148782	PIPERINE	rxcui:1311146	PIPERINE	TRUE	FALSE	FALSE
CDC25B	hgnc:1726	CDC25B	DTC	9/2/20	NULL	5.000730593875666	NSC-71881	chembl:CHEMBL357170	CHEMBL:CHEMBL357170	FALSE	FALSE	FALSE
APP	hgnc:620	APP	DTC	9/2/20	NULL	1.615620653405984	NSC-649410	chembl:CHEMBL177126	CHEMBL:CHEMBL177126	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	PYRAZOPHOS	chembl:CHEMBL1537719	PYRAZOPHOS	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.013286354	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	PERUVOSIDE	drugbank:DB13756	PERUVOSIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	HESPERETIN	rxcui:1314255	HESPERETIN	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.00399693	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.027870314	PD-81723	chembl:CHEMBL59532	CHEMBL:CHEMBL59532	FALSE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	FDA	10-Apr-24	NULL	0.2125816649218401	Fosphenytoin	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	MyCancerGenome	20-Jun-17	inhibitor	0.3889457128569963	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	MyCancerGenome	20-Jun-17	inhibitor	0.049349315	AEE788	iuphar.ligand:7643	AEE788	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	MyCancerGenome	20-Jun-17	inhibitor	0.2711239478607289	PLX3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenome	20-Jun-17	inhibitor	0.7143900848393808	REFAMETINIB	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	MyCancerGenome	20-Jun-17	inhibitor	0.440315901	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	MyCancerGenome	20-Jun-17	inhibitor	0.013695272	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	MyCancerGenome	20-Jun-17	inhibitor	0.1406455479527531	TANDUTINIB	ncit:C48404	TANDUTINIB	FALSE	FALSE	TRUE
PIK3R2	hgnc:8980	PIK3R2	MyCancerGenome	20-Jun-17	inhibitor	0.049864835	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PIK3R4	hgnc:8982	PIK3R4	MyCancerGenome	20-Jun-17	inhibitor	0.108040476	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenome	20-Jun-17	inhibitor	0.027010119	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1183271464466354	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.1000146118775133	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.2465148884304905	TIVOZANIB	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.1041818873724097	LENVATINIB	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.150021918	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.097236428	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.024309107	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
FLT1	hgnc:3763	FLT1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.075442056	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.5903640284436551	GDC-0973	rxcui:1722365	COBIMETINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.039598545	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.1495945049449985	BIOCHANIN A	ncit:C28201	BIOCHANIN A	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.017260904	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.023014539	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
AGT	hgnc:333	AGT	NCI	14-Sep-17	NULL	0.3070624048871023	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
APOA2	hgnc:601	APOA2	NCI	14-Sep-17	NULL	0.3387591692625452	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.056826484	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
ANXA1	hgnc:533	ANXA1	NCI	14-Sep-17	NULL	0.3409589041278863	PPD	rxcui:1362740	4-PHENYLENEDIAMINE	FALSE	FALSE	FALSE
APOE	hgnc:613	APOE	NCI	14-Sep-17	NULL	0.095295229	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
APP	hgnc:620	APP	NCI	14-Sep-17	NULL	1.615620653405984	BAF	ncit:C1258	TRIAZINATE	FALSE	FALSE	FALSE
APOB	hgnc:603	APOB	NCI	14-Sep-17	NULL	0.1035654265003836	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
AR	hgnc:644	AR	NCI	14-Sep-17	NULL	0.017541538	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.08334551	FLUTAMIDE	rxcui:4508	FLUTAMIDE	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.02587222	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.022467981	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.025111273	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.035574303	TRAMADOL	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	NCI	14-Sep-17	NULL	0.034151331	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
BIRC5	hgnc:593	BIRC5	NCI	14-Sep-17	NULL	0.1325951293830669	SCH 66336	rxcui:2467553	LONAFARNIB	TRUE	FALSE	FALSE
CAMK4	hgnc:1464	CAMK4	NCI	14-Sep-17	NULL	5.250767124	ESTRADIOL BENZOATE	rxcui:60661	ESTRADIOL 3-BENZOATE	TRUE	FALSE	FALSE
COL18A1	hgnc:2195	COL18A1	NCI	14-Sep-17	NULL	3.750547945	CSF	ncit:C387	RECOMBINANT COLONY STIMULATING FACTOR	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.2333674277141977	4-HYDROPEROXYCYCLOPHOSPHAMIDE	ncit:C1423	PERFOSFAMIDE	FALSE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.2287915957982331	RITONAVIR	rxcui:85762	RITONAVIR	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.192335792	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.2692701089009974	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	NCI	14-Sep-17	NULL	0.005366413	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	NCI	14-Sep-17	NULL	0.212152207	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
CYP1A1	hgnc:2595	CYP1A1	NCI	14-Sep-17	NULL	0.052246439	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	NCI	14-Sep-17	NULL	1.346350544504987	SOY PROTEIN	ncit:C1803	SOY PROTEIN ISOLATE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	NCI	14-Sep-17	NULL	0.017709164	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
CYP3A43	hgnc:17450	CYP3A43	NCI	14-Sep-17	NULL	1.875273972703375	SHO-SAIKO-TO	ncit:C2690	SHO-SAIKO-TO	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	NCI	14-Sep-17	NULL	0.023813003	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.001753236	RISPERIDONE	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
DDIT3	hgnc:2726	DDIT3	NCI	14-Sep-17	NULL	0.2220197515251353	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
CYR61	hgnc:2654	CCN1	NCI	14-Sep-17	NULL	11.66837138570988	INTERLEUKIN-8	rxcui:1426866	INTERLEUKIN-8	FALSE	FALSE	FALSE
DCK	hgnc:2704	DCK	NCI	14-Sep-17	NULL	0.4565884455277783	CLADRIBINE	rxcui:44157	CLADRIBINE	TRUE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.1790034246671403	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.1981421556063943	BIOMODULATORS	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
DNMT1	hgnc:2976	DNMT1	NCI	14-Sep-17	NULL	0.095468493	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
DPYD	hgnc:3012	DPYD	NCI	14-Sep-17	NULL	0.1071038678953482	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
EDN3	hgnc:3178	EDN3	NCI	14-Sep-17	NULL	5.527123287967842	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
EPO	hgnc:3415	EPO	NCI	14-Sep-17	NULL	0.7895890411382631	HUMAN CHORIONIC GONADOTROPIN	rxcui:340705	HUMAN CHORIONIC GONADOTROPIN	TRUE	FALSE	FALSE
EIF4G1	hgnc:3296	EIF4G1	NCI	14-Sep-17	NULL	0.068324881	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.038382801	AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
ERCC1	hgnc:3433	ERCC1	NCI	14-Sep-17	NULL	1.093909817410302	HERBIMYCIN A	iuphar.ligand:5984	HERBIMYCIN A	FALSE	FALSE	FALSE
F9	hgnc:3551	F9	NCI	14-Sep-17	NULL	0.032134438	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.012486961	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
FCGR1A	hgnc:3613	FCGR1A	NCI	14-Sep-17	NULL	15.75230137070834	MDX-447	chembl:CHEMBL2109391	MDX-447	FALSE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	NCI	14-Sep-17	NULL	0.9907107780319716	CA19-9 ANTIGEN	ncit:C327	CA19-9 ANTIGEN	FALSE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.099446347	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
FCGR3B	hgnc:3620	FCGR3B	NCI	14-Sep-17	NULL	0.1060761035064535	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.06823609	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
GGT1	hgnc:4250	GGT1	NCI	14-Sep-17	NULL	0.4321619031744403	N-METHYL-N-NITROSOUREA	ncit:C645	METHYLNITROSOUREA	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	NCI	14-Sep-17	NULL	0.017198713	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.7955707762984013	LEVOFLOXACIN	rxcui:1546009	LEVOFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	0.080471527	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.1646008502686348	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
GSTA1	hgnc:4626	GSTA1	NCI	14-Sep-17	NULL	0.6563458904461812	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
GRP	hgnc:4605	GRP	NCI	14-Sep-17	NULL	1.296485709523321	EGFR TYROSINE KINASE INHIBITORS	ncit:C2167	EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR	FALSE	FALSE	TRUE
GSR	hgnc:4623	GSR	NCI	14-Sep-17	NULL	0.2983390411119005	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.3512218811752141	NITROGLYCERIN	rxcui:4917	NITROGLYCERIN	TRUE	FALSE	TRUE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1093909817410302	ETHACRYNIC ACID	rxcui:4109	ETHACRYNIC ACID	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	NCI	14-Sep-17	NULL	0.5707355569097228	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1093909817410302	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
IL17F	hgnc:16404	IL17F	NCI	14-Sep-17	NULL	0.9376369863516875	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
IL17RC	hgnc:18358	IL17RC	NCI	14-Sep-17	NULL	35.00511415712966	IL-17	ncit:C1684	RECOMBINANT INTERLEUKIN-17	FALSE	FALSE	FALSE
IL27	hgnc:19157	IL27	NCI	14-Sep-17	NULL	4.773424657790409	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.059532507	CGP41251	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	2.059124362184098	TXP	ncit:C2649	DHA-PACLITAXEL	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.3241214273808302	MBL	ncit:C1151	MANNOSE-BINDING LECTIN	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.044706404	LANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
IRAK4	hgnc:17967	IRAK4	NCI	14-Sep-17	NULL	0.2651902587661338	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
IRS2	hgnc:6126	IRS2	NCI	14-Sep-17	NULL	1.238388472539964	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.2917092846427472	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
ITGAX	hgnc:6152	ITGAX	NCI	14-Sep-17	NULL	1.944728564284981	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	NCI	14-Sep-17	NULL	0.729273212	FAS-LIGAND	ncit:C1538	RECOMBINANT FAS LIGAND	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	NCI	14-Sep-17	NULL	0.7242437411819932	RTX	ncit:C1214	RESINIFERATOXIN	FALSE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.546954909	DMSO	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	2.187819634820604	LIAROZOLE	ncit:C1433	LIAROZOLE	FALSE	FALSE	FALSE
KCNA2	hgnc:6220	KCNA2	NCI	14-Sep-17	NULL	0.6563458904461813	6-OHDA	ncit:C1316	OXIDOPAMINE	FALSE	FALSE	FALSE
KCNA4	hgnc:6222	KCNA4	NCI	14-Sep-17	NULL	0.3333820395917111	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
KCNQ1	hgnc:6294	KCNQ1	NCI	14-Sep-17	NULL	0.090064616	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
LAMB1	hgnc:6486	LAMB1	NCI	14-Sep-17	NULL	4.375639269641208	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.5048814541893701	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.8468979231563628	TRIBUTYRIN	ncit:C1260	TRIBUTYRIN	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	NCI	14-Sep-17	NULL	0.260583976	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	NCI	14-Sep-17	NULL	0.1037701012563132	BFGF	ncit:C1674	RECOMBINANT FIBROBLAST GROWTH FACTOR 2	FALSE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.2287915957982331	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.1029562181092049	PLATINUM	rxcui:1311280	PLATINUM	FALSE	FALSE	FALSE
MDH2	hgnc:6971	MDH2	NCI	14-Sep-17	NULL	26.25383561784724	EXPECTORANT	ncit:C29767	EXPECTORANT	FALSE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	4.375639269641208	MELANOMA VACCINE	ncit:C2517	MELANOMA VACCINE	FALSE	FALSE	FALSE
MMP2	hgnc:7166	MMP2	NCI	14-Sep-17	NULL	0.4487835148349957	4-HYDROPEROXYCYCLOPHOSPHAMIDE	ncit:C1423	PERFOSFAMIDE	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	3.500511415712966	CI-921	ncit:C1050	ASULACRINE ISETHIONATE	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.1875273972703375	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.037505479	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
GRIN1	hgnc:4584	GRIN1	PharmGKB	4/5/24	NULL	0.028199609	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.3454452054979901	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.002075566	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.009685975	HYPERICIN	rxcui:1546455	HYPERICIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.023609564	DICUMAROL	rxcui:1598	DICUMAROL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.011110383	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
NPPC	hgnc:7941	NPPC	NCI	14-Sep-17	NULL	0.7501095890813501	IMMUNOMODULATORS	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.2051080907644316	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.729273212	INTERLEUKIN-8	rxcui:1426866	INTERLEUKIN-8	FALSE	FALSE	FALSE
NRG1	hgnc:7997	NRG1	NCI	14-Sep-17	NULL	0.1562728310586145	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
P2RY2	hgnc:8541	P2RY2	NCI	14-Sep-17	NULL	0.1154014752432846	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
OXTR	hgnc:8529	OXTR	NCI	14-Sep-17	NULL	0.325124899	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
PCSK1	hgnc:8743	PCSK1	NCI	14-Sep-17	NULL	6.563458904461812	PHOSPHODIESTERASE INHIBITOR	ncit:C744	PHOSPHODIESTERASE INHIBITOR	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	NCI	14-Sep-17	NULL	0.024309107	FLAVOPIRIDOL	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	0.4605936073306535	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
PLA2G2A	hgnc:9031	PLA2G2A	NCI	14-Sep-17	NULL	1.750255707856483	DIFLUOROMETHYLORNITHINE	ncit:C226	EFLORNITHINE	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	NCI	14-Sep-17	NULL	0.1682938180631233	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1346350544504987	ZINC SULFATE	rxcui:1299928	ZINC SULFATE ANHYDROUS	TRUE	FALSE	FALSE
NKX6-1	hgnc:7839	NKX6-1	PharmGKB	4/5/24	NULL	0.6908904109959803	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.036770078	IRESSA	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
PPIA	hgnc:9253	PPIA	NCI	14-Sep-17	NULL	0.8334550989792778	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
PLTP	hgnc:9093	PLTP	NCI	14-Sep-17	NULL	4.773424657790409	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	1.458546423213736	ANTI-PROGESTIN	ncit:C1891	PROGESTERONE ANTAGONIST	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	1.458546423213736	BUPROPION HCL	chembl:CHEMBL1698	BUPROPION HYDROCHLORIDE	FALSE	FALSE	FALSE
PTPRC	hgnc:9666	PTPRC	NCI	14-Sep-17	NULL	0.4861821410712453	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.2822993077187876	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.1562728310586145	DMSO	rxcui:3455	DIMETHYL SULFOXIDE	TRUE	FALSE	FALSE
RBP3	hgnc:9921	RBP3	NCI	14-Sep-17	NULL	1.458546423213736	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
RORA	hgnc:10258	RORA	NCI	14-Sep-17	NULL	1.357957014716237	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
SHBG	hgnc:10839	SHBG	NCI	14-Sep-17	NULL	1.050153425	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.4039051633514961	FDG	rxcui:1362737	FLUORODEOXYGLUCOSE F18	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.201952582	LIF	iuphar.ligand:5016	LIF	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	PharmGKB	4/5/24	NULL	0.025588534	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.3088686543276147	SELENIUM	rxcui:9641	SELENIUM	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	NCI	14-Sep-17	NULL	0.4907258993990139	TYROSINE HYDROXYLASE INHIBITOR	ncit:C2155	TYROSINE HYDROXYLASE INHIBITOR	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.064624826	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.1346350544504987	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	NCI	14-Sep-17	NULL	0.08780547	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
GRIK4	hgnc:4582	GRIK4	PharmGKB	4/5/24	NULL	0.09869863	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
STAR	hgnc:11359	STAR	NCI	14-Sep-17	NULL	17.50255707856483	BDNF	iuphar.ligand:4872	BDNF	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1047012387551236	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1483267549030917	BRDU	ncit:C318	BROXURIDINE	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.8899605294185507	BOVINE CARTILAGE	ncit:C2418	BOVINE CARTILAGE	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.1495945049449985	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
THBS1	hgnc:11785	THBS1	NCI	14-Sep-17	NULL	0.123644438	ALL-TRANS RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.192335792	VASCULAR ENDOTHELIAL GROWTH FACTOR	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.074797252	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	1.346350544504987	RICIN	ncit:C809	RICIN	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.6731752722524935	CHINESE HERBS	ncit:C2663	CHINESE HERBS	FALSE	FALSE	FALSE
XDH	hgnc:12805	XDH	NCI	14-Sep-17	NULL	0.1121958787087489	FOLIC ACID	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.049349315	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
XRCC1	hgnc:12828	XRCC1	NCI	14-Sep-17	NULL	0.8678953923255289	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	OncoKB	23-Jul-20	NULL	0.1331836936859721	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CDKN2A	hgnc:1787	CDKN2A	OncoKB	23-Jul-20	NULL	0.5609793935437446	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
MDM2	hgnc:6973	MDM2	OncoKB	23-Jul-20	NULL	1.312691780892362	RO5045337	ncit:C91724	MDM2 ANTAGONIST RO5045337	FALSE	FALSE	TRUE
ARAF	hgnc:646	ARAF	OncoKB	23-Jul-20	NULL	0.075369863	Sorafenib	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	OncoKB	23-Jul-20	NULL	0.049723174	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	OncoKB	23-Jul-20	NULL	0.3642372228836055	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	OncoKB	23-Jul-20	NULL	0.1176247115494948	Ribociclib	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	OncoKB	23-Jul-20	NULL	0.4089382494991783	Erdafitinib	rxcui:2123125	ERDAFITINIB	TRUE	FALSE	TRUE
EIF2AK4	hgnc:19687	EIF2AK4	PharmGKB	4/5/24	NULL	0.3454452054979901	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
HSPG2	hgnc:5273	HSPG2	PharmGKB	4/5/24	NULL	0.4605936073306535	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
GRIN2A	hgnc:4585	GRIN2A	PharmGKB	4/5/24	NULL	0.020025809	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
ARID5B	hgnc:17362	ARID5B	PharmGKB	4/5/24	NULL	0.4605936073306535	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
PLEKHA6	hgnc:17053	PLEKHA6	PharmGKB	4/5/24	NULL	1.381780822	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
CYP2J2	hgnc:2634	CYP2J2	PharmGKB	4/5/24	NULL	0.2692701089009974	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EDN1	hgnc:3176	EDN1	PharmGKB	4/5/24	NULL	0.9723642821424906	muraglitazar	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	PharmGKB	4/5/24	NULL	0.017715139	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
STN1	hgnc:26200	STN1	PharmGKB	4/5/24	NULL	2.917092846427472	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.072324616	hydroxyprogesterone	ncit:C87242	HYDROXYPROGESTERONE	FALSE	FALSE	FALSE
APOC3	hgnc:610	APOC3	PharmGKB	4/5/24	NULL	0.2500365296937833	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.08854582	acetaminophen / caffeine / dihydrocodeine	wikidata:Q48566647	ACETAMINOPHEN / CAFFEINE / DIHYDROCODEINE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.001591431	dipyridamole	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
CYP3A43	hgnc:17450	CYP3A43	PharmGKB	4/5/24	NULL	0.1119566550867686	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
HOMER1	hgnc:17512	HOMER1	PharmGKB	4/5/24	NULL	1.381780822	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
UGT1A10	hgnc:12531	UGT1A10	PharmGKB	4/5/24	NULL	0.4251633298436802	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
ADH1A	hgnc:249	ADH1A	PharmGKB	4/5/24	NULL	1.312691780892362	acetaldehyde	rxcui:1311137	ACETALDEHYDE	TRUE	FALSE	FALSE
CDCA3	hgnc:14624	CDCA3	PharmGKB	4/5/24	NULL	6.563458904461812	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.014299475	dronabinol	rxcui:10402	DRONABINOL	TRUE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.030015818	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
KLRD1	hgnc:6378	KLRD1	PharmGKB	4/5/24	NULL	3.000438356325399	certolizumab pegol	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
SLC22A1	hgnc:10963	SLC22A1	PharmGKB	4/5/24	NULL	0.182318303	levodopa	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
SLCO2B1	hgnc:10962	SLCO2B1	PharmGKB	4/5/24	NULL	0.2625383561784725	chloroquine	rxcui:2393	CHLOROQUINE	TRUE	FALSE	TRUE
RRM2B	hgnc:17296	RRM2B	PharmGKB	4/5/24	NULL	0.1296485709523321	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	PharmGKB	4/5/24	NULL	0.069180068	Ergot alkaloids	rxcui:4023	ERGOT ALKALOIDS	FALSE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	PharmGKB	4/5/24	NULL	0.3509871071904712	olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
IL13	hgnc:5973	IL13	PharmGKB	4/5/24	NULL	0.2651902587661338	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.025891357	crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.014024485	nicardipine	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.029918901	amlodipine	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
IRS1	hgnc:6125	IRS1	PharmGKB	4/5/24	NULL	0.1600843635234588	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.024932417	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.016027983	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.02804897	propranolol	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.017260904	quinine	rxcui:9071	QUININE	TRUE	FALSE	FALSE
NPPA	hgnc:7939	NPPA	PharmGKB	4/5/24	NULL	1.750255707856483	amlodipine	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
FOLR1	hgnc:3791	FOLR1	PharmGKB	4/5/24	NULL	0.5469549087051511	mirvetuximab soravtansine	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
UGT1A3	hgnc:12535	UGT1A3	PharmGKB	4/5/24	NULL	0.4751825451194073	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
HTR1A	hgnc:5286	HTR1A	PharmGKB	4/5/24	NULL	0.018672714	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.1121958787087489	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.052481431	lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
TLR9	hgnc:15633	TLR9	PharmGKB	4/5/24	NULL	0.1187956362798518	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	0.4487835148349958	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
NFATC2	hgnc:7776	NFATC2	PharmGKB	4/5/24	NULL	0.6731752722524936	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
GBP6	hgnc:25395	GBP6	PharmGKB	4/5/24	NULL	4.039051633514962	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
RYR3	hgnc:10485	RYR3	PharmGKB	4/5/24	NULL	0.8751278539282417	amlodipine	rxcui:104416	AMLODIPINE BESYLATE	TRUE	FALSE	FALSE
ZNF816	hgnc:26995	ZNF816	PharmGKB	4/5/24	NULL	0.7955707762984016	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
CD69	hgnc:1694	CD69	PharmGKB	4/5/24	NULL	3.500511415712967	tocilizumab	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
KCNE2	hgnc:6242	KCNE2	PharmGKB	4/5/24	NULL	4.039051633514962	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	PharmGKB	4/5/24	NULL	0.026458892	atezolizumab	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
SLCO1A2	hgnc:10956	SLCO1A2	PharmGKB	4/5/24	NULL	1.093909817410302	celiprolol	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.040275444	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NOS1AP	hgnc:16859	NOS1AP	PharmGKB	4/5/24	NULL	0.3106962795011509	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	PharmGKB	4/5/24	NULL	0.1025540453822158	phenylephrine	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
DMD	hgnc:2928	DMD	PharmGKB	4/5/24	NULL	7.501095891	viltolarsen	rxcui:2389840	VILTOLARSEN	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.043137707	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.00804962	fluphenazine	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
DBH	hgnc:2689	DBH	PharmGKB	4/5/24	NULL	0.1944728564284981	levodopa	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.003849818	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	PharmGKB	4/5/24	NULL	0.033919684	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
CD58	hgnc:1688	CD58	PharmGKB	4/5/24	NULL	3.500511415712967	interferon beta-1b	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
CD58	hgnc:1688	CD58	PharmGKB	4/5/24	NULL	2.333674277141977	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.098513454	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
TNFSF13B	hgnc:11929	TNFSF13B	PharmGKB	4/5/24	NULL	32.81729452230906	belimumab	rxcui:1092437	BELIMUMAB	TRUE	TRUE	TRUE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.078840347	levodopa	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
IL1RN	hgnc:6000	IL1RN	PharmGKB	4/5/24	NULL	0.3454452054979901	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	PharmGKB	4/5/24	NULL	0.0287871	dextroamphetamine	rxcui:3287	DEXTROAMPHETAMINE SULFATE	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.2651902587661338	anakinra	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.1620607136904151	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
MIR4268	hgnc:38352	MIR4268	PharmGKB	4/5/24	NULL	0.1600843635234588	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.01235184	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	PharmGKB	4/5/24	NULL	0.001493605	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	PharmGKB	4/5/24	NULL	0.032412143	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
JAG1	hgnc:6188	JAG1	PharmGKB	4/5/24	NULL	8.751278539282415	maralixibat	rxcui:2571074	MARALIXIBAT	TRUE	FALSE	FALSE
MISP	hgnc:27000	MISP	PharmGKB	4/5/24	NULL	0.4268916360625569	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
MUTYH	hgnc:7527	MUTYH	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.08334551	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CUX2	hgnc:19347	CUX2	PharmGKB	4/5/24	NULL	3.750547945406749	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CYP27B1	hgnc:2606	CYP27B1	PharmGKB	4/5/24	NULL	0.2885036881082115	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	0.1014640990061729	brentuximab vedotin	rxcui:1147320	BRENTUXIMAB VEDOTIN	TRUE	FALSE	FALSE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.1296485709523321	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.7001022831425934	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
SULT2B1	hgnc:11459	SULT2B1	PharmGKB	4/5/24	NULL	2.625383561784725	gemtuzumab ozogamicin	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
SLC22A12	hgnc:17989	SLC22A12	PharmGKB	4/5/24	NULL	0.8078103267029924	gemtuzumab ozogamicin	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
ADGRL3	hgnc:20974	ADGRL3	PharmGKB	4/5/24	NULL	0.172722603	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
RPTOR	hgnc:30287	RPTOR	PharmGKB	4/5/24	NULL	0.086361301	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1458546423213736	sacituzumab govitecan	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
BLMH	hgnc:1059	BLMH	PharmGKB	4/5/24	NULL	0.090530468	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.061412481	fluticasone propionate	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
PTPRD	hgnc:9668	PTPRD	PharmGKB	4/5/24	NULL	0.7721716358190368	pioglitazone	rxcui:259319	PIOGLITAZONE HYDROCHLORIDE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.017859752	everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
UGT1A9	hgnc:12541	UGT1A9	PharmGKB	4/5/24	NULL	0.3512218811752141	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.069454592	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
KCNMA1	hgnc:6284	KCNMA1	PharmGKB	4/5/24	NULL	0.3241214273808303	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
DPYS	hgnc:3013	DPYS	PharmGKB	4/5/24	NULL	0.045579576	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	PharmGKB	4/5/24	NULL	0.7343730242754476	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	PharmGKB	4/5/24	NULL	0.012945678	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
ALK	hgnc:427	ALK	PharmGKB	4/5/24	NULL	2.493675356344019	lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	1.250182648468916	terbinafine	rxcui:37801	TERBINAFINE	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.3671865121377238	losartan	rxcui:203160	LOSARTAN POTASSIUM	TRUE	FALSE	FALSE
GLDC	hgnc:4313	GLDC	PharmGKB	4/5/24	NULL	1.000146118775133	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.02726255	sacituzumab govitecan	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
AURKA	hgnc:11393	AURKA	TALC	12-May-16	inhibitor	1.779921058837101	MK5108	ncit:C90585	AURORA A KINASE INHIBITOR MK5108	FALSE	FALSE	TRUE
HDAC5	hgnc:14068	HDAC5	TALC	12-May-16	inhibitor	0.218327115	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
HDAC6	hgnc:14064	HDAC6	TALC	12-May-16	inhibitor	0.2817943000126717	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
HDAC8	hgnc:13315	HDAC8	TALC	12-May-16	inhibitor	0.1495945049449985	CHR-3996	iuphar.ligand:8391	CHR-3996	FALSE	FALSE	TRUE
ITGB1	hgnc:6153	ITGB1	TALC	12-May-16	antibody	4.375639269641208	VOLOCIXIMAB	ncit:C48426	VOLOCIXIMAB	FALSE	FALSE	TRUE
ITGA5	hgnc:6141	ITGA5	TALC	12-May-16	antibody	6.563458904461812	PF-04605412	chembl:CHEMBL2109622	PF-04605412	FALSE	FALSE	TRUE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	0.9907107780319716	AVE1642	ncit:C79798	VELIGROTUG	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.3642372228836055	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.2692701089009974	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
UNIPROT:P22102	hgnc:4163	GART	TdgClinicalTrial	Jan-14	NULL	0.1536809889825205	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
UNIPROT:P41143	hgnc:8153	OPRD1	TdgClinicalTrial	Jan-14	NULL	0.3889457128569962	ALKS 37	chembl:CHEMBL2364619	METHYLSAMIDORPHAN	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.079197091	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.05387244	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.057197899	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.05387244	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.055155117	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.051478109	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TdgClinicalTrial	Jan-14	NULL	0.040275444	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.042073455	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.057700738	AMISULPRIDE	rxcui:46303	AMISULPRIDE	TRUE	FALSE	FALSE
UNIPROT:P01031	hgnc:1331	C5	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	ARC1905	iuphar.ligand:12857	AVACINCAPTAD PEGOL	FALSE	FALSE	FALSE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	ARBACLOFEN	ncit:C90890	ARBACLOFEN	FALSE	FALSE	FALSE
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.1325951293830669	ARRY-614	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	ARRY-797	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
UNIPROT:P42701	hgnc:5971	IL12RB1	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	AS1409	drugbank:DB05182	AS1409	FALSE	FALSE	FALSE
CYB5R4	hgnc:20147	CYB5R4	PharmGKB	4/5/24	NULL	0.7501095890813498	metoclopramide	rxcui:267036	METOCLOPRAMIDE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q99665	hgnc:5972	IL12RB2	TdgClinicalTrial	Jan-14	NULL	8.751278539282415	AS1409	drugbank:DB05182	AS1409	FALSE	FALSE	FALSE
UNIPROT:P00748	hgnc:3530	F12	TdgClinicalTrial	Jan-14	NULL	0.9723642821424908	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	0.1389091831632129	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
NPY5R	hgnc:7958	NPY5R	PharmGKB	4/5/24	NULL	0.4412409347537353	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.8751278539282416	BECAPLERMIN	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	1.615620653405984	BAN2401	iuphar.ligand:12202	LECANEMAB	FALSE	FALSE	FALSE
UNIPROT:Q02880	hgnc:11990	TOP2B	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	BECATECARIN	ncit:C1620	BECATECARIN	FALSE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	BMS-582949	drugbank:DB12696	BMS-582949	FALSE	FALSE	FALSE
UNIPROT:P34972	hgnc:2160	CNR2	TdgClinicalTrial	Jan-14	NULL	2.019525817	PRS-211375	chembl:CHEMBL3545290	PRS-211375	FALSE	FALSE	FALSE
UNIPROT:P05231	hgnc:6018	IL6	TdgClinicalTrial	Jan-14	NULL	4.286340509036285	CDP6038	ncit:C172654	OLOKIZUMAB	FALSE	FALSE	FALSE
UNIPROT:P15509	hgnc:2435	CSF2RA	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	CG0070	drugbank:DB05148	CG0070	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.088396753	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1223955040459079	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P06756	hgnc:6150	ITGAV	TdgClinicalTrial	Jan-14	NULL	2.692701089009974	CNTO-95	ncit:C61070	INTETUMUMAB	FALSE	FALSE	FALSE
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	SEMAPIMOD	ncit:C96535	SEMAPIMOD	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.097236428	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
UNIPROT:P49356	hgnc:3785	FNTB	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	CP-609,754	ncit:C2551	CP-609,754	FALSE	FALSE	FALSE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.3241214273808303	hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.192335792	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
UNIPROT:P56817	hgnc:933	BACE1	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	CTS-21166	drugbank:DB06073	CTS-21166	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.029235897	DROSPIRENONE	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.3443125982668492	NORETHISTERONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
ALDH2	hgnc:404	ALDH2	PharmGKB	4/5/24	NULL	0.4565884455277783	acetaldehyde	rxcui:1311137	ACETALDEHYDE	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.1226814748497534	DIENOGEST	rxcui:22968	DIENOGEST	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.057732459	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
UNIPROT:P47989	hgnc:12805	XDH	TdgClinicalTrial	Jan-14	NULL	0.7249579855026854	FEBUXOSTAT	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
UNIPROT:Q00535	hgnc:1774	CDK5	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
SLC19A1	hgnc:10937	SLC19A1	PharmGKB	4/5/24	NULL	0.364636606	folic acid	rxcui:4511	FOLIC ACID	TRUE	FALSE	FALSE
UNIPROT:P49336	hgnc:1779	CDK8	TdgClinicalTrial	Jan-14	NULL	0.1312691780892362	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
UNIPROT:P50613	hgnc:1778	CDK7	TdgClinicalTrial	Jan-14	NULL	0.525076712	ALVOCIDIB	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
DSP	hgnc:3052	DSP	PharmGKB	4/5/24	NULL	1.400204566285186	nintedanib	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	1.381780822	FLOVAGATRAN	ncit:C80843	FLOVAGATRAN	FALSE	FALSE	FALSE
UNIPROT:P13945	hgnc:288	ADRB3	TdgClinicalTrial	Jan-14	NULL	3.000438356	KUC-7483	chembl:CHEMBL2107773	RITOBEGRON	FALSE	FALSE	FALSE
UNIPROT:P10827	hgnc:11796	THRA	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.42006137	NAVEGLITAZAR	ncit:C75191	NAVEGLITAZAR	FALSE	FALSE	FALSE
UNIPROT:Q9NR96	hgnc:15633	TLR9	TdgClinicalTrial	Jan-14	NULL	4.633029815	MGN1703	ncit:C94207	LEFITOLIMOD	FALSE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TdgClinicalTrial	Jan-14	NULL	21.00306849427779	METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA	rxcui:729596	METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA	TRUE	FALSE	FALSE
UNIPROT:O14920	hgnc:5960	IKBKB	TdgClinicalTrial	Jan-14	NULL	5.000730593875666	MLN-0415	chembl:CHEMBL3545265	MLN-0415	FALSE	FALSE	FALSE
UNIPROT:P04275	hgnc:12726	VWF	TdgClinicalTrial	Jan-14	NULL	0.6908904109959803	FACTOR VIII	rxcui:11274	VON WILLEBRAND FACTOR	TRUE	FALSE	FALSE
ADH1B	hgnc:250	ADH1B	PharmGKB	4/5/24	NULL	7.001022831425934	acetaldehyde	rxcui:1311137	ACETALDEHYDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.1158257453728555	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
UNIPROT:P04141	hgnc:2434	CSF2	TdgClinicalTrial	Jan-14	NULL	2.100306849	MT203	ncit:C97943	NAMILUMAB	FALSE	FALSE	FALSE
UNIPROT:P09693	hgnc:1675	CD3G	TdgClinicalTrial	Jan-14	NULL	0.42006137	MT-103	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
UNIPROT:P16422	hgnc:11529	EPCAM	TdgClinicalTrial	Jan-14	NULL	1.575230137070835	MT110	ncit:C77854	SOLITOMAB	FALSE	FALSE	TRUE
UNIPROT:P09172	hgnc:2689	DBH	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	NEPICASTAT	ncit:C84003	NEPICASTAT	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.034981793	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.08854582	dextromethorphan / quinidine	wikidata:Q5268496	DEXTROMETHORPHAN/QUINIDINE	FALSE	FALSE	FALSE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.1331836936859721	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:P15056	hgnc:1097	BRAF	TdgClinicalTrial	Jan-14	NULL	0.091636424	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:Q16445	hgnc:4080	GABRA6	TdgClinicalTrial	Jan-14	NULL	0.032899543	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
UNIPROT:P43119	hgnc:9602	PTGIR	TdgClinicalTrial	Jan-14	NULL	5.625821918110125	NS-304	rxcui:1729002	SELEXIPAG	TRUE	FALSE	FALSE
UNIPROT:P41180	hgnc:1514	CASR	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	NPS-2143	drugbank:DB05695	NPS-2143	FALSE	FALSE	FALSE
UNIPROT:Q9UBN7	hgnc:14064	HDAC6	TdgClinicalTrial	Jan-14	NULL	0.2817943000126717	CRA-024781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.078136416	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.2243917574174978	Cremophor EL	chembl:CHEMBL2074614	CREMOPHOR EL	FALSE	FALSE	FALSE
UNIPROT:P05129	hgnc:9402	PRKCG	TdgClinicalTrial	Jan-14	NULL	0.1426838892274307	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.3571950424196904	2-O, 3-O DESULFATED HEPARIN	drugbank:DB17569	2-O, 3-O DESULFATED HEPARIN	FALSE	FALSE	FALSE
UNIPROT:Q16512	hgnc:9405	PKN1	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.089756703	cannabinoids	chembl:CHEMBL3833333	NABIXIMOLS	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.032055965	vecuronium	rxcui:11153	VECURONIUM BROMIDE	TRUE	FALSE	FALSE
UNIPROT:P14784	hgnc:6009	IL2RB	TdgClinicalTrial	Jan-14	NULL	0.4039051633514962	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
UNIPROT:P31785	hgnc:6010	IL2RG	TdgClinicalTrial	Jan-14	NULL	0.5250767123569451	ALDESLEUKIN	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
UNIPROT:Q96DB2	hgnc:19086	HDAC11	TdgClinicalTrial	Jan-14	NULL	0.1060761035064535	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.7095631248066824	SVT-40776	chembl:CHEMBL1779046	TARAFENACIN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.011810092	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	TC-6499	chembl:CHEMBL4594254	SIMPINICLINE	FALSE	FALSE	FALSE
UNIPROT:Q99250	hgnc:10588	SCN2A	TdgClinicalTrial	Jan-14	NULL	0.08334551	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.1193356164447602	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TdgClinicalTrial	Jan-14	NULL	0.082043236	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.057073556	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
UNIPROT:Q9BQB6	hgnc:23663	VKORC1	TdgClinicalTrial	Jan-14	NULL	0.3621218705909965	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.037398626	methylprednisolone	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
UNIPROT:P05093	hgnc:2593	CYP17A1	TdgClinicalTrial	Jan-14	NULL	3.750547945	GALETERONE	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
NLRP3	hgnc:16400	NLRP3	PharmGKB	4/5/24	NULL	1.944728564284981	anakinra	rxcui:72435	ANAKINRA	TRUE	FALSE	TRUE
UNIPROT:Q96RI0	hgnc:3540	F2RL3	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	RUSALATIDE	ncit:C152274	RUSALATIDE	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.073089743	GALETERONE	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.088248187	MELEVODOPA	ncit:C83927	MELEVODOPA	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
UNIPROT:P52895	hgnc:385	AKR1C2	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.0296486	MELEVODOPA	ncit:C83927	MELEVODOPA	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.1084869240406911	norclobazam	drugbank:DB17092	NORCLOBAZAM	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.1805819381121768	PANITUMUMAB	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
UNIPROT:P10721	hgnc:6342	KIT	TdgClinicalTrial	Jan-14	NULL	0.1405827877796372	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
UNIPROT:P43235	hgnc:2536	CTSK	TdgClinicalTrial	Jan-14	NULL	11.66837138570988	VEL-0230	chembl:CHEMBL1085282	CHEMBL:CHEMBL1085282	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.007341677	nicardipine	rxcui:7396	NICARDIPINE	TRUE	FALSE	FALSE
UNIPROT:P25116	hgnc:3537	F2R	TdgClinicalTrial	Jan-14	NULL	1.009762908	VORAPAXAR	rxcui:1537034	VORAPAXAR	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	0.5933070196123671	CANDOXATRIL	ncit:C171870	CANDOXATRIL	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.3040984820600068	CEVIMELINE	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.054695491	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.091583148	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TdgClinicalTrial	Jan-14	NULL	0.089501712	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
UNIPROT:Q14181	hgnc:30073	POLA2	TdgClinicalTrial	Jan-14	NULL	1.000146118775133	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TdgClinicalTrial	Jan-14	NULL	0.075496292	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.020873652	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.021715331	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TdgClinicalTrial	Jan-14	NULL	0.2419708351875322	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:P30049	hgnc:837	ATP5F1D	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	HALOTHANE	rxcui:5095	HALOTHANE	TRUE	FALSE	FALSE
UNIPROT:P26358	hgnc:2976	DNMT1	TdgClinicalTrial	Jan-14	NULL	0.1704794520639431	IFOSFAMIDE	rxcui:5657	IFOSFAMIDE	TRUE	FALSE	TRUE
UNIPROT:Q13936	hgnc:1390	CACNA1C	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
ABCC5	hgnc:56	ABCC5	PharmGKB	4/5/24	NULL	0.072424374	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.1988926940746003	MEPHENYTOIN	rxcui:6757	MEPHENYTOIN	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.042504861	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.2004109589148645	MEDRYSONE	rxcui:29439	MEDRYSONE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	1.221108633388244	METHOHEXITAL	rxcui:6847	METHOHEXITAL	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.1154014752432845	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TdgClinicalTrial	Jan-14	NULL	0.596678082	MEXILETINE	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.056097939	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.05913026	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.033919684	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	NEOSTIGMINE	rxcui:7315	NEOSTIGMINE	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.1141471113819445	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.081407242	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	PharmGKB	4/5/24	NULL	1.628144844517658	pemigatinib	rxcui:2359268	PEMIGATINIB	TRUE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.096050618	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
UNIPROT:P00747	hgnc:9071	PLG	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	TENECTEPLASE	rxcui:259280	TENECTEPLASE	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.2031244535229961	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P36544	hgnc:1960	CHRNA7	TdgClinicalTrial	Jan-14	NULL	0.2075402025126264	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.1864177677006905	TERAZOSIN	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.040235763	lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	TORASEMIDE	rxcui:38413	TORSEMIDE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TdgClinicalTrial	Jan-14	NULL	0.1025540453822158	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.2302968036653267	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.2187819634820604	TOLAZOLINE	rxcui:10634	TOLAZOLINE	TRUE	FALSE	FALSE
UNIPROT:P47901	hgnc:896	AVPR1B	TdgClinicalTrial	Jan-14	NULL	0.5770073762164232	VASOPRESSIN	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.8204323630577265	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.077827576	TRIFLUPROMAZINE	rxcui:10805	TRIFLUPROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.5303805175322677	TROPICAMIDE	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
SLCO1C1	hgnc:13819	SLCO1C1	PharmGKB	4/5/24	NULL	0.5048814541893702	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.054695491	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.092988792	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.1840222122746302	CLOMIFENE	rxcui:2596	CLOMIPHENE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.088396753	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.044611445	DIETHYLSTILBESTROL	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.7026004179620139	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
UNIPROT:P12268	hgnc:6053	IMPDH2	TEND	1-Aug-11	NULL	1.312691780892362	MYCOPHENOLATE MOFETIL	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
UNIPROT:P22303	hgnc:108	ACHE	TEND	1-Aug-11	NULL	1.158257453728555	EDROPHONIUM	rxcui:1546421	EDROPHONIUM CATION	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TEND	1-Aug-11	NULL	0.6819178082557726	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
PKLR	hgnc:9020	PKLR	PharmGKB	4/5/24	NULL	11.66837138570988	mitapivat	rxcui:2594468	MITAPIVAT	TRUE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TEND	1-Aug-11	NULL	0.1103102336884338	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
UNIPROT:P47989	hgnc:12805	XDH	TEND	1-Aug-11	NULL	0.7249579855026854	FEBUXOSTAT	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
UNIPROT:P09884	hgnc:9173	POLA1	TEND	1-Aug-11	NULL	0.5791287268642776	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.03729238	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.096167896	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
MECP2	hgnc:6990	MECP2	PharmGKB	4/5/24	NULL	0.1810609352954982	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.055344054	FLUPENTHIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.054695491	FLUPENTHIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.028300937	FLUPHENAZINE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14780	hgnc:7176	MMP9	TEND	1-Aug-11	NULL	0.42006137	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	PharmGKB	4/5/24	NULL	0.546954909	sotorasib	rxcui:2550714	SOTORASIB	TRUE	FALSE	TRUE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.1640864726115453	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TEND	1-Aug-11	NULL	4.375639269641208	GLYCODIAZINE	rxcui:102848	GLYMIDINE	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TEND	1-Aug-11	NULL	0.086361301	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TEND	1-Aug-11	NULL	0.6250913242344582	ILOPROST	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.4234489615781814	KETOTIFEN	rxcui:11404	KETOTIFEN FUMARATE	TRUE	FALSE	FALSE
PGM1	hgnc:8905	PGM1	PharmGKB	4/5/24	NULL	0.6646540662746139	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TEND	1-Aug-11	NULL	0.0701037	LEVONORGESTREL	rxcui:6373	LEVONORGESTREL	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.042073455	LOXAPINE	rxcui:6475	LOXAPINE	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.2983390411119005	LOTEPREDNOL ETABONATE	rxcui:237027	LOTEPREDNOL	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.059085902	METHYLDOPA	rxcui:1545996	METHYLDOPA ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TEND	1-Aug-11	NULL	5.000730593875666	METOCURINE	rxcui:29950	METOCURINE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TEND	1-Aug-11	NULL	0.1121958787087489	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TEND	1-Aug-11	NULL	0.054020238	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q96P88	hgnc:16341	GNRHR2	TEND	1-Aug-11	NULL	5.834185692854944	NAFARELIN	rxcui:28656	NAFARELIN	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.021036727	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.2386712328895204	NABUMETONE	rxcui:31448	NABUMETONE	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TEND	1-Aug-11	NULL	0.3443125982668492	NORETHINDRONE	rxcui:7514	NORETHINDRONE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.046518424	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.090922374	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.3454452054979901	PROCAINE	rxcui:8701	PROCAINE	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.049457775	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.055155117	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.2778183663264258	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
MET	hgnc:7029	MET	PharmGKB	4/5/24	NULL	0.384671584	crizotinib	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.0296486	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.1013661606866689	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TEND	1-Aug-11	NULL	0.088248187	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.1154014752432845	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	PharmGKB	4/5/24	NULL	0.1187188949127459	propranolol	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1556551518844698	ZUCLOPENTHIXOL	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.5877724392055355	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
GABA TRANSAMINASE	hgnc:23	ABAT	TTD	2020.06.01	NULL	0.3017682254924971	CPP-115	iuphar.ligand:8284	CPP-115	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.4167275494896388	ASP8273	ncit:C115110	NAQUOTINIB	FALSE	FALSE	TRUE
HELODERMIN-PREFERRING VIP RECEPTOR	hgnc:12695	VIPR2	TTD	2020.06.01	NULL	26.25383561784724	PB1046	ncit:C179114	PEMZIVIPTADIL	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.2656374598770379	ethylmorphine	rxcui:4166	ETHYLMORPHINE	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-XL	hgnc:992	BCL2L1	TTD	2020.06.01	NULL	1.875273972703375	APG-1252	ncit:C148488	PELCITOCLAX	FALSE	FALSE	FALSE
INDUCED MYELOID LEUKEMIA CELL DIFFERENTIATION PROTEIN MCL-1	hgnc:32041	ADAMTSL4-AS1	TTD	2020.06.01	NULL	0.3125456621172291	AZD5991	iuphar.ligand:11783	AZD5991	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	1.897867635025102	BLU-285	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.04427291	oliceridine	rxcui:2392230	OLICERIDINE	TRUE	FALSE	FALSE
ENHANCER OF ZESTE HOMOLOG 1	hgnc:3526	EZH1	TTD	2020.06.01	NULL	8.751278539282415	DS-3201	ncit:C127114	VALEMETOSTAT	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.1193356164447602	Sulfatinib	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
STIMULATOR OF INTERFERON GENES PROTEIN	hgnc:27962	STING1	TTD	2020.06.01	NULL	26.25383561784724	MK-1454	drugbank:DB14721	MK-1454	FALSE	FALSE	FALSE
SCNN1G	hgnc:10602	SCNN1G	PharmGKB	4/5/24	NULL	1.620607136904151	triamterene	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE UFO	hgnc:905	AXL	TTD	2020.06.01	NULL	0.364636606	ONO-7475	chembl:CHEMBL4650414	ONO-7475	FALSE	FALSE	FALSE
BROMODOMAIN AND EXTRATERMINAL DOMAIN PROTEIN	hgnc:24456	DNER	TTD	2020.06.01	NULL	4.039051633514961	RG6146	ncit:C112500	BET INHIBITOR RO6870810	FALSE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	0.7192831676122533	ONO-7579	drugbank:DB17236	ONO-7579	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	0.5048814541893701	MP0250	ncit:C117236	VEGF/HGF-TARGETING DARPIN MP0250	FALSE	FALSE	FALSE
RETINOIC ACID RECEPTOR ALPHA	hgnc:9864	RARA	TTD	2020.06.01	NULL	0.8334550989792776	SY-1425	ncit:C71025	TAMIBAROTENE	FALSE	FALSE	TRUE
SCNN1B	hgnc:10600	SCNN1B	PharmGKB	4/5/24	NULL	1.823183029	triamterene	rxcui:10763	TRIAMTERENE	TRUE	FALSE	FALSE
MAP KINASE SIGNAL-INTEGRATING KINASE 2	hgnc:7111	MKNK2	TTD	2020.06.01	NULL	2.625383561784724	EFT508	ncit:C125062	TOMIVOSERTIB	FALSE	FALSE	FALSE
CALGRANULIN D	hgnc:10489	S100A12	TTD	2020.06.01	NULL	5.250767123569449	Atogepant	rxcui:2571813	ATOGEPANT	TRUE	FALSE	FALSE
XRCC3	hgnc:12830	XRCC3	PharmGKB	4/5/24	NULL	0.1207072901969988	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SURVIVAL MOTOR NEURON PROTEIN	hgnc:11117	SMN1	TTD	2020.06.01	NULL	0.3977853881492007	LMI070	chembl:CHEMBL4290141	BRANAPLAM	FALSE	FALSE	FALSE
TYK2 TYROSINE KINASE	hgnc:12440	TYK2	TTD	2020.06.01	NULL	0.8468979231563628	PF-06826647	ncit:C180657	ROPSACITINIB	FALSE	FALSE	FALSE
TISSUE KALLIKREIN	hgnc:6363	KLK2	TTD	2020.06.01	NULL	13.12691780892362	Avoralstat	ncit:C169799	AVORALSTAT	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.00804962	promethazine	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	0.4375639269641208	Conatumumab	ncit:C71015	CONATUMUMAB	FALSE	TRUE	TRUE
PANCREATIC TRIACYLGLYCEROL LIPASE	hgnc:9155	PNLIP	TTD	2020.06.01	NULL	6.563458904461812	MS-1819	drugbank:DB15004	MS-1819	FALSE	FALSE	FALSE
HEAT SHOCK PROTEIN 90 ALPHA	hgnc:5253	HSP90AA1	TTD	2020.06.01	NULL	0.3621218705909965	Debio 0932	ncit:C92572	HSP90 INHIBITOR DEBIO 0932	FALSE	FALSE	FALSE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.5385402178019949	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BMX	hgnc:1079	BMX	TTD	2020.06.01	NULL	0.3182283105193606	Ibrutinib	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.073089743	TOK-001	ncit:C84866	GALETERONE	FALSE	FALSE	FALSE
HYALURONIC ACID RECEPTOR	hgnc:14687	LYVE1	TTD	2020.06.01	NULL	52.50767123569449	Hyaluronate sodium	ncit:C83761	HYALURONATE SODIUM	FALSE	FALSE	FALSE
CALGRANULIN B	hgnc:10499	S100A9	TTD	2020.06.01	NULL	26.25383561784724	Tasquinimod	ncit:C74080	TASQUINIMOD	FALSE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	PharmGKB	4/5/24	NULL	0.172722603	enalapril	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 1	hgnc:4584	GRIN1	TTD	2020.06.01	NULL	0.2678962818147678	ELIPRODIL	ncit:C80994	ELIPRODIL	FALSE	FALSE	FALSE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	0.1630673019742065	Alprostadil	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	Levomethadyl Acetate	rxcui:237005	LEVOMETHADYL	TRUE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.5	hgnc:10593	SCN5A	TTD	2020.06.01	NULL	0.596678082	Mexiletine	rxcui:6926	MEXILETINE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.096758608	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
MAPK/ERK KINASE KINASE 2	hgnc:6854	MAP3K2	TTD	2020.06.01	NULL	2.917092846427472	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
GLUCOCORTICOID RECEPTOR	hgnc:7978	NR3C1	TTD	2020.06.01	NULL	0.2226788432387383	Mometasone	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	2.386712328895204	NCX 1022	drugbank:DB05410	NCX 1022	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.041508041	Tolazoline	rxcui:10634	TOLAZOLINE	TRUE	FALSE	FALSE
MTHFR	hgnc:7436	MTHFR	PharmGKB	4/5/24	NULL	0.078840347	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-12	hgnc:7158	MMP12	TTD	2020.06.01	NULL	0.2333674277141977	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
PRESENILIN 2	hgnc:9509	PSEN2	TTD	2020.06.01	NULL	0.7955707762984013	R-flurbiprofen	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
PRESENILIN 1	hgnc:9508	PSEN1	TTD	2020.06.01	NULL	0.6731752722524935	R-flurbiprofen	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-21	hgnc:14357	MMP21	TTD	2020.06.01	NULL	2.100306849	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
FATTY ALDEHYDE DEHYDROGENASE	hgnc:403	ALDH3A2	TTD	2020.06.01	NULL	0.1356787370431382	Disulfiram	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	1.381780822	Dextofisopam	ncit:C76460	DEXTOFISOPAM	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2	hgnc:281	ADRA2A	TTD	2020.06.01	NULL	0.6105543166941221	Fipamezole	ncit:C65684	FIPAMEZOLE	FALSE	FALSE	FALSE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	0.4167275494896389	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	Met-enkephalin	rxcui:1349278	METENKEFALIN	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Denopamine	ncit:C77934	DENOPAMINE	FALSE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	2.282942227638891	MEM-3454	chembl:CHEMBL5095032	RG3487	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 12 MEMBER 1	hgnc:10910	SLC12A1	TTD	2020.06.01	NULL	1.875273972703375	Bendroflumethiazide	rxcui:1369	BENDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	0.305277158	Picrotoxin	rxcui:2539172	PICROTOXIN	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-1	hgnc:4075	GABRA1	TTD	2020.06.01	NULL	1.221108633388244	Methohexital	rxcui:6847	METHOHEXITAL	TRUE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.7395446652914718	SALVINORIN A	drugbank:DB12327	SALVINORIN A	FALSE	FALSE	FALSE
5-HT 3A RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	0.1666910197958555	Levetiracetam	rxcui:114477	LEVETIRACETAM	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.3040984820600068	Cevimeline	rxcui:44281	CEVIMELINE	TRUE	FALSE	FALSE
GTPASE NRAS	hgnc:7989	NRAS	TTD	2020.06.01	NULL	0.07699072	Salirasib	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
IMMUNOGLOBULIN GAMMA FC RECEPTOR III	hgnc:3619	FCGR3A	TTD	2020.06.01	NULL	0.9907107780319716	GMA-161	drugbank:DB15397	GMA-161	FALSE	FALSE	FALSE
FATTY ACID-BINDING PROTEIN 1	hgnc:3555	FABP1	TTD	2020.06.01	NULL	0.7721716358190367	FENOFIBRIC ACID	rxcui:24852	FENOFIBRIC ACID	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-2	hgnc:1956	CHRNA2	TTD	2020.06.01	NULL	0.750109589	Carbachol	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
MATRIX METALLOPROTEINASE-2	hgnc:7166	MMP2	TTD	2020.06.01	NULL	0.053854022	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-14	hgnc:7160	MMP14	TTD	2020.06.01	NULL	0.300043836	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	PharmGKB	4/5/24	NULL	0.5303805175322677	cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
CYTOCHROME P450 26	hgnc:2603	CYP26A1	TTD	2020.06.01	NULL	15.75230137070834	Rambazole	ncit:C90792	TALAROZOLE	FALSE	FALSE	FALSE
CALCINEURIN	hgnc:9314	PPP3CA	TTD	2020.06.01	NULL	4.375639269641208	Pimecrolimus	rxcui:321952	PIMECROLIMUS	TRUE	FALSE	FALSE
CYCLIN-DEPENDENT KINASE 4	hgnc:1773	CDK4	TTD	2020.06.01	NULL	0.2778183663264258	AG-024322	ncit:C52182	CDK1/2/4 INHIBITOR AG-024322	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1848861663228679	E-7050	ncit:C82363	GOLVATINIB	FALSE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.3697723326457359	Nalfurafine hcl	chembl:CHEMBL490665	NALFURAFINE HYDROCHLORIDE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.5585922471882393	Nebracetam	ncit:C66223	NEBRACETAM	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	0.1875273972703375	Tesofensine	ncit:C66589	TESOFENSINE	FALSE	FALSE	FALSE
GONADOTROPIN-RELEASING HORMONE RECEPTOR	hgnc:4421	GNRHR	TTD	2020.06.01	NULL	1.193356164447602	Ozarelix	ncit:C95214	OZARELIX	FALSE	FALSE	FALSE
VITAMIN K EPOXIDE REDUCTASE COMPLEX 1	hgnc:23663	VKORC1	TTD	2020.06.01	NULL	15.75230137070834	Tecarfarin	ncit:C152523	TECARFARIN	FALSE	FALSE	FALSE
LEUKOTRIENE A-4 HYDROLASE	hgnc:6710	LTA4H	TTD	2020.06.01	NULL	0.8334550989792776	Bestatin	ncit:C1015	UBENIMEX	FALSE	FALSE	FALSE
PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA	hgnc:8803	PDGFRA	TTD	2020.06.01	NULL	0.033106981	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
GAPVD1	hgnc:23375	GAPVD1	PharmGKB	4/5/24	NULL	3.500511415712966	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.000146118775133	PF-4217903	chembl:CHEMBL2001019	PF-04217903	FALSE	FALSE	TRUE
N-ACETYLGALACTOSAMINE-4-SULFATASE	hgnc:714	ARSB	TTD	2020.06.01	NULL	6.563458904461812	Galsulfase	rxcui:578033	GALSULFASE	TRUE	FALSE	FALSE
NEURONAL ACETYLCHOLINE RECEPTOR ALPHA-7	hgnc:1960	CHRNA7	TTD	2020.06.01	NULL	2.282942227638891	JNJ-39393406	drugbank:DB11867	JNJ-39393406	FALSE	FALSE	FALSE
HUS1	hgnc:5309	HUS1	PharmGKB	4/5/24	NULL	3.281729452230906	mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.073437302	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
FIBRONECTIN	hgnc:3778	FN1	TTD	2020.06.01	NULL	0.212581665	Ocriplasmin	rxcui:29998	OCRIPLASMIN	TRUE	FALSE	FALSE
NUCLEAR FACTOR ERYTHROID 2-RELATED FACTOR 2	hgnc:4071	GABPA	TTD	2020.06.01	NULL	8.751278539282415	OT-551	drugbank:DB05650	OT-551	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	0.8247278204559345	PLX8394	drugbank:DB16038	PLX8394	FALSE	FALSE	TRUE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.6819178082557726	Dyphylline	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 2	hgnc:4594	GRM2	TTD	2020.06.01	NULL	3.750547945	ADX71149	iuphar.ligand:8946	JNJ-40411813	FALSE	FALSE	FALSE
B1 BRADYKININ RECEPTOR	hgnc:1029	BDKRB1	TTD	2020.06.01	NULL	11.66837138570988	Safotibant	ncit:C152283	SAFOTIBANT	FALSE	FALSE	FALSE
ANGIOTENSIN II RECEPTOR TYPE-2	hgnc:338	AGTR2	TTD	2020.06.01	NULL	1.193356164447602	ANGIOTENSIN II	rxcui:1999003	ANGIOTENSIN II	TRUE	FALSE	FALSE
SOMATOTROPIN	hgnc:4261	GH1	TTD	2020.06.01	NULL	8.751278539282415	VRS-317	chembl:CHEMBL3707323	SOMAVARATAN	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.8204323630577265	MSC2363318A	ncit:C112004	P70S6K/AKT INHIBITOR M-2698	FALSE	FALSE	FALSE
SLC39A8	hgnc:20862	SLC39A8	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
TRANSMEMBRANE ACTIVATOR AND CAML INTERACTOR	hgnc:18153	TNFRSF13B	TTD	2020.06.01	NULL	26.25383561784724	AUTO2	ncit:C150509	AUTOLOGOUS BCMA/TACI-TARGETED CAR T CELLS AUTO2	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR A	hgnc:12680	VEGFA	TTD	2020.06.01	NULL	1.413668071730236	Aflibercept	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
TYROSINE-PROTEIN KINASE KIT	hgnc:6342	KIT	TTD	2020.06.01	NULL	0.3642372228836055	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
CARBONIC ANHYDRASE I	hgnc:1368	CA1	TTD	2020.06.01	NULL	0.7501095890813498	Acetazolamide	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1584738568481725	Brivanib	ncit:C67040	BRIVANIB	FALSE	FALSE	TRUE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.4526523382387456	Sabarubicin	ncit:C1706	SABARUBICIN	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.097308509	XL880	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	1.093909817410302	TCN-P	ncit:C1262	TRICIRIBINE PHOSPHATE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M1	hgnc:1950	CHRM1	TTD	2020.06.01	NULL	0.3351553483129436	Metixene	rxcui:29682	METHIXENE	TRUE	FALSE	FALSE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	2.763561643983921	TLN-4601	ncit:C62508	DIAZEPINOMICIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	0.046549354	Dipyridamole	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
MULTIDRUG RESISTANCE PROTEIN 1	hgnc:40	ABCB1	TTD	2020.06.01	NULL	0.2243917574174978	CBT-1	ncit:C67042	MDR MODULATOR CBT-1	FALSE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.2465148884304905	brimonidine	rxcui:134615	BRIMONIDINE	TRUE	FALSE	FALSE
TYROSINE-PROTEIN KINASE ABL1	hgnc:76	ABL1	TTD	2020.06.01	NULL	0.066662299	Adenosine triphosphate	rxcui:318	ADENOSINE TRIPHOSPHATE	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.099446347	Atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.4293851619741372	Atomoxetine	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME	hgnc:2707	ACE	TTD	2020.06.01	NULL	0.4449802647092754	Benazepril	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	1.591141552596802	Crofelemer	rxcui:1364449	CROFELEMER	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.1312691780892362	glimepiride	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	0.5000730593875666	Clevidipine butyrate	rxcui:233603	CLEVIDIPINE	TRUE	FALSE	FALSE
FYN TYROSINE PROTEIN KINASE	hgnc:4037	FYN	TTD	2020.06.01	NULL	0.075768645	Dasatinib	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	1.029562181092048	Neostigmine	rxcui:7315	NEOSTIGMINE	TRUE	FALSE	FALSE
CORTICOSTEROID-BINDING GLOBULIN	hgnc:1540	SERPINA6	TTD	2020.06.01	NULL	6.563458904461812	Paramethasone	rxcui:7910	PARAMETHASONE	TRUE	FALSE	FALSE
GASTRIC H(+)/K(+) ATPASE ALPHA	hgnc:819	ATP4A	TTD	2020.06.01	NULL	0.2243917574174979	Rabeprazole	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	0.080471527	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
BETA-CATENIN	hgnc:2514	CTNNB1	TTD	2020.06.01	NULL	0.7955707762984014	Recombinant human endostatin	ncit:C45515	RECOMBINANT HUMAN ENDOSTATIN	FALSE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.111481255	RO-23-7553	ncit:C1883	VITAMIN D3 ANALOGUE ILX23-7553	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.7	hgnc:10597	SCN9A	TTD	2020.06.01	NULL	1.250182648468916	RG7893	chembl:CHEMBL3707353	RG7893	FALSE	FALSE	FALSE
FK506-BINDING PROTEIN 1A	hgnc:3711	FKBP1A	TTD	2020.06.01	NULL	4.375639269641208	AP1903	ncit:C82412	RIMIDUCID	FALSE	FALSE	FALSE
PURINE NUCLEOSIDE PHOSPHORYLASE	hgnc:7892	PNP	TTD	2020.06.01	NULL	8.751278539282415	BCX-3408	chembl:CHEMBL269864	ULODESINE	FALSE	FALSE	FALSE
TRAIL RECEPTOR 2	hgnc:11905	TNFRSF10B	TTD	2020.06.01	NULL	5.834185692854944	Conatumumab	ncit:C71015	CONATUMUMAB	FALSE	TRUE	TRUE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.037398626	celiprolol	rxcui:20498	CELIPROLOL	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.7778914257139926	APD-334	rxcui:2668045	ETRASIMOD	TRUE	FALSE	FALSE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	1.944728564284981	KRP-203	ncit:C106368	MOCRAVIMOD HYDROCHLORIDE	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	1.029562181092049	M2951	ncit:C141427	EVOBRUTINIB	FALSE	FALSE	FALSE
NEUROMEDIN-K RECEPTOR	hgnc:11528	TACR3	TTD	2020.06.01	NULL	1.944728564284981	Senktide	iuphar.ligand:2127	SENKTIDE	FALSE	FALSE	FALSE
REEP5	hgnc:30077	REEP5	PharmGKB	4/5/24	NULL	0.750109589	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
MAP KINASE P38	hgnc:6874	MAPK12	TTD	2020.06.01	NULL	0.3241214273808302	VX-745	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	2.423430980108977	Gantenerumab	ncit:C88580	GANTENERUMAB	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	3.500511415712966	DIPROTEVERINE HYDROCHLORIDE	ncit:C73025	DIPROTEVERINE	FALSE	FALSE	FALSE
INDOLEAMINE 2,3-DIOXYGENASE 1	hgnc:6059	IDO1	TTD	2020.06.01	NULL	3.750547945	Epacadostat	ncit:C92582	EPACADOSTAT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.015608701	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.2108741816694558	IUPHAR.LIGAND:16	iuphar.ligand:16	L-772,405	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.063262255	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
REEP5	hgnc:30077	REEP5	PharmGKB	4/5/24	NULL	0.9376369863516874	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	inhibitor	0.2108741816694558	IUPHAR.LIGAND:113	iuphar.ligand:113	GR-55562	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.1223955040459079	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:5	ncbigene:5	A12M2	GuideToPharmacology	2024.1	agonist	0.017715139	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1241316104862754	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	PharmGKB	4/5/24	NULL	0.076934317	everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.011575765	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.011575765	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.027781837	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:9825	iuphar.ligand:9825	COMPOUND 3B [PMID:28943244]	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.055271233	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.078958904	IUPHAR.LIGAND:152	iuphar.ligand:152	&ALPHA;-METHYL-5-HT	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	agonist	0.1842374429322613	IUPHAR.LIGAND:171	iuphar.ligand:171	ORG-37684	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.025739055	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:9	hgnc:7645	NAT1	GuideToPharmacology	2024.1	inhibitor	0.097236428	IUPHAR.LIGAND:260	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:7356	ncit:C169839	CERLAPIRDINE	FALSE	FALSE	FALSE
NCBIGENE:779	hgnc:1397	CACNA1S	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:10372	iuphar.ligand:10372	COMPOUND 14 [PMID: 30925062]	FALSE	FALSE	FALSE
NCBIGENE:768	hgnc:1383	CA9	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10372	iuphar.ligand:10372	COMPOUND 14 [PMID: 30925062]	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.2206204673768676	IUPHAR.LIGAND:7709	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	PharmGKB	4/5/24	NULL	0.5780661053470953	cannabinoids	chembl:CHEMBL3833333	NABIXIMOLS	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:11874	iuphar.ligand:11874	ENVONALKIB	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:500	iuphar.ligand:500	[125I]HEAT (BE2254)	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.1415301111474245	IUPHAR.LIGAND:499	iuphar.ligand:499	WB 4101	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.3977853881492006	IUPHAR.LIGAND:500	iuphar.ligand:500	[125I]HEAT (BE2254)	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:499	iuphar.ligand:499	WB 4101	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.066297565	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	PharmGKB	4/5/24	NULL	0.004931224	temazepam	rxcui:10355	TEMAZEPAM	TRUE	FALSE	FALSE
NT5C3A	hgnc:17820	NT5C3A	PharmGKB	4/5/24	NULL	0.6482428547616604	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
RAC2	hgnc:9802	RAC2	PharmGKB	4/5/24	NULL	0.3201687270469177	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
SLC22A8	hgnc:10972	SLC22A8	PharmGKB	4/5/24	NULL	0.2027323213733378	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.009572521	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
ADRA2C	hgnc:283	ADRA2C	PharmGKB	4/5/24	NULL	0.2275522047050683	clonidine	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
BMP7	hgnc:1074	BMP7	PharmGKB	4/5/24	NULL	0.1296485709523321	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:498	iuphar.ligand:498	SNAP5089	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	PharmGKB	4/5/24	NULL	0.1909369863116163	sitagliptin	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.094438258	IUPHAR.LIGAND:526	iuphar.ligand:526	RX821002	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	inhibitor	0.062958838	IUPHAR.LIGAND:313	iuphar.ligand:313	MUSCARINIC TOXIN 3	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.018887652	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:526	iuphar.ligand:526	RX821002	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.1704794520639431	IUPHAR.LIGAND:499	iuphar.ligand:499	WB 4101	FALSE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	agonist	0.059667808	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.067317527	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:2767	hgnc:4379	GNA11	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9346	iuphar.ligand:9346	PXS-4728A	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6455	rxcui:1546379	TRANDOLAPRILAT	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1207072901969988	IUPHAR.LIGAND:5612	ncit:C152892	VIPADENANT	FALSE	FALSE	FALSE
PNPLA3	hgnc:18590	PNPLA3	PharmGKB	4/5/24	NULL	0.5834185692854944	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:410	iuphar.ligand:410	GALANGIN	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.084146909	IUPHAR.LIGAND:5596	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.045898314	IUPHAR.LIGAND:5615	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.090219366	IUPHAR.LIGAND:5596	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1804387327687096	IUPHAR.LIGAND:433	iuphar.ligand:433	VISNAGIN	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:5604	ncit:C96195	ROLOFYLLINE	FALSE	FALSE	FALSE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.1750255707856483	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.067664525	IUPHAR.LIGAND:5605	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.1539814405738841	IUPHAR.LIGAND:592	rxcui:73494	TELMISARTAN	TRUE	FALSE	FALSE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	0.760980743	IUPHAR.LIGAND:6170	iuphar.ligand:6170	MK-5046	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:5571	iuphar.ligand:5571	(-)-RO 363	FALSE	FALSE	FALSE
NCBIGENE:1789	hgnc:2979	DNMT3B	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8144	iuphar.ligand:8144	COMPOUND 13R [PMID: 23639540]	FALSE	FALSE	FALSE
IGHMBP2	hgnc:5542	IGHMBP2	PharmGKB	4/5/24	NULL	0.7778914257139926	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:11866	iuphar.ligand:11866	AMREDOBRESIB	FALSE	FALSE	FALSE
NCBIGENE:2729	hgnc:4311	GCLC	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:7511	iuphar.ligand:7511	(+)-JQ1	FALSE	FALSE	FALSE
NCBIGENE:2728	ncbigene:2728	GLC3B	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8824	iuphar.ligand:8824	COMPOUND 50 [PMID: 24313754]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9857	iuphar.ligand:9857	BMS-986142	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.2019525816757481	IUPHAR.LIGAND:8148	iuphar.ligand:8148	COMPOUND 31 [PMID: 24915291]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9869	iuphar.ligand:9869	BRANEBRUTINIB	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9263	iuphar.ligand:9263	GDC-0834	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:645	iuphar.ligand:645	[DES-ARG11]T-KININ	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:648	iuphar.ligand:648	[DES-PRO8,DES-PHE9,DES-ARG10]KALLIDIN	FALSE	FALSE	FALSE
NCBIGENE:41	hgnc:100	ASIC1	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:641	iuphar.ligand:641	[LEU8,DES-ARG9]BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:31	hgnc:84	ACACA	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:3640	iuphar.ligand:3640	C3A	FALSE	FALSE	FALSE
NCBIGENE:2471	hgnc:3881	FRA20A	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:6687	rxcui:10318	TACRINE	TRUE	FALSE	FALSE
NCBIGENE:939	hgnc:11922	CD27	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:11228	iuphar.ligand:11228	INHIBITOR E18	FALSE	FALSE	FALSE
NCBIGENE:2471	hgnc:3881	FRA20A	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:6598	rxcui:8299	PHYSOSTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:678	iuphar.ligand:678	[THI5,8,D-PHE7]BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:9450	iuphar.ligand:9450	AVACOPAN	FALSE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:578	iuphar.ligand:578	NDT9520492	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12258	iuphar.ligand:12258	MONNA	FALSE	FALSE	FALSE
NCBIGENE:708	hgnc:1243	C1QBP	GuideToPharmacology	2024.1	blocker	3.281729452230906	IUPHAR.LIGAND:4173	iuphar.ligand:4173	DCDPC	FALSE	FALSE	FALSE
NCBIGENE:1594	hgnc:2606	CYP27B1	GuideToPharmacology	2024.1	inhibitor	2.019525817	IUPHAR.LIGAND:8623	iuphar.ligand:8623	COMPOUND 4 [PMID: 19954973]	FALSE	FALSE	FALSE
NCBIGENE:1617	hgnc:2682	DAZ1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:6467	ncit:C76768	PRALNACASAN	FALSE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7718	iuphar.ligand:7718	Z944	FALSE	FALSE	FALSE
NCBIGENE:529	hgnc:857	ATP6V1E1	GuideToPharmacology	2024.1	activator	1.458546423213736	IUPHAR.LIGAND:4065	iuphar.ligand:4065	(-)-(S)-BAYK8644	FALSE	FALSE	FALSE
NCBIGENE:535	hgnc:865	ATP6V0A1	GuideToPharmacology	2024.1	blocker	0.3281729452230906	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:11515	iuphar.ligand:11515	K777	FALSE	FALSE	FALSE
NCBIGENE:58	hgnc:129	ACTA1	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:753	iuphar.ligand:753	CCL14	FALSE	FALSE	FALSE
NCBIGENE:60	hgnc:132	ACTB	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:789	iuphar.ligand:789	RO116-4875/608	FALSE	FALSE	FALSE
NCBIGENE:1990	hgnc:3308	CELA1	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:8055	drugbank:DB08691	ETHYL 3-[(E)-2-AMINO-1-CYANOETHENYL]-6,7-DICHLORO-1-METHYL-1H-INDOLE-2-CARBOXYLATE	FALSE	FALSE	FALSE
NCBIGENE:2744	hgnc:4331	GLS	GuideToPharmacology	2024.1	NULL	0.1479089330582944	IUPHAR.LIGAND:6891	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	blocker	0.041150213	IUPHAR.LIGAND:2414	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	inhibitor	1.591141552596802	IUPHAR.LIGAND:7453	rxcui:1364449	CROFELEMER	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.02926849	IUPHAR.LIGAND:2713	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.1268301237577161	IUPHAR.LIGAND:2893	rxcui:232158	ROFECOXIB	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.054355767	IUPHAR.LIGAND:5425	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
NCBIGENE:720	hgnc:1323	C4A	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:719	hgnc:1319	C3AR1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:716	hgnc:1247	C1S	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:69	hgnc:142	ACTBP9	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8501	iuphar.ligand:8501	SX-517	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.021215221	IUPHAR.LIGAND:5932	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:5946	drugbank:DB07664	K-00546	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.018359326	IUPHAR.LIGAND:5932	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:10531	iuphar.ligand:10531	BSJ-04-132	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:12074	iuphar.ligand:12074	ASNUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.2263261691193728	IUPHAR.LIGAND:5945	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	1.810609352954982	IUPHAR.LIGAND:11686	iuphar.ligand:11686	ENITOCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:10467	ncit:C139552	MEVOCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1319	ncbigene:1319	CORD1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8748	iuphar.ligand:8748	5H3'FPE	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
NCBIGENE:3133	hgnc:4962	HLA-E	GuideToPharmacology	2024.1	inhibitor	0.3500511415712966	IUPHAR.LIGAND:11101	rxcui:15657	DECITABINE	TRUE	FALSE	TRUE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:7435	rxcui:1433212	LEVOMILNACIPRAN	TRUE	FALSE	FALSE
NCBIGENE:2002	hgnc:3321	ELK1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.083744292	IUPHAR.LIGAND:7317	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1625	ncit:C80578	ETORPHINE	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1619	iuphar.ligand:1619	DYNORPHIN A-(1-13)	FALSE	FALSE	FALSE
NCBIGENE:1397	hgnc:2361	CRIP2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10245	iuphar.ligand:10245	KT-109	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:12105	iuphar.ligand:12105	COMPOUND 19 [PMID: 35925768]	FALSE	FALSE	FALSE
NCBIGENE:1397	hgnc:2361	CRIP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10243	iuphar.ligand:10243	DO34	FALSE	FALSE	FALSE
NCBIGENE:2604	hgnc:2867	DHODH	GuideToPharmacology	2024.1	inhibitor	2.763561643983921	IUPHAR.LIGAND:11469	iuphar.ligand:11469	BRD9185	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.019447286	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1400204566285186	IUPHAR.LIGAND:94	ncit:C152139	RACLOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:2833	hgnc:4540	CXCR3	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11828	ncit:C169944	ENARODUSTAT	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:11672	ncit:C167205	SUNVOZERTINIB	FALSE	FALSE	FALSE
NCBIGENE:644	hgnc:1062	BLVRA	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:3048	drugbank:DB04714	ISOPENTENYL PYROPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:2826	hgnc:4474	CCR10	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:8026	iuphar.ligand:8026	BMS-214662	FALSE	FALSE	FALSE
NCBIGENE:2533	hgnc:4036	FYB1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8797	iuphar.ligand:8797	COMPOUND 13 [PMID: 17502136]	FALSE	FALSE	FALSE
NCBIGENE:2933	ncbigene:2933	GSM1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:9557	iuphar.ligand:9557	IGE HEAVY CHAIN	FALSE	FALSE	FALSE
NCBIGENE:2022	hgnc:3349	ENG	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:8137	iuphar.ligand:8137	COMPOUND 8E [PMID: 24432909]	FALSE	FALSE	FALSE
NCBIGENE:2023	hgnc:3350	ENO1	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:8137	iuphar.ligand:8137	COMPOUND 8E [PMID: 24432909]	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1061	drugbank:DB02406	N-VALERIC ACID	FALSE	FALSE	FALSE
NCBIGENE:226	hgnc:414	ALDOA	GuideToPharmacology	2024.1	agonist	0.1293292394967845	IUPHAR.LIGAND:1059	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.1973972602845657	IUPHAR.LIGAND:8104	iuphar.ligand:8104	LY2874455	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:6043	drugbank:DB08009	SU-11652	FALSE	FALSE	FALSE
NCBIGENE:1808	hgnc:3014	DPYSL2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:9785	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12313	iuphar.ligand:12313	COMPOUND 29 [PMID: 36356320]	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:9785	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.01439355	IUPHAR.LIGAND:5679	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	NULL	0.1367387271762877	IUPHAR.LIGAND:5085	iuphar.ligand:5085	VEGFA	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.062509132	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:608	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:11024	iuphar.ligand:11024	BMS-986235	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.1312691780892362	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:1960	iuphar.ligand:1960	LATANOPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.067839369	IUPHAR.LIGAND:4146	ncit:C72111	BRETAZENIL	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.1325951293830669	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.054243462	IUPHAR.LIGAND:4360	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	agonist	0.1325951293830669	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:405	hgnc:700	ARNT	GuideToPharmacology	2024.1	modulator	0.1988926940746003	IUPHAR.LIGAND:4146	ncit:C72111	BRETAZENIL	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.2917092846427472	IUPHAR.LIGAND:3594	iuphar.ligand:3594	GALANIN-LIKE PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:643	hgnc:1060	CXCR5	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:3196	iuphar.ligand:3196	BPH-715	FALSE	FALSE	FALSE
NCBIGENE:929	hgnc:1628	CD14	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:4705	iuphar.ligand:4705	SKF89976A	FALSE	FALSE	FALSE
NCBIGENE:447	hgnc:765	ASS1P2	GuideToPharmacology	2024.1	inhibitor	0.3281729452230906	IUPHAR.LIGAND:4210	iuphar.ligand:4210	GYKI53784	FALSE	FALSE	FALSE
NCBIGENE:251	hgnc:441	ALPG	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:9479	iuphar.ligand:9479	ADOMEGLIVANT	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.305277158	IUPHAR.LIGAND:7474	rxcui:23043	DIFLUPREDNATE	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:11901	iuphar.ligand:11901	LEO 134310	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.067839369	IUPHAR.LIGAND:7088	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
NCBIGENE:452	hgnc:4581	GRIK3	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:4092	iuphar.ligand:4092	[3H]UBP310	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	modulator	0.6731752722524935	IUPHAR.LIGAND:12156	iuphar.ligand:12156	ONFASPRODIL	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.070574827	IUPHAR.LIGAND:727	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.056097939	IUPHAR.LIGAND:4084	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.070574827	IUPHAR.LIGAND:4084	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.094099769	IUPHAR.LIGAND:4268	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
NCBIGENE:256	hgnc:4421	GNRHR	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:1181	iuphar.ligand:1181	D-24710	FALSE	FALSE	FALSE
NCBIGENE:221	hgnc:410	ALDH3B1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:1014	iuphar.ligand:1014	G-1	FALSE	FALSE	FALSE
NCBIGENE:37	hgnc:92	ACADVL	GuideToPharmacology	2024.1	agonist	0.4773424657790409	IUPHAR.LIGAND:608	rxcui:2323	CHENODEOXYCHOLIC ACID	TRUE	FALSE	FALSE
NCBIGENE:1748	hgnc:2917	DLX4	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:9068	rxcui:2586354	VOSORITIDE	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	0.4565884455277783	IUPHAR.LIGAND:5786	rxcui:1546433	MONOMETHYL FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:400	hgnc:692	ARL1	GuideToPharmacology	2024.1	blocker	2.100306849	IUPHAR.LIGAND:2359	iuphar.ligand:2359	ZD7288	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:8305	iuphar.ligand:8305	TUCIDINOSTAT	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.130291988	IUPHAR.LIGAND:8366	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2615	hgnc:4161	LRRC32	GuideToPharmacology	2024.1	inhibitor	0.1909369863116163	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.058406753	IUPHAR.LIGAND:1059	rxcui:1362696	BUTYRIC ACID	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.060492709	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.1411496538593938	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.075010959	IUPHAR.LIGAND:7006	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.046425881	IUPHAR.LIGAND:1204	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:1199	iuphar.ligand:1199	OXO-ARPROMIDINE	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.067059606	IUPHAR.LIGAND:1223	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	inhibitor	0.172722603	IUPHAR.LIGAND:1234	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1257	iuphar.ligand:1257	UCL-2138	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:1263	iuphar.ligand:1263	VUF 4904	FALSE	FALSE	FALSE
NCBIGENE:2763	ncbigene:2763	GMFA	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:7695	iuphar.ligand:7695	AZD4017	FALSE	FALSE	FALSE
NCBIGENE:2763	ncbigene:2763	GMFA	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:7357	iuphar.ligand:7357	ABT-384	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2980	iuphar.ligand:2980	GLPDGG PEPTIDE [PMID: 20494585]	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:5748	iuphar.ligand:5748	COMPOUND 58 [PMID: 21273063]	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.1875273972703375	IUPHAR.LIGAND:3317	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
NCBIGENE:102	hgnc:188	ADAM10	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:9743	rxcui:28859	LODOXAMIDE TROMETHAMINE	TRUE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5561	iuphar.ligand:5561	GSK575594A	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:3622	rxcui:2001986	PALMIDROL	FALSE	FALSE	FALSE
KCNQ1	hgnc:6294	KCNQ1	PharmGKB	4/5/24	NULL	0.9546849315580819	sitagliptin	rxcui:593411	SITAGLIPTIN	TRUE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:4056	iuphar.ligand:4056	PAMP-12 (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2371	hgnc:3879	FRA1L	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8597	iuphar.ligand:8597	NTE-2	FALSE	FALSE	FALSE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
NCBIGENE:345	hgnc:610	APOC3	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:8314	ncit:C166506	ESUBERAPROST	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	0.04464938	IUPHAR.LIGAND:8741	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:5993	iuphar.ligand:5993	JAK3 INHIBITOR II	FALSE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.027433475	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
CASP3	hgnc:1504	CASP3	PharmGKB	4/5/24	NULL	0.016094305	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.075442056	IUPHAR.LIGAND:7949	iuphar.ligand:7949	AT-9283	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:12871	iuphar.ligand:12871	LEPZACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:5994	iuphar.ligand:5994	JAK3 INHIBITOR IV	FALSE	FALSE	FALSE
NCBIGENE:974	hgnc:1699	CD79B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4589	iuphar.ligand:4589	DIOA	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.006694845	IUPHAR.LIGAND:7885	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.025942525	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10383	iuphar.ligand:10383	ARS-1620	FALSE	FALSE	TRUE
TRPV1	hgnc:12716	TRPV1	PharmGKB	4/5/24	NULL	0.5122699632750684	cannabinoids	chembl:CHEMBL3833333	NABIXIMOLS	FALSE	FALSE	FALSE
TMEM43	hgnc:28472	TMEM43	PharmGKB	4/5/24	NULL	0.7242437411819931	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:7648	drugbank:DB14765	RIVOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:380	hgnc:657	ARF4P1	GuideToPharmacology	2024.1	activator	0.596678082	IUPHAR.LIGAND:2307	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:2318	iuphar.ligand:2318	NS8593	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.063568609	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:570	hgnc:932	BAAT	GuideToPharmacology	2024.1	blocker	2.386712328895204	IUPHAR.LIGAND:2606	iuphar.ligand:2606	LY97241	FALSE	FALSE	FALSE
GRIA3	hgnc:4573	GRIA3	PharmGKB	4/5/24	NULL	0.2083637747448194	venlafaxine	rxcui:39786	VENLAFAXINE	TRUE	FALSE	FALSE
NCBIGENE:538	hgnc:869	ATP7A	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:2547	iuphar.ligand:2547	MARGATOXIN	FALSE	FALSE	FALSE
NCBIGENE:539	hgnc:850	ATP5PO	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:571	hgnc:1282	GRIK1-AS2	GuideToPharmacology	2024.1	blocker	8.751278539282415	IUPHAR.LIGAND:2606	iuphar.ligand:2606	LY97241	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	blocker	2.019525817	IUPHAR.LIGAND:2592	iuphar.ligand:2592	L735821	FALSE	FALSE	FALSE
NCBIGENE:563	hgnc:910	AZGP1	GuideToPharmacology	2024.1	activator	0.546954909	IUPHAR.LIGAND:2307	ncit:C76778	FLINDOKALNER	FALSE	FALSE	FALSE
NCBIGENE:561	ncbigene:561	AZF2	GuideToPharmacology	2024.1	modulator	0.577007376	IUPHAR.LIGAND:2601	rxcui:1112990	EZOGABINE	TRUE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6717	iuphar.ligand:6717	COMPOUND 10 [PMID: 22533316]	FALSE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6722	iuphar.ligand:6722	COMPOUND 1 [GOTTELAND ET AL., 1997]	FALSE	FALSE	FALSE
NCBIGENE:2434	hgnc:3832	FRA10D	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6716	iuphar.ligand:6716	COMPOUND 8 [PMID: 22533316]	FALSE	FALSE	FALSE
SELP	hgnc:10721	SELP	PharmGKB	4/5/24	NULL	13.12691780892362	crizanlizumab-tmca	rxcui:2262279	CRIZANLIZUMAB	TRUE	FALSE	FALSE
NCBIGENE:2053	hgnc:3402	EPHX2	GuideToPharmacology	2024.1	inhibitor	0.050007306	IUPHAR.LIGAND:9404	iuphar.ligand:9404	PP2	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	2.500365296937833	IUPHAR.LIGAND:11663	iuphar.ligand:11663	MLI-2	FALSE	FALSE	FALSE
NCBIGENE:602	hgnc:998	BCL3	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:7725	iuphar.ligand:7725	AZ12260493	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	0.2187819634820604	IUPHAR.LIGAND:2755	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
NCBIGENE:2055	hgnc:2079	CLN8	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:8153	iuphar.ligand:8153	COMPOUND 22M [PMID: 19831390]	FALSE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:9500	iuphar.ligand:9500	TCLPA5	FALSE	FALSE	FALSE
NCBIGENE:2664	hgnc:4226	GDI1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:7488	iuphar.ligand:7488	MG149	FALSE	FALSE	FALSE
GSTM4	hgnc:4636	GSTM4	PharmGKB	4/5/24	NULL	0.3621218705909965	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:1217	hgnc:26439	SLC47A2	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:1231	rxcui:2541	CIMETIDINE	TRUE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1309	iuphar.ligand:1309	S36540	FALSE	FALSE	FALSE
NCBIGENE:2847	hgnc:4479	MCHR1	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:8318	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
NCBIGENE:282	hgnc:482	ANCR	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:1325	iuphar.ligand:1325	SHU9119	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6365	iuphar.ligand:6365	COMPOUND 10I [PMID: 23084894]	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	NULL	0.6177373086552294	IUPHAR.LIGAND:4949	iuphar.ligand:4949	HEPATOCYTE GROWTH FACTOR	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.061773731	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3215	drugbank:DB02509	FARNESOL	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.1458546423213736	meloxicam	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	modulator	0.3860858179095183	IUPHAR.LIGAND:6226	iuphar.ligand:6226	RO4491533	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.3860858179095183	IUPHAR.LIGAND:11614	iuphar.ligand:11614	LY395756	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6474	iuphar.ligand:6474	CIS-10 [PMID: 15771457]	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	agonist	0.077217164	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:1373	iuphar.ligand:1373	(+)-MCPG	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.2573905452730122	IUPHAR.LIGAND:1373	iuphar.ligand:1373	(+)-MCPG	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.03070624	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	modulator	0.6250913242344582	IUPHAR.LIGAND:10606	iuphar.ligand:10606	COMPOUND 3 [PMID: 31804822]	FALSE	FALSE	FALSE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.2678962818147679	IUPHAR.LIGAND:7836	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:7128	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	modulator	0.1193356164447602	IUPHAR.LIGAND:343	iuphar.ligand:343	BRUCINE N-OXIDE	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:8584	iuphar.ligand:8584	AQ-RA 741	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:6937	iuphar.ligand:6937	IPEROXO	FALSE	FALSE	FALSE
FASLG	hgnc:11936	FASLG	PharmGKB	4/5/24	NULL	0.009529523	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.2983390411119005	IUPHAR.LIGAND:6938	iuphar.ligand:6938	LY2119620	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.013259513	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.059667808	IUPHAR.LIGAND:367	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:312	iuphar.ligand:312	MUSCARINIC TOXIN 2	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:367	rxcui:69120	TIOTROPIUM	TRUE	FALSE	FALSE
SNX9	hgnc:14973	SNX9	PharmGKB	4/5/24	NULL	1.458546423213736	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
SNX9	hgnc:14973	SNX9	PharmGKB	4/5/24	NULL	4.039051633514962	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:314	iuphar.ligand:314	MUSCARINIC TOXIN 7	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1325951293830669	IUPHAR.LIGAND:313	iuphar.ligand:313	MUSCARINIC TOXIN 3	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:10667	iuphar.ligand:10667	UCSF4226	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:10667	iuphar.ligand:10667	UCSF4226	FALSE	FALSE	FALSE
NCBIGENE:287	hgnc:493	ANK2	GuideToPharmacology	2024.1	agonist	0.7095631248066824	IUPHAR.LIGAND:1350	iuphar.ligand:1350	IIK7	FALSE	FALSE	FALSE
AQP4	hgnc:637	AQP4	PharmGKB	4/5/24	NULL	0.1256164383629055	eculizumab	rxcui:591781	ECULIZUMAB	TRUE	TRUE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:1619	iuphar.ligand:1619	DYNORPHIN A-(1-13)	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.024041974	IUPHAR.LIGAND:8286	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	agonist	0.192335792	IUPHAR.LIGAND:9005	iuphar.ligand:9005	AR-M1000390	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	modulator	0.5770073762164231	IUPHAR.LIGAND:9156	iuphar.ligand:9156	BMS-986121	FALSE	FALSE	FALSE
NCBIGENE:3005	hgnc:4714	H1-0	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9931	iuphar.ligand:9931	COMPOUND 7C [PMID: 22041175]	FALSE	FALSE	FALSE
NCBIGENE:580	hgnc:952	BARD1	GuideToPharmacology	2024.1	blocker	0.6819178082557726	IUPHAR.LIGAND:10355	iuphar.ligand:10355	GNE-616	FALSE	FALSE	FALSE
NCBIGENE:581	hgnc:959	BAX	GuideToPharmacology	2024.1	blocker	0.7001022831425933	IUPHAR.LIGAND:2630	iuphar.ligand:2630	&MU;-CONOTOXIN GIIIA	FALSE	FALSE	FALSE
NCBIGENE:579	hgnc:951	NKX3-2	GuideToPharmacology	2024.1	inhibitor	0.8751278539282416	IUPHAR.LIGAND:12644	ncit:C174600	FUNAPIDE	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	activator	3.750547945	IUPHAR.LIGAND:2632	iuphar.ligand:2632	&BETA;-SCORPION TOXIN CN2	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:5733	iuphar.ligand:5733	N-ME-AMINOPYRIMIDINONE 9	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	activator	0.1562728310586145	IUPHAR.LIGAND:2626	iuphar.ligand:2626	VERATRIDINE	FALSE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	blocker	0.089298761	IUPHAR.LIGAND:10355	iuphar.ligand:10355	GNE-616	FALSE	FALSE	FALSE
NCBIGENE:583	hgnc:967	BBS2	GuideToPharmacology	2024.1	inhibitor	0.7501095890813501	IUPHAR.LIGAND:10003	iuphar.ligand:10003	GNE-131	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	modulator	0.6035364509849942	IUPHAR.LIGAND:2373	rxcui:6069	IVERMECTIN	TRUE	FALSE	FALSE
NCBIGENE:466	hgnc:783	ATF1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:4011	iuphar.ligand:4011	&ALPHA;-CONOTOXIN TXIA	FALSE	FALSE	FALSE
NCBIGENE:469	hgnc:789	ATF4P1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9472	iuphar.ligand:9472	RGIA4	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:2088	iuphar.ligand:2088	KASSININ	FALSE	FALSE	FALSE
NCBIGENE:298	hgnc:4518	NMUR1	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:7926	iuphar.ligand:7926	COMPOUND 8D [PMID: 24999562]	FALSE	FALSE	FALSE
NCBIGENE:2129	hgnc:14311	NUAK1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
P2RY12	hgnc:18124	P2RY12	PharmGKB	4/5/24	NULL	0.040515178	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	inhibitor	1.050153425	IUPHAR.LIGAND:6193	ncit:C96714	VERLUKAST	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2244	iuphar.ligand:2244	L-366,875	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2242	iuphar.ligand:2242	L-366,509	FALSE	FALSE	FALSE
NCBIGENE:323	hgnc:582	APBB2	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:5807	iuphar.ligand:5807	GLAXOSMITHKLINE COMPOUND 5H [PMID:20542694]	FALSE	FALSE	FALSE
NCBIGENE:2877	hgnc:4554	GPX2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8625	iuphar.ligand:8625	O-F-AMIDINE	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2665	iuphar.ligand:2665	TZD18	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:8907	ncit:C75189	EDAGLITAZONE	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2710	iuphar.ligand:2710	[125I]SB-236636	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:2665	iuphar.ligand:2665	TZD18	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2704	iuphar.ligand:2704	GW7845	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:2698	iuphar.ligand:2698	SB-219993	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	inhibitor	0.078136416	IUPHAR.LIGAND:3442	drugbank:DB07863	2-CHLORO-5-NITRO-N-PHENYLBENZAMIDE	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.5899738341089269	IUPHAR.LIGAND:8243	iuphar.ligand:8243	HS-173	FALSE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.5899738341089269	IUPHAR.LIGAND:12382	iuphar.ligand:12382	RISOVALISIB	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:10598	iuphar.ligand:10598	COMPOUND 41 [PMID: 31855425]	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.075768645	IUPHAR.LIGAND:7875	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:8242	iuphar.ligand:8242	PI-3065	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:6653	iuphar.ligand:6653	CZC 24832	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:8916	rxcui:2478439	UMBRALISIB	TRUE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.028598949	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	0.3070624048871023	IUPHAR.LIGAND:7202	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
NCBIGENE:1301	hgnc:2186	COL11A1	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:6962	rxcui:1091836	ROFLUMILAST	TRUE	FALSE	FALSE
NCBIGENE:1309	hgnc:8795	PDE9A	GuideToPharmacology	2024.1	inhibitor	0.5048814541893702	IUPHAR.LIGAND:2919	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:8156	iuphar.ligand:8156	COMPOUND 20 [PMID: 22136433]	FALSE	FALSE	FALSE
CYB5R1	hgnc:13397	CYB5R1	PharmGKB	4/5/24	NULL	2.100306849	rasburicase	rxcui:283821	RASBURICASE	TRUE	FALSE	FALSE
NCBIGENE:2171	hgnc:3560	FABP5	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:12396	iuphar.ligand:12396	CZS-241	FALSE	FALSE	FALSE
NCBIGENE:2171	hgnc:3560	FABP5	GuideToPharmacology	2024.1	inhibitor	0.4773424657790409	IUPHAR.LIGAND:5659	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.042689164	IUPHAR.LIGAND:2879	rxcui:1000112	MEDROXYPROGESTERONE ACETATE	TRUE	FALSE	FALSE
ADORA2A	hgnc:263	ADORA2A	PharmGKB	4/5/24	NULL	0.078840347	levodopa	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	agonist	0.4268916360625568	IUPHAR.LIGAND:3454	iuphar.ligand:3453	ORG2058	FALSE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:6489	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
NCBIGENE:627	hgnc:1033	BDNF	GuideToPharmacology	2024.1	inhibitor	0.2134458180312784	IUPHAR.LIGAND:2883	ncit:C91054	ASOPRISNIL	FALSE	FALSE	FALSE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	0.093763699	IUPHAR.LIGAND:7499	rxcui:1547545	PEMBROLIZUMAB	TRUE	TRUE	TRUE
NCBIGENE:2382	hgnc:3894	FRA2J	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:6564	iuphar.ligand:6564	PHENYLACETYL-ARG-VAL-ARG-4-AMIDINOBENZYLAMIDE	FALSE	FALSE	FALSE
PDE4D	hgnc:8783	PDE4D	PharmGKB	4/5/24	NULL	0.069454592	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:2161	hgnc:3530	F12	GuideToPharmacology	2024.1	activator	8.751278539282415	IUPHAR.LIGAND:13011	iuphar.ligand:13011	MTK458	FALSE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:4022	iuphar.ligand:4022	[125I]PRRP31	FALSE	FALSE	FALSE
NCBIGENE:337	hgnc:602	APOA4	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1557	iuphar.ligand:1557	NPY-(18-36) (HUMAN, PIG)	FALSE	FALSE	FALSE
EPM2A	hgnc:3413	EPM2A	PharmGKB	4/5/24	NULL	0.4167275494896389	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	inhibitor	0.8334550989792777	IUPHAR.LIGAND:1818	iuphar.ligand:1818	TIP39-(9-39) (HUMAN/BOVINE)	FALSE	FALSE	FALSE
NCBIGENE:331	hgnc:592	XIAP	GuideToPharmacology	2024.1	agonist	0.8334550989792777	IUPHAR.LIGAND:1813	iuphar.ligand:1813	[TYR36]-PTHRP-(1-36) AMIDE (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:736	hgnc:8600	PANX2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:1828	iuphar.ligand:1828	TIP39-(7-39) (MOUSE)	FALSE	FALSE	FALSE
NCBIGENE:332	hgnc:593	BIRC5	GuideToPharmacology	2024.1	agonist	0.2983390411119005	IUPHAR.LIGAND:1815	iuphar.ligand:1815	TIP39	FALSE	FALSE	FALSE
NCBIGENE:3006	hgnc:4716	H1-2	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:10493	iuphar.ligand:10493	COMPOUND 1 [PMID: 31465224]	FALSE	FALSE	FALSE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:12420	iuphar.ligand:12420	LV-2211	FALSE	FALSE	FALSE
NCBIGENE:598	hgnc:992	BCL2L1	GuideToPharmacology	2024.1	agonist	0.2344092465879218	IUPHAR.LIGAND:2755	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.1618110053488274	sildenafil	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:2755	drugbank:DB07080	TO-901317	FALSE	FALSE	FALSE
NCBIGENE:1527	hgnc:2563	TEX28	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:9549	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8037	iuphar.ligand:8037	GSK269962A	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:11914	iuphar.ligand:11914	INSL3 [A(5-26):B(7-27)]	FALSE	FALSE	FALSE
NCBIGENE:1525	hgnc:2559	CXADR	GuideToPharmacology	2024.1	inhibitor	7.501095891	IUPHAR.LIGAND:8248	iuphar.ligand:8248	LY2584702	FALSE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	PharmGKB	4/5/24	NULL	0.027584802	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:6997	iuphar.ligand:6997	NIBR-0213	FALSE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	0.5147810905460244	IUPHAR.LIGAND:8709	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
NCBIGENE:278	hgnc:476	AMY1C	GuideToPharmacology	2024.1	agonist	3.088686543276147	IUPHAR.LIGAND:12572	iuphar.ligand:12572	SLB736	FALSE	FALSE	FALSE
NCBIGENE:2510	hgnc:3997	FTH1P21	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:6664	iuphar.ligand:6664	MYRIOCIN	FALSE	FALSE	FALSE
NCBIGENE:279	hgnc:477	AMY2A	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:8709	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
NCBIGENE:2197	hgnc:3597	FAU	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:8049	iuphar.ligand:8049	HG-9-91-01	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	PharmGKB	4/5/24	NULL	1.944728564284981	pralsetinib	rxcui:2394936	PRALSETINIB	TRUE	FALSE	TRUE
NCBIGENE:2213	hgnc:3618	FCGR2B	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8210	iuphar.ligand:8210	COMPOUND 27 [PMID: 21123062]	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.034888818	IUPHAR.LIGAND:4621	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	PharmGKB	4/5/24	NULL	0.1715936968486748	sacituzumab govitecan	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.012822386	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:2520	hgnc:4164	GAST	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8835	iuphar.ligand:8835	COMPOUND 1J [PMID: 26314925]	FALSE	FALSE	FALSE
DDIT4	hgnc:24944	DDIT4	PharmGKB	4/5/24	NULL	0.192335792	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:1116	hgnc:1932	CHI3L1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8837	iuphar.ligand:8837	COMPOUND 16 [PMID: 19097778]	FALSE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:4587	iuphar.ligand:4587	SERGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:3235	hgnc:5140	HOXD9	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:12746	iuphar.ligand:12746	COMPOUND 14I [PMID: 37204466]	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.3500511415712967	IUPHAR.LIGAND:7957	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2024	iuphar.ligand:2024	[125I]TYR10-CST14	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5631	iuphar.ligand:5631	MALTOTRIOSE-[125I][TYR3,THR8]OCTREOTIDE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2032	iuphar.ligand:2032	BIM 23023	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.3723948314588262	IUPHAR.LIGAND:2032	iuphar.ligand:2032	BIM 23023	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:3513	iuphar.ligand:3513	NNC269100	FALSE	FALSE	FALSE
NCBIGENE:2715	ncbigene:2715	GKP5	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8388	iuphar.ligand:8388	CHAETOCIN	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.2548916079402645	IUPHAR.LIGAND:2638	drugbank:DB03176	KB-141	FALSE	FALSE	FALSE
NCBIGENE:2244	hgnc:3662	FGB	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8192	iuphar.ligand:8192	COMPOUND 5 [PMID: 23232060]	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	inhibitor	0.3241214273808302	IUPHAR.LIGAND:8144	iuphar.ligand:8144	COMPOUND 13R [PMID: 23639540]	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:10274	iuphar.ligand:10274	ASP7663	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6292	iuphar.ligand:6292	CHLOROPICRIN	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:6294	iuphar.ligand:6294	BENZYL BROMIDE	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.1084869240406911	IUPHAR.LIGAND:6281	ncit:C71146	SALIRASIB	FALSE	FALSE	TRUE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.091159151	IUPHAR.LIGAND:7088	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.7721716358190367	IUPHAR.LIGAND:4191	iuphar.ligand:4191	FLUFENAMATE	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	0.172722603	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	blocker	0.5048814541893702	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	blocker	1.458546423213736	IUPHAR.LIGAND:11860	iuphar.ligand:11860	ESTRADIOL 3-METHYL ETHER	FALSE	FALSE	FALSE
NCBIGENE:501	hgnc:877	ALDH7A1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:11860	iuphar.ligand:11860	ESTRADIOL 3-METHYL ETHER	FALSE	FALSE	FALSE
NCBIGENE:500	hgnc:17961	TRPM8	GuideToPharmacology	2024.1	blocker	2.763561643983921	IUPHAR.LIGAND:10300	iuphar.ligand:10300	PF-05105679	FALSE	FALSE	FALSE
NCBIGENE:497	hgnc:14323	TRPM5	GuideToPharmacology	2024.1	modulator	6.563458904461812	IUPHAR.LIGAND:12540	iuphar.ligand:12540	APV207094A	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	1.944728564284981	IUPHAR.LIGAND:4205	iuphar.ligand:4205	GSK1016790A	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	0.6482428547616604	IUPHAR.LIGAND:12553	drugbank:DB12290	PUERARIN	FALSE	FALSE	FALSE
NCBIGENE:509	hgnc:833	ATP5F1C	GuideToPharmacology	2024.1	blocker	4.773424657790408	IUPHAR.LIGAND:12550	iuphar.ligand:12550	VERBASCOSIDE	FALSE	FALSE	FALSE
NCBIGENE:2264	hgnc:3691	FGFR4	GuideToPharmacology	2024.1	inhibitor	1.117184494376478	IUPHAR.LIGAND:11664	iuphar.ligand:11664	LUVIXASERTIB	FALSE	FALSE	FALSE
NCBIGENE:1836	hgnc:10994	SLC26A2	GuideToPharmacology	2024.1	NULL	2.500365296937833	IUPHAR.LIGAND:4935	iuphar.ligand:4935	GROWTH ARREST SPECIFIC PROTEIN 6	FALSE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:9285	iuphar.ligand:9285	PRN694	FALSE	FALSE	FALSE
NCBIGENE:1031	hgnc:1789	CDKN2C	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:7673	rxcui:1731031	LESINURAD	TRUE	FALSE	FALSE
NCBIGENE:2246	hgnc:3665	FGF1	GuideToPharmacology	2024.1	inhibitor	0.8334550989792776	IUPHAR.LIGAND:10947	iuphar.ligand:10947	NIK INHIBITOR 12F	FALSE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:2152	iuphar.ligand:2152	U-II-(4-11) (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:2528	hgnc:4017	FUT6	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:11935	iuphar.ligand:11935	T-690	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:3842	iuphar.ligand:3842	[LYS15,ARG16,LEU27]VIP-(1-7)/GRF-(8-27)-NH2	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	agonist	0.2778183663264258	IUPHAR.LIGAND:10444	iuphar.ligand:10444	LIT-001	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1517	iuphar.ligand:1517	PYY-(3-36)	FALSE	FALSE	FALSE
NCBIGENE:308	hgnc:543	ANXA5	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1563	iuphar.ligand:1563	FMS586	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.3472729579080324	ROCILETINIB	ncit:C99905	ROCILETINIB	FALSE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	CIViC	10-Apr-24	NULL	0.023744802	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
CFLAR	hgnc:1876	CFLAR	CIViC	10-Apr-24	NULL	0.6563458904461813	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	CIViC	10-Apr-24	NULL	1.165474011072658	FGFR INHIBITOR AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.364636606	ANTI-ERBB3 MONOCLONAL ANTIBODY AV-203	ncit:C102535	ANTI-ERBB3 MONOCLONAL ANTIBODY AV-203	FALSE	TRUE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.011762471	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	2.493675356344019	LORLATINIB	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
DDR2	hgnc:2731	DDR2	CIViC	10-Apr-24	NULL	0.9546849315580819	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.011444567	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ASS1	hgnc:758	ASS1	CIViC	10-Apr-24	NULL	1.875273972703375	PEGARGIMINASE	ncit:C91702	PEGARGIMINASE	FALSE	FALSE	TRUE
KDM6A	hgnc:12637	KDM6A	CIViC	10-Apr-24	NULL	0.5000730593875666	VENETOCLAX	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
CDKN2B	hgnc:1788	CDKN2B	CIViC	10-Apr-24	NULL	0.5357925636295356	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
FANCC	hgnc:3584	FANCC	CIViC	10-Apr-24	NULL	0.112919723	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
FANCC	hgnc:3584	FANCC	CIViC	10-Apr-24	NULL	0.1448487482363986	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	0.099446347	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.546954909	MEK INHIBITOR GDC-0623	ncit:C95738	MEK INHIBITOR GDC-0623	FALSE	FALSE	TRUE
AR	hgnc:644	AR	CIViC	10-Apr-24	NULL	0.064318974	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.056826484	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
HDAC9	hgnc:14065	HDAC9	CIViC	10-Apr-24	NULL	0.2545826484154885	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
ARAF	hgnc:646	ARAF	CIViC	10-Apr-24	NULL	0.075369863	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
CIP2A	hgnc:29302	CIP2A	CIViC	10-Apr-24	NULL	0.5645986154375753	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
RRM1	hgnc:10451	RRM1	CIViC	10-Apr-24	NULL	0.1187956362798518	VINORELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
TNC	hgnc:5318	TNC	CIViC	10-Apr-24	NULL	0.070574827	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
SMARCA4	hgnc:11100	SMARCA4	CIViC	10-Apr-24	NULL	0.2524407270946851	VINORELBINE	rxcui:39541	VINORELBINE	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	1.389091831632129	RINDOPEPIMUT	ncit:C69076	RINDOPEPIMUT	FALSE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DoCM	10-Apr-24	NULL	0.8008364246019593	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.9131768910555564	Ficonalkib	ncit:C199050	FICONALKIB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.5498185469706229	BI 882370	ncit:C187123	PAN-RAF INHIBITOR XP-102	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.008206247	Celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1832728489902076	PF-07284892	ncit:C178469	SHP2 INHIBITOR PF-07284892	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	LY294002	ncit:C148229	PI3K/BET INHIBITOR LY294002	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.068727318	SAR260301	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.091636424	GSK2334470	iuphar.ligand:8008	GSK2334470	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.8561033353645842	Iruplinalkib	ncit:C154279	IRUPLINALKIB	FALSE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.6848826682916673	TAE684	ncit:C171615	ALK INHIBITOR TAE684	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.5233322714521047	Rogaratinib	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.2035181055647073	ICP-192	ncit:C178318	GUNAGRATINIB	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.033002936	Leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.2442217266776488	PHA-665752	iuphar.ligand:5700	PHA-665752	FALSE	FALSE	TRUE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.9158314750411831	Bemarituzumab	ncit:C120040	BEMARITUZUMAB	FALSE	FALSE	FALSE
KEAP1	hgnc:23177	KEAP1	JAX-CKB	10-Apr-24	NULL	1.050153425	Camrelizumab	ncit:C123816	CAMRELIZUMAB	FALSE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.1785975212098452	LY3214996	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
MDM2	hgnc:6973	MDM2	JAX-CKB	10-Apr-24	NULL	1.312691780892362	Nutlin-3a	ncit:C74594	REBEMADLIN	FALSE	FALSE	TRUE
MAP2K1	hgnc:6840	MAP2K1	JAX-CKB	10-Apr-24	NULL	0.2678962818147679	E6201	iuphar.ligand:7836	E6201	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.07699072	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2117244807890907	CCT241161	iuphar.ligand:9814	CCT241161	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.1323278004931817	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.014857858	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.1215455352678113	PF-04691502	drugbank:DB11974	PF-04691502	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.05913026	SF1126	drugbank:DB05210	SF1126	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1621858570986702	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1330430859012529	SAR260301	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.070956312	2-Methoxyestradiol	ncit:C965	2-METHOXYESTRADIOL	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.032252869	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.014906788	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.01448088	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CancerCommons	25-Jul-13	inhibitor	0.099220845	BEZ235	ncit:C74072	DACTOLISIB	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.070717402	Cediranib	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
DRD2	hgnc:3023	DRD2	ChEMBL	33	agonist	0.051885051	ROPINIROLE HYDROCHLORIDE	rxcui:236553	ROPINIROLE HYDROCHLORIDE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.1041818873724097	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
PRKCG	hgnc:9402	PRKCG	DTC	9/2/20	NULL	0.078722146	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.1648592503475494	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
SLC2A4	hgnc:11009	SLC2A4	NCI	14-Sep-17	NULL	0.021258166	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
PPP2R2A	hgnc:9304	PPP2R2A	PharmGKB	4/5/24	NULL	1.193356164447602	olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	0.33338204	ACY-1215	ncit:C96431	RICOLINOSTAT	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.2365210416022274	Methacholine Chloride	rxcui:40165	METHACHOLINE CHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	0.05073205	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:493	hgnc:817	ATP2B4	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
PALB2	hgnc:26144	PALB2	CIViC	10-Apr-24	NULL	0.546954909	MITOMYCIN	rxcui:632	MITOMYCIN	TRUE	FALSE	TRUE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.061197752	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003001553	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	ChEMBL	33	inhibitor	0.1562728310586146	AZD-8186	drugbank:DB15029	AZD-8186	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TCMDC-124353	chembl:CHEMBL529918	CHEMBL:CHEMBL529918	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.002337414	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	DNDI1416988	chembl:CHEMBL1389794	CHEMBL:CHEMBL1389794	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.069824031	ML-10302	iuphar.ligand:235	ML 10302	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.005722283	OMEPRAZOLE	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
S1PR4	hgnc:3170	S1PR4	DTC	9/2/20	NULL	0.364636606	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
CCL2	hgnc:10618	CCL2	PharmGKB	4/5/24	NULL	0.3918482928036903	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.022136455	darifenacin	rxcui:136198	DARIFENACIN	TRUE	FALSE	FALSE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.2386712328895204	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
UNIPROT:Q9UHC9	hgnc:7898	NPC1L1	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	EZETIMIBE	rxcui:341248	EZETIMIBE	TRUE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	JCAR015	ncit:C133718	VADACABTAGENE LERALEUCEL	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	3.387591692625451	TC-99M MIBI	rxcui:1482913	TECHNETIUM TC 99M SESTAMIBI	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:10185	iuphar.ligand:10185	NFP	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	DEXTROMORAMIDE	rxcui:3290	DEXTROMORAMIDE	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	agonist	0.040021091	CIPEPOFOL	ncit:C188595	CIPEPOFOL	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.029498692	WAY-100135	iuphar.ligand:79	WAY-100135	FALSE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.010975684	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	VISNAGIN	iuphar.ligand:433	VISNAGIN	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	MyCancerGenome	20-Jun-17	inhibitor	0.048083948	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	blocker	0.1630673019742065	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:1837	hgnc:3057	DTNA	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:12375	iuphar.ligand:12375	ADRIXETINIB	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.024141458	IUPHAR.LIGAND:22	rxcui:784649	ASENAPINE	TRUE	FALSE	FALSE
PLEKHH2	hgnc:30506	PLEKHH2	PharmGKB	4/5/24	NULL	1.458546423213736	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
UNIPROT:P47901	hgnc:896	AVPR1B	TdgClinicalTrial	Jan-14	NULL	3.750547945	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
RHO-ASSOCIATED PROTEIN KINASE 2	hgnc:10252	ROCK2	TTD	2020.06.01	NULL	0.3365876361262467	GSK269962A	iuphar.ligand:8037	GSK269962A	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1354	iuphar.ligand:1354	S24773	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:3977	iuphar.ligand:3976	[125I]EPIBATIDINE	FALSE	FALSE	FALSE
NCBIGENE:587	hgnc:977	BCAT2	GuideToPharmacology	2024.1	inhibitor	0.7955707762984016	IUPHAR.LIGAND:2294	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
MYCN	hgnc:7559	MYCN	CIViC	10-Apr-24	NULL	0.5000730593875667	GSK126	iuphar.ligand:7012	GSK126	FALSE	FALSE	TRUE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	(S)-ISRADIPINE	rxcui:33910	ISRADIPINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.006419031	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
GALNT18	hgnc:30488	GALNT18	PharmGKB	4/5/24	NULL	10.50153425	tocilizumab	rxcui:612865	TOCILIZUMAB	TRUE	TRUE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	DNDI1417147	chembl:CHEMBL2094484	CHEMBL:CHEMBL2094484	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	NCI	14-Sep-17	NULL	0.082043236	FLAVOPIRIDOL	ncit:C74940	ALVOCIDIB	FALSE	FALSE	TRUE
UNIPROT:O15392	hgnc:593	BIRC5	TdgClinicalTrial	Jan-14	NULL	0.1491695205559502	HGS1029	ncit:C78484	IAP INHIBITOR HGS1029	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	CIViC	10-Apr-24	NULL	0.089103927	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
RAPGEF4	hgnc:16626	RAPGEF4	DTC	9/2/20	NULL	0.077789143	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
SOD1	hgnc:11179	SOD1	PharmGKB	4/5/24	NULL	10.50153424713889	tofersen	rxcui:2634995	TOFERSEN	TRUE	FALSE	FALSE
MYLK	hgnc:7590	MYLK	DTC	9/2/20	inhibitor	0.4795221117415023	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.030527716	AG-34	chembl:CHEMBL80155	CHEMBL:CHEMBL80155	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	DIMERCAPROL	rxcui:3445	DIMERCAPROL	TRUE	FALSE	FALSE
NCBIGENE:446	hgnc:4573	GRIA3	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:4248	iuphar.ligand:4248	LY392098	FALSE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	DTC	9/2/20	NULL	0.7395446652914718	SALVINORIN A	drugbank:DB12327	SALVINORIN A	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.09669921	3,5 DIBROMOTYROSINE	chembl:CHEMBL1232132	DIBROMOTYROSINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	MINOXIDIL	rxcui:6984	MINOXIDIL	TRUE	FALSE	FALSE
MAP2K4	hgnc:6844	MAP2K4	PharmGKB	4/5/24	NULL	0.1477009036165808	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
BIRC3	hgnc:591	BIRC3	TALC	12-May-16	inhibitor	0.6250913242344582	TL 32711	ncit:C88295	BIRINAPANT	FALSE	FALSE	TRUE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.1944728564284981	SOLIFENACIN	rxcui:322167	SOLIFENACIN	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TEND	1-Aug-11	NULL	0.070197421	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.012971263	Phenylephrine	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
CYB5R4	hgnc:20147	CYB5R4	PharmGKB	4/5/24	NULL	1.050153425	isosorbide mononitrate	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.021846337	Haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
DPP6	hgnc:3010	DPP6	PharmGKB	4/5/24	NULL	0.026586163	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.032899543	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:Q02880	hgnc:11990	TOP2B	TdgClinicalTrial	Jan-14	NULL	0.036062961	DAUNORUBICIN	rxcui:214468	DAUNORUBICIN LIPOSOMAL	TRUE	FALSE	TRUE
UNIPROT:P06729	hgnc:1639	CD2	TdgClinicalTrial	Jan-14	NULL	17.50255707856483	SIPLIZUMAB	ncit:C38685	SIPLIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.090530468	IUPHAR.LIGAND:9	iuphar.ligand:9	BMY-7378	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:9619	ncit:C171928	DELGOCITINIB	FALSE	FALSE	FALSE
CREB1	hgnc:2345	CREB1	PharmGKB	4/5/24	NULL	0.4091506849534637	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	PHENFORMIN HYDROCHLORIDE	rxcui:235288	PHENFORMIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ENDOTHELIN B RECEPTOR	hgnc:3180	EDNRB	TTD	2020.06.01	NULL	3.750547945	Bosentan	rxcui:1468845	BOSENTAN ANHYDROUS	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.2738340090518618	metoprolol	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:12211	iuphar.ligand:12211	LY3023703	FALSE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.2536602475154323	METARAMINOL BITARTRATE	rxcui:6806	METARAMINOL BITARTRATE	TRUE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.2958178661165888	GSPE	ncit:C2689	IH636 GRAPE SEED PROANTHOCYANIDIN EXTRACT	FALSE	FALSE	FALSE
ABCG2	hgnc:74	ABCG2	PharmGKB	4/5/24	NULL	0.07458476	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
ADRA1D	hgnc:280	ADRA1D	PharmGKB	4/5/24	NULL	0.100976291	phenylephrine	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
HLA-DQA1	hgnc:4942	HLA-DQA1	PharmGKB	4/5/24	NULL	0.7001022831425934	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	OZARELIX	ncit:C95214	OZARELIX	FALSE	FALSE	FALSE
LONG TRANSIENT RECEPTOR POTENTIAL CHANNEL 8	hgnc:17961	TRPM8	TTD	2020.06.01	NULL	2.763561643983921	PF-05105679	drugbank:DB15450	PF-05105679	FALSE	FALSE	FALSE
NCBIGENE:2142	hgnc:8810	PDK2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:9362	iuphar.ligand:9362	AZD7545	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	NCI	14-Sep-17	NULL	0.031650194	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
TPMT	hgnc:12014	TPMT	PharmGKB	4/5/24	NULL	0.5000730593875666	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.02103111	everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TdgClinicalTrial	Jan-14	NULL	0.089756703	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.2083637747448194	LENVATINIB MESYLATE	rxcui:1604346	LENVATINIB MESYLATE	TRUE	FALSE	FALSE
UNIPROT:O75899	hgnc:4507	GABBR2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	ARBACLOFEN	ncit:C90890	ARBACLOFEN	FALSE	FALSE	FALSE
NCBIGENE:1814	hgnc:3024	DRD3	GuideToPharmacology	2024.1	inhibitor	0.027781837	IUPHAR.LIGAND:7426	rxcui:1603296	LENVATINIB	TRUE	FALSE	TRUE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:1919	ncit:C84191	SULPROSTONE	FALSE	FALSE	FALSE
HDAC3	hgnc:4854	HDAC3	TALC	12-May-16	inhibitor	0.295540363	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
FYN	hgnc:4037	FYN	NCI	14-Sep-17	NULL	0.2083637747448194	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
UNIPROT:P30542	hgnc:262	ADORA1	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	T-62	drugbank:DB12919	T-62	FALSE	FALSE	FALSE
UNIPROT:P05067	hgnc:620	APP	TdgClinicalTrial	Jan-14	NULL	2.423430980108977	GANTENERUMAB	ncit:C88580	GANTENERUMAB	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.1058622403945453	BENZQUINAMIDE	rxcui:19041	BENZQUINAMIDE	TRUE	FALSE	FALSE
UNIPROT:P28476	hgnc:4091	GABRR2	TdgClinicalTrial	Jan-14	NULL	0.1121958787087489	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
ADA	hgnc:186	ADA	ChEMBL	33	inhibitor	3.043922970185188	PENTOSTATIN	rxcui:8011	PENTOSTATIN	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	FDA	10-Apr-24	NULL	0.2333674277141977	Imatinib	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
PTGDR2	hgnc:4502	PTGDR2	ChEMBL	33	inhibitor	0.9211872146613068	FEVIPIPRANT	ncit:C166588	FEVIPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:537	hgnc:868	ATP6AP1	GuideToPharmacology	2024.1	blocker	1.750255707856483	IUPHAR.LIGAND:7718	iuphar.ligand:7718	Z944	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002436325	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.6482428547616604	N-(3-OXODODECANOYL)HOMOSERINELACTONE	chembl:CHEMBL8483	CHEMBL:CHEMBL8483	FALSE	FALSE	FALSE
HDAC4	hgnc:14063	HDAC4	TALC	12-May-16	inhibitor	0.2403097081725148	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.105015342	OLSALAZINE SODIUM	rxcui:104123	OLSALAZINE SODIUM	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	ChEMBL	33	inhibitor	0.08572681	TEMUTERKIB	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
PDE7B	hgnc:8792	PDE7B	ChEMBL	33	inhibitor	1.640864726115453	FLAVOXATE HYDROCHLORIDE	rxcui:142437	FLAVOXATE HYDROCHLORIDE	TRUE	FALSE	FALSE
HDAC7	hgnc:14067	HDAC7	TALC	12-May-16	inhibitor	0.218327115	PCI-24781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
PDE2A	hgnc:8777	PDE2A	ChEMBL	33	inhibitor	0.375054795	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.069454592	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	GNF-PF-1083	chembl:CHEMBL530361	CHEMBL:CHEMBL530361	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.047561296	2-AMINOETHOXYDIPHENYL BORATE	iuphar.ligand:2433	2-APB	FALSE	FALSE	FALSE
JAK2	hgnc:6192	JAK2	TALC	12-May-16	inhibitor	0.1037701012563132	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
TUBA3E	hgnc:20765	TUBA3E	ChEMBL	33	inhibitor	0.040021091	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.5147810905460245	SHO-SAIKO-TO	ncit:C2690	SHO-SAIKO-TO	FALSE	FALSE	FALSE
NCBIGENE:1988	hgnc:16627	CHEK2	GuideToPharmacology	2024.1	inhibitor	0.5147810905460244	IUPHAR.LIGAND:9549	ncit:C91392	PREXASERTIB	FALSE	FALSE	TRUE
ACHE	hgnc:108	ACHE	ChEMBL	33	activator	1.544343271638073	PRALIDOXIME CHLORIDE	rxcui:55322	PRALIDOXIME CHLORIDE	TRUE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.018860514	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.011834048	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2191733444543002	SALBUTAMOL	rxcui:142153	ALBUTEROL SULFATE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.1215455352678113	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
PIK3R1	hgnc:8979	PIK3R1	ChEMBL	33	inhibitor	0.1682938180631233	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.010470124	MIBEFRADIL	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.001276813	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	0.375054795	dactinomycin	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
UNIPROT:P43220	hgnc:4324	GLP1R	TdgClinicalTrial	Jan-14	NULL	0.9546849315580818	ALBIGLUTIDE	rxcui:1534763	ALBIGLUTIDE	TRUE	FALSE	FALSE
MELANOMA-ASSOCIATED ANTIGEN 3	hgnc:6801	MAGEA3	TTD	2020.06.01	NULL	17.50255707856483	GL-0817	ncit:C166968	BIROPEPIMUT-S	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008345148	PYRROLIDINE DITHIOCARBAMATE	chembl:CHEMBL399491	PYRROLIDINE DITHIOCARBAMATE	FALSE	FALSE	FALSE
NCBIGENE:33	hgnc:88	ACADL	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:9384	iuphar.ligand:9384	P32 [PMID: 27108698]	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	modulator	0.040021091	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
CBFB	hgnc:1539	CBFB	DTC	9/2/20	NULL	0.1262203635473425	D-DOPA	chembl:CHEMBL211670	CHEMBL:CHEMBL211670	FALSE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	0.525076712	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2051080907644316	FURAFYLLINE	ncit:C65779	FURAFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P16234	hgnc:8803	PDGFRA	TdgClinicalTrial	Jan-14	NULL	0.1434635826111871	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE SGK1	hgnc:10810	SGK1	TTD	2020.06.01	NULL	0.9723642821424908	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.056500364	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
PROTEIN TYROSINE PHOSPHATASE	hgnc:10989	SLC25A3	TTD	2020.06.01	NULL	13.12691780892362	INCB13739	drugbank:DB05064	INCB13739	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.069824031	ETHOPROPAZINE	rxcui:4134	PROFENAMINE	TRUE	FALSE	FALSE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1912847768149162	PIRARUBICIN	rxcui:33764	PIRARUBICIN	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.059397818	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
DHODH	hgnc:2867	DHODH	NCI	14-Sep-17	NULL	0.3070624048871023	IMMUNOSUPPRESSIVE	ncit:C574	IMMUNOSUPPRESSANT	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.035098711	IUPHAR.LIGAND:320	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
UNIPROT:P08069	hgnc:5465	IGF1R	TdgClinicalTrial	Jan-14	NULL	0.440315901	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.058645947	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:1991	hgnc:3309	ELANE	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:9655	iuphar.ligand:9655	TAKINIB	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4168	iuphar.ligand:4168	D-AP5	FALSE	FALSE	FALSE
UNIPROT:P07900	hgnc:5253	HSP90AA1	TdgClinicalTrial	Jan-14	NULL	0.3621218705909965	ALVESPIMYCIN	ncit:C38142	ALVESPIMYCIN	FALSE	FALSE	TRUE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:12472	iuphar.ligand:12472	3&BETA;-HYDROXYDIHYDROCOSTUNOLIDE	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	activator	1.312691780892362	IUPHAR.LIGAND:4303	iuphar.ligand:4303	RYANODINE	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:4303	iuphar.ligand:4303	RYANODINE	FALSE	FALSE	FALSE
UNIPROT:P06756	hgnc:6150	ITGAV	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	CILENGITIDE	ncit:C1834	CILENGITIDE	FALSE	FALSE	TRUE
RET	hgnc:9967	RET	DTC	9/2/20	NULL	0.015434354	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
NCBIGENE:244	hgnc:4133	GALR2	GuideToPharmacology	2024.1	agonist	0.8751278539282416	IUPHAR.LIGAND:6135	iuphar.ligand:6135	GALANIN(9-29) (RAT/MOUSE)	FALSE	FALSE	FALSE
UNIPROT:P34995	hgnc:9593	PTGER1	TdgClinicalTrial	Jan-14	NULL	0.4892019059226195	ALPROSTADIL	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
NCBIGENE:669	hgnc:1093	BPGM	GuideToPharmacology	2024.1	agonist	7.501095891	IUPHAR.LIGAND:12451	iuphar.ligand:12451	D-(-)-AMYGDALIN	FALSE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.06466462	IUPHAR.LIGAND:5677	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.019490598	TRITON X	chembl:CHEMBL39763	TRITON X	FALSE	FALSE	FALSE
POLE3	hgnc:13546	POLE3	ChEMBL	33	inhibitor	0.094099769	GEMCITABINE HYDROCHLORIDE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.025147352	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.6105543166941221	IUPHAR.LIGAND:7901	ncit:C75168	DAPOXETINE	TRUE	FALSE	FALSE
UNIPROT:Q8TCU5	hgnc:16767	GRIN3A	TdgClinicalTrial	Jan-14	NULL	0.3195192975802911	KETAMINE	rxcui:203184	KETAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	agonist	1.014640990061729	DESMOPRESSIN ACETATE	rxcui:3251	DESMOPRESSIN	TRUE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.1548898856510162	DNDI1417692	chembl:CHEMBL1481509	CHEMBL:CHEMBL1481509	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.8334550989792777	Zalutumumab	ncit:C64620	ZALUTUMUMAB	FALSE	FALSE	TRUE
NCBIGENE:1937	hgnc:3213	EEF1G	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:8355	iuphar.ligand:8355	COMPOUND 46 [PMID: 16451062]	FALSE	FALSE	FALSE
UNIPROT:Q13258	hgnc:9591	PTGDR	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	AM-461	iuphar.ligand:10170	AM-461	FALSE	FALSE	FALSE
MCL1	hgnc:32041	ADAMTSL4-AS1	DTC	9/2/20	NULL	0.093763699	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	NCI	14-Sep-17	NULL	0.084553416	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1232574442152452	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
NCBIGENE:3096	hgnc:4920	HIVEP1	GuideToPharmacology	2024.1	NULL	10.50153424713889	IUPHAR.LIGAND:11966	iuphar.ligand:11966	MRTX0902	FALSE	FALSE	FALSE
DRD3	hgnc:3024	DRD3	PharmGKB	4/5/24	NULL	0.069454592	levodopa	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
UNIPROT:P34913	hgnc:3402	EPHX2	TdgClinicalTrial	Jan-14	NULL	2.250328767244049	AR9281	drugbank:DB06345	AR-9281	FALSE	FALSE	FALSE
UNIPROT:P25942	hgnc:11919	CD40	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	LUCATUMUMAB	ncit:C48405	LUCATUMUMAB	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	CIViC	10-Apr-24	NULL	0.8643238063488805	LESTAURTINIB	ncit:C48402	LESTAURTINIB	FALSE	FALSE	TRUE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.3684748858645228	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.1254663589861278	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
CD33	hgnc:1659	CD33	PharmGKB	4/5/24	NULL	2.423430980108977	gemtuzumab ozogamicin	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
UNIPROT:P07099	hgnc:3401	EPHX1	TdgClinicalTrial	Jan-14	NULL	2.019525817	AR9281	drugbank:DB06345	AR-9281	FALSE	FALSE	FALSE
UNIPROT:Q15842	hgnc:6269	KCNJ8	TdgClinicalTrial	Jan-14	NULL	3.281729452230906	THIAMYLAL	rxcui:10464	THIAMYLAL	TRUE	FALSE	FALSE
ACE	hgnc:2707	ACE	PharmGKB	4/5/24	NULL	0.7026004179620139	enalapril	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
INTERFERON-BETA	hgnc:5434	IFNB1	TTD	2020.06.01	NULL	26.25383561784724	PF-06823859	chembl:CHEMBL4297808	PF-06823859	FALSE	FALSE	FALSE
UNIPROT:Q16539	hgnc:6876	MAPK14	TdgClinicalTrial	Jan-14	NULL	0.1902451856365742	ARRY-797	iuphar.ligand:11095	ARRY-371797	FALSE	FALSE	FALSE
TLR4	hgnc:11850	TLR4	NCI	14-Sep-17	NULL	0.4565884455277783	HEAT SHOCK PROTEIN 70	ncit:C28696	RECOMBINANT 70-KD HEAT-SHOCK PROTEIN	FALSE	FALSE	FALSE
NCBIGENE:227	hgnc:4499	FFAR3	GuideToPharmacology	2024.1	agonist	3.281729452230906	IUPHAR.LIGAND:1061	drugbank:DB02406	N-VALERIC ACID	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.00389812	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.075714018	IL-6	iuphar.ligand:4998	IL-6	FALSE	FALSE	FALSE
UNIPROT:Q02763	hgnc:11724	TEK	TdgClinicalTrial	Jan-14	NULL	0.364636606	ARRY-614	ncit:C85481	PEXMETINIB	FALSE	FALSE	FALSE
ATG16L1	hgnc:21498	ATG16L1	PharmGKB	4/5/24	NULL	3.182283105193606	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:1613	iuphar.ligand:1613	[LEU]ENKEPHALIN	FALSE	FALSE	FALSE
UNIPROT:Q9UGN5	hgnc:272	PARP2	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	MK-4827	rxcui:1918231	NIRAPARIB	TRUE	FALSE	TRUE
UNIPROT:Q96GD4	hgnc:11390	AURKB	TdgClinicalTrial	Jan-14	NULL	0.284980577	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.9211872146613069	DOXACURIUM	rxcui:23651	DOXACURIUM	TRUE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.046798281	IUPHAR.LIGAND:320	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.016558711	Duvelisib	rxcui:2058509	DUVELISIB	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	TCMDC-125142	chembl:CHEMBL528791	CHEMBL:CHEMBL528791	FALSE	FALSE	FALSE
NFIB	hgnc:7785	NFIB	PharmGKB	4/5/24	NULL	0.3918482928036902	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.020423054	ZINC 02849675	chembl:CHEMBL605959	CHEMBL:CHEMBL605959	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.016206071	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
FOS	hgnc:3796	FOS	NCI	14-Sep-17	NULL	0.2625383561784725	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
MAP2K1	hgnc:6840	MAP2K1	TALC	12-May-16	inhibitor	0.7143900848393808	RDEA119	ncit:C74059	REFAMETINIB	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.045265234	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
MST1R	hgnc:7381	MST1R	DTC	9/2/20	NULL	0.039778539	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	FDA	10-Apr-24	NULL	0.030996264	Flibanserin	rxcui:1665509	FLIBANSERIN	TRUE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.750109589	PIXY	ncit:C1477	MILODISTIM	FALSE	FALSE	FALSE
UNIPROT:P02751	hgnc:3778	FN1	TdgClinicalTrial	Jan-14	NULL	1.346350544504987	AS1409	drugbank:DB05182	AS1409	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.036212187	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	MMV667491	chembl:CHEMBL1437888	CHEMBL:CHEMBL1437888	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.2800409132570373	PROSTAGLANDIN D2	drugbank:DB02056	PROSTAGLANDIN D2	FALSE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.1591141552596803	NITROGEN MUSTARD	rxcui:6674	MECHLORETHAMINE	TRUE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.9376369863516875	PEFLOXACIN	rxcui:7960	PEFLOXACIN	TRUE	FALSE	FALSE
UNIPROT:P09871	hgnc:1247	C1S	TdgClinicalTrial	Jan-14	NULL	0.5834185692854945	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
CPT1A	hgnc:2328	CPT1A	PharmGKB	4/5/24	NULL	0.09972967	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:9635	rxcui:1988390	LATANOPROSTENE BUNOD	TRUE	FALSE	FALSE
EML4	hgnc:1316	EML4	JAX-CKB	10-Apr-24	NULL	0.5707355569097228	NUV-655	ncit:C188054	ALK INHIBITOR NVL-655	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1193356164447602	MMV667491	chembl:CHEMBL1437888	CHEMBL:CHEMBL1437888	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	3,6-DIMETHOXYFLAVONE	chembl:CHEMBL1331521	3,6-DIMETHOXYFLAVONE	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	PharmGKB	4/5/24	NULL	0.01524613	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	2.940429589198891	rasburicase	rxcui:283821	RASBURICASE	TRUE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.004636439	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	0.3070624048871023	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	ChEMBL	33	inhibitor	0.036463661	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.2692701089009974	NIALAMIDE	rxcui:7394	NIALAMIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.004197256	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
MLANA	hgnc:7124	MLANA	NCI	14-Sep-17	NULL	0.7778914257139926	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
PSMC1P1	hgnc:30147	PSMC1P1	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
GRK4	hgnc:4543	GRK4	PharmGKB	4/5/24	NULL	1.458546423213736	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
TUMOR-ASSOCIATED CALCIUM SIGNAL TRANSDUCER 1	hgnc:11529	EPCAM	TTD	2020.06.01	NULL	6.300920548	Citatuzumab bogatox	ncit:C71694	CITATUZUMAB BOGATOX	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.012649403	DIHYDREXIDINE	drugbank:DB12890	DIHYDREXIDINE	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.025111273	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
UNIPROT:P03951	hgnc:3529	F11	TdgClinicalTrial	Jan-14	NULL	0.3070624048871023	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	3.500511415712966	NABILONE	rxcui:31447	NABILONE	TRUE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	1.050153425	IUPHAR.LIGAND:720	rxcui:426	ALANINE	TRUE	FALSE	FALSE
KCNK18	hgnc:19439	KCNK18	ChEMBL	33	potentiator	0.2838252499226729	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P08684	hgnc:2637	CYP3A4	TdgClinicalTrial	Jan-14	NULL	0.058733413	AVI-4557	drugbank:DB05447	AVI-4557	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.019332721	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.016027983	fluoxetine	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.079557078	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.06375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
NOREPINEPHRINE TRANSPORTER	hgnc:11048	SLC6A2	TTD	2020.06.01	NULL	0.2453629496995069	TD-9855	chembl:CHEMBL4297646	AMPRELOXETINE	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:4150	rxcui:2045371	CANNABIDIOL	TRUE	FALSE	FALSE
NCBIGENE:2191	hgnc:3590	FAP	GuideToPharmacology	2024.1	inhibitor	0.4039051633514962	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	SJ000031505	chembl:CHEMBL589479	CHEMBL:CHEMBL589479	FALSE	FALSE	FALSE
HDAC11	hgnc:19086	HDAC11	DTC	9/2/20	NULL	0.2447910080918158	PSAMMAPLIN A	chembl:CHEMBL83747	PSAMMAPLIN A	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	7-CHLOROKYNURENIC ACID	chembl:CHEMBL311389	7-CHLOROKYNURENIC ACID	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.008504644	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.009659248	CHELERYTHRINE	drugbank:DB17024	CHELERYTHRINE	FALSE	FALSE	FALSE
PRKCA	hgnc:9393	PRKCA	MyCancerGenome	20-Jun-17	inhibitor	0.027693919	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
BGLAP	hgnc:1043	BGLAP	NCI	14-Sep-17	NULL	0.2580229544751573	CLODRONATE	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.1226814748497534	CYCLOFENIL	rxcui:2983	CYCLOFENIL	TRUE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.082043236	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1666910197958555	IZORLISIB	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
KCNJ8	hgnc:6269	KCNJ8	ChEMBL	33	potentiator	1.640864726115453	SARAKALIM	ncit:C72978	SARAKALIM	FALSE	FALSE	FALSE
NCBIGENE:269	hgnc:465	AMHR2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3334	ncit:C96710	POBILUKAST	FALSE	FALSE	FALSE
NCBIGENE:671	hgnc:1095	BPI	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:7163	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
UNIPROT:Q9H4B7	hgnc:16257	TUBB1	TdgClinicalTrial	Jan-14	NULL	0.077789143	OMBRABULIN	ncit:C78480	OMBRABULIN	FALSE	FALSE	FALSE
NCBIGENE:1392	hgnc:2355	CRH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:10265	iuphar.ligand:10265	GGSTOP	FALSE	FALSE	FALSE
CDKN1B	hgnc:1785	CDKN1B	NCI	14-Sep-17	NULL	0.8334550989792776	TOMUDEX	rxcui:196239	RALTITREXED	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.020936073	DAIDZEIN	ncit:C1060	DAIDZEIN	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.013532905	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.099446347	NORTRIPTYLINE HYDROCHLORIDE	rxcui:203130	NORTRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	agonist	0.1193356164447602	IUPHAR.LIGAND:6937	iuphar.ligand:6937	IPEROXO	FALSE	FALSE	FALSE
VCAM1	hgnc:12663	VCAM1	NCI	14-Sep-17	NULL	0.3804903712731485	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
UNIPROT:Q09470	hgnc:6218	KCNA1	TEND	1-Aug-11	NULL	0.2419708351875322	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
UNIPROT:P26010	hgnc:6162	ITGB7	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	R1295	drugbank:DB05122	R1295	FALSE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TdgClinicalTrial	Jan-14	NULL	0.2237542808339254	PHENACEMIDE	rxcui:33253	PHENACEMIDE	TRUE	FALSE	FALSE
NCBIGENE:29	hgnc:81	ABR	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:546	iuphar.ligand:546	NIP	FALSE	FALSE	FALSE
NCBIGENE:981	hgnc:23089	SLC13A5	GuideToPharmacology	2024.1	inhibitor	10.50153424713889	IUPHAR.LIGAND:12849	iuphar.ligand:12849	PF-06649298	FALSE	FALSE	FALSE
CD4	hgnc:1678	CD4	NCI	14-Sep-17	NULL	3.281729452230906	HERBIMYCIN	ncit:C1124	HERBIMYCIN	FALSE	FALSE	FALSE
UNIPROT:P05106	hgnc:6156	ITGB3	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	GANTOFIBAN	ncit:C73227	GANTOFIBAN	FALSE	FALSE	FALSE
PROLACTIN RECEPTOR	hgnc:9446	PRLR	TTD	2020.06.01	NULL	8.751278539282415	Prolanta	drugbank:DB18431	PROLACTIN G129R	FALSE	FALSE	FALSE
CA7	hgnc:1381	CA7	ChEMBL	33	inhibitor	1.458546423213736	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	OncoKB	23-Jul-20	NULL	1.374546367426557	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.101562227	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
NCBIGENE:890	hgnc:1578	CCNA2	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:8737	iuphar.ligand:8737	IGN523	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	DROMETRIZOLE	rxcui:1426903	DROMETRIZOLE	FALSE	FALSE	FALSE
ARAP1	hgnc:16925	ARAP1	PharmGKB	4/5/24	NULL	2.917092846427472	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
UNIPROT:P00742	hgnc:3528	F10	TdgClinicalTrial	Jan-14	NULL	0.2381300282797936	ANTITHROMBIN	rxcui:1427179	ANTITHROMBIN ALFA	TRUE	FALSE	FALSE
PRKD1	hgnc:9407	PRKD1	MyCancerGenome	20-Jun-17	inhibitor	0.066465407	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.1143957978991165	BGJ398	rxcui:2550729	INFIGRATINIB	TRUE	FALSE	TRUE
DEFB4	hgnc:2767	DEFB4A	NCI	14-Sep-17	NULL	0.8751278539282416	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
ITGA5	hgnc:6141	ITGA5	TALC	12-May-16	antibody	4.375639269641208	VOLOCIXIMAB	ncit:C48426	VOLOCIXIMAB	FALSE	FALSE	TRUE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.010097629	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.057197899	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
UNIPROT:P00734	hgnc:3535	F2	TdgClinicalTrial	Jan-14	NULL	2.763561643983921	BIVALIRUDIN	rxcui:60819	BIVALIRUDIN	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.0403388	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:P41597	hgnc:1603	CCR2	TdgClinicalTrial	Jan-14	NULL	3.424413341458336	CCX140	ncit:C175798	ILACIRNON	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.2019525816757481	IUPHAR.LIGAND:5443	rxcui:5033	GUANABENZ	TRUE	FALSE	FALSE
NCBIGENE:1835	hgnc:905	AXL	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:10574	iuphar.ligand:10574	COMPOUND 1 [CRUZ-L&OACUTE;PEZ ET AL., 2019]	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.085796848	IUPHAR.LIGAND:1223	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	inhibitor	1.944728564284981	IUPHAR.LIGAND:1547	iuphar.ligand:1547	BIIE0246	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	NSC-405662	chembl:CHEMBL118378	CHEMBL:CHEMBL118378	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.033487035	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TdgClinicalTrial	Jan-14	NULL	0.083257407	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	FDA	10-Apr-24	NULL	5.966780822238011	Elexacaftor	rxcui:2256951	ELEXACAFTOR	TRUE	FALSE	FALSE
PPP1R18	hgnc:29413	PPP1R18	PharmGKB	4/5/24	NULL	0.5966780822238011	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ADRB3	hgnc:288	ADRB3	ChEMBL	33	agonist	1.500219178	AMIBEGRON HYDROCHLORIDE	ncit:C97276	AMIBEGRON HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TdgClinicalTrial	Jan-14	NULL	0.100976291	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	vaccine	4.375639269641208	TECEMOTIDE	ncit:C2195	EMEPEPIMUT-S	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.090634645	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.025588534	THYROXINE	chembl:CHEMBL42115	THYROXINE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.00524657	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.025427444	N6-PHENYLADENOSINE	chembl:CHEMBL262083	N6-PHENYLADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:432	hgnc:742	ASGR1	GuideToPharmacology	2024.1	inhibitor	0.2885036881082116	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	0.2957715794844315	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	CIViC	10-Apr-24	NULL	0.1364544470782081	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.1187956362798518	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
POLA1	hgnc:9173	POLA1	ChEMBL	33	inhibitor	0.546954909	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
NCBIGENE:2844	hgnc:4476	GPR21	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8320	iuphar.ligand:8320	ABT-737	FALSE	FALSE	FALSE
NCBIGENE:1395	hgnc:2358	CRHR2	GuideToPharmacology	2024.1	activator	3.750547945	IUPHAR.LIGAND:10562	iuphar.ligand:10562	4-OME-ARM1	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:9586	iuphar.ligand:9586	AZ7188	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	0.4839416703750644	MAPK INHIBITORS	ncit:C2149	MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.047049885	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.007416338	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P09884	hgnc:9173	POLA1	TdgClinicalTrial	Jan-14	NULL	1.036335616	CLOFARABINE	rxcui:44151	CLOFARABINE	TRUE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.005569924	BUTHIONINE SULFOXIMINE	ncit:C1029	BUTHIONINE SULFOXIMINE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.039598545	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.061197752	IUPHAR.LIGAND:6511	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:9192	iuphar.ligand:9192	PROBE 2.1 [PMID: 24187130]	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.059667808	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
TNF SUPERFAMILY RECEPTOR 12A	hgnc:18152	TNFRSF12A	TTD	2020.06.01	NULL	105.0153424713889	Enavatuzumab	ncit:C80045	ENAVATUZUMAB	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	NCI	14-Sep-17	NULL	0.07699072	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
CDK15	hgnc:14434	CDK15	ChEMBL	33	inhibitor	0.4688184931758437	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.023110771	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.053145416	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
MATK	hgnc:6906	MATK	DTC	9/2/20	NULL	0.063568609	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.5000730593875666	NOCICEPTIN	iuphar.ligand:1681	NOCICEPTIN/ORPHANIN FQ	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.087318744	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
CTLA4	hgnc:2505	CTLA4	NCI	14-Sep-17	NULL	0.1141471113819445	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
UNIPROT:P51168	hgnc:10600	SCNN1B	TEND	1-Aug-11	NULL	1.544343271638073	AMILORIDE	rxcui:644	AMILORIDE	TRUE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.02271093	TRICETIN	rxcui:1994358	TRICETIN	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.027276712	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.014985066	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	GLICLAZIDE	rxcui:4816	GLICLAZIDE	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.048083948	ZOLPIDEM TARTRATE	rxcui:221183	ZOLPIDEM TARTRATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	NALTALIMIDE	ncit:C174856	NALTALIMIDE	FALSE	FALSE	FALSE
PSEN1	hgnc:9508	PSEN1	ChEMBL	33	modulator	0.6731752722524935	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	agonist	0.2011788169949981	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:10277	iuphar.ligand:10277	YNT-185	FALSE	FALSE	FALSE
UNIPROT:P22894	hgnc:7175	MMP8	TdgClinicalTrial	Jan-14	NULL	0.2678962818147678	COLLAGENASE	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.1474934585272317	IUPHAR.LIGAND:12075	iuphar.ligand:12075	VULOLISIB	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.1304538415793652	TAE226	iuphar.ligand:9382	NVP-TAE 226	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.1154014752432846	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
PAX8	hgnc:8622	PAX8	DTC	9/2/20	NULL	0.2651902587661338	BETA-NAPHTHOFLAVONE	ncit:C29812	BETA-NAPHTHOFLAVONE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	(S)-NIMODIPINE	chembl:CHEMBL255033	(S)-NIMODIPINE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.1458546423213736	TCMDC-124240	chembl:CHEMBL582764	CHEMBL:CHEMBL582764	FALSE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.1014640990061729	AMITRIPTYLINE	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	TALC	12-May-16	inhibitor	0.440315901	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	2.187819634820604	BENZTHIAZIDE	rxcui:19008	BENZTHIAZIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	CEFDITORIN PIVOXIL	chembl:CHEMBL1514735	CEFDITORIN PIVOXIL	FALSE	FALSE	FALSE
PIK3CB	hgnc:8976	PIK3CB	NCI	14-Sep-17	NULL	0.2778183663264258	BACILLUS CALMETTE-GUERIN	hemonc:59	BCG VACCINE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	5-CHLORO-[1,10]PHENANTHROLINE	chembl:CHEMBL317115	CHEMBL:CHEMBL317115	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	positive modulator	2.282942227638891	JNJ-39393406	drugbank:DB11867	JNJ-39393406	FALSE	FALSE	FALSE
HTR3B	hgnc:5298	HTR3B	ChEMBL	33	inhibitor	0.4412409347537352	MOSAPRIDE	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
UNIPROT:A5X5Y0	hgnc:24005	HTR3E	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	DDP225	chembl:CHEMBL5095232	DDP-225	FALSE	FALSE	FALSE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.059397818	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
UNIPROT:P26439	hgnc:5218	HSD3B2	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	TRILOSTANE	rxcui:38668	TRILOSTANE	TRUE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	2.983390411119005	IUPHAR.LIGAND:4342	rxcui:1243041	IVACAFTOR	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.032837818	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
COMT	hgnc:2228	COMT	PharmGKB	4/5/24	NULL	0.1562728310586145	propranolol	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
BLM	hgnc:1058	BLM	DTC	9/2/20	NULL	0.050978322	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
UNIPROT:P03956	hgnc:7155	MMP1	TdgClinicalTrial	Jan-14	NULL	0.093763699	COLLAGENASE	rxcui:2475861	COLLAGENASE CLOSTRIDIUM HISTOLYTICUM-AAES	TRUE	FALSE	FALSE
PDGFB	hgnc:8800	PDGFB	CancerCommons	25-Jul-13	inhibitor	0.3977853881492008	AXITINIB	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.1472177698197042	OSPEMIFENE	rxcui:1370971	OSPEMIFENE	TRUE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	0.729273212	SIMPINICLINE	ncit:C179121	SIMPINICLINE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.024932417	Arsenic trioxide	rxcui:18330	ARSENIC TRIOXIDE	TRUE	FALSE	TRUE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.017502557	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.5147810905460245	PODOCARIC ACID	chembl:CHEMBL421115	PODOCARIC ACID	FALSE	FALSE	FALSE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.2083637747448194	CUDC-101	drugbank:DB12174	CUDC-101	FALSE	FALSE	TRUE
UNIPROT:Q96KS0	hgnc:14660	EGLN2	TdgClinicalTrial	Jan-14	NULL	3.500511415712966	FG-2216	drugbank:DB08687	FG-2216	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.7876150685354175	Tafenoquine	rxcui:2054023	TAFENOQUINE	TRUE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.036951211	LARGAZOLE	chembl:CHEMBL1173445	LARGAZOLE	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	TALC	12-May-16	inhibitor	1.165474011072658	AZD4547	ncit:C88272	FEXAGRATINIB	FALSE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.4817217544559128	REMIFENTANIL	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
NOS3	hgnc:7876	NOS3	PharmGKB	4/5/24	NULL	0.4688184931758437	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
GLI1	hgnc:4317	GLI1	NCI	14-Sep-17	NULL	0.064111931	ALL-TRANS RETINOIC ACID	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
UNIPROT:Q9GZT9	hgnc:1232	EGLN1	TdgClinicalTrial	Jan-14	NULL	1.591141552596802	FG-2216	drugbank:DB08687	FG-2216	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	inhibitor	0.087222045	BRIVANIB ALANINATE	ncit:C53397	BRIVANIB ALANINATE	FALSE	FALSE	FALSE
TFRC	hgnc:11763	TFRC	ChEMBL	33	inhibitor	17.50255707856483	A27.15	chembl:CHEMBL2109494	A27.15	FALSE	FALSE	FALSE
RPL11	hgnc:10301	RPL11	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TdgClinicalTrial	Jan-14	NULL	0.062608511	ALPRAZOLAM	rxcui:596	ALPRAZOLAM	TRUE	FALSE	FALSE
NCBIGENE:531	hgnc:1393	CACNA1F	GuideToPharmacology	2024.1	activator	0.3125456621172291	IUPHAR.LIGAND:4065	iuphar.ligand:4065	(-)-(S)-BAYK8644	FALSE	FALSE	FALSE
NCBIGENE:1566	ncbigene:1566	CYP2D7BP	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9683	iuphar.ligand:9683	COMPOUND 3V [PMID: 27390066]	FALSE	FALSE	FALSE
NCBIGENE:1483	ncbigene:1483	CTAA1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:5263	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
ACP5	hgnc:124	ACP5	NCI	14-Sep-17	NULL	0.4039051633514962	ANALGESICS	ncit:C241	ANALGESIC AGENT	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.064347636	PSEUDOEPHEDRINE	rxcui:8896	PSEUDOEPHEDRINE	TRUE	FALSE	FALSE
UNIPROT:P20138	hgnc:1659	CD33	TEND	1-Aug-11	NULL	2.423430980108977	GEMTUZUMAB OZOGAMICIN	rxcui:1294580	GEMTUZUMAB OZOGAMICIN	TRUE	FALSE	TRUE
ITGAM	hgnc:6149	ITGAM	NCI	14-Sep-17	NULL	0.5147810905460245	CLARITHROMYCIN	rxcui:21212	CLARITHROMYCIN	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	S-166659	chembl:CHEMBL252417	CHEMBL:CHEMBL252417	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.014883127	L-NOREPINEPHRINE	chembl:CHEMBL18824	L-NOREPINEPHRINE	FALSE	FALSE	FALSE
LEPR	hgnc:6554	LEPR	ChEMBL	33	agonist	3.500511415712967	METRELEPTIN	rxcui:1491625	METRELEPTIN	TRUE	FALSE	FALSE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.3889457128569963	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
UGT1A5	hgnc:12537	UGT1A5	PharmGKB	4/5/24	NULL	0.5385402178019949	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004216468	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
UNIPROT:P31751	hgnc:392	AKT2	TdgClinicalTrial	Jan-14	NULL	0.6482428547616604	GDC-0068	ncit:C91072	IPATASERTIB	FALSE	FALSE	TRUE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	2.500365296937833	IUPHAR.LIGAND:2332	iuphar.ligand:2332	MAUROTOXIN	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	ChEMBL	33	inhibitor	0.4039051633514962	LITHIUM CARBONATE	rxcui:42351	LITHIUM CARBONATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.069180068	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.1491695205559502	PROPRANOLOL	rxcui:82084	PROPRANOLOL HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:11316	iuphar.ligand:11316	RADIOPROTECTIN-1	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	SJ000079774	chembl:CHEMBL601192	CHEMBL:CHEMBL601192	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.042276708	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.3889457128569962	TDR77225	chembl:CHEMBL1353528	CHEMBL:CHEMBL1353528	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.064190307	SJ000072878	chembl:CHEMBL601400	CHEMBL:CHEMBL601400	FALSE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	inhibitor	0.1302273592155121	FULVESTRANT	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	1.250182648468916	PF-05089771	drugbank:DB14856	PF-05089771	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	modulator	0.072927321	EPOTHILONE D	ncit:C2672	EPOTHILONE D	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.042174836	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
GRIN3A	hgnc:16767	GRIN3A	PharmGKB	4/5/24	NULL	0.078722146	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.024651489	SCLEROTIORIN	chembl:CHEMBL1095515	SCLEROTIORIN	FALSE	FALSE	FALSE
UNIPROT:P11802	hgnc:1773	CDK4	TdgClinicalTrial	Jan-14	NULL	0.3704244884352345	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
ATIC	hgnc:794	ATIC	DTC	9/2/20	NULL	1.680245479542224	PEMETREXED	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
CACNA2D2	hgnc:1400	CACNA2D2	ChEMBL	33	modulator	0.1442518440541058	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.015498132	FLOXURIDINE	rxcui:4488	FLOXURIDINE	TRUE	FALSE	TRUE
MAP3K10	hgnc:6849	MAP3K10	DTC	9/2/20	NULL	0.1198805279353755	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.021805511	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
ANKK1	hgnc:21027	ANKK1	PharmGKB	4/5/24	NULL	0.4167275494896389	quetiapine	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.3125456621172291	CC-1088	ncit:C2210	SELECTIVE CYTOKINE INHIBITORY DRUG CC-1088	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	8-GERANYLOXY PSORALEN	chembl:CHEMBL1412710	CHEMBL:CHEMBL1412710	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	ChEMBL	33	inhibitor	0.042619863	SU-9516	drugbank:DB03428	SU9516	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	0.4412409347537352	IUPHAR.LIGAND:7890	ncit:C82390	AFURESERTIB	FALSE	FALSE	FALSE
NCBIGENE:294	hgnc:4598	GRM6	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:3359	iuphar.ligand:3359	HOMO-AMPA	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.050488145	IUPHAR.LIGAND:333	iuphar.ligand:333	N-DESMETHYLCLOZAPINE	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	OncoKB	23-Jul-20	NULL	0.2041114528112516	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	0.4449802647092754	BENAZEPRIL	rxcui:18867	BENAZEPRIL	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1458546423213736	VU001171	iuphar.ligand:6228	VU0001171	FALSE	FALSE	FALSE
CDH1	hgnc:1748	CDH1	TALC	12-May-16	NULL	13.12691780892362	COMBRETASTATIN-A4 PHOSPHATE	chembl:CHEMBL2105643	FOSBRETABULIN TROMETHAMINE	FALSE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.1037701012563132	LURASIDONE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	inhibitor	0.4605936073306534	CANRENONE	rxcui:1982	CANRENONE	TRUE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:3413	iuphar.ligand:3413	[3H]LTB4	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.037505479	GF-109203	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
RNF8	hgnc:10071	RNF8	PharmGKB	4/5/24	NULL	0.7778914257139925	trastuzumab	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
RECQL	hgnc:9948	RECQL	NCI	14-Sep-17	NULL	0.00416232	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
PDE5A	hgnc:8784	PDE5A	ChEMBL	33	inhibitor	0.1406455479527531	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	ChEMBL	33	inhibitor	0.056826484	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	GUAIFENESIN	rxcui:5032	GUAIFENESIN	TRUE	FALSE	FALSE
L3MBTL1	hgnc:15905	L3MBTL1	DTC	9/2/20	NULL	0.2386712328895204	NSC-175743	chembl:CHEMBL1609016	CHEMBL:CHEMBL1609016	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.036062961	SILMITASERTIB	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	CRUFOMATE	ncit:C75214	CRUFOMATE	FALSE	FALSE	FALSE
TXNIP	hgnc:16952	TXNIP	NCI	14-Sep-17	NULL	26.25383561784724	FAS-LIGAND	ncit:C1538	RECOMBINANT FAS LIGAND	FALSE	FALSE	FALSE
UNIPROT:P11387	hgnc:11986	TOP1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344583	CAMPTOTHECIN	ncit:C338	CAMPTOTHECIN	TRUE	FALSE	TRUE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.4449802647092754	IUPHAR.LIGAND:279	ncit:C73316	FLUPERLAPINE	FALSE	FALSE	FALSE
RTKN2	hgnc:19364	RTKN2	PharmGKB	4/5/24	NULL	1.381780822	haloperidol	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	ChEMBL	33	inhibitor	0.056826484	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
TYRO3	hgnc:12446	TYRO3	DTC	9/2/20	NULL	0.091159151	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.037398626	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
FIBROBLAST GROWTH FACTOR RECEPTOR 4	hgnc:3691	FGFR4	TTD	2020.06.01	NULL	1.117184494376478	INCB62079	ncit:C143067	FGFR4 ANTAGONIST INCB062079	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.021431703	ERIBULIN MESYLATE	rxcui:1045452	ERIBULIN MESYLATE	TRUE	FALSE	TRUE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.049442252	OXCARBAZEPINE	rxcui:32624	OXCARBAZEPINE	TRUE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.09869863	IUPHAR.LIGAND:11691	iuphar.ligand:11691	ICI-199441	FALSE	FALSE	FALSE
NCBIGENE:2824	hgnc:4461	GPM6B	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:12931	iuphar.ligand:12931	LUNA18	FALSE	FALSE	FALSE
NCBIGENE:1240	hgnc:2121	CMKLR1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:5240	ncit:C81112	FENCLONINE	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	modulator	0.6035364509849942	IUPHAR.LIGAND:4000	iuphar.ligand:4000	NS1738	FALSE	FALSE	FALSE
NCBIGENE:2909	hgnc:4591	ARHGAP35	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9261	iuphar.ligand:9261	LUMINESPIB	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	PharmGKB	4/5/24	NULL	0.029515273	protriptyline	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
ADA	hgnc:186	ADA	NCI	14-Sep-17	NULL	0.108711535	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.7143900848393808	RETINYL PALMITATE	rxcui:35406	VITAMIN A PALMITATE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	NCI	14-Sep-17	NULL	0.021846337	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.2083637747448194	TG100-115	drugbank:DB05552	TG100-115	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.039420174	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
UNIPROT:Q01726	hgnc:6929	MC1R	TdgClinicalTrial	Jan-14	NULL	1.071585127259071	BREMELANOTIDE	rxcui:2176312	BREMELANOTIDE	TRUE	FALSE	FALSE
NCBIGENE:1921	hgnc:19679	AAK1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11688	iuphar.ligand:11688	BMS-911172	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.043180651	Fulvestrant	rxcui:282357	FULVESTRANT	TRUE	FALSE	TRUE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.08914715	Loratadine	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:6946	iuphar.ligand:6946	COMPOUND 11D  [PMID: 23981898]	FALSE	FALSE	FALSE
NCBIGENE:536	hgnc:1395	CACNA1H	GuideToPharmacology	2024.1	blocker	0.07631929	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:1377	hgnc:9599	PTGES	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9709	iuphar.ligand:9709	COMPOUND III [PMID: 24045148]	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3822	iuphar.ligand:3822	[3H]GR100679	FALSE	FALSE	FALSE
UNIPROT:Q00534	hgnc:1777	CDK6	TdgClinicalTrial	Jan-14	NULL	0.9723642821424906	LEE011	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
TRANSLOCATOR PROTEIN	hgnc:1158	TSPO	TTD	2020.06.01	NULL	0.062808219	Prazepam	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.8468979231563628	(R)-EDELFOSINE	chembl:CHEMBL107514	(R)-EDELFOSINE	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TdgClinicalTrial	Jan-14	NULL	0.2465148884304905	ALKS 37	chembl:CHEMBL2364619	METHYLSAMIDORPHAN	FALSE	FALSE	FALSE
UNIPROT:P21397	hgnc:6833	MAOA	TdgClinicalTrial	Jan-14	NULL	1.795134059339982	ISOCARBOXAZID	rxcui:6011	ISOCARBOXAZID	TRUE	FALSE	FALSE
NCBIGENE:2873	hgnc:4549	GPS1	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8606	iuphar.ligand:8606	JZL195	FALSE	FALSE	FALSE
PCGF3	hgnc:10066	PCGF3	PharmGKB	4/5/24	NULL	5.527123287967842	enalapril	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.022296251	METHANANDAMIDE	iuphar.ligand:2506	R-(+)-METHANANDAMIDE	FALSE	FALSE	FALSE
UNIPROT:P49810	hgnc:9509	PSEN2	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	SEMAGACESTAT	ncit:C81115	SEMAGACESTAT	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	DIMETHYL GAMBOGATE	chembl:CHEMBL1436860	DIMETHYL GAMBOGATE	FALSE	FALSE	FALSE
LINC00251	hgnc:31950	LINC00251	PharmGKB	4/5/24	NULL	0.7001022831425934	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
VASOPRESSIN V1B RECEPTOR	hgnc:896	AVPR1B	TTD	2020.06.01	NULL	0.6250913242344582	Mozavaptan	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
RAD50	hgnc:9816	RAD50	CGI	2/1/22	NULL	0.8334550989792777	Irinotecan	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
TIE1	hgnc:11809	TIE1	ChEMBL	33	inhibitor	6.563458904461812	CP-459632	chembl:CHEMBL3545300	CP-459632	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1232574442152452	KRN-633	iuphar.ligand:6057	VEGF RECEPTOR TYROSINE KINASE INHIBITOR III	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.084146909	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:3451	iuphar.ligand:3451	RU28318	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:7780	iuphar.ligand:7780	CIFEA	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	agonist	0.5585922471882393	IUPHAR.LIGAND:2060	iuphar.ligand:2060	[125I]TYR11-SRIF-14	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.1092771513750145	RETINOIDS	ncit:C804	RETINOIC ACID AGENT	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.019142425	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	1.432027397337122	CIMICOXIB	ncit:C77551	CIMICOXIB	FALSE	FALSE	FALSE
NHLH1	hgnc:7817	NHLH1	PharmGKB	4/5/24	NULL	0.7242437411819931	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.290901226	METHYLENE BLUE	rxcui:2198975	METHYLENE BLUE ANHYDROUS	TRUE	FALSE	FALSE
PTGER3	hgnc:9595	PTGER3	ChEMBL	33	agonist	1.458546423213736	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:Q07869	hgnc:9232	PPARA	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	NAVEGLITAZAR	ncit:C75191	NAVEGLITAZAR	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.1052961321571413	ETOMIDATE	rxcui:4177	ETOMIDATE	TRUE	FALSE	FALSE
NCBIGENE:365	hgnc:4468	UTS2R	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:9436	iuphar.ligand:9436	[3-IODO-TYR6]U-II-(4-11) (HUMAN)	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.001255969	ASPIRIN	rxcui:1191	ASPIRIN	TRUE	FALSE	TRUE
NCBIGENE:1396	hgnc:2360	CRIP1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10246	iuphar.ligand:10246	LEI105	FALSE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	0.3671865121377238	IUPHAR.LIGAND:7907	iuphar.ligand:7907	7-HYDROXYSTAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:2198	iuphar.ligand:2198	RWJ-351647	FALSE	FALSE	FALSE
NT5C2	hgnc:8022	NT5C2	CIViC	10-Apr-24	NULL	0.7778914257139925	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.03233231	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.3500511415712966	MELANOMA VACCINE	ncit:C2517	MELANOMA VACCINE	FALSE	FALSE	FALSE
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	SUVN-502	drugbank:DB06140	SUVN-502	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.025676123	BROXYQUINOLINE	ncit:C73253	BROXYQUINOLINE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.038382801	NSC-175743	chembl:CHEMBL1609016	CHEMBL:CHEMBL1609016	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.6731752722524935	RAMIPRIL	rxcui:35296	RAMIPRIL	TRUE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.018288983	7,8,2'-TRIHYDROXYFLAVONE	chembl:CHEMBL244707	CHEMBL:CHEMBL244707	FALSE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.052229116	THIORIDAZINE HYDROCHLORIDE	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
CDK13	hgnc:1733	CDK13	ChEMBL	33	inhibitor	0.5000730593875666	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
SSTR3	hgnc:11332	SSTR3	ChEMBL	33	agonist	0.8334550989792776	VAPREOTIDE	ncit:C1429	VAPREOTIDE	TRUE	FALSE	TRUE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.7001022831425934	pegaspargase	rxcui:34132	PEGASPARGASE	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.058997383	SULISOBENZONE	rxcui:1311567	SULISOBENZONE	TRUE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	DTC	9/2/20	NULL	0.012466209	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.010216825	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
ADENOSINE A2A RECEPTOR	hgnc:263	ADORA2A	TTD	2020.06.01	NULL	0.7095631248066824	AMP-579	chembl:CHEMBL1950650	CHEMBL:CHEMBL1950650	FALSE	FALSE	FALSE
SRPK1	hgnc:11305	SRPK1	DTC	9/2/20	NULL	0.040515178	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
DRD3	hgnc:3024	DRD3	DTC	9/2/20	NULL	0.1666910197958555	SKF-75670 HYDROBROMIDE	chembl:CHEMBL1256698	CHEMBL:CHEMBL1256698	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	SJ000154295	chembl:CHEMBL578502	CHEMBL:CHEMBL578502	FALSE	FALSE	FALSE
FFAR1	hgnc:4498	FFAR1	DTC	9/2/20	NULL	1.875273972703375	AMG-837	iuphar.ligand:6485	AMG-837	FALSE	FALSE	FALSE
PNPT1	hgnc:23166	PNPT1	PharmGKB	4/5/24	NULL	5.527123287967842	enalapril	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
HEAT SHOCK PROTEIN 20	hgnc:26511	HSPB6	TTD	2020.06.01	NULL	52.50767123569449	AZX-100	drugbank:DB06323	AZX-100	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:8439	iuphar.ligand:8439	ABT-670	FALSE	FALSE	FALSE
NCBIGENE:2833	hgnc:4540	CXCR3	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11831	ncit:C152811	VADADUSTAT	FALSE	FALSE	FALSE
TRANSTHYRETIN	hgnc:12405	TTR	TTD	2020.06.01	NULL	17.50255707856483	ISIS-TTRRx	rxcui:2099289	INOTERSEN	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:7206	rxcui:11404	KETOTIFEN FUMARATE	TRUE	FALSE	FALSE
NQO1	hgnc:2874	NQO1	DTC	9/2/20	NULL	2.019525817	NSC-640559	chembl:CHEMBL1287866	CHEMBL:CHEMBL1287866	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.003934927	LEVOTHYROXINE	rxcui:10582	LEVOTHYROXINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	DTC	9/2/20	NULL	0.9546849315580818	VALDECOXIB	rxcui:278567	VALDECOXIB	TRUE	FALSE	FALSE
CREBBP	hgnc:2348	CREBBP	DTC	9/2/20	NULL	0.045898314	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
PARP2	hgnc:272	PARP2	ChEMBL	33	inhibitor	2.187819634820604	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	1.712206670729168	MACITENTAN	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
ACVR2B	hgnc:174	ACVR2B	ChEMBL	33	inhibitor	8.751278539282415	BIMAGRUMAB	ncit:C116852	BIMAGRUMAB	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	MIRVETUXIMAB SORAVTANSINE	rxcui:2621548	MIRVETUXIMAB SORAVTANSINE	TRUE	FALSE	FALSE
UNIPROT:O14746	hgnc:11730	TERT	TdgClinicalTrial	Jan-14	NULL	3.000438356	IMETELSTAT	ncit:C49084	IMETELSTAT	FALSE	FALSE	TRUE
NCBIGENE:2104	hgnc:3474	ESRRG	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:4907	iuphar.ligand:4907	DORSOMORPHIN	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	inhibitor	0.019490598	IUPHAR.LIGAND:2210	iuphar.ligand:2210	[PHAA1,D-TYR(ME)2,ARG6,TYR-NH29]AVP	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	2.386712328895204	Felbinac	rxcui:262307	FELBINAC	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.02550154	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
SRGN	hgnc:9361	SRGN	NCI	14-Sep-17	NULL	3.281729452230906	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	CancerCommons	25-Jul-13	inhibitor	0.2041114528112516	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1193356164447602	OLSALAZINE SODIUM	rxcui:104123	OLSALAZINE SODIUM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.065092154	MESALAZINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	ChEMBL	33	binder	2.019525817	YTTRIUM Y 90 TACATUZUMAB TETRAXETAN	chembl:CHEMBL2108669	YTTRIUM Y 90 TACATUZUMAB TETRAXETAN	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.4526523382387456	HT-0712	drugbank:DB11650	HT-0712	FALSE	FALSE	FALSE
UNIPROT:P38435	hgnc:4247	GGCX	TdgClinicalTrial	Jan-14	NULL	0.7242437411819931	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
UNIPROT:P21917	hgnc:3025	DRD4	TdgClinicalTrial	Jan-14	NULL	0.06502498	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
NCBIGENE:32	hgnc:85	ACACB	GuideToPharmacology	2024.1	agonist	1.693795846312725	IUPHAR.LIGAND:572	iuphar.ligand:572	N-METHYL-PHE-LYS-PRO-D-CHA-CHA-D-ARG-CO2H	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:12277	iuphar.ligand:12277	COMPOUND 5G [PMID: 36385925]	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:4031	iuphar.ligand:4031	DODECYLPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:12484	iuphar.ligand:12484	YL5084	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.030746697	APOMORPHINE	rxcui:1043	APOMORPHINE	TRUE	FALSE	FALSE
CHRM3	hgnc:1952	CHRM3	ChEMBL	33	inhibitor	0.2660861718025059	UMECLIDINIUM BROMIDE	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
AVPR2	hgnc:897	AVPR2	ChEMBL	33	inhibitor	0.7955707762984013	MOZAVAPTAN	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
RPL32	hgnc:10336	RPL32	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.3017682254924971	ENSIFENTRINE	ncit:C166674	ENSIFENTRINE	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	OT-730	drugbank:DB16112	OT-730	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.054020238	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.4605936073306534	IUPHAR.LIGAND:4146	ncit:C72111	BRETAZENIL	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.00630647	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.175610941	GEMFIBROZIL	rxcui:4719	GEMFIBROZIL	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.012001753	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.023598953	DNDI1416975	chembl:CHEMBL1415851	CHEMBL:CHEMBL1415851	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.023987059	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.6543011991986852	PHENTERMINE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.068369364	TAK-715	drugbank:DB16108	TAK-715	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	ZK-164015	chembl:CHEMBL184074	CHEMBL:CHEMBL184074	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.4167275494896388	PKI-166	iuphar.ligand:7642	PKI166	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007441563	MICONAZOLE	rxcui:42790	MICONAZOLE NITRATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.010824092	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	MyCancerGenome	20-Jun-17	inhibitor	0.005112724	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
GFAP	hgnc:4235	GFAP	NCI	14-Sep-17	NULL	0.1000146118775133	TCDD	iuphar.ligand:9642	TCDD	FALSE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.42006137	METAGLIDASEN	chembl:CHEMBL451321	METAGLIDASEN	FALSE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.044878351	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	PharmGKB	4/5/24	NULL	0.049349315	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:P36888	hgnc:3765	FLT3	TdgClinicalTrial	Jan-14	NULL	0.5672124979164529	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
UNIPROT:P01579	hgnc:5438	IFNG	TdgClinicalTrial	Jan-14	NULL	3.750547945	FONTOLIZUMAB	ncit:C87765	FONTOLIZUMAB	FALSE	FALSE	FALSE
UNIPROT:P17181	hgnc:5432	IFNAR1	TEND	1-Aug-11	NULL	0.8751278539282416	INTERFERON BETA-1B	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
TRANSFORMATION-SENSITIVE PROTEIN P120	hgnc:497	TRPA1	TTD	2020.06.01	NULL	4.375639269641208	Menthol	rxcui:1430390	RACEMENTHOL	TRUE	FALSE	FALSE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:2765	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	0.2430910705356226	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.3571950424196904	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.007308974	BITHIONOLATE SODIUM	ncit:C171717	BITHIONOLATE SODIUM	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	CIS-4-AMINOCROTONIC ACID	iuphar.ligand:4148	CACA	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.1367387271762877	BUTACLAMOL	ncit:C81088	BUTACLAMOL	FALSE	FALSE	FALSE
UNIPROT:Q00613	hgnc:5224	HSF1	TdgClinicalTrial	Jan-14	NULL	13.12691780892362	BIMOCLOMOL	ncit:C171764	BIMOCLOMOL	FALSE	FALSE	FALSE
UNIPROT:P25103	hgnc:11526	TACR1	TdgClinicalTrial	Jan-14	NULL	2.838252499226729	CASOPITANT	ncit:C71635	CASOPITANT	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	1.250182648468916	MF101	drugbank:DB05052	MF101	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:12048	iuphar.ligand:12048	COMPOUND 13 [PMID: 35653642]	FALSE	FALSE	FALSE
AR	hgnc:644	AR	CancerCommons	25-Jul-13	inhibitor	0.035982643	ENZALUTAMIDE	rxcui:1307298	ENZALUTAMIDE	TRUE	FALSE	TRUE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1193356164447602	AMOXAPINE	rxcui:722	AMOXAPINE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1193356164447602	BENZYDAMINE	rxcui:1425	BENZYDAMINE	TRUE	FALSE	FALSE
GRM4	hgnc:4596	GRM4	DTC	9/2/20	NULL	7.501095891	N-(3-(TRIFLUOROMETHOXY)PHENYL)PICOLINAMIDE	chembl:CHEMBL559271	CHEMBL:CHEMBL559271	FALSE	FALSE	FALSE
UNIPROT:P03372	hgnc:3467	ESR1	TdgClinicalTrial	Jan-14	NULL	0.2453629496995069	FISPEMIFENE	ncit:C65687	FISPEMIFENE	FALSE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.038608582	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
NCBIGENE:2379	hgnc:3891	FRA2G	GuideToPharmacology	2024.1	antibody	4.375639269641208	IUPHAR.LIGAND:9094	rxcui:2055640	LANADELUMAB-FLYO	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.108711535	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	0.4102161815288632	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	KRT-232	ncit:C116624	NAVTEMADLIN	FALSE	FALSE	FALSE
MPO	hgnc:7218	MPO	NCI	14-Sep-17	NULL	0.2059124362184098	LIDOCAINE	rxcui:6387	LIDOCAINE	TRUE	FALSE	FALSE
BRCA2	hgnc:1101	BRCA2	CGI	2/1/22	NULL	0.3509871071904712	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CGI	2/1/22	NULL	1.389091831632129	Rindopepimut	ncit:C69076	RINDOPEPIMUT	FALSE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.065092154	MESALAMINE	rxcui:52582	MESALAMINE	TRUE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	CGI	2/1/22	NULL	0.2041114528112516	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
UNIPROT:P04233	hgnc:1697	CD74	TdgClinicalTrial	Jan-14	NULL	52.50767123569449	MILATUZUMAB	ncit:C66983	MILATUZUMAB	FALSE	TRUE	TRUE
NOTCH1	hgnc:7881	NOTCH1	CGI	2/1/22	NULL	1.406455479527531	Pf-03084014	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
NF1	hgnc:7765	NF1	CGI	2/1/22	NULL	0.2739530673166669	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CGI	2/1/22	NULL	0.011762471	Gemcitabine	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
CCND1	hgnc:1582	CCND1	CGI	2/1/22	NULL	0.063784829	Palbociclib	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	CGI	2/1/22	NULL	0.046059361	Osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	CGI	2/1/22	NULL	0.007555061	Trametinib	rxcui:1425098	TRAMETINIB DIMETHYL SULFOXIDE	TRUE	FALSE	TRUE
UNIPROT:Q01959	hgnc:11049	SLC6A3	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	MODAFINIL	rxcui:30125	MODAFINIL	TRUE	FALSE	FALSE
PTCH1	hgnc:9585	PTCH1	CGI	2/1/22	NULL	0.6908904109959803	Foretinib	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
TPMT	hgnc:12014	TPMT	CGI	2/1/22	NULL	0.051731696	Cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HRH1	hgnc:5182	HRH1	ChEMBL	33	inhibitor	0.08914715	LORATADINE	rxcui:28889	LORATADINE	TRUE	FALSE	FALSE
HRH1	hgnc:5182	HRH1	ChEMBL	33	agonist	0.2117244807890907	HISTAMINE PHOSPHATE	rxcui:26925	HISTAMINE PHOSPHATE	TRUE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1848861663228679	MP0112	iuphar.ligand:8371	ABICIPAR PEGOL	FALSE	FALSE	FALSE
IMPDH1	hgnc:6052	IMPDH1	ChEMBL	33	inhibitor	0.1842374429322614	RIBAVIRIN	rxcui:9344	RIBAVIRIN	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	ChEMBL	33	inhibitor	0.3226277802500429	CERTOLIZUMAB PEGOL	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.0296486	PROCHLORPERAZINE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
CALCR	hgnc:1440	CALCR	ChEMBL	33	agonist	13.12691780892362	CALCITONIN SALMON	rxcui:36118	SALMON CALCITONIN	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	ChEMBL	33	inhibitor	0.3860858179095183	OLSALAZINE SODIUM	rxcui:104123	OLSALAZINE SODIUM	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.068191781	ESCITALOPRAM OXALATE	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	1.419126249613364	MN-305	drugbank:DB05339	MN-305	FALSE	FALSE	FALSE
IGF1R	hgnc:5465	IGF1R	ChEMBL	33	agonist	0.9907107780319716	MECASERMIN	rxcui:274403	MECASERMIN	TRUE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	ChEMBL	33	inhibitor	0.8334550989792776	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
INSR	hgnc:6091	INSR	ChEMBL	33	agonist	0.042459033	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
GHR	hgnc:4263	GHR	ChEMBL	33	agonist	5.250767123569449	SOMATREM	rxcui:56570	SOMATREM	TRUE	FALSE	FALSE
HTR2A	hgnc:5293	HTR2A	ChEMBL	33	inhibitor	0.1262203635473425	PALIPERIDONE PALMITATE	rxcui:679314	PALIPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P15391	hgnc:1633	CD19	TdgClinicalTrial	Jan-14	NULL	0.5122699632750684	MT-103	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
DPEP1	hgnc:3002	DPEP1	ChEMBL	33	inhibitor	4.375639269641208	CILASTATIN SODIUM	rxcui:82128	CILASTATIN SODIUM	TRUE	FALSE	FALSE
NR3C2	hgnc:7979	NR3C2	ChEMBL	33	agonist	1.381780822	DESOXYCORTICOSTERONE ACETATE	rxcui:258333	DESOXYCORTICOSTERONE ACETATE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	ChEMBL	33	modulator	0.087512785	RALOXIFENE HYDROCHLORIDE	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.2408608772279564	PROPOXYPHENE HYDROCHLORIDE	rxcui:71517	PROPOXYPHENE HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	REMIFENTANIL HYDROCHLORIDE	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.4817217544559128	DIHYDROCODEINE BITARTRATE	rxcui:104966	DIHYDROCODEINE BITARTRATE	TRUE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	other/unknown	0.3241214273808302	DEXTROAMPHETAMINE SACCHARATE	rxcui:221088	DEXTROAMPHETAMINE SACCHARATE	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.3006164383722967	LOTEPREDNOL ETABONATE	rxcui:237027	LOTEPREDNOL	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2226788432387383	MOMETASONE FUROATE	rxcui:108118	MOMETASONE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.030850571	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	ChEMBL	33	agonist	0.2404931506978374	FLUOCINOLONE ACETONIDE	rxcui:4461	FLUOCINOLONE ACETONIDE	TRUE	FALSE	FALSE
DHFR	hgnc:2861	DHFR	ChEMBL	33	inhibitor	2.734774543525755	PRALATREXATE	rxcui:662019	PRALATREXATE	TRUE	FALSE	TRUE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	other/unknown	0.1635752997996713	DEXTROAMPHETAMINE SACCHARATE	rxcui:221088	DEXTROAMPHETAMINE SACCHARATE	TRUE	FALSE	FALSE
PDE4A	hgnc:8780	PDE4A	ChEMBL	33	inhibitor	0.6819178082557726	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P20963	hgnc:1677	CD247	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	MT-103	rxcui:1597258	BLINATUMOMAB	TRUE	FALSE	FALSE
HMGCR	hgnc:5006	HMGCR	ChEMBL	33	inhibitor	1.458546423213736	CERIVASTATIN SODIUM	rxcui:221072	CERIVASTATIN SODIUM	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.9376369863516875	ESOMEPRAZOLE MAGNESIUM	rxcui:283562	ESOMEPRAZOLE MAGNESIUM	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.1875273972703375	PANTOPRAZOLE SODIUM	rxcui:253191	PANTOPRAZOLE SODIUM	TRUE	FALSE	FALSE
ATP4B	hgnc:820	ATP4B	ChEMBL	33	inhibitor	0.06466462	DEXLANSOPRAZOLE	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
OPRD1	hgnc:8153	OPRD1	ChEMBL	33	agonist	0.3889457128569962	CODEINE POLISTIREX	rxcui:1545976	CODEINE ANHYDROUS	TRUE	FALSE	FALSE
OPRK1	hgnc:8154	OPRK1	ChEMBL	33	agonist	0.2465148884304905	CODEINE SULFATE	rxcui:91104	CODEINE SULFATE	TRUE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	inhibitor	0.1605739181519709	NALMEFENE HYDROCHLORIDE	rxcui:236069	NALMEFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TdgClinicalTrial	Jan-14	NULL	0.351221881	SUMATRIPTAN	rxcui:37418	SUMATRIPTAN	TRUE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	ChEMBL	33	inhibitor	0.6731752722524935	LITHIUM CITRATE	rxcui:52105	LITHIUM CITRATE	TRUE	FALSE	FALSE
GRIN3B	hgnc:16768	GRIN3B	ChEMBL	33	inhibitor	0.106290832	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2C	hgnc:4587	GRIN2C	ChEMBL	33	inhibitor	0.044573575	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
GRIN2B	hgnc:4586	GRIN2B	ChEMBL	33	inhibitor	0.035430277	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1684738114514262	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
GRIN2D	hgnc:4588	GRIN2D	ChEMBL	33	inhibitor	0.1023541349623674	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2B	hgnc:282	ADRA2B	ChEMBL	33	agonist	0.3125456621172291	APRACLONIDINE HYDROCHLORIDE	rxcui:91350	APRACLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	ChEMBL	33	agonist	0.1902451856365742	ALFUZOSIN HYDROCHLORIDE	rxcui:46043	ALFUZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.2692701089009974	PHENYLEPHRINE BITARTRATE	rxcui:91167	PHENYLEPHRINE BITARTRATE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	agonist	0.182318303	METARAMINOL BITARTRATE	rxcui:6806	METARAMINOL BITARTRATE	TRUE	FALSE	FALSE
UNIPROT:P20594	hgnc:7944	NPR2	TdgClinicalTrial	Jan-14	NULL	4.375639269641208	NESIRITIDE	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	agonist	0.2692701089009974	METARAMINOL BITARTRATE	rxcui:6806	METARAMINOL BITARTRATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1193356164447602	BISMUTH SUBSALICYLATE	rxcui:19478	BISMUTH SUBSALICYLATE	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.3818739726232327	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	ChEMBL	33	inhibitor	0.3938075342677087	DIFLUNISAL	rxcui:3393	DIFLUNISAL	TRUE	FALSE	FALSE
PTGS2	hgnc:9605	PTGS2	ChEMBL	33	inhibitor	0.1591141552596802	TOLMETIN SODIUM	rxcui:42935	TOLMETIN SODIUM	TRUE	FALSE	FALSE
GUCY1A2	hgnc:4684	GUCY1A2	ChEMBL	33	activator	0.2917092846427472	ISOSORBIDE MONONITRATE	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	ChEMBL	33	blocker	0.7501095890813498	REPAGLINIDE	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
ADRA1D	hgnc:280	ADRA1D	ChEMBL	33	inhibitor	0.089756703	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ADRA2A	hgnc:281	ADRA2A	ChEMBL	33	inhibitor	0.067839369	TOLAZOLINE HYDROCHLORIDE	rxcui:235450	TOLAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	3.938075342677087	NBI-98854	rxcui:1918219	VALBENAZINE	TRUE	FALSE	FALSE
RRM1	hgnc:10451	RRM1	ChEMBL	33	inhibitor	0.4412409347537352	GALLIUM NITRATE	rxcui:25544	GALLIUM NITRATE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.1436598392221464	FELODIPINE	rxcui:4316	FELODIPINE	TRUE	FALSE	FALSE
ADRB2	hgnc:286	ADRB2	ChEMBL	33	agonist	0.4070362111294147	PIRBUTEROL ACETATE	rxcui:221142	PIRBUTEROL ACETATE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	inhibitor	0.064318974	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	0.595325071	RIVAROXABAN	rxcui:1114195	RIVAROXABAN	TRUE	FALSE	FALSE
CHRM2	hgnc:1951	CHRM2	ChEMBL	33	inhibitor	0.1842374429322614	PROPANTHELINE BROMIDE	rxcui:8762	PROPANTHELINE BROMIDE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	agonist	0.5250767123569451	DECAMETHONIUM BROMIDE	ncit:C65365	DECAMETHONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNB1	hgnc:1961	CHRNB1	ChEMBL	33	inhibitor	0.5250767123569451	PIPECURONIUM BROMIDE	rxcui:66983	PIPECURONIUM BROMIDE	TRUE	FALSE	FALSE
CHRNG	hgnc:1967	CHRNG	ChEMBL	33	inhibitor	0.7501095890813501	PIPECURONIUM BROMIDE	rxcui:66983	PIPECURONIUM BROMIDE	TRUE	FALSE	FALSE
GLRA1	hgnc:4326	GLRA1	ChEMBL	33	positive modulator	0.1290114772375786	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
UNIPROT:P16066	hgnc:7943	NPR1	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	NESIRITIDE	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.1193356164447602	MAZINDOL	rxcui:6664	MAZINDOL	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1962903597596056	MAZINDOL	rxcui:6664	MAZINDOL	TRUE	FALSE	FALSE
PTGER4	hgnc:9596	PTGER4	ChEMBL	33	agonist	0.7721716358190367	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:P17342	hgnc:7945	NPR3	TdgClinicalTrial	Jan-14	NULL	6.563458904461812	NESIRITIDE	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
PDE1C	hgnc:8776	PDE1C	ChEMBL	33	inhibitor	0.750109589	PENTOXIFYLLINE	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
ITGB2	hgnc:6155	ITGB2	ChEMBL	33	inhibitor	0.4861821410712453	EFALIZUMAB	rxcui:356988	EFALIZUMAB	TRUE	TRUE	FALSE
KCNK9	hgnc:6283	KCNK9	ChEMBL	33	blocker	4.375639269641208	DOXAPRAM HYDROCHLORIDE	rxcui:82011	DOXAPRAM HYDROCHLORIDE	TRUE	FALSE	FALSE
KCNK3	hgnc:6278	KCNK3	ChEMBL	33	blocker	3.750547945	DOXAPRAM HYDROCHLORIDE	rxcui:82011	DOXAPRAM HYDROCHLORIDE	TRUE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	ChEMBL	33	inhibitor	0.0296486	PROCHLORPERAZINE EDISYLATE	rxcui:8704	PROCHLORPERAZINE	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.090374649	SU-014813	chembl:CHEMBL1721885	SU-014813	FALSE	FALSE	FALSE
NR1H2	hgnc:7965	NR1H2	ChEMBL	33	agonist	1.346350544504987	LXR-623	chembl:CHEMBL456237	LXR-623	FALSE	FALSE	FALSE
NR1H3	hgnc:7966	NR1H3	ChEMBL	33	agonist	0.8334550989792776	LXR-623	chembl:CHEMBL456237	LXR-623	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	inhibitor	0.8607814956671229	PF-05019702	chembl:CHEMBL3545239	PF-05019702	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.84012274	CLX-0921	drugbank:DB05854	CLX-0921	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.6563458904461812	NAPROXEN ETEMESIL	ncit:C166529	NAPROXEN ETEMESIL	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	ChEMBL	33	agonist	0.1973972602845657	AVE0847	chembl:CHEMBL3545295	AVE0847	FALSE	FALSE	FALSE
AR	hgnc:644	AR	ChEMBL	33	modulator	0.058471794	LY2452473	chembl:CHEMBL3542265	LY2452473	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	ChEMBL	33	inhibitor	1.250182648468916	AS-602868	chembl:CHEMBL129857	AS-602868	FALSE	FALSE	FALSE
PIK3R5	hgnc:30035	PIK3R5	ChEMBL	33	inhibitor	0.1875273972703375	AZD-6482	drugbank:DB14980	AZD-6482	FALSE	FALSE	FALSE
ALK	hgnc:427	ALK	ChEMBL	33	inhibitor	0.2282942227638891	CEP-37440	drugbank:DB13060	CEP-37440	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.2218633995874415	OSI-930	drugbank:DB05913	OSI-930	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.030368809	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
SRC	hgnc:11283	SRC	ChEMBL	33	inhibitor	0.018699313	PD-0166285	chembl:CHEMBL3545196	PD-0166285	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	ChEMBL	33	inhibitor	0.056826484	PHA-793887	drugbank:DB12686	PHA-793887	FALSE	FALSE	FALSE
MAPK14	hgnc:6876	MAPK14	ChEMBL	33	inhibitor	0.5707355569097228	SD-0006	drugbank:DB07943	SD-0006	FALSE	FALSE	FALSE
PIK3CD	hgnc:8977	PIK3CD	ChEMBL	33	inhibitor	0.4167275494896388	RP-6530	chembl:CHEMBL3545141	RP-6530	FALSE	FALSE	FALSE
UNIPROT:P28472	hgnc:4083	GABRB3	TdgClinicalTrial	Jan-14	NULL	0.034118045	NG2-73	chembl:CHEMBL2103791	ADIPIPLON	FALSE	FALSE	FALSE
CHKA	hgnc:1937	CHKA	ChEMBL	33	inhibitor	52.50767123569449	TCD-717	chembl:CHEMBL3545084	TCD-717	FALSE	FALSE	FALSE
PTK2	hgnc:9611	PTK2	ChEMBL	33	inhibitor	3.889457128569962	VS-4718	drugbank:DB15273	VS-4718	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.1479089330582944	TAK-593	drugbank:DB13093	TAK-593	FALSE	FALSE	FALSE
UNIPROT:O00311	hgnc:1745	CDC7	TdgClinicalTrial	Jan-14	NULL	8.078103267029922	NMS-1116354	chembl:CHEMBL3545321	NMS-1116354	FALSE	FALSE	FALSE
CHRNA4	hgnc:1958	CHRNA4	ChEMBL	33	modulator	0.5585922471882393	ABT-560	drugbank:DB06093	ABT-560	FALSE	FALSE	FALSE
KCNJ11	hgnc:6257	KCNJ11	ChEMBL	33	potentiator	0.4526523382387456	SARAKALIM	ncit:C72978	SARAKALIM	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	positive modulator	0.3977853881492007	CX1739	chembl:CHEMBL3707399	CX1739	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	ChEMBL	33	modulator	0.2453629496995069	FISPEMIFENE	ncit:C65687	FISPEMIFENE	FALSE	FALSE	FALSE
PGR	hgnc:8910	PGR	ChEMBL	33	inhibitor	0.4303907478335614	ONAPRISTONE	ncit:C170255	ONAPRISTONE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.42006137	NAVEGLITAZAR	ncit:C75191	NAVEGLITAZAR	FALSE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	2.019525817	ARHALOFENATE	ncit:C83536	ARHALOFENATE	FALSE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.116943588	OXANDROLONE	rxcui:7779	OXANDROLONE	TRUE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	ChEMBL	33	agonist	0.7955707762984014	GW590735	chembl:CHEMBL219586	GW590735	FALSE	FALSE	FALSE
CDK15	hgnc:14434	CDK15	ChEMBL	33	inhibitor	0.6250913242344582	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.3241214273808302	AKN-028	drugbank:DB12746	AKN-028	FALSE	FALSE	FALSE
ROCK2	hgnc:10252	ROCK2	ChEMBL	33	inhibitor	0.6731752722524935	VEROSUDIL	ncit:C152866	VEROSUDIL	FALSE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	ChEMBL	33	inhibitor	0.092606122	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
ROCK1	hgnc:10251	ROCK1	ChEMBL	33	inhibitor	0.7721716358190367	VEROSUDIL	ncit:C152866	VEROSUDIL	FALSE	FALSE	FALSE
CDK3	hgnc:1772	CDK3	ChEMBL	33	inhibitor	0.4167275494896388	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
CDK10	hgnc:1770	CDK10	ChEMBL	33	inhibitor	0.5000730593875666	AT-7519	drugbank:DB08142	AT-7519	FALSE	FALSE	FALSE
CDK8	hgnc:1779	CDK8	ChEMBL	33	inhibitor	0.093763699	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK20	hgnc:21420	CDK20	ChEMBL	33	inhibitor	0.4688184931758437	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK14	hgnc:8883	CDK14	ChEMBL	33	inhibitor	0.4688184931758437	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK7	hgnc:1778	CDK7	ChEMBL	33	inhibitor	0.075010959	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	0.1041818873724097	RONICICLIB	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.033295923	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
GSK3B	hgnc:4617	GSK3B	ChEMBL	33	inhibitor	0.043902735	LY-2090314	drugbank:DB11913	LY-2090314	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	0.3431873936973496	POZIOTINIB	ncit:C98838	POZIOTINIB	FALSE	FALSE	TRUE
UNIPROT:P30874	hgnc:11331	SSTR2	TdgClinicalTrial	Jan-14	NULL	0.729273212	PASIREOTIDE	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
MAPKAPK5	hgnc:6889	MAPKAPK5	ChEMBL	33	inhibitor	17.50255707856483	GLPG-0259	drugbank:DB15190	GLPG-0259	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1428780169678761	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
FLT4	hgnc:3767	FLT4	ChEMBL	33	inhibitor	0.065799087	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
FGFR4	hgnc:3691	FGFR4	ChEMBL	33	inhibitor	0.101562227	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	ChEMBL	33	inhibitor	0.1041818873724097	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	0.05751114	XL-999	chembl:CHEMBL3545285	XL-999	FALSE	FALSE	FALSE
PIK3R3	hgnc:8981	PIK3R3	ChEMBL	33	inhibitor	0.1071585127259071	SAMOTOLISIB	ncit:C121817	SAMOTOLISIB	FALSE	FALSE	FALSE
OXTR	hgnc:8529	OXTR	ChEMBL	33	inhibitor	3.088686543276147	RETOSIBAN	ncit:C76681	RETOSIBAN	FALSE	FALSE	FALSE
HTR1F	hgnc:5292	HTR1F	ChEMBL	33	agonist	14.32027397337122	LASMIDITAN	rxcui:2256930	LASMIDITAN	TRUE	FALSE	FALSE
TACR1	hgnc:11526	TACR1	ChEMBL	33	inhibitor	2.838252499226729	ORVEPITANT	ncit:C90613	ORVEPITANT	FALSE	FALSE	FALSE
BDKRB1	hgnc:1029	BDKRB1	ChEMBL	33	inhibitor	11.66837138570988	SAFOTIBANT	ncit:C152283	SAFOTIBANT	FALSE	FALSE	FALSE
UNIPROT:Q99062	hgnc:2439	CSF3R	TdgClinicalTrial	Jan-14	NULL	4.039051633514961	PEGFILGRASTIM	rxcui:2048018	PEGFILGRASTIM-JMDB	TRUE	FALSE	FALSE
HRH4	hgnc:17383	HRH4	ChEMBL	33	inhibitor	9.546849315580817	UR-63325	chembl:CHEMBL3545345	UR-63325	FALSE	FALSE	FALSE
OPRM1	hgnc:8156	OPRM1	ChEMBL	33	agonist	0.1605739181519709	FAXELADOL	ncit:C80579	FAXELADOL	FALSE	FALSE	FALSE
GRM5	hgnc:4597	GRM5	ChEMBL	33	negative modulator	5.834185692854944	STX107	chembl:CHEMBL3642985	STX107	FALSE	FALSE	FALSE
CHRNA7	hgnc:1960	CHRNA7	ChEMBL	33	agonist	1.141471113819445	ND0801	chembl:CHEMBL3707316	ND0801	FALSE	FALSE	FALSE
GRIA2	hgnc:4572	GRIA2	ChEMBL	33	inhibitor	0.3182283105193606	DASOLAMPANEL	ncit:C166510	DASOLAMPANEL	FALSE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	agonist	0.044347695	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.1400204566285186	MURAGLITAZAR	ncit:C75190	MURAGLITAZAR	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	ChEMBL	33	inhibitor	0.09753747	MASITINIB	ncit:C79910	MASITINIB	TRUE	FALSE	TRUE
GABRP	hgnc:4089	GABRP	ChEMBL	33	agonist	0.041540879	DARIGABAT	ncit:C175766	DARIGABAT	FALSE	FALSE	FALSE
INSR	hgnc:6091	INSR	ChEMBL	33	inhibitor	0.1071585127259071	LINSITINIB	ncit:C70982	LINSITINIB	FALSE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	ChEMBL	33	inhibitor	0.012836492	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	ChEMBL	33	inhibitor	0.2778183663264259	SIMOTINIB	iuphar.ligand:7640	SIMOTINIB	FALSE	FALSE	FALSE
ACHE	hgnc:108	ACHE	ChEMBL	33	inhibitor	0.7721716358190367	ECHOTHIOPHATE	ncit:C76040	ECHOTHIOPHATE	TRUE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	ChEMBL	33	inhibitor	0.8899605294185507	OLMESARTAN	rxcui:118463	OLMESARTAN MEDOXOMIL	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	modulator	0.042174836	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	modulator	0.042689164	DAVUNETIDE	ncit:C169878	DAVUNETIDE	FALSE	FALSE	FALSE
F10	hgnc:3528	F10	ChEMBL	33	inhibitor	1.071585127259071	IDRAPARINUX SODIUM	ncit:C170051	IDRAPARINUX SODIUM	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	ChEMBL	33	inhibitor	0.2224901323546377	LUSPATERCEPT	rxcui:2262543	LUSPATERCEPT-AAMT	TRUE	FALSE	FALSE
KIT	hgnc:6342	KIT	ChEMBL	33	inhibitor	1.897867635025102	AVAPRITINIB	rxcui:2272107	AVAPRITINIB	TRUE	FALSE	TRUE
MTNR1B	hgnc:7464	MTNR1B	ChEMBL	33	agonist	1.086365611772989	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	ChEMBL	33	inhibitor	0.192335792	IPRONIAZID	rxcui:5981	IPRONIAZID	TRUE	FALSE	FALSE
TBXA2R	hgnc:11608	TBXA2R	ChEMBL	33	inhibitor	1.071585127259071	RAMATROBAN	ncit:C76400	RAMATROBAN	FALSE	FALSE	FALSE
ATP4A	hgnc:819	ATP4A	ChEMBL	33	inhibitor	0.729273212	VONOPRAZAN FUMARATE	rxcui:2604576	VONOPRAZAN FUMARATE	TRUE	FALSE	FALSE
SLC5A2	hgnc:11037	SLC5A2	ChEMBL	33	inhibitor	3.281729452230906	SERGLIFLOZIN ETABONATE	ncit:C78129	SERGLIFLOZIN ETABONATE	FALSE	FALSE	FALSE
GP	hgnc:18280	RNF130	ChEMBL	33	inhibitor	7.501095891	ATOLTIVIMAB	rxcui:2461338	ATOLTIVIMAB	TRUE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	ChEMBL	33	inhibitor	0.040021091	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.033487035	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
SLC34A2	hgnc:11020	SLC34A2	ChEMBL	33	binder	3.281729452230906	LIFASTUZUMAB VEDOTIN	ncit:C116747	LIFASTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
GUCY2C	hgnc:4688	GUCY2C	ChEMBL	33	binder	1.640864726115453	INDUSATUMAB VEDOTIN	ncit:C101524	INDUSATUMAB VEDOTIN	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	ChEMBL	33	inhibitor	0.596678082	SELUMETINIB SULFATE	rxcui:2361596	SELUMETINIB SULFATE	TRUE	FALSE	FALSE
CACNA1D	hgnc:1391	CACNA1D	ChEMBL	33	blocker	0.1744440904840348	CILNIDIPINE	ncit:C171754	CILNIDIPINE	FALSE	FALSE	FALSE
PSMD6	hgnc:9564	PSMD6	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMD3	hgnc:9560	PSMD3	ChEMBL	33	inhibitor	0.2500365296937833	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMB9	hgnc:9546	PSMB9	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMA5	hgnc:9534	PSMA5	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMB10	hgnc:9538	PSMB10	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
PSMA7	hgnc:9536	PSMA7	ChEMBL	33	inhibitor	0.2083637747448194	IXAZOMIB	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
AVPR1A	hgnc:895	AVPR1A	ChEMBL	33	inhibitor	1.141471113819445	PECAVAPTAN	ncit:C166718	PECAVAPTAN	FALSE	FALSE	FALSE
RPL31	hgnc:10334	RPL31	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPS25	hgnc:10413	RPS25	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPS21	hgnc:10409	RPS21	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL12	hgnc:10302	RPL12	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL13	hgnc:10303	RPL13	ChEMBL	33	inhibitor	0.092606122	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL4	hgnc:10353	RPL4	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL23	hgnc:10316	RPL23	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL8	hgnc:10368	RPL8	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL27	hgnc:10328	RPL27	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
RPL39	hgnc:10350	RPL39	ChEMBL	33	inhibitor	0.1296485709523321	MT-3724	chembl:CHEMBL4297789	MT-3724	FALSE	FALSE	FALSE
TNNC2	hgnc:11944	TNNC2	ChEMBL	33	activator	11.66837138570988	RELDESEMTIV	ncit:C166781	RELDESEMTIV	FALSE	FALSE	FALSE
HDAC9	hgnc:14065	HDAC9	ChEMBL	33	inhibitor	0.1060761035064535	QUISINOSTAT	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
SLC22A12	hgnc:17989	SLC22A12	ChEMBL	33	inhibitor	4.039051633514961	SHR-4640	chembl:CHEMBL3746329	SHR-4640	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	ChEMBL	33	inhibitor	0.1434635826111871	SERALUTINIB	ncit:C175203	SERALUTINIB	FALSE	FALSE	FALSE
SSTR5	hgnc:11334	SSTR5	ChEMBL	33	agonist	0.8751278539282418	SOMATOSTATIN	rxcui:9939	SOMATOSTATIN	FALSE	FALSE	FALSE
PDE4C	hgnc:8782	PDE4C	ChEMBL	33	inhibitor	0.3621218705909966	REVAMILAST	ncit:C95233	REVAMILAST	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.6563458904461812	KARENITECIN	chembl:CHEMBL1743260	KARENITECIN	FALSE	FALSE	FALSE
RPMJ	hgnc:14490	MRPL36	ChEMBL	33	inhibitor	0.3860858179095183	JOSAMYCIN	rxcui:6084	JOSAMYCIN	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	ChEMBL	33	inhibitor	0.042689164	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
TUBB1	hgnc:16257	TUBB1	ChEMBL	33	inhibitor	0.038894571	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	ChEMBL	33	inhibitor	0.035719504	PLOCABULIN	ncit:C95888	PLOCABULIN	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.091636424	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.031317948	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.014243231	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
HDAC10	hgnc:18128	HDAC10	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2917092846427472	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.032492371	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PI3KCD	hgnc:8977	PIK3CD	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.2083637747448194	PKI-594	ncit:C84837	PI3K/MTOR KINASE INHIBITOR PF-04691502	FALSE	FALSE	TRUE
PI3KCA	hgnc:8975	PIK3CA	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.1715936968486748	GDC-0941	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
PI3KCG	hgnc:8978	PIK3CG	ClearityFoundationClinicalTrial	15-Jun-13	inhibitor	0.100976291	PKI-593	ncit:C84837	PI3K/MTOR KINASE INHIBITOR PF-04691502	FALSE	FALSE	TRUE
ALK	hgnc:427	ALK	COSMIC	4-Sep-20	NULL	2.493675356344019	Lorlatinib	rxcui:2103164	LORLATINIB	TRUE	FALSE	TRUE
CAMK2G	hgnc:1463	CAMK2G	DTC	9/2/20	NULL	0.025776962	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.015299438	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.018131102	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.040275444	AMIODARONE HYDROCHLORIDE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.021301287	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.031254566	DNDI1417467	chembl:CHEMBL1997335	CHEMBL:CHEMBL1997335	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.003614115	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.036718651	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
CAMKK2	hgnc:1470	CAMKK2	DTC	9/2/20	NULL	0.097236428	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2822993077187876	LEAD DIACETATE TRIHYDRATE	chembl:CHEMBL1350036	LEAD DIACETATE TRIHYDRATE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.032412143	CB7969312	chembl:CHEMBL599255	CHEMBL:CHEMBL599255	FALSE	FALSE	FALSE
CDK7	hgnc:1778	CDK7	DTC	9/2/20	NULL	0.019447286	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	DNDI1417165	chembl:CHEMBL1406948	CHEMBL:CHEMBL1406948	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.097236428	IRINOTECAN	rxcui:153329	IRINOTECAN HYDROCHLORIDE	TRUE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.012591768	TRIBUTYLTIN-OXIDE	chembl:CHEMBL511667	TRIBUTYLTIN-OXIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.064318974	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.011804782	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.01875274	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
GSK3B	hgnc:4617	GSK3B	DTC	9/2/20	NULL	0.02075402	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.1143957978991165	HYDROQUINONE	rxcui:5509	HYDROQUINONE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.007378818	PIRIBEDIL	rxcui:8353	PIRIBEDIL	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.3182283105193605	TCMDC-123702	chembl:CHEMBL548286	CHEMBL:CHEMBL548286	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.017709164	PROCARBAZINE	rxcui:8702	PROCARBAZINE	TRUE	FALSE	FALSE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.027390543	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.00804962	L-741626	iuphar.ligand:177	L-741,626	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.005208578	LEVOBUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.022136455	ATOMOXETINE	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CSNK1G3	hgnc:2456	CSNK1G3	DTC	9/2/20	NULL	0.088996053	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.009972967	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
TUBB3	hgnc:20772	TUBB3	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
TUBA4A	hgnc:12407	TUBA4A	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.037160418	ZOMEPIRAC SODIUM	rxcui:58331	ZOMEPIRAC SODIUM	TRUE	FALSE	FALSE
PRKACA	hgnc:9380	PRKACA	DTC	9/2/20	NULL	0.02706581	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
TUBB4A	hgnc:20774	TUBB4A	DTC	9/2/20	NULL	0.1108276362854715	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	DTC	9/2/20	NULL	0.04321619	DACARBAZINE	rxcui:3098	DACARBAZINE	TRUE	FALSE	TRUE
PRKX	hgnc:9441	PRKX	DTC	9/2/20	NULL	0.2785552850699973	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.045421861	SKF-83565 HYDROBROMIDE	chembl:CHEMBL541585	CHEMBL:CHEMBL541585	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.012154554	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.019059046	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004713012	DNDI1417156	chembl:CHEMBL1504679	CHEMBL:CHEMBL1504679	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.009944635	SJ000029642	chembl:CHEMBL591126	CHEMBL:CHEMBL591126	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.013411921	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.038187397	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.007866318	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.1274458039701322	PACHYRRIZINE	chembl:CHEMBL479689	PACHYRRIZINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TAZOBACTAM SODIUM	rxcui:221167	TAZOBACTAM SODIUM	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	2',4'-DIHYDROXY FLAVONE	chembl:CHEMBL1374610	CHEMBL:CHEMBL1374610	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	2-AMINO-ANTHRAQUINONE	chembl:CHEMBL84685	CHEMBL:CHEMBL84685	FALSE	FALSE	FALSE
TUBA1C	hgnc:20768	TUBA1C	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
NTSR1	hgnc:8039	NTSR1	DTC	9/2/20	NULL	0.546954909	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
TUBB	hgnc:20778	TUBB	DTC	9/2/20	NULL	0.069454592	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011143394	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
TUBB6	hgnc:20776	TUBB6	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.006496866	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	DTC	9/2/20	NULL	0.022249013	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
NR1H2	hgnc:7965	NR1H2	DTC	9/2/20	NULL	1.009762908	GW3965	iuphar.ligand:2754	GW3965	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.077077657	PACLITAXEL	rxcui:56946	PACLITAXEL	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	ONONIN	chembl:CHEMBL465980	ONONIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	JNJ-1661010	iuphar.ligand:5206	JNJ1661010	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.010698385	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	APTIGANEL	ncit:C79861	APTIGANEL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	AG-528	chembl:CHEMBL56542	CHEMBL:CHEMBL56542	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.007441563	TCMDC-123916	chembl:CHEMBL493863	CHEMBL:CHEMBL493863	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.106290832	ALOXISTATIN	ncit:C76907	ALOXISTATIN	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	GNF-PF-3286	chembl:CHEMBL581880	CHEMBL:CHEMBL581880	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	3-HYDROXYEVODIAMINE	chembl:CHEMBL2171793	CHEMBL:CHEMBL2171793	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.018131102	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.025390557	NSC-19063	chembl:CHEMBL1310138	CHEMBL:CHEMBL1310138	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004084611	CID 4101591	chembl:CHEMBL428789	CHEMBL:CHEMBL428789	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.04907259	CETRIMONIUM BROMIDE	rxcui:288999	CETRIMONIUM BROMIDE	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	TICLOPIDINE	rxcui:10594	TICLOPIDINE	TRUE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.020002922	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.054695491	FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.093596562	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.1190650141398968	RATANIAPHENOL II	chembl:CHEMBL463574	RATANIAPHENOL II	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.013350539	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	0.4487835148349957	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.012282496	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	MAKALUVAMINE E	chembl:CHEMBL509186	MAKALUVAMINE E	FALSE	FALSE	FALSE
MPHOSPH8	hgnc:29810	MPHOSPH8	DTC	9/2/20	NULL	0.009673484	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	TCMDC-124240	chembl:CHEMBL582764	CHEMBL:CHEMBL582764	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	DTC	9/2/20	NULL	0.760980743	PLERIXAFOR	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
LTA4H	hgnc:6710	LTA4H	DTC	9/2/20	NULL	11.66837138570988	DIPHENYLETHER	chembl:CHEMBL38934	DIPHENYLETHER	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	(S)-NIMODIPINE	chembl:CHEMBL255033	(S)-NIMODIPINE	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.014985066	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
CNR1	hgnc:2159	CNR1	DTC	9/2/20	NULL	0.2500365296937833	WIN-552122	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.006560179	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
GNAS	hgnc:4392	GNAS	DTC	9/2/20	NULL	0.375054795	S-166659	chembl:CHEMBL252417	CHEMBL:CHEMBL252417	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008023788	ISOVELLERAL	iuphar.ligand:6287	ISOVELLERAL	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.1193356164447602	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	THEONELLASTEROL E	chembl:CHEMBL1782601	THEONELLASTEROL E	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.009745299	MK-2206	drugbank:DB16828	MK-2206	FALSE	FALSE	TRUE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.1973972602845657	THIOSEMICARBAZIDE	chembl:CHEMBL256250	THIOSEMICARBAZIDE	FALSE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.4375639269641208	CHRYSENE	chembl:CHEMBL85685	CHRYSENE	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	CLEMIZOLE	ncit:C81139	CLEMIZOLE	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.002763853	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	DTC	9/2/20	NULL	0.1282238613814273	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
NFKBIA	hgnc:7797	NFKBIA	DTC	9/2/20	NULL	2.917092846427472	DIOSCIN	iuphar.ligand:840	DIOSCIN	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.017059022	2-AMINOPHENOXAZINONE	chembl:CHEMBL146710	CHEMBL:CHEMBL146710	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.004762601	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	FLUDROCORTISONE	rxcui:4452	FLUDROCORTISONE	TRUE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.016027983	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV000653	chembl:CHEMBL592344	CHEMBL:CHEMBL592344	FALSE	FALSE	FALSE
FRK	hgnc:3955	FRK	DTC	9/2/20	NULL	0.017363648	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.039688338	INDINAVIR SULFATE	rxcui:203153	INDINAVIR SULFATE	TRUE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.2625383561784725	GARCINONE E	chembl:CHEMBL454580	GARCINONE E	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.073954467	INDOCYANINE GREEN	rxcui:2199577	INDOCYANINE GREEN ACID FORM	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.031822831	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.077789143	ONONIN	chembl:CHEMBL465980	ONONIN	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.045461187	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	CALOTHRIXIN B	chembl:CHEMBL362573	CALOTHRIXIN B	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.004176557	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.015268296	CEPHALOCHROMIN	chembl:CHEMBL463175	CEPHALOCHROMIN	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.021760328	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.093346971	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.1367387271762877	PLERIXAFOR	rxcui:733003	PLERIXAFOR	TRUE	FALSE	FALSE
UNIPROT:P34969	hgnc:5302	HTR7	TdgClinicalTrial	Jan-14	NULL	0.2500365296937833	PARDOPRUNOX	ncit:C80765	PARDOPRUNOX	FALSE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	DTC	9/2/20	NULL	1.029562181092048	5-OXO-ETE	iuphar.ligand:3391	5-OXO-ETE	FALSE	FALSE	FALSE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.060772768	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	1.363835616511545	GAMMA-PROPARGYLAMINO-ATP	chembl:CHEMBL557670	CHEMBL:CHEMBL557670	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.013887244	ENALAPRIL	rxcui:203123	ENALAPRIL MALEATE	TRUE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.010223456	BITHIONOL	ncit:C77030	BITHIONOL	TRUE	FALSE	FALSE
UNIPROT:Q13547	hgnc:4852	HDAC1	TdgClinicalTrial	Jan-14	NULL	0.2286255641612242	CRA-024781	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
STK32B	hgnc:14217	STK32B	DTC	9/2/20	NULL	2.917092846427472	MIDOSTAURIN	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	GNF-PF-4832	chembl:CHEMBL601137	CHEMBL:CHEMBL601137	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.011557929	3',4'-DIHYDROXYFLAVONE	chembl:CHEMBL222556	CHEMBL:CHEMBL222556	FALSE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.044498026	2-HYDROXY-NAPHTHALDEHYDE THIOSEMICARBAZONE	chembl:CHEMBL505209	CHEMBL:CHEMBL505209	FALSE	FALSE	FALSE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	1.312691780892362	GW459057A	chembl:CHEMBL1909354	GW459057A	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1209854175937661	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	INDIUM CHLORIDE	chembl:CHEMBL1447815	INDIUM CHLORIDE	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.01013466	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TCMDC-125310	chembl:CHEMBL582030	CHEMBL:CHEMBL582030	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011143394	FENTICLOR	ncit:C65671	FENTICLOR	FALSE	FALSE	FALSE
CDC42BPA	hgnc:1737	CDC42BPA	DTC	9/2/20	NULL	0.044198376	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.012386806	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.021878196	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
UNIPROT:P30872	hgnc:11330	SSTR1	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	PASIREOTIDE	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
SOD1	hgnc:11179	SOD1	DTC	9/2/20	NULL	0.5250767123569451	OXYTETRACYCLINE	rxcui:1545999	OXYTETRACYCLINE ANHYDROUS	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.033832262	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.1071585127259071	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
CAMK1D	hgnc:19341	CAMK1D	DTC	9/2/20	NULL	0.2051080907644316	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.014757637	ROPINIROLE	rxcui:72302	ROPINIROLE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	HOMATROPINE METHYLBROMIDE	rxcui:1546413	METHYLHOMATROPINE	TRUE	FALSE	FALSE
UNIPROT:Q04759	hgnc:9410	PRKCQ	TdgClinicalTrial	Jan-14	NULL	0.1640864726115453	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.008345148	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008176218	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.008475815	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.015557829	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	TEMEFOS	drugbank:DB12231	TEMEFOS	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.7836965856073805	NERVIANO	chembl:CHEMBL1172241	NERVIANO	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.077217164	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.007869855	RETINYL ACETATE	ncit:C1216	RETINYL ACETATE	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	DTC	9/2/20	NULL	0.02926849	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.1271372184883644	NAPHTHYLAMINE	chembl:CHEMBL278164	NAPHTHYLAMINE	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.021396769	TCMDC-123868	chembl:CHEMBL548615	CHEMBL:CHEMBL548615	FALSE	FALSE	FALSE
UNIPROT:Q05513	hgnc:9412	PRKCZ	TdgClinicalTrial	Jan-14	NULL	0.2734774543525755	INGENOL MEBUTATE	rxcui:1242806	INGENOL MEBUTATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001924909	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TILNOPROFEN ARBAMEL	ncit:C76820	TILNOPROFEN ARBAMEL	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW831090X	chembl:CHEMBL103104	GW831090X	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	DERRUSNIN	chembl:CHEMBL1526572	DERRUSNIN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.016067219	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	1.521961485092594	YEZOQUINOLIDE	chembl:CHEMBL1668776	YEZOQUINOLIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	FIPEXIDE	ncit:C65685	FIPEXIDE	TRUE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.00663646	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.019665794	2-ARACHIDONOYLGLYCEROL	iuphar.ligand:729	2-ARACHIDONOYLGLYCEROL	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.010848692	QUINIDINE	rxcui:9068	QUINIDINE	TRUE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.043976274	2S,1'S,2'S)-2-(CARBOXYCYCLOPROPYL)GLYCINE	iuphar.ligand:1368	L-CCG-I	FALSE	FALSE	FALSE
MAOA	hgnc:6833	MAOA	DTC	9/2/20	NULL	0.092851762	MENADIONE	rxcui:6728	VITAMIN K3	TRUE	FALSE	FALSE
LRRK2	hgnc:18618	LRRK2	DTC	9/2/20	NULL	0.028771327	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
UNIPROT:P29274	hgnc:263	ADORA2A	TdgClinicalTrial	Jan-14	NULL	0.8514757497680189	PRELADENANT	ncit:C76394	PRELADENANT	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.06638138	GNF-PF-2298	chembl:CHEMBL578905	CHEMBL:CHEMBL578905	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.012442576	STREPTONIGRIN	ncit:C844	STREPTONIGRIN	FALSE	FALSE	FALSE
UNIPROT:Q969S8	hgnc:18128	HDAC10	TdgClinicalTrial	Jan-14	NULL	0.097236428	PRACINOSTAT	ncit:C71708	PRACINOSTAT	FALSE	FALSE	TRUE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.006557721	NISOLDIPINE	rxcui:7435	NISOLDIPINE	TRUE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.099446347	METHYLBENZETHONIUM CHLORIDE	rxcui:1796444	METHYLBENZETHONIUM CHLORIDE	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.016537849	SANGUINARIUM	ncit:C81358	SANGUINARIUM	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.014099804	FLUOXETINE HYDROCHLORIDE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.182318303	NSC-44661	chembl:CHEMBL571228	CHEMBL:CHEMBL571228	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001250391	RESVERATROL	rxcui:1000492	RESVERATROL	TRUE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1041818873724097	GNF-PF-3537	chembl:CHEMBL601110	CHEMBL:CHEMBL601110	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.025776962	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	TCMDC-124395	chembl:CHEMBL534047	CHEMBL:CHEMBL534047	FALSE	FALSE	FALSE
UNIPROT:O75888	hgnc:11928	TNFSF13	TdgClinicalTrial	Jan-14	NULL	39.38075342677087	TACI-IG	ncit:C81166	ATACICEPT	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005787883	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
AURKB	hgnc:11390	AURKB	DTC	9/2/20	NULL	0.1741547968016401	BMS-754807	drugbank:DB15399	BMS-754807	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.002623285	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
MINK1	hgnc:17565	MINK1	DTC	9/2/20	NULL	0.2778183663264258	SB-242235	chembl:CHEMBL95692	SB-242235	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.025427444	(+)-THALIPORPHINE	chembl:CHEMBL1397308	CHEMBL:CHEMBL1397308	FALSE	FALSE	FALSE
TUBA3D	hgnc:24071	TUBA3D	DTC	9/2/20	NULL	0.3125456621172291	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
TUBA1B	hgnc:18809	TUBA1B	DTC	9/2/20	NULL	0.080042182	4-(PHENYLCARBAMOYL)BENZYLNITRATE	chembl:CHEMBL1795737	CHEMBL:CHEMBL1795737	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.036463661	GNF-PF-3641	chembl:CHEMBL599098	CHEMBL:CHEMBL599098	FALSE	FALSE	FALSE
NQO2	hgnc:7856	NQO2	DTC	9/2/20	NULL	3.088686543276147	NSC-640353	chembl:CHEMBL1288253	CHEMBL:CHEMBL1288253	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.008575481	E324	chembl:CHEMBL172064	E324	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.005209094	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.03292017	GNF-PF-2657	chembl:CHEMBL578944	CHEMBL:CHEMBL578944	FALSE	FALSE	FALSE
HSP90AA1	hgnc:5253	HSP90AA1	DTC	9/2/20	NULL	0.060353645	8-FLUOROTRYPTANTHRIN	chembl:CHEMBL1098875	CHEMBL:CHEMBL1098875	FALSE	FALSE	FALSE
ENPP2	hgnc:3357	ENPP2	DTC	9/2/20	NULL	17.50255707856483	NSC-1698	chembl:CHEMBL1093490	CHEMBL:CHEMBL1093490	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	LY-2183240	drugbank:DB17035	LY-2183240	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002349337	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	LIOTHYRONINE SODIUM	rxcui:142448	LIOTHYRONINE SODIUM	TRUE	FALSE	FALSE
DAO	hgnc:2671	DAO	DTC	9/2/20	NULL	10.50153424713889	3-HYDROXYCOUMARIN	chembl:CHEMBL150372	3-HYDROXYCOUMARIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006807685	HISPIDIN	chembl:CHEMBL1224512	HISPIDIN	FALSE	FALSE	FALSE
UNIPROT:P09919	hgnc:2438	CSF3	TdgClinicalTrial	Jan-14	NULL	1.750255707856483	TALABOSTAT	ncit:C48264	TALABOSTAT	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	CEFPODOXIME PROXETIL	rxcui:47835	CEFPODOXIME PROXETIL	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.023813003	SJ000114740	chembl:CHEMBL592068	CHEMBL:CHEMBL592068	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	DITHIANON	chembl:CHEMBL2228641	DITHIANON	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	DTC	9/2/20	NULL	0.2344092465879218	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.006295884	TOLFENAMIC ACID	rxcui:38377	TOLFENAMIC ACID	FALSE	FALSE	FALSE
APAF1	hgnc:576	APAF1	DTC	9/2/20	NULL	0.042242696	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.055563673	DNDI1417195	chembl:CHEMBL1303948	CHEMBL:CHEMBL1303948	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.07643038	FANGCHINOLINE	chembl:CHEMBL504256	FANGCHINOLINE	FALSE	FALSE	FALSE
RXFP1	hgnc:19718	RXFP1	DTC	9/2/20	NULL	1.875273972703375	N6-METHYLADENOSINE	chembl:CHEMBL383144	CHEMBL:CHEMBL383144	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.078136416	AM-251	iuphar.ligand:3317	AM251	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.032755877	SJ000147784	chembl:CHEMBL590186	CHEMBL:CHEMBL590186	FALSE	FALSE	FALSE
MAP2K2	hgnc:6842	MAP2K2	DTC	9/2/20	NULL	0.016347345	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.023182195	CID 752709	chembl:CHEMBL429335	CHEMBL:CHEMBL429335	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	FURAFYLLINE	ncit:C65779	FURAFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	1.117184494376478	ISPRONICLINE	ncit:C65986	ISPRONICLINE	FALSE	FALSE	FALSE
MAP4K4	hgnc:6866	MAP4K4	DTC	9/2/20	NULL	0.025802295	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	AZOXYSTROBIN	drugbank:DB07401	AZOXYSTROBIN	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	HTS-05058	chembl:CHEMBL261692	CHEMBL:CHEMBL261692	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.018580209	PH-011685	chembl:CHEMBL126804	CHEMBL:CHEMBL126804	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.062958838	METACRESOL	rxcui:1367170	METACRESOL	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.00675253	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	(TRICYCLO[5.2.1.0~2,6~]DEC-8-YLOXY)CARBONOTHIOYLSULFIDE	chembl:CHEMBL404954	CHEMBL:CHEMBL404954	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.4526523382387456	SJ000040549	chembl:CHEMBL589421	CHEMBL:CHEMBL589421	FALSE	FALSE	FALSE
ABCC8	hgnc:59	ABCC8	DTC	9/2/20	NULL	0.7501095890813498	GLIQUIDONE	rxcui:25793	GLIQUIDONE	FALSE	FALSE	FALSE
CLK2	hgnc:2069	CLK2	DTC	9/2/20	NULL	0.2187819634820604	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003262967	PRASTERONE	rxcui:3143	PRASTERONE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.012713722	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
PPARD	hgnc:9235	PPARD	DTC	9/2/20	NULL	0.015184405	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	2.100306849	TETRABENAZINE	rxcui:10390	TETRABENAZINE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	0.1944728564284981	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
HDAC1	hgnc:4852	HDAC1	DTC	9/2/20	NULL	0.1801292323694494	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
HDAC8	hgnc:13315	HDAC8	DTC	9/2/20	NULL	0.2447910080918158	PHENYLBUTYRYLHYDROXAMIC ACID	chembl:CHEMBL55895	PHENYLBUTYRYLHYDROXAMIC ACID	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.08334551	GNF-PF-321	chembl:CHEMBL581044	CHEMBL:CHEMBL581044	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.008916229	MAPROTILINE	rxcui:6646	MAPROTILINE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.043902735	CETYLPYRIDINIUM BROMIDE	ncit:C83617	CETYLPYRIDINIUM BROMIDE	FALSE	FALSE	FALSE
LIMK1	hgnc:6613	LIMK1	DTC	9/2/20	NULL	0.2169738480813822	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.004427291	OXYMETAZOLINE	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.008725103	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.9907107780319716	TDR78274	chembl:CHEMBL1594756	CHEMBL:CHEMBL1594756	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.023182195	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
DYRK1A	hgnc:3091	DYRK1A	DTC	9/2/20	NULL	0.058212496	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.031254566	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.013505059	GW1929	iuphar.ligand:2703	GW1929	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	4-HYDROXYESTRADIOL	chembl:CHEMBL1412489	CHEMBL:CHEMBL1412489	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.1058622403945453	FPL-55712	chembl:CHEMBL267475	FPL-55712	FALSE	FALSE	FALSE
PRKD2	hgnc:17293	PRKD2	DTC	9/2/20	NULL	0.013087655	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TdgClinicalTrial	Jan-14	NULL	0.069089041	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.1530835896084387	GATIFLOXACIN	rxcui:1546025	GATIFLOXACIN ANHYDROUS	TRUE	FALSE	FALSE
RAB9A	hgnc:9792	RAB9A	DTC	9/2/20	NULL	0.033148782	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.049864835	L-745870	iuphar.ligand:3303	L745870	FALSE	FALSE	FALSE
ANXA2	hgnc:537	ANXA2	DTC	9/2/20	NULL	0.6250913242344582	WITHAFERIN A	iuphar.ligand:13097	WITHAFERIN A	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.022929114	GNF-PF-78	chembl:CHEMBL579318	CHEMBL:CHEMBL579318	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.1187956362798518	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	TCMDC-124585	chembl:CHEMBL587856	CHEMBL:CHEMBL587856	FALSE	FALSE	FALSE
UNIPROT:Q9NY46	hgnc:10590	SCN3A	TdgClinicalTrial	Jan-14	NULL	0.087512785	TETRODOTOXIN	ncit:C78845	TETRODOTOXIN	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.4102161815288632	BRYOSTATIN	chembl:CHEMBL449158	BRYOSTATIN	FALSE	FALSE	TRUE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.1259176768242074	GO-Y022	chembl:CHEMBL128729	CHEMBL:CHEMBL128729	FALSE	FALSE	FALSE
XBP1	hgnc:12801	XBP1	DTC	9/2/20	NULL	0.2386712328895204	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
PRKCQ	hgnc:9410	PRKCQ	DTC	9/2/20	NULL	0.090530468	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.2292911407672248	SJ000100732	chembl:CHEMBL592819	CHEMBL:CHEMBL592819	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.2083637747448194	SJ000196127	chembl:CHEMBL605084	CHEMBL:CHEMBL605084	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.006286838	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.024108205	BUTYLATED HYDROXYTOLUENE	rxcui:1848	BUTYLATED HYDROXYTOLUENE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	U-73122	iuphar.ligand:5283	U73122	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.007432084	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.034184682	NAN-190	iuphar.ligand:73	NAN 190	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	HYDRAZOBENZENE	chembl:CHEMBL558459	HYDRAZOBENZENE	FALSE	FALSE	FALSE
FLT1	hgnc:3763	FLT1	DTC	9/2/20	NULL	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:P37288	hgnc:895	AVPR1A	TdgClinicalTrial	Jan-14	NULL	3.043922970185188	TERLIPRESSIN	rxcui:57048	TERLIPRESSIN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.003068829	GENISTEIN	rxcui:25696	GENISTEIN	TRUE	FALSE	FALSE
CDK1	hgnc:1722	CDK1	DTC	9/2/20	NULL	0.008725103	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.2117244807890907	DIOTYROSINE	iuphar.ligand:6651	3,5-DIIODO-L-TYROSINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-741905	chembl:CHEMBL407113	CHEMBL:CHEMBL407113	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	SUVANINE'S SODIUM SALT	chembl:CHEMBL1818099	SUVANINE'S SODIUM SALT	FALSE	FALSE	FALSE
TOP2A	hgnc:11989	TOP2A	DTC	9/2/20	NULL	0.9053046764774912	(+)-9-DEMETHOXYELEUTHERIN	chembl:CHEMBL594379	CHEMBL:CHEMBL594379	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.072927321	3,5-DIPHENYLISOXAZOLE	chembl:CHEMBL1374535	3,5-DIPHENYLISOXAZOLE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	DTC	9/2/20	NULL	0.00444002	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.3889457128569963	GNF-PF-1702	chembl:CHEMBL600313	CHEMBL:CHEMBL600313	FALSE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.033658764	TERGURIDE	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
ALOX15B	hgnc:434	ALOX15B	DTC	9/2/20	NULL	0.084553416	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
PPARA	hgnc:9232	PPARA	DTC	9/2/20	NULL	0.7955707762984014	MYRISTIC ACID	rxcui:1356758	MYRISTIC ACID	TRUE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.090064616	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
TOP1	hgnc:11986	TOP1	DTC	9/2/20	NULL	0.8751278539282416	3-AMINOEVODIAMINE	chembl:CHEMBL2171795	CHEMBL:CHEMBL2171795	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.029766254	GNF-PF-186	chembl:CHEMBL601140	CHEMBL:CHEMBL601140	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.011068227	TCMDC-123869	chembl:CHEMBL546597	CHEMBL:CHEMBL546597	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.022789788	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
WEE1	hgnc:12761	WEE1	DTC	9/2/20	NULL	0.041639708	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TdgClinicalTrial	Jan-14	NULL	0.060585775	EPINEPHRINE	rxcui:3992	EPINEPHRINE	TRUE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.019799273	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	5,7,3',5'-TETRAHYDROXYFLAVANONE	iuphar.ligand:12442	(+/-)-ERIODICTYOL	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	CAMBENDAZOLE	rxcui:1951	CAMBENDAZOLE	FALSE	FALSE	FALSE
MAPK10	hgnc:6872	MAPK10	DTC	9/2/20	NULL	0.012466209	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CTNNB1	hgnc:2514	CTNNB1	DTC	9/2/20	NULL	0.7955707762984014	(+/-)-HYDNOCARPIN	chembl:CHEMBL91638	CHEMBL:CHEMBL91638	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW301784X	chembl:CHEMBL410072	GW301784X	FALSE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.2263261691193728	SJ000040549	chembl:CHEMBL589421	CHEMBL:CHEMBL589421	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.016047577	CID 3237815	chembl:CHEMBL410484	CHEMBL:CHEMBL410484	FALSE	FALSE	FALSE
APEX1	hgnc:587	APEX1	DTC	9/2/20	NULL	0.016491103	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.016027983	FLUOXETINE HYDROCHLORIDE	rxcui:227224	FLUOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.05293112	LY-255283	chembl:CHEMBL15766	LY-255283	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.015325238	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	TRIMETHYL-OCTADECYL-AMMONIUM CHLORIDE	chembl:CHEMBL118745	TRIMETHYL-OCTADECYL-AMMONIUM CHLORIDE	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.01864619	MYCOPHENOLIC ACID	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.009437037	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.088996053	NU-6027	chembl:CHEMBL303958	CHEMBL:CHEMBL303958	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.005723531	CADMIUM DICHLORIDE	chembl:CHEMBL1458880	CADMIUM DICHLORIDE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	GNF-PF-1401	iuphar.ligand:1376	AIDA	FALSE	FALSE	FALSE
SMN2	hgnc:11118	SMN2	DTC	9/2/20	NULL	0.045579576	GNF-PF-992	chembl:CHEMBL602561	CHEMBL:CHEMBL602561	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.007341677	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.004207345	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.03070624	OXYQUINOLINE	rxcui:110	OXYQUINOLINE	TRUE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.021138354	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.020257589	TIRATRICOL	rxcui:13982	TIRATRICOL	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.046798281	S-(P-AZIDOPHENACYL)GLUTATHIONE	chembl:CHEMBL1256813	CHEMBL:CHEMBL1256813	FALSE	FALSE	FALSE
ERBB4	hgnc:3432	ERBB4	DTC	9/2/20	NULL	0.3621218705909966	DIMETHYLCURCUMIN	drugbank:DB06133	DIMETHYLCURCUMIN	FALSE	FALSE	FALSE
GLP1R	hgnc:4324	GLP1R	DTC	9/2/20	NULL	0.026519026	PINAFIDE	ncit:C76757	PINAFIDE	FALSE	FALSE	FALSE
MAP4K2	hgnc:6864	MAP4K2	DTC	9/2/20	NULL	0.025244073	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
LYN	hgnc:6735	LYN	DTC	9/2/20	NULL	0.079557078	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.005953251	JUGLONE	chembl:CHEMBL43612	JUGLONE	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	1,3-DI(4-AMINOPHENYLCARBOXAMIDO)BENZENE	chembl:CHEMBL421431	CHEMBL:CHEMBL421431	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.019844169	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	chembl:CHEMBL1449651	PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT	FALSE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.032173818	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
TYK2	hgnc:12440	TYK2	DTC	9/2/20	NULL	0.008730906	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
MAPKAPK5	hgnc:6889	MAPKAPK5	DTC	9/2/20	NULL	0.4487835148349957	GW843682X	chembl:CHEMBL514499	GW843682X	FALSE	FALSE	FALSE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.045265234	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.001825687	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
SGK2	hgnc:13900	SGK2	DTC	9/2/20	NULL	0.1293292394967845	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
OPRM1	hgnc:8156	OPRM1	DTC	9/2/20	NULL	0.3211478363039418	ENDOMORPHIN-1	iuphar.ligand:1623	ENDOMORPHIN-1	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	FANGCHINOLINE	chembl:CHEMBL504256	FANGCHINOLINE	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	DTC	9/2/20	NULL	0.016083624	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.033529803	DITHIAZANINE	ncit:C72743	DITHIAZANINE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.091159151	TRIMETREXATE	rxcui:42333	TRIMETREXATE	TRUE	FALSE	TRUE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.031861451	GF-109203	iuphar.ligand:5193	GF109203X	FALSE	FALSE	TRUE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.014699796	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
PDGFRA	hgnc:8803	PDGFRA	DTC	9/2/20	NULL	0.007294758	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
PRKD3	hgnc:9408	PRKD3	DTC	9/2/20	NULL	0.013532905	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PLA2G1B	hgnc:9030	PLA2G1B	DTC	9/2/20	NULL	0.6731752722524935	SJ000196127	chembl:CHEMBL605084	CHEMBL:CHEMBL605084	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.006614723	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
NEK2	hgnc:7745	NEK2	DTC	9/2/20	NULL	0.036087747	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.3596415838061266	SJ000089102	chembl:CHEMBL606460	CHEMBL:CHEMBL606460	FALSE	FALSE	FALSE
AKT1	hgnc:391	AKT1	DTC	9/2/20	NULL	0.007624172	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.2917092846427472	TCMDC-125317	chembl:CHEMBL528373	CHEMBL:CHEMBL528373	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	MMV665814	chembl:CHEMBL586033	CHEMBL:CHEMBL586033	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.2625383561784725	Potassium Chloride	rxcui:8591	POTASSIUM CHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.022136455	Atomoxetine	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	FDA	10-Apr-24	NULL	0.035418328	Cariprazine	rxcui:1667655	CARIPRAZINE	TRUE	FALSE	FALSE
IFNL3	hgnc:18365	IFNL3	FDA	10-Apr-24	NULL	4.200613699	Dasabuvir	rxcui:1597381	DASABUVIR	TRUE	FALSE	FALSE
UNIPROT:P25116	hgnc:3537	F2R	TdgClinicalTrial	Jan-14	NULL	0.6731752722524935	RUSALATIDE	ncit:C152274	RUSALATIDE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.095468493	Chlorpropamide	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	FDA	10-Apr-24	NULL	0.058341857	Dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.5509279467829125	Erlotinib	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
FGF2	hgnc:3676	FGF2	NCI	14-Sep-17	NULL	0.2580229544751573	LAK CELLS	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	NCI	14-Sep-17	NULL	0.089222891	VACCINE	ncit:C923	VACCINE	FALSE	FALSE	FALSE
UNIPROT:Q86V86	hgnc:19310	PIM3	TdgClinicalTrial	Jan-14	NULL	1.029562181092048	VADIMEZAN	ncit:C2504	VADIMEZAN	FALSE	FALSE	TRUE
FGF3	hgnc:3681	FGF3	NCI	14-Sep-17	NULL	2.187819634820604	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	NCI	14-Sep-17	NULL	0.4861821410712453	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	NCI	14-Sep-17	NULL	0.2287915957982331	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
GADD45A	hgnc:4095	GADD45A	NCI	14-Sep-17	NULL	15.00219178	NB1011	ncit:C1882	BRIVUDINE PHOSPHORAMIDATE	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	NCI	14-Sep-17	NULL	0.036212187	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
GCG	hgnc:4191	GCG	NCI	14-Sep-17	NULL	0.6731752722524935	FDG	rxcui:1362737	FLUORODEOXYGLUCOSE F18	TRUE	FALSE	FALSE
GSTP1	hgnc:4638	GSTP1	NCI	14-Sep-17	NULL	0.038894571	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
HMGB1	hgnc:4983	HMGB1	NCI	14-Sep-17	NULL	0.502465753	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
UNIPROT:O76074	hgnc:8784	PDE5A	TdgClinicalTrial	Jan-14	NULL	8.204323630577266	UDENAFIL	ncit:C74086	UDENAFIL	TRUE	FALSE	FALSE
HLA-A	hgnc:4931	HLA-A	NCI	14-Sep-17	NULL	3.750547945	PMCV	ncit:C1633	POLYVALENT MELANOMA VACCINE	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	NCI	14-Sep-17	NULL	0.041872146	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.03015083	CYTARABINE	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.128537751	FLUTICASONE PROPIONATE	rxcui:41126	FLUTICASONE	TRUE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.1061833594250647	KETANSERIN	rxcui:6131	KETANSERIN	FALSE	FALSE	FALSE
HSPA4	hgnc:5237	HSPA4	NCI	14-Sep-17	NULL	0.016842878	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P00750	hgnc:9051	PLAT	TdgClinicalTrial	Jan-14	NULL	0.596678082	UROKINASE	rxcui:11055	UROKINASE	TRUE	FALSE	FALSE
ICAM3	hgnc:5346	ICAM3	NCI	14-Sep-17	NULL	0.8204323630577265	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
IFNG	hgnc:5438	IFNG	NCI	14-Sep-17	NULL	0.2344092465879218	URSODEOXYCHOLIC ACID	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	1.022876712383659	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
IL10	hgnc:5962	IL10	NCI	14-Sep-17	NULL	1.312691780892362	SHO-SAIKO-TO	ncit:C2690	SHO-SAIKO-TO	FALSE	FALSE	FALSE
IL15	hgnc:5977	IL15	NCI	14-Sep-17	NULL	1.022876712383659	LYMPHOKINE-ACTIVATED KILLER CELLS	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
IGFBP5	hgnc:5474	IGFBP5	NCI	14-Sep-17	NULL	2.763561643983921	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
IL17A	hgnc:5981	IL17A	NCI	14-Sep-17	NULL	0.080781033	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
IL1B	hgnc:5992	IL1B	NCI	14-Sep-17	NULL	0.5147810905460245	CHINESE HERBS	ncit:C2663	CHINESE HERBS	FALSE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	NCI	14-Sep-17	NULL	0.2059124362184098	GARLIC	ncit:C38706	GARLIC	FALSE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.071439008	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.014247096	ATRA	rxcui:10753	TRETINOIN	TRUE	FALSE	TRUE
IL7	hgnc:6023	IL7	NCI	14-Sep-17	NULL	17.50255707856483	HIV VACCINE	ncit:C1325	HIV VACCINE	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1736364789540161	VATALANIB	ncit:C1868	VATALANIB	FALSE	FALSE	TRUE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.2381300282797936	SAQUINAVIR	rxcui:83395	SAQUINAVIR	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	NCI	14-Sep-17	NULL	0.5357925636295356	SIGNAL TRANSDUCTION INHIBITORS	ncit:C2189	SIGNAL TRANSDUCTION INHIBITOR	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.1178623372293928	CEFTRIAXONE	rxcui:2193	CEFTRIAXONE	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	1.29648571	TALC	rxcui:10323	TALC	TRUE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.036013492	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
IL8RB	hgnc:6027	CXCR2	NCI	14-Sep-17	NULL	0.5303805175322677	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
UNIPROT:P12004	hgnc:8729	PCNA	TdgClinicalTrial	Jan-14	NULL	10.50153424713889	VIT-100	drugbank:DB05865	VIT-100	FALSE	FALSE	FALSE
IL8	hgnc:6025	CXCL8	NCI	14-Sep-17	NULL	0.072026984	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
LEP	hgnc:6553	LEP	NCI	14-Sep-17	NULL	0.076765601	VALPROIC ACID	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
LIF	hgnc:6596	LIF	NCI	14-Sep-17	NULL	0.057177137	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.2885036881082116	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
LPL	hgnc:6677	LPL	NCI	14-Sep-17	NULL	0.3409589041278864	LAK	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
MAOB	hgnc:6834	MAOB	NCI	14-Sep-17	NULL	0.037345428	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
MAPK8	hgnc:6881	MAPK8	NCI	14-Sep-17	NULL	0.2573905452730122	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
UNIPROT:P55011	hgnc:10911	SLC12A2	TdgClinicalTrial	Jan-14	NULL	5.834185692854945	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
MAZ	hgnc:6914	MAZ	NCI	14-Sep-17	NULL	5.834185692854945	IL-1	ncit:C586	RECOMBINANT INTERLEUKIN-1	FALSE	FALSE	FALSE
MGMT	hgnc:7059	MGMT	NCI	14-Sep-17	NULL	0.03292017	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
MIA	hgnc:7076	MIA	NCI	14-Sep-17	NULL	3.182283105193606	LYMPHOKINE-ACTIVATED KILLER CELL	ncit:C13008	LYMPHOKINE-ACTIVATED KILLER CELLS	FALSE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TdgClinicalTrial	Jan-14	NULL	0.093763699	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
MIF	hgnc:7097	MIF	NCI	14-Sep-17	NULL	0.3804903712731485	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
MYC	hgnc:7553	MYC	NCI	14-Sep-17	NULL	0.2143170254518142	BESTATIN	ncit:C1015	UBENIMEX	FALSE	FALSE	FALSE
NEUROD1	hgnc:7762	NEUROD1	NCI	14-Sep-17	NULL	2.059124362184098	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
MYOD1	hgnc:7611	MYOD1	NCI	14-Sep-17	NULL	0.4688184931758437	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TdgClinicalTrial	Jan-14	NULL	0.086551106	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.031479419	PYRAZOLE	drugbank:DB02757	PYRAZOLE	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	NCI	14-Sep-17	NULL	0.002518354	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.3697723326457359	DIETHYLDITHIOCARBAMIC ACID	ncit:C432	DITIOCARB	FALSE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TdgClinicalTrial	Jan-14	NULL	0.1346350544504987	CLOTIAZEPAM	rxcui:2622	CLOTIAZEPAM	TRUE	FALSE	FALSE
NOL1	hgnc:7867	NOP2	NCI	14-Sep-17	NULL	0.3889457128569963	ADJUVANT	ncit:C2140	ADJUVANT	FALSE	FALSE	FALSE
NOS1	hgnc:7872	NOS1	NCI	14-Sep-17	NULL	0.092443083	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
NR5A1	hgnc:7983	NR5A1	NCI	14-Sep-17	NULL	0.2734774543525755	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	NCI	14-Sep-17	NULL	0.007157534	MTX	rxcui:6851	METHOTREXATE	TRUE	FALSE	TRUE
NTF3	hgnc:8023	NTF3	NCI	14-Sep-17	NULL	4.039051633514961	VANILLOID	ncit:C1955	VANILLOID	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.030598876	DESIPRAMINE	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TdgClinicalTrial	Jan-14	NULL	1.166837138570988	ENPROFYLLINE	ncit:C74327	ENPROFYLLINE	FALSE	FALSE	FALSE
NTF4	hgnc:8024	NTF4	NCI	14-Sep-17	NULL	17.50255707856483	BDNF	iuphar.ligand:4872	BDNF	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.21578495	GAMMA-INTERFERON	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.089910396	PHENYLEPHRINE	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	NCI	14-Sep-17	NULL	0.2397610558707511	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.1346350544504987	BDNF	iuphar.ligand:4872	BDNF	FALSE	FALSE	FALSE
PIK3CG	hgnc:8978	PIK3CG	NCI	14-Sep-17	NULL	0.067317527	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
UNIPROT:P28222	hgnc:5287	HTR1B	TdgClinicalTrial	Jan-14	NULL	0.280789686	ERGOTAMINE	rxcui:4025	ERGOTAMINE	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.092606122	RETINOL	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
PLAU	hgnc:9052	PLAU	NCI	14-Sep-17	NULL	0.2273059360852575	BCNU	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
PPY	hgnc:9327	PPY	NCI	14-Sep-17	NULL	8.751278539282415	CORTISONE	rxcui:2878	CORTISONE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.037398626	LOVASTATIN	rxcui:6472	LOVASTATIN	TRUE	FALSE	TRUE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.729273212	DEXAMETHASONE ACETATE	rxcui:22690	DEXAMETHASONE ACETATE	TRUE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.1121958787087489	CLONIDINE	rxcui:142432	CLONIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P30556	hgnc:336	AGTR1	TdgClinicalTrial	Jan-14	NULL	2.669881588255652	FORASARTAN	ncit:C65749	FORASARTAN	FALSE	FALSE	FALSE
PRL	hgnc:9445	PRL	NCI	14-Sep-17	NULL	0.091159151	PHENOTHIAZINE	ncit:C740	PHENOTHIAZINE	FALSE	FALSE	FALSE
PTGS1	hgnc:9604	PTGS1	NCI	14-Sep-17	NULL	0.028536778	HYDROCHLOROTHIAZIDE	rxcui:5487	HYDROCHLOROTHIAZIDE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.074797252	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.070860555	AZATHIOPRINE	rxcui:1256	AZATHIOPRINE	TRUE	FALSE	TRUE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	2.692701089009974	POTASSIUM CITRATE	rxcui:1374802	POTASSIUM CITRATE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	FONDAPARINUX	rxcui:321208	FONDAPARINUX	TRUE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.1121958787087489	LAMIVUDINE	rxcui:68244	LAMIVUDINE	TRUE	FALSE	FALSE
PTHR1	hgnc:9608	PTH1R	NCI	14-Sep-17	NULL	0.087222045	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
MTR	hgnc:7468	MTR	PharmGKB	4/5/24	NULL	0.1600843635234588	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
UNIPROT:P47871	hgnc:4192	GCGR	TdgClinicalTrial	Jan-14	NULL	1.670698630226643	GLUCAGON RECOMBINANT	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.006106608	lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
NRXN1	hgnc:8008	NRXN1	PharmGKB	4/5/24	NULL	1.141471113819445	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
XDH	hgnc:12805	XDH	PharmGKB	4/5/24	NULL	0.7249579855026854	febuxostat	rxcui:73689	FEBUXOSTAT	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	PharmGKB	4/5/24	NULL	0.047304208	omeprazole	rxcui:7646	OMEPRAZOLE	TRUE	FALSE	FALSE
FGG	hgnc:3694	FGG	PharmGKB	4/5/24	NULL	2.625383561784725	eptifibatide	rxcui:75635	EPTIFIBATIDE	TRUE	FALSE	FALSE
HMMR	hgnc:5012	HMMR	PharmGKB	4/5/24	NULL	0.3201687270469177	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.00445925	raloxifene	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
ESR2	hgnc:3468	ESR2	PharmGKB	4/5/24	NULL	0.087512785	raloxifene	rxcui:166551	RALOXIFENE HYDROCHLORIDE	TRUE	FALSE	FALSE
FNTB	hgnc:3785	FNTB	PharmGKB	4/5/24	NULL	0.2386712328895204	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.2983390411119005	ISOETHARINE	rxcui:6023	ISOETHARINE	TRUE	FALSE	FALSE
HLA-E	hgnc:4962	HLA-E	PharmGKB	4/5/24	NULL	2.500365296937833	certolizumab pegol	rxcui:709271	CERTOLIZUMAB PEGOL	TRUE	FALSE	FALSE
VDR	hgnc:12679	VDR	PharmGKB	4/5/24	NULL	0.3251536612259921	calcitriol	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.023493365	fesoterodine	rxcui:797195	FESOTERODINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.006525935	hydroxychloroquine	rxcui:5521	HYDROXYCHLOROQUINE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.011294887	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.010488109	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.01305187	itraconazole	rxcui:28031	ITRACONAZOLE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.2234869519440402	vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
UNIPROT:P15382	hgnc:6240	KCNE1	TdgClinicalTrial	Jan-14	NULL	3.000438356	INDAPAMIDE	rxcui:5764	INDAPAMIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	PharmGKB	4/5/24	NULL	0.016780975	trimethoprim	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	PharmGKB	4/5/24	NULL	0.005840675	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ALOX5	hgnc:435	ALOX5	PharmGKB	4/5/24	NULL	1.887530665335423	zileuton	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
GNB3	hgnc:4400	GNB3	PharmGKB	4/5/24	NULL	0.7955707762984016	sildenafil	rxcui:136411	SILDENAFIL	TRUE	FALSE	FALSE
DRD4	hgnc:3025	DRD4	PharmGKB	4/5/24	NULL	0.013429072	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
HLA-B	hgnc:4932	HLA-B	PharmGKB	4/5/24	NULL	0.1973972602845657	acetazolamide	rxcui:167	ACETAZOLAMIDE	TRUE	FALSE	FALSE
BDKRB2	hgnc:1030	BDKRB2	PharmGKB	4/5/24	NULL	0.546954909	imidapril	rxcui:60245	IMIDAPRIL	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.07458476	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	0.1363835616511545	MECLOFENAMIC ACID	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.1262203635473425	pyrazinamide	rxcui:8987	PYRAZINAMIDE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.068369364	midazolam	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP2B6	hgnc:2615	CYP2B6	PharmGKB	4/5/24	NULL	0.087903467	rifampin	rxcui:9384	RIFAMPIN	TRUE	FALSE	FALSE
CYP4F2	hgnc:2645	CYP4F2	PharmGKB	4/5/24	NULL	2.651902587661338	Vitamin K	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	PharmGKB	4/5/24	NULL	0.017835486	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
UNIPROT:P04150	hgnc:7978	NR3C1	TdgClinicalTrial	Jan-14	NULL	0.066803653	METHYLPREDNISOLONE	rxcui:6902	METHYLPREDNISOLONE	TRUE	FALSE	FALSE
GAPVD1	hgnc:23375	GAPVD1	PharmGKB	4/5/24	NULL	5.250767124	interferon beta-1b	rxcui:72257	INTERFERON BETA-1B	TRUE	TRUE	FALSE
TNFRSF1B	hgnc:11917	TNFRSF1B	PharmGKB	4/5/24	NULL	0.4773424657790409	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
TLR2	hgnc:11848	TLR2	PharmGKB	4/5/24	NULL	0.2273059360852576	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.078136416	METHOTRIMEPRAZINE	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
TF	hgnc:11740	TF	PharmGKB	4/5/24	NULL	0.7955707762984016	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
CCNY	hgnc:23354	CCNY	PharmGKB	4/5/24	NULL	3.182283105193606	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.5073204950308646	METHOXAMINE	rxcui:6853	METHOXAMINE	TRUE	FALSE	FALSE
CDSN	hgnc:1802	CDSN	PharmGKB	4/5/24	NULL	0.2983390411119005	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
EMSY	hgnc:18071	EMSY	PharmGKB	4/5/24	NULL	3.182283105193606	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
SERPINC1	hgnc:775	SERPINC1	PharmGKB	4/5/24	NULL	0.033148782	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
SERPINA5	hgnc:8723	SERPINA5	PharmGKB	4/5/24	NULL	0.2983390411119005	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UNIPROT:P48169	hgnc:4078	GABRA4	TdgClinicalTrial	Jan-14	NULL	0.053361455	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	PharmGKB	4/5/24	NULL	0.02339914	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
UGT1A1	hgnc:12530	UGT1A1	PharmGKB	4/5/24	NULL	0.029833904	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
MAP3K1	hgnc:6848	MAP3K1	PharmGKB	4/5/24	NULL	0.1325951293830669	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
HLA-DRB1	hgnc:4948	HLA-DRB1	PharmGKB	4/5/24	NULL	0.1591141552596803	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
FTO	hgnc:24678	FTO	PharmGKB	4/5/24	NULL	0.364636606	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
BCR	hgnc:1014	BCR	PharmGKB	4/5/24	NULL	1.250182648468916	asciminib	rxcui:2584304	ASCIMINIB	TRUE	FALSE	TRUE
CES1	hgnc:1863	CES1	PharmGKB	4/5/24	NULL	0.060077427	clomipramine	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
RABGAP1L	hgnc:24663	RABGAP1L	PharmGKB	4/5/24	NULL	1.329308132549227	ethanol	rxcui:1310469	DEHYDRATED ALCOHOL	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.4605936073306534	DACOMITINIB	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	TALC	12-May-16	inhibitor	0.053445395	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	inhibitor	0.1151484018326633	AEE 788	ncit:C48369	MULTIKINASE INHIBITOR AEE788	FALSE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	TALC	12-May-16	vaccine	0.086361301	EP-2101	ncit:C26645	MULTI-NEO-EPITOPE VACCINE OSE 2101	FALSE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	TALC	12-May-16	inhibitor	0.3571950424196904	TELATINIB	ncit:C80869	TELATINIB	FALSE	FALSE	TRUE
HDAC1	hgnc:4852	HDAC1	TALC	12-May-16	inhibitor	0.104285345	DACINOSTAT	ncit:C81158	DACINOSTAT	FALSE	FALSE	TRUE
JAK3	hgnc:6193	JAK3	TALC	12-May-16	inhibitor	0.1037701012563132	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.023110771	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
KIT	hgnc:6342	KIT	TALC	12-May-16	inhibitor	0.1331836936859721	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.097308509	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	TALC	12-May-16	inhibitor	0.1232574442152452	AEE 788	ncit:C48369	MULTIKINASE INHIBITOR AEE788	FALSE	FALSE	TRUE
MST1R	hgnc:7381	MST1R	TALC	12-May-16	inhibitor	0.1151484018326633	FORETINIB	ncit:C80058	FORETINIB	FALSE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	TALC	12-May-16	inhibitor	0.5877724392055355	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
AURKC	hgnc:11391	AURKC	TALC	12-May-16	inhibitor	0.8751278539282416	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.032492371	DOVITINIB	ncit:C76199	DOVITINIB	FALSE	FALSE	TRUE
PARP2	hgnc:272	PARP2	TALC	12-May-16	inhibitor	2.187819634820604	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
PDGFRB	hgnc:8804	PDGFRB	TALC	12-May-16	inhibitor	0.3281729452230906	XL820	drugbank:DB05146	XL820	FALSE	FALSE	TRUE
BCR	hgnc:1014	BCR	TALC	12-May-16	inhibitor	0.2333674277141977	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
TERT	hgnc:11730	TERT	TALC	12-May-16	inhibitor	3.000438356	IMETELSTAT	ncit:C49084	IMETELSTAT	FALSE	FALSE	TRUE
TERT	hgnc:11730	TERT	TALC	12-May-16	inhibitor	3.000438356	SODIUM METAARSENITE	ncit:C91098	SODIUM METAARSENITE	FALSE	FALSE	TRUE
TLR9	hgnc:15633	TLR9	TALC	12-May-16	agonist	3.088686543276147	PF-3512676	ncit:C28580	AGATOLIMOD SODIUM	FALSE	FALSE	TRUE
SRC	hgnc:11283	SRC	TALC	12-May-16	inhibitor	0.7778914257139926	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
C14ORF129	hgnc:20343	GSKIP	TALC	12-May-16	inhibitor	4.773424657790409	AT9283	drugbank:DB05169	AT9283	FALSE	FALSE	TRUE
ZHX2	hgnc:18513	ZHX2	TALC	12-May-16	inhibitor	0.3182283105193606	REGORAFENIB	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
ZHX2	hgnc:18513	ZHX2	TALC	12-May-16	inhibitor	0.1842374429322613	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
VEGFA	hgnc:12680	VEGFA	TALC	12-May-16	NULL	0.027290889	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
FGFR3	hgnc:3690	FGFR3	TALC	12-May-16	antibody	0.276356164	FP-1039	iuphar.ligand:11581	FP-1039	FALSE	FALSE	TRUE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.112036283	ARIPIPRAZOLE	rxcui:1673265	ARIPIPRAZOLE LAUROXIL	TRUE	FALSE	FALSE
UNIPROT:P52732	hgnc:6388	KIF11	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	4SC-205	ncit:C90557	EG5 KINESIN-RELATED MOTOR PROTEIN INHIBITOR 4SC-205	FALSE	FALSE	FALSE
PSMC2	hgnc:9548	PSMC2	TALC	12-May-16	inhibitor	0.4487835148349957	MLN9708	rxcui:1723734	IXAZOMIB CITRATE	TRUE	FALSE	TRUE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.251232877	OXYBUTYNIN	rxcui:32675	OXYBUTYNIN	TRUE	FALSE	FALSE
UNIPROT:P08514	hgnc:6138	ITGA2B	TdgClinicalTrial	Jan-14	NULL	3.646366058	ABCIXIMAB	rxcui:83929	ABCIXIMAB	TRUE	FALSE	FALSE
UNIPROT:O43451	hgnc:7043	MGAM	TdgClinicalTrial	Jan-14	NULL	3.182283105193605	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
UNIPROT:P10253	hgnc:4065	GAA	TdgClinicalTrial	Jan-14	NULL	0.364636606	ACARBOSE	rxcui:16681	ACARBOSE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.092118721	ACLIDINIUM	rxcui:1303098	ACLIDINIUM	TRUE	FALSE	FALSE
UNIPROT:P48039	hgnc:7463	MTNR1A	TdgClinicalTrial	Jan-14	NULL	1.875273972703375	AGOMELATINE	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
UNIPROT:P41595	hgnc:5294	HTR2B	TdgClinicalTrial	Jan-14	NULL	0.2734774543525755	AGOMELATINE	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
UNIPROT:P49286	hgnc:7464	MTNR1B	TdgClinicalTrial	Jan-14	NULL	2.625383561784724	AGOMELATINE	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
UNIPROT:Q15759	hgnc:6873	MAPK11	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	BMS-582949	drugbank:DB12696	BMS-582949	FALSE	FALSE	FALSE
UNIPROT:P35968	hgnc:6307	KDR	TdgClinicalTrial	Jan-14	NULL	0.1183271464466354	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
UNIPROT:P53778	hgnc:6874	MAPK12	TdgClinicalTrial	Jan-14	NULL	0.3241214273808302	BMS-582949	drugbank:DB12696	BMS-582949	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.08334551	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
UNIPROT:Q92731	hgnc:3468	ESR2	TdgClinicalTrial	Jan-14	NULL	0.093098708	ESTRADIOL	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.2365210416022274	BIFEPRUNOX	ncit:C65262	BIFEPRUNOX	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.1000146118775133	NINTEDANIB	rxcui:1592736	NINTEDANIB ESYLATE	TRUE	FALSE	TRUE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.064318974	BICALUTAMIDE	rxcui:83008	BICALUTAMIDE	TRUE	FALSE	TRUE
UNIPROT:P49810	hgnc:9509	PSEN2	TdgClinicalTrial	Jan-14	NULL	1.193356164447602	BMS-708163	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
UNIPROT:P49768	hgnc:9508	PSEN1	TdgClinicalTrial	Jan-14	NULL	1.009762908	BMS-708163	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
UNIPROT:P18825	hgnc:283	ADRA2C	TdgClinicalTrial	Jan-14	NULL	0.092443083	LURASIDONE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.088695391	LURASIDONE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P19235	hgnc:3416	EPOR	TdgClinicalTrial	Jan-14	NULL	5.250767123569449	ERYTHROPOIESIS-STIMULATING AGENT	wikidata:Q1363798	ERYTHROPOIESIS-STIMULATING AGENT	FALSE	FALSE	FALSE
UNIPROT:P49327	hgnc:3594	FASN	TdgClinicalTrial	Jan-14	NULL	0.2991890098899972	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
UNIPROT:P30518	hgnc:897	AVPR2	TdgClinicalTrial	Jan-14	NULL	2.386712328895204	OPC-51803	drugbank:DB05838	OPC-51803	FALSE	FALSE	FALSE
UNIPROT:P16233	hgnc:9155	PNLIP	TdgClinicalTrial	Jan-14	NULL	3.029288725136221	ORLISTAT	rxcui:37925	ORLISTAT	TRUE	FALSE	FALSE
UNIPROT:P10415	hgnc:990	BCL2	TdgClinicalTrial	Jan-14	NULL	0.2134458180312784	ORTATAXEL	ncit:C1867	ORTATAXEL	FALSE	FALSE	FALSE
UNIPROT:Q9UKV0	hgnc:14065	HDAC9	TdgClinicalTrial	Jan-14	NULL	0.2651902587661338	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
UNIPROT:Q92769	hgnc:4853	HDAC2	TdgClinicalTrial	Jan-14	NULL	0.2841324201065719	BELINOSTAT	rxcui:1543543	BELINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P48039	hgnc:7463	MTNR1A	TdgClinicalTrial	Jan-14	NULL	7.501095891	RAMELTEON	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.4817217544559128	REMIFENTANIL	rxcui:236540	REMIFENTANIL HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28223	hgnc:5293	HTR2A	TdgClinicalTrial	Jan-14	NULL	0.050488145	RENZAPRIDE	ncit:C152191	RENZAPRIDE	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	1.389091831632129	RINDOPEPIMUT	ncit:C69076	RINDOPEPIMUT	FALSE	FALSE	TRUE
UNIPROT:P15391	hgnc:1633	CD19	TdgClinicalTrial	Jan-14	NULL	3.842024724563012	SAR3419	ncit:C71009	COLTUXIMAB RAVTANSINE	FALSE	FALSE	FALSE
UNIPROT:P08246	hgnc:3309	ELANE	TdgClinicalTrial	Jan-14	NULL	3.804903712731485	SIVELESTAT	ncit:C66539	SIVELESTAT	FALSE	FALSE	FALSE
UNIPROT:P13945	hgnc:288	ADRB3	TdgClinicalTrial	Jan-14	NULL	0.750109589	SOLABEGRON	ncit:C96754	SOLABEGRON	FALSE	FALSE	FALSE
UNIPROT:P05546	hgnc:4838	SERPIND1	TdgClinicalTrial	Jan-14	NULL	26.25383561784724	SULODEXIDE	ncit:C152467	SULODEXIDE	TRUE	FALSE	FALSE
UNIPROT:P17787	hgnc:1962	CHRNB2	TdgClinicalTrial	Jan-14	NULL	2.917092846427472	ISPRONICLINE	ncit:C65986	ISPRONICLINE	FALSE	FALSE	FALSE
UNIPROT:P00374	hgnc:2861	DHFR	TdgClinicalTrial	Jan-14	NULL	0.546954909	TALOTREXIN	ncit:C29341	TALOTREXIN	FALSE	FALSE	FALSE
UNIPROT:P00533	hgnc:3236	EGFR	TdgClinicalTrial	Jan-14	NULL	0.5509279467829125	ERLOTINIB	rxcui:337525	ERLOTINIB	TRUE	FALSE	TRUE
UNIPROT:P25101	hgnc:3179	EDNRA	TdgClinicalTrial	Jan-14	NULL	1.521961485092594	SITAXSENTAN	ncit:C73038	SITAXENTAN	TRUE	FALSE	FALSE
UNIPROT:O14965	hgnc:11393	AURKA	TdgClinicalTrial	Jan-14	NULL	0.2542744369767287	XL228	drugbank:DB05184	XL228	FALSE	FALSE	TRUE
UNIPROT:P08514	hgnc:6138	ITGA2B	TdgClinicalTrial	Jan-14	NULL	2.187819634820604	GANTOFIBAN	ncit:C73227	GANTOFIBAN	FALSE	FALSE	FALSE
UNIPROT:P35916	hgnc:3767	FLT4	TdgClinicalTrial	Jan-14	NULL	0.053887183	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
UNIPROT:P61073	hgnc:2561	CXCR4	TdgClinicalTrial	Jan-14	NULL	3.150460274	BL-8040	rxcui:2664896	MOTIXAFORTIDE	TRUE	FALSE	FALSE
UNIPROT:P06729	hgnc:1639	CD2	TdgClinicalTrial	Jan-14	NULL	11.66837138570988	ALEFACEPT	rxcui:299635	ALEFACEPT	TRUE	TRUE	FALSE
UNIPROT:P05023	hgnc:799	ATP1A1	TdgClinicalTrial	Jan-14	NULL	1.555782851427985	ACETYLDIGITOXIN	rxcui:132871	ACETYLDIGITOXIN	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TdgClinicalTrial	Jan-14	NULL	0.9845188356692718	ALSEROXYLON	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
UNIPROT:P02671	hgnc:3661	FGA	TdgClinicalTrial	Jan-14	NULL	1.591141552596802	ANISTREPLASE	rxcui:40028	ANISTREPLASE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.4189441853911795	BENZTROPINE	rxcui:1424	BENZTROPINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.6351734423672721	BUCLIZINE	rxcui:59636	BUCLIZINE	TRUE	FALSE	FALSE
UNIPROT:O00555	hgnc:1388	CACNA1A	TdgClinicalTrial	Jan-14	NULL	0.5834185692854944	BEPRIDIL	rxcui:1436	BEPRIDIL	TRUE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.1250182648468916	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.1166837138570989	BUTETHAL	rxcui:19874	BUTOBARBITAL	FALSE	FALSE	FALSE
UNIPROT:P42262	hgnc:4572	GRIA2	TEND	1-Aug-11	NULL	0.1591141552596803	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.079197091	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TEND	1-Aug-11	NULL	0.07182992	ADINAZOLAM	ncit:C76531	ADINAZOLAM	FALSE	FALSE	FALSE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.036531311	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.4234489615781814	CHLORPHENIRAMINE	rxcui:221074	CHLORPHENIRAMINE POLISTIREX	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.083016081	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.068191781	CITALOPRAM	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
UNIPROT:A8MPY1	hgnc:17969	GABRR3	TEND	1-Aug-11	NULL	0.1223955040459079	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P04035	hgnc:5006	HMGCR	TEND	1-Aug-11	NULL	0.7425327245451747	ATORVASTATIN	rxcui:1297766	ATORVASTATIN CALCIUM TRIHYDRATE	TRUE	FALSE	FALSE
UNIPROT:P30939	hgnc:5292	HTR1F	TEND	1-Aug-11	NULL	1.060761035064535	NARATRIPTAN	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:Q12809	hgnc:6251	KCNH2	TEND	1-Aug-11	NULL	0.080550887	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
UNIPROT:P01583	hgnc:5991	IL1A	TEND	1-Aug-11	NULL	3.500511415712966	RILONACEPT	rxcui:763450	RILONACEPT	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TEND	1-Aug-11	NULL	0.2027323213733378	DIPHENIDOL	rxcui:23370	DIPHENIDOL	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.9211872146613069	DOXACURIUM	rxcui:23651	DOXACURIUM	TRUE	FALSE	FALSE
UNIPROT:P18507	hgnc:4087	GABRG2	TEND	1-Aug-11	NULL	0.093763699	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P01008	hgnc:775	SERPINC1	TEND	1-Aug-11	NULL	0.1367387271762877	HEPARIN	rxcui:5224	HEPARIN	TRUE	FALSE	FALSE
UNIPROT:P18505	hgnc:4081	GABRB1	TEND	1-Aug-11	NULL	0.096050618	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TEND	1-Aug-11	NULL	0.1022876712383659	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.087512785	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.1653584607713247	ISOPROTERENOL	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TEND	1-Aug-11	NULL	0.8334550989792776	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.3006164383722967	LOTEPREDNOL ETABONATE	rxcui:237027	LOTEPREDNOL	TRUE	FALSE	FALSE
UNIPROT:Q13131	hgnc:9376	PRKAA1	TEND	1-Aug-11	NULL	1.640864726115453	PHENFORMIN	rxcui:8129	PHENFORMIN	TRUE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.1037701012563132	LURASIDONE	rxcui:1040027	LURASIDONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.1875273972703374	MECLOFENAMIC ACID	rxcui:588003	MECLOFENAMATE	TRUE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.042504861	METHADONE	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.063415062	METHAMPHETAMINE	rxcui:6816	METHAMPHETAMINE	TRUE	FALSE	FALSE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.056097939	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TEND	1-Aug-11	NULL	0.033919684	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.091159151	MINAPRINE	rxcui:30031	MINAPRINE	TRUE	FALSE	FALSE
UNIPROT:Q9UN88	hgnc:14454	GABRQ	TEND	1-Aug-11	NULL	0.05913026	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P28221	hgnc:5289	HTR1D	TEND	1-Aug-11	NULL	0.4487835148349957	NARATRIPTAN	rxcui:141366	NARATRIPTAN	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.0701037	NEFAZODONE	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
UNIPROT:P29074	hgnc:9656	PTPN4	TEND	1-Aug-11	NULL	4.375639269641208	ALENDRONATE	rxcui:203152	ALENDRONATE SODIUM	TRUE	FALSE	TRUE
UNIPROT:P08185	hgnc:1540	SERPINA6	TEND	1-Aug-11	NULL	6.563458904461812	PARAMETHASONE	rxcui:7910	PARAMETHASONE	TRUE	FALSE	FALSE
UNIPROT:P46098	hgnc:5297	HTR3A	TEND	1-Aug-11	NULL	1.166837138570988	PALONOSETRON	rxcui:1552337	NETUPITANT	TRUE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.033701971	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P47869	hgnc:4076	GABRA2	TEND	1-Aug-11	NULL	0.030368809	PHENOBARBITAL	rxcui:8134	PHENOBARBITAL	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.3977853881492006	PHENTERMINE	rxcui:221138	PHENTERMINE RESIN	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TEND	1-Aug-11	NULL	1.186614039224734	PERINDOPRIL	rxcui:54552	PERINDOPRIL	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TEND	1-Aug-11	NULL	0.8334550989792778	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
UNIPROT:P38435	hgnc:4247	GGCX	TEND	1-Aug-11	NULL	3.500511415712966	PHYTONADIONE	rxcui:11258	VITAMIN K	TRUE	FALSE	FALSE
TYROSINASE	hgnc:12442	TYR	TTD	2020.06.01	NULL	1.193356164447602	Melanoma vaccine	ncit:C2517	MELANOMA VACCINE	FALSE	FALSE	FALSE
CD70 ANTIGEN	hgnc:11937	CD70	TTD	2020.06.01	NULL	4.039051633514961	AMG 172	ncit:C106266	ANTI-CD27L ANTIBODY-DRUG CONJUGATE AMG 172	FALSE	FALSE	FALSE
TELOMERASE REVERSE TRANSCRIPTASE	hgnc:11730	TERT	TTD	2020.06.01	NULL	3.000438356	KML-001	ncit:C91098	SODIUM METAARSENITE	FALSE	FALSE	TRUE
GLUCAGON-LIKE PEPTIDE 2 RECEPTOR	hgnc:4325	GLP2R	TTD	2020.06.01	NULL	26.25383561784724	ZP-1848	iuphar.ligand:10885	GLEPAGLUTIDE	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.092443083	Sulfatinib	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 1	hgnc:3763	FLT1	TTD	2020.06.01	NULL	0.1562728310586145	Sulfatinib	ncit:C116066	SULFATINIB	FALSE	FALSE	FALSE
INTERLEUKIN 13 RECEPTOR ALPHA-2	hgnc:5975	IL13RA2	TTD	2020.06.01	NULL	13.12691780892362	ICT-107	ncit:C124054	MULTI-GLIOBLASTOMA-PEPTIDE-TARGETING AUTOLOGOUS DENDRITIC CELL VACCINE ICT-107	FALSE	FALSE	FALSE
CYTOKINE RECEPTOR UNSPECIFIC	hgnc:2355	CRH	TTD	2020.06.01	NULL	6.563458904461812	IRX-2	drugbank:DB05643	IRX-2	FALSE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.8334550989792777	ABT-414	ncit:C105612	DEPATUXIZUMAB MAFODOTIN	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	4.286340509036285	Olokizumab	ncit:C172654	OLOKIZUMAB	FALSE	FALSE	FALSE
T-CELL RECEPTOR	hgnc:12197	TRBV20OR9-2	TTD	2020.06.01	NULL	4.200613698855561	TOL-101	drugbank:DB16980	TOL-101	FALSE	FALSE	FALSE
ANGIOTENSIN-CONVERTING ENZYME 2	hgnc:13557	ACE2	TTD	2020.06.01	NULL	10.50153424713889	GSK2586881	iuphar.ligand:11320	ALUNACEDASE ALFA	FALSE	FALSE	FALSE
HISTAMINE H4 RECEPTOR	hgnc:17383	HRH4	TTD	2020.06.01	NULL	7.160136986685614	JNJ-38518168	ncit:C152698	TOREFORANT	FALSE	FALSE	FALSE
ERBB3 TYROSINE KINASE RECEPTOR	hgnc:3431	ERBB3	TTD	2020.06.01	NULL	2.059124362184098	KTN3379	ncit:C113333	ANTI-ERBB3 MONOCLONAL ANTIBODY CDX-3379	FALSE	FALSE	FALSE
B-CELL RECEPTOR CD22	hgnc:1643	CD22	TTD	2020.06.01	NULL	8.751278539282417	OspA lipoprotein	rxcui:54214	OSPA PROTEIN	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 4D	hgnc:8783	PDE4D	TTD	2020.06.01	NULL	0.08334551	Papaverine	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
GLUTAMATE RECEPTOR IONOTROPIC NMDA 2B	hgnc:4586	GRIN2B	TTD	2020.06.01	NULL	0.1682938180631233	ELIPRODIL	ncit:C80994	ELIPRODIL	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.3365876361262467	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
ARACHIDONATE 5-LIPOXYGENASE	hgnc:435	ALOX5	TTD	2020.06.01	NULL	0.5147810905460244	Silymarin	rxcui:9794	SILYMARIN	FALSE	FALSE	FALSE
LCK TYROSINE PROTEIN KINASE	hgnc:6524	LCK	TTD	2020.06.01	NULL	0.057197899	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.041085815	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
DIHYDROTHYMINE DEHYDROGENASE	hgnc:3012	DPYD	TTD	2020.06.01	NULL	1.486066167047957	Eniluracil	ncit:C1773	ENILURACIL	FALSE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV3.2	hgnc:1395	CACNA1H	TTD	2020.06.01	NULL	0.1436598392221464	Mibefradil	rxcui:83213	MIBEFRADIL	FALSE	FALSE	FALSE
GTP CYCLOHYDROLASE-I	hgnc:4193	GCH1	TTD	2020.06.01	NULL	26.25383561784724	Guanine	rxcui:1372539	GUANINE	FALSE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.075010959	GBR-12909	ncit:C81084	VANOXERINE	FALSE	FALSE	FALSE
INTERLEUKIN-8	hgnc:6025	CXCL8	TTD	2020.06.01	NULL	1.29648571	ABX-IL8	chembl:CHEMBL2109616	ABX-IL8	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	0.1093909817410302	Papaverine	rxcui:7895	PAPAVERINE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.2187819634820604	Tafluposide	ncit:C152490	TAFLUPOSIDE	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	6.300920548	MSX-122	drugbank:DB12715	MSX-122	FALSE	FALSE	FALSE
INWARD RECTIFIER POTASSIUM CHANNEL KIR1.2	hgnc:6256	KCNJ10	TTD	2020.06.01	NULL	0.6819178082557728	Chlorpropamide	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
SUBSTANCE-K RECEPTOR	hgnc:11527	TACR2	TTD	2020.06.01	NULL	2.100306849	Rambazole	ncit:C90792	TALAROZOLE	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.9	hgnc:10583	SCN11A	TTD	2020.06.01	NULL	0.084689792	Flecainide	rxcui:42686	FLECAINIDE ACETATE	TRUE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.8751278539282416	Edotecarin	ncit:C2665	EDOTECARIN	FALSE	FALSE	FALSE
VOLTAGE-GATED POTASSIUM CHANNEL KV1.5	hgnc:6224	KCNA5	TTD	2020.06.01	NULL	1.166837138570988	T-226296	iuphar.ligand:1314	T-226296	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR BETA	hgnc:3468	ESR2	TTD	2020.06.01	NULL	1.875273972703375	AUS-131	chembl:CHEMBL198877	AUS-131	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.03849536	Tranilast	rxcui:57330	TRANILAST	FALSE	FALSE	FALSE
VOLTAGE-GATED SODIUM CHANNEL ALPHA NAV1.4	hgnc:10591	SCN4A	TTD	2020.06.01	NULL	0.8078103267029922	Lanperisone	ncit:C79785	LANPERISONE	FALSE	FALSE	FALSE
ORPHAN NUCLEAR RECEPTOR NR1I3	hgnc:7969	NR1I3	TTD	2020.06.01	NULL	0.5357925636295356	Meclizine	rxcui:6676	MECLIZINE	TRUE	FALSE	FALSE
PROSTAGLANDIN D2 RECEPTOR	hgnc:9591	PTGDR	TTD	2020.06.01	NULL	2.917092846427472	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1962903597596056	Quinestrol	rxcui:9066	QUINESTROL	TRUE	FALSE	FALSE
DELTA-AMINOLEVULINIC ACID DEHYDRATASE	hgnc:395	ALAD	TTD	2020.06.01	NULL	52.50767123569449	Porphobilinogen	drugbank:DB02272	PORPHOBILINOGEN	FALSE	FALSE	FALSE
LIPOPROTEIN LIPASE	hgnc:6677	LPL	TTD	2020.06.01	NULL	0.1172046232939609	Clofibrate	rxcui:2594	CLOFIBRATE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.1280674908187671	MCI-186	rxcui:1921877	EDARAVONE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	2.316514907	Ambenonium	rxcui:623	AMBENONIUM	TRUE	FALSE	FALSE
SODIUM CHANNEL UNSPECIFIC	hgnc:12811	XK	TTD	2020.06.01	NULL	0.067751834	Zonisamide	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	5.834185692854944	Anti-Mesothelin CAR-T cells	ncit:C201275	ANTI-MESOTHELIN CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
CYCLIC ADP-RIBOSE HYDROLASE 1	hgnc:1667	CD38	TTD	2020.06.01	NULL	5.834185692854944	Anti-CD38 CAR-T cells	ncit:C201510	ANTI-CD38 CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.055740628	Calcifediol	rxcui:1855064	CALCIFEDIOL ANHYDROUS	TRUE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.030176823	Doxorubicin	rxcui:142433	DOXORUBICIN HYDROCHLORIDE	TRUE	FALSE	TRUE
RIBONUCLEOSIDE-DIPHOSPHATE REDUCTASE M2	hgnc:10452	RRM2	TTD	2020.06.01	NULL	0.384671584	Hydroxyurea	rxcui:5552	HYDROXYUREA	TRUE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.0296486	Levomepromazine	rxcui:6852	METHOTRIMEPRAZINE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	1.544343271638073	Pralidoxime Chloride	rxcui:55322	PRALIDOXIME CHLORIDE	TRUE	FALSE	FALSE
OPIOID RECEPTOR MU	hgnc:14449	OPN4	TTD	2020.06.01	NULL	0.375054795	Eluxadoline	rxcui:1653781	ELUXADOLINE	TRUE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE RAF	hgnc:18513	ZHX2	TTD	2020.06.01	NULL	3.500511415712966	RO-5126766	drugbank:DB15254	AVUTOMETINIB	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-1	hgnc:285	ADRB1	TTD	2020.06.01	NULL	0.99446347	Betaxolol	rxcui:1520	BETAXOLOL	TRUE	FALSE	FALSE
P2Y PURINOCEPTOR 12	hgnc:18124	P2RY12	TTD	2020.06.01	NULL	0.2812910959055062	Clopidogrel	rxcui:32968	CLOPIDOGREL	TRUE	FALSE	FALSE
INTEGRIN ALPHA-L	hgnc:6148	ITGAL	TTD	2020.06.01	NULL	1.357957014716237	lifitegrast	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-2	hgnc:286	ADRB2	TTD	2020.06.01	NULL	0.1653584607713247	Isoproterenol	rxcui:6054	ISOPROTERENOL	TRUE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.086861325	Lenalidomide	rxcui:342369	LENALIDOMIDE	TRUE	FALSE	TRUE
ANGIOTENSIN II RECEPTOR TYPE-1	hgnc:336	AGTR1	TTD	2020.06.01	NULL	0.4449802647092754	Irbesartan	rxcui:83818	IRBESARTAN	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.4773424657790409	Lornoxicam	rxcui:20890	LORNOXICAM	TRUE	FALSE	FALSE
VASOPRESSIN V2 RECEPTOR	hgnc:897	AVPR2	TTD	2020.06.01	NULL	0.7955707762984013	Mozavaptan	ncit:C77018	MOZAVAPTAN	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR BETA-3	hgnc:288	ADRB3	TTD	2020.06.01	NULL	0.750109589	Rimiterol	rxcui:9388	RIMITEROL	TRUE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-1D	hgnc:280	ADRA1D	TTD	2020.06.01	NULL	0.1864177677006905	Terazosin	rxcui:37798	TERAZOSIN	TRUE	FALSE	TRUE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1556551518844698	Zuclopenthixol	rxcui:114176	ZUCLOPENTHIXOL	TRUE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	2.625383561784724	MGD006	ncit:C117238	FLOTETUZUMAB	FALSE	FALSE	FALSE
LEUKOTRIENE B4 RECEPTOR 1	hgnc:6713	LTB4R	TTD	2020.06.01	NULL	6.563458904461812	Amelubant	ncit:C73299	AMELUBANT	FALSE	FALSE	FALSE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	1.071585127259071	GW-813893	drugbank:DB07278	GW-813893	FALSE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	0.4039051633514961	T-817MA	chembl:CHEMBL4297438	T-817 MALEATE	FALSE	FALSE	FALSE
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 2	hgnc:2358	CRHR2	TTD	2020.06.01	NULL	7.501095891	Urocortin 2	iuphar.ligand:3545	UROCORTIN 2	FALSE	FALSE	FALSE
METABOTROPIC GLUTAMATE RECEPTOR 3	hgnc:4595	GRM3	TTD	2020.06.01	NULL	5.250767123569449	LY404039	chembl:CHEMBL375611	LY404039	FALSE	FALSE	FALSE
ADENOSINE A3 RECEPTOR	hgnc:268	ADORA3	TTD	2020.06.01	NULL	1.973972602845657	IB-MECA	ncit:C166615	PICLIDENOSON	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE	hgnc:9612	PTK2B	TTD	2020.06.01	NULL	0.095122593	KD019	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
SPHINGOSINE-1-PHOSPHATE RECEPTOR 1	hgnc:3165	S1PR1	TTD	2020.06.01	NULL	0.6482428547616604	Ozanimod	rxcui:2288236	OZANIMOD	TRUE	FALSE	FALSE
NCBIGENE:1388	hgnc:2349	ATF6B	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8751	iuphar.ligand:8751	COMPOUND 34 [PMID: 20866075]	FALSE	FALSE	FALSE
MATRIX METALLOPROTEINASE-3	hgnc:7173	MMP3	TTD	2020.06.01	NULL	0.150021918	GM6001	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:16	iuphar.ligand:16	L-772,405	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.4526523382387456	IUPHAR.LIGAND:18	iuphar.ligand:18	LY 165,163	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.055387839	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1207072901969988	IUPHAR.LIGAND:5593	iuphar.ligand:5593	GS9667	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.100589408	IUPHAR.LIGAND:5596	rxcui:1546015	REGADENOSON ANHYDROUS	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.100976291	IUPHAR.LIGAND:5595	ncit:C174671	BINODENOSON	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.033658764	IUPHAR.LIGAND:2844	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:415	iuphar.ligand:415	(S)-PIA	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.045461187	IUPHAR.LIGAND:2844	rxcui:296	ADENOSINE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:5610	iuphar.ligand:5610	MSX-2	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:5611	ncit:C152704	TOZADENANT	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:10193	iuphar.ligand:10193	PBF-509	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:5604	ncit:C96195	ROLOFYLLINE	FALSE	FALSE	FALSE
UNIPROT:P07101	hgnc:11782	TH	TdgClinicalTrial	Jan-14	NULL	0.9616789603607051	METYROSINE	rxcui:266604	METYROSINE	TRUE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	inhibitor	0.063110182	IUPHAR.LIGAND:5605	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:5590	iuphar.ligand:5590	TCPA	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.6819178082557726	IUPHAR.LIGAND:442	iuphar.ligand:442	AS96	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	agonist	0.1704794520639431	IUPHAR.LIGAND:415	iuphar.ligand:415	(S)-PIA	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.061992528	IUPHAR.LIGAND:5615	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1082632396612257	IUPHAR.LIGAND:5601	iuphar.ligand:5601	MRS3558	FALSE	FALSE	FALSE
NCBIGENE:20	hgnc:32	ABCA2	GuideToPharmacology	2024.1	inhibitor	0.019483366	IUPHAR.LIGAND:7095	rxcui:8013	PENTOXIFYLLINE	TRUE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1082632396612257	IUPHAR.LIGAND:5593	iuphar.ligand:5593	GS9667	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1082632396612257	IUPHAR.LIGAND:5595	ncit:C174671	BINODENOSON	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	agonist	0.1353290495765322	IUPHAR.LIGAND:415	iuphar.ligand:415	(S)-PIA	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1804387327687096	IUPHAR.LIGAND:3285	iuphar.ligand:3285	PSB36	FALSE	FALSE	FALSE
NCBIGENE:21	hgnc:33	ABCA3	GuideToPharmacology	2024.1	inhibitor	0.1082632396612257	IUPHAR.LIGAND:5612	ncit:C152892	VIPADENANT	FALSE	FALSE	FALSE
NCBIGENE:2594	hgnc:59	ABCC8	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:6841	rxcui:73044	REPAGLINIDE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.6141248097742046	MIVACURIUM	rxcui:30077	MIVACURIUM	TRUE	FALSE	FALSE
NCBIGENE:849	ncbigene:849	CATHL1L	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:12008	ncit:C152542	TEGOPRAZAN	FALSE	FALSE	FALSE
NCBIGENE:2720	hgnc:4298	GLB1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:9521	iuphar.ligand:9521	GSK8814	FALSE	FALSE	FALSE
NCBIGENE:3245	hgnc:115	ACLY	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:12855	iuphar.ligand:12855	BMS-303141	FALSE	FALSE	FALSE
NCBIGENE:39	hgnc:94	ACAT2	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:12494	iuphar.ligand:12494	[D-PHE6, STAT13, LEU14}BN(6-14)	FALSE	FALSE	FALSE
NCBIGENE:2330	hgnc:3773	FMO5	GuideToPharmacology	2024.1	inhibitor	0.7955707762984014	IUPHAR.LIGAND:9822	iuphar.ligand:9822	NB-360	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7856	iuphar.ligand:7856	EXAMPLE 92 [WO2012095521]	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8688	iuphar.ligand:8688	HYDROXYETHYLAMINE TRANSITION-STATE INHIBITOR 1	FALSE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	2.500365296937833	MIVACURIUM	rxcui:30077	MIVACURIUM	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:7178	rxcui:49737	ESMOLOL	TRUE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:546	iuphar.ligand:546	NIP	FALSE	FALSE	FALSE
NCBIGENE:1789	hgnc:2979	DNMT3B	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:11888	ncit:C175551	ZILURGISERTIB	FALSE	FALSE	FALSE
NCBIGENE:2749	hgnc:4338	GLUD1P3	GuideToPharmacology	2024.1	activator	0.3106962795011509	IUPHAR.LIGAND:1204	rxcui:5333	HISTAMINE	TRUE	FALSE	FALSE
NCBIGENE:3055	hgnc:4840	HCK	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10149	iuphar.ligand:10149	SLC-0111	FALSE	FALSE	FALSE
NCBIGENE:1619	hgnc:1504	CASP3	GuideToPharmacology	2024.1	inhibitor	0.2333674277141978	IUPHAR.LIGAND:8654	iuphar.ligand:8654	M826	FALSE	FALSE	FALSE
NCBIGENE:1621	hgnc:2689	DBH	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9901	iuphar.ligand:9901	URACIL 20	FALSE	FALSE	FALSE
NCBIGENE:2343	ncbigene:2343	FNTBL1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11515	iuphar.ligand:11515	K777	FALSE	FALSE	FALSE
NCBIGENE:2351	ncbigene:2351	FOLR2L	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:11515	iuphar.ligand:11515	K777	FALSE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7861	iuphar.ligand:7861	BALICATIB	FALSE	FALSE	FALSE
NCBIGENE:390	hgnc:671	RND3	GuideToPharmacology	2024.1	activator	2.187819634820604	IUPHAR.LIGAND:5412	iuphar.ligand:5412	PGF1&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:56	hgnc:127	ACRV1	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:9234	ncit:C174784	IBIPINABANT	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:11890	iuphar.ligand:11890	VICASINABIN	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	0.063110182	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	agonist	2.019525817	IUPHAR.LIGAND:12751	iuphar.ligand:12751	LY2828360	FALSE	FALSE	FALSE
NCBIGENE:76	hgnc:1570	CCKAR	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:3888	iuphar.ligand:3888	JMV180	FALSE	FALSE	FALSE
NCBIGENE:57	hgnc:2160	CNR2	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:9234	ncit:C174784	IBIPINABANT	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	1.141471113819445	IUPHAR.LIGAND:8440	iuphar.ligand:8440	ML398	FALSE	FALSE	FALSE
NCBIGENE:1232	hgnc:1604	CCR3	GuideToPharmacology	2024.1	antibody	5.834185692854944	IUPHAR.LIGAND:9596	iuphar.ligand:9596	OLECLUMAB	FALSE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TdgClinicalTrial	Jan-14	NULL	0.1117184494376478	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12711	iuphar.ligand:12711	DBPR112	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:7422	rxcui:2058848	DACOMITINIB ANHYDROUS	TRUE	FALSE	TRUE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.7001022831425933	IUPHAR.LIGAND:1919	ncit:C84191	SULPROSTONE	FALSE	FALSE	FALSE
NCBIGENE:340	ncbigene:340	APOBER1	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:1915	rxcui:8814	EPOPROSTENOL	TRUE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	NULL	0.5000730593875666	IUPHAR.LIGAND:4864	iuphar.ligand:4864	AMPHIREGULIN	FALSE	FALSE	FALSE
NCBIGENE:2970	hgnc:4660	GTF2IP1	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:10002	iuphar.ligand:10002	TRIPLE MODULATOR 10 [PMID: 29878767]	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.084553416	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
UNIPROT:P20309	hgnc:1952	CHRM3	TdgClinicalTrial	Jan-14	NULL	0.3547815624033412	OXYPHENCYCLIMINE	rxcui:32698	OXYPHENCYCLIMINE	TRUE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.3241214273808302	IUPHAR.LIGAND:1881	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	0.1620607136904151	IUPHAR.LIGAND:1895	rxcui:40138	ILOPROST	TRUE	FALSE	TRUE
NCBIGENE:341	hgnc:607	APOC1	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1947	iuphar.ligand:1947	19(R)-OH-PGE2	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.2134458180312784	IUPHAR.LIGAND:1892	iuphar.ligand:1892	BUTAPROST (FREE ACID FORM)	FALSE	FALSE	FALSE
NCBIGENE:343	hgnc:642	AQP8	GuideToPharmacology	2024.1	agonist	0.3201687270469177	IUPHAR.LIGAND:1915	rxcui:8814	EPOPROSTENOL	TRUE	FALSE	FALSE
NCBIGENE:342	hgnc:608	APOC1P1	GuideToPharmacology	2024.1	agonist	0.7955707762984013	IUPHAR.LIGAND:1919	ncit:C84191	SULPROSTONE	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	antibody	0.036463661	IUPHAR.LIGAND:5046	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:7883	iuphar.ligand:7883	CP-724714	FALSE	FALSE	FALSE
NCBIGENE:1799	hgnc:3432	ERBB4	GuideToPharmacology	2024.1	NULL	0.4526523382387456	IUPHAR.LIGAND:4918	iuphar.ligand:4918	EPIREGULIN	FALSE	FALSE	FALSE
NCBIGENE:2019	hgnc:3342	EN1	GuideToPharmacology	2024.1	inhibitor	0.1367387271762877	IUPHAR.LIGAND:7944	ncit:C62496	TESEVATINIB	FALSE	FALSE	TRUE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	agonist	0.7955707762984014	IUPHAR.LIGAND:2825	iuphar.ligand:2825	DIARYLPROPIONITRILE	FALSE	FALSE	FALSE
NCBIGENE:1798	hgnc:2995	DPAGT1	GuideToPharmacology	2024.1	NULL	2.917092846427472	IUPHAR.LIGAND:5027	iuphar.ligand:5027	NEUREGULIN-1	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.074006584	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:10204	iuphar.ligand:10204	NORENDOXIFEN	FALSE	FALSE	FALSE
NCBIGENE:620	hgnc:1024	BCYRN1P2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:12715	iuphar.ligand:12715	GIREDESTRANT	FALSE	FALSE	FALSE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	agonist	0.076934317	IUPHAR.LIGAND:1016	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:621	hgnc:3468	ESR2	GuideToPharmacology	2024.1	inhibitor	0.076934317	IUPHAR.LIGAND:1016	rxcui:10324	TAMOXIFEN	TRUE	FALSE	TRUE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:7352	rxcui:1442132	MACITENTAN	TRUE	FALSE	FALSE
NCBIGENE:219	hgnc:407	ALDH1B1	GuideToPharmacology	2024.1	inhibitor	0.9376369863516875	IUPHAR.LIGAND:3539	ncit:C48430	ZIBOTENTAN	FALSE	FALSE	TRUE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:10198	iuphar.ligand:10198	INT-767	FALSE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.2035181055647073	THIAMYLAL	rxcui:10464	THIAMYLAL	TRUE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	agonist	0.1535312024435511	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.062808219	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	modulator	0.2302968036653267	IUPHAR.LIGAND:4146	ncit:C72111	BRETAZENIL	FALSE	FALSE	FALSE
NCBIGENE:406	hgnc:701	BMAL1	GuideToPharmacology	2024.1	blocker	0.060077427	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:4227	iuphar.ligand:4227	ISONIPECOTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:407	hgnc:710	ARR3	GuideToPharmacology	2024.1	modulator	0.4605936073306534	IUPHAR.LIGAND:4365	iuphar.ligand:4296	RO15-4513	FALSE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.058212496	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TdgClinicalTrial	Jan-14	NULL	0.1060761035064535	THIOPENTAL	rxcui:10493	THIOPENTAL	TRUE	FALSE	FALSE
NCBIGENE:408	hgnc:711	ARRB1	GuideToPharmacology	2024.1	modulator	0.2134458180312784	IUPHAR.LIGAND:4368	iuphar.ligand:4368	[18F]FLUOROETHYLFLUMAZENIL	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	modulator	0.3017682254924971	IUPHAR.LIGAND:4146	ncit:C72111	BRETAZENIL	FALSE	FALSE	FALSE
NCBIGENE:410	hgnc:713	ARSA	GuideToPharmacology	2024.1	blocker	0.095122593	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:409	hgnc:712	ARRB2	GuideToPharmacology	2024.1	blocker	0.078722146	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:421	hgnc:728	ARVCF	GuideToPharmacology	2024.1	agonist	0.4167275494896389	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:418	hgnc:724	ART2P	GuideToPharmacology	2024.1	blocker	1.141471113819445	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:3594	iuphar.ligand:3594	GALANIN-LIKE PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.9907107780319716	IUPHAR.LIGAND:6082	iuphar.ligand:6082	[SAR1, D-ALA12]GALANIN(1-16)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	agonist	0.3302369260106572	IUPHAR.LIGAND:6095	iuphar.ligand:6095	GALANIN(D-TRP2) (PIG)	FALSE	FALSE	FALSE
NCBIGENE:243	hgnc:431	ALOX12P1	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:3861	iuphar.ligand:3861	C7	FALSE	FALSE	FALSE
NCBIGENE:248	hgnc:437	ALPI	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:11998	iuphar.ligand:11998	MGIPANT-1	FALSE	FALSE	FALSE
NCBIGENE:444	hgnc:757	ASPH	GuideToPharmacology	2024.1	agonist	0.5000730593875667	IUPHAR.LIGAND:4077	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
NCBIGENE:445	hgnc:758	ASS1	GuideToPharmacology	2024.1	agonist	0.375054795	IUPHAR.LIGAND:4077	iuphar.ligand:4077	[3H]AMPA	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.043611023	IUPHAR.LIGAND:2866	rxcui:8638	PREDNISOLONE	TRUE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.056097939	IUPHAR.LIGAND:727	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.013836014	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	modulator	0.760980743	IUPHAR.LIGAND:11289	iuphar.ligand:11289	NYX-2925	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	agonist	0.069180068	IUPHAR.LIGAND:6511	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:456	hgnc:4585	GRIN2A	GuideToPharmacology	2024.1	blocker	0.1902451856365742	IUPHAR.LIGAND:4260	iuphar.ligand:4260	N1-DANSYL-SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	blocker	0.2822993077187876	IUPHAR.LIGAND:7595	rxcui:6378	LEVORPHANOL	TRUE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.1693795846312726	IUPHAR.LIGAND:3309	rxcui:1169	ASPARTIC ACID	TRUE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	inhibitor	0.4234489615781814	IUPHAR.LIGAND:4208	iuphar.ligand:4208	GV196771A	FALSE	FALSE	FALSE
NCBIGENE:459	hgnc:764	ASS1P14	GuideToPharmacology	2024.1	agonist	0.1881995384791917	IUPHAR.LIGAND:4268	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
NCBIGENE:2891	hgnc:4572	GRIA2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:12712	iuphar.ligand:12712	IPN60090	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	inhibitor	0.1842374429322614	IUPHAR.LIGAND:260	rxcui:27392	TROPISETRON	TRUE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	blocker	0.6908904109959803	IUPHAR.LIGAND:4286	iuphar.ligand:4286	PICROTIN	FALSE	FALSE	FALSE
NCBIGENE:424	ncbigene:424	ARVD3	GuideToPharmacology	2024.1	blocker	0.6908904109959803	IUPHAR.LIGAND:1862	iuphar.ligand:1862	GINKGOLIDE B	FALSE	FALSE	FALSE
NCBIGENE:427	hgnc:735	ASAH1	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:1862	iuphar.ligand:1862	GINKGOLIDE B	FALSE	FALSE	FALSE
NCBIGENE:936	hgnc:1647	CD24P2	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11297	iuphar.ligand:11297	GT-0198	FALSE	FALSE	FALSE
NCBIGENE:311	hgnc:535	ANXA11	GuideToPharmacology	2024.1	agonist	6.563458904461812	IUPHAR.LIGAND:2934	drugbank:DB03066	D-LACTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:401	hgnc:691	PHOX2A	GuideToPharmacology	2024.1	blocker	2.625383561784725	IUPHAR.LIGAND:2359	iuphar.ligand:2359	ZD7288	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TdgClinicalTrial	Jan-14	NULL	0.036463661	TRIFLUOPERAZINE	rxcui:10800	TRIFLUOPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:2907	hgnc:4589	GRINA	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9261	iuphar.ligand:9261	LUMINESPIB	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.4234489615781814	TRIPROLIDINE	rxcui:10849	TRIPROLIDINE	TRUE	FALSE	FALSE
NCBIGENE:2905	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	inhibitor	0.8468979231563628	IUPHAR.LIGAND:9828	iuphar.ligand:9828	ALVESPIMYCIN	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.1121958787087489	IUPHAR.LIGAND:8366	ncit:C68920	ABEXINOSTAT	FALSE	FALSE	TRUE
NCBIGENE:2614	ncbigene:2614	GAPDHL17	GuideToPharmacology	2024.1	inhibitor	0.1060761035064535	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2616	hgnc:4159	GAPDHP1	GuideToPharmacology	2024.1	inhibitor	0.061197752	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	1.346350544504987	IUPHAR.LIGAND:11072	ncit:C152324	SELIFORANT	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	inhibitor	0.4487835148349957	IUPHAR.LIGAND:8985	iuphar.ligand:8985	ADRIFORANT	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.1495945049449985	IUPHAR.LIGAND:1223	iuphar.ligand:1223	CLOBENPROPIT	FALSE	FALSE	FALSE
NCBIGENE:87	hgnc:163	ACTN1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:10568	iuphar.ligand:10568	GPR15L (71-81)	FALSE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:7799	iuphar.ligand:7799	COMPOUND 1A [PMID: 24900311]	FALSE	FALSE	FALSE
NCBIGENE:130	hgnc:255	ADH6	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:8773	iuphar.ligand:8773	LP-360924	FALSE	FALSE	FALSE
NCBIGENE:89	hgnc:165	ACTN3	GuideToPharmacology	2024.1	agonist	0.364636606	IUPHAR.LIGAND:2364	iuphar.ligand:2364	ANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:120	hgnc:245	ADD3	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:11212	iuphar.ligand:11212	6-NONYLPYRIDINE-2,4-DIOL	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:5560	iuphar.ligand:5560	T1117	FALSE	FALSE	FALSE
NCBIGENE:109	hgnc:234	ADCY3	GuideToPharmacology	2024.1	agonist	0.2500365296937833	IUPHAR.LIGAND:2661	iuphar.ligand:2661	N-OLEOYLETHANOLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:261	ncbigene:261	AMCN	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:12240	iuphar.ligand:12240	TALQUETAMAB	FALSE	FALSE	FALSE
UNIPROT:P18089	hgnc:282	ADRA2B	TdgClinicalTrial	Jan-14	NULL	0.1654653505326507	YOHIMBINE	rxcui:220982	YOHIMBINE	TRUE	FALSE	FALSE
NCBIGENE:2741	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	antibody	1.591141552596803	IUPHAR.LIGAND:8997	iuphar.ligand:8997	LIGELIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:122	ncbigene:122	ADFN	GuideToPharmacology	2024.1	agonist	2.500365296937833	IUPHAR.LIGAND:2906	iuphar.ligand:2906	LPA	FALSE	FALSE	FALSE
NCBIGENE:2741	hgnc:4326	GLRA1	GuideToPharmacology	2024.1	antibody	0.3977853881492007	IUPHAR.LIGAND:6890	rxcui:302379	OMALIZUMAB	TRUE	FALSE	FALSE
NCBIGENE:578	hgnc:949	BAK1	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:10355	iuphar.ligand:10355	GNE-616	FALSE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.039420174	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.2027323213733378	IUPHAR.LIGAND:7436	rxcui:588250	MILNACIPRAN	TRUE	FALSE	FALSE
NCBIGENE:926	hgnc:1707	CD8B	GuideToPharmacology	2024.1	inhibitor	0.1013661606866689	IUPHAR.LIGAND:7247	rxcui:31565	NEFAZODONE	TRUE	FALSE	FALSE
NCBIGENE:1817	hgnc:3027	DRD5P1	GuideToPharmacology	2024.1	inhibitor	0.3621218705909966	IUPHAR.LIGAND:336	drugbank:DB02152	K-252A	FALSE	FALSE	FALSE
NCBIGENE:1251	hgnc:7872	NOS1	GuideToPharmacology	2024.1	inhibitor	0.2465148884304905	IUPHAR.LIGAND:9849	iuphar.ligand:9849	GW274150	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.9053046764774912	VALRUBICIN	rxcui:31435	VALRUBICIN	TRUE	FALSE	TRUE
NCBIGENE:1611	hgnc:2672	DAP	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:7858	iuphar.ligand:7858	SACUBITRILAT	FALSE	FALSE	FALSE
NCBIGENE:470	ncbigene:470	ATHS	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9472	iuphar.ligand:9472	RGIA4	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:3970	iuphar.ligand:3970	&ALPHA;-CONOTOXIN MII	FALSE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	blocker	0.1325951293830669	IUPHAR.LIGAND:3990	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
NCBIGENE:464	hgnc:1957	CHRNA3	GuideToPharmacology	2024.1	agonist	0.3182283105193606	IUPHAR.LIGAND:5459	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
NCBIGENE:463	hgnc:777	ZFHX3	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:3977	iuphar.ligand:3976	[125I]EPIBATIDINE	FALSE	FALSE	FALSE
NCBIGENE:463	hgnc:777	ZFHX3	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:3976	iuphar.ligand:3976	[125I]EPIBATIDINE	FALSE	FALSE	FALSE
NCBIGENE:468	hgnc:786	ATF4	GuideToPharmacology	2024.1	agonist	0.9053046764774912	IUPHAR.LIGAND:7371	iuphar.ligand:7371	AQW051	FALSE	FALSE	FALSE
NCBIGENE:467	hgnc:785	ATF3	GuideToPharmacology	2024.1	blocker	0.6250913242344582	IUPHAR.LIGAND:3990	rxcui:6673	MECAMYLAMINE	TRUE	FALSE	FALSE
UNIPROT:P47871	hgnc:4192	GCGR	TEND	1-Aug-11	NULL	1.670698630226643	GLUCAGON RECOMBINANT	rxcui:261716	GLUCAGON (RDNA)	TRUE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2093	iuphar.ligand:2093	PHYLLOMEDUSIN	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:3835	iuphar.ligand:3835	[3H]SP (HUMAN, MOUSE, RAT)	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:2121	iuphar.ligand:2121	YM44781	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	agonist	0.4605936073306534	IUPHAR.LIGAND:2089	iuphar.ligand:2089	NEUROKININ A	FALSE	FALSE	FALSE
NCBIGENE:320	hgnc:578	APBA1	GuideToPharmacology	2024.1	agonist	1.280674908	IUPHAR.LIGAND:1685	iuphar.ligand:1685	UFP-102	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:1582	ncit:C156766	MECLINERTANT	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	inhibitor	0.596678082	IUPHAR.LIGAND:1486	iuphar.ligand:1486	RF9	FALSE	FALSE	FALSE
NCBIGENE:301	hgnc:533	ANXA1	GuideToPharmacology	2024.1	agonist	0.596678082	IUPHAR.LIGAND:1479	iuphar.ligand:1479	NEUROPEPTIDE FF	FALSE	FALSE	FALSE
NCBIGENE:300	hgnc:17425	NPFFR1	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:1486	iuphar.ligand:1486	RF9	FALSE	FALSE	FALSE
NCBIGENE:1873	hgnc:11918	TNFRSF4	GuideToPharmacology	2024.1	NULL	3.500511415712966	IUPHAR.LIGAND:5076	iuphar.ligand:5076	OX-40 LIGAND	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:9122	iuphar.ligand:9122	ACT-335827	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1705	iuphar.ligand:1705	SB-410220	FALSE	FALSE	FALSE
NCBIGENE:321	hgnc:579	APBA2	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1706	iuphar.ligand:1706	[3H]SB-674042	FALSE	FALSE	FALSE
NCBIGENE:322	hgnc:581	APBB1	GuideToPharmacology	2024.1	inhibitor	0.5834185692854944	IUPHAR.LIGAND:1706	iuphar.ligand:1706	[3H]SB-674042	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
NCBIGENE:2133	ncbigene:2133	EXT3	GuideToPharmacology	2024.1	modulator	5.250767123569449	IUPHAR.LIGAND:12266	iuphar.ligand:12266	BJG-05-039	FALSE	FALSE	FALSE
NCBIGENE:2134	hgnc:3515	EXTL1	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:8941	iuphar.ligand:8941	COMPOUND 4 [PMID: 24432870]	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:4115	iuphar.ligand:4115	A317491	FALSE	FALSE	FALSE
NCBIGENE:480	hgnc:14073	ATP1A4	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:11232	iuphar.ligand:11232	CAMLIPIXANT	FALSE	FALSE	FALSE
NCBIGENE:327	hgnc:586	APEH	GuideToPharmacology	2024.1	agonist	1.544343271638073	IUPHAR.LIGAND:1756	iuphar.ligand:1756	AR-C67085	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:1769	iuphar.ligand:1769	INS49266	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.2638576444004749	IUPHAR.LIGAND:6147	iuphar.ligand:6147	[3H]PSB-0413	FALSE	FALSE	FALSE
NCBIGENE:328	hgnc:587	APEX1	GuideToPharmacology	2024.1	inhibitor	0.1319288222002374	IUPHAR.LIGAND:1770	rxcui:1313722	REGRELOR	FALSE	FALSE	FALSE
NCBIGENE:329	hgnc:590	BIRC2	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:1725	iuphar.ligand:1725	PPADS	FALSE	FALSE	FALSE
NCBIGENE:324	hgnc:583	APC	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:1738	iuphar.ligand:1738	AR-C126313	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1746	iuphar.ligand:1746	INS48823	FALSE	FALSE	FALSE
NCBIGENE:326	hgnc:360	AIRE	GuideToPharmacology	2024.1	inhibitor	0.5250767123569451	IUPHAR.LIGAND:1725	iuphar.ligand:1725	PPADS	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:8910	iuphar.ligand:8910	SAR407899	FALSE	FALSE	FALSE
NCBIGENE:353	hgnc:626	APRT	GuideToPharmacology	2024.1	agonist	0.9376369863516875	IUPHAR.LIGAND:11906	iuphar.ligand:11906	COMPOUND 10D [PMID: 34855388]	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:11922	iuphar.ligand:11922	RLF-(A11-B10)-ISOPEPTIDE AMIDEA26 (XA11-B10)	FALSE	FALSE	FALSE
NCBIGENE:354	hgnc:6364	KLK3	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:3907	iuphar.ligand:3907	R3(B&DELTA;23-27)R/I5 CHIMERIC PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:747	hgnc:1165	DAGLA	GuideToPharmacology	2024.1	blocker	1.312691780892362	IUPHAR.LIGAND:4291	rxcui:8701	PROCAINE	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	inhibitor	0.750109589	IUPHAR.LIGAND:3324	iuphar.ligand:3324	VPC23019	FALSE	FALSE	FALSE
NCBIGENE:749	hgnc:10485	RYR3	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:4172	rxcui:3105	DANTROLENE	TRUE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	1.500219178	IUPHAR.LIGAND:11493	iuphar.ligand:11493	BMS-986166	FALSE	FALSE	FALSE
NCBIGENE:2994	hgnc:4703	GYPB	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:7972	iuphar.ligand:7972	WP1066	FALSE	FALSE	FALSE
NCBIGENE:916	hgnc:1674	CD3E	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:11905	ncit:C171901	ENAVOGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:355	hgnc:11920	FAS	GuideToPharmacology	2024.1	agonist	0.1810609352954983	IUPHAR.LIGAND:2004	iuphar.ligand:2004	BIM 23052	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.053038052	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:10708	iuphar.ligand:10708	SI306	FALSE	FALSE	FALSE
NCBIGENE:2206	hgnc:7316	MS4A2	GuideToPharmacology	2024.1	inhibitor	0.056459862	IUPHAR.LIGAND:7885	iuphar.ligand:7885	ENMD-2076	FALSE	FALSE	TRUE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:5646	iuphar.ligand:5646	ANALOG 3 [PMID:18543899]	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.525076712	IUPHAR.LIGAND:2035	iuphar.ligand:2035	BIM 23034	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.084689792	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:5634	iuphar.ligand:5634	SIFA-ASN(ACNH-&BETA;-GLC)-PEG-TYR3-OCTREOTATE	FALSE	FALSE	FALSE
NCBIGENE:357	hgnc:630	SHROOM2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:2053	iuphar.ligand:2053	NOC-ATE	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:2004	iuphar.ligand:2004	BIM 23052	FALSE	FALSE	FALSE
NCBIGENE:359	hgnc:634	AQP2	GuideToPharmacology	2024.1	inhibitor	0.2234368988752957	IUPHAR.LIGAND:2026	iuphar.ligand:2026	BIM 23454	FALSE	FALSE	FALSE
NCBIGENE:2902	hgnc:4584	GRIN1	GuideToPharmacology	2024.1	agonist	1.071585127259071	IUPHAR.LIGAND:11960	iuphar.ligand:11960	COMPOUND 53 [PMID: 33038794]	FALSE	FALSE	FALSE
NCBIGENE:166	hgnc:307	TLE5	GuideToPharmacology	2024.1	agonist	2.386712328895204	IUPHAR.LIGAND:3637	rxcui:37255	SUCCINIC ACID	TRUE	FALSE	FALSE
NCBIGENE:3108	hgnc:4934	HLA-DMA	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10676	iuphar.ligand:10676	AZ1366	FALSE	FALSE	FALSE
NCBIGENE:2419	hgnc:3930	FRA8B	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8853	iuphar.ligand:8853	YZM18	FALSE	FALSE	FALSE
NCBIGENE:1758	hgnc:2932	DMP1	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:9026	ncit:C80521	MOTOLIMOD	FALSE	FALSE	TRUE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1982	iuphar.ligand:1982	[125I]SAP	FALSE	FALSE	FALSE
NCBIGENE:1788	hgnc:2978	DNMT3A	GuideToPharmacology	2024.1	agonist	0.9723642821424906	IUPHAR.LIGAND:9713	iuphar.ligand:9713	H. POLYGYRUS TGF-&BETA; MIMIC	FALSE	FALSE	FALSE
NCBIGENE:346	hgnc:611	APOC4	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:1985	iuphar.ligand:1985	[3H]SQ-29548	FALSE	FALSE	FALSE
NCBIGENE:2420	ncbigene:2420	FRDA2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8670	iuphar.ligand:8670	COMPOUND 5 [PMID: 21741839]	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.2983390411119005	IUPHAR.LIGAND:2420	iuphar.ligand:2420	ALLYL ISOTHIOCYANATE	FALSE	FALSE	FALSE
NCBIGENE:2422	hgnc:3932	FRA8D	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8624	iuphar.ligand:8624	INHIBITOR 1 [COLOMBO ET AL., 2012]	FALSE	FALSE	FALSE
NCBIGENE:2851	hgnc:12405	TTR	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:8378	rxcui:1545063	TAFAMIDIS	TRUE	FALSE	FALSE
NCBIGENE:3009	hgnc:4719	H1-5	GuideToPharmacology	2024.1	antibody	26.25383561784724	IUPHAR.LIGAND:9947	iuphar.ligand:9947	ANATUMOMAB MAFENATOX	FALSE	FALSE	FALSE
NCBIGENE:489	hgnc:813	ATP2A3	GuideToPharmacology	2024.1	blocker	2.187819634820604	IUPHAR.LIGAND:10291	iuphar.ligand:10291	PICO145	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:10276	iuphar.ligand:10276	AM-0902	FALSE	FALSE	FALSE
UNIPROT:P48169	hgnc:4078	GABRA4	TEND	1-Aug-11	NULL	0.087318744	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	blocker	0.3088686543276147	IUPHAR.LIGAND:7091	rxcui:31994	NORGESTIMATE	TRUE	FALSE	FALSE
NCBIGENE:494	ncbigene:494	ATP3	GuideToPharmacology	2024.1	activator	1.381780822	IUPHAR.LIGAND:2451	ncit:C87339	NADIDE	FALSE	FALSE	FALSE
NCBIGENE:505	hgnc:9011	PKD2L1	GuideToPharmacology	2024.1	blocker	1.093909817410302	IUPHAR.LIGAND:4281	iuphar.ligand:4281	PHENAMIL	FALSE	FALSE	FALSE
NCBIGENE:512	hgnc:14006	TRPV6	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:12561	iuphar.ligand:12561	TRPV6 INHIBITOR CIS-22 A	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:11240	iuphar.ligand:11240	NSC600684	FALSE	FALSE	FALSE
NCBIGENE:3063	ncbigene:3063	HCVS	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10201	iuphar.ligand:10201	EXAMPLE 25 [WO2018228934]	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.078510274	CLOMIPRAMINE	rxcui:2597	CLOMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:605	hgnc:1004	BCL7A	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:2786	iuphar.ligand:2786	CALCITRIOL-26,23-LACTONE	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2204	iuphar.ligand:2204	YM 218	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:2198	iuphar.ligand:2198	RWJ-351647	FALSE	FALSE	FALSE
NCBIGENE:366	hgnc:643	AQP9	GuideToPharmacology	2024.1	inhibitor	0.2778183663264258	IUPHAR.LIGAND:2211	iuphar.ligand:2211	[PHAA1,D-TYR2,VAL4,ARG6,ARG-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:367	hgnc:644	AR	GuideToPharmacology	2024.1	agonist	0.002248915	IUPHAR.LIGAND:2176	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	agonist	0.033658764	IUPHAR.LIGAND:2176	rxcui:1098	ARGIPRESSIN	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2212	iuphar.ligand:2212	[TBAA1,D-TYR(ET)2,VAL4,LYS6,ARG-NH28,DES-GLY9]AVP	FALSE	FALSE	FALSE
UNIPROT:P47870	hgnc:4082	GABRB2	TEND	1-Aug-11	NULL	0.083257407	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
NCBIGENE:368	hgnc:57	ABCC6	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:2210	iuphar.ligand:2210	[PHAA1,D-TYR(ME)2,ARG6,TYR-NH29]AVP	FALSE	FALSE	FALSE
NCBIGENE:306	hgnc:541	ANXA3	GuideToPharmacology	2024.1	agonist	1.944728564284981	IUPHAR.LIGAND:1536	iuphar.ligand:1536	NPY-(16-36) (PIG)	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.6351734423672721	CYCLIZINE	rxcui:2977	CYCLIZINE	TRUE	FALSE	FALSE
NCBIGENE:587	hgnc:977	BCAT2	GuideToPharmacology	2024.1	agonist	0.3977853881492008	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	CIViC	10-Apr-24	NULL	0.2041114528112516	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
CD44	hgnc:1681	CD44	CIViC	10-Apr-24	NULL	0.019059046	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
UNIPROT:P04150	hgnc:7978	NR3C1	TEND	1-Aug-11	NULL	0.03262504	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NECTIN4	hgnc:19688	NECTIN4	CIViC	10-Apr-24	NULL	4.118248724368196	ENFORTUMAB VEDOTIN	rxcui:2268306	ENFORTUMAB VEDOTIN-EJFV	TRUE	FALSE	TRUE
ATRX	hgnc:886	ATRX	CIViC	10-Apr-24	NULL	0.030176823	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	CIViC	10-Apr-24	NULL	0.1331836936859721	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
TFF3	hgnc:11757	TFF3	CIViC	10-Apr-24	NULL	3.281729452230906	AMINOGLUTETHIMIDE	rxcui:677	AMINOGLUTETHIMIDE	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	CIViC	10-Apr-24	NULL	0.006137659	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
HMOX1	hgnc:5013	HMOX1	CIViC	10-Apr-24	NULL	0.051177067	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
UNIPROT:Q14524	hgnc:10593	SCN5A	TEND	1-Aug-11	NULL	0.2983390411119005	DIBUCAINE	rxcui:3339	DIBUCAINE	TRUE	FALSE	FALSE
FOXP3	hgnc:6106	FOXP3	CIViC	10-Apr-24	NULL	0.7292732116068681	EPIRUBICIN	rxcui:3995	EPIRUBICIN	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	CIViC	10-Apr-24	NULL	0.3454452054979901	MTOR KINASE INHIBITOR AZD8055	ncit:C78856	MTOR KINASE INHIBITOR AZD8055	FALSE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	CIViC	10-Apr-24	NULL	0.1176247115494948	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
TP53	hgnc:11998	TP53	CIViC	10-Apr-24	NULL	0.008429889	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.4907258993990139	DIETHYLPROPION	rxcui:3389	DIETHYLPROPION	TRUE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.2430910705356226	MTOR KINASE INHIBITOR PP242	ncit:C128632	MTOR KINASE INHIBITOR PP242	FALSE	FALSE	TRUE
IGF2	hgnc:5466	IGF2	CIViC	10-Apr-24	NULL	0.03136659	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	1.270346884734544	EMEDASTINE	rxcui:28144	EMEDASTINE	TRUE	FALSE	FALSE
ZHX2	hgnc:18513	ZHX2	CIViC	10-Apr-24	NULL	0.1842374429322613	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
AURKB	hgnc:11390	AURKB	CIViC	10-Apr-24	NULL	0.3562257207306275	BARASERTIB	ncit:C62502	BARASERTIB	FALSE	FALSE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.062808219	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
APC	hgnc:583	APC	JAX-CKB	10-Apr-24	NULL	0.7955707762984013	STP1002	ncit:C174060	BASROPARIB	FALSE	FALSE	FALSE
ATM	hgnc:795	ATM	JAX-CKB	10-Apr-24	NULL	0.038880171	Leucovorin	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TEND	1-Aug-11	NULL	0.3763990769583835	ENFLURANE	rxcui:3920	ENFLURANE	TRUE	FALSE	FALSE
ATR	hgnc:882	ATR	JAX-CKB	10-Apr-24	NULL	0.9723642821424907	Berzosertib	ncit:C116355	BERZOSERTIB	FALSE	FALSE	FALSE
ATR	hgnc:882	ATR	JAX-CKB	10-Apr-24	NULL	0.8751278539282416	Ceralasertib	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.06109095	CI-1040	drugbank:DB12429	CI-1040	FALSE	FALSE	TRUE
UNIPROT:Q07343	hgnc:8781	PDE4B	TEND	1-Aug-11	NULL	0.5000730593875666	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:O95069	hgnc:6277	KCNK2	TEND	1-Aug-11	NULL	1.154014752432846	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.068369364	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P21918	hgnc:3026	DRD5	TEND	1-Aug-11	NULL	0.2625383561784725	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P08913	hgnc:281	ADRA2A	TEND	1-Aug-11	NULL	0.030527716	FENOLDOPAM	rxcui:203151	FENOLDOPAM MESYLATE	TRUE	FALSE	FALSE
UNIPROT:P18405	hgnc:11284	SRD5A1	TEND	1-Aug-11	NULL	1.250182648468916	FINASTERIDE	rxcui:25025	FINASTERIDE	TRUE	FALSE	FALSE
UNIPROT:P31644	hgnc:4079	GABRA5	TEND	1-Aug-11	NULL	0.099446347	FLUMAZENIL	rxcui:4457	FLUMAZENIL	TRUE	FALSE	FALSE
UNIPROT:P08254	hgnc:7173	MMP3	TEND	1-Aug-11	NULL	0.7501095890813501	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.037734582	FLUSPIRILENE	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1376949420516464	FLUVOXAMINE	rxcui:42355	FLUVOXAMINE	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.2983390411119005	FLURBIPROFEN	rxcui:4502	FLURBIPROFEN	TRUE	FALSE	FALSE
UNIPROT:Q00975	hgnc:1389	CACNA1B	TEND	1-Aug-11	NULL	0.1230648544586589	GABAPENTIN	rxcui:25480	GABAPENTIN	TRUE	FALSE	FALSE
UNIPROT:P08253	hgnc:7166	MMP2	TEND	1-Aug-11	NULL	0.3590268118679965	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
UNIPROT:Q8N1C3	hgnc:4086	GABRG1	TEND	1-Aug-11	NULL	0.100976291	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.1074020548002842	INDOMETHACIN	rxcui:5781	INDOMETHACIN	TRUE	FALSE	FALSE
UNIPROT:Q9Y5Y9	hgnc:10582	SCN10A	TEND	1-Aug-11	NULL	0.1219218372345847	LEVOBUPIVACAINE	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
PATTERN RECOGNITION RECEPTOR NOD2	hgnc:5331	NOD2	TTD	2020.06.01	NULL	1.875273972703375	MIS-416	ncit:C127934	MICROPARTICLE MDP/BACTERIAL DNA-CONTAINING MIS416	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.000146118775133	EMD-1204831	chembl:CHEMBL3545053	EMD-1204831	FALSE	FALSE	FALSE
AURORA KINASE A	hgnc:11393	AURKA	TTD	2020.06.01	NULL	0.1582152052299645	MLN8237	ncit:C71717	ALISERTIB	FALSE	FALSE	TRUE
TAX TRANSCRIPTIONALLY-ACTIVATED GLYCOPROTEIN 1	hgnc:11918	TNFRSF4	TTD	2020.06.01	NULL	3.500511415712966	MEDI6383	ncit:C118282	EFIZONERIMOD	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.045226246	LABETALOL	rxcui:6185	LABETALOL	TRUE	FALSE	FALSE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.5834185692854944	MK-1496	drugbank:DB12763	MK-1496	FALSE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.1930429089547592	Milataxel	ncit:C77880	MILATAXEL	FALSE	FALSE	FALSE
DIHYDROOROTATE DEHYDROGENASE	hgnc:2867	DHODH	TTD	2020.06.01	NULL	2.763561643983921	BAY2402234	ncit:C153137	ORLUDODSTAT	FALSE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.3201687270469177	APG-1252	ncit:C148488	PELCITOCLAX	FALSE	FALSE	FALSE
UNIPROT:Q13946	hgnc:8791	PDE7A	TEND	1-Aug-11	NULL	3.000438356325399	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
APOPTOSIS REGULATOR BCL-2	hgnc:990	BCL2	TTD	2020.06.01	NULL	0.6403374540938354	BCL201	ncit:C125603	BCL-2 INHIBITOR BCL201	FALSE	FALSE	FALSE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.4907258993990139	AZD9496	ncit:C122834	SELECTIVE ESTROGEN RECEPTOR DEGRADER AZD9496	FALSE	FALSE	TRUE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	0.2500365296937833	CBT-101	ncit:C129717	VEBRELTINIB	FALSE	FALSE	FALSE
APOPTOSIS INHIBITOR SURVIVIN	hgnc:593	BIRC5	TTD	2020.06.01	NULL	0.596678082	SurVaxM	drugbank:DB17397	SURVAXM	FALSE	FALSE	FALSE
MACROPHAGE COLONY-STIMULATING FACTOR 1 RECEPTOR	hgnc:2433	CSF1R	TTD	2020.06.01	NULL	0.3182283105193605	PLX7486	iuphar.ligand:9104	PLX7486	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE MER	hgnc:7027	MERTK	TTD	2020.06.01	NULL	3.500511415712966	ONO-7475	chembl:CHEMBL4650414	ONO-7475	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE SYK	hgnc:11491	SYK	TTD	2020.06.01	NULL	0.1666910197958555	GSK2646264	iuphar.ligand:10108	GSK2646264	FALSE	FALSE	FALSE
TYROSINE-PROTEIN KINASE BTK	hgnc:1133	BTK	TTD	2020.06.01	NULL	0.5147810905460245	LOU064	ncit:C175851	REMIBRUTINIB	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.2263261691193728	Gepotidacin	ncit:C170025	GEPOTIDACIN	FALSE	FALSE	FALSE
CHOLINERGIC RECEPTOR UNSPECIFIC	ncbigene:1125	CHR	TTD	2020.06.01	NULL	4.375639269641208	Sofpironium bromide	ncit:C152384	SOFPIRONIUM BROMIDE	FALSE	FALSE	FALSE
RETINAL PIGMENT EPITHELIUM PROTEIN	hgnc:10294	RPE65	TTD	2020.06.01	NULL	15.00219178	Emixustat	ncit:C171669	EMIXUSTAT	FALSE	FALSE	FALSE
KININOGEN	hgnc:6383	KNG1	TTD	2020.06.01	NULL	13.12691780892362	Avoralstat	ncit:C169799	AVORALSTAT	FALSE	FALSE	FALSE
MINERALOCORTICOID RECEPTOR	hgnc:7979	NR3C2	TTD	2020.06.01	NULL	2.763561643983921	XL550	chembl:CHEMBL3545393	XL550	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TEND	1-Aug-11	NULL	0.055387839	MIDAZOLAM	rxcui:203128	MIDAZOLAM HYDROCHLORIDE	TRUE	FALSE	FALSE
STRESS-ACTIVATED PROTEIN KINASE	hgnc:1189	AHSA1	TTD	2020.06.01	NULL	4.375639269641208	LY-2228820	ncit:C105853	RALIMETINIB MESYLATE	FALSE	FALSE	TRUE
COAGULATION FACTOR XA	hgnc:3528	F10	TTD	2020.06.01	NULL	0.6429510763554428	DU-176b	rxcui:1599538	EDOXABAN	TRUE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.4039051633514961	CLR-1401	chembl:CHEMBL208375	IOPOFOSINE	FALSE	FALSE	FALSE
UNIPROT:P41145	hgnc:8154	OPRK1	TEND	1-Aug-11	NULL	0.4930297768609811	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SOMATOSTATIN RECEPTOR TYPE 1	hgnc:11330	SSTR1	TTD	2020.06.01	NULL	1.093909817410302	Pasireotide	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
SOMATOSTATIN RECEPTOR TYPE 2	hgnc:11331	SSTR2	TTD	2020.06.01	NULL	0.729273212	Pasireotide	rxcui:1364105	PASIREOTIDE	TRUE	FALSE	TRUE
ESTROGEN-RELATED RECEPTOR-ALPHA	hgnc:3471	ESRRA	TTD	2020.06.01	NULL	8.751278539282415	Corticosteroid	wikidata:Q210420	CORTICOSTEROID	FALSE	FALSE	FALSE
SOLUTE CARRIER FAMILY 40 MEMBER 1	hgnc:10909	SLC40A1	TTD	2020.06.01	NULL	157.5230137070835	LY2928057	iuphar.ligand:8416	LY2928057	FALSE	FALSE	FALSE
FATTY ACID SYNTHASE	hgnc:3594	FASN	TTD	2020.06.01	NULL	3.889457128569962	TVB-2640	ncit:C118285	DENIFANSTAT	FALSE	FALSE	FALSE
UNIPROT:P35354	hgnc:9605	PTGS2	TEND	1-Aug-11	NULL	0.1684738114514262	NAPROXEN	rxcui:142442	NAPROXEN SODIUM	TRUE	FALSE	FALSE
VASOPRESSIN V1A RECEPTOR	hgnc:895	AVPR1A	TTD	2020.06.01	NULL	1.369765336583334	RG7314	ncit:C169802	BALOVAPTAN	FALSE	FALSE	FALSE
CARBONIC ANHYDRASE II	hgnc:1373	CA2	TTD	2020.06.01	NULL	0.2692701089009974	Ethoxzolamide	ncit:C65561	ETHOXZOLAMIDE	TRUE	FALSE	FALSE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.1223955040459079	Fenofibrate	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.037734582	Fluspirilene	rxcui:4507	FLUSPIRILENE	TRUE	FALSE	FALSE
CASPASE-1	hgnc:1499	CASP1	TTD	2020.06.01	NULL	1.009762908	PRALNACASAN	ncit:C76768	PRALNACASAN	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.3117023117067671	NALOXONE	rxcui:203192	NALOXONE HYDROCHLORIDE	TRUE	FALSE	FALSE
5-HT 3 RECEPTOR	hgnc:5297	HTR3A	TTD	2020.06.01	NULL	1.166837138570988	Pancopride	ncit:C87213	PANCOPRIDE	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.2573905452730122	Anisotropine Methylbromide	rxcui:17945	OCTOTROPINE METHYLBROMIDE	TRUE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.7721716358190367	Amocarzine	ncit:C72145	AMOCARZINE	FALSE	FALSE	FALSE
UNIPROT:P35372	hgnc:8156	OPRM1	TEND	1-Aug-11	NULL	0.1605739181519709	NALBUPHINE	rxcui:154985	NALBUPHINE HYDROCHLORIDE	TRUE	FALSE	FALSE
ROTAMASE B	hgnc:9255	PPIB	TTD	2020.06.01	NULL	13.12691780892362	L-Proline	rxcui:8737	PROLINE	TRUE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TEND	1-Aug-11	NULL	0.6105543166941221	ORCIPRENALINE	rxcui:7688	METAPROTERENOL	TRUE	FALSE	FALSE
CASPASE	hgnc:2379	CRTAP	TTD	2020.06.01	NULL	52.50767123569449	NCX-1000	drugbank:DB16026	NCX-1000	FALSE	FALSE	FALSE
MHC CLASS II ANTIGEN DRB1*1	hgnc:4948	HLA-DRB1	TTD	2020.06.01	NULL	0.5114383561918295	Glatiramer Acetate	rxcui:214582	GLATIRAMER	TRUE	FALSE	FALSE
TUBULIN	hgnc:12406	TUB	TTD	2020.06.01	NULL	0.039538909	Docetaxel	rxcui:1299922	DOCETAXEL ANHYDROUS	TRUE	FALSE	TRUE
ADENYLATE CYCLASE TYPE 1	hgnc:232	ADCY1	TTD	2020.06.01	NULL	8.751278539282415	Adenosine monophosphate	rxcui:309	ADENOSINE MONOPHOSPHATE	TRUE	FALSE	FALSE
P2Y PURINOCEPTOR 2	hgnc:8541	P2RY2	TTD	2020.06.01	NULL	3.500511415712966	Diquafosol	ncit:C65436	DIQUAFOSOL	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.1037701012563132	Umespirone	ncit:C152798	UMESPIRONE	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II BETA	hgnc:11990	TOP2B	TTD	2020.06.01	NULL	1.312691780892362	Dexrazoxane	rxcui:42736	DEXRAZOXANE	TRUE	FALSE	FALSE
PROTO-ONCOGENE C-SRC	hgnc:11283	SRC	TTD	2020.06.01	NULL	0.3241214273808302	SKI-758	chembl:CHEMBL219557	CHEMBL:CHEMBL219557	FALSE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Flutropium bromide	ncit:C80960	FLUTROPIUM BROMIDE	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.1881995384791917	CPL-7075	ncit:C174799	LENABASUM	FALSE	FALSE	FALSE
THROMBOXANE A2 RECEPTOR	hgnc:11608	TBXA2R	TTD	2020.06.01	NULL	0.4167275494896389	LAROPIPRANT	ncit:C87372	LAROPIPRANT	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.9907107780319716	Chlamydocin	chembl:CHEMBL2371450	CHLAMYDOCIN	FALSE	FALSE	FALSE
SARCOPLASMIC/ENDOPLASMIC RETICULUM CALCIUM ATPASE	hgnc:811	ATP2A1	TTD	2020.06.01	NULL	0.8751278539282416	Artesunate	rxcui:18346	ARTESUNATE	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.8334550989792777	Matuzumab	ncit:C2012	MATUZUMAB	FALSE	FALSE	TRUE
ESTROGEN RECEPTOR	hgnc:3467	ESR1	TTD	2020.06.01	NULL	0.1090501998664475	Mestranol	rxcui:6782	MESTRANOL	TRUE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.3889457128569962	SALVINORIN A	drugbank:DB12327	SALVINORIN A	FALSE	FALSE	FALSE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.2895643634321387	Pyridostigmine	rxcui:9000	PYRIDOSTIGMINE	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.4773424657790409	IMRECOXIB	drugbank:DB12354	IMRECOXIB	FALSE	FALSE	FALSE
HISTONE DEACETYLASE	hgnc:14065	HDAC9	TTD	2020.06.01	NULL	1.166837138570988	CXD-101	chembl:CHEMBL4297489	CXD-101	FALSE	FALSE	FALSE
A PROLIFERATION-INDUCING LIGAND	hgnc:11928	TNFSF13	TTD	2020.06.01	NULL	39.38075342677087	Atacicept	ncit:C81166	ATACICEPT	FALSE	FALSE	FALSE
AROMATASE	hgnc:2594	CYP19A1	TTD	2020.06.01	NULL	0.9376369863516875	LIAROZOLE	ncit:C1433	LIAROZOLE	FALSE	FALSE	FALSE
XANTHINE DEHYDROGENASE/OXIDASE	hgnc:12805	XDH	TTD	2020.06.01	NULL	0.6731752722524935	Cyclic pyranopterin monophosphate	rxcui:2531288	FOSDENOPTERIN	TRUE	FALSE	FALSE
OPIOID RECEPTOR KAPPA	hgnc:8154	OPRK1	TTD	2020.06.01	NULL	0.1479089330582944	CHLOROXINE	rxcui:20875	CHLOROXINE	TRUE	FALSE	FALSE
BETA-SECRETASE	hgnc:933	BACE1	TTD	2020.06.01	NULL	2.019525817	AZD-3839	drugbank:DB12368	AZD-3839	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.8751278539282416	Gimatecan	ncit:C65804	GIMATECAN	FALSE	FALSE	FALSE
CHECKPOINT KINASE-1	hgnc:1925	CHEK1	TTD	2020.06.01	NULL	2.072671233	LY2603618	ncit:C81937	RABUSERTIB	FALSE	FALSE	TRUE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	1.479089330582943	ORM-12741	drugbank:DB12057	ORM-12741	FALSE	FALSE	FALSE
GLUTAMINASE	hgnc:4331	GLS	TTD	2020.06.01	NULL	0.3697723326457359	CB-839	ncit:C114381	TELAGLENASTAT	FALSE	FALSE	FALSE
PROTO-ONCOGENE C-MET	hgnc:7029	MET	TTD	2020.06.01	NULL	1.000146118775133	AMG 208	ncit:C82677	C-MET INHIBITOR AMG 208	FALSE	FALSE	TRUE
COAGULATION FACTOR IX	hgnc:3551	F9	TTD	2020.06.01	NULL	0.6908904109959803	Emicizumab	rxcui:1989794	EMICIZUMAB	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	0.16256245	Promazine	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
BETA-GLUCURONIDASE	hgnc:4696	GUSB	TTD	2020.06.01	NULL	26.25383561784724	Vestronidase alfa	rxcui:1989818	VESTRONIDASE ALFA-VJBK	TRUE	FALSE	FALSE
CALCITONIN GENE-RELATED PEPTIDE RECEPTOR	hgnc:16709	CALCRL	TTD	2020.06.01	NULL	1.166837138570988	Galcanezumab	rxcui:2058846	GALCANEZUMAB	TRUE	FALSE	FALSE
PLASMA KALLIKREIN	hgnc:6371	KLKB1	TTD	2020.06.01	NULL	7.501095891	Lanadelumab	rxcui:2055640	LANADELUMAB-FLYO	TRUE	FALSE	FALSE
INTESTINAL MALTASE-GLUCOAMYLASE	hgnc:7043	MGAM	TTD	2020.06.01	NULL	1.193356164447602	Deoxynojirimycin	ncit:C87373	DUVOGLUSTAT	FALSE	FALSE	FALSE
5-HT 4 RECEPTOR	hgnc:5299	HTR4	TTD	2020.06.01	NULL	0.6731752722524935	Lintopride	ncit:C66018	LINTOPRIDE	FALSE	FALSE	FALSE
PROTEIN-TYROSINE PHOSPHATASE SIGMA	hgnc:9681	PTPRS	TTD	2020.06.01	NULL	3.750547945406749	Etidronic acid	rxcui:1356715	ETIDRONIC ACID	TRUE	FALSE	TRUE
PHOSPHODIESTERASE 4A	hgnc:8780	PDE4A	TTD	2020.06.01	NULL	0.2983390411119005	CC-1088	ncit:C2210	SELECTIVE CYTOKINE INHIBITORY DRUG CC-1088	FALSE	FALSE	FALSE
ADRENERGIC RECEPTOR ALPHA-2C	hgnc:283	ADRA2C	TTD	2020.06.01	NULL	0.082171629	TNX-102	rxcui:21949	CYCLOBENZAPRINE	TRUE	FALSE	FALSE
UNIPROT:P43681	hgnc:1958	CHRNA4	TEND	1-Aug-11	NULL	0.063839114	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
B-CELL MATURATION PROTEIN	hgnc:11913	TNFRSF17	TTD	2020.06.01	NULL	2.763561643983921	Autologous Anti-BCMA-CAR-expressing CD4+/CD8+ T-lymphocytes FCARH143	ncit:C142807	AUTOLOGOUS ANTI-BCMA-CAR-EXPRESSING CD4+/CD8+ T-LYMPHOCYTES FCARH143	FALSE	FALSE	FALSE
B-LYMPHOCYTE SURFACE ANTIGEN B4	hgnc:1633	CD19	TTD	2020.06.01	NULL	1.280674908	SJCAR19	ncit:C142887	AUTOLOGOUS ANTI-CD19 CHIMERIC ANTIGEN RECEPTOR T-CELLS SJCAR19	FALSE	FALSE	FALSE
PHOSPHODIESTERASE 5A	hgnc:8784	PDE5A	TTD	2020.06.01	NULL	4.922594178346359	Avanafil	rxcui:1291301	AVANAFIL	TRUE	FALSE	FALSE
PLACENTA GROWTH FACTOR	hgnc:8893	PGF	TTD	2020.06.01	NULL	7.001022831425934	Aflibercept	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.067231333	Regorafenib	rxcui:1312397	REGORAFENIB	TRUE	FALSE	TRUE
SERINE/THREONINE-PROTEIN KINASE B-RAF	hgnc:1097	BRAF	TTD	2020.06.01	NULL	1.657092009619794	Vemurafenib	rxcui:1147220	VEMURAFENIB	TRUE	FALSE	TRUE
INTERLEUKIN-2	hgnc:6001	IL2	TTD	2020.06.01	NULL	0.027347745	Aldesleukin	rxcui:70223	ALDESLEUKIN	TRUE	FALSE	TRUE
5-HT 1A RECEPTOR	hgnc:5286	HTR1A	TTD	2020.06.01	NULL	0.3547815624033412	OPC-14523	drugbank:DB05422	OPC-14523	FALSE	FALSE	FALSE
OPIOID RECEPTOR SIGMA 1	hgnc:8157	SIGMAR1	TTD	2020.06.01	NULL	1.050153425	OPC-14523	drugbank:DB05422	OPC-14523	FALSE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.035083077	Dihydrotestosterone	ncit:C29619	DIHYDROTESTOSTERONE	FALSE	FALSE	FALSE
SPHINGOSINE KINASE 1	hgnc:11240	SPHK1	TTD	2020.06.01	NULL	3.750547945406749	Phenoxodiol	ncit:C2642	IDRONOXIL	FALSE	FALSE	TRUE
ALK TYROSINE KINASE RECEPTOR	hgnc:427	ALK	TTD	2020.06.01	NULL	2.407466349146467	AP26113	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
FRUCTOSE-1,6-BISPHOSPHATASE	hgnc:3606	FBP1	TTD	2020.06.01	NULL	26.25383561784724	MB07803	chembl:CHEMBL4297400	MB-07803	FALSE	FALSE	FALSE
DNA TOPOISOMERASE II	hgnc:11989	TOP2A	TTD	2020.06.01	NULL	0.9053046764774912	Pixantrone	ncit:C26663	PIXANTRONE	TRUE	FALSE	TRUE
PARATHYROID HORMONE	hgnc:9606	PTH	TTD	2020.06.01	NULL	0.4487835148349957	Ostabolin-C	chembl:CHEMBL4802222	OSTABOLIN-C	FALSE	FALSE	FALSE
DUAL-SPECIFICITY TYROSINE-PHOSPHORYLATION REGULATED KINASE 3	hgnc:3094	DYRK3	TTD	2020.06.01	NULL	0.3182283105193606	HARMINE	ncit:C97713	HARMINE	FALSE	FALSE	FALSE
S-MEPHENYTOIN 4-HYDROXYLASE	hgnc:2623	CYP2C9	TTD	2020.06.01	NULL	0.045579576	Sulfaphenazole	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
COAGULATION FACTOR IIA	hgnc:3535	F2	TTD	2020.06.01	NULL	2.763561643983921	Bivalirudin	rxcui:60819	BIVALIRUDIN	TRUE	FALSE	FALSE
CORTICOSTEROID-BINDING GLOBULIN	hgnc:1540	SERPINA6	TTD	2020.06.01	NULL	3.281729452230906	Ciclesonide	rxcui:274964	CICLESONIDE	TRUE	FALSE	FALSE
VITAMIN D3 RECEPTOR	hgnc:12679	VDR	TTD	2020.06.01	NULL	0.027870314	Cholecalciferol	rxcui:2418	CHOLECALCIFEROL	TRUE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE	hgnc:2294	COX8A	TTD	2020.06.01	NULL	0.070197421	Diclofenac	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.158793361	Diphenhydramine	rxcui:3498	DIPHENHYDRAMINE	TRUE	FALSE	FALSE
CATECHOL-O-METHYL-TRANSFERASE	hgnc:2228	COMT	TTD	2020.06.01	NULL	1.500219178	Entacapone	rxcui:60307	ENTACAPONE	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M5	hgnc:1954	CHRM5	TTD	2020.06.01	NULL	1.029562181092049	Propiverine	rxcui:55175	PROPIVERINE	FALSE	FALSE	FALSE
DOPAMINE D2 RECEPTOR	hgnc:3023	DRD2	TTD	2020.06.01	NULL	0.028626235	Thioridazine	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.007496384	Testosterone	rxcui:10379	TESTOSTERONE	TRUE	FALSE	FALSE
BILIVERDIN REDUCTASE A	hgnc:1062	BLVRA	TTD	2020.06.01	NULL	0.1367387271762877	Ursodeoxycholic acid	rxcui:11065	URSODIOL	TRUE	FALSE	FALSE
MUSCARINIC ACETYLCHOLINE RECEPTOR M3	hgnc:1952	CHRM3	TTD	2020.06.01	NULL	0.2365210416022274	Tolterodine	rxcui:119565	TOLTERODINE	TRUE	FALSE	FALSE
TROPOMYOSIN-RELATED KINASE A	hgnc:8031	NTRK1	TTD	2020.06.01	NULL	0.2397610558707511	PLX7486	iuphar.ligand:9104	PLX7486	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.067231333	VS-5584	drugbank:DB12986	VS-5584	FALSE	FALSE	FALSE
INTERLEUKIN 3 RECEPTOR ALPHA	hgnc:6012	IL3RA	TTD	2020.06.01	NULL	5.250767123569449	UCART123	ncit:C146806	ALLOGENEIC CD123-SPECIFIC UNIVERSAL CAR123-EXPRESSING T-LYMPHOCYTES	FALSE	FALSE	FALSE
ERBB2 TYROSINE KINASE RECEPTOR	hgnc:3430	ERBB2	TTD	2020.06.01	NULL	0.1480479452134243	AZD8931	ncit:C77887	SAPITINIB	FALSE	FALSE	TRUE
POLO-LIKE KINASE 1	hgnc:9077	PLK1	TTD	2020.06.01	NULL	0.2917092846427472	BI 2536	drugbank:DB16107	BI 2536	FALSE	FALSE	FALSE
MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN	hgnc:7467	MTTP	TTD	2020.06.01	NULL	13.12691780892362	Implitapide	ncit:C65901	IMPLITAPIDE	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.3889457128569962	Met-enkephalin	rxcui:1349278	METENKEFALIN	FALSE	FALSE	FALSE
GLUCOKINASE	hgnc:4195	GCK	TTD	2020.06.01	NULL	7.001022831425932	PF-04991532	drugbank:DB11765	PF-04991532	FALSE	FALSE	FALSE
SERINE/THREONINE-PROTEIN KINASE MTOR	hgnc:3942	MTOR	TTD	2020.06.01	NULL	0.069332312	SAR245409	ncit:C71704	VOXTALISIB	FALSE	FALSE	TRUE
ADENOSINE A1 RECEPTOR	hgnc:262	ADORA1	TTD	2020.06.01	NULL	0.5469549087051511	Tonapofylline	ncit:C96194	TONAPOFYLLINE	FALSE	FALSE	FALSE
GLUTATHIONE S-TRANSFERASE P	hgnc:4638	GSTP1	TTD	2020.06.01	NULL	1.750255707856483	Canfosfamide	ncit:C83581	CANFOSFAMIDE	FALSE	FALSE	FALSE
ALDOSE REDUCTASE	hgnc:381	AKR1B1	TTD	2020.06.01	NULL	4.039051633514961	Fidarestat	ncit:C81355	FIDARESTAT	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.0403388	Cediranib	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA	hgnc:9232	PPARA	TTD	2020.06.01	NULL	0.3182283105193606	CS-038	iuphar.ligand:12287	CHIGLITAZAR	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.1265245090016735	IUPHAR.LIGAND:7191	rxcui:228783	FROVATRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.008323981	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.070291394	IUPHAR.LIGAND:40	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.037884323	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	agonist	0.1389091831632129	IUPHAR.LIGAND:2941	rxcui:1300701	LORCASERIN	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:198	ncit:C72684	AGOMELATINE	TRUE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:136	iuphar.ligand:136	RAUWOLSCINE	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:176	iuphar.ligand:176	EGIS-7625	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:176	iuphar.ligand:176	EGIS-7625	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	inhibitor	0.1286952726365061	IUPHAR.LIGAND:194	iuphar.ligand:194	SB 243213	FALSE	FALSE	FALSE
NCBIGENE:11	hgnc:15	NATP	GuideToPharmacology	2024.1	inhibitor	0.2966535098061835	IUPHAR.LIGAND:274	iuphar.ligand:274	RO 04-6790	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613069	IUPHAR.LIGAND:272	iuphar.ligand:272	2-BROMO-LSD	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.2302968036653267	IUPHAR.LIGAND:283	ncit:C66417	PIRENPERONE	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.031765076	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:2465	hgnc:3862	FRA17A	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:6602	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:1787	hgnc:2977	TRDMT1	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10662	iuphar.ligand:10662	BMS-986260	FALSE	FALSE	FALSE
NCBIGENE:1264	hgnc:2155	CNN1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:8884	iuphar.ligand:8884	COMPOUND 21 [PMID: 23981033]	FALSE	FALSE	FALSE
NCBIGENE:1792	hgnc:174	ACVR2B	GuideToPharmacology	2024.1	antibody	8.751278539282415	IUPHAR.LIGAND:8086	iuphar.ligand:8086	BIMAGRUMAB	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:12084	iuphar.ligand:12084	PIFUSERTIB	FALSE	FALSE	FALSE
NCBIGENE:1839	hgnc:3059	HBEGF	GuideToPharmacology	2024.1	inhibitor	0.065145994	IUPHAR.LIGAND:4903	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
NCBIGENE:2919	hgnc:4602	CXCL1	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:10245	iuphar.ligand:10245	KT-109	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.2561349816375342	IUPHAR.LIGAND:9	iuphar.ligand:9	BMY-7378	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.3201687270469177	IUPHAR.LIGAND:506	iuphar.ligand:506	L-765314	FALSE	FALSE	FALSE
NCBIGENE:23	hgnc:70	ABCF1	GuideToPharmacology	2024.1	inhibitor	0.1829535583125243	IUPHAR.LIGAND:499	iuphar.ligand:499	WB 4101	FALSE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.079557078	IUPHAR.LIGAND:5385	rxcui:8629	PRAZOSIN	TRUE	FALSE	FALSE
NCBIGENE:24	hgnc:34	ABCA4	GuideToPharmacology	2024.1	inhibitor	0.2386712328895204	IUPHAR.LIGAND:9	iuphar.ligand:9	BMY-7378	FALSE	FALSE	FALSE
NCBIGENE:25	hgnc:76	ABL1	GuideToPharmacology	2024.1	agonist	0.075550606	IUPHAR.LIGAND:5443	rxcui:5033	GUANABENZ	TRUE	FALSE	FALSE
NCBIGENE:26	hgnc:80	AOC1	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:12577	iuphar.ligand:12577	MK-912	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.067317527	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	agonist	0.050488145	IUPHAR.LIGAND:124	rxcui:106101	OXYMETAZOLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:27	hgnc:77	ABL2	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:2741	iuphar.ligand:2741	ALL-TRANS-4-OXO-RETINOIC ACID	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	0.6035364509849942	IUPHAR.LIGAND:6949	rxcui:31494	NANDROLONE DECANOATE	TRUE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	agonist	1.810609352954982	IUPHAR.LIGAND:3455	drugbank:DB02901	STANOLONE	FALSE	FALSE	FALSE
NCBIGENE:1613	hgnc:2676	DAPK3	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:6344	rxcui:1546377	RAMIPRILAT	TRUE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.05486695	IUPHAR.LIGAND:5615	iuphar.ligand:5615	CVT-6883	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:5610	iuphar.ligand:5610	MSX-2	FALSE	FALSE	FALSE
NCBIGENE:19	hgnc:29	ABCA1	GuideToPharmacology	2024.1	agonist	0.045898314	IUPHAR.LIGAND:372	iuphar.ligand:372	2-CHLOROADENOSINE	FALSE	FALSE	FALSE
NCBIGENE:34	hgnc:89	ACADM	GuideToPharmacology	2024.1	inhibitor	0.5645986154375752	IUPHAR.LIGAND:3937	rxcui:69749	VALSARTAN	TRUE	FALSE	FALSE
NCBIGENE:2938	hgnc:4626	GSTA1	GuideToPharmacology	2024.1	antibody	5.250767123569449	IUPHAR.LIGAND:9589	iuphar.ligand:9589	ENOBLITUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2845	hgnc:4477	GPR22	GuideToPharmacology	2024.1	inhibitor	0.4167275494896388	IUPHAR.LIGAND:8318	rxcui:1747556	VENETOCLAX	TRUE	FALSE	TRUE
NCBIGENE:40	hgnc:99	ASIC2	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:8508	iuphar.ligand:8508	COMPOUND 9F [PMID: 24412111]	FALSE	FALSE	FALSE
NCBIGENE:2845	hgnc:4477	GPR22	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:11102	iuphar.ligand:11102	A-1331852	FALSE	FALSE	FALSE
NCBIGENE:2331	hgnc:3774	FMOD	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:9822	iuphar.ligand:9822	NB-360	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.4688184931758437	IUPHAR.LIGAND:132	iuphar.ligand:132	CYANOPINDOLOL	FALSE	FALSE	FALSE
NCBIGENE:28	hgnc:79	ABO	GuideToPharmacology	2024.1	inhibitor	0.072125922	IUPHAR.LIGAND:553	rxcui:6918	METOPROLOL	TRUE	FALSE	FALSE
NCBIGENE:30	hgnc:82	ACAA1	GuideToPharmacology	2024.1	inhibitor	1.693795846312725	IUPHAR.LIGAND:3463	iuphar.ligand:3463	L-748328	FALSE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:3405	iuphar.ligand:3405	12R-HETE	FALSE	FALSE	FALSE
NCBIGENE:267	hgnc:463	AMFR	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3351	iuphar.ligand:3351	LY255283	FALSE	FALSE	FALSE
NCBIGENE:1940	ncbigene:1940	EEGV1	GuideToPharmacology	2024.1	inhibitor	0.5357925636295356	IUPHAR.LIGAND:9285	iuphar.ligand:9285	PRN694	FALSE	FALSE	FALSE
NCBIGENE:1943	hgnc:3222	EFNA2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:11806	iuphar.ligand:11806	GSK329	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:7515	iuphar.ligand:7515	BZT-7	FALSE	FALSE	FALSE
NCBIGENE:1946	hgnc:3225	EFNA5	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8215	iuphar.ligand:8215	CCT244747	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	1.221108633388244	IUPHAR.LIGAND:9120	iuphar.ligand:9120	PELABRESIB	FALSE	FALSE	FALSE
NCBIGENE:1945	hgnc:3224	EFNA4	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:7511	iuphar.ligand:7511	(+)-JQ1	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	0.252440727	IUPHAR.LIGAND:9861	rxcui:2262435	ZANUBRUTINIB	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9262	iuphar.ligand:9262	LFM-A13	FALSE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.050007306	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:11203	iuphar.ligand:11203	COMPOUND 71 [WO2018191577A1]	FALSE	FALSE	FALSE
NCBIGENE:1948	hgnc:3227	EFNB2	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:9264	iuphar.ligand:9264	CGI560	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:649	iuphar.ligand:649	BRADYKININ	FALSE	FALSE	FALSE
NCBIGENE:42	hgnc:1030	BDKRB2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:675	iuphar.ligand:675	NPC-349	FALSE	FALSE	FALSE
NCBIGENE:2471	hgnc:3881	FRA20A	GuideToPharmacology	2024.1	inhibitor	1.500219178162699	IUPHAR.LIGAND:6602	rxcui:183379	RIVASTIGMINE	TRUE	FALSE	FALSE
NCBIGENE:1949	hgnc:3228	EFNB3	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9127	iuphar.ligand:9127	BAY-524	FALSE	FALSE	FALSE
UNIPROT:P55017	hgnc:10912	SLC12A3	TEND	1-Aug-11	NULL	5.834185692854944	BENDROFLUMETHIAZIDE	rxcui:1369	BENDROFLUMETHIAZIDE	TRUE	FALSE	FALSE
NCBIGENE:1957	ncbigene:1957	EGI	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:5274	iuphar.ligand:5274	STO609	FALSE	FALSE	FALSE
NCBIGENE:1997	hgnc:3316	ELF1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10357	iuphar.ligand:10357	CDK INHIBITOR 4.35	FALSE	FALSE	FALSE
UNIPROT:Q16445	hgnc:4080	GABRA6	TEND	1-Aug-11	NULL	0.053579256	PRIMIDONE	rxcui:8691	PRIMIDONE	TRUE	FALSE	FALSE
NCBIGENE:1549	hgnc:2611	CYP2A7	GuideToPharmacology	2024.1	inhibitor	1.875273972703374	IUPHAR.LIGAND:8126	ncit:C98054	SILMITASERTIB	FALSE	FALSE	FALSE
NCBIGENE:531	hgnc:1393	CACNA1F	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:2334	rxcui:7441	NITRENDIPINE	TRUE	FALSE	FALSE
NCBIGENE:534	hgnc:862	ATP6V1G2	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:4315	iuphar.ligand:4315	SNX482	FALSE	FALSE	FALSE
NCBIGENE:1581	hgnc:2651	CYP7A1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:7876	rxcui:1102129	BOCEPREVIR	TRUE	FALSE	FALSE
NCBIGENE:2350	hgnc:3793	FOLR2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:7860	iuphar.ligand:7860	L873724	FALSE	FALSE	FALSE
NCBIGENE:389	hgnc:669	RHOC	GuideToPharmacology	2024.1	activator	0.3804903712731485	IUPHAR.LIGAND:1882	rxcui:598	ALPROSTADIL	TRUE	FALSE	FALSE
NCBIGENE:77	hgnc:1571	CCKBR	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:910	iuphar.ligand:910	TETRONOTHIODIN	FALSE	FALSE	FALSE
NCBIGENE:3086	hgnc:30185	CRBN	GuideToPharmacology	2024.1	NULL	1.458546423213736	IUPHAR.LIGAND:12000	iuphar.ligand:12000	MS40	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	activator	1.193356164447602	IUPHAR.LIGAND:4152	iuphar.ligand:4152	CBIQ	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	blocker	1.193356164447602	IUPHAR.LIGAND:4202	iuphar.ligand:4202	GLYH-101	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.079798892	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:9420	ncit:C80544	ESFLURBIPROFEN	FALSE	FALSE	FALSE
NCBIGENE:1376	hgnc:2330	CPT2	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:10242	iuphar.ligand:10242	SC-236	FALSE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.073540156	IUPHAR.LIGAND:5425	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
NCBIGENE:728	hgnc:1338	C5AR1	GuideToPharmacology	2024.1	inhibitor	0.2734774543525755	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.1666910197958555	IUPHAR.LIGAND:10357	iuphar.ligand:10357	CDK INHIBITOR 4.35	FALSE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.078136416	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.3889457128569962	IUPHAR.LIGAND:5950	iuphar.ligand:5950	CDK4 INHIBITOR	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.1315981735230438	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.5048814541893701	IUPHAR.LIGAND:12277	iuphar.ligand:12277	COMPOUND 5G [PMID: 36385925]	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.3365876361262467	IUPHAR.LIGAND:10095	iuphar.ligand:10095	RO3306	FALSE	FALSE	FALSE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.036062961	IUPHAR.LIGAND:7874	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
NCBIGENE:1973	hgnc:3282	EIF4A1	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:5945	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.1041818873724097	IUPHAR.LIGAND:5945	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
NCBIGENE:1976	hgnc:1773	CDK4	GuideToPharmacology	2024.1	inhibitor	0.3704244884352345	IUPHAR.LIGAND:7383	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
NCBIGENE:1977	hgnc:3287	EIF4E	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:9095	iuphar.ligand:9095	ZOTIRACICLIB	FALSE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TEND	1-Aug-11	NULL	0.108711535	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:1978	hgnc:3288	EIF4EBP1	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:11409	iuphar.ligand:11409	CIMPUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1980	hgnc:3292	EIF4EP1	GuideToPharmacology	2024.1	inhibitor	4.039051633514961	IUPHAR.LIGAND:11842	iuphar.ligand:11842	DS96432529	FALSE	FALSE	FALSE
NCBIGENE:1979	hgnc:3289	EIF4EBP2	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:5945	iuphar.ligand:5945	CGP74514A	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:12074	iuphar.ligand:12074	ASNUCICLIB	FALSE	FALSE	FALSE
NCBIGENE:1981	hgnc:3296	EIF4G1	GuideToPharmacology	2024.1	inhibitor	0.2586584789935689	IUPHAR.LIGAND:10357	iuphar.ligand:10357	CDK INHIBITOR 4.35	FALSE	FALSE	FALSE
NCBIGENE:1318	hgnc:11017	SLC31A2	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:8748	iuphar.ligand:8748	5H3'FPE	FALSE	FALSE	FALSE
NCBIGENE:1326	hgnc:6860	MAP3K8	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:11352	ncit:C66569	SULFAPHENAZOLE	TRUE	FALSE	FALSE
UNIPROT:P21728	hgnc:3020	DRD1	TEND	1-Aug-11	NULL	0.039068208	PROPIOMAZINE	rxcui:8770	PROPIOMAZINE	TRUE	FALSE	FALSE
NCBIGENE:1320	hgnc:2597	CYP1B1	GuideToPharmacology	2024.1	inhibitor	0.5303805175322676	IUPHAR.LIGAND:8748	iuphar.ligand:8748	5H3'FPE	FALSE	FALSE	FALSE
NCBIGENE:270	hgnc:468	AMPD1	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:10580	iuphar.ligand:10580	ONO-2570366	FALSE	FALSE	FALSE
NCBIGENE:2743	hgnc:4329	GLRB	GuideToPharmacology	2024.1	antibody	5.250767123569449	IUPHAR.LIGAND:12992	iuphar.ligand:12992	NURULIMAB	FALSE	FALSE	FALSE
UNIPROT:P31645	hgnc:11050	SLC6A4	TEND	1-Aug-11	NULL	0.1325951293830669	PROTRIPTYLINE	rxcui:8886	PROTRIPTYLINE	TRUE	FALSE	FALSE
NCBIGENE:927	hgnc:1708	CD8B2	GuideToPharmacology	2024.1	inhibitor	0.16256245	IUPHAR.LIGAND:7135	rxcui:203204	BUPROPION HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.2323348284765243	IUPHAR.LIGAND:7824	iuphar.ligand:7824	AZD7268	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.4646696569530486	IUPHAR.LIGAND:1615	iuphar.ligand:1615	DELTORPHIN II	FALSE	FALSE	FALSE
NCBIGENE:317	hgnc:576	APAF1	GuideToPharmacology	2024.1	agonist	0.1548898856510162	IUPHAR.LIGAND:1617	ncit:C166495	DIPRENORPHINE	FALSE	FALSE	FALSE
NCBIGENE:2821	hgnc:4458	GPI	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7828	iuphar.ligand:7828	T863	FALSE	FALSE	FALSE
NCBIGENE:1612	hgnc:2674	DAPK1	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:9627	iuphar.ligand:9627	ZY15557	FALSE	FALSE	FALSE
UNIPROT:P35498	hgnc:10585	SCN1A	TEND	1-Aug-11	NULL	0.098451884	ZONISAMIDE	rxcui:39998	ZONISAMIDE	TRUE	FALSE	FALSE
NCBIGENE:642	hgnc:1059	BLMH	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:3205	iuphar.ligand:3205	6-FLUOROMEVALONATE 5-DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.009211872	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:216	hgnc:402	ALDH1A1	GuideToPharmacology	2024.1	inhibitor	0.023598953	IUPHAR.LIGAND:94	ncit:C152139	RACLOPRIDE	FALSE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.2853677784548614	IUPHAR.LIGAND:9215	rxcui:1373	BENPERIDOL	TRUE	FALSE	FALSE
NCBIGENE:217	hgnc:404	ALDH2	GuideToPharmacology	2024.1	inhibitor	0.076098074	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:2735	hgnc:4317	GLI1	GuideToPharmacology	2024.1	inhibitor	1.458546423213736	IUPHAR.LIGAND:7529	iuphar.ligand:7529	SGC-CBP30	FALSE	FALSE	FALSE
NCBIGENE:1567	hgnc:29499	ERAP2	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9683	iuphar.ligand:9683	COMPOUND 3V [PMID: 27390066]	FALSE	FALSE	FALSE
NCBIGENE:2834	hgnc:4464	PRLHR	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8796	iuphar.ligand:8796	COMPOUND 6EE [PMID: 22364528]	FALSE	FALSE	FALSE
NCBIGENE:2654	hgnc:3527	EZH2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8237	iuphar.ligand:8237	UNC1999	FALSE	FALSE	TRUE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:5939	iuphar.ligand:5939	BPIQ-I	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:12986	iuphar.ligand:12986	JND3229	FALSE	FALSE	FALSE
NCBIGENE:1797	hgnc:2992	DXO	GuideToPharmacology	2024.1	inhibitor	0.5000730593875666	IUPHAR.LIGAND:7641	drugbank:DB11737	ICOTINIB	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:10187	iuphar.ligand:10187	COMPOUND 3F [FESTA ET AL., 2019]	FALSE	FALSE	FALSE
NCBIGENE:603	ncbigene:603	BCL5	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:10655	ncit:C174657	NIDUFEXOR	FALSE	FALSE	FALSE
NCBIGENE:3017	hgnc:4747	H2BC5	GuideToPharmacology	2024.1	antibody	13.12691780892362	IUPHAR.LIGAND:11278	iuphar.ligand:11278	BEMARITUZUMAB	FALSE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1848861663228679	CYC116	drugbank:DB05198	CYC116	FALSE	FALSE	TRUE
NCBIGENE:2935	hgnc:4621	GSPT1	GuideToPharmacology	2024.1	agonist	26.25383561784724	IUPHAR.LIGAND:9557	iuphar.ligand:9557	IGE HEAVY CHAIN	FALSE	FALSE	FALSE
NCBIGENE:2534	hgnc:4037	FYN	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:11124	ncit:C96701	BINDARIT	FALSE	FALSE	FALSE
NCBIGENE:225	hgnc:66	ABCD2	GuideToPharmacology	2024.1	agonist	2.763561643983921	IUPHAR.LIGAND:10668	iuphar.ligand:10668	HWL-088	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.6035364509849942	IUPHAR.LIGAND:1215	iuphar.ligand:1215	(S)-CETIRIZINE	FALSE	FALSE	FALSE
NCBIGENE:1194	hgnc:10909	SLC40A1	GuideToPharmacology	2024.1	antibody	157.5230137070835	IUPHAR.LIGAND:8416	iuphar.ligand:8416	LY2928057	FALSE	FALSE	FALSE
NCBIGENE:127	hgnc:252	ADH4	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:11195	iuphar.ligand:11195	TUG-1197	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	agonist	0.3125456621172291	IUPHAR.LIGAND:6954	rxcui:196319	PALIFERMIN	TRUE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	antibody	1.250182648468916	IUPHAR.LIGAND:11278	iuphar.ligand:11278	BEMARITUZUMAB	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12313	iuphar.ligand:12313	COMPOUND 29 [PMID: 36356320]	FALSE	FALSE	FALSE
NCBIGENE:1809	hgnc:3015	DPYSL3	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:8104	iuphar.ligand:8104	LY2874455	FALSE	FALSE	FALSE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.3125456621172291	IUPHAR.LIGAND:9785	ncit:C104267	DERAZANTINIB	FALSE	FALSE	TRUE
NCBIGENE:1810	hgnc:3017	DR1	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:9788	iuphar.ligand:9788	PRN1371	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.034184682	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.054695491	IUPHAR.LIGAND:5712	iuphar.ligand:5712	SU-14813	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.4102161815288632	IUPHAR.LIGAND:10574	iuphar.ligand:10574	COMPOUND 1 [CRUZ-L&OACUTE;PEZ ET AL., 2019]	FALSE	FALSE	FALSE
NCBIGENE:1812	hgnc:3020	DRD1	GuideToPharmacology	2024.1	inhibitor	0.030386384	IUPHAR.LIGAND:6058	rxcui:2534233	TIVOZANIB	TRUE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:5982	iuphar.ligand:5982	GTP-14564	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:8784	iuphar.ligand:8784	SGI-1776	FALSE	FALSE	FALSE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	inhibitor	0.1640864726115453	IUPHAR.LIGAND:7918	ncit:C143162	ONVANSERTIB	FALSE	FALSE	TRUE
NCBIGENE:1807	hgnc:3013	DPYS	GuideToPharmacology	2024.1	NULL	0.8204323630577265	IUPHAR.LIGAND:4932	iuphar.ligand:4932	FMS-RELATED TYROSINE KINASE 3 LIGAND	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:5828	iuphar.ligand:5828	3570-0208 [PMID:19807662]	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.1930429089547591	IUPHAR.LIGAND:8983	iuphar.ligand:8983	ST-1006	FALSE	FALSE	FALSE
NCBIGENE:3212	hgnc:5113	HOXB2	GuideToPharmacology	2024.1	antibody	52.50767123569449	IUPHAR.LIGAND:12250	iuphar.ligand:12250	MIRVETUXIMAB SORAVTANSINE	FALSE	FALSE	FALSE
NCBIGENE:222	hgnc:411	ALDH3B2	GuideToPharmacology	2024.1	inhibitor	1.591141552596803	IUPHAR.LIGAND:1025	iuphar.ligand:1025	CYCLOSPORIN H	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:3934	iuphar.ligand:3934	RESOLVIN D1	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6247	iuphar.ligand:6247	F PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:6250	iuphar.ligand:6250	MHC BINDING PEPTIDE	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	2.100306849	IUPHAR.LIGAND:1955	iuphar.ligand:1955	13,14-DIHYDRO-16-M-CHLOROPHENOXY-W-TETRANOR-PGF1&ALPHA;	FALSE	FALSE	FALSE
NCBIGENE:344	hgnc:609	APOC2	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:1881	iuphar.ligand:1881	PGD2	FALSE	FALSE	FALSE
NCBIGENE:223	hgnc:412	ALDH9A1	GuideToPharmacology	2024.1	modulator	1.166837138570988	IUPHAR.LIGAND:1043	iuphar.ligand:1043	PBP10	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1243	iuphar.ligand:1243	GR 175737	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	1.628144844517658	IUPHAR.LIGAND:4221	ncit:C74385	INDIPLON	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.045226246	IUPHAR.LIGAND:4226	iuphar.ligand:4226	ISOGUVACINE	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	agonist	0.045226246	IUPHAR.LIGAND:4259	iuphar.ligand:4090	[3H]MUSCIMOL	FALSE	FALSE	FALSE
NCBIGENE:2026	hgnc:3353	ENO2	GuideToPharmacology	2024.1	inhibitor	0.083744292	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	blocker	0.017697227	IUPHAR.LIGAND:4051	drugbank:DB00466	PICROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:404	hgnc:4075	GABRA1	GuideToPharmacology	2024.1	modulator	0.037003292	IUPHAR.LIGAND:4360	rxcui:4460	FLUNITRAZEPAM	TRUE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:9180	iuphar.ligand:9180	C108297	FALSE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	inhibitor	0.3860858179095183	IUPHAR.LIGAND:12571	iuphar.ligand:12571	ST-1478	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	1.221108633388244	IUPHAR.LIGAND:11780	iuphar.ligand:11780	AZD2906	FALSE	FALSE	FALSE
NCBIGENE:625	ncbigene:625	BDM	GuideToPharmacology	2024.1	agonist	0.6105543166941221	IUPHAR.LIGAND:9731	iuphar.ligand:9731	BENZODROCORTISONE	FALSE	FALSE	FALSE
NCBIGENE:458	hgnc:4587	GRIN2C	GuideToPharmacology	2024.1	agonist	0.07699072	IUPHAR.LIGAND:6511	iuphar.ligand:4698	[3H]D-ASPARTIC ACID	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	agonist	0.074797252	IUPHAR.LIGAND:4268	iuphar.ligand:4268	NMDA	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	blocker	0.1682938180631233	IUPHAR.LIGAND:4260	iuphar.ligand:4260	N1-DANSYL-SPERMINE	FALSE	FALSE	FALSE
NCBIGENE:457	hgnc:4586	GRIN2B	GuideToPharmacology	2024.1	inhibitor	0.1682938180631233	IUPHAR.LIGAND:4168	iuphar.ligand:4168	D-AP5	FALSE	FALSE	FALSE
NCBIGENE:1747	hgnc:2916	DLX3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:4890	rxcui:19666	NESIRITIDE	TRUE	FALSE	FALSE
NCBIGENE:1720	hgnc:52354	DHFRP3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:12013	iuphar.ligand:12013	SOMATROGON	FALSE	FALSE	FALSE
NCBIGENE:55	hgnc:125	ACP3	GuideToPharmacology	2024.1	agonist	0.4375639269641208	IUPHAR.LIGAND:727	rxcui:4919	GLYCINE	TRUE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:1592	iuphar.ligand:1592	5-METHYL NICOTINIC ACID	FALSE	FALSE	FALSE
NCBIGENE:312	hgnc:536	ANXA13	GuideToPharmacology	2024.1	agonist	2.282942227638891	IUPHAR.LIGAND:5790	iuphar.ligand:5790	COMPOUND (+)17A [PMID: 20363624]	FALSE	FALSE	FALSE
NCBIGENE:400	hgnc:692	ARL1	GuideToPharmacology	2024.1	blocker	2.625383561784724	IUPHAR.LIGAND:2358	ncit:C66687	ZATEBRADINE	FALSE	FALSE	FALSE
NCBIGENE:2658	hgnc:4217	GDF2	GuideToPharmacology	2024.1	inhibitor	0.4861821410712453	IUPHAR.LIGAND:7501	iuphar.ligand:7501	RGFP109	FALSE	FALSE	FALSE
NCBIGENE:265	hgnc:461	AMELX	GuideToPharmacology	2024.1	agonist	0.3365876361262467	IUPHAR.LIGAND:8983	iuphar.ligand:8983	ST-1006	FALSE	FALSE	FALSE
NCBIGENE:2617	hgnc:4162	GARS1	GuideToPharmacology	2024.1	inhibitor	0.030796288	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.182318303	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:2659	hgnc:14063	HDAC4	GuideToPharmacology	2024.1	inhibitor	0.095122593	IUPHAR.LIGAND:8894	iuphar.ligand:8894	CUDC-101	FALSE	FALSE	FALSE
NCBIGENE:2618	hgnc:4163	GART	GuideToPharmacology	2024.1	inhibitor	0.038808331	IUPHAR.LIGAND:7489	rxcui:1603350	PANOBINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2660	hgnc:4223	MSTN	GuideToPharmacology	2024.1	inhibitor	0.039778539	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:2619	hgnc:4165	GAS1	GuideToPharmacology	2024.1	inhibitor	0.038187397	IUPHAR.LIGAND:6852	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3023	iuphar.ligand:3023	DFGYVAE	FALSE	FALSE	FALSE
NCBIGENE:2033	hgnc:3373	EP300	GuideToPharmacology	2024.1	inhibitor	0.5147810905460245	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2028	hgnc:3355	ENPEP	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:8784	iuphar.ligand:8784	SGI-1776	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3014	iuphar.ligand:3014	COMPOUND 11NN [PMID: 1656041]	FALSE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.020811602	IUPHAR.LIGAND:100	rxcui:10502	THIORIDAZINE	TRUE	FALSE	FALSE
NCBIGENE:262	hgnc:457	AMD1	GuideToPharmacology	2024.1	inhibitor	0.007941269	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:264	hgnc:5184	HRH3	GuideToPharmacology	2024.1	agonist	0.7721716358190367	IUPHAR.LIGAND:1244	ncit:C76618	CIPRALISANT	FALSE	FALSE	FALSE
NCBIGENE:263	hgnc:460	AMD1P2	GuideToPharmacology	2024.1	agonist	0.6908904109959803	IUPHAR.LIGAND:8983	iuphar.ligand:8983	ST-1006	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3007	iuphar.ligand:3007	COMPOUND 2F [PMID: 2153213]	FALSE	FALSE	FALSE
NCBIGENE:3006	hgnc:4716	H1-2	GuideToPharmacology	2024.1	activator	7.501095891	IUPHAR.LIGAND:10555	iuphar.ligand:10555	TEPP-46	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:3024	iuphar.ligand:3024	FPYVAE PEPTIDE [PMID: 20494585]	FALSE	FALSE	FALSE
NCBIGENE:600	hgnc:996	BAK1P1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:2740	iuphar.ligand:2740	ALRT 1550	FALSE	FALSE	FALSE
NCBIGENE:2874	hgnc:4550	GPS2	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8607	iuphar.ligand:8607	ALA(1-NAPH)-PRO-CN	FALSE	FALSE	FALSE
NCBIGENE:639	hgnc:9346	PRDM1	GuideToPharmacology	2024.1	inhibitor	1.500219178	IUPHAR.LIGAND:2995	iuphar.ligand:2995	COMPOUND 29 [PMID: 15686906]	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	2.386712328895204	IUPHAR.LIGAND:12245	iuphar.ligand:12245	GSK3145095	FALSE	FALSE	FALSE
NCBIGENE:1523	hgnc:2557	CUX1	GuideToPharmacology	2024.1	inhibitor	13.12691780892362	IUPHAR.LIGAND:8131	iuphar.ligand:8131	COMPOUND 24 [PMID: 15955699]	FALSE	FALSE	FALSE
NCBIGENE:351	hgnc:620	APP	GuideToPharmacology	2024.1	agonist	0.8078103267029922	IUPHAR.LIGAND:8349	iuphar.ligand:8349	A(4-24)(F23A)H2	FALSE	FALSE	FALSE
NCBIGENE:352	ncbigene:352	APPL1	GuideToPharmacology	2024.1	inhibitor	2.282942227638891	IUPHAR.LIGAND:8332	iuphar.ligand:8332	A(&DELTA;10/15C)INSL3	FALSE	FALSE	FALSE
NCBIGENE:275	hgnc:473	AMT	GuideToPharmacology	2024.1	agonist	0.750109589	IUPHAR.LIGAND:12571	iuphar.ligand:12571	ST-1478	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	inhibitor	3.088686543276147	IUPHAR.LIGAND:10310	iuphar.ligand:10310	TY-52156	FALSE	FALSE	FALSE
NCBIGENE:277	hgnc:475	AMY1B	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:3324	iuphar.ligand:3324	VPC23019	FALSE	FALSE	FALSE
NCBIGENE:126	hgnc:251	ADH1C	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:4027	iuphar.ligand:4027	AS1269574	FALSE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	0.546954909	IUPHAR.LIGAND:2020	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:2513	hgnc:24045	SPTSSB	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:11157	iuphar.ligand:11157	COMPOUND 18 [PMID: 32330443]	FALSE	FALSE	FALSE
NCBIGENE:2219	hgnc:3623	FCN1	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11811	iuphar.ligand:11811	SBP-3264	FALSE	FALSE	FALSE
NCBIGENE:2219	hgnc:3623	FCN1	GuideToPharmacology	2024.1	inhibitor	0.7721716358190368	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2214	hgnc:3619	FCGR3A	GuideToPharmacology	2024.1	inhibitor	0.2476776945079929	IUPHAR.LIGAND:10167	iuphar.ligand:10167	TOMIVOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.027135747	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:1536	hgnc:2578	CYBB	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:9423	iuphar.ligand:9423	COMPOUND 14N [PMID: 25589934]	FALSE	FALSE	FALSE
NCBIGENE:2553	hgnc:4074	GABPB1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:6685	iuphar.ligand:6684	1,3-DITOLYLGUANIDINE	FALSE	FALSE	FALSE
NCBIGENE:928	hgnc:1709	CD9	GuideToPharmacology	2024.1	inhibitor	0.037003292	IUPHAR.LIGAND:7317	rxcui:10834	TRIMIPRAMINE	TRUE	FALSE	FALSE
NCBIGENE:915	hgnc:1673	CD3D	GuideToPharmacology	2024.1	inhibitor	0.8204323630577265	IUPHAR.LIGAND:4587	iuphar.ligand:4587	SERGLIFLOZIN	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3070	iuphar.ligand:3070	J-104118	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3136	iuphar.ligand:3136	1-ALLYL-2-[3-(ISOPROPYLAMINO)PROPOXY]-9H-CARBAZOLE	FALSE	FALSE	FALSE
NCBIGENE:3048	hgnc:4832	HBG2	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12695	iuphar.ligand:12695	SLF1081851	FALSE	FALSE	FALSE
NCBIGENE:157	hgnc:290	GRK3	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:9567	iuphar.ligand:9567	TAN-67	FALSE	FALSE	FALSE
NCBIGENE:645	hgnc:1063	BLVRB	GuideToPharmacology	2024.1	inhibitor	1.875273972703375	IUPHAR.LIGAND:3105	iuphar.ligand:3105	COMPOUND 1C [BROWN ET AL., 1997]	FALSE	FALSE	FALSE
NCBIGENE:2433	hgnc:3831	FRA10C	GuideToPharmacology	2024.1	inhibitor	52.50767123569449	IUPHAR.LIGAND:8794	iuphar.ligand:8794	COMPOUND 1B [PMID: 9871762]	FALSE	FALSE	FALSE
NCBIGENE:356	hgnc:11936	FASLG	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:2053	iuphar.ligand:2053	NOC-ATE	FALSE	FALSE	FALSE
NCBIGENE:2040	hgnc:3383	STOM	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:9580	iuphar.ligand:9580	MPI-0485520	FALSE	FALSE	FALSE
NCBIGENE:358	hgnc:633	AQP1	GuideToPharmacology	2024.1	agonist	0.172722603	IUPHAR.LIGAND:2020	iuphar.ligand:2020	SRIF-28	FALSE	FALSE	FALSE
NCBIGENE:3109	hgnc:4935	HLA-DMB	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:10674	iuphar.ligand:10674	NVP‐TNKS656	FALSE	FALSE	FALSE
NCBIGENE:2238	hgnc:11719	TEC	GuideToPharmacology	2024.1	inhibitor	0.577007376	IUPHAR.LIGAND:9285	iuphar.ligand:9285	PRN694	FALSE	FALSE	FALSE
NCBIGENE:589	hgnc:11799	THRB	GuideToPharmacology	2024.1	agonist	0.5097832158805291	IUPHAR.LIGAND:12028	iuphar.ligand:12028	COMPOUND 16G [PMID: 35507418]	FALSE	FALSE	FALSE
NCBIGENE:1842	hgnc:3154	ECM2	GuideToPharmacology	2024.1	NULL	4.773424657790408	IUPHAR.LIGAND:4868	iuphar.ligand:4868	ANGIOPOIETIN-4	FALSE	FALSE	FALSE
NCBIGENE:614	hgnc:7972	NR2C2	GuideToPharmacology	2024.1	agonist	0.9723642821424907	IUPHAR.LIGAND:4053	rxcui:11246	VITAMIN A	TRUE	FALSE	FALSE
NCBIGENE:2244	hgnc:3662	FGB	GuideToPharmacology	2024.1	inhibitor	0.2059124362184098	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:485	hgnc:809	ATP1B1P1	GuideToPharmacology	2024.1	activator	0.596678082	IUPHAR.LIGAND:2419	iuphar.ligand:2419	ALLICIN	FALSE	FALSE	FALSE
NCBIGENE:486	hgnc:4026	FXYD2	GuideToPharmacology	2024.1	blocker	0.546954909	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
NCBIGENE:491	hgnc:815	ATP2B2	GuideToPharmacology	2024.1	activator	0.7721716358190367	IUPHAR.LIGAND:2764	iuphar.ligand:2764	HYPERFORIN	FALSE	FALSE	FALSE
NCBIGENE:490	hgnc:814	ATP2B1	GuideToPharmacology	2024.1	activator	0.2051080907644316	IUPHAR.LIGAND:2426	iuphar.ligand:2426	GD3+	FALSE	FALSE	FALSE
NCBIGENE:498	hgnc:823	ATP5F1A	GuideToPharmacology	2024.1	activator	0.8078103267029924	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:499	ncbigene:499	ATP5A2	GuideToPharmacology	2024.1	activator	1.346350544504987	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	activator	0.9723642821424906	IUPHAR.LIGAND:7000	iuphar.ligand:7000	CURCUMIN	FALSE	FALSE	FALSE
NCBIGENE:510	hgnc:18083	TRPV4	GuideToPharmacology	2024.1	blocker	1.944728564284981	IUPHAR.LIGAND:6465	iuphar.ligand:6465	GSK2193874	FALSE	FALSE	FALSE
NCBIGENE:2268	hgnc:3697	FGR	GuideToPharmacology	2024.1	inhibitor	0.075768645	IUPHAR.LIGAND:6912	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
NCBIGENE:2640	ncbigene:2640	GCF1	GuideToPharmacology	2024.1	inhibitor	0.081030357	IUPHAR.LIGAND:6785	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
NCBIGENE:2528	hgnc:4017	FUT6	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:11550	ncit:C152852	VENGLUSTAT	FALSE	FALSE	FALSE
NCBIGENE:371	ncbigene:371	ARCN2	GuideToPharmacology	2024.1	agonist	1.250182648468916	IUPHAR.LIGAND:2276	iuphar.ligand:2276	RO 25-1392	FALSE	FALSE	FALSE
NCBIGENE:305	hgnc:540	ANXA2P3	GuideToPharmacology	2024.1	agonist	1.009762908	IUPHAR.LIGAND:1522	iuphar.ligand:1522	[ALA31,AIB32]NPY (PIG)	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	0.7001022831425934	IUPHAR.LIGAND:1514	iuphar.ligand:1514	PEPTIDE YY	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	modulator	3.500511415712966	IUPHAR.LIGAND:12608	iuphar.ligand:12608	(S)-VU0637120	FALSE	FALSE	FALSE
NCBIGENE:307	hgnc:542	ANXA4	GuideToPharmacology	2024.1	agonist	3.500511415712966	IUPHAR.LIGAND:1511	iuphar.ligand:1511	PANCREATIC POLYPEPTIDE	FALSE	FALSE	FALSE
CCNE1	hgnc:1589	CCNE1	CIViC	10-Apr-24	NULL	0.4039051633514962	TASELISIB	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	CIViC	10-Apr-24	NULL	0.2639729920045843	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
MDM4	hgnc:6974	MDM4	CIViC	10-Apr-24	NULL	0.4167275494896388	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
FGF3	hgnc:3681	FGF3	CIViC	10-Apr-24	NULL	0.1151484018326633	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
FN1	hgnc:3778	FN1	CIViC	10-Apr-24	NULL	4.039051633514961	DAROMUN	ncit:C154627	DAROMUN	FALSE	FALSE	TRUE
NTRK3	hgnc:8033	NTRK3	CIViC	10-Apr-24	NULL	0.020696756	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
ERCC1	hgnc:3433	ERCC1	CIViC	10-Apr-24	NULL	0.3319450480417468	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	CIViC	10-Apr-24	NULL	2.407466349146467	BRIGATINIB	rxcui:1921217	BRIGATINIB	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.007544206	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
NRG1	hgnc:7997	NRG1	CIViC	10-Apr-24	NULL	0.070574827	LAPATINIB	rxcui:480167	LAPATINIB	TRUE	FALSE	TRUE
DDIT3	hgnc:2726	DDIT3	CIViC	10-Apr-24	NULL	0.2442217266776488	NVP-AEW541	iuphar.ligand:8067	NVP-AEW541	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	CIViC	10-Apr-24	NULL	0.2749092734853114	MEK INHIBITOR HL-085	ncit:C173437	TUNLAMETINIB	FALSE	FALSE	TRUE
ABL2	hgnc:77	ABL2	CIViC	10-Apr-24	NULL	0.039341412	DASATINIB	rxcui:1546019	DASATINIB ANHYDROUS	TRUE	FALSE	TRUE
EGFR	hgnc:3236	EGFR	CIViC	10-Apr-24	NULL	0.2778183663264259	FUTUXIMAB/MODOTUXIMAB MIXTURE	ncit:C91381	FUTUXIMAB/MODOTUXIMAB MIXTURE	FALSE	TRUE	TRUE
BARD1	hgnc:952	BARD1	CIViC	10-Apr-24	NULL	0.1767935058440892	APITOLISIB	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
ERCC2	hgnc:3434	ERCC2	CIViC	10-Apr-24	NULL	0.1646008502686348	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SF3B1	hgnc:10768	SF3B1	CIViC	10-Apr-24	NULL	0.2966535098061836	ETOPOSIDE	rxcui:4179	ETOPOSIDE	TRUE	FALSE	TRUE
NTRK1	hgnc:8031	NTRK1	CIViC	10-Apr-24	NULL	0.7192831676122533	TRK INHIBITOR	ncit:C155765	TRK INHIBITOR	FALSE	FALSE	TRUE
ASS1	hgnc:758	ASS1	CIViC	10-Apr-24	NULL	0.012932924	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
KDM6A	hgnc:12637	KDM6A	CIViC	10-Apr-24	NULL	0.2386712328895204	OLAPARIB	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	CIViC	10-Apr-24	NULL	0.073922431	SORAFENIB	rxcui:495881	SORAFENIB	TRUE	FALSE	TRUE
PBRM1	hgnc:30064	PBRM1	CIViC	10-Apr-24	NULL	0.3947945205691315	ATEZOLIZUMAB	rxcui:1792776	ATEZOLIZUMAB	TRUE	TRUE	TRUE
PIK3CA	hgnc:8975	PIK3CA	CIViC	10-Apr-24	NULL	0.054020238	RIBOCICLIB	rxcui:1873916	RIBOCICLIB	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.011162345	PALBOCICLIB	rxcui:1601374	PALBOCICLIB	TRUE	FALSE	TRUE
XRCC1	hgnc:12828	XRCC1	CIViC	10-Apr-24	NULL	0.051327147	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
KRAS	hgnc:6407	KRAS	CIViC	10-Apr-24	NULL	0.003772103	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
WEE1	hgnc:12761	WEE1	CIViC	10-Apr-24	NULL	0.043430663	GEMCITABINE	rxcui:12574	GEMCITABINE	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	CIViC	10-Apr-24	NULL	0.047647615	PAZOPANIB	rxcui:714438	PAZOPANIB	TRUE	FALSE	TRUE
RRM1	hgnc:10451	RRM1	CIViC	10-Apr-24	NULL	0.06390386	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
EZH2	hgnc:3527	EZH2	CIViC	10-Apr-24	NULL	2.917092846427472	UNC1999	iuphar.ligand:8237	UNC1999	FALSE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	DoCM	10-Apr-24	NULL	0.2639729920045843	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
MTOR	hgnc:3942	MTOR	DoCM	10-Apr-24	NULL	0.090821275	RAPAMYCIN	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
MET	hgnc:7029	MET	DoCM	10-Apr-24	NULL	0.384671584	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
PDGFRA	hgnc:8803	PDGFRA	DoCM	10-Apr-24	NULL	1.090323227845022	CRENOLANIB	ncit:C64639	CRENOLANIB	FALSE	FALSE	TRUE
ERBB3	hgnc:3431	ERBB3	DoCM	10-Apr-24	NULL	0.1372749574789398	PERTUZUMAB	rxcui:121191	RITUXIMAB	TRUE	TRUE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.05073205	Octreotide	rxcui:221130	OCTREOTIDE ACETATE	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.073054151	Pemetrexed Disodium	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
ALK	hgnc:427	ALK	JAX-CKB	10-Apr-24	NULL	0.016020647	Sirolimus	rxcui:35302	SIROLIMUS	TRUE	TRUE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	Spartalizumab	ncit:C121625	SPARTALIZUMAB	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1374546367426557	FCN-159	ncit:C172382	MEK 1/2 INHIBITOR FCN-159	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.009645939	Valproic acid	rxcui:11118	VALPROIC ACID	TRUE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.2749092734853114	BGB3245	ncit:C173633	BRAF INHIBITOR BGB-3245	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.4015030085991933	Futibatinib	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	JAX-CKB	10-Apr-24	NULL	0.5608295993131588	Rogaratinib	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.3947945205691315	Rogaratinib	ncit:C112205	ROGARATINIB	FALSE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.5527123287967841	S-49076	drugbank:DB16821	S-49076	FALSE	FALSE	FALSE
JAK3	hgnc:6193	JAK3	JAX-CKB	10-Apr-24	NULL	0.7134194461371536	ASP015K	ncit:C170291	PEFICITINIB	FALSE	FALSE	FALSE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.4906052389860809	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
KIT	hgnc:6342	KIT	JAX-CKB	10-Apr-24	NULL	0.1725334213659184	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
MLH1	hgnc:7127	MLH1	JAX-CKB	10-Apr-24	NULL	0.029416062	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
MSH6	hgnc:7329	MSH6	JAX-CKB	10-Apr-24	NULL	0.082732675	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.4234489615781814	BMF-219	ncit:C185864	ICOVAMENIB	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.729273212	RLY-2608	drugbank:DB16751	RLY-2608	FALSE	FALSE	FALSE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.044198376	Futibatinib	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.218327115	Temsirolimus	rxcui:657797	TEMSIROLIMUS	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1995646288518794	GSK2636771	drugbank:DB11795	GSK-2636771	FALSE	FALSE	TRUE
PMS2	hgnc:9122	PMS2	JAX-CKB	10-Apr-24	NULL	0.03394161	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.024189652	Olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.078840347	M2698	drugbank:DB15431	M-2698	FALSE	FALSE	FALSE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.1182605208011137	MEN1611	ncit:C158603	IZORLISIB	FALSE	FALSE	TRUE
VHL	hgnc:12687	VHL	JAX-CKB	10-Apr-24	NULL	0.1666910197958555	Everolimus	rxcui:141704	EVEROLIMUS	TRUE	TRUE	TRUE
GABRA1	hgnc:4075	GABRA1	ChEMBL	33	positive modulator	0.023943307	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.038131933	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.03591496	GLUTETHIMIDE	rxcui:4903	GLUTETHIMIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.081365193	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.087318744	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRG2	hgnc:4087	GABRG2	ChEMBL	33	positive modulator	0.085239726	PRAZEPAM	rxcui:8627	PRAZEPAM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.035478156	PENTOBARBITAL	rxcui:203085	PENTOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.01924768	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.021715331	PROPOFOL	rxcui:8782	PROPOFOL	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.03729238	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	positive modulator	0.038159645	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRG1	hgnc:4086	GABRG1	ChEMBL	33	positive modulator	0.042073455	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRA4	hgnc:4078	GABRA4	ChEMBL	33	positive modulator	0.040021091	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	positive modulator	0.044347695	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.017963623	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.038159645	SECOBARBITAL SODIUM	rxcui:91110	SECOBARBITAL SODIUM	TRUE	FALSE	FALSE
GABRB3	hgnc:4083	GABRB3	ChEMBL	33	positive modulator	0.017520077	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GABRA2	hgnc:4076	GABRA2	ChEMBL	33	positive modulator	0.046784382	SEVOFLURANE	rxcui:36453	SEVOFLURANE	TRUE	FALSE	FALSE
GABRB2	hgnc:4082	GABRB2	ChEMBL	33	positive modulator	0.03591496	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.036770078	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRP	hgnc:4089	GABRP	ChEMBL	33	positive modulator	0.041540879	FLURAZEPAM HYDROCHLORIDE	rxcui:71484	FLURAZEPAM HYDROCHLORIDE	TRUE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	positive modulator	0.035098711	THIOPENTAL SODIUM	rxcui:282416	THIOPENTAL SODIUM	TRUE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.087512785	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABRB1	hgnc:4081	GABRB1	ChEMBL	33	positive modulator	0.096050618	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABRA6	hgnc:4080	GABRA6	ChEMBL	33	positive modulator	0.031254566	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
GABRD	hgnc:4084	GABRD	ChEMBL	33	positive modulator	0.1022876712383659	HALAZEPAM	rxcui:26412	HALAZEPAM	TRUE	FALSE	FALSE
PPAT	hgnc:9238	PPAT	ChEMBL	33	inhibitor	0.7778914257139925	MERCAPTOPURINE	rxcui:103	MERCAPTOPURINE	TRUE	FALSE	TRUE
RPSA	hgnc:6502	RPSA	ChEMBL	33	inhibitor	0.3500511415712966	TETRACYCLINE PHOSPHATE COMPLEX	rxcui:2105975	TETRACYCLINE PHOSPHATE COMPLEX	TRUE	FALSE	FALSE
IL2RA	hgnc:6008	IL2RA	ChEMBL	33	binder	0.8579684842433742	DENILEUKIN DIFTITOX	rxcui:214470	DENILEUKIN DIFTITOX	TRUE	FALSE	TRUE
CACNA2D3	hgnc:15460	CACNA2D3	ChEMBL	33	modulator	0.2019525816757481	PREGABALIN	rxcui:187832	PREGABALIN	TRUE	FALSE	FALSE
SCN1A	hgnc:10585	SCN1A	ChEMBL	33	blocker	0.068369364	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.074163377	MORICIZINE HYDROCHLORIDE	rxcui:221126	MORICIZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN11A	hgnc:10583	SCN11A	ChEMBL	33	blocker	0.044573575	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN8A	hgnc:10596	SCN8A	ChEMBL	33	blocker	0.046840028	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.036362653	ORPHENADRINE HYDROCHLORIDE	rxcui:202723	ORPHENADRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.014883127	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.016449772	PHENYTOIN	rxcui:71227	PHENYTOIN SODIUM	TRUE	FALSE	FALSE
SCN10A	hgnc:10582	SCN10A	ChEMBL	33	blocker	0.053145416	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.048083948	FOSPHENYTOIN SODIUM	rxcui:72236	FOSPHENYTOIN	TRUE	FALSE	FALSE
SCN9A	hgnc:10597	SCN9A	ChEMBL	33	blocker	0.028413242	LAMOTRIGINE	rxcui:28439	LAMOTRIGINE	TRUE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	ChEMBL	33	inhibitor	2.414145803939977	EFALIZUMAB	rxcui:356988	EFALIZUMAB	TRUE	TRUE	FALSE
GABBR1	hgnc:4070	GABBR1	ChEMBL	33	agonist	2.187819634820604	ARBACLOFEN	ncit:C90890	ARBACLOFEN	FALSE	FALSE	FALSE
PARP3	hgnc:273	PARP3	ChEMBL	33	inhibitor	0.729273212	VELIPARIB	ncit:C60768	VELIPARIB	FALSE	FALSE	TRUE
GABBR2	hgnc:4507	GABBR2	ChEMBL	33	agonist	2.917092846427472	ARBACLOFEN	ncit:C90890	ARBACLOFEN	FALSE	FALSE	FALSE
CASP6	hgnc:1507	CASP6	ChEMBL	33	inhibitor	0.1442518440541058	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
CASP9	hgnc:1511	CASP9	ChEMBL	33	inhibitor	0.5048814541893702	EMRICASAN	ncit:C76660	EMRICASAN	FALSE	FALSE	FALSE
PSEN2	hgnc:9509	PSEN2	ChEMBL	33	modulator	0.7955707762984013	TARENFLURBIL	ncit:C26666	TARENFLURBIL	FALSE	FALSE	FALSE
SELE	hgnc:10718	SELE	ChEMBL	33	inhibitor	4.773424657790408	BIMOSIAMOSE	ncit:C72942	BIMOSIAMOSE	FALSE	FALSE	FALSE
ITGAL	hgnc:6148	ITGAL	ChEMBL	33	inhibitor	1.357957014716237	LIFITEGRAST	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.3271505995993426	DASOTRALINE	ncit:C166750	DASOTRALINE	FALSE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	ChEMBL	33	inhibitor	0.1635752997996713	LIAFENSINE	ncit:C170121	LIAFENSINE	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.6482428547616604	DASOTRALINE	ncit:C166750	DASOTRALINE	FALSE	FALSE	FALSE
SLC6A4	hgnc:11050	SLC6A4	ChEMBL	33	inhibitor	0.3977853881492006	DASOTRALINE	ncit:C166750	DASOTRALINE	FALSE	FALSE	FALSE
SLC6A3	hgnc:11049	SLC6A3	ChEMBL	33	inhibitor	0.3241214273808302	LIAFENSINE	ncit:C170121	LIAFENSINE	FALSE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	1.346350544504987	POLMACOXIB	ncit:C170335	POLMACOXIB	FALSE	FALSE	FALSE
CRBN	hgnc:30185	CRBN	ChEMBL	33	inhibitor	0.1576806944014849	THALIDOMIDE	rxcui:10432	THALIDOMIDE	TRUE	TRUE	TRUE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	positive modulator	0.064824285	GANAXOLONE	rxcui:2604689	GANAXOLONE	TRUE	FALSE	FALSE
MMP9	hgnc:7176	MMP9	ChEMBL	33	inhibitor	0.42006137	MARIMASTAT	ncit:C1652	MARIMASTAT	FALSE	FALSE	TRUE
POLD4	hgnc:14106	POLD4	ChEMBL	33	inhibitor	0.729273212	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
PDK1	hgnc:8809	PDK1	ChEMBL	33	inhibitor	1.875273972703375	SODIUM DICHLOROACETATE	rxcui:1366930	SODIUM DICHLOROACETATE	TRUE	FALSE	FALSE
PRIM2	hgnc:9370	PRIM2	ChEMBL	33	inhibitor	0.729273212	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
POLD3	hgnc:20932	POLD3	ChEMBL	33	inhibitor	0.729273212	TROXACITABINE	ncit:C1438	TROXACITABINE	FALSE	FALSE	FALSE
PDK2	hgnc:8810	PDK2	ChEMBL	33	inhibitor	3.281729452230906	SODIUM DICHLOROACETATE	rxcui:1366930	SODIUM DICHLOROACETATE	TRUE	FALSE	FALSE
ITGAV	hgnc:6150	ITGAV	ChEMBL	33	inhibitor	1.346350544504987	ABITUZUMAB	ncit:C82422	ABITUZUMAB	FALSE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	ChEMBL	33	binder	0.172722603	GANCOTAMAB	ncit:C170020	GANCOTAMAB	FALSE	FALSE	FALSE
DPP4	hgnc:3009	DPP4	ChEMBL	33	inhibitor	1.050153425	BEGELOMAB	ncit:C125608	BEGELOMAB	FALSE	FALSE	FALSE
KIR2DL2	hgnc:6330	KIR2DL2	ChEMBL	33	inhibitor	3.281729452230906	LIRILUMAB	ncit:C103820	LIRILUMAB	FALSE	FALSE	FALSE
TBXAS1	hgnc:11609	TBXAS1	ChEMBL	33	inhibitor	3.281729452230906	TERBOGREL	ncit:C96923	TERBOGREL	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	ChEMBL	33	inhibitor	0.8334550989792777	RIBOCICLIB SUCCINATE	rxcui:1873978	RIBOCICLIB SUCCINATE	TRUE	FALSE	FALSE
CDK6	hgnc:1777	CDK6	ChEMBL	33	inhibitor	2.917092846427472	RIBOCICLIB SUCCINATE	rxcui:1873978	RIBOCICLIB SUCCINATE	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	ChEMBL	33	agonist	0.105015342	BEZAFIBRATE	rxcui:1525	BEZAFIBRATE	TRUE	FALSE	FALSE
ADRA1A	hgnc:277	ADRA1A	ChEMBL	33	inhibitor	0.1367387271762877	ISOXSUPRINE HYDROCHLORIDE	rxcui:82033	ISOXSUPRINE HYDROCHLORIDE	TRUE	FALSE	FALSE
HNF4A	hgnc:5024	HNF4A	ChEMBL	33	activator	1.640864726115453	ALVERINE	rxcui:17627	ALVERINE	TRUE	FALSE	FALSE
NS3	hgnc:6407	KRAS	ChEMBL	33	inhibitor	0.182318303	VOXILAPREVIR	rxcui:1939323	VOXILAPREVIR	TRUE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	binder	3.889457128569962	MLN-2704	chembl:CHEMBL2109556	MLN-2704	FALSE	FALSE	FALSE
FOLH1	hgnc:3788	FOLH1	ChEMBL	33	binder	1.944728564284981	CYT-500 177LU	chembl:CHEMBL2109553	CYT-500 177LU	FALSE	FALSE	FALSE
CSF1R	hgnc:2433	CSF1R	ChEMBL	33	inhibitor	1.909369863116163	IMC-CS4	chembl:CHEMBL2109323	IMC-CS4	FALSE	FALSE	FALSE
KDR	hgnc:6307	KDR	ChEMBL	33	inhibitor	0.3697723326457359	IMC-1C11	ncit:C2037	IMC-1C11	FALSE	FALSE	FALSE
ITGA5	hgnc:6141	ITGA5	ChEMBL	33	inhibitor	6.563458904461812	PF-04605412	chembl:CHEMBL2109622	PF-04605412	FALSE	FALSE	TRUE
TSG101	hgnc:15971	TSG101	ChEMBL	33	inhibitor	8.078103267029922	FGI-101-1A6	chembl:CHEMBL2109593	FGI-101-1A6	FALSE	FALSE	FALSE
MUC1	hgnc:7508	MUC1	ChEMBL	33	binder	2.187819634820604	EPITUMOMAB	chembl:CHEMBL2108403	EPITUMOMAB	FALSE	FALSE	FALSE
GPA33	hgnc:4445	GPA33	ChEMBL	33	binder	26.25383561784724	HUA33	chembl:CHEMBL2109435	HUA33	FALSE	FALSE	FALSE
STEAP1	hgnc:11378	STEAP1	ChEMBL	33	binder	9.845188356692718	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
IFNA13	hgnc:5419	IFNA13	ChEMBL	33	binder	8.751278539282415	FARALIMOMAB	ncit:C188538	FARALIMOMAB	FALSE	FALSE	FALSE
MFGE8	hgnc:7036	MFGE8	ChEMBL	33	binder	26.25383561784724	BRE-3 90Y	chembl:CHEMBL2109363	BRE-3 90Y	FALSE	FALSE	FALSE
POL	hgnc:39043	ERVW-4	ChEMBL	33	inhibitor	0.4773424657790409	ELVUCITABINE	ncit:C73201	ELVUCITABINE	FALSE	FALSE	FALSE
POLD1	hgnc:9175	POLD1	ChEMBL	33	inhibitor	0.3977853881492008	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
POLD4	hgnc:14106	POLD4	ChEMBL	33	inhibitor	0.7955707762984016	ASPACYTARABINE	ncit:C153327	ASPACYTARABINE	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	inhibitor	0.5147810905460245	ZENOCUTUZUMAB	ncit:C152948	ZENOCUTUZUMAB	FALSE	FALSE	FALSE
E2F6	hgnc:3120	E2F6	ChEMBL	33	inhibitor	2.187819634820604	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
E2F2	hgnc:3114	E2F2	ChEMBL	33	inhibitor	1.312691780892362	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
MKNK2	hgnc:7111	MKNK2	ChEMBL	33	inhibitor	2.625383561784724	TOMIVOSERTIB	ncit:C125062	TOMIVOSERTIB	FALSE	FALSE	FALSE
NCBIGENE:2884	hgnc:4561	GPX1P2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:10663	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
PARC	hgnc:10616	CCL18	ChEMBL	33	inhibitor	1.810609352954982	AVAROFLOXACIN	ncit:C171788	ACORAFLOXACIN	FALSE	FALSE	FALSE
E2F8	hgnc:24727	E2F8	ChEMBL	33	inhibitor	3.281729452230906	EDIFOLIGIDE	ncit:C166786	EDIFOLIGIDE	FALSE	FALSE	FALSE
FCGRT	hgnc:3621	FCGRT	ChEMBL	33	inhibitor	1.296485709523321	EFGARTIGIMOD ALFA	rxcui:2587717	EFGARTIGIMOD ALFA	TRUE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	ChEMBL	33	binder	0.1144789343801478	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
TUBB2A	hgnc:12412	TUBB2A	ChEMBL	33	inhibitor	0.039068208	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
TUBA3C	hgnc:12408	TUBA3C	ChEMBL	33	inhibitor	0.040021091	APRUTUMAB IXADOTIN	ncit:C121212	APRUTUMAB IXADOTIN	FALSE	FALSE	FALSE
TUBB4B	hgnc:20771	TUBB4B	ChEMBL	33	inhibitor	0.039538909	ASG-5ME	chembl:CHEMBL2109574	ASG-5ME	FALSE	FALSE	FALSE
NPM1	hgnc:7910	NPM1	ChEMBL	33	inhibitor	0.2885036881082116	CRIZOTINIB	rxcui:1148495	CRIZOTINIB	TRUE	FALSE	TRUE
BCR	hgnc:1014	BCR	ChEMBL	33	inhibitor	0.2333674277141977	IMATINIB MESYLATE	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
TUBA1C	hgnc:20768	TUBA1C	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
TUBB2B	hgnc:30829	TUBB2B	ChEMBL	33	inhibitor	0.040021091	VANDORTUZUMAB VEDOTIN	ncit:C116748	VANDORTUZUMAB VEDOTIN	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	ChEMBL	33	inhibitor	0.1226814748497534	INFIGRATINIB PHOSPHATE	ncit:C175088	INFIGRATINIB PHOSPHATE	TRUE	FALSE	FALSE
ADH5	hgnc:253	ADH5	ChEMBL	33	inhibitor	7.501095891	CAVOSONSTAT	ncit:C174782	CAVOSONSTAT	FALSE	FALSE	FALSE
CA2	hgnc:1373	CA2	ChEMBL	33	inhibitor	0.3365876361262467	SULTHIAME	rxcui:10240	SULTHIAME	TRUE	FALSE	FALSE
GABRQ	hgnc:14454	GABRQ	ChEMBL	33	agonist	0.037345428	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
GABRG3	hgnc:4088	GABRG3	ChEMBL	33	agonist	0.032134438	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
GABRA3	hgnc:4077	GABRA3	ChEMBL	33	agonist	0.03070624	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
GABRA5	hgnc:4079	GABRA5	ChEMBL	33	agonist	0.03140411	PADSEVONIL	ncit:C166432	PADSEVONIL	FALSE	FALSE	FALSE
CHRM1	hgnc:1950	CHRM1	ChEMBL	33	agonist	0.032858367	XANOMELINE	ncit:C152926	XANOMELINE	FALSE	FALSE	FALSE
AGT	hgnc:333	AGT	ChEMBL	33	cleavage	2.917092846427472	GSK-2586881	chembl:CHEMBL4297887	GSK-2586881	FALSE	FALSE	FALSE
NCBIGENE:668	hgnc:1092	FOXL2	GuideToPharmacology	2024.1	agonist	2.187819634820604	IUPHAR.LIGAND:5344	iuphar.ligand:5344	(-)-&ALPHA;-THUJONE	FALSE	FALSE	FALSE
CFTR	hgnc:1884	CFTR	ChEMBL	33	positive modulator	1.193356164447602	GALICAFTOR	ncit:C170018	GALICAFTOR	FALSE	FALSE	FALSE
ERBB3	hgnc:3431	ERBB3	ChEMBL	33	binder	1.029562181092049	PATRITUMAB DERUXTECAN	ncit:C136987	PATRITUMAB DERUXTECAN	FALSE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	ChEMBL	33	inhibitor	0.2187819634820604	DS-1062	chembl:CHEMBL4297939	DS-1062	FALSE	FALSE	FALSE
CHRNB2	hgnc:1962	CHRNB2	ChEMBL	33	agonist	0.5834185692854945	VARENICLINE	rxcui:591622	VARENICLINE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	ChEMBL	33	inhibitor	0.1604757678352521	VORASIDENIB	ncit:C152914	VORASIDENIB	FALSE	FALSE	TRUE
NR1H4	hgnc:7967	NR1H4	ChEMBL	33	agonist	0.760980743	TERN-101	drugbank:DB16045	TERN-101	FALSE	FALSE	FALSE
CDC7	hgnc:1745	CDC7	ChEMBL	33	inhibitor	4.039051633514961	SIMUROSERTIB	ncit:C126641	SIMUROSERTIB	FALSE	FALSE	FALSE
ATP1A1	hgnc:799	ATP1A1	ChEMBL	33	inhibitor	0.2333674277141977	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
ATP1B2	hgnc:805	ATP1B2	ChEMBL	33	inhibitor	0.5834185692854944	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1293292394967844	IUPHAR.LIGAND:10947	iuphar.ligand:10947	NIK INHIBITOR 12F	FALSE	FALSE	FALSE
ATP1A2	hgnc:800	ATP1A2	ChEMBL	33	inhibitor	0.5000730593875666	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
GPRC5D	hgnc:13310	GPRC5D	ChEMBL	33	binder	13.12691780892362	TALQUETAMAB	rxcui:2644447	TALQUETAMAB	TRUE	FALSE	FALSE
NCBIGENE:2049	hgnc:3394	EPHB3	GuideToPharmacology	2024.1	inhibitor	0.1508841127462485	IUPHAR.LIGAND:5992	drugbank:DB04716	2-TERT-BUTYL-9-FLUORO-1,6-DIHYDROBENZO[H]IMIDAZO[4,5-F]ISOQUINOLIN-7-ONE	FALSE	FALSE	TRUE
ADH5	hgnc:253	ADH5	ChEMBL	33	inhibitor	3.750547945	N6022	chembl:CHEMBL1738699	N6022	FALSE	FALSE	FALSE
HTR4	hgnc:5299	HTR4	ChEMBL	33	agonist	0.5770073762164231	MOSAPRIDE	rxcui:135091	MOSAPRIDE	FALSE	FALSE	FALSE
GSK3A	hgnc:4616	GSK3A	DTC	9/2/20	NULL	0.020819854	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.1019566431761058	(+)-THALIPORPHINE	chembl:CHEMBL1397308	CHEMBL:CHEMBL1397308	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.2302968036653267	IUPHAR.LIGAND:1619	iuphar.ligand:1619	DYNORPHIN A-(1-13)	FALSE	FALSE	FALSE
TSHR	hgnc:12373	TSHR	DTC	9/2/20	NULL	0.5585922471882393	DECANOIC ACID	rxcui:22380	DECANOIC ACID	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004660306	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	HARMAN	chembl:CHEMBL12014	HARMAN	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.2822993077187876	INDIUM CHLORIDE	chembl:CHEMBL1447815	INDIUM CHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003915561	CHLORANIL	chembl:CHEMBL192627	CHLORANIL	FALSE	FALSE	FALSE
NCBIGENE:318	hgnc:8049	NUDT2	GuideToPharmacology	2024.1	agonist	0.0287871	IUPHAR.LIGAND:8286	rxcui:10689	TRAMADOL	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	DNDI1417529	chembl:CHEMBL1990783	CHEMBL:CHEMBL1990783	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.015925894	SOFALCONE	ncit:C81118	SOFALCONE	FALSE	FALSE	FALSE
EYA2	hgnc:3520	EYA2	DTC	9/2/20	NULL	0.022583945	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NLRP3	hgnc:16400	NLRP3	DTC	9/2/20	NULL	5.834185692854944	SJ000290236	chembl:CHEMBL602526	CHEMBL:CHEMBL602526	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.004894451	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.3302369260106572	IUPHAR.LIGAND:9691	iuphar.ligand:9691	KBP-7018	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.2117244807890907	PEUCENIN	chembl:CHEMBL1415085	PEUCENIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.023524942	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
NCBIGENE:1805	hgnc:3011	DPT	GuideToPharmacology	2024.1	inhibitor	0.1238388472539964	IUPHAR.LIGAND:10475	iuphar.ligand:10475	IBCASERTIB	FALSE	FALSE	FALSE
FEN1	hgnc:3650	FEN1	DTC	9/2/20	NULL	0.013097449	AG-494	drugbank:DB16774	TYRPHOSTIN B48	FALSE	FALSE	FALSE
F2RL1	hgnc:3538	F2RL1	DTC	9/2/20	NULL	1.193356164447602	MINOCYCLINE	rxcui:6980	MINOCYCLINE	TRUE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.034912015	2-HYDROXYPHENAZINE 5,10-DIOXIDE	chembl:CHEMBL179611	CHEMBL:CHEMBL179611	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.013622434	DOFETILIDE	rxcui:49247	DOFETILIDE	TRUE	FALSE	FALSE
RXRA	hgnc:10477	RXRA	DTC	9/2/20	NULL	0.3500511415712966	BROMETHALIN	chembl:CHEMBL1901818	BROMETHALIN	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2317	iuphar.ligand:2317	NS309	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002338872	PAROXETINE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.007003824	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.002642294	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
GFER	hgnc:4236	GFER	DTC	9/2/20	NULL	0.1166837138570989	AMSACRINE HYDROCHLORIDE	chembl:CHEMBL1256655	AMSACRINE HYDROCHLORIDE	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.5556367326528519	GRACILIN A	chembl:CHEMBL449214	GRACILIN A	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.005524797	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
NCBIGENE:386	hgnc:18866	KCNT2	GuideToPharmacology	2024.1	inhibitor	1.166837138570988	IUPHAR.LIGAND:2341	iuphar.ligand:2341	PHORBOL 12-MYRISTATE 13-ACETATE	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.063722902	PD-81723	chembl:CHEMBL59532	CHEMBL:CHEMBL59532	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.1209854175937661	NORSTICTIC ACID	chembl:CHEMBL228281	NORSTICTIC ACID	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.003224693	ARACHIDONOYL GLYCINE	iuphar.ligand:3635	N-ARACHIDONOYLGLYCINE	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.015193192	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.011762471	KAEMPFEROL	drugbank:DB01852	KAEMPHEROL	FALSE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.010687497	OXIDOPAMINE HYDROCHLORIDE	chembl:CHEMBL451197	OXIDOPAMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.003248433	ZAFIRLUKAST	rxcui:114970	ZAFIRLUKAST	TRUE	FALSE	FALSE
RGS4	hgnc:10000	RGS4	DTC	9/2/20	NULL	0.042898424	BAY-11-7085	chembl:CHEMBL270299	BAY-11-7085	FALSE	FALSE	FALSE
DRD2	hgnc:3023	DRD2	DTC	9/2/20	NULL	0.055344054	FLUPENTIXOL	rxcui:4495	FLUPENTHIXOL	FALSE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	activator	1.640864726115453	IUPHAR.LIGAND:7660	iuphar.ligand:7660	NS3623	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.014757637	IODOMELATONIN	drugbank:DB08190	N-[2-(2-IODO-5-METHOXY-1H-INDOL-3-YL)ETHYL]ACETAMIDE	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.364636606	GNF-PF-5037	chembl:CHEMBL585828	CHEMBL:CHEMBL585828	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.02617531	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.018006746	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.053579256	GNF-PF-3996	chembl:CHEMBL584458	CHEMBL:CHEMBL584458	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.1000146118775133	GNF-PF-2301	chembl:CHEMBL578061	CHEMBL:CHEMBL578061	FALSE	FALSE	FALSE
PRKCD	hgnc:9399	PRKCD	DTC	9/2/20	NULL	0.013905633	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002542252	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
NCBIGENE:572	hgnc:936	BAD	GuideToPharmacology	2024.1	blocker	0.071341945	IUPHAR.LIGAND:2326	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.002784371	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003356195	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
SLK	hgnc:11088	SLK	DTC	9/2/20	NULL	0.042689164	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.008143249	APIGENIN	rxcui:1368130	APIGENIN	TRUE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.053579256	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NTRK1	hgnc:8031	NTRK1	DTC	9/2/20	NULL	0.006660029	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
NCBIGENE:1391	hgnc:6719	LTC4S	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:9556	iuphar.ligand:9556	TK05	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.014172111	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
TTR	hgnc:12405	TTR	DTC	9/2/20	NULL	8.751278539282415	DIHYDROGUAIARETIC ACID	chembl:CHEMBL1976696	DIHYDROGUAIARETIC ACID	FALSE	FALSE	FALSE
NR1H4	hgnc:7967	NR1H4	DTC	9/2/20	NULL	0.760980743	THEONELLASTEROL C	chembl:CHEMBL1782599	THEONELLASTEROL C	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW827105X	chembl:CHEMBL186213	GW827105X	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.029366707	RESORCINOL	rxcui:35382	RESORCINOL	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.011124507	EUPAFOLIN	chembl:CHEMBL172350	EUPAFOLIN	FALSE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	DTC	9/2/20	NULL	0.5585922471882393	DNDI1418024	chembl:CHEMBL1333798	CHEMBL:CHEMBL1333798	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.129648571	N-(3,4-DICHLOROPHENYL)BENZAMIDE	chembl:CHEMBL560296	CHEMBL:CHEMBL560296	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.007292732	DNDI1417614	chembl:CHEMBL1567571	CHEMBL:CHEMBL1567571	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003174779	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.3017682254924971	GNF-PF-3314	chembl:CHEMBL582287	CHEMBL:CHEMBL582287	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.053145416	(+/-)-OCTOCLOTHEPIN MALEATE	chembl:CHEMBL1256660	CHEMBL:CHEMBL1256660	FALSE	FALSE	FALSE
SNCA	hgnc:11138	SNCA	DTC	9/2/20	NULL	0.1060761035064535	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	1,3-DIPHENYLTHIOUREA	chembl:CHEMBL275260	CHEMBL:CHEMBL275260	FALSE	FALSE	FALSE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.00701037	DACTINOMYCIN	rxcui:3100	DACTINOMYCIN	TRUE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.026045472	METHYLTHIONINIUM CHLORIDE	chembl:CHEMBL405110	METHYLTHIONINIUM CHLORIDE	FALSE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.013394814	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.002917579	METITEPINE	ncit:C166815	METITEPINE	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	EXIFONE	ncit:C81567	EXIFONE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.020187494	1,2-NAPHTHOQUINONE	rxcui:1661328	1,2-NAPHTHOQUINONE	FALSE	FALSE	FALSE
IRAK1	hgnc:6112	IRAK1	DTC	9/2/20	NULL	0.036847489	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:2054	hgnc:3403	STX2	GuideToPharmacology	2024.1	inhibitor	2.917092846427472	IUPHAR.LIGAND:8151	iuphar.ligand:8151	COMPOUND 14 [PMID: 19831390]	FALSE	FALSE	FALSE
TUBB8	hgnc:20773	TUBB8	DTC	9/2/20	NULL	0.080042182	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
TUBA1A	hgnc:20766	TUBA1A	DTC	9/2/20	NULL	0.079077818	NSC-753582	chembl:CHEMBL2036124	CHEMBL:CHEMBL2036124	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.028413242	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00731101	TYRPHOSTIN 23	chembl:CHEMBL76904	TYRPHOSTIN 23	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.019577804	CIS-2,4,3',5'-TETRAMETHOXYSTILBENE	chembl:CHEMBL221300	CHEMBL:CHEMBL221300	FALSE	FALSE	FALSE
NCBIGENE:2059	hgnc:3420	EPS8	GuideToPharmacology	2024.1	inhibitor	0.3571950424196904	IUPHAR.LIGAND:10947	iuphar.ligand:10947	NIK INHIBITOR 12F	FALSE	FALSE	FALSE
RAD54L	hgnc:9826	RAD54L	DTC	9/2/20	NULL	0.525076712	TCMDC-124395	chembl:CHEMBL534047	CHEMBL:CHEMBL534047	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.013229446	4-METHOXYDALBERGIONE	chembl:CHEMBL1554531	4-METHOXYDALBERGIONE	FALSE	FALSE	FALSE
HTT	hgnc:4851	HTT	DTC	9/2/20	NULL	0.347732922	CALYCULIN A	drugbank:DB02860	CALYCULIN A	FALSE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	DTC	9/2/20	NULL	0.016837477	IBRUTINIB	rxcui:1442981	IBRUTINIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	DTC	9/2/20	NULL	0.04907259	ENDOSULFAN	chembl:CHEMBL194399	ENDOSULFAN	FALSE	FALSE	FALSE
POLH	hgnc:9181	POLH	DTC	9/2/20	NULL	0.061055432	N-PHENETHYLCINNAMAMIDE	chembl:CHEMBL1305393	CHEMBL:CHEMBL1305393	FALSE	FALSE	FALSE
NCBIGENE:601	hgnc:997	BAK1P2	GuideToPharmacology	2024.1	agonist	1.750255707856483	IUPHAR.LIGAND:7725	iuphar.ligand:7725	AZ12260493	FALSE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.017709164	SJ000173328	chembl:CHEMBL591613	CHEMBL:CHEMBL591613	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.022136455	METIZOLINE	ncit:C99577	METIZOLINE	FALSE	FALSE	FALSE
BCR	hgnc:1014	BCR	DTC	9/2/20	NULL	0.2333674277141977	IMATINIB	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
HIF1A	hgnc:4910	HIF1A	DTC	9/2/20	NULL	0.016460085	TYRPHOSTIN A9	ncit:C2026	TYRPHOSTIN A9	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01573971	SUFENTANIL CITRATE	rxcui:58964	SUFENTANIL CITRATE	TRUE	FALSE	FALSE
RPS6KA3	hgnc:10432	RPS6KA3	DTC	9/2/20	NULL	0.027276712	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
DAPK3	hgnc:2676	DAPK3	DTC	9/2/20	NULL	0.042107194	FASUDIL	ncit:C65624	FASUDIL	FALSE	FALSE	TRUE
SENP6	hgnc:20944	SENP6	DTC	9/2/20	NULL	0.7001022831425934	XANTHOANGELOL B	chembl:CHEMBL494082	XANTHOANGELOL B	FALSE	FALSE	FALSE
NCBIGENE:273	hgnc:471	AMPH	GuideToPharmacology	2024.1	agonist	4.039051633514961	IUPHAR.LIGAND:4030	iuphar.ligand:4030	DECYL DIHYDROGEN PHOSPHATE	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00808059	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
POLK	hgnc:9183	POLK	DTC	9/2/20	NULL	0.050294704	ISOORIENTIN	chembl:CHEMBL239559	ISOORIENTIN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	CEFPIROME	rxcui:27130	CEFPIROME	TRUE	FALSE	FALSE
GLI1	hgnc:4317	GLI1	DTC	9/2/20	NULL	5.834185692854944	2,3-DIHYDROWITHAFERIN A	chembl:CHEMBL1934585	CHEMBL:CHEMBL1934585	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.024309107	NONIVAMIDE	rxcui:31945	NONIVAMIDE	TRUE	FALSE	FALSE
NCBIGENE:272	hgnc:470	AMPD3	GuideToPharmacology	2024.1	inhibitor	0.5707355569097228	IUPHAR.LIGAND:2916	iuphar.ligand:2916	DIOCTANOYLGLYCEROL PYROPHOSPHATE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.2051080907644316	NSC-123414	chembl:CHEMBL16751	CHEMBL:CHEMBL16751	FALSE	FALSE	FALSE
TEK	hgnc:11724	TEK	DTC	9/2/20	NULL	0.5966780822238011	AMPICILLIN	rxcui:221058	AMPICILLIN (ANHYDROUS)	TRUE	FALSE	FALSE
THRB	hgnc:11799	THRB	DTC	9/2/20	NULL	0.026830696	INAMRINONE	rxcui:738	INAMRINONE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.021878196	DIMERCAPROL	rxcui:3445	DIMERCAPROL	TRUE	FALSE	FALSE
ALOX5	hgnc:435	ALOX5	DTC	9/2/20	NULL	1.887530665335423	ZILEUTON	rxcui:40575	ZILEUTON	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.059063747	NORSTICTIC ACID	chembl:CHEMBL228281	NORSTICTIC ACID	FALSE	FALSE	FALSE
ALOX15	hgnc:433	ALOX15	DTC	9/2/20	NULL	0.017059022	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.012196904	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.023274677	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004674828	COLCHICINE	rxcui:2683	COLCHICINE	TRUE	FALSE	FALSE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:7036	iuphar.ligand:7036	LYS-COA	FALSE	FALSE	FALSE
IKBKB	hgnc:5960	IKBKB	DTC	9/2/20	NULL	2.500365296937833	6-METHOXYCOMAPARVIN 5-METHYL ETHER	chembl:CHEMBL256967	CHEMBL:CHEMBL256967	FALSE	FALSE	FALSE
TAOK1	hgnc:29259	TAOK1	DTC	9/2/20	NULL	0.1539814405738841	BMS-345541	iuphar.ligand:5669	BMS-345541	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.021554873	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.020510809	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
CCNA2	hgnc:1578	CCNA2	DTC	9/2/20	NULL	0.9376369863516874	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
NCBIGENE:2737	hgnc:4319	GLI3	GuideToPharmacology	2024.1	inhibitor	0.364636606	IUPHAR.LIGAND:7002	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
RAD52	hgnc:9824	RAD52	DTC	9/2/20	NULL	0.1193356164447602	SJ000114961	chembl:CHEMBL590168	CHEMBL:CHEMBL590168	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	FENPYROXYMATE	chembl:CHEMBL365100	FENPYROXYMATE	FALSE	FALSE	FALSE
TARDBP	hgnc:11571	TARDBP	DTC	9/2/20	NULL	0.1172046232939609	REV-5901	chembl:CHEMBL8747	REV-5901	FALSE	FALSE	FALSE
NPSR1	hgnc:23631	NPSR1	DTC	9/2/20	NULL	0.029766254	WIN-55212-2	iuphar.ligand:733	WIN55212-2	FALSE	FALSE	FALSE
STK17A	hgnc:11395	STK17A	DTC	9/2/20	NULL	0.3088686543276147	KD-025	rxcui:2564025	BELUMOSUDIL	TRUE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.021036727	GNF-PF-1969	chembl:CHEMBL601364	CHEMBL:CHEMBL601364	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.001331938	NORDIHYDROGUAIARETIC ACID	rxcui:227239	MASOPROCOL	TRUE	FALSE	FALSE
CSNK1A1	hgnc:2451	CSNK1A1	DTC	9/2/20	NULL	0.4688184931758437	SB-242235	chembl:CHEMBL95692	SB-242235	FALSE	FALSE	FALSE
AGTR1	hgnc:336	AGTR1	DTC	9/2/20	NULL	0.055622533	HELENALIN	chembl:CHEMBL338474	HELENALIN	FALSE	FALSE	FALSE
MET	hgnc:7029	MET	DTC	9/2/20	NULL	0.009092237	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
TAAR1	hgnc:17734	TAAR1	DTC	9/2/20	NULL	0.9053046764774912	ANTAZOLINE PHOSPHATE	rxcui:866	ANTAZOLINE PHOSPHATE	TRUE	FALSE	FALSE
KDM4E	hgnc:37098	KDM4E	DTC	9/2/20	NULL	0.090843722	TCMDC-125548	chembl:CHEMBL528045	CHEMBL:CHEMBL528045	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.007571402	TOZASERTIB	ncit:C98053	TOZASERTIB	FALSE	FALSE	TRUE
POLI	hgnc:9182	POLI	DTC	9/2/20	NULL	0.035216413	DAPHNORIN	chembl:CHEMBL1209491	DAPHNORIN	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	DTC	9/2/20	NULL	0.4487835148349957	VOACAMINE	drugbank:DB04877	VOACAMINE	FALSE	FALSE	FALSE
NR3C1	hgnc:7978	NR3C1	DTC	9/2/20	NULL	0.2004109589148645	BETAMETHASONE	rxcui:1514	BETAMETHASONE	TRUE	TRUE	FALSE
S1PR4	hgnc:3170	S1PR4	DTC	9/2/20	NULL	0.6482428547616605	TCMDC-123713	chembl:CHEMBL586135	CHEMBL:CHEMBL586135	FALSE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	DTC	9/2/20	NULL	0.4646696569530486	SUVANINE'S SODIUM SALT	chembl:CHEMBL1818099	SUVANINE'S SODIUM SALT	FALSE	FALSE	FALSE
TDP1	hgnc:18884	TDP1	DTC	9/2/20	NULL	0.4234489615781814	DEMETHYLENCECALIN	chembl:CHEMBL443462	DEMETHYLENCECALIN	FALSE	FALSE	FALSE
HPGD	hgnc:5154	HPGD	DTC	9/2/20	NULL	0.021172448	KOPARIN	chembl:CHEMBL1354502	KOPARIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009862448	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
GAA	hgnc:4065	GAA	DTC	9/2/20	NULL	0.1458546423213736	HONOKIOL	rxcui:2562546	HONOKIOL	FALSE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.023813003	GNF-PF-372	chembl:CHEMBL580155	CHEMBL:CHEMBL580155	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.054695491	CAMBENDAZOLE	rxcui:1951	CAMBENDAZOLE	FALSE	FALSE	FALSE
UBA1	hgnc:12469	UBA1	DTC	9/2/20	NULL	52.50767123569449	HIMEIC ACID A	chembl:CHEMBL2046773	HIMEIC ACID A	FALSE	FALSE	FALSE
LCK	hgnc:6524	LCK	DTC	9/2/20	NULL	0.032173818	TCMDC-125758	chembl:CHEMBL546797	CHEMBL:CHEMBL546797	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.060772768	MENTHOFURAN	chembl:CHEMBL1522900	MENTHOFURAN	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	(+)-HYDRASTINE	chembl:CHEMBL1256868	CHEMBL:CHEMBL1256868	FALSE	FALSE	FALSE
CHRM5	hgnc:1954	CHRM5	DTC	9/2/20	NULL	0.2059124362184098	PIPERTRAMINE	chembl:CHEMBL127273	PIPERTRAMINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.058733413	2,4,6-TRICHLOROPHENOL	chembl:CHEMBL309917	CHEMBL:CHEMBL309917	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.030634581	NORDEXFENFLURAMINE	iuphar.ligand:216	(+)-NORFENFLURAMINE	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.029766254	(+/-)-OCTOCLOTHEPIN MALEATE	chembl:CHEMBL1256660	CHEMBL:CHEMBL1256660	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.023620185	SAQUINAVIR MESYLATE	rxcui:859857	SAQUINAVIR MESYLATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.013957382	SR-2640	iuphar.ligand:3329	SR2640	FALSE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.008558708	LANATOSIDE C	rxcui:27929	LANATOSIDE C	TRUE	FALSE	FALSE
MAPT	hgnc:6893	MAPT	DTC	9/2/20	NULL	0.006614723	OLEOYL DOPAMINE	iuphar.ligand:5552	N-OLEOYLDOPAMINE	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	SB-409514	chembl:CHEMBL160333	CHEMBL:CHEMBL160333	FALSE	FALSE	FALSE
PTK2B	hgnc:9612	PTK2B	DTC	9/2/20	NULL	0.1037701012563132	BAS03450373	chembl:CHEMBL1576310	CHEMBL:CHEMBL1576310	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.027121731	FIPEXIDE	ncit:C65685	FIPEXIDE	TRUE	FALSE	FALSE
MGLL	hgnc:17038	MGLL	DTC	9/2/20	NULL	17.50255707856483	OCTHILINONE	chembl:CHEMBL1922512	OCTHILINONE	FALSE	FALSE	FALSE
F2	hgnc:3535	F2	DTC	9/2/20	NULL	1.381780822	CYANIN	chembl:CHEMBL2425137	CYANIN	FALSE	FALSE	FALSE
MAPK1	hgnc:6871	MAPK1	DTC	9/2/20	NULL	0.037505479	SANGUINARIUM CHLORIDE	ncit:C80864	SANGUINARIUM CHLORIDE	FALSE	FALSE	FALSE
DRD1	hgnc:3020	DRD1	DTC	9/2/20	NULL	0.012430793	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.059532507	NITRILOTRIACETIC ACID	drugbank:DB03040	NITRILOTRIACETIC ACID	FALSE	FALSE	FALSE
TRPV1	hgnc:12716	TRPV1	DTC	9/2/20	NULL	2.561349816375341	N-ARACHIDONOYLSEROTONIN	chembl:CHEMBL191534	CHEMBL:CHEMBL191534	FALSE	FALSE	FALSE
MITF	hgnc:7105	MITF	DTC	9/2/20	NULL	0.1651184630053286	DNDI1416934	chembl:CHEMBL1989750	CHEMBL:CHEMBL1989750	FALSE	FALSE	FALSE
RECQL	hgnc:9948	RECQL	DTC	9/2/20	NULL	0.015882538	AG-555	drugbank:DB16773	TYRPHOSTIN AG 555	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GLYCYROL	chembl:CHEMBL132695	GLYCYROL	FALSE	FALSE	FALSE
ABL1	hgnc:76	ABL1	DTC	9/2/20	NULL	0.8008364246019593	PONATINIB	rxcui:1364347	PONATINIB	TRUE	FALSE	TRUE
CAMK2B	hgnc:1461	CAMK2B	DTC	9/2/20	NULL	0.032817295	LINIFANIB	ncit:C71759	LINIFANIB	FALSE	FALSE	TRUE
HBB	hgnc:4827	HBB	DTC	9/2/20	NULL	0.1131630845596864	PHENAZOPYRIDINE HYDROCHLORIDE	rxcui:203197	PHENAZOPYRIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.010113188	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.051177067	DNDI1417529	chembl:CHEMBL1990783	CHEMBL:CHEMBL1990783	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	HYDROXYFLUTAMIDE	ncit:C63948	HYDROXYFLUTAMIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.014683353	NOSCAPINE	rxcui:7533	NOSCAPINE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.003262967	TYRPHOSTIN AG 879	ncit:C1491	TYRPHOSTIN AG 879	FALSE	FALSE	FALSE
MAPK12	hgnc:6874	MAPK12	DTC	9/2/20	NULL	0.7778914257139926	PH-797804	drugbank:DB07941	PH-797804	FALSE	FALSE	FALSE
POLB	hgnc:9174	POLB	DTC	9/2/20	NULL	0.020721259	METHACYCLINE HYDROCHLORIDE	rxcui:235554	METHACYCLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
CDK9	hgnc:1780	CDK9	DTC	9/2/20	NULL	0.2287915957982331	BMS-387032	iuphar.ligand:5670	BMS-387032	FALSE	FALSE	FALSE
RACGAP1	hgnc:9804	RACGAP1	DTC	9/2/20	NULL	0.750109589	LASSBIO-1183	chembl:CHEMBL1173141	CHEMBL:CHEMBL1173141	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.035358701	NSC-234945	chembl:CHEMBL260311	CHEMBL:CHEMBL260311	FALSE	FALSE	FALSE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.00505903	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	GLAUCINE METHIODIDE	chembl:CHEMBL225852	GLAUCINE METHIODIDE	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.030386384	DEXTROTHYROXINE	rxcui:3292	DEXTROTHYROXINE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.031479419	GNF-PF-1008	chembl:CHEMBL602424	CHEMBL:CHEMBL602424	FALSE	FALSE	FALSE
SMAD3	hgnc:6769	SMAD3	DTC	9/2/20	NULL	0.045858228	DNDI1416975	chembl:CHEMBL1415851	CHEMBL:CHEMBL1415851	FALSE	FALSE	FALSE
CBX1	hgnc:1551	CBX1	DTC	9/2/20	NULL	0.2792961235941196	OXOLINIC ACID	rxcui:7798	OXOLINIC ACID	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	DTC	9/2/20	NULL	0.079920352	MITOTANE	rxcui:7004	MITOTANE	TRUE	FALSE	FALSE
RAPGEF3	hgnc:16629	RAPGEF3	DTC	9/2/20	NULL	0.066297565	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.01049314	GNF-PF-3756	chembl:CHEMBL597035	CHEMBL:CHEMBL597035	FALSE	FALSE	FALSE
NPC1	hgnc:7897	NPC1	DTC	9/2/20	NULL	0.1944728564284981	3,6-DIPHENYL-[1,2,4,5]TETRAZINE	chembl:CHEMBL17784	CHEMBL:CHEMBL17784	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	1.093909817410302	BISACODYL	rxcui:1596	BISACODYL	TRUE	FALSE	FALSE
HIPK2	hgnc:14402	HIPK2	DTC	9/2/20	NULL	0.027811267	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
JUN	hgnc:6204	JUN	DTC	9/2/20	NULL	0.08780547	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.059330702	TDR77225	chembl:CHEMBL1353528	CHEMBL:CHEMBL1353528	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.00479785	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.061269161	AZEPEXOLE	ncit:C72919	AZEPEXOLE	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.00703008	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
NCBIGENE:2060	hgnc:3419	EPS15	GuideToPharmacology	2024.1	inhibitor	0.8751278539282418	IUPHAR.LIGAND:7906	ncit:C62516	BAFETINIB	FALSE	FALSE	TRUE
APOBEC3G	hgnc:17357	APOBEC3G	DTC	9/2/20	NULL	0.2263261691193728	GLAUCINE METHIODIDE	chembl:CHEMBL225852	GLAUCINE METHIODIDE	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.1093909817410302	GNF-PF-5058	chembl:CHEMBL601180	CHEMBL:CHEMBL601180	FALSE	FALSE	FALSE
AXL	hgnc:905	AXL	DTC	9/2/20	NULL	0.016086909	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
MAPK14	hgnc:6876	MAPK14	DTC	9/2/20	NULL	0.00839317	GEFITINIB	rxcui:328134	GEFITINIB	TRUE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005135225	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010235413	2-PHENYLAMINO-[1,4]NAPHTHOQUINONE	chembl:CHEMBL84010	CHEMBL:CHEMBL84010	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	PHENYLETHYL ALCOHOL	rxcui:8126	PHENYLETHYL ALCOHOL	TRUE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.010966514	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.009040577	ISOLIQUIRITIGENIN	drugbank:DB03285	ISOLIQUIRITIGENIN	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.004786261	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
PLK4	hgnc:11397	PLK4	DTC	9/2/20	NULL	0.03409589	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
NFKB2	hgnc:7795	NFKB2	DTC	9/2/20	NULL	0.9460841664089098	TAMARIXETIN	chembl:CHEMBL226034	TAMARIXETIN	FALSE	FALSE	FALSE
CYP19A1	hgnc:2594	CYP19A1	DTC	9/2/20	NULL	0.8334550989792776	LETROZOLE	rxcui:72965	LETROZOLE	TRUE	FALSE	TRUE
NCBIGENE:2105	hgnc:7111	MKNK2	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:10167	iuphar.ligand:10167	TOMIVOSERTIB	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.029235897	OXIGLUTATIONE	ncit:C62624	OXIGLUTATIONE	TRUE	FALSE	FALSE
THPO	hgnc:11795	THPO	DTC	9/2/20	NULL	0.068191781	CLEMASTINE	rxcui:2578	CLEMASTINE	TRUE	FALSE	FALSE
RELA	hgnc:9955	RELA	DTC	9/2/20	NULL	0.6604738520213144	TAMARIXETIN	chembl:CHEMBL226034	TAMARIXETIN	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.006126916	BAY-11-7082	iuphar.ligand:5934	BAY 11-7082	FALSE	FALSE	FALSE
BAZ2B	hgnc:963	BAZ2B	DTC	9/2/20	NULL	0.025588534	DNDI1417420	chembl:CHEMBL1546223	CHEMBL:CHEMBL1546223	FALSE	FALSE	FALSE
KDM4A	hgnc:22978	KDM4A	DTC	9/2/20	NULL	0.005412046	FLUPHENAZINE HYDROCHLORIDE	rxcui:203207	FLUPHENAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NFE2L2	hgnc:7782	NFE2L2	DTC	9/2/20	NULL	0.020986279	ROSIGLITAZONE MALEATE	rxcui:253198	ROSIGLITAZONE MALEATE	TRUE	FALSE	FALSE
CYP2D6	hgnc:2625	CYP2D6	DTC	9/2/20	NULL	0.04427291	VESAMICOL	iuphar.ligand:4759	VESAMICOL	FALSE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.036463661	DIPHENOXYLATE HYDROCHLORIDE	rxcui:82005	DIPHENOXYLATE HYDROCHLORIDE	TRUE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.012253832	HARMINE HYDROCHLORIDE	chembl:CHEMBL1593867	HARMINE HYDROCHLORIDE	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.011746683	DIMETHYL GAMBOGATE	chembl:CHEMBL1436860	DIMETHYL GAMBOGATE	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:1313	iuphar.ligand:1313	SNAP-7941	FALSE	FALSE	FALSE
PLK1	hgnc:9077	PLK1	DTC	9/2/20	NULL	0.097236428	NSC-135810	chembl:CHEMBL1605629	CHEMBL:CHEMBL1605629	FALSE	FALSE	FALSE
CYP2C19	hgnc:2621	CYP2C19	DTC	9/2/20	NULL	0.013560866	SILVER SULFADIAZINE	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
CASP3	hgnc:1504	CASP3	DTC	9/2/20	NULL	2.333674277141977	PHATHALIMIDE	chembl:CHEMBL261567	PHATHALIMIDE	FALSE	FALSE	FALSE
MAP4K5	hgnc:6867	MAP4K5	DTC	9/2/20	NULL	0.029833904	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.011670965	DNDI1417086	chembl:CHEMBL1224755	CHEMBL:CHEMBL1224755	FALSE	FALSE	FALSE
CDK5	hgnc:1774	CDK5	DTC	9/2/20	NULL	0.1704794520639431	AR-A014418	drugbank:DB01950	AR-AO-14418	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:7756	iuphar.ligand:7756	PYRROLIDINE MCHR1 ANTAGONIST 1	FALSE	FALSE	FALSE
IKBKE	hgnc:14552	IKBKE	DTC	9/2/20	NULL	0.05413162	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.014488872	NIGULDIPINE	ncit:C84018	NIGULDIPINE	FALSE	FALSE	FALSE
KMT2A	hgnc:7132	KMT2A	DTC	9/2/20	NULL	0.054695491	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
GPR55	hgnc:4511	GPR55	DTC	9/2/20	NULL	1.458546423213736	DNDI1417434	chembl:CHEMBL394883	CHEMBL:CHEMBL394883	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	DTC	9/2/20	NULL	0.011591097	SERTRALINE HYDROCHLORIDE	rxcui:155137	SERTRALINE HYDROCHLORIDE	TRUE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.027563082	CONGO RED	chembl:CHEMBL116955	CONGO RED	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.012466209	PD-169316	drugbank:DB17040	PD-169316	FALSE	FALSE	FALSE
NCBIGENE:280	hgnc:478	AMY2B	GuideToPharmacology	2024.1	inhibitor	1.381780822	IUPHAR.LIGAND:7754	iuphar.ligand:7754	COMPOUND (R)-10H [PMID: 22490048]	FALSE	FALSE	FALSE
BRSK1	hgnc:18994	BRSK1	DTC	9/2/20	NULL	0.028490326	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
YES1	hgnc:12841	YES1	DTC	9/2/20	NULL	0.252440727	GW695874X	chembl:CHEMBL205158	GW695874X	FALSE	FALSE	FALSE
ALDH1A1	hgnc:402	ALDH1A1	DTC	9/2/20	NULL	0.1179947668217853	DNDI1417943	chembl:CHEMBL1326758	CHEMBL:CHEMBL1326758	FALSE	FALSE	FALSE
FER	hgnc:3655	FER	DTC	9/2/20	NULL	0.038665443	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.040515178	CARBIMAZOLE	rxcui:2020	CARBIMAZOLE	TRUE	FALSE	FALSE
NCBIGENE:284	hgnc:484	ANGPT1	GuideToPharmacology	2024.1	inhibitor	0.6563458904461812	IUPHAR.LIGAND:1325	iuphar.ligand:1325	SHU9119	FALSE	FALSE	FALSE
CXCR4	hgnc:2561	CXCR4	DTC	9/2/20	NULL	4.200613699	SPERMINE TRIS-2-NAPG	chembl:CHEMBL2347633	CHEMBL:CHEMBL2347633	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.035430277	NSC-695801	chembl:CHEMBL461193	CHEMBL:CHEMBL461193	FALSE	FALSE	FALSE
TBK1	hgnc:11584	TBK1	DTC	9/2/20	NULL	0.055622533	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.002447226	PODOFILOX	rxcui:8463	PODOFILOX	TRUE	FALSE	TRUE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.028413242	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
BRD2	hgnc:1103	BRD2	DTC	9/2/20	NULL	0.1553481397505754	ACETAMINOPHEN	rxcui:161	ACETAMINOPHEN	TRUE	FALSE	FALSE
PPARG	hgnc:9236	PPARG	DTC	9/2/20	NULL	0.84012274	(-)-GRACILIOETHER B	chembl:CHEMBL2178596	CHEMBL:CHEMBL2178596	FALSE	FALSE	FALSE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:5057	iuphar.ligand:5057	SU11274	FALSE	FALSE	TRUE
FGFR1	hgnc:3688	FGFR1	DTC	9/2/20	NULL	0.004543758	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.058471794	SULFACARBAMIDE	ncit:C152453	SULFACARBAMIDE	TRUE	FALSE	FALSE
GMNN	hgnc:17493	GMNN	DTC	9/2/20	NULL	0.010939098	DNDI1417309	chembl:CHEMBL1341830	CHEMBL:CHEMBL1341830	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	DTC	9/2/20	NULL	0.005698065	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.011068227	SILVER SULFADIAZINE	rxcui:9793	SILVER SULFADIAZINE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	DTC	9/2/20	NULL	0.004961042	CARBAMAZEPINE	rxcui:2002	CARBAMAZEPINE	TRUE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	DTC	9/2/20	NULL	0.016632142	BAY-613606	iuphar.ligand:9693	BAY 61-3606	FALSE	FALSE	FALSE
HSD17B10	hgnc:4800	HSD17B10	DTC	9/2/20	NULL	0.021189536	TERAZOSIN HYDROCHLORIDE	rxcui:235224	TERAZOSIN HYDROCHLORIDE	TRUE	FALSE	FALSE
AHR	hgnc:348	AHR	DTC	9/2/20	NULL	0.1093909817410302	COLFORSIN	ncit:C166496	COLFORSIN	FALSE	FALSE	FALSE
AKR1C1	hgnc:384	AKR1C1	DTC	9/2/20	NULL	17.50255707856483	2-(4-CHLOROBENZYLIDENE)CYCLOPENTANONE	chembl:CHEMBL562352	CHEMBL:CHEMBL562352	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	inhibitor	0.1829535583125243	IUPHAR.LIGAND:1378	iuphar.ligand:1378	LY341495	FALSE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	DTC	9/2/20	NULL	0.1495945049449985	RPR-260243	iuphar.ligand:7657	RPR260243	FALSE	FALSE	FALSE
SMN1	hgnc:11117	SMN1	DTC	9/2/20	NULL	0.079557078	CID 752709	chembl:CHEMBL429335	CHEMBL:CHEMBL429335	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.004376369	CAFFEIC ACID PHENETHYL ESTER	ncit:C63756	CAFFEIC ACID PHENETHYL ESTER	FALSE	FALSE	FALSE
ATXN2	hgnc:10555	ATXN2	DTC	9/2/20	NULL	0.008503267	PAROXETINE HYDROCHLORIDE	rxcui:1298842	PAROXETINE HYDROCHLORIDE, HEMIHYDRATE	TRUE	FALSE	FALSE
CSNK1D	hgnc:2452	CSNK1D	DTC	9/2/20	NULL	0.024605282	CYC-116	chembl:CHEMBL482967	CYC-116	FALSE	FALSE	FALSE
AR	hgnc:644	AR	DTC	9/2/20	NULL	0.014617949	FLUMETHASONE	rxcui:25113	FLUMETHASONE PIVALATE	TRUE	FALSE	FALSE
IDH1	hgnc:5382	IDH1	DTC	9/2/20	NULL	0.005349192	GNF-PF-1947	chembl:CHEMBL585591	CHEMBL:CHEMBL585591	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.01531729	METIZOLINE	ncit:C99577	METIZOLINE	FALSE	FALSE	FALSE
SLC5A7	hgnc:14025	SLC5A7	DTC	9/2/20	NULL	0.1293292394967844	ERBSTATIN	chembl:CHEMBL47986	ERBSTATIN	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	agonist	0.2763561643983921	IUPHAR.LIGAND:1369	rxcui:25916	GLUTAMIC ACID	TRUE	FALSE	FALSE
UBE2N	hgnc:12492	UBE2N	DTC	9/2/20	NULL	0.080781033	PERPHENAZINE	rxcui:8076	PERPHENAZINE	TRUE	FALSE	FALSE
CLK4	hgnc:13659	CLK4	DTC	9/2/20	NULL	0.00908123	CENISERTIB	ncit:C64540	CENISERTIB	FALSE	FALSE	TRUE
CYP1A2	hgnc:2596	CYP1A2	DTC	9/2/20	NULL	0.006811217	DIAZOXIDE	rxcui:3327	DIAZOXIDE	TRUE	FALSE	FALSE
RORC	hgnc:10260	RORC	DTC	9/2/20	NULL	0.1141471113819445	POTASSIUM DICHROMATE	rxcui:8595	POTASSIUM DICHROMATE	FALSE	FALSE	FALSE
MARK3	hgnc:6897	MARK3	DTC	9/2/20	NULL	0.023151531	PF-562271	iuphar.ligand:9381	PF-562271	FALSE	FALSE	TRUE
CYP3A4	hgnc:2637	CYP3A4	DTC	9/2/20	NULL	0.009788902	MRS-1523	iuphar.ligand:474	MRS1523	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	modulator	2.763561643983921	IUPHAR.LIGAND:10237	iuphar.ligand:10237	VU0650786	FALSE	FALSE	FALSE
KAT2A	hgnc:4201	KAT2A	DTC	9/2/20	NULL	0.012920195	MITOXANTRONE DIHYDROCHLORIDE	rxcui:203129	MITOXANTRONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NTRK2	hgnc:8032	NTRK2	DTC	9/2/20	NULL	0.019889269	JNJ-7706621	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
GLS	hgnc:4331	GLS	DTC	9/2/20	NULL	0.1232574442152452	2-HYDROXYESTRADIOL	ncit:C120474	2-HYDROXYESTRADIOL	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.111481255	DALBERGIONE	chembl:CHEMBL1514569	DALBERGIONE	FALSE	FALSE	FALSE
EHMT2	hgnc:14129	EHMT2	DTC	9/2/20	NULL	0.008752737	TOLAZAMIDE	rxcui:10633	TOLAZAMIDE	TRUE	FALSE	FALSE
ATAD5	hgnc:25752	ATAD5	DTC	9/2/20	NULL	0.029665351	GNF-PF-3756	chembl:CHEMBL597035	CHEMBL:CHEMBL597035	FALSE	FALSE	FALSE
USP1	hgnc:12607	USP1	DTC	9/2/20	NULL	0.025489161	TANSHINONE I	drugbank:DB16886	TANSHINONE I	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	DTC	9/2/20	NULL	0.011148126	GUANIDINONALTRINDOLE	iuphar.ligand:1669	5'-GUANIDINONALTRINDOLE	FALSE	FALSE	FALSE
TTR	hgnc:12405	TTR	FDA	10-Apr-24	NULL	17.50255707856483	Inotersen	rxcui:2099289	INOTERSEN	TRUE	FALSE	FALSE
EGFR	hgnc:3236	EGFR	FDA	10-Apr-24	NULL	0.1805819381121768	Panitumumab	rxcui:263034	PANITUMUMAB	TRUE	TRUE	TRUE
OTC	hgnc:8512	OTC	FDA	10-Apr-24	NULL	1.750255707856483	Sodium Phenylbutyrate	rxcui:1546447	4-PHENYLBUTYRIC ACID	TRUE	FALSE	TRUE
ERBB2	hgnc:3430	ERBB2	FDA	10-Apr-24	NULL	0.025588534	Talazoparib	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
AURKA	hgnc:11393	AURKA	MyCancerGenome	20-Jun-17	inhibitor	1.779921058837101	MK5108	ncit:C90585	AURORA A KINASE INHIBITOR MK5108	FALSE	FALSE	TRUE
CDK9	hgnc:1780	CDK9	MyCancerGenome	20-Jun-17	inhibitor	0.4167275494896389	SELICICLIB	ncit:C62783	SELICICLIB	FALSE	FALSE	TRUE
CSF1R	hgnc:2433	CSF1R	MyCancerGenome	20-Jun-17	inhibitor	0.272767123	PLX3397	rxcui:2183102	PEXIDARTINIB	TRUE	FALSE	TRUE
PIK3R1	hgnc:8979	PIK3R1	MyCancerGenome	20-Jun-17	inhibitor	0.017042412	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PKN2	hgnc:9406	PKN2	MyCancerGenome	20-Jun-17	inhibitor	0.031650194	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3C2A	hgnc:8971	PIK3C2A	MyCancerGenome	20-Jun-17	inhibitor	0.039097298	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3R5	hgnc:30035	PIK3R5	MyCancerGenome	20-Jun-17	inhibitor	0.018990116	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
PIK3CD	hgnc:8977	PIK3CD	MyCancerGenome	20-Jun-17	inhibitor	0.010550065	SOPHORETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
RET	hgnc:9967	RET	MyCancerGenome	20-Jun-17	inhibitor	0.3968833804663227	SUNITINIB	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
FLT4	hgnc:3767	FLT4	MyCancerGenome	20-Jun-17	inhibitor	0.048083948	ORANTINIB	ncit:C1884	ORANTINIB	FALSE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.06375385	VANDETANIB	rxcui:1098413	VANDETANIB	TRUE	FALSE	TRUE
KDR	hgnc:6307	KDR	MyCancerGenome	20-Jun-17	inhibitor	0.1232574442152452	RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	immunotherapy	1.280674908	PIDILIZUMAB	ncit:C71014	PIDILIZUMAB	FALSE	TRUE	TRUE
PDCD1	hgnc:8760	PDCD1	MyCancerGenome	20-Jun-17	antibody	1.280674908	PIDILIZUMAB	ncit:C71014	PIDILIZUMAB	FALSE	TRUE	TRUE
NOTCH1	hgnc:7881	NOTCH1	MyCancerGenome	20-Jun-17	other/unknown	1.406455479527531	PF-03084014	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
PSENEN	hgnc:30100	PSENEN	MyCancerGenome	20-Jun-17	other/unknown	0.4375639269641209	MK0752	ncit:C49175	NOTCH SIGNALING PATHWAY INHIBITOR MK0752	FALSE	FALSE	TRUE
HSP90AA1	hgnc:5253	HSP90AA1	MyCancerGenome	20-Jun-17	other/unknown	0.4828291607879953	AUY922	drugbank:DB11881	AUY922	FALSE	FALSE	TRUE
NOTCH4	hgnc:7884	NOTCH4	MyCancerGenome	20-Jun-17	other/unknown	0.6250913242344582	PF-03084014	rxcui:2670631	NIROGACESTAT	TRUE	FALSE	TRUE
PSMA3	hgnc:9532	PSMA3	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSME2	hgnc:9569	PSME2	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD9	hgnc:9567	PSMD9	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMC5	hgnc:9552	PSMC5	MyCancerGenome	20-Jun-17	other/unknown	0.4884434533552976	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB5	hgnc:9542	PSMB5	MyCancerGenome	20-Jun-17	other/unknown	0.4273880216858854	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSME4	hgnc:20635	PSME4	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMA6	hgnc:9535	PSMA6	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB2	hgnc:9539	PSMB2	MyCancerGenome	20-Jun-17	other/unknown	0.4579157375205915	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMC3IP	hgnc:17928	PSMC3IP	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMB3	hgnc:9540	PSMB3	MyCancerGenome	20-Jun-17	other/unknown	0.4070362111294147	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
PSMD10P2	hgnc:30151	PSMD10P2	MyCancerGenome	20-Jun-17	other/unknown	0.305277158	BORTEZOMIB	rxcui:358258	BORTEZOMIB	TRUE	FALSE	TRUE
MAP2K6	hgnc:6846	MAP2K6	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.1591141552596803	AZD6244	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
TOP1	hgnc:11986	TOP1	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.8751278539282416	NKTR-102	ncit:C74069	ETIRINOTECAN PEGOL	FALSE	FALSE	TRUE
PIK3CB	hgnc:8976	PIK3CB	MyCancerGenomeClinicalTrial	30-Feburary-2014	inhibitor	0.041672755	BUPARLISIB HYDROCHLORIDE	ncit:C142973	BUPARLISIB HYDROCHLORIDE	FALSE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	NCI	14-Sep-17	NULL	0.084770219	VERAPAMIL	rxcui:11170	VERAPAMIL	TRUE	FALSE	TRUE
ABCC1	hgnc:51	ABCC1	NCI	14-Sep-17	NULL	0.1912847768149162	VM-26	rxcui:10362	TENIPOSIDE	TRUE	FALSE	TRUE
ABCC4	hgnc:55	ABCC4	NCI	14-Sep-17	NULL	0.091556532	LEUCOVORIN	rxcui:225852	LEUCOVORIN CALCIUM	TRUE	FALSE	TRUE
ABL1	hgnc:76	ABL1	NCI	14-Sep-17	NULL	0.009563368	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
ACHE	hgnc:108	ACHE	NCI	14-Sep-17	NULL	0.3088686543276147	6-AMINONICOTINAMIDE	ncit:C38127	6-AMINONICOTINAMIDE	FALSE	FALSE	FALSE
ADIPOQ	hgnc:13633	ADIPOQ	NCI	14-Sep-17	NULL	0.4953553890159858	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
ADCYAP1R1	hgnc:242	ADCYAP1R1	NCI	14-Sep-17	NULL	0.094353407	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
AFP	hgnc:317	AFP	NCI	14-Sep-17	NULL	0.100976291	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
ALOX5	hgnc:435	ALOX5	NCI	14-Sep-17	NULL	0.1065064325267636	MELATONIN	rxcui:6711	MELATONIN	TRUE	FALSE	FALSE
ANPEP	hgnc:500	ANPEP	NCI	14-Sep-17	NULL	0.020320306	HALOPERIDOL	rxcui:26420	HALOPERIDOL DECANOATE	TRUE	FALSE	FALSE
ANGPT2	hgnc:485	ANGPT2	NCI	14-Sep-17	NULL	0.2500365296937833	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
ARNT	hgnc:700	ARNT	NCI	14-Sep-17	NULL	0.056826484	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
ARF6	hgnc:659	ARF6	NCI	14-Sep-17	NULL	0.1238388472539964	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
ATF4	hgnc:786	ATF4	NCI	14-Sep-17	NULL	0.2263261691193728	VITAMIN E	rxcui:11256	VITAMIN E	TRUE	FALSE	FALSE
AQP9	hgnc:643	AQP9	NCI	14-Sep-17	NULL	0.011495932	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	0.073694977	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	0.1164249916534246	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
BAX	hgnc:959	BAX	NCI	14-Sep-17	NULL	1.400204566285186	XK469	ncit:C2662	TOPOISOMERASE-II-BETA INHIBITOR RACEMIC XK469	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	1.280674908	5-AMINOLAEVULINIC ACID	ncit:C234	AMINOLEVULINIC ACID	FALSE	FALSE	FALSE
BCL2	hgnc:990	BCL2	NCI	14-Sep-17	NULL	1.280674908	MICELLAR PACLITAXEL	ncit:C29256	MICELLAR PACLITAXEL	FALSE	FALSE	FALSE
CCL17	hgnc:10615	CCL17	NCI	14-Sep-17	NULL	1.750255707856483	POLY IC	ncit:C758	POLY IC	FALSE	FALSE	FALSE
CCL21	hgnc:10620	CCL21	NCI	14-Sep-17	NULL	6.563458904461812	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
CCL14	hgnc:10612	CCL14	NCI	14-Sep-17	NULL	4.375639269641208	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
CCL18	hgnc:10616	CCL18	NCI	14-Sep-17	NULL	0.3621218705909966	IMMUNOMODULATORS	ncit:C308	IMMUNOTHERAPEUTIC AGENT	FALSE	FALSE	FALSE
CCKBR	hgnc:1571	CCKBR	NCI	14-Sep-17	NULL	0.082300425	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
CCND1	hgnc:1582	CCND1	NCI	14-Sep-17	NULL	0.026045472	GOSSYPOL	ncit:C529	GOSSYPOL	FALSE	FALSE	FALSE
CCR2	hgnc:1603	CCR2	NCI	14-Sep-17	NULL	0.091317689	SIMVASTATIN	rxcui:36567	SIMVASTATIN	TRUE	FALSE	TRUE
CD34	hgnc:1662	CD34	NCI	14-Sep-17	NULL	10.50153424713889	BOVINE PITUITARY EXTRACT	ncit:C29784	BOVINE PITUITARY EXTRACT	FALSE	FALSE	FALSE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	0.1286952726365061	FLUDARABINE	rxcui:24698	FLUDARABINE	TRUE	FALSE	TRUE
CD40	hgnc:11919	CD40	NCI	14-Sep-17	NULL	1.093909817410302	MBL	ncit:C1151	MANNOSE-BINDING LECTIN	FALSE	FALSE	FALSE
CDH17	hgnc:1756	CDH17	NCI	14-Sep-17	NULL	0.1207072901969988	CISPLATIN	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.015858554	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.1389091831632129	17-AAG	ncit:C37899	TANESPIMYCIN	FALSE	FALSE	TRUE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	0.056826484	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
NCBIGENE:291	hgnc:10990	SLC25A4	GuideToPharmacology	2024.1	modulator	1.381780822	IUPHAR.LIGAND:6226	iuphar.ligand:6226	RO4491533	FALSE	FALSE	FALSE
CDK2	hgnc:1771	CDK2	NCI	14-Sep-17	NULL	2.045753424767318	PURINE INHIBITORS	ncit:C1556	PURINE ANTAGONIST	FALSE	FALSE	FALSE
CDKN1A	hgnc:1784	CDKN1A	NCI	14-Sep-17	NULL	1.129197231	CASPASE INHIBITOR	ncit:C38461	CASPASE INHIBITOR	FALSE	FALSE	FALSE
CDK4	hgnc:1773	CDK4	NCI	14-Sep-17	NULL	0.029074015	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
CGA	hgnc:1885	CGA	NCI	14-Sep-17	NULL	0.090530468	CIS-DIAMMINEDICHLOROPLATINUM	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	1.400204566285186	TRIVALENT INFLUENZA VACCINE	ncit:C2643	TRIVALENT INFLUENZA VACCINE	FALSE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.03043923	STREPTOZOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
CSF2	hgnc:2434	CSF2	NCI	14-Sep-17	NULL	0.1750255707856483	IMMUNOTOXIN	ncit:C575	IMMUNOTOXIN	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.4327555321623173	VEGF	ncit:C1272	RECOMBINANT VASCULAR ENDOTHELIAL GROWTH FACTOR	FALSE	FALSE	FALSE
CTGF	hgnc:2500	CCN2	NCI	14-Sep-17	NULL	0.212581665	DHT	ncit:C29618	THERAPEUTIC ANDROSTANOLONE	FALSE	FALSE	FALSE
CXCL10	hgnc:10637	CXCL10	NCI	14-Sep-17	NULL	0.3860858179095183	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
CTSG	hgnc:2532	CTSG	NCI	14-Sep-17	NULL	0.546954909	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.011294887	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A4	hgnc:2637	CYP3A4	NCI	14-Sep-17	NULL	0.003915561	FENTANYL	rxcui:142436	FENTANYL CITRATE	TRUE	FALSE	FALSE
E2F1	hgnc:3113	E2F1	NCI	14-Sep-17	NULL	0.045838211	QUERCETIN	rxcui:9060	QUERCETIN	TRUE	FALSE	TRUE
EDN1	hgnc:3176	EDN1	NCI	14-Sep-17	NULL	5.834185692854944	ANTIPLATELET AGENT	ncit:C1327	ANTIPLATELET AGENT	FALSE	FALSE	FALSE
ENO2	hgnc:3353	ENO2	NCI	14-Sep-17	NULL	0.4605936073306534	NERVE GROWTH FACTOR	rxcui:7327	NERVE GROWTH FACTOR	FALSE	FALSE	FALSE
ENOSF1	hgnc:30365	ENOSF1	NCI	14-Sep-17	NULL	0.7778914257139926	AZT	rxcui:11413	ZIDOVUDINE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.020936073	DES	rxcui:3390	DIETHYLSTILBESTROL	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	NCI	14-Sep-17	NULL	0.024674658	DEPSIPEPTIDE	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
FAS	hgnc:11920	FAS	NCI	14-Sep-17	NULL	0.3017682254924971	BISPECIFIC ANTIBODY	ncit:C1454	BISPECIFIC ANTIBODY	FALSE	FALSE	FALSE
FASN	hgnc:3594	FASN	NCI	14-Sep-17	NULL	0.2778183663264258	ANTINEOPLASTIC	ncit:C274	ANTINEOPLASTIC AGENT	FALSE	FALSE	FALSE
PTH	hgnc:9606	PTH	NCI	14-Sep-17	NULL	0.4487835148349957	SOY PROTEIN	ncit:C1803	SOY PROTEIN ISOLATE	FALSE	FALSE	FALSE
RARA	hgnc:9864	RARA	NCI	14-Sep-17	NULL	0.029074015	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
PTPRZ1	hgnc:9685	PTPRZ1	NCI	14-Sep-17	NULL	0.760980743	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
PTPN6	hgnc:9658	PTPN6	NCI	14-Sep-17	NULL	5.834185692854944	HEN EGG LYSOZYME	ncit:C1925	LYSOZYME	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.1930429089547591	GM-CSF	iuphar.ligand:4942	GM-CSF	FALSE	FALSE	FALSE
SAG	hgnc:10521	SAG	NCI	14-Sep-17	NULL	0.2035181055647073	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
NCBIGENE:2062	hgnc:6840	MAP2K1	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:12872	iuphar.ligand:12872	NEDOMETINIB	FALSE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	0.2375912725597036	CAPTOPRIL	rxcui:1998	CAPTOPRIL	TRUE	FALSE	FALSE
SERPINE1	hgnc:8583	SERPINE1	NCI	14-Sep-17	NULL	1.029562181092048	DEFIBROTIDE	rxcui:1311089	DEFIBROTIDE	TRUE	FALSE	FALSE
SHH	hgnc:10848	SHH	NCI	14-Sep-17	NULL	0.7095631248066824	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
SLC16A1	hgnc:10922	SLC16A1	NCI	14-Sep-17	NULL	0.760980743	PMA	ncit:C866	TETRADECANOYLPHORBOL ACETATE	FALSE	FALSE	FALSE
SLC2A1	hgnc:11005	SLC2A1	NCI	14-Sep-17	NULL	0.1810609352954982	DIAZEPAM	rxcui:3322	DIAZEPAM	TRUE	FALSE	FALSE
TAC1	hgnc:11517	TAC1	NCI	14-Sep-17	NULL	0.4023576339899962	8-MOP	rxcui:6854	METHOXSALEN	TRUE	FALSE	FALSE
TAGLN	hgnc:11553	TAGLN	NCI	14-Sep-17	NULL	1.312691780892362	5-AZACYTIDINE	rxcui:1251	AZACITIDINE	TRUE	FALSE	TRUE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.3387591692625452	GAMMA-INTERFERON	rxcui:1421648	GAMMA-INTERFERON	FALSE	FALSE	FALSE
TG	hgnc:11764	TG	NCI	14-Sep-17	NULL	0.130291988	AMIODARONE	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
TFPI	hgnc:11760	TFPI	NCI	14-Sep-17	NULL	0.2125816649218401	FENOFIBRATE	rxcui:221100	FENOFIBRATE MICRONIZED	TRUE	FALSE	FALSE
TFAP2A	hgnc:11742	TFAP2A	NCI	14-Sep-17	NULL	0.729273212	TNF-ALPHA	chembl:CHEMBL265582	TNF-ALPHA	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1618110053488274	ALPHA-TOCOPHEROL	ncit:C74960	ALPHA-TOCOPHEROL	FALSE	FALSE	FALSE
TGFB1	hgnc:11766	TGFB1	NCI	14-Sep-17	NULL	0.1483267549030917	HEPARAN SULFATE	rxcui:2603494	HEPARAN SULFATE	FALSE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.1682938180631233	13-CIS RETINOIC ACID	rxcui:6064	ISOTRETINOIN	TRUE	FALSE	FALSE
TGM2	hgnc:11778	TGM2	NCI	14-Sep-17	NULL	0.1583941817064691	DEFEROXAMINE	rxcui:3131	DEFEROXAMINE	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	1.129197231	PNEUMOCOCCAL POLYSACCHARIDE VACCINE	ncit:C1643	PNEUMOCOCCAL POLYVALENT VACCINE	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	1.129197231	COPTIS	ncit:C2626	HUANG LIAN	FALSE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.031958412	INSULIN	rxcui:253182	INSULIN, REGULAR, HUMAN	TRUE	FALSE	FALSE
TNF	hgnc:11892	TNF	NCI	14-Sep-17	NULL	0.03136659	CGP41251	rxcui:1919083	MIDOSTAURIN	TRUE	FALSE	TRUE
TNFRSF8	hgnc:11923	TNFRSF8	NCI	14-Sep-17	NULL	0.546954909	CHEMOKINES	ncit:C1593	RECOMBINANT CHEMOKINE	FALSE	FALSE	FALSE
TRH	hgnc:12298	TRH	NCI	14-Sep-17	NULL	4.200613698855561	6-AMINONICOTINAMIDE	ncit:C38127	6-AMINONICOTINAMIDE	FALSE	FALSE	FALSE
TSC22D3	hgnc:3051	TSC22D3	NCI	14-Sep-17	NULL	0.4167275494896388	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
TRPC1	hgnc:12333	TRPC1	NCI	14-Sep-17	NULL	2.838252499226729	CAFFEINE	rxcui:1886	CAFFEINE	TRUE	FALSE	FALSE
TYMS	hgnc:12441	TYMS	NCI	14-Sep-17	NULL	0.053199262	HYDROCORTISONE	rxcui:103468	HYDROCORTISONE BUTYRATE	TRUE	FALSE	FALSE
TSPO	hgnc:1158	TSPO	NCI	14-Sep-17	NULL	0.6908904109959803	PYRAZOLE	drugbank:DB02757	PYRAZOLE	FALSE	FALSE	FALSE
NCBIGENE:1497	hgnc:2518	CTNS	GuideToPharmacology	2024.1	inhibitor	1.193356164447602	IUPHAR.LIGAND:5273	iuphar.ligand:5273	SP600125	FALSE	FALSE	FALSE
UBR1	hgnc:16808	UBR1	NCI	14-Sep-17	NULL	1.221108633388244	DEXAMETHASONE	rxcui:3264	DEXAMETHASONE	TRUE	FALSE	TRUE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.013115442	ANDROGENS	ncit:C243	THERAPEUTIC ANDROGEN	FALSE	FALSE	FALSE
VDR	hgnc:12679	VDR	NCI	14-Sep-17	NULL	0.021234525	9-CIS RETINOIC ACID	rxcui:81864	ALITRETINOIN	TRUE	FALSE	TRUE
VHL	hgnc:12687	VHL	NCI	14-Sep-17	NULL	0.09972967	IBUPROFEN	rxcui:1429044	IBUPROFEN, SODIUM SALT	TRUE	FALSE	TRUE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.1802322811293861	STREPTOZOCIN	rxcui:10114	STREPTOZOCIN	TRUE	FALSE	FALSE
VWF	hgnc:12726	VWF	NCI	14-Sep-17	NULL	0.2125816649218401	PTK INHIBITORS	ncit:C1967	TYROSINE KINASE INHIBITOR	FALSE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	1.166837138570988	sodium nitrite	rxcui:9894	SODIUM NITRITE	TRUE	FALSE	FALSE
ERBB2	hgnc:3430	ERBB2	PharmGKB	4/5/24	NULL	0.011776541	carboplatin	rxcui:40048	CARBOPLATIN	TRUE	FALSE	TRUE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.1682938180631234	lacosamide	rxcui:623400	LACOSAMIDE	TRUE	FALSE	FALSE
ABCC2	hgnc:53	ABCC2	PharmGKB	4/5/24	NULL	0.078136416	SN-38	drugbank:DB05482	SN-38	FALSE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.1411496538593938	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
LDLR	hgnc:6547	LDLR	PharmGKB	4/5/24	NULL	0.8468979231563628	mipomersen	rxcui:1367839	MIPOMERSEN	TRUE	FALSE	FALSE
ABCC3	hgnc:54	ABCC3	PharmGKB	4/5/24	NULL	0.04573839	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
NR1I2	hgnc:7968	NR1I2	PharmGKB	4/5/24	NULL	0.016023092	lansoprazole	rxcui:17128	LANSOPRAZOLE	TRUE	FALSE	FALSE
RORA	hgnc:10258	RORA	PharmGKB	4/5/24	NULL	1.750255707856483	interferon beta-1a	rxcui:75917	INTERFERON BETA-1A	TRUE	FALSE	FALSE
USP5	hgnc:12628	USP5	PharmGKB	4/5/24	NULL	4.375639269641208	diuretics	ncit:C448	DIURETIC	FALSE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.011049594	oxymorphone	rxcui:7814	OXYMORPHONE	TRUE	FALSE	FALSE
CYP2C9	hgnc:2623	CYP2C9	PharmGKB	4/5/24	NULL	0.1215455352678113	meloxicam	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
KCNE1	hgnc:6240	KCNE1	PharmGKB	4/5/24	NULL	0.5770073762164232	amiodarone	rxcui:203114	AMIODARONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	agonist	0.1262203635473425	IUPHAR.LIGAND:301	ncit:C132273	MILAMELINE	FALSE	FALSE	FALSE
SULT1A2	hgnc:11454	SULT1A2	PharmGKB	4/5/24	NULL	7.001022831425934	4-hydroxytamoxifen	drugbank:DB04468	AFIMOXIFENE	FALSE	FALSE	FALSE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.032055965	cyanocobalamin	rxcui:11248	VITAMIN B12	TRUE	FALSE	FALSE
AKT1	hgnc:391	AKT1	PharmGKB	4/5/24	NULL	0.018962684	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.064944553	adalimumab	rxcui:2103477	ADALIMUMAB-ADBM	TRUE	FALSE	FALSE
PGR	hgnc:8910	PGR	PharmGKB	4/5/24	NULL	0.039126432	olaparib	rxcui:1597582	OLAPARIB	TRUE	FALSE	TRUE
ABCB1	hgnc:40	ABCB1	PharmGKB	4/5/24	NULL	0.023620185	abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
ESR1	hgnc:3467	ESR1	PharmGKB	4/5/24	NULL	0.038741518	abemaciclib	rxcui:1946825	ABEMACICLIB	TRUE	FALSE	TRUE
IL6	hgnc:6018	IL6	PharmGKB	4/5/24	NULL	0.082429625	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.2059124362184098	bupivacaine	rxcui:1815	BUPIVACAINE	TRUE	FALSE	FALSE
CYB5R3	hgnc:2873	CYB5R3	PharmGKB	4/5/24	NULL	0.4375639269641208	meloxicam	rxcui:41493	MELOXICAM	TRUE	FALSE	FALSE
BDNF	hgnc:1033	BDNF	PharmGKB	4/5/24	NULL	0.1422972120208522	Ergot alkaloids	rxcui:4023	ERGOT ALKALOIDS	FALSE	FALSE	FALSE
TCL1A	hgnc:11648	TCL1A	PharmGKB	4/5/24	NULL	1.117184494376478	estradiol	rxcui:24395	ESTRADIOL VALERATE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.095468493	chlorpropamide	rxcui:2404	CHLORPROPAMIDE	TRUE	FALSE	FALSE
CYP2A6	hgnc:2610	CYP2A6	PharmGKB	4/5/24	NULL	5.527123287967841	pilocarpine	rxcui:235426	PILOCARPINE HYDROCHLORIDE	TRUE	FALSE	FALSE
FCGR2B	hgnc:3618	FCGR2B	PharmGKB	4/5/24	NULL	0.2524407270946851	etanercept	rxcui:2103480	ETANERCEPT-SZZS	TRUE	TRUE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.525076712	sodium nitrate	rxcui:36700	SODIUM NITRATE	TRUE	FALSE	FALSE
GSTM1	hgnc:4632	GSTM1	PharmGKB	4/5/24	NULL	0.083522277	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.095468493	carmustine	rxcui:2105	CARMUSTINE	TRUE	FALSE	TRUE
STAT3	hgnc:11364	STAT3	PharmGKB	4/5/24	NULL	0.2333674277141977	osimertinib	rxcui:1721560	OSIMERTINIB	TRUE	FALSE	TRUE
CYP3A	ncbigene:1574	CYP3A	PharmGKB	4/5/24	NULL	0.049256727	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
PAPLN	hgnc:19262	PAPLN	PharmGKB	4/5/24	NULL	3.000438356	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
BRCA1	hgnc:1100	BRCA1	PharmGKB	4/5/24	NULL	0.062065805	sacituzumab govitecan	rxcui:2360232	SACITUZUMAB GOVITECAN	TRUE	FALSE	FALSE
VEGFA	hgnc:12680	VEGFA	PharmGKB	4/5/24	NULL	1.413668071730236	aflibercept	rxcui:1232150	AFLIBERCEPT	TRUE	TRUE	TRUE
MIR1912	hgnc:35396	MIR1912	PharmGKB	4/5/24	NULL	0.3918482928036902	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
SLC6A2	hgnc:11048	SLC6A2	PharmGKB	4/5/24	NULL	0.075496292	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYB5R1	hgnc:13397	CYB5R1	PharmGKB	4/5/24	NULL	1.050153425	isosorbide mononitrate	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
MC1R	hgnc:6929	MC1R	PharmGKB	4/5/24	NULL	0.384671584	desipramine	rxcui:3247	DESIPRAMINE	TRUE	FALSE	FALSE
CYB5R2	hgnc:24376	CYB5R2	PharmGKB	4/5/24	NULL	1.050153425	isosorbide mononitrate	rxcui:28004	ISOSORBIDE MONONITRATE	TRUE	FALSE	FALSE
CHAT	hgnc:1912	CHAT	PharmGKB	4/5/24	NULL	0.2536602475154323	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
KCNH2	hgnc:6251	KCNH2	PharmGKB	4/5/24	NULL	0.013199515	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
FMO1	hgnc:3769	FMO1	PharmGKB	4/5/24	NULL	0.760980743	nicotine	rxcui:31765	NICOTINE POLACRILEX	TRUE	FALSE	FALSE
CXCL8	hgnc:6025	CXCL8	PharmGKB	4/5/24	NULL	0.015810801	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
CYP1B1	hgnc:2597	CYP1B1	PharmGKB	4/5/24	NULL	0.047496763	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
SLC4A1	hgnc:11027	SLC4A1	PharmGKB	4/5/24	NULL	1.458546423213736	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
SLC1A1	hgnc:10939	SLC1A1	PharmGKB	4/5/24	NULL	0.1119566550867686	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
MSANTD1	hgnc:33741	MSANTD1	PharmGKB	4/5/24	NULL	1.567393171214761	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
UGT1A8	hgnc:12540	UGT1A8	PharmGKB	4/5/24	NULL	0.104492878	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
HTT	hgnc:4851	HTT	PharmGKB	4/5/24	NULL	0.010380087	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
TJP1	hgnc:11827	TJP1	PharmGKB	4/5/24	NULL	0.3918482928036902	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
PPA2	hgnc:28883	PPA2	PharmGKB	4/5/24	NULL	1.567393171214761	risperidone	rxcui:35636	RISPERIDONE	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.027840759	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
FCGR3A	hgnc:3619	FCGR3A	PharmGKB	4/5/24	NULL	0.024163678	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
DOK5	hgnc:16173	DOK5	PharmGKB	4/5/24	NULL	0.128067491	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
CYP4X1	hgnc:20244	CYP4X1	PharmGKB	4/5/24	NULL	0.6403374540938354	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
CBR3	hgnc:1549	CBR3	PharmGKB	4/5/24	NULL	0.1422972120208523	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
PIK3R2	hgnc:8980	PIK3R2	PharmGKB	4/5/24	NULL	0.032837818	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
FGFR4	hgnc:3691	FGFR4	PharmGKB	4/5/24	NULL	0.027248402	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
FCGR2A	hgnc:3616	FCGR2A	PharmGKB	4/5/24	NULL	0.2134458180312784	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
ATM	hgnc:795	ATM	PharmGKB	4/5/24	NULL	0.017543492	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
IKZF3	hgnc:13178	IKZF3	PharmGKB	4/5/24	NULL	1.280674908	cyclophosphamide	rxcui:1545988	CYCLOPHOSPHAMIDE ANHYDROUS	TRUE	FALSE	FALSE
RRM2	hgnc:10452	RRM2	PharmGKB	4/5/24	NULL	0.09972967	cytarabine	rxcui:3041	CYTARABINE	TRUE	FALSE	TRUE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.029698909	IUPHAR.LIGAND:320	rxcui:1223	ATROPINE	TRUE	FALSE	FALSE
CYP2C8	hgnc:2622	CYP2C8	PharmGKB	4/5/24	NULL	0.4475085616678508	mycophenolate mofetil	rxcui:68149	MYCOPHENOLATE MOFETIL	TRUE	TRUE	FALSE
SEMA6A	hgnc:10738	SEMA6A	PharmGKB	4/5/24	NULL	0.7242437411819931	cisplatin	rxcui:2555	CISPLATIN	TRUE	FALSE	TRUE
SLC22A2	hgnc:10966	SLC22A2	PharmGKB	4/5/24	NULL	1.875273972703374	trimethoprim	rxcui:10180	SULFAMETHOXAZOLE	TRUE	FALSE	FALSE
CYP1A2	hgnc:2596	CYP1A2	PharmGKB	4/5/24	NULL	0.013281873	imipramine	rxcui:150816	IMIPRAMINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UGT1A7	hgnc:12539	UGT1A7	PharmGKB	4/5/24	NULL	0.280789686	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
OR2B11	hgnc:31249	OR2B11	PharmGKB	4/5/24	NULL	4.773424657790409	axitinib	rxcui:1242999	AXITINIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.105015342	nicorandil	rxcui:31748	NICORANDIL	FALSE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.7876150685354175	tafenoquine	rxcui:2054023	TAFENOQUINE	TRUE	FALSE	FALSE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.058341857	dabrafenib	rxcui:1424911	DABRAFENIB	TRUE	FALSE	TRUE
G6PD	hgnc:4057	G6PD	PharmGKB	4/5/24	NULL	0.525076712	sulfacetamide	rxcui:10169	SULFACETAMIDE	TRUE	FALSE	FALSE
PROX1	hgnc:9459	PROX1	PharmGKB	4/5/24	NULL	2.917092846427472	atenolol	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
H2AFX	hgnc:4739	H2AX	PharmGKB	4/5/24	NULL	0.4412409347537353	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
IKBKG	hgnc:5961	IKBKG	PharmGKB	4/5/24	NULL	4.375639269641208	artesunate	rxcui:18346	ARTESUNATE	TRUE	FALSE	FALSE
RFK	hgnc:30324	RFK	PharmGKB	4/5/24	NULL	3.000438356	citalopram	rxcui:2556	CITALOPRAM	TRUE	FALSE	FALSE
UGT2B7	hgnc:12554	UGT2B7	PharmGKB	4/5/24	NULL	0.3231241306811969	lorazepam	rxcui:6470	LORAZEPAM	TRUE	FALSE	FALSE
SLCO1B1	hgnc:10959	SLCO1B1	PharmGKB	4/5/24	NULL	0.034590034	mitoxantrone	rxcui:7005	MITOXANTRONE	TRUE	FALSE	TRUE
RHBDF2	hgnc:20788	RHBDF2	PharmGKB	4/5/24	NULL	4.039051633514961	oxycodone	rxcui:7804	OXYCODONE	TRUE	FALSE	FALSE
KCNJ6	hgnc:6267	KCNJ6	PharmGKB	4/5/24	NULL	0.7721716358190368	methadone	rxcui:218337	METHADONE HYDROCHLORIDE	TRUE	FALSE	FALSE
CYP3A5	hgnc:2638	CYP3A5	PharmGKB	4/5/24	NULL	0.2333674277141978	salmeterol	rxcui:36117	SALMETEROL	TRUE	FALSE	FALSE
ADRA1B	hgnc:278	ADRA1B	PharmGKB	4/5/24	NULL	0.1426838892274307	phenylephrine	rxcui:8163	PHENYLEPHRINE	TRUE	FALSE	FALSE
UNIPROT:Q9NZ42	hgnc:30100	PSENEN	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	BMS-708163	ncit:C96305	AVAGACESTAT	FALSE	FALSE	FALSE
UNIPROT:P07550	hgnc:286	ADRB2	TdgClinicalTrial	Jan-14	NULL	0.2035181055647073	BUCINDOLOL	ncit:C142971	BUCINDOLOL HYDROCHLORIDE	FALSE	FALSE	FALSE
UNIPROT:P32246	hgnc:1602	CCR1	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	CCX354	iuphar.ligand:10164	CCX354	FALSE	FALSE	FALSE
UNIPROT:P17948	hgnc:3763	FLT1	TdgClinicalTrial	Jan-14	NULL	0.056826484	CEDIRANIB	ncit:C80867	CEDIRANIB	FALSE	FALSE	TRUE
UNIPROT:P35354	hgnc:9605	PTGS2	TdgClinicalTrial	Jan-14	NULL	1.432027397337122	CIMICOXIB	ncit:C77551	CIMICOXIB	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TdgClinicalTrial	Jan-14	NULL	0.057912873	DICLOFENAC	rxcui:203214	DICLOFENAC SODIUM	TRUE	FALSE	FALSE
UNIPROT:O14764	hgnc:4084	GABRD	TdgClinicalTrial	Jan-14	NULL	0.092988792	CLOBAZAM	rxcui:21241	CLOBAZAM	TRUE	FALSE	FALSE
UNIPROT:P37231	hgnc:9236	PPARG	TdgClinicalTrial	Jan-14	NULL	0.84012274	CLX-0921	drugbank:DB05854	CLX-0921	FALSE	FALSE	FALSE
UNIPROT:P12235	hgnc:10990	SLC25A4	TdgClinicalTrial	Jan-14	NULL	0.502465753	CLODRONATE	rxcui:3350	CLODRONIC ACID	TRUE	FALSE	FALSE
UNIPROT:P29275	hgnc:264	ADORA2B	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	CVT-6883	drugbank:DB05936	CVT-6883	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.084146909	IUPHAR.LIGAND:313	iuphar.ligand:313	MUSCARINIC TOXIN 3	FALSE	FALSE	FALSE
UNIPROT:O95264	hgnc:5298	HTR3B	TdgClinicalTrial	Jan-14	NULL	0.5147810905460244	DDP225	chembl:CHEMBL5095232	DDP-225	FALSE	FALSE	FALSE
UNIPROT:P30872	hgnc:11330	SSTR1	TdgClinicalTrial	Jan-14	NULL	0.6250913242344582	DG3173	ncit:C152846	VELDOREOTIDE	FALSE	FALSE	FALSE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.1666910197958555	DEXPRAMIPEXOLE	ncit:C169899	DEXPRAMIPEXOLE	FALSE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.069180068	DEXPRAMIPEXOLE	ncit:C169899	DEXPRAMIPEXOLE	FALSE	FALSE	FALSE
UNIPROT:A5X5Y0	hgnc:24005	HTR3E	TdgClinicalTrial	Jan-14	NULL	0.4375639269641208	DOLASETRON	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
UNIPROT:Q8WXA8	hgnc:24003	HTR3C	TdgClinicalTrial	Jan-14	NULL	0.4688184931758437	DOLASETRON	rxcui:68091	DOLASETRON	TRUE	FALSE	FALSE
UNIPROT:P06401	hgnc:8910	PGR	TdgClinicalTrial	Jan-14	NULL	0.6455861217503421	DROSPIRENONE	rxcui:11636	DROSPIRENONE	TRUE	FALSE	FALSE
UNIPROT:Q12882	hgnc:3012	DPYD	TdgClinicalTrial	Jan-14	NULL	1.486066167047957	ENILURACIL	ncit:C1773	ENILURACIL	FALSE	FALSE	FALSE
UNIPROT:P30968	hgnc:4421	GNRHR	TdgClinicalTrial	Jan-14	NULL	0.3977853881492007	LEUPROLIDE	rxcui:203217	LEUPROLIDE ACETATE	TRUE	FALSE	TRUE
UNIPROT:P35462	hgnc:3024	DRD3	TdgClinicalTrial	Jan-14	NULL	0.069454592	LEVODOPA	rxcui:6375	LEVODOPA	TRUE	FALSE	FALSE
UNIPROT:P48048	hgnc:6255	KCNJ1	TdgClinicalTrial	Jan-14	NULL	1.093909817410302	GLIMEPIRIDE	rxcui:25789	GLIMEPIRIDE	TRUE	FALSE	FALSE
UNIPROT:P01116	hgnc:6407	KRAS	TdgClinicalTrial	Jan-14	NULL	0.2734774543525755	GI-4000	drugbank:DB05698	GI-4000	FALSE	FALSE	FALSE
UNIPROT:P11388	hgnc:11989	TOP2A	TdgClinicalTrial	Jan-14	NULL	0.4526523382387456	GPX-100	ncit:C2494	13-DEOXYDOXORUBICIN	FALSE	FALSE	FALSE
UNIPROT:Q9Y478	hgnc:9378	PRKAB1	TdgClinicalTrial	Jan-14	NULL	1.009762908	METFORMIN	rxcui:6809	METFORMIN	TRUE	FALSE	TRUE
UNIPROT:P07098	hgnc:6622	LIPF	TdgClinicalTrial	Jan-14	NULL	5.834185692854944	GT 389-255	drugbank:DB05894	GT 389-255	FALSE	FALSE	FALSE
UNIPROT:P09619	hgnc:8804	PDGFRB	TdgClinicalTrial	Jan-14	NULL	0.8751278539282416	PDGF-BB	rxcui:115238	BECAPLERMIN	TRUE	FALSE	FALSE
UNIPROT:P04049	hgnc:9829	RAF1	TdgClinicalTrial	Jan-14	NULL	2.019525817	ICO-007	drugbank:DB05268	ICO-007	FALSE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TdgClinicalTrial	Jan-14	NULL	0.020164236	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P08908	hgnc:5286	HTR1A	TdgClinicalTrial	Jan-14	NULL	0.03378872	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P50406	hgnc:5301	HTR6	TdgClinicalTrial	Jan-14	NULL	0.1666910197958555	ILOPERIDONE	rxcui:73178	ILOPERIDONE	TRUE	FALSE	FALSE
UNIPROT:P04626	hgnc:3430	ERBB2	TdgClinicalTrial	Jan-14	NULL	0.3454452054979901	INSM-18	chembl:CHEMBL3545025	INSM-18	FALSE	FALSE	FALSE
UNIPROT:P12931	hgnc:11283	SRC	TdgClinicalTrial	Jan-14	NULL	0.7778914257139926	KX2-391	rxcui:2471078	TIRBANIBULIN	TRUE	FALSE	TRUE
UNIPROT:P35372	hgnc:8156	OPRM1	TdgClinicalTrial	Jan-14	NULL	0.1070492787679806	BUTORPHANOL	rxcui:1841	BUTORPHANOL	TRUE	FALSE	FALSE
UNIPROT:Q13621	hgnc:10910	SLC12A1	TdgClinicalTrial	Jan-14	NULL	0.8334550989792778	BUMETANIDE	rxcui:1808	BUMETANIDE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.750109589	CARBACHOL	rxcui:1546387	CARBAMOYLCHOLINE	TRUE	FALSE	FALSE
UNIPROT:Q12791	hgnc:6284	KCNMA1	TdgClinicalTrial	Jan-14	NULL	1.944728564284981	CHLORZOXAZONE	rxcui:2410	CHLORZOXAZONE	TRUE	FALSE	FALSE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	0.9376369863516875	CISATRACURIUM BESYLATE	rxcui:136561	CISATRACURIUM BESYLATE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TdgClinicalTrial	Jan-14	NULL	0.083016081	CHLORPROTHIXENE	rxcui:2406	CHLORPROTHIXENE	TRUE	FALSE	FALSE
UNIPROT:P05091	hgnc:404	ALDH2	TdgClinicalTrial	Jan-14	NULL	0.07963752	DISULFIRAM	rxcui:3554	DISULFIRAM	TRUE	FALSE	FALSE
UNIPROT:P43115	hgnc:9595	PTGER3	TdgClinicalTrial	Jan-14	NULL	1.458546423213736	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:P35408	hgnc:9596	PTGER4	TdgClinicalTrial	Jan-14	NULL	0.7721716358190367	DINOPROSTONE	rxcui:3478	DINOPROSTONE	TRUE	FALSE	FALSE
UNIPROT:P27815	hgnc:8780	PDE4A	TdgClinicalTrial	Jan-14	NULL	0.6819178082557726	DYPHYLLINE	rxcui:3714	DYPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P10275	hgnc:644	AR	TdgClinicalTrial	Jan-14	NULL	0.116943588	DROMOSTANOLONE	rxcui:23678	DROMOSTANOLONE	TRUE	FALSE	TRUE
UNIPROT:P78334	hgnc:4085	GABRE	TdgClinicalTrial	Jan-14	NULL	0.079197091	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:Q99928	hgnc:4088	GABRG3	TdgClinicalTrial	Jan-14	NULL	0.07182992	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:O00591	hgnc:4089	GABRP	TdgClinicalTrial	Jan-14	NULL	0.078194596	FLUDIAZEPAM	ncit:C65709	FLUDIAZEPAM	FALSE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TdgClinicalTrial	Jan-14	NULL	0.2792961235941196	OXYPHENCYCLIMINE	rxcui:32698	OXYPHENCYCLIMINE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	0.3977853881492006	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
UNIPROT:Q13131	hgnc:9376	PRKAA1	TdgClinicalTrial	Jan-14	NULL	1.640864726115453	PHENFORMIN	rxcui:8129	PHENFORMIN	TRUE	FALSE	TRUE
UNIPROT:Q15822	hgnc:1956	CHRNA2	TdgClinicalTrial	Jan-14	NULL	7.501095891	PIPECURONIUM	rxcui:33742	PIPECURONIUM	TRUE	FALSE	FALSE
UNIPROT:P14867	hgnc:4075	GABRA1	TdgClinicalTrial	Jan-14	NULL	0.305277158	PICROTOXIN	rxcui:2539172	PICROTOXIN	FALSE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TdgClinicalTrial	Jan-14	NULL	1.790034246671403	PRACTOLOL	rxcui:8620	PRACTOLOL	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.4565884455277782	PROPERICIAZINE	rxcui:8766	PERICIAZINE	FALSE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.096967075	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TdgClinicalTrial	Jan-14	NULL	0.083744292	PROMETHAZINE	rxcui:142445	PROMETHAZINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P35368	hgnc:278	ADRA1B	TdgClinicalTrial	Jan-14	NULL	0.080103236	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P28335	hgnc:5295	HTR2C	TdgClinicalTrial	Jan-14	NULL	0.040640612	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TdgClinicalTrial	Jan-14	NULL	0.2047082699247349	PROMAZINE	rxcui:8742	PROMAZINE	TRUE	FALSE	FALSE
UNIPROT:P12821	hgnc:2707	ACE	TdgClinicalTrial	Jan-14	NULL	1.334940794127826	SPIRAPRIL	rxcui:36908	SPIRAPRIL	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1215455352678113	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
UNIPROT:P25100	hgnc:280	ADRA1D	TEND	1-Aug-11	NULL	0.2692701089009974	ALFUZOSIN	rxcui:17300	ALFUZOSIN	TRUE	FALSE	FALSE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.2983390411119005	ALCLOMETASONE	rxcui:108088	ALCLOMETASONE	TRUE	FALSE	FALSE
UNIPROT:P42081	hgnc:1705	CD86	TEND	1-Aug-11	NULL	3.500511415712966	ABATACEPT	rxcui:614391	ABATACEPT	TRUE	FALSE	FALSE
UNIPROT:P11511	hgnc:2594	CYP19A1	TEND	1-Aug-11	NULL	0.7693431682885642	ANASTROZOLE	rxcui:84857	ANASTROZOLE	TRUE	FALSE	TRUE
UNIPROT:P04083	hgnc:533	ANXA1	TEND	1-Aug-11	NULL	0.1704794520639431	AMCINONIDE	rxcui:17652	AMCINONIDE	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.099446347	ATENOLOL	rxcui:1202	ATENOLOL	TRUE	FALSE	FALSE
UNIPROT:P15509	hgnc:2435	CSF2RA	TEND	1-Aug-11	NULL	11.66837138570988	SARGRAMOSTIM	rxcui:69634	SARGRAMOSTIM	TRUE	TRUE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.5527123287967841	IUPHAR.LIGAND:364	iuphar.ligand:364	[3H]DIMETHYL-W84	FALSE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.4293851619741372	ATOMOXETINE	rxcui:353103	ATOMOXETINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:P23975	hgnc:11048	SLC6A2	TEND	1-Aug-11	NULL	0.1226814748497534	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P35348	hgnc:277	ADRA1A	TEND	1-Aug-11	NULL	0.1367387271762877	BETHANIDINE	rxcui:1523	BETHANIDINE	TRUE	FALSE	FALSE
UNIPROT:P14416	hgnc:3023	DRD2	TEND	1-Aug-11	NULL	0.020084536	BROMOCRIPTINE	rxcui:1760	BROMOCRIPTINE	TRUE	FALSE	FALSE
UNIPROT:P34903	hgnc:4077	GABRA3	TEND	1-Aug-11	NULL	0.087512785	BUTALBITAL	rxcui:19860	BUTALBITAL	TRUE	FALSE	FALSE
UNIPROT:P11473	hgnc:12679	VDR	TEND	1-Aug-11	NULL	0.3251536612259921	CALCITRIOL	rxcui:1894	CALCITRIOL	TRUE	FALSE	FALSE
UNIPROT:P08588	hgnc:285	ADRB1	TEND	1-Aug-11	NULL	0.3977853881492006	PINDOLOL	rxcui:8332	PINDOLOL	TRUE	FALSE	FALSE
UNIPROT:Q9UBS5	hgnc:4070	GABBR1	TEND	1-Aug-11	NULL	4.375639269641208	PROGABIDE	rxcui:34568	PROGABIDE	FALSE	FALSE	FALSE
UNIPROT:P48039	hgnc:7463	MTNR1A	TEND	1-Aug-11	NULL	7.501095891	RAMELTEON	rxcui:596205	RAMELTEON	TRUE	FALSE	FALSE
UNIPROT:P25021	hgnc:5183	HRH2	TEND	1-Aug-11	NULL	0.8204323630577265	RANITIDINE	rxcui:203136	RANITIDINE HYDROCHLORIDE	TRUE	FALSE	FALSE
UNIPROT:Q05940	hgnc:10935	SLC18A2	TEND	1-Aug-11	NULL	0.4039051633514962	RESERPINE	rxcui:9260	RESERPINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	modulator	0.276356164	IUPHAR.LIGAND:6938	iuphar.ligand:6938	LY2119620	FALSE	FALSE	FALSE
UNIPROT:P23219	hgnc:9604	PTGS1	TEND	1-Aug-11	NULL	0.4922594178346359	SUPROFEN	rxcui:10255	SUPROFEN	TRUE	FALSE	FALSE
UNIPROT:P05546	hgnc:4838	SERPIND1	TEND	1-Aug-11	NULL	26.25383561784724	SULODEXIDE	ncit:C152467	SULODEXIDE	TRUE	FALSE	FALSE
UNIPROT:P11229	hgnc:1950	CHRM1	TEND	1-Aug-11	NULL	0.101562227	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:7354	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
UNIPROT:Q07343	hgnc:8781	PDE4B	TEND	1-Aug-11	NULL	0.1296485709523321	THEOPHYLLINE	rxcui:10438	THEOPHYLLINE	TRUE	FALSE	FALSE
UNIPROT:P35367	hgnc:5182	HRH1	TEND	1-Aug-11	NULL	0.07699072	THIETHYLPERAZINE	rxcui:10471	THIETHYLPERAZINE	TRUE	FALSE	FALSE
UNIPROT:P16473	hgnc:12373	TSHR	TEND	1-Aug-11	NULL	0.9309870786470656	THYROTROPIN ALFA	rxcui:4952	THYROTROPIN ALFA	TRUE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:3264	iuphar.ligand:3264	AFDX384	FALSE	FALSE	FALSE
UNIPROT:P08173	hgnc:1953	CHRM4	TEND	1-Aug-11	NULL	0.5303805175322677	TROPICAMIDE	rxcui:10869	TROPICAMIDE	TRUE	FALSE	FALSE
UNIPROT:P08172	hgnc:1951	CHRM2	TEND	1-Aug-11	NULL	0.4605936073306534	TRIDIHEXETHYL	rxcui:38617	TRIDIHEXETHYL	TRUE	FALSE	FALSE
UNIPROT:P07437	hgnc:20778	TUBB	TEND	1-Aug-11	NULL	0.046303061	VINCRISTINE	rxcui:11202	VINCRISTINE	TRUE	FALSE	TRUE
UNIPROT:Q9BY41	hgnc:13315	HDAC8	TEND	1-Aug-11	NULL	0.29374921	VORINOSTAT	rxcui:194337	VORINOSTAT	TRUE	FALSE	TRUE
TRANSIENT RECEPTOR POTENTIAL CATION CHANNEL V1	hgnc:12716	TRPV1	TTD	2020.06.01	NULL	2.561349816375341	MR-1817	chembl:CHEMBL3707397	MR-1817	FALSE	FALSE	FALSE
NCBIGENE:15	hgnc:19	AANAT	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:7459	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
CYTOCHROME P450 24	hgnc:2602	CYP24A1	TTD	2020.06.01	NULL	1.944728564284981	Lunacalcipol	iuphar.ligand:11382	LUNACALCIPOL	FALSE	FALSE	FALSE
CHYMOTRYPSIN	hgnc:1440	CALCR	TTD	2020.06.01	NULL	2.187819634820604	Liprotamase	chembl:CHEMBL2108703	LIPROTAMASE	FALSE	FALSE	FALSE
PI3-KINASE GAMMA	hgnc:8978	PIK3CG	TTD	2020.06.01	NULL	0.062139256	GDC-0032	ncit:C116876	TASELISIB	FALSE	FALSE	TRUE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:7128	rxcui:1589	BIPERIDEN	TRUE	FALSE	FALSE
MANNAN-BINDING LECTIN SERINE PROTEASE-2	hgnc:6902	MASP2	TTD	2020.06.01	NULL	105.0153424713889	OMS721	ncit:C119952	NARSOPLIMAB	FALSE	FALSE	FALSE
INTERLEUKIN-6	hgnc:6018	IL6	TTD	2020.06.01	NULL	1.071585127259071	PF-04236921	chembl:CHEMBL2109613	PF-04236921	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:324	iuphar.ligand:324	HIMBACINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	modulator	0.035098711	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
MICRORNA HSA-MIR-155	hgnc:31542	MIR155	TTD	2020.06.01	NULL	13.12691780892362	MRG-201	chembl:CHEMBL4594491	REMLARSEN	FALSE	FALSE	FALSE
COLLAGEN	hgnc:633	AQP1	TTD	2020.06.01	NULL	0.6908904109959803	MRG-201	chembl:CHEMBL4594491	REMLARSEN	FALSE	FALSE	FALSE
C-X-C CHEMOKINE RECEPTOR TYPE 4	hgnc:2561	CXCR4	TTD	2020.06.01	NULL	2.100306849	PF-06747143	chembl:CHEMBL4297806	PF-06747143	FALSE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-5	hgnc:4079	GABRA5	TTD	2020.06.01	NULL	0.2983390411119005	Basmisanil	ncit:C167009	BASMISANIL	FALSE	FALSE	FALSE
MYELOID CELL SURFACE ANTIGEN CD33	hgnc:1659	CD33	TTD	2020.06.01	NULL	4.039051633514961	Vadastuximab talirine	ncit:C111039	VADASTUXIMAB TALIRINE	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:314	iuphar.ligand:314	MUSCARINIC TOXIN 7	FALSE	FALSE	FALSE
DIHYDROOROTATE DEHYDROGENASE	hgnc:2867	DHODH	TTD	2020.06.01	NULL	1.658136986390352	Vidofludimus	ncit:C152873	VIDOFLUDIMUS	FALSE	FALSE	FALSE
CANNABINOID RECEPTOR 1	hgnc:2159	CNR1	TTD	2020.06.01	NULL	1.166837138570988	TM38837	iuphar.ligand:8705	TM38837	FALSE	FALSE	FALSE
TUMOR NECROSIS FACTOR	hgnc:11892	TNF	TTD	2020.06.01	NULL	0.051327147	Nafamostat	ncit:C96292	NAFAMOSTAT	FALSE	FALSE	FALSE
NCBIGENE:16	hgnc:20	AARS1	GuideToPharmacology	2024.1	inhibitor	0.07458476	IUPHAR.LIGAND:7354	rxcui:1487512	UMECLIDINIUM BROMIDE	TRUE	FALSE	FALSE
B7 HOMOLOG 3	hgnc:19137	CD276	TTD	2020.06.01	NULL	10.50153424713889	124I-8H9	ncit:C99632	IODINE I 124 OMBURTAMAB	FALSE	FALSE	FALSE
MART-1 MELANOMA ANTIGEN	hgnc:7124	MLANA	TTD	2020.06.01	NULL	4.375639269641208	Melanoma vaccine	ncit:C2517	MELANOMA VACCINE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 1	hgnc:3688	FGFR1	TTD	2020.06.01	NULL	0.061340737	KW-2449	iuphar.ligand:5691	KW-2449	FALSE	FALSE	FALSE
COLLAGEN	hgnc:633	AQP1	TTD	2020.06.01	NULL	0.053145416	Vitamin C	rxcui:1151	ASCORBIC ACID	TRUE	FALSE	FALSE
HISTONE DEACETYLASE 1	hgnc:4852	HDAC1	TTD	2020.06.01	NULL	0.1769126389342806	Romidepsin	rxcui:877510	ROMIDEPSIN	TRUE	FALSE	TRUE
CARBONIC ANHYDRASE XII	hgnc:1371	CA12	TTD	2020.06.01	NULL	0.9376369863516875	PARABEN	chembl:CHEMBL441343	PARABEN	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	modulator	0.1591141552596803	IUPHAR.LIGAND:343	iuphar.ligand:343	BRUCINE N-OXIDE	FALSE	FALSE	FALSE
FIBROBLAST GROWTH FACTOR RECEPTOR 3	hgnc:3690	FGFR3	TTD	2020.06.01	NULL	0.042516333	E-3810	rxcui:114979	RABEPRAZOLE	TRUE	FALSE	TRUE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	1.389091831632129	Rindopepimut	ncit:C69076	RINDOPEPIMUT	FALSE	FALSE	TRUE
PROSTACYCLIN RECEPTOR	hgnc:9602	PTGIR	TTD	2020.06.01	NULL	5.625821918110125	Selexipag	rxcui:1729002	SELEXIPAG	TRUE	FALSE	FALSE
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2	hgnc:6307	KDR	TTD	2020.06.01	NULL	0.1232574442152452	RAF265	ncit:C61311	B-RAF/VEGFR-2 INHIBITOR RAF265	FALSE	FALSE	TRUE
AURORA KINASE B	hgnc:11390	AURKB	TTD	2020.06.01	NULL	0.020268015	ABT-348	ncit:C116729	ILORASERTIB	FALSE	FALSE	TRUE
ACETYLCHOLINESTERASE	hgnc:108	ACHE	TTD	2020.06.01	NULL	0.7721716358190367	Methanesulfonyl fluoride	drugbank:DB13058	METHANESULFONYL FLUORIDE	FALSE	FALSE	FALSE
SEROTONIN TRANSPORTER	hgnc:11050	SLC6A4	TTD	2020.06.01	NULL	0.596678082	DA-8031	chembl:CHEMBL5095175	DA-8031	FALSE	FALSE	FALSE
NCBIGENE:17	hgnc:22	AAVS1	GuideToPharmacology	2024.1	inhibitor	0.1591141552596803	IUPHAR.LIGAND:3264	iuphar.ligand:3264	AFDX384	FALSE	FALSE	FALSE
RAC-ALPHA SERINE/THREONINE-PROTEIN KINASE	hgnc:391	AKT1	TTD	2020.06.01	NULL	0.3697723326457359	CMX-2043	drugbank:DB12795	CMX-2043	FALSE	FALSE	FALSE
CELL SURFACE A33 ANTIGEN	hgnc:4445	GPA33	TTD	2020.06.01	NULL	39.38075342677087	KRN-330	chembl:CHEMBL2109293	KRN-330	FALSE	FALSE	FALSE
DNA TOPOISOMERASE I	hgnc:11986	TOP1	TTD	2020.06.01	NULL	0.8751278539282416	AR-67	iuphar.ligand:8919	AR-67	FALSE	FALSE	FALSE
INSULIN RECEPTOR	hgnc:6091	INSR	TTD	2020.06.01	NULL	0.2500365296937833	Mitoglitazone	drugbank:DB11721	MITOGLITAZONE	FALSE	FALSE	FALSE
NCBIGENE:1552	hgnc:7590	MYLK	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8152	iuphar.ligand:8152	RKI-1447	FALSE	FALSE	FALSE
INTERCELLULAR ADHESION MOLECULE ICAM-1	hgnc:5344	ICAM1	TTD	2020.06.01	NULL	6.563458904461812	lifitegrast	rxcui:1801820	LIFITEGRAST	TRUE	FALSE	FALSE
AMYLOID BETA A4 PROTEIN	hgnc:620	APP	TTD	2020.06.01	NULL	1.615620653405984	BAN2401	iuphar.ligand:12202	LECANEMAB	FALSE	FALSE	FALSE
RAC-GAMMA SERINE/THREONINE-PROTEIN KINASE	hgnc:393	AKT3	TTD	2020.06.01	NULL	0.4688184931758437	AZD5363	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9	hgnc:20001	PCSK9	TTD	2020.06.01	NULL	6.058577450272442	AMG 145	rxcui:1665684	EVOLOCUMAB	TRUE	FALSE	FALSE
T-CELL SURFACE GLYCOPROTEIN CD4	hgnc:1678	CD4	TTD	2020.06.01	NULL	3.281729452230906	BT-061	iuphar.ligand:9864	TREGALIZUMAB	FALSE	FALSE	FALSE
INTERLEUKIN 11 RECEPTOR ALPHA	hgnc:5967	IL11RA	TTD	2020.06.01	NULL	26.25383561784724	BMTP-11	ncit:C82370	BONE METASTASIS TARGETING PEPTIDE-11	FALSE	FALSE	FALSE
PI3-KINASE DELTA	hgnc:8977	PIK3CD	TTD	2020.06.01	NULL	0.1894216134043813	BAY 80-6946	rxcui:1945077	COPANLISIB	TRUE	FALSE	TRUE
ANDROGEN RECEPTOR	hgnc:644	AR	TTD	2020.06.01	NULL	0.1461794856227575	ARN-509	rxcui:1999574	APALUTAMIDE	TRUE	FALSE	TRUE
NCBIGENE:582	hgnc:966	BBS1	GuideToPharmacology	2024.1	blocker	0.4688184931758437	IUPHAR.LIGAND:10355	iuphar.ligand:10355	GNE-616	FALSE	FALSE	FALSE
POTASSIUM CHANNEL UNSPECIFIC	hgnc:1437	CALCA	TTD	2020.06.01	NULL	0.2160809515872201	Dronedarone	rxcui:233698	DRONEDARONE	TRUE	FALSE	FALSE
GABA(A) RECEPTOR ALPHA-5	hgnc:4079	GABRA5	TTD	2020.06.01	NULL	0.596678082	RG-7816	chembl:CHEMBL5095259	ALOGABAT	FALSE	FALSE	FALSE
CAMP-DEPENDENT CHLORIDE CHANNEL	hgnc:1884	CFTR	TTD	2020.06.01	NULL	1.193356164447602	GLPG-1837	drugbank:DB16835	GLPG-1837	FALSE	FALSE	FALSE
HISTAMINE H1 RECEPTOR	hgnc:5182	HRH1	TTD	2020.06.01	NULL	0.6351734423672721	Carbinoxamine	rxcui:20220	CARBINOXAMINE	TRUE	FALSE	FALSE
VOLTAGE-GATED CALCIUM CHANNEL ALPHA CAV1.2	hgnc:1390	CACNA1C	TTD	2020.06.01	NULL	0.1396480617970598	RAUWOLFIA SERPENTINA ROOT	rxcui:317836	RAUWOLFIA SERPENTINA (USP)	TRUE	FALSE	FALSE
NCBIGENE:584	hgnc:10597	SCN9A	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:10003	iuphar.ligand:10003	GNE-131	FALSE	FALSE	FALSE
CALCIUM CHANNEL UNSPECIFIC	hgnc:1421	SLC25A20	TTD	2020.06.01	NULL	3.500511415712966	Nexopamil	ncit:C66239	NEXOPAMIL	FALSE	FALSE	FALSE
OPIOID RECEPTOR DELTA	hgnc:8153	OPRD1	TTD	2020.06.01	NULL	0.3889457128569962	LY-25582	chembl:CHEMBL300662	CHEMBL:CHEMBL300662	FALSE	FALSE	FALSE
PROSTAGLANDIN G/H SYNTHASE 2	hgnc:9605	PTGS2	TTD	2020.06.01	NULL	0.1363835616511545	Mefenamic acid	rxcui:6693	MEFENAMIC ACID	TRUE	FALSE	FALSE
EPIDERMAL GROWTH FACTOR RECEPTOR	hgnc:3236	EGFR	TTD	2020.06.01	NULL	0.2778183663264259	S-222611	chembl:CHEMBL3545200	S-222611	FALSE	FALSE	FALSE
ADENOSINE DEAMINASE	hgnc:186	ADA	TTD	2020.06.01	NULL	2.282942227638891	EZN-2279	chembl:CHEMBL3990026	ELAPEGADEMASE	FALSE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	5.834185692854944	Anti-mesothelin CAR T Cells	ncit:C201275	ANTI-MESOTHELIN CAR T CELLS PREPARATION	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	agonist	1.093909817410302	IUPHAR.LIGAND:2095	iuphar.ligand:2095	SEPTIDE	FALSE	FALSE	FALSE
MESOTHELIN	hgnc:7371	MSLN	TTD	2020.06.01	NULL	5.834185692854944	Hu-CART meso cells	ncit:C148160	AUTOLOGOUS MESOTHELIN-SPECIFIC CAR-T CELLS	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.050294704	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.030176823	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	agonist	0.030176823	IUPHAR.LIGAND:52	ncit:C90625	ROXINDOLE	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.4526523382387456	IUPHAR.LIGAND:81	iuphar.ligand:81	[3H]P-MPPF	FALSE	FALSE	FALSE
NCBIGENE:1	hgnc:5	A1BG	GuideToPharmacology	2024.1	inhibitor	0.1131630845596864	IUPHAR.LIGAND:79	iuphar.ligand:79	WAY-100135	FALSE	FALSE	FALSE
NCBIGENE:2	hgnc:7	A2M	GuideToPharmacology	2024.1	agonist	0.070291394	IUPHAR.LIGAND:10	iuphar.ligand:10	BRL-15572	FALSE	FALSE	FALSE
NCBIGENE:361	hgnc:637	AQP4	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:2114	iuphar.ligand:2114	FK-888	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	modulator	0.3125456621172291	IUPHAR.LIGAND:137	iuphar.ligand:137	5-HT-MODULINE	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.6250913242344582	IUPHAR.LIGAND:139	iuphar.ligand:139	LYSERGIC ACID	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.062509132	IUPHAR.LIGAND:29	ncit:C77256	CAPESEROD	FALSE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	agonist	0.017363648	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:3	hgnc:8	A2MP1	GuideToPharmacology	2024.1	inhibitor	0.2083637747448194	IUPHAR.LIGAND:16	iuphar.ligand:16	L-772,405	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.031032903	IUPHAR.LIGAND:50	rxcui:221153	QUETIAPINE FUMARATE	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.101562227	IUPHAR.LIGAND:7	iuphar.ligand:31	[3H]8-OH-DPAT	FALSE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	0.1241316104862754	IUPHAR.LIGAND:40	rxcui:231049	ELETRIPTAN	TRUE	FALSE	FALSE
NCBIGENE:4	ncbigene:4	A12M1	GuideToPharmacology	2024.1	agonist	1.117184494376478	IUPHAR.LIGAND:146	iuphar.ligand:146	5-FLUOROTRYPTAMINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.08334551	IUPHAR.LIGAND:206	ncit:C83940	MESULERGINE	FALSE	FALSE	FALSE
NCBIGENE:6	ncbigene:6	A12M3	GuideToPharmacology	2024.1	inhibitor	0.1389091831632129	IUPHAR.LIGAND:191	iuphar.ligand:191	SB 221284	FALSE	FALSE	FALSE
NCBIGENE:7	ncbigene:7	A12M4	GuideToPharmacology	2024.1	inhibitor	0.1842374429322613	IUPHAR.LIGAND:186	iuphar.ligand:186	GLEMANSERIN	FALSE	FALSE	FALSE
NCBIGENE:360	hgnc:636	AQP3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5746	iuphar.ligand:5746	T2328	FALSE	FALSE	FALSE
NCBIGENE:8	hgnc:5295	HTR2C	GuideToPharmacology	2024.1	agonist	0.1286952726365061	IUPHAR.LIGAND:153	iuphar.ligand:153	(+)-DOI	FALSE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.012120884	IUPHAR.LIGAND:47	rxcui:61381	OLANZAPINE	TRUE	FALSE	FALSE
NCBIGENE:12	hgnc:16	SERPINA3	GuideToPharmacology	2024.1	inhibitor	0.1842374429322614	IUPHAR.LIGAND:206	ncit:C83940	MESULERGINE	FALSE	FALSE	FALSE
NCBIGENE:362	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:5766	iuphar.ligand:5766	PD 154740	FALSE	FALSE	FALSE
NCBIGENE:1791	hgnc:2983	DNTT	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:8086	iuphar.ligand:8086	BIMAGRUMAB	FALSE	FALSE	FALSE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	modulator	0.5527123287967842	IUPHAR.LIGAND:5921	iuphar.ligand:5921	AKT INHIBITOR VIII	FALSE	FALSE	FALSE
NCBIGENE:1480	hgnc:2486	CSTP1	GuideToPharmacology	2024.1	inhibitor	1.029562181092048	IUPHAR.LIGAND:12112	iuphar.ligand:12112	NTQ1062	FALSE	FALSE	FALSE
NCBIGENE:2286	hgnc:3718	FKBP2	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:7709	rxcui:2669967	CAPIVASERTIB	TRUE	FALSE	TRUE
NCBIGENE:1479	hgnc:2485	CSTF3	GuideToPharmacology	2024.1	inhibitor	0.9211872146613068	IUPHAR.LIGAND:12112	iuphar.ligand:12112	NTQ1062	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.4953553890159858	IUPHAR.LIGAND:498	iuphar.ligand:498	SNAP5089	FALSE	FALSE	FALSE
NCBIGENE:309	hgnc:544	ANXA6	GuideToPharmacology	2024.1	agonist	4.375639269641208	IUPHAR.LIGAND:1575	iuphar.ligand:1575	CONTULAKIN-G	FALSE	FALSE	FALSE
NCBIGENE:22	hgnc:48	ABCB7	GuideToPharmacology	2024.1	inhibitor	0.055039488	IUPHAR.LIGAND:135	rxcui:6929	MIANSERIN	FALSE	FALSE	FALSE
NCBIGENE:628	ncbigene:628	BEVI	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:11992	iuphar.ligand:11992	PRUXELUTAMIDE	FALSE	FALSE	FALSE
NCBIGENE:694	hgnc:1130	BTG1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
NCBIGENE:310	hgnc:545	ANXA7	GuideToPharmacology	2024.1	agonist	3.750547945	IUPHAR.LIGAND:1572	iuphar.ligand:1572	JMV458	FALSE	FALSE	FALSE
NCBIGENE:692	hgnc:638	AQP5	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:4215	iuphar.ligand:4215	HG2+	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:3761	iuphar.ligand:3761	[125I][GLP65NLE75,TYR77]APELIN-13	FALSE	FALSE	FALSE
NCBIGENE:36	hgnc:91	ACADSB	GuideToPharmacology	2024.1	agonist	1.640864726115453	IUPHAR.LIGAND:6311	iuphar.ligand:6311	CYCLO APELIN-12 (7-12)	FALSE	FALSE	FALSE
NCBIGENE:685	hgnc:1121	BTC	GuideToPharmacology	2024.1	activator	0.5048814541893702	IUPHAR.LIGAND:2346	iuphar.ligand:2346	H+	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1207072901969988	IUPHAR.LIGAND:5601	iuphar.ligand:5601	MRS3558	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.1508841127462485	IUPHAR.LIGAND:5590	iuphar.ligand:5590	TCPA	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	inhibitor	0.3017682254924971	IUPHAR.LIGAND:381	iuphar.ligand:381	AS100	FALSE	FALSE	FALSE
NCBIGENE:18	hgnc:23	ABAT	GuideToPharmacology	2024.1	agonist	0.3017682254924971	IUPHAR.LIGAND:11222	iuphar.ligand:11222	NELADENOSON	FALSE	FALSE	FALSE
NCBIGENE:62	hgnc:135	ACTBP2	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:7686	iuphar.ligand:7686	AZD5672	FALSE	FALSE	FALSE
NCBIGENE:1221	hgnc:10961	SLCO1B3	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:4570	rxcui:35616	RIFAMYCIN SV	TRUE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	0.4688184931758437	IUPHAR.LIGAND:6889	rxcui:42405	MUROMONAB-CD3	TRUE	TRUE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	1.640864726115453	IUPHAR.LIGAND:10353	iuphar.ligand:10353	TEPODITAMAB	FALSE	FALSE	FALSE
NCBIGENE:2742	hgnc:4327	GLRA2	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:12969	iuphar.ligand:12969	TARLATAMAB	FALSE	FALSE	FALSE
NCBIGENE:2628	hgnc:4175	GATM	GuideToPharmacology	2024.1	antibody	3.750547945	IUPHAR.LIGAND:12690	iuphar.ligand:12690	ODRONEXTAMAB	FALSE	FALSE	FALSE
NCBIGENE:2744	hgnc:4331	GLS	GuideToPharmacology	2024.1	NULL	0.1479089330582944	IUPHAR.LIGAND:6892	rxcui:1112973	BELATACEPT	TRUE	FALSE	FALSE
NCBIGENE:79	hgnc:152	ACTG1P7	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:2945	iuphar.ligand:2945	CHEMERIN	FALSE	FALSE	FALSE
NCBIGENE:707	hgnc:1884	CFTR	GuideToPharmacology	2024.1	NULL	5.966780822238011	IUPHAR.LIGAND:10552	rxcui:2256951	ELEXACAFTOR	TRUE	FALSE	FALSE
NCBIGENE:698	ncbigene:698	BTS1	GuideToPharmacology	2024.1	blocker	0.3409589041278864	IUPHAR.LIGAND:566	iuphar.ligand:566	ZN2+	FALSE	FALSE	FALSE
NCBIGENE:2362	hgnc:3870	FRA1C	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:6380	rxcui:1546356	DABIGATRAN	TRUE	FALSE	FALSE
NCBIGENE:1375	hgnc:2329	CPT1B	GuideToPharmacology	2024.1	inhibitor	0.7721716358190367	IUPHAR.LIGAND:10241	iuphar.ligand:10241	FK-881	FALSE	FALSE	FALSE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	inhibitor	0.525076712	IUPHAR.LIGAND:4570	rxcui:35616	RIFAMYCIN SV	TRUE	FALSE	FALSE
NCBIGENE:2842	hgnc:4473	GPR19	GuideToPharmacology	2024.1	antibody	6.563458904461812	IUPHAR.LIGAND:8294	iuphar.ligand:8294	LAMPALIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:2734	hgnc:4316	GLG1	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:7529	iuphar.ligand:7529	SGC-CBP30	FALSE	FALSE	FALSE
NCBIGENE:2876	hgnc:4553	GPX1	GuideToPharmacology	2024.1	NULL	26.25383561784724	IUPHAR.LIGAND:8609	iuphar.ligand:8609	KL044	FALSE	FALSE	FALSE
NCBIGENE:1994	hgnc:3312	ELAVL1	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:7648	drugbank:DB14765	RIVOCERANIB	FALSE	FALSE	FALSE
NCBIGENE:725	hgnc:1328	C4BPB	GuideToPharmacology	2024.1	inhibitor	0.546954909	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:68	hgnc:141	ACTBP8	GuideToPharmacology	2024.1	agonist	2.917092846427472	IUPHAR.LIGAND:8496	iuphar.ligand:8496	VCXCL1	FALSE	FALSE	FALSE
NCBIGENE:1224	hgnc:10962	SLCO2B1	GuideToPharmacology	2024.1	inhibitor	0.072424374	IUPHAR.LIGAND:2414	rxcui:4815	GLYBURIDE	TRUE	FALSE	FALSE
NCBIGENE:727	hgnc:1331	C5	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
NCBIGENE:1961	hgnc:3241	EGR4	GuideToPharmacology	2024.1	inhibitor	0.041672755	IUPHAR.LIGAND:7874	ncit:C92579	RONICICLIB	FALSE	FALSE	TRUE
NCBIGENE:1341	hgnc:2642	CYP4A11	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:11371	ncit:C72762	EPALRESTAT	FALSE	FALSE	FALSE
NCBIGENE:1337	hgnc:2277	COX6A1	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:10209	rxcui:10864	TROLEANDOMYCIN	TRUE	FALSE	FALSE
NCBIGENE:2356	hgnc:3824	FPGS	GuideToPharmacology	2024.1	inhibitor	4.773424657790408	IUPHAR.LIGAND:6536	iuphar.ligand:6536	COMPOUND 18 [PMID: 15664838]	FALSE	FALSE	FALSE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	0.046673486	IUPHAR.LIGAND:5687	rxcui:282388	IMATINIB	TRUE	FALSE	TRUE
NCBIGENE:1843	hgnc:3064	DUSP1	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:9354	iuphar.ligand:9354	DDR-IN-1	FALSE	FALSE	FALSE
NCBIGENE:369	hgnc:646	ARAF	GuideToPharmacology	2024.1	inhibitor	0.9546849315580818	IUPHAR.LIGAND:2247	iuphar.ligand:2247	L-367,938	FALSE	FALSE	FALSE
NCBIGENE:1844	hgnc:3068	DUSP2	GuideToPharmacology	2024.1	inhibitor	0.5834185692854945	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	agonist	0.1312691780892362	IUPHAR.LIGAND:1884	rxcui:3477	DINOPROST	FALSE	FALSE	FALSE
NCBIGENE:339	hgnc:604	APOBEC1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425933	IUPHAR.LIGAND:8995	ncit:C166588	FEVIPIPRANT	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.046673486	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.046673486	IUPHAR.LIGAND:56	ncit:C152567	TERGURIDE	FALSE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.070010228	IUPHAR.LIGAND:7427	rxcui:1086768	VILAZODONE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	inhibitor	0.1750255707856483	IUPHAR.LIGAND:9215	rxcui:1373	BENPERIDOL	TRUE	FALSE	FALSE
NCBIGENE:215	hgnc:61	ABCD1	GuideToPharmacology	2024.1	agonist	0.3500511415712966	IUPHAR.LIGAND:3949	ncit:C76651	SUMANIROLE	FALSE	FALSE	FALSE
NCBIGENE:334	hgnc:598	APLP2	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:1852	iuphar.ligand:1852	CV-6209	FALSE	FALSE	FALSE
NCBIGENE:1250	hgnc:7873	NOS2	GuideToPharmacology	2024.1	inhibitor	0.9460841664089098	IUPHAR.LIGAND:9849	iuphar.ligand:9849	GW274150	FALSE	FALSE	FALSE
NCBIGENE:2624	hgnc:4171	GATA2	GuideToPharmacology	2024.1	inhibitor	0.2983390411119005	IUPHAR.LIGAND:6832	rxcui:265323	MYCOPHENOLATE	TRUE	TRUE	FALSE
NCBIGENE:2045	hgnc:3390	EPHA7	GuideToPharmacology	2024.1	inhibitor	0.729273212	IUPHAR.LIGAND:9655	iuphar.ligand:9655	TAKINIB	FALSE	FALSE	FALSE
NCBIGENE:348	hgnc:613	APOE	GuideToPharmacology	2024.1	inhibitor	0.9053046764774912	IUPHAR.LIGAND:9570	iuphar.ligand:9570	C391	FALSE	FALSE	FALSE
NCBIGENE:1449	hgnc:14897	ITPKC	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:9548	iuphar.ligand:9548	GNF362	FALSE	FALSE	FALSE
NCBIGENE:744	hgnc:1180	MPPED2	GuideToPharmacology	2024.1	activator	3.500511415712966	IUPHAR.LIGAND:4222	iuphar.ligand:4222	IP3	FALSE	FALSE	FALSE
NCBIGENE:743	hgnc:6180	ITPR1	GuideToPharmacology	2024.1	activator	2.917092846427472	IUPHAR.LIGAND:4223	iuphar.ligand:4223	INOSITOL 2,4,5-TRISPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:165	hgnc:303	AEBP1	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:2916	iuphar.ligand:2916	DIOCTANOYLGLYCEROL PYROPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:659	hgnc:1078	BMPR2	GuideToPharmacology	2024.1	agonist	0.8204323630577265	IUPHAR.LIGAND:6953	rxcui:236146	DEXTROMETHORPHAN POLISTIREX	TRUE	FALSE	FALSE
NCBIGENE:678	hgnc:1108	ZFP36L2	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:12460	rxcui:1310546	ACESULFAME	TRUE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	1.591141552596803	IUPHAR.LIGAND:2676	iuphar.ligand:2676	PRISTANIC ACID	FALSE	FALSE	FALSE
NCBIGENE:662	hgnc:1082	BNIP1	GuideToPharmacology	2024.1	agonist	0.9723642821424908	IUPHAR.LIGAND:7002	iuphar.ligand:7002	EPIGALLOCATECHIN-3-GALLATE	FALSE	FALSE	FALSE
NCBIGENE:679	hgnc:18877	TAS2R46	GuideToPharmacology	2024.1	agonist	1.458546423213736	IUPHAR.LIGAND:9675	drugbank:DB05767	ANDROGRAPHOLIDE	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2917092846427472	IUPHAR.LIGAND:10744	iuphar.ligand:10744	GOLIDOCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.072927321	IUPHAR.LIGAND:8957	ncit:C113173	CERDULATINIB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:12871	iuphar.ligand:12871	LEPZACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1458546423213736	IUPHAR.LIGAND:5993	iuphar.ligand:5993	JAK3 INHIBITOR II	FALSE	FALSE	TRUE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:8364	iuphar.ligand:8364	ITACITINIB	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.2187819634820604	IUPHAR.LIGAND:10631	iuphar.ligand:10631	LORPUCITINIB	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.012561644	IUPHAR.LIGAND:5932	iuphar.ligand:5932	JNJ-7706621	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.1562728310586145	IUPHAR.LIGAND:11135	ncit:C166574	ELAFIBRANOR	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.4375639269641208	IUPHAR.LIGAND:12621	iuphar.ligand:12621	WXFL10203614	FALSE	FALSE	FALSE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.062509132	IUPHAR.LIGAND:5677	rxcui:1357536	TOFACITINIB	TRUE	FALSE	TRUE
NCBIGENE:2047	hgnc:3392	EPHB1	GuideToPharmacology	2024.1	inhibitor	0.1250182648468916	IUPHAR.LIGAND:10947	iuphar.ligand:10947	NIK INHIBITOR 12F	FALSE	FALSE	FALSE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.1151484018326633	IUPHAR.LIGAND:5993	iuphar.ligand:5993	JAK3 INHIBITOR II	FALSE	FALSE	TRUE
NCBIGENE:2048	hgnc:3393	EPHB2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:8364	iuphar.ligand:8364	ITACITINIB	FALSE	FALSE	FALSE
NCBIGENE:972	hgnc:1697	CD74	GuideToPharmacology	2024.1	inhibitor	3.281729452230906	IUPHAR.LIGAND:4589	iuphar.ligand:4589	DIOA	FALSE	FALSE	FALSE
NCBIGENE:1813	hgnc:3023	DRD2	GuideToPharmacology	2024.1	inhibitor	0.0296486	IUPHAR.LIGAND:8104	iuphar.ligand:8104	LY2874455	FALSE	FALSE	FALSE
NCBIGENE:521	hgnc:846	ATP5ME	GuideToPharmacology	2024.1	activator	3.750547945	IUPHAR.LIGAND:10336	iuphar.ligand:10336	BL-1249	FALSE	FALSE	FALSE
NCBIGENE:515	hgnc:840	ATP5PB	GuideToPharmacology	2024.1	blocker	8.751278539282415	IUPHAR.LIGAND:11206	iuphar.ligand:11206	AVE1231	FALSE	FALSE	FALSE
NCBIGENE:520	hgnc:844	ATP5MC2P1	GuideToPharmacology	2024.1	inhibitor	2.625383561784725	IUPHAR.LIGAND:2506	iuphar.ligand:2506	R-(+)-METHANANDAMIDE	FALSE	FALSE	FALSE
NCBIGENE:381	hgnc:658	ARF5	GuideToPharmacology	2024.1	activator	0.6563458904461812	IUPHAR.LIGAND:2335	iuphar.ligand:2335	SKA-31	FALSE	FALSE	FALSE
NCBIGENE:382	hgnc:659	ARF6	GuideToPharmacology	2024.1	activator	0.8204323630577265	IUPHAR.LIGAND:2335	iuphar.ligand:2335	SKA-31	FALSE	FALSE	FALSE
NCBIGENE:383	hgnc:663	ARG1	GuideToPharmacology	2024.1	activator	0.6250913242344582	IUPHAR.LIGAND:2335	iuphar.ligand:2335	SKA-31	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	blocker	2.500365296937833	IUPHAR.LIGAND:2336	iuphar.ligand:2336	TRAM-34	FALSE	FALSE	FALSE
NCBIGENE:384	hgnc:664	ARG2	GuideToPharmacology	2024.1	activator	0.108711535	IUPHAR.LIGAND:2326	rxcui:35623	RILUZOLE	TRUE	FALSE	FALSE
NCBIGENE:434	hgnc:745	ASIP	GuideToPharmacology	2024.1	activator	2.625383561784724	IUPHAR.LIGAND:2340	iuphar.ligand:2340	NA+	FALSE	FALSE	FALSE
NCBIGENE:386	hgnc:18866	KCNT2	GuideToPharmacology	2024.1	activator	0.6731752722524936	IUPHAR.LIGAND:2439	rxcui:7418	NIFLUMIC ACID	FALSE	FALSE	FALSE
NCBIGENE:435	hgnc:746	ASL	GuideToPharmacology	2024.1	activator	4.375639269641208	IUPHAR.LIGAND:2340	iuphar.ligand:2340	NA+	FALSE	FALSE	FALSE
NCBIGENE:438	hgnc:750	ASMT	GuideToPharmacology	2024.1	blocker	26.25383561784724	IUPHAR.LIGAND:11821	iuphar.ligand:11821	VU0134992	FALSE	FALSE	FALSE
NCBIGENE:543	hgnc:880	ALDH7A1P3	GuideToPharmacology	2024.1	blocker	13.12691780892362	IUPHAR.LIGAND:2563	iuphar.ligand:2563	&ALPHA;-DENDROTOXIN	FALSE	FALSE	FALSE
NCBIGENE:94	hgnc:175	ACVRL1	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:2906	iuphar.ligand:2906	LPA	FALSE	FALSE	FALSE
NCBIGENE:1242	hgnc:20692	TPH2	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:5126	iuphar.ligand:5126	6-FLUOROTRYPTOPHAN	FALSE	FALSE	FALSE
NCBIGENE:124	hgnc:249	ADH1A	GuideToPharmacology	2024.1	agonist	0.4688184931758437	IUPHAR.LIGAND:2906	iuphar.ligand:2906	LPA	FALSE	FALSE	FALSE
NCBIGENE:1243	ncbigene:1243	CMM	GuideToPharmacology	2024.1	inhibitor	4.375639269641208	IUPHAR.LIGAND:5095	iuphar.ligand:5095	&ALPHA;-PROPYLDOPACETAMIDE	FALSE	FALSE	FALSE
NCBIGENE:285	hgnc:485	ANGPT2	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:1340	iuphar.ligand:1340	MCL0129	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.3977853881492007	IUPHAR.LIGAND:11135	ncit:C166574	ELAFIBRANOR	FALSE	FALSE	FALSE
NCBIGENE:2109	hgnc:3482	ETFB	GuideToPharmacology	2024.1	inhibitor	0.2442217266776488	IUPHAR.LIGAND:7743	iuphar.ligand:7743	IZORLISIB	FALSE	FALSE	FALSE
NCBIGENE:3136	hgnc:4965	HLA-H	GuideToPharmacology	2024.1	inhibitor	5.834185692854944	IUPHAR.LIGAND:9599	drugbank:DB14793	RO-5045337	FALSE	FALSE	TRUE
NCBIGENE:1815	hgnc:3025	DRD4	GuideToPharmacology	2024.1	inhibitor	0.6177373086552294	IUPHAR.LIGAND:12391	iuphar.ligand:12391	VABAMETKIB	FALSE	FALSE	FALSE
NCBIGENE:593	hgnc:986	BCKDHA	GuideToPharmacology	2024.1	agonist	0.2651902587661338	IUPHAR.LIGAND:2661	iuphar.ligand:2661	N-OLEOYLETHANOLAMIDE	FALSE	FALSE	FALSE
NCBIGENE:289	ncbigene:289	ANOP1	GuideToPharmacology	2024.1	modulator	1.280674908	IUPHAR.LIGAND:6357	iuphar.ligand:6357	COMPOUND 12E [PMID: 22266036]	FALSE	FALSE	FALSE
NCBIGENE:640	hgnc:1057	BLK	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:3051	drugbank:DB02552	GERANYL DIPHOSPHATE	FALSE	FALSE	FALSE
NCBIGENE:290	hgnc:500	ANPEP	GuideToPharmacology	2024.1	inhibitor	0.1103102336884338	IUPHAR.LIGAND:1378	iuphar.ligand:1378	LY341495	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.5357925636295356	IUPHAR.LIGAND:6439	iuphar.ligand:6439	AZD9272	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:10002	iuphar.ligand:10002	TRIPLE MODULATOR 10 [PMID: 29878767]	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	inhibitor	0.2500365296937833	IUPHAR.LIGAND:1378	iuphar.ligand:1378	LY341495	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	0.5357925636295356	IUPHAR.LIGAND:9309	ncit:C166619	BASIMGLURANT	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6232	iuphar.ligand:6232	COMPOUND 7 [PMID: 20638279]	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6419	iuphar.ligand:6419	COMPOUND 24 [PMID: 23374867]	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	1.750255707856483	IUPHAR.LIGAND:6230	iuphar.ligand:6230	VU0359516	FALSE	FALSE	FALSE
NCBIGENE:2152	hgnc:3541	F3	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:10598	iuphar.ligand:10598	COMPOUND 41 [PMID: 31855425]	FALSE	FALSE	FALSE
NCBIGENE:292	hgnc:10991	SLC25A5	GuideToPharmacology	2024.1	modulator	0.4375639269641208	IUPHAR.LIGAND:6227	iuphar.ligand:6227	VU0080241	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	modulator	1.071585127259071	IUPHAR.LIGAND:6406	iuphar.ligand:6406	COMPOUND 47 [PMID: 21295468]	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:3388	iuphar.ligand:3388	ACDPP	FALSE	FALSE	FALSE
NCBIGENE:295	ncbigene:295	ANTP2	GuideToPharmacology	2024.1	agonist	0.8334550989792776	IUPHAR.LIGAND:6706	iuphar.ligand:6706	LSP4-2022	FALSE	FALSE	FALSE
NCBIGENE:293	hgnc:10992	SLC25A6	GuideToPharmacology	2024.1	inhibitor	1.071585127259071	IUPHAR.LIGAND:3344	iuphar.ligand:1425	[3H]M-MPEP	FALSE	FALSE	FALSE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	agonist	1.381780822	IUPHAR.LIGAND:2872	iuphar.ligand:2872	ALDOSTERONE	FALSE	FALSE	FALSE
NCBIGENE:595	hgnc:1582	CCND1	GuideToPharmacology	2024.1	inhibitor	0.052090944	IUPHAR.LIGAND:2807	rxcui:233272	BEXAROTENE	TRUE	FALSE	TRUE
NCBIGENE:626	hgnc:7979	NR3C2	GuideToPharmacology	2024.1	inhibitor	0.3454452054979901	IUPHAR.LIGAND:2882	ncit:C170255	ONAPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:1495	hgnc:2509	CTNNA1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:11727	iuphar.ligand:11727	ASTX029	FALSE	FALSE	FALSE
NCBIGENE:3024	hgnc:4715	H1-1	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:10917	rxcui:235559	NITROFURANTOIN, MACROCRYSTALS	TRUE	FALSE	FALSE
NCBIGENE:2153	hgnc:3542	F5	GuideToPharmacology	2024.1	inhibitor	0.084281976	IUPHAR.LIGAND:8011	iuphar.ligand:8011	KU-0060648	FALSE	FALSE	TRUE
NCBIGENE:1062	hgnc:1856	CENPE	GuideToPharmacology	2024.1	inhibitor	17.50255707856483	IUPHAR.LIGAND:4572	iuphar.ligand:4572	CARBOXYATRACTYLOSIDE	FALSE	FALSE	FALSE
NCBIGENE:3023	ncbigene:3023	H4F3	GuideToPharmacology	2024.1	inhibitor	1.009762908	IUPHAR.LIGAND:2919	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
NCBIGENE:1500	hgnc:2515	CTNND1	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:5719	ncit:C170207	NEFLAMAPIMOD	FALSE	FALSE	FALSE
NCBIGENE:1498	hgnc:2513	CTNNA1P1	GuideToPharmacology	2024.1	inhibitor	0.7001022831425934	IUPHAR.LIGAND:9989	iuphar.ligand:9989	COMPOUND 11 [PMID: 26431428]	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.059532507	IUPHAR.LIGAND:8011	iuphar.ligand:8011	KU-0060648	FALSE	FALSE	TRUE
NCBIGENE:1496	hgnc:2510	CTNNA2	GuideToPharmacology	2024.1	inhibitor	0.6250913242344582	IUPHAR.LIGAND:9836	ncit:C152510	TANZISERTIB	FALSE	FALSE	FALSE
NCBIGENE:2065	hgnc:3431	ERBB3	GuideToPharmacology	2024.1	inhibitor	0.060562481	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:2080	hgnc:6857	MAP3K5	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:10430	iuphar.ligand:10430	GS-444217	FALSE	FALSE	FALSE
NCBIGENE:2154	hgnc:8976	PIK3CB	GuideToPharmacology	2024.1	inhibitor	0.049026771	IUPHAR.LIGAND:5682	ncit:C165479	PICTILISIB	FALSE	FALSE	TRUE
NCBIGENE:2081	hgnc:3449	ERN1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:8133	iuphar.ligand:8133	COMPOUND 10 [PMID: 23147077]	FALSE	FALSE	FALSE
NCBIGENE:2074	hgnc:3438	ERCC6	GuideToPharmacology	2024.1	inhibitor	0.7501095890813498	IUPHAR.LIGAND:10947	iuphar.ligand:10947	NIK INHIBITOR 12F	FALSE	FALSE	FALSE
NCBIGENE:2072	hgnc:3436	ERCC4	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:8173	iuphar.ligand:8173	CEP-1347	FALSE	FALSE	FALSE
NCBIGENE:2087	ncbigene:2087	ERVK2	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:10389	iuphar.ligand:10389	RIPK3 INHIBITOR 18	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:12075	iuphar.ligand:12075	VULOLISIB	FALSE	FALSE	FALSE
NCBIGENE:2106	hgnc:26617	MLKL	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:12194	iuphar.ligand:12194	COMPOUND 56 [PMID: 36136378]	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:2288	hgnc:3720	FKBP4	GuideToPharmacology	2024.1	inhibitor	2.187819634820604	IUPHAR.LIGAND:8793	iuphar.ligand:8793	SAR260301	FALSE	FALSE	TRUE
NCBIGENE:1641	hgnc:2714	DCX	GuideToPharmacology	2024.1	inhibitor	2.100306849	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:1637	hgnc:2708	DCR	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:5170	iuphar.ligand:5170	CL82198	FALSE	FALSE	FALSE
NCBIGENE:1629	hgnc:2698	DBT	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:5140	iuphar.ligand:5140	ARP100	FALSE	FALSE	FALSE
NCBIGENE:2489	ncbigene:2489	FSHMD1A	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6637	ncit:C77519	BEFLOXATONE	FALSE	FALSE	FALSE
NCBIGENE:1399	hgnc:2363	CRKL	GuideToPharmacology	2024.1	inhibitor	1.750255707856483	IUPHAR.LIGAND:12994	iuphar.ligand:12994	CAY10499	FALSE	FALSE	FALSE
NCBIGENE:1632	hgnc:2703	ECI1	GuideToPharmacology	2024.1	inhibitor	0.2625383561784725	IUPHAR.LIGAND:7409	ncit:C96286	ILOMASTAT	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	1.875273972703375	IUPHAR.LIGAND:1452	iuphar.ligand:1452	[BPA1,ILE13]MOTILIN (HUMAN)	FALSE	FALSE	FALSE
NCBIGENE:297	ncbigene:297	ANTP4	GuideToPharmacology	2024.1	agonist	0.2083637747448194	IUPHAR.LIGAND:1465	rxcui:9478	ROXITHROMYCIN	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.100976291	IUPHAR.LIGAND:343	iuphar.ligand:343	BRUCINE N-OXIDE	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	inhibitor	0.100976291	IUPHAR.LIGAND:8584	iuphar.ligand:8584	AQ-RA 741	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.252440727	IUPHAR.LIGAND:338	iuphar.ligand:338	KT 5823	FALSE	FALSE	FALSE
NCBIGENE:13	hgnc:17	AADAC	GuideToPharmacology	2024.1	modulator	0.5048814541893701	IUPHAR.LIGAND:3261	iuphar.ligand:3261	VU0029767	FALSE	FALSE	FALSE
NCBIGENE:1304	hgnc:8784	PDE5A	GuideToPharmacology	2024.1	inhibitor	0.1262203635473425	IUPHAR.LIGAND:2919	ncit:C66685	ZAPRINAST	FALSE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.012282496	IUPHAR.LIGAND:200	rxcui:203168	AMITRIPTYLINE HYDROCHLORIDE	TRUE	FALSE	FALSE
NCBIGENE:14	hgnc:18	AAMP	GuideToPharmacology	2024.1	inhibitor	0.069089041	IUPHAR.LIGAND:7459	rxcui:1546438	GLYCOPYRRONIUM	TRUE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:7924	iuphar.ligand:7924	BOMPPA	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	0.5834185692854944	IUPHAR.LIGAND:1350	iuphar.ligand:1350	IIK7	FALSE	FALSE	FALSE
NCBIGENE:288	hgnc:494	ANK3	GuideToPharmacology	2024.1	agonist	1.166837138570988	IUPHAR.LIGAND:9226	iuphar.ligand:9226	UCM1014	FALSE	FALSE	FALSE
NCBIGENE:319	hgnc:615	APOF	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:1603	iuphar.ligand:1603	(-)-BREMAZOCINE	FALSE	FALSE	FALSE
NCBIGENE:350	hgnc:616	APOH	GuideToPharmacology	2024.1	agonist	5.250767123569449	IUPHAR.LIGAND:3739	iuphar.ligand:3739	GYPGQV-NH2	FALSE	FALSE	FALSE
NCBIGENE:2158	hgnc:3551	F9	GuideToPharmacology	2024.1	inhibitor	0.4605936073306534	IUPHAR.LIGAND:12708	iuphar.ligand:12708	GDC-0339	FALSE	FALSE	FALSE
NCBIGENE:2894	hgnc:4575	GRID1	GuideToPharmacology	2024.1	inhibitor	8.751278539282415	IUPHAR.LIGAND:8625	iuphar.ligand:8625	O-F-AMIDINE	FALSE	FALSE	FALSE
NCBIGENE:2155	hgnc:3544	F7	GuideToPharmacology	2024.1	inhibitor	0.023151531	IUPHAR.LIGAND:7888	ncit:C91731	APITOLISIB	FALSE	FALSE	TRUE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1544343271638073	IUPHAR.LIGAND:8974	iuphar.ligand:8974	OMIPALISIB	FALSE	FALSE	FALSE
NCBIGENE:2156	hgnc:3545	F7R	GuideToPharmacology	2024.1	inhibitor	0.1930429089547591	IUPHAR.LIGAND:9928	iuphar.ligand:9928	PUQUITINIB	FALSE	FALSE	FALSE
NCBIGENE:1298	hgnc:2218	COL9A2	GuideToPharmacology	2024.1	inhibitor	0.9723642821424906	IUPHAR.LIGAND:9063	rxcui:49626	ENOXIMONE	TRUE	FALSE	FALSE
NCBIGENE:2402	hgnc:3913	FRA6B	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:8848	iuphar.ligand:8848	SCH-900229	FALSE	FALSE	FALSE
NCBIGENE:335	hgnc:600	APOA1	GuideToPharmacology	2024.1	agonist	1.141471113819445	IUPHAR.LIGAND:8522	iuphar.ligand:8522	[125I]BH-MIT1	FALSE	FALSE	FALSE
NCBIGENE:2945	ncbigene:2945	GSTM5P1	GuideToPharmacology	2024.1	inhibitor	26.25383561784724	IUPHAR.LIGAND:10112	iuphar.ligand:10112	DOOKU1	FALSE	FALSE	FALSE
NCBIGENE:2394	hgnc:3906	FRA5B	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:6537	iuphar.ligand:6537	BIS-TRIAZOLE DERIVATIVE 10	FALSE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:1865	iuphar.ligand:1865	MIT1	FALSE	FALSE	FALSE
NCBIGENE:336	hgnc:601	APOA2	GuideToPharmacology	2024.1	agonist	2.625383561784724	IUPHAR.LIGAND:8522	iuphar.ligand:8522	[125I]BH-MIT1	FALSE	FALSE	FALSE
NCBIGENE:1804	hgnc:3010	DPP6	GuideToPharmacology	2024.1	inhibitor	0.210030685	IUPHAR.LIGAND:5982	iuphar.ligand:5982	GTP-14564	FALSE	FALSE	FALSE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	0.6177373086552295	IUPHAR.LIGAND:7918	ncit:C143162	ONVANSERTIB	FALSE	FALSE	TRUE
NCBIGENE:2168	hgnc:3555	FABP1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:10072	iuphar.ligand:10072	DUAL BRD4/PLK1 INHIBITOR 23	FALSE	FALSE	FALSE
NCBIGENE:2171	hgnc:3560	FABP5	GuideToPharmacology	2024.1	inhibitor	2.625383561784724	IUPHAR.LIGAND:8057	iuphar.ligand:8057	XMD8-92	FALSE	FALSE	FALSE
NCBIGENE:2772	hgnc:4386	GNAI2P1	GuideToPharmacology	2024.1	inhibitor	0.1944728564284981	IUPHAR.LIGAND:8313	rxcui:2099704	TALAZOPARIB	TRUE	FALSE	TRUE
NCBIGENE:606	hgnc:1007	NBEAP1	GuideToPharmacology	2024.1	agonist	0.1041818873724097	IUPHAR.LIGAND:2805	rxcui:6964	MIFEPRISTONE	TRUE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	0.1562728310586145	IUPHAR.LIGAND:8450	rxcui:1723735	IXAZOMIB	TRUE	FALSE	FALSE
NCBIGENE:2406	hgnc:3917	FRA6F	GuideToPharmacology	2024.1	inhibitor	1.640864726115453	IUPHAR.LIGAND:10409	iuphar.ligand:10409	ZETOMIPZOMIB	FALSE	FALSE	FALSE
NCBIGENE:1476	hgnc:2482	CSTB	GuideToPharmacology	2024.1	inhibitor	3.500511415712967	IUPHAR.LIGAND:10423	ncit:C152226	RIPASUDIL	FALSE	FALSE	FALSE
NCBIGENE:1477	hgnc:2483	CSTF1	GuideToPharmacology	2024.1	inhibitor	1.544343271638073	IUPHAR.LIGAND:346	drugbank:DB02010	STAUROSPORINE	FALSE	FALSE	FALSE
NCBIGENE:1486	hgnc:2496	CTBS	GuideToPharmacology	2024.1	inhibitor	3.750547945	IUPHAR.LIGAND:5953	iuphar.ligand:5953	CHELERYTHRINE	FALSE	FALSE	FALSE
NCBIGENE:1482	hgnc:2488	NKX2-5	GuideToPharmacology	2024.1	inhibitor	0.9546849315580819	IUPHAR.LIGAND:5192	iuphar.ligand:5192	G&OUML; 6983	FALSE	FALSE	FALSE
NCBIGENE:1484	ncbigene:1484	CTAA2	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:5263	ncit:C66524	RUBOXISTAURIN	FALSE	FALSE	FALSE
NCBIGENE:2388	hgnc:3900	FRA4A	GuideToPharmacology	2024.1	antibody	7.501095891	IUPHAR.LIGAND:12517	iuphar.ligand:12517	TAFOLECIMAB	FALSE	FALSE	FALSE
NCBIGENE:1520	hgnc:2545	CTSS	GuideToPharmacology	2024.1	inhibitor	3.500511415712966	IUPHAR.LIGAND:8156	iuphar.ligand:8156	COMPOUND 20 [PMID: 22136433]	FALSE	FALSE	FALSE
NCBIGENE:2801	hgnc:4425	GOLGA2	GuideToPharmacology	2024.1	inhibitor	6.563458904461812	IUPHAR.LIGAND:11558	iuphar.ligand:11558	COMPOUND I [PMID: 29351497]	FALSE	FALSE	FALSE
NCBIGENE:2189	hgnc:3588	FANCG	GuideToPharmacology	2024.1	inhibitor	0.7955707762984013	IUPHAR.LIGAND:10388	iuphar.ligand:10388	SZM594	FALSE	FALSE	FALSE
NCBIGENE:2190	hgnc:10020	RIPK2	GuideToPharmacology	2024.1	inhibitor	5.250767123569449	IUPHAR.LIGAND:9134	iuphar.ligand:9134	GSK583	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	0.3281729452230906	IUPHAR.LIGAND:9962	rxcui:2205637	TRIFAROTENE	TRUE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	agonist	1.312691780892362	IUPHAR.LIGAND:2649	iuphar.ligand:2649	AGN193836	FALSE	FALSE	FALSE
NCBIGENE:590	hgnc:983	BCHE	GuideToPharmacology	2024.1	inhibitor	1.312691780892362	IUPHAR.LIGAND:2643	iuphar.ligand:2643	BMS614	FALSE	FALSE	FALSE
NCBIGENE:610	hgnc:4846	HCN2	GuideToPharmacology	2024.1	inhibitor	0.192335792	IUPHAR.LIGAND:5425	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
NCBIGENE:2760	hgnc:4367	GM2A	GuideToPharmacology	2024.1	antibody	3.281729452230906	IUPHAR.LIGAND:12989	iuphar.ligand:12989	TORIPALIMAB	FALSE	FALSE	FALSE
NCBIGENE:596	hgnc:990	BCL2	GuideToPharmacology	2024.1	agonist	0.2134458180312784	IUPHAR.LIGAND:2903	iuphar.ligand:2903	GSK4112	FALSE	FALSE	FALSE
NCBIGENE:1503	hgnc:2519	CTPS1	GuideToPharmacology	2024.1	inhibitor	0.6908904109959803	IUPHAR.LIGAND:8037	iuphar.ligand:8037	GSK269962A	FALSE	FALSE	FALSE
NCBIGENE:1504	hgnc:2521	CTRB1	GuideToPharmacology	2024.1	inhibitor	1.250182648468916	IUPHAR.LIGAND:10498	iuphar.ligand:10498	COMPOUND 8 [PMID: 25898023]	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.1527273741585063	TAK-632	iuphar.ligand:10387	TAK-632	FALSE	FALSE	FALSE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.8247278204559345	PLX8394	drugbank:DB16038	PLX8394	FALSE	FALSE	TRUE
BRAF	hgnc:1097	BRAF	JAX-CKB	10-Apr-24	NULL	0.049983504	Futibatinib	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.6177373086552294	Spartalizumab	ncit:C121625	SPARTALIZUMAB	FALSE	FALSE	FALSE
CD274	hgnc:17635	CD274	JAX-CKB	10-Apr-24	NULL	0.7721716358190368	Camrelizumab	ncit:C123816	CAMRELIZUMAB	FALSE	FALSE	FALSE
NCBIGENE:737	hgnc:20573	PANX3	GuideToPharmacology	2024.1	inhibitor	1.093909817410302	IUPHAR.LIGAND:4151	ncit:C63669	CARBENOXOLONE	FALSE	FALSE	FALSE
FGFR2	hgnc:3689	FGFR2	JAX-CKB	10-Apr-24	NULL	0.010261417	Fluorouracil	rxcui:4492	FLUOROURACIL	TRUE	FALSE	TRUE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.050246575	Quisinostat	ncit:C77912	QUISINOSTAT	FALSE	FALSE	FALSE
FGFR3	hgnc:3690	FGFR3	JAX-CKB	10-Apr-24	NULL	0.3517260274161354	Futibatinib	rxcui:2628190	FUTIBATINIB	TRUE	FALSE	TRUE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.4321619031744402	FF-10101	chembl:CHEMBL4650283	FF-10101	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.6482428547616604	SKI-G-801	ncit:C155773	DENFIVONTINIB HYDROCHLORIDE	FALSE	FALSE	FALSE
FLT3	hgnc:3765	FLT3	JAX-CKB	10-Apr-24	NULL	0.044198376	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.1535312024435511	LY3009120	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
HRAS	hgnc:5173	HRAS	JAX-CKB	10-Apr-24	NULL	0.1973972602845657	LY3214996	ncit:C131335	TEMUTERKIB	FALSE	FALSE	FALSE
IDH2	hgnc:5383	IDH2	JAX-CKB	10-Apr-24	NULL	0.729273212	Dubermatinib	ncit:C127116	DUBERMATINIB	FALSE	FALSE	FALSE
NCBIGENE:2184	hgnc:3579	FAH	GuideToPharmacology	2024.1	inhibitor	0.1193356164447602	IUPHAR.LIGAND:8072	iuphar.ligand:8072	GW5074	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.094099769	RO5126766	ncit:C80060	AVUTOMETINIB	FALSE	FALSE	FALSE
NRAS	hgnc:7989	NRAS	JAX-CKB	10-Apr-24	NULL	0.2822993077187876	PLX8394	drugbank:DB16038	PLX8394	FALSE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.03683198	Selumetinib	rxcui:2289380	SELUMETINIB	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.057878826	Sulindac	rxcui:10237	SULINDAC	TRUE	FALSE	TRUE
PIK3CA	hgnc:8975	PIK3CA	JAX-CKB	10-Apr-24	NULL	0.010884675	Celecoxib	rxcui:140587	CELECOXIB	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.028382525	Pemetrexed Disodium	rxcui:282443	PEMETREXED DISODIUM	TRUE	FALSE	TRUE
PTEN	hgnc:9588	PTEN	JAX-CKB	10-Apr-24	NULL	0.044347695	GSK690693	iuphar.ligand:5196	GSK690693	FALSE	FALSE	FALSE
RET	hgnc:9967	RET	JAX-CKB	10-Apr-24	NULL	0.3968833804663227	Sunitinib	rxcui:357977	SUNITINIB	TRUE	FALSE	TRUE
RB1	hgnc:9884	RB1	JAX-CKB	10-Apr-24	NULL	1.207072901969988	Nutlin-3a	ncit:C74594	REBEMADLIN	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.077273983	Ceralasertib	ncit:C111993	CERALASERTIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.014488872	PD-0325901	ncit:C52195	MIRDAMETINIB	FALSE	FALSE	TRUE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.1159109740302306	ALRN-6924	ncit:C118669	SULANEMADLIN	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.025757994	LY3009120	iuphar.ligand:8943	LY3009120	FALSE	FALSE	FALSE
TP53	hgnc:11998	TP53	JAX-CKB	10-Apr-24	NULL	0.010537361	Cabozantinib	rxcui:1363267	CABOZANTINIB S-MALATE	TRUE	FALSE	TRUE
NCBIGENE:333	hgnc:597	APLP1	GuideToPharmacology	2024.1	agonist	5.834185692854944	IUPHAR.LIGAND:10252	iuphar.ligand:10252	LV-2186	FALSE	FALSE	FALSE
